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Citius Pharmaceuticals, Inc.

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FY2018 Annual Report · Citius Pharmaceuticals, Inc.
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UNITED STATES
SECURITIES AND EXCHANGE COMMISSION
Washington, D.C. 20549

FORM 10-K

☒ ANNUAL REPORT PURSUANT TO SECTION 13 OR 15(d) OF THE SECURITIES EXCHANGE ACT OF 1934

For the Fiscal Year Ended September 30, 2018

☐ TRANSITION REPORT PURSUANT TO SECTION 13 OR 15(d) OF THE SECURITIES EXCHANGE ACT OF 1934

Commission File Number 333-170781

Citius Pharmaceuticals, Inc.
(Exact name of Registrant as specified in its Charter)

Nevada
(State or other jurisdiction of
incorporation or organization)

27-3425913
(I.R.S. Employer
Identification No.)

11 Commerce Drive, First Floor, Cranford, NJ 07016
(Address of principal executive offices) (Zip Code)

(908) 967-6677
(Registrant’s telephone number, including area code)

(Former name and address, if changed since last report)

Securities registered pursuant to Section 12(b) of the Exchange Act:

Common Stock, par value $0.001 per share
Warrants to purchase Common Stock

The NASDAQ Capital Market
The NASDAQ Capital Market

(Title or Class)

Indicate by check mark if the registrant is a well-known seasoned issuer, as defined in Rule 405 of the Securities Act. ☐ Yes ☒ No

Indicate by check mark if the registrant is not required to file reports pursuant to Section 13 or 15(d) of the Act. ☐ Yes ☒ No

Indicate by check mark whether the registrant (1) has filed all reports required to be filed by Section 13 or 15(d) of the Exchange Act of 1934 during the
preceding 12 months (or for such shorter period that the registrant was required to file such reports), and (2) has been subject to such filing requirements
for the past ninety (90) days. ☒ Yes ☐ No

Indicate  by  check  mark  whether  the  registrant  has  submitted  electronically  and  posted  on  its  corporate  Website,  if  any,  every  Interactive  Data  File
required  to  be  submitted  and  posted  pursuant  to  Rule  405  of  Regulation  S-T  during  the  preceding  12  months  (or  for  such  shorter  period  that  the
registrant was required to submit and post such files). ☒ Yes ☐ No

Indicate by check mark if disclosure of delinquent filers pursuant to Item 405 of Regulation S-K is not contained herein, and will not be contained, to the
best of registrant’s knowledge, in definitive proxy or information statements incorporated by reference in Part III of this Form 10-K or any amendments
to this Form 10-K. ☐

Indicate by check mark whether the registrant is a large accelerated filer, an accelerated filer, a non-accelerated filer, smaller reporting company, or an
emerging  growth  company.  See  the  definitions  of  “large  accelerated  filer,”  “accelerated  filer,”  “smaller  reporting  company,”  and  “emerging  growth
company” in Rule 12b-2 of the Exchange Act.

Large accelerated filer
Non-accelerated filer

☐
☒

Accelerated filer
Smaller reporting company
Emerging growth company

☐
☒
☐

If an emerging growth company, indicate by check mark if the registrant has elected not to use the extended transition period for complying with any
new or revised financial accounting standards provided pursuant to Section 13(a) of the Exchange Act. ☐

Indicate by check mark whether the registrant is a shell company (as defined in Rule 12b-2 of the Exchange Act). ☐ Yes ☒ No

The  aggregate  market  value  of  the  voting  and  non-voting  common  equity  held  by  non-affiliates*  computed  by  reference  to  the  price  at  which  the
common equity was last sold, or the average bid and asked price of such common equity, as of the last business day of the registrant’s most recently
completed second fiscal quarter (March 31, 2018) was $19.7 million.

Affiliates for the purpose of this item refers to the issuer’s officers and directors and/or any persons or firms (excluding those brokerage firms and/or
clearing houses and/or depository companies holding issuer’s securities as record holders only for their respective clienteles’ beneficial interest) owning
10% or more of the issuer’s common stock, both of record and beneficially.

Indicate the number of shares outstanding of each of the registrant’s classes of Common Stock, as of the latest practicable date:

APPLICABLE ONLY TO CORPORATE REGISTRANTS

17,798,791 shares as of December 1, 2018, all of one class of Common Stock, $0.001 par value.

DOCUMENTS INCORPORATED BY REFERENCE

Portions  of  the  Company’s  Proxy  Statement  for  the Annual  Meeting  of  Shareholders  expected  to  be  held  on  February  13,  2019  are  incorporated  by
reference in Part III of this Report.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Citius Pharmaceuticals, Inc.
FORM 10-K
September 30, 2018

TABLE OF CONTENTS

Business
Risk Factors
Unresolved Staff Comments
Properties
Legal Proceedings
Mine Safety Disclosures

Market for Registrant’s Common Equity, Related Stockholder Matters and Issuer Purchases of Equity Securities
Selected Financial Data
Management’s Discussion and Analysis of Financial Condition and Results of Operations
Quantitative and Qualitative Disclosures About Market Risk
Financial Statements and Supplementary Data
Changes in and Disagreements With Accountants on Accounting and Financial Disclosure
Controls and Procedures
Other Information

Directors, Executive Officers and Corporate Governance
Executive Compensation
Security Ownership of Certain Beneficial Owners and Management and Related Stockholder Matters
Certain Relationships and Related Transactions and Director Independence
Principal Accounting Fees and Services

PART I

Item 1.
Item 1A.
Item 1B
Item 2.
Item 3.
Item 4.

PART II

Item 5.
Item 6.
Item 7.
Item 7A.
Item 8.
Item 9.
Item 9A.
Item 9B.

PART III

Item 10.
Item 11.
Item 12.
Item 13.
Item 14.

PART IV  

Item 15.

Exhibits, Financial Statement Schedules

Signatures

i

Page

1
12
30
30
30
30

31
31
31
37
F-1
38
38
38

39
39
39
39
39

40

43

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
  
NOTES

In  this  annual  report  on  Form  10-K,  and  unless  the  context  otherwise  requires  the  “Company,”  “we,”  “us”  and  “our”  refer  to  Citius
Pharmaceuticals,  Inc.  and  its  wholly-owned  subsidiaries,  Citius  Pharmaceuticals,  LLC  and  Leonard-Meron  Biosciences,  Inc.,  taken  as  a
whole.

Mino-Lok® is our registered trademark. All other trade names, trademarks and service marks appearing in this prospectus are the property
of their respective owners. We have assumed that the reader understands that all such terms are source-indicating. Accordingly, such terms,
when first mentioned in this prospectus, appear with the trade name, trademark or service mark notice and then throughout the remainder of
this prospectus without trade name, trademark or service mark notices for convenience only and should not be construed as being used in a
descriptive or generic sense.

FORWARD-LOOKING STATEMENTS

This Annual  Report  on  Form  10-K  contains  “forward-looking  statements.”  Forward-looking  statements  include,  but  are  not  limited  to,
statements that express our intentions, beliefs, expectations, strategies, predictions or any other statements relating to our future activities or
other future events or conditions. These statements are based on current expectations, estimates and projections about our business based,
in part, on assumptions made by management. These statements are not guarantees of future performance and involve risks, uncertainties
and assumptions that are difficult to predict. Therefore, actual outcomes and results may, and are likely to, differ materially from what is
expressed or forecasted in the forward-looking statements due to numerous factors discussed from time to time in this report, including the
risks described under Item 1A - “Risk Factors,” and Item 7 - “Management’s Discussion and Analysis of Financial Condition and Results
of  Operations”  in  this  report  and  in  other  documents  which  we  file  with  the  Securities  and  Exchange  Commission.  In  addition,  such
statements could be affected by risks and uncertainties related to:

● our ability to raise funds for general corporate purposes and operations, including our clinical trials;

● the cost, timing and results of our clinical trials;

● our ability to obtain and maintain required regulatory approvals for our product candidates;

● the commercial feasibility and success of our technology;

● our ability to recruit qualified management and technical personnel to carry out our operations; and

● the other factors discussed in the “Risk Factors” section and elsewhere in this report.

Any  forward-looking  statements  speak  only  as  of  the  date  on  which  they  are  made,  and,  except  as  may  be  required  under  applicable
securities laws, we do not undertake any obligation to update any forward-looking statement to reflect events or circumstances after the
filing date of this report.

ii

 
 
 
 
 
 
 
 
 
 
 
 
 
 
Item 1. Business

Overview

PART I

Citius Pharmaceuticals, Inc., headquartered in Cranford, New Jersey, is a specialty pharmaceutical company dedicated to the development
and commercialization of critical care products targeting important medical needs with a focus on anti-infective products in adjunct cancer
care and unique prescription products. Our goal is to achieve leading market positions by providing therapeutic products that address unmet
medical  needs  yet  have  a  lower  development  risk  than  is  associated  with  new  chemical  entities.  New  formulations  or  combinations  of
previously approved drugs with substantial existing safety and efficacy data are a core focus as we seek to reduce development and clinical
risks  associated  with  drug  development.  Our  strategy  centers  on  products  that  have  intellectual  property  and  regulatory  exclusivity
protection, while providing competitive advantages over other existing therapeutic approaches.

The  Company  was  founded  as  Citius  Pharmaceuticals,  LLC,  a  Massachusetts  limited  liability  company,  on  January  23,  2007.  On
September  12,  2014,  Citius  Pharmaceuticals,  LLC  entered  into  a  Share  Exchange  and  Reorganization  Agreement,  with  Citius
Pharmaceuticals,  Inc.  (formerly  Trail  One,  Inc.),  a  publicly  traded  company  incorporated  under  the  laws  of  the  State  of  Nevada.  Citius
Pharmaceuticals, LLC became a wholly-owned subsidiary of Citius. On March 30, 2016, Citius acquired Leonard-Meron Biosciences, Inc.
as  a  wholly-owned  subsidiary.  LMB  was  a  pharmaceutical  company  focused  on  the  development  and  commercialization  of  critical  care
products with a concentration on anti-infectives.

Since  its  inception,  the  Company  has  devoted  substantially  all  of  its  efforts  to  business  planning,  research  and  development,  recruiting
management  and  technical  staff,  and  raising  capital.  We  are  developing  two  proprietary  products:  Mino-Lok,  an  antibiotic  lock  solution
used to treat patients with catheter-related bloodstream infections by salvaging the infected catheter, and a hydrocortisone-lidocaine topical
formulation that is intended to provide anti-inflammatory and anesthetic relief to individuals suffering from hemorrhoids. We believe the
markets for our products are large, growing, and underserved by the current prescription products or procedures.

Citius is subject to a number of risks common to companies in the pharmaceutical industry including, but not limited to, risks related to the
development by Citius or its competitors of research and development stage products, market acceptance of its products, competition from
larger  companies,  dependence  on  key  personnel,  dependence  on  key  suppliers  and  strategic  partners,  the  Company’s  ability  to  obtain
additional financing and the Company’s compliance with governmental and other regulations.

Mino-Lok®

Overview

Mino-Lok is a patented solution containing minocycline, disodium ethylenediaminetetraacetic acid (edetate), and ethyl alcohol, all of which
act synergistically to treat and salvage infected central venous catheters (“CVCs”) in patients with catheter related bloodstream infections
(“CRBSIs”).  Mino-Lok  breaks  down  biofilm  barriers  formed  by  bacterial  colonies,  eradicates  the  bacteria,  and  provides  anti-clotting
properties to maintain patency in CVCs.

The administration of Mino-Lok consists of filling the lumen of the catheter with 0.8 ml to 2.0 ml of Mino-Lok solution. The catheter is
then “locked”, meaning that the solution remains in the catheter without flowing into the vein. the lock is maintained for a dwell-time of
two hours while the catheter is not in use. If the catheter has multiple lumens, all lumens may be locked with the Mino-Lok solution either
simultaneously or sequentially. If patients are receiving continuous infusion therapy, the catheters alternate between being locked with the
Mino-Lok solution and delivering therapy. The Mino-Lok therapy is two hours per day for at least five days, usually with two additional
locks in the subsequent two weeks. After locking the catheter for two hours, the Mino-Lok solution is aspirated, and the catheter is flushed
with normal saline. At that time, either the infusion will be continued, or will be locked with the standard-of-care lock solution until further
use of the catheter is required. In a clinical study conducted by MD Anderson Cancer Center (“MDACC”), there were no serum levels of
either  minocycline  or  edetate  detected  in  the  sera  of  several  patients  who  underwent  daily  catheter  lock  solution  with  minocycline  and
edetate (“M-EDTA”) at the concentration level proposed in Mino-Lok treatment. Thus, it has been demonstrated that the amount of either
minocycline or edetate that leaks into the serum is very low or none at all.

1

 
 
 
 
 
 
 
 
 
 
 
 
 
Phase 2b Results

From April 2013 to July 2014, 30 patients with CVC-related bloodstream infection were enrolled at MDACC in a prospective Phase 2b
study.  Patients  received  Mino-Lok  therapy  for  two  hours  once  daily  for  a  minimum  of  five  days  within  the  first  week  followed  by  two
additional  locks  within  the  next  two  weeks.  Patients  were  followed  for  one  month  post  lock  therapy.  Demographic  information,  clinical
characteristics, laboratory data, therapy, as well as adverse events and outcome were collected for each patient. Median age at diagnosis
was  56  years  (range:  21-73  years).  In  all  patients,  prior  to  the  use  of  lock  therapy,  systemic  treatment  with  a  culture-directed,  first-line
intravenous  antibiotic  was  started.  Microbiological  eradication  was  achieved  at  the  end  of  therapy  in  all  cases.  None  of  the  patients
experienced any serious adverse event related to the lock therapy.

The active arm, which is the Mino-Lok treated group of patients, was then compared to 60 patients in a matched cohort that experienced
removal and replacement of their CVCs within the same contemporaneous timeframe. The patients were matched for cancer type, infecting
organism, and level of neutropenia. All patients were cancer patients and treated at the MDACC. The efficacy of Mino-Lok therapy was
100% in salvaging CVCs, demonstrating equal effectiveness to removing the infected CVC and replacing with a new catheter.

The main purpose of the study was to show that Mino-Lok therapy was at least as effective as the removal and replacement of CVCs when
CRBSIs are present, and that the safety was better, that is, the complications of removing an infected catheter and replacing with a new one
could be avoided. In addition to having a 100% efficacy rate with all CVCs being salvaged, Mino-Lok therapy had no significant adverse
events  (“SAEs”),  compared  to  an  18%  SAE  rate  in  the  matched  cohort  where  patients  had  the  infected  CVCs  removed  and  replaced
(“R&R”) with a fresh catheter. There were no overall complication rates in the Mino-Lok arm group compared to 11 patients with events
(18%)  in  the  control  group.  These  events  included  bacterial  relapse  (5%)  at  four  (4)  weeks  post-intervention,  and  a  number  of
complications associated with mechanical manipulation in the removal or replacement procedure for the catheter (10%) or development of
deep  seated  infections  such  as  septic  thrombophlebitis  and  osteomyelitis  (8%).  As  footnoted,  six  (6)  patients  had  more  than  one  (1)
complication in the control arm group.

Parameter

Patients
Cancer type

- Hematologic
- Solid tumor
ICU Admission
Mech.Ventilator
Bacteremia
- Gram+
- Gram-

Neutropenia (<500)
Microbiologic Eradication

- Relapse
Complications
SAEs related R&R
Overall Complication Rate

Mino-Lok® Arm
(%)
N

Control Arm

N

(%)

30     

20     
10     
4     
3     

17     
14     
19     
30     
0     
0     
0     
0     

(100%)   

(67)
(33)
(13)
(10)

(57)*    
(47)*    
(63)
(100)
(0)
(0)
(0)
(0%)   

60 

48 
12 
4 
0 

32 
28 
36 
60 
3 
8 
6 
11**   

(100%)

(80)
(20)
(7)
(0)

(53)
(47)
(60)
(100)
(5)
(13)
(10)
(18%)

* 1 Polymicrobial patient had a Gram+ and a Gram- organism cultured
** 6 Patients had > 1 complication

Source: Dr. Issam Raad, Antimicrobial Agents and Chemotherapy, June 2016, Vol. 60 No. 6, Page 3429

2

 
 
 
 
 
 
 
 
 
 
 
 
   
 
 
 
 
 
   
   
   
      
  
   
  
   
  
   
   
   
   
   
   
   
   
   
   
   
   
   
      
  
   
  
   
  
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
 
 
 
Phase 3 Initiation

In  November  2016,  the  Company  initiated  site  recruitment  for  Phase  3  clinical  trials.  From  initiation  through  first  quarter  2017,  the
Company  received  input  from  several  sites  related  to  the  control  arm  as  being  less  than  standard  of  care  for  some  of  the  respective
institutions. The Company worked closely with the U.S. Food and Drug Administration (“FDA”) with respect to the design of the phase 3
trial, and received feedback on August 17, 2017. The FDA stated that they recognized that there is an unmet medical need in salvaging
infected catheters and agreed that an open label, superiority design would address the Company’s concerns and would be acceptable to meet
the  requirements  of  a  new  drug  application.  The  Company  amended  the  phase  3  study  design  to  remove  the  saline  and  heparin  placebo
control  arm  and  to  use  an  active  control  arm  that  conforms  with  today’s  current  standard  of  care.  Patient  enrollment  commenced  in
February 2018.

The Mino-Lok Phase 3 Trial is planned to enroll 700 patients in 50 participating institutions, all located in the U.S. There will be interim
analyses at both the 50% and 75% points of the trial as measured by the number of patients treated. As of December 2018, there are 20
active  sites  currently  enrolling  patients  including  such  academic  centers  as  MD Anderson  Cancer  Center,  Henry  Ford  Health  Center,
Georgetown  University  Medical  Center,  University  of  Chicago,  and  others.  There  are  15  additional  well  renowned  medical  centers  in
startup mode. When these study centers are activated, site recruitment will have reached 75% of the target institutions planned; and there
are another 30 centers in feasibility stage as of December 1, 2018.

Fast Track Designation

In October 2017, the Company received official notice from FDA that the investigational program for Mino-Lok was granted “Fast Track”
status. Fast Track is a designation that expedites FDA review to facilitate development of drugs which treat a serious or life-threatening
condition and fill an unmet medical need. A drug that receives Fast Track designation is eligible for the following:

● More frequent  meetings  with  FDA  to  discuss  the  drug’s  development  plan  and  ensure  collection  of  appropriate  data  needed  to

support drug approval;

● More frequent written correspondence from FDA about the design of the clinical trials;

● Priority review to shorten the FDA review process for a new drug from ten months to six months; and,

● Rolling review,  which  means  Citius  can  submit  completed  sections  of  its  New  Drug Application  (“NDA”)  for  review  by  FDA,

rather than waiting until every section of the application is completed before the entire application can be reviewed.

Mino-Lok International Study

In October 2017, data from an international study on Mino-Lok was presented at the Infectious Disease Conference, (“ID Week”), in San
Diego,  California.  The  44  patient  study  was  conducted  in  Brazil,  Lebanon,  and  Japan  and  showed  Mino-Lok  therapy  was  an  effective
intervention to salvage long term, infected central venous catheters (CVCs) in catheter related bloodstream infections in patients who had
cancer with limited vascular access. This study showed 95% effectiveness for Mino-Lok therapy in achieving microbiological eradication
of the CVCs as compared to 83% for the control.

Stability Patent Application for Mino-Lok

In July 2018, the Company received notice from the MD Anderson Cancer Center that the U.S. Patent and Trademark Office has reviewed
and  examined  the  patent  application  US  2017/051373 A1  and  that  it  is  allowed  for  issuance  as  a  patent.  The  new  invention  overcomes
limitations  in  mixing  antimicrobial  solutions  in  which  components  have  precipitated  because  of  physical  and/or  chemical  factors,  thus
limiting the stability of the post-mix solutions.

Citius holds the exclusive worldwide license which provides access to this patented technology for development and commercialization of
Mino-Lok.

3

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Market Opportunity

In  spite  of  best  clinical  practice,  catheters  contribute  to  approximately  70%  of  blood  stream  infections  that  occur  in  the  ICU,  or  are
associated  with  hemodialysis  or  cancer  patients  (approximately  470,000  per  year).  Bacteria  enter  the  catheter  either  from  the  skin  or
intraluminally  through  the  catheter  hub.  Once  in  the  catheter,  bacteria  tend  to  form  a  protective  biofilm  on  the  interior  surface  of  the
catheter that is resistant to most antimicrobial solutions. The most frequently used maintenance flush, heparin, actually stimulates biofilm
formation. Heparin is widely used as a prophylactic lock solution, in spite of the evidence that it contributes to the promotion of biofilm
formation. The formation of bacterial biofilm usually precedes CRBSIs.

The SOC in the management of CRBSI patients consists of removing the infected CVC and replacing it with a new catheter at a different
vascular access site. However, in cancer and hemodialysis patients with long-term surgically implantable silicone catheters, removal of the
CVC and reinsertion of a new one at a different site might be difficult, or even impossible, because of the unavailability of other accessible
vascular sites and the need to maintain infusion therapy. Furthermore, critically ill patients with short-term catheters often have underlying
coagulopathy,  which  makes  reinsertion  of  a  new  CVC  at  a  different  site,  in  the  setting  of  CRBSIs,  risky  in  terms  of  mechanical
complications,  such  as  pneumothorax,  misplacement,  or  arterial  puncture.  Studies  have  also  revealed  that  CRBSI  patients  may  be
associated  with  serious  complications,  including  septic  thrombosis,  endocarditis  and  disseminated  infection,  particularly  if  caused  by
Staphylococcus aureus  or Candida  species.  Furthermore,  catheter  retention  in  patients  with  CRBSIs  is  associated  with  a  higher  risk  of
relapse and poor response to antimicrobial therapy.

According to Maki et al., published in the Mayo Clinic Proceedings in 2006, there are approximately 250,000 CRBSIs annually in the U.S.
Subsequent to this study, our estimates have ranged upwards to over 450,000 CLABSIs annually (see analysis in the table below). CRBSIs
are associated with a 12% to 35% mortality rate and an attributable cost of $35,000 to $56,000 per episode.

We estimate that the potential market for Mino-Lok in the U.S. to be approximately $500 million to $1 billion as shown in the table below
based on a target price of up to $300 per dose of each salvage flush treatment.

No. of Catheters
Avg. Duration (Days)
Catheter Days
Infection Rate
Catheters Infected
Flushes/Catheter
Total Salvage Flushes

Long-Term
CVC
 4 million     
100     

Short-Term
CVC
3 million     
12     

Total
7 million 
N/A 
36 million      400 million      436 million 
 N/A 
472,000 
6.7 
3,160,000 

    2/1,000 days      1/1,000 days     
400,000     
7     
2,800,000     

72,000     
5     
360,000     

Sources: Ann Intern Med 2000; 132:391-402, Clev Clin J Med 2011; 78(1):10-17, JAVA 2007; 12(1):17-27, J Inf Nurs 2004;27(4):245-
250, Joint Commission website Monograph, CLABSI and Internal Estimates.

Under various plausible pricing scenarios, we believe that Mino-Lok would be cost saving to the healthcare system given that the removal
of an infected CVC and replacement of a new catheter in a different venous access site is estimated by the Company to cost between $8,000
and  $10,000.  Furthermore,  there  are  potential  additional  medical  benefits,  a  reduction  in  patient  discomfort  and  avoidance  of  serious
adverse events with the Mino-Lok approach since the catheter remains in place and is not subject to manipulation. We believe there will be
an economic argument to enhance the adoption of Mino-Lok by infection control committees at acute care institutions.

4

 
 
 
 
 
 
 
 
 
   
   
 
   
   
   
   
   
   
 
 
 
In January of 2017, the Company commissioned a primary market research study with MEDACore, a subsidiary of Leerink, a healthcare
focused  network  with  more  than  35,000  healthcare  professionals,  including  key  opinion  leaders,  experienced  practitioners  and  other
healthcare  professionals  throughout  North  America,  Europe,  Asia  and  other  locations  around  the  world.  This  network  includes
approximately 55 clinical specialties, 21 basic sciences and 20 business specialties. As part of this market research project, the Company
commissioned  a  third  party  survey  of  31  physicians  to  qualify  the  need  for  catheter  salvage  in  patients  with  infected,  indwelling  central
venous lines, especially when the catheter is a tunneled or an implanted port. There were 19 infectious disease experts and 12 intensivists
surveyed  who  all  agreed  that  salvage  would  be  preferable  to  catheter  exchange  to  avoid  catheter  misplacements,  blood  clots,  or  vessel
punctures that can potentially occur during reinsertion. Most were also concerned that viable venous access may not be available in patients
who were vitally dependent on a central line.

Hydro-Lido

Overview

Hydro-Lido is a topical formulation of hydrocortisone and lidocaine that is intended for the treatment of hemorrhoids. To our knowledge,
there are currently no FDA-approved prescription drug products for the treatment of hemorrhoids. Some physicians are known to prescribe
topical  steroids  for  the  treatment  of  hemorrhoids.  In  addition,  there  are  various  strengths  of  topical  combination  prescription  products
containing hydrocortisone along with lidocaine or pramoxine, each a topical anesthetic, that are prescribed by physicians for the treatment
of  hemorrhoids.  These  products  contain  drugs  that  were  in  use  prior  to  the  start  of  the  Drug  Efficacy  Study  Implementation  (“DESI”)
program  and  are  commonly  referred  to  as  DESI  drugs.  However,  none  of  these  single-agent  or  combination  prescription  products  have
been  clinically  evaluated  for  safety  and  efficacy  and  approved  by  the  FDA  for  the  treatment  of  hemorrhoids.  Further,  many  hemorrhoid
patients  use  over  the  counter  (“OTC”)  products  as  their  first  line  therapy.  OTC  products  contain  any  one  of  several  active  ingredients
including glycerin, phenylephrine, pramoxine, white petrolatum, shark liver oil and/or witch hazel, for symptomatic relief.

Development of Hemorrhoids Drugs

Hemorrhoids  are  a  common  gastrointestinal  disorder,  characterized  by  anal  itching,  pain,  swelling,  tenderness,  bleeding  and  difficulty
defecating.  In  the  U.S.,  hemorrhoids  affect  nearly  5%  of  the  population,  with  approximately  10  million  persons  annually  admitting  to
having symptoms of hemorrhoidal disease. Of these persons, approximately one third visit a physician for evaluation and treatment of their
hemorrhoids. The data also indicate that for both sexes a peak of prevalence occurs from age 45 to 65 years with a subsequent decrease after
age 65 years. Caucasian populations are affected significantly more frequently than African Americans, and increased prevalence rates are
associated with higher socioeconomic status in men but not women. Development of hemorrhoids before age 20 is unusual. In addition,
between 50% and 90% of the general U.S., Canadian and European population will experience hemorrhoidal disease at least once in life.
Although hemorrhoids and other anorectal diseases are not life-threatening, individual patients can suffer from agonizing symptoms which
can limit social activities and have a negative impact on the quality of life.

Hemorrhoids  are  defined  as  internal  or  external  according  to  their  position  relative  to  the  dentate  line.  Classification  is  important  for
selecting  the  optimal  treatment  for  an  individual  patient. Accordingly,  physicians  use  the  following  grading  system  referred  to  as  the
Goligher’s classification of internal hemorrhoids:

Grade I

Hemorrhoids not prolapsed but bleeding.

Grade II

Hemorrhoids prolapse and reduce spontaneously with or without bleeding.

Grade III

Prolapsed hemorrhoids that require reduction manually.

Grade IV

Prolapsed and  cannot  be  reduced  including  both  internal  and  external  hemorrhoids  that  are  confluent  from  skin  tag  to  inner
anal canal.

5

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Development Activities to Date

In  the  fall  of  2015,  we  completed  dosing  patients  in  a  double-blind  dose  ranging  placebo  controlled  Phase  2a  study  where  six  different
formulations  containing  hydrocortisone  and  lidocaine  in  various  strengths  (“CITI-001”)  were  tested  against  the  vehicle  control.  The
objectives  of  this  study  were  to:  1)  demonstrate  the  safety  and  efficacy  of  the  formulations  when  applied  twice  daily  for  two  weeks  in
subjects  with  Grade  I  or  II  hemorrhoids  and  2)  assess  the  potential  contribution  of  lidocaine  hydrochloride  and  hydrocortisone  acetate,
alone or in combination for the treatment of symptoms of Goligher’s Classification Grade I or II hemorrhoids.

Symptom improvement was observed based on a global score of disease severity (“GSDS”), and based on some of the individual signs and
symptoms  of  hemorrhoids,  specifically  itching  and  overall  pain  and  discomfort.  Within  the  first  few  days  of  treatment,  the  combination
products  (containing  both  hydrocortisone  and  lidocaine)  were  directionally  favorable  versus  the  placebo  and  their  respective  individual
active treatment groups (e.g., hydrocortisone or lidocaine alone) in achieving ‘almost symptom free’ or ’symptom free’ status according to
the GSDS scale. These differences suggest the possibility of a benefit for the combination product formulation.

Overall, results from adverse event reporting support the safety profile of all test articles evaluated in this study and demonstrate similar
safety profiles as compared to the vehicle. The safety findings were unremarkable. There was a low occurrence of adverse events and a
similar rate of treatment related adverse events across all treatment groups. The majority of adverse events were mild and only one was
severe. None of the adverse events were serious and the majority of adverse events were recovered/resolved at the end of the study. There
were only two subjects who were discontinued from the study due to adverse events.

In addition to the safety and dose-ranging information, information was obtained relating to the use of the GSDS as an assessment tool for
measuring  the  effectiveness  of  the  test  articles.  Individual  signs  and  symptoms  were  also  assessed  but  can  vary  from  patient  to  patient.
Therefore,  the  goal  of  the  GSDS  was  to  provide  an  assessment  tool  that  could  be  used  for  all  patients  regardless  of  which  signs  and
symptoms  they  are  experiencing.  The  GSDS  proved  to  be  a  more  effective  tool  for  assessing  the  severity  of  the  disease  and  the
effectiveness of the drug when compared to the assessment of the individual signs and symptoms. Citius believes that we can continue to
develop this assessment tool as well as other patient reported outcome endpoints for use in the next trials and in the pivotal trial.

Information was also obtained about the formulation of the drug and the vehicle. As a result of this study, we believe that the performance
of  the  active  arms  of  the  study  relative  to  the  vehicle  can  be  improved  by  re-formulating  our  topical  preparation.  Therefore,  we  have
initiated work on vehicle formulation and evaluation of higher potency steroids.

In June and July 2016, the Company engaged the Dominion Group, a leading provider of healthcare and pharmaceutical marketing research
services. The primary market research was conducted to understand the symptoms that are most bothersome to patients better in order to
develop  meaningful  endpoints  for  the  clinical  trials.  We  also  learned  about  the  factors  that  drive  patients  to  seek  medical  attention  for
hemorrhoids in an effort to understand the disease impact on quality of life. The results of this survey are able to help us develop patient
reported  outcome  evaluation  tools.  These  tools  can  be  used  in  clinical  trials  to  evaluate  the  patients’  conditions  and  to  assess  the
performance of the test articles.

In March 2018, we announced that we are selecting a higher potency corticosteroid in our steroid/anesthetic topical formulation program
for the treatment of hemorrhoids. The original topical preparation, CITI-001, which was used in the Phase 2a study, was a combination of
hydrocortisone  acetate  and  lidocaine  hydrochloride.  The  new  formulation,  CITI-002,  which  we  refer  to  as  Halo-Lido,  will  combine
lidocaine with the higher potency corticosteroid for symptomatic relief of the pain and discomfort of hemorrhoids.

We held a Type C meeting with the FDA in December 2017 to discuss the results of the Phase 2a study and to obtain the FDA’s view on
development plans to support the potential formulation change for the planned Phase 2b study. We also requested the FDA’s feedback on
our  Phase  2b  study  design,  including  target  patient  population,  inclusion/exclusion  criteria,  and  efficacy  endpoints.  The  pre-clinical  and
clinical development programs for CITI-002 are planned to be similar to those conducted for the development of CITI-001 to support the
design for a planned Phase 3 clinical trial.

6

 
 
 
 
 
 
 
 
 
 
 
Market Opportunity

The current market for OTC and topical prescription (“Rx”) products for the symptomatic treatment of hemorrhoids is highly fragmented,
and  includes  approximately  20  million  units  of  OTC  and  over  4  million  prescriptions.  None  of  the  Rx  products  have  received  FDA
approval  and  are  only  available  due  to  the  Drug  Efficacy  Study  Implementation  (“DESI”)  program,  which  started  decades  ago  after
enactment of the 1962 Kefauver-Harris Drug Amendments. These DESI products have no FDA reviewed evidence of efficacy or safety,
and may be subject to withdrawal if an approved product were to be introduced. Several topical combination prescription products for the
treatment  of  hemorrhoids  are  available  containing  hydrocortisone  in  strengths  ranging  from  0.5%  to  3.0%,  combined  with  lidocaine  in
strengths  ranging  from  1.0%  to  3.0%.  The  various  topical  formulations  include  creams,  ointments,  gels,  lotions,  enemas,  pads,  and
suppositories.  The  most  commonly  prescribed  topical  combination  gel  is  sold  as  a  branded  generic  product  and  contains  2.5%
hydrocortisone and 3.0% lidocaine.

We believe there are currently no FDA-approved prescription drug products for the treatment of hemorrhoids. Although there are numerous
Rx  and  OTC  products  commonly  used  to  treat  hemorrhoids,  none  possess  proven  safety  and  efficacy  data  generated  from  rigorously
conducted  clinical  trials.  We  believe  that  a  novel  topical  formulation  of  hydrocortisone  and  lidocaine  designed  to  provide  anti-
inflammatory and anesthetic relief and which has an FDA-approved label specifically claiming the treatment of hemorrhoids will become
an important treatment option for physicians who want to provide their patients with a therapy that has demonstrated safety and efficacy in
treating  this  uncomfortable  and  often  recurring  disease.  We  believe  that  our  CITI-002  product  represents  an  attractive,  low-risk  product
opportunity with meaningful upside potential.

Market Exclusivity

We  believe  that  we  will  be  the  first  company  to  conduct  rigorous  clinical  trials  and  receive  FDA  approval  of  a  topical  hydrocortisone-
lidocaine  combination  product  for  the  treatment  of  hemorrhoids.  If  we  receive  FDA  approval,  we  will  qualify  for  3  years  of  market
exclusivity for our dosage strength and formulation. In addition, we will also be the only product on the market specifically proven to be
safe and effective for the treatment of hemorrhoids. Generally, if a company conducts clinical trials and receives FDA approval of a product
for which there are similar, but non FDA-approved, prescription products on the market, the manufacturers of the unapproved but marketed
products  are  required  to  withdraw  them  from  the  market.  However,  the  FDA  has  significant  latitude  in  determining  how  to  enforce  its
regulatory powers in these circumstances. We have not had any communication with the FDA regarding this matter and cannot predict what
action, if any, the FDA will take with respect to the unapproved products.

We believe that should our product receive an FDA approval and demonstrate, proven safety and efficacy data, and if our products obtain 3
years of market exclusivity based on our dosage strength and formulation, we are likely to have a meaningful advantage in our pursuit of
achieving a significant position in the market for topical combination prescription products for the treatment of hemorrhoids.

Sales and Marketing

We are primarily focused on identifying opportunities within the critical care and cancer care market segments. In our product acquisition
criteria, we concentrate on markets that are highly influenced by key opinion leaders (KOLs) and have products that are prescribed by a
relatively small number of physicians, yet provide large opportunities for growth and market share. This strategy allows for a manageable
commercialization effort for our Company in terms of resources and capital. We also seek to provide cost-effective therapies that would be
endorsed by payers, patients, and providers. We believe that we will be able to commercialize products within the scope of these criteria
ourselves, and that we can create marketing synergies by having a common narrow audience for our marketing efforts (“several products in
the bag for the same customer”).

For products that we own that fall out of the narrow scope criteria, we have identified pharmaceutical companies with large sales forces,
experienced sales and marketing management teams, direct-to-consumer (“DTC”) capabilities, significantly larger resources than ours, and
non-competing product portfolios that we believe would make excellent sales and marketing partners for us. We intend to license our mass
audience, non-specialty products to such companies for sales and marketing.

7

 
 
 
 
 
 
  
 
 
 
 
Intellectual Property

We rely on a combination of patent, trade secret, copyright, and trademark laws, as well as confidentiality, licensing and other agreements,
to establish and protect our proprietary rights. Our policy is to actively seek to obtain, where appropriate, the broadest intellectual property
protection  possible  for  our  current  product  candidates  and  any  future  product  candidates  both  in  the  U.S.  and  abroad.  However,  patent
protection  may  not  provide  us  with  complete  protection  against  competitors  who  seek  to  circumvent  our  patents.  To  help  protect  our
proprietary know-how that is not patentable, and for inventions for which patents may be difficult to enforce, we currently rely and will in
the future rely on trade secret protection and confidentiality agreements to protect our interests.

Mino-Lok Intellectual Property

Mino-Lok is covered by an issued U.S. patent (no. 7,601,731), “Antimicrobials in Combination with Chelators and Ethanol for the Rapid
Eradication  of  Microorganisms  Embedded  in  Biofilm,”  which  was  issued  on  October  13,  2009.  This  patent  is  a  composition  of  matter
patent and provides intellectual property protection until June 7, 2024. There are corresponding applications pending in Europe and Canada
(European Application No. EP 1644024; Canadian Patent Application No. 0252852). On April 15, 2014, a patent application was filed for
an enhanced formulation that provides greater stability of the reconstituted Mino-Lok solution. In June 2017, the Company was notified
that US Patent Application 15/344,113 has been published by the US Patent Office with a publication date of June 1, 2017. This patent is a
step  forward  for  Mino-Lok  as  it  overcomes  limitations  in  mixing  antimicrobial  solutions  where  components  may  precipitate  because  of
physical and/or chemical factors, thus limiting the stability of the post-mix solutions.

In July 2018, the Company received notice from the MD Anderson Cancer Center that the U.S. Patent and Trademark Office has reviewed
and  examined  the  patent  application  US  2017/051373 A1  and  that  it  is  allowed  for  issuance  as  a  patent.  The  new  invention  overcomes
limitations  in  mixing  antimicrobial  solutions  in  which  components  have  precipitated  because  of  physical  and/or  chemical  factors,  thus
limiting the stability of the post-mix solutions.

On May 14, 2014, LMB entered into a patent and technology license agreement with Novel Anti-Infective Therapeutics, Inc. (“NAT”) to
develop and commercialize Mino-Lok on an exclusive, worldwide (except for South America), sub licensable basis. LMB incurred a one-
time license fee in May 2014. On March 20, 2017, LMB entered into an amendment to the license agreement that expanded the licensed
territory  to  include  South America,  providing  LMB  with  worldwide  rights.  Under  the  license  agreement,  the  Company  will  pay  (i)  an
annual maintenance fee until commercial sales of a product subject to the license, (ii) upon commercialization, we will pay annual royalties
on  net  sales  of  licensed  products,  and  (iii)  certain  regulatory  and  milestone  payments.  Unless  earlier  terminated  by  NAT  based  on  the
failure  to  achieve  certain  development  or  commercial  milestones,  the  license  agreement  remains  in  effect  until  the  date  that  all  patents
licensed under the agreement have expired and all patent applications within the licensed patent rights have been cancelled, withdrawn or
expressly abandoned.

Mino-Lok  has  received  a  Qualified  Infectious  Disease  Product  (“QIDP”)  designation.  The  QIDP  designation  provides  New  Drug
Applications an additional five years of market exclusivity, which together with the potential three years of exclusivity for the new strength
and formulation of Mino-Lok, would result in a combined total of eight years of market exclusivity regardless of patent protection

Hydro-Lido Intellectual Property

We  are  developing  a  new  formulation  of  Hydro-Lido,  CITI-002,  which  will  have  a  unique  combination  of  excipients  as  well  as  unique
concentrations  of  the  active  ingredients.  The  goal  is  to  have  a  product  that  is  optimized  for  stability  and  activity.  Once  the  formulation
development is completed and data is obtained, we intend to apply for a patent on this new topical formulation.

We  seek  to  achieve  approval  for  Hydro-Lido  by  utilizing  the  FDA’s  505(b)(2)  pathway.  This  pathway  will  provide  3  years  of  market
exclusivity.

8

 
 
 
 
 
 
 
 
 
 
 
 
Competition

We operate in a highly competitive and regulated industry which is subject to rapid and frequent changes. We face significant competition
from organizations that are pursuing drugs that would compete with the drug candidates that we are developing and the same or similar
products  that  target  the  same  conditions  we  intend  to  treat.  Due  to  our  limited  resources,  we  may  not  be  able  to  compete  successfully
against  these  organizations,  which  include  many  large,  well-financed  and  experienced  pharmaceutical  and  biotechnology  companies,  as
well as academic and research institutions and government agencies.

Mino-Lok Competition

Currently, the only alternative to Mino-Lok in the treatment of infected CVCs in CRBSI/CLABSI patients of which we are aware, is the
SOC of removing the culprit CVC and replacing a new CVC at a different vascular site. Citius is not aware of any Investigational New
Drug Applications  (“INDs”)  for  a  salvage  antibiotic  lock  solution  and  does  not  expect  any  to  be  forthcoming  due  to  the  difficulty  of
meeting the necessary criteria to be effective and practical.

At  this  time,  there  are  no  pharmacologic  agents  approved  in  the  U.S.  for  the  prevention  or  treatment  of  CLABSIs  in  central  venous
catheters. Citius is aware that there are several agents in development for prevention but none for salvage. The most prominent of these
appear to be Neutrolin from CorMedix and B-Lock from Great Lakes Pharmaceuticals, Inc. (“GLP”).

Neutrolin® (CorMedix Inc.)

Neutrolin  is  a  formulation  of  Taurolidine  1.35%,  Citrate  3.5%,  and  Heparin  1000  units/mL.  Neutrolin  is  an  anti-microbial  catheter  lock
solution being developed by CorMedix to prevent CRBSIs and to prevent clotting. In January 2015, the U.S. Food and Drug Administration
(the  “FDA”)  granted  Fast  Track  and  Qualified  Infectious  Disease  Product  (“QIDP”)  designations  for  Neutrolin.  In  December  2015,
CorMedix initiated its Phase 3 clinical trial in hemodialysis patients in the United States. The clinical trial named Catheter Lock Solution
Investigational  Trial,  or  LOCK-IT-100  is  a  prospective,  multicenter,  randomized,  double-blind,  placebo-controlled,  active  control  trial
designed to show efficacy and safety of Neutrolin in preventing CRBSIs in subjects receiving hemodialysis therapy. On April 20, 2017,
CorMedix provided an update on the LOCK-IT-100 trial. CorMedix had enrolled 368 patients to date and completed a safety review by an
independent Data and Safety Monitoring Board (“DSMB”) of the first 279 patients. The DSMB concluded that it was safe to continue the
trial as designed; however, CorMedix initiated discussions with the FDA to make some protocol changes to include one or more interim
efficacy analyses. According to CorMedix, the FDA accepted the CorMedix proposal.

On  June  20,  2018,  CorMedix  announced  that  it  had  completed  its  review  and  source-verification  of  the  data  required  for  the  interim
analysis of the Phase 3 LOCK-IT-100 study for Neutrolin®. The data was then locked and transferred to the independent biostatistician for
un-blinding and analysis, who then provided the results to the independent Data Safety Monitoring Board (DSMB) for its review.

On  July  25,  2018  CorMedix  announced  that  the  independent  Data  Safety  Monitoring  Board  (DSMB)  had  completed  its  review  of  the
interim  analysis  of  the  data  from  the  currently  ongoing  Phase  3  LOCK-IT-100  study  for  Neutrolin®.  Because  the  pre-specified  level  of
statistical significance was reached and efficacy had been demonstrated, the DSMB recommended the study be terminated early. No safety
concerns were reported by the DSMB based on the interim analysis. The company will submit the results of the interim analysis to the U.S.
Food and Drug Administration for its review.

9

 
 
 
 
 
 
 
 
 
 
 
B-Lock™ (Great Lakes Pharmaceuticals, Inc.)

B-Lock is a triple combination of trimethoprim, EDTA and ethanol from Great Lakes Pharmaceuticals, Inc. (“GLP”). On July 24, 2012,
GLP announced the initiation of a clinical study of B-Lock. We are unaware as to the progress or results of these studies. In addition, we
are not aware of any IND being filed in the US for B-Lock, nor are we aware of any clinical studies to support salvage of infected catheters
in bacteremic patients.

Neither of these lock solutions have been shown to be effective in salvaging catheters in bacteremic patients as Mino-Lok is intended to do,
and Citius does not expect that either would be pursued for this indication.

There has been no further public information available on GLP. GLP’s web site and phone number are no longer active and the Company
believes that they have ceased operations.

Hydro-Lido Competition

The primary competition in the hemorrhoid market is non-prescription over the counter products. When approved, Hydro-Lido will be the
only prescription product for the treatment of hemorrhoids.

Supply and Manufacturing

We  do  not  currently  have  and  we  do  not  intend  to  set  up  our  own  manufacturing  facilities.  We  expect  to  use  approved  contract
manufacturers  for  manufacturing  our  products  in  all  stages  of  development  after  we  file  for  FDA  approval.  Each  of  our  domestic  and
foreign contract manufacturing establishments, including any contract manufacturers we may decide to use, must be listed in the New Drug
Application (“NDA”) and must be registered with the FDA. Also, the FDA imposes substantial annual fees on manufacturers of branded
products.

In  general,  our  suppliers  purchase  raw  materials  and  supplies  on  the  open  market.  Substantially  all  such  materials  are  obtainable  from  a
number of sources so that the loss of any one source of supply would not have a material adverse effect on us.

If  we  elect  to  conduct  product  development  and  manufacturing,  we  will  be  subject  to  regulation  under  various  federal  and  state  laws,
including  the  Occupational  Safety  and  Health Act,  the  Environmental  Protection Act,  the  Toxic  Substances  Control Act,  the  Resource
Conservation and Recovery Act, the Controlled Substances Act and other present and potential future federal, state or local regulations.

We  have  contracted  with  proven  suppliers  and  manufacturers  for  active  pharmaceutical  ingredient,  development  and  packaging.  We  are
confident that all materials meet or will meet specifications discussed at the chemistry, manufacturing and controls meeting with the FDA.

Regulatory Strategy

United States Government Regulation

The research, development, testing, manufacture, labeling, promotion, advertising, distribution and marketing, among other things, of our
products are extensively regulated by governmental authorities in the United States and other countries. Our products may be classified by
the FDA as a drug or a medical device depending upon the indications for use or claims. Because certain of our  product  candidates  are
considered as medical devices and others are considered as drugs for regulatory purposes, we intend to submit applications to regulatory
agencies for approval or clearance of both medical device and pharmaceutical product candidates.

In  the  United  States,  the  FDA  regulates  drugs  and  medical  devices  under  the  Federal  Food,  Drug,  and  Cosmetic Act  and  the  agency’s
implementing regulations. If we fail to comply with the applicable United States requirements at any time during the product development
process, clinical testing, and the approval process or after approval, we may become subject to administrative or judicial sanctions. These
sanctions could include the FDA’s refusal to approve pending applications, license suspension or revocation, withdrawal of an approval,
warning  letters,  adverse  publicity,  product  recalls,  product  seizures,  total  or  partial  suspension  of  production  or  distribution,  injunctions,
fines, civil penalties or criminal prosecution. Any agency enforcement action could have a material adverse effect on our company.

10

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Foreign Regulatory Requirements

We and any collaborative partners may be subject to widely varying foreign regulations, which may be different from those of the FDA,
governing clinical trials, manufacture, product registration and approval and pharmaceutical sales. Whether or not FDA approval has been
obtained, we or our collaboration partners must obtain a separate approval for a product by the comparable regulatory authorities of foreign
countries  prior  to  the  commencement  of  product  marketing  in  such  countries.  In  certain  countries,  regulatory  authorities  also  establish
pricing and reimbursement criteria. The approval process varies from country to country, and the time may be longer or shorter than that
required for FDA approval. In addition, under current United States law, there are restrictions on the export of products not approved by the
FDA, depending on the country involved and the status of the product in that country.

International  sales  of  medical  devices  manufactured  in  the  U.S.  that  are  not  approved  by  the  FDA  for  use  in  the  U.S.,  or  are  banned  or
deviate  from  lawful  performance  standards,  are  subject  to  FDA  export  requirements.  Exported  devices  are  subject  to  the  regulatory
requirements of each country to which the device is exported. Some countries do not have medical device regulations, but in most foreign
countries, medical devices are regulated. Frequently, regulatory approval may first be obtained in a foreign country prior to application in
the  U.S.  to  take  advantage  of  differing  regulatory  requirements.  Most  countries  outside  of  the  U.S.  require  that  product  approvals  be
recertified on a regular basis, generally every 5 years. The recertification process requires that we evaluate any device changes and any new
regulations  or  standards  relevant  to  the  device  and  conduct  appropriate  testing  to  document  continued  compliance.  Where  recertification
applications are required, they must be approved in order to continue selling our products in those countries.

In the European Union, in order for a product to be marketed and sold, it is required to comply with the Medical Devices Directive and
obtain CE Mark certification. The CE Mark certification encompasses an extensive review of the applicant’s quality management system
which is inspected by a notified body’s auditor as part of a stage 1 and 2 International Organization for Standardization (“ISO”) 13485:2016
audit,  in  accordance  with  worldwide  recognized  ISO  standards  and  applicable  European  Medical  Devices  Directives  for  quality
management  systems  for  medical  device  manufacturers.  Once  the  quality  management  system  and  design  dossier  has  been  successfully
audited by a notified body and reviewed and approved  by  a  competent  authority,  a  CE  certificate  for  the  medical  device  will  be  issued.
Applicants  are  also  required  to  comply  with  other  foreign  regulations  such  as  the  requirement  to  obtain  Ministry  of  Health,  Labor  and
Welfare  approval  before  a  new  product  can  be  launched  in  Japan.  The  time  required  to  obtain  these  foreign  approvals  to  market  our
products may vary from U.S. approvals, and requirements for these approvals may differ from those required by the FDA.

Medical device laws and regulations are in effect in many of the countries in which we may do business outside the United States. These
laws and regulations range from comprehensive device approval requirements for our medical device product to requests for product data
or certifications. The number and scope of these requirements are increasing. We may not be able to obtain regulatory approvals in such
countries and may be required to incur significant costs in obtaining or maintaining its foreign regulatory approvals. In addition, the export
of certain of our products which have not yet been cleared for domestic commercial distribution may be subject to FDA export restrictions.
Any failure to obtain product approvals in a timely fashion or to comply with state or foreign medical device laws and regulations may have
a serious adverse effect on our business, financial condition or results of operations.

Employees

As of September 30, 2018, we had seven employees and various consultants providing support. Through our consulting and collaboration
arrangements,  and  including  our  Scientific  Advisory  Board,  we  have  access  to  more  than  30  additional  professionals,  who  possess
significant  expertise  in  business  development,  legal,  accounting,  regulatory  affairs,  clinical  operations  and  manufacturing.  We  also  rely
upon a network of consultants to support our clinical studies and manufacturing efforts.

11

 
 
 
 
 
 
 
 
 
Executive Officers of Citius

Myron Holubiak, President, Chief Executive Officer and Director – Mr. Holubiak, 71, was appointed President, Chief Executive Officer
and Director in March 2016. He previously served as a Director of Citius since October 2015 and was the founder and Chief Executive
Officer and President of Leonard-Meron Biosciences, Inc., an acquired subsidiary of Citius, from March 2013 until March 2016.

Leonard Mazur, Executive Chairman and Secretary – Mr. Mazur, 73, has been a member of the Board since September 2014. Mr. Mazur
previously served as Chief Executive Officer, President, and Chief Operating Officer from September 2014 until March 2016.

Jaime Bartushak, Chief Financial Officer and Principal Financial Officer – Mr. Bartushak, 51, was appointed as Chief Financial Officer in
November  2017.  Previously,  he  was  one  of  the  founders  and  Chief  Financial  Officer  of  Leonard-Meron  Biosciences,  Inc.,  an  acquired
subsidiary of Citius,

Other Information

We make available, free of charge through our website, our annual report on Form 10-K, quarterly reports on Form 10-Q, current reports
on  Form  8-K  and  all  amendments  to  those  reports  as  soon  as  is  reasonably  practicable  after  such  material  is  electronically  filed  with  or
furnished to the Securities and Exchange Commission (the “SEC”) pursuant to Section 13(a) or 15(d) of the Securities Exchange Act of
1934, as amended (the “Exchange Act”). The SEC maintains an Internet site that contains these reports at www.sec.gov.

Our website address is http://www.citiuspharma.com. The information contained in, or that can be accessed through, our website is not part
of this report.

Item 1A. Risk Factors

This  report  contains  forward-looking  statements  that  involve  risks  and  uncertainties.  Our  actual  results  could  differ  materially  from
those discussed in this report. Factors that could cause or contribute to these differences include, but are not limited to, those discussed
below and elsewhere in this report and in any documents incorporated in this report by reference.

If  any  of  the  following  risks,  or  other  risks  not  presently  known  to  us  or  that  we  currently  believe  to  not  be  significant,  develop  into
actual events, then our business, financial condition, results of operations or prospects could be materially adversely affected. If that
happens, the market price of our common stock could decline, and stockholders may lose all or part of their investment.

Risks related to our Business and our Industry

We have a history of net losses and expect to incur losses for the foreseeable future. We may never generate revenues or, if we are able
to generate revenues, achieve profitability.

We were formed as a limited liability company in 2007 and since our inception have incurred a net loss in each of our previous operating
years. Our ability to become profitable depends upon our ability to obtain marketing approval for and generate revenues from sales of our
product candidates. We have been focused on product development and have not generated any revenues to date. We have incurred losses
in each period of our operations, and we expect to continue to incur losses for the foreseeable future. These losses are likely to continue to
adversely  affect  our  working  capital,  total  assets  and  shareholders’  equity  (deficit).  The  process  of  developing  our  products  requires
significant  clinical,  development  and  laboratory  testing  and  clinical  trials.  In  addition,  commercialization  of  our  product  candidates  will
require that we obtain necessary regulatory approvals and establish sales, marketing and manufacturing capabilities, either through internal
hiring  or  through  contractual  relationships  with  others.  We  expect  to  incur  substantial  losses  for  the  foreseeable  future  as  a  result  of
anticipated  increases  in  our  research  and  development  costs,  including  costs  associated  with  conducting  preclinical  testing  and  clinical
trials,  and  regulatory  compliance  activities.  We  incurred  net  losses  of  $12,536,638,  $10,384,953,  and  $8,295,698  for  the  years  ended
September 30, 2018, 2017 and 2016, respectively. At September 30, 2018, we had stockholders’ equity of $27,865,684 and an accumulated
deficit  of  $40,257,838.  Our  net  cash  used  for  operating  activities  was  $11,318,138,  $7,971,205,  and  $5,900,421  for  the  years  ended
September 30, 2018, 2017 and 2016, respectively.

12

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Our ability to generate revenues and achieve profitability will depend on numerous factors, including success in:

● developing and testing product candidates;

● receiving regulatory approvals for our product candidates;

● commercializing our product candidates;

● manufacturing commercial quantities of our product candidates at acceptable cost levels; and

● establishing a favorable competitive position for our product candidates.

Many of these factors will depend on circumstances beyond our control. We cannot assure you that any of our products will be approved
by the FDA, that we will successfully bring any product to market or, if so, that we will ever become profitable.

There is substantial doubt about our ability to continue as a going concern.

Currently, we do not have sufficient capital to continue our operations after the first nine months of fiscal 2019. You should not rely on our
consolidated balance sheet as an indication of the amount of proceeds that would be available to satisfy claims of creditors, and potentially
be available for distribution to shareholders, in the event of liquidation.

Our audited consolidated financial statements included within have been prepared assuming that we will continue as a going concern and
do not include any adjustments to reflect the possible future effects on the recoverability and classification of assets, or the amounts and
classification of liabilities that may result if we do not continue as a going concern. We have concluded that substantial doubt about our
ability to continue as a going concern exists and our auditors have made reference to this in their audit report on our audited consolidated
financial statements for the year ended September 30, 2018.

We need to secure additional financing.

We  anticipate  that  we  will  incur  operating  losses  for  the  foreseeable  future.  We  have  received  gross  proceeds  of  approximately  $35.6
million from our public and private placement offerings through September 30, 2018. Additionally, in connection with the acquisition of
LMB our Executive Chairman, Leonard Mazur, made an equity investment of $3.0 million in March 2016. Mr. Mazur has also loaned us
$4,710,000 pursuant to convertible promissory notes. On August 8, 2017, these notes and accrued interest of $76,240 were converted into
1,547,067 shares of common stock at a price of $3.09 per share as part of an underwritten public offering which closed on the same date.

The amount and timing of our future funding requirements will depend on many factors, including, but not limited to:

● the rate of progress and cost of our trials and other product development programs for our product candidates;

● the costs and timing of obtaining licenses for additional product candidates or acquiring other complementary technologies;

● the timing of any regulatory approvals of our product candidates;

● the costs of establishing sales, marketing and distribution capabilities; and

● the status, terms and timing of any collaborative, licensing, co-promotion or other arrangements.

13

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
We  will  need  to  access  the  capital  markets  in  the  future  for  additional  capital  for  research  and  development  and  for  operations.
Traditionally,  pharmaceutical  companies  have  funded  their  research  and  development  expenditures  through  raising  capital  in  the  equity
markets.  Declines  and  uncertainties  in  these  markets  over  the  past  several  years  have  severely  restricted  raising  new  capital  and  have
affected companies’ ability to continue to expand or fund existing research and development efforts. If these economic conditions continue
or  become  worse,  our  future  cost  of  equity  or  debt  capital  and  access  to  the  capital  markets  could  be  adversely  affected.  If  we  are  not
successful in securing additional financing, we may be required to delay significantly, reduce the scope of or eliminate one or more of our
research  or  development  programs,  downsize  our  general  and  administrative  infrastructure,  or  seek  alternative  measures  to  avoid
insolvency,  including  arrangements  with  collaborative  partners  or  others  that  may  require  us  to  relinquish  rights  to  certain  of  our
technologies or product candidates.

We are a late-stage development company with an unproven business strategy and may never achieve commercialization of our
therapeutic products or profitability.

Our  strategy  of  using  collaborative  partners  to  assist  us  in  the  development  of  our  therapeutic  products  is  unproven.  Our  success  will
depend upon our ability to enter into additional collaboration agreements on favorable terms and to select an appropriate commercialization
strategy for each product candidate that we and our collaborators choose to pursue. If we are not successful in implementing our strategy to
commercialize our product candidates, we may never achieve, maintain or increase profitability. Our ability to successfully commercialize
any of our products or product candidates will depend, among other things, on our ability to:

● successfully complete clinical trials for our product candidates;

● produce, through a validated process, sufficiently large quantities of our drug compound(s) to permit successful commercialization

of our product candidates;

● receive marketing approvals from the FDA and similar foreign regulatory authorities for our product candidates;

● establish commercial manufacturing arrangements with third-party manufacturers for our product candidates;

● build and  maintain  strong  sales,  distribution  and  marketing  capabilities  sufficient  to  launch  commercial  sales  of  any  approved

products or establish collaborations with third parties for such commercialization;

● secure acceptance of any approved products from physicians, health care payers, patients and the medical community; and

● manage our  spending  as  costs  and  expenses  increase  due  to  clinical  trials,  regulatory  applications  and  development  and

commercialization activities.

There are no guarantees that we will be successful in completing these tasks. If we are unable to successfully complete these tasks, we may
not  be  able  to  commercialize  any  of  our  product  candidates  in  a  timely  manner,  or  at  all,  in  which  case  we  may  be  unable  to  generate
sufficient  revenues  to  sustain  and  grow  our  business.  If  we  experience  unanticipated  delays  or  problems,  our  development  costs  could
substantially increase and our business, financial condition and results of operations will be adversely affected.

We face significant risks in our product candidate development efforts.

Our business depends on the successful development and commercialization of our product candidates. We are not permitted to market any
of our product candidates in the United States until we receive approval of an NDA from the FDA, or in any foreign jurisdiction until we
receive  the  requisite  approvals  from  such  jurisdiction.  The  process  of  developing  new  drugs  and/or  therapeutic  products  is  inherently
complex, unpredictable, time-consuming, expensive and uncertain. We must make long-term investments and commit significant resources
before  knowing  whether  our  development  programs  will  result  in  drugs  that  will  receive  regulatory  approval  and  achieve  market
acceptance. Product candidates that appear to be promising at all stages of development may not reach the market for a number of reasons
that may not be predictable based on results and data of the clinical program. Product candidates may be found ineffective or may cause
harmful side effects during clinical trials, may take longer to progress through clinical trials than had been anticipated, may not be able to
achieve  the  pre-defined  clinical  endpoints  due  to  statistical  anomalies  even  though  clinical  benefit  may  have  been  achieved,  may  fail  to
receive  necessary  regulatory  approvals,  may  prove  impracticable  to  manufacture  in  commercial  quantities  at  reasonable  cost  and  with
acceptable quality, or may fail to achieve market acceptance.

14

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
We  cannot  predict  whether  or  when  we  will  obtain  regulatory  approval  to  commercialize  our  product  candidates  that  are  under
development  and  we  cannot,  therefore,  predict  the  timing  of  any  future  revenues  from  these  product  candidates,  if  any.  The  FDA  has
substantial discretion in the drug approval process, including the ability to delay, limit or deny approval of a product candidate for many
reasons. For example, the FDA:

● could determine that we cannot rely on Section 505(b)(2) for Mino-Lok or Hydro-Lido or any future product candidates;

● could determine  that  the  information  provided  by  us  was  inadequate,  contained  clinical  deficiencies  or  otherwise  failed  to

demonstrate the safety and effectiveness of any of our product candidates for any indication;

● may not  find  the  data  from  clinical  trials  sufficient  to  support  the  submission  of  an  NDA  or  to  obtain  marketing  approval  in  the

United States, including any findings that the clinical and other benefits of our product candidates outweigh their safety risks;

● may disagree  with  our  trial  design  or  our  interpretation  of  data  from  preclinical  studies  or  clinical  trials,  or  may  change  the

requirements for approval even after it has reviewed and commented on the design for our trials;

● may determine that we have identified the wrong reference listed drug or drugs or that approval of our Section 505(b)(2) application

for any of our product candidates is blocked by patent or non-patent exclusivity of the reference listed drug or drugs;

● may identify  deficiencies  in  the  manufacturing  processes  or  facilities  of  third-party  manufacturers  with  which  we  enter  into

agreements for the manufacturing of our product candidates;

● may approve our product candidates for fewer or more limited indications than we request, or may grant approval contingent on the

performance of costly post-approval clinical trials;

● m a y change  its  approval  policies  or  adopt  new  regulations  that  could  adversely  impact  our  product  candidate  development

programs; or

● may not approve the labeling claims that we believe are necessary or desirable for the successful commercialization of our product

candidates.

Any failure to obtain regulatory approval of our product candidates would significantly limit our ability to generate revenues, and any
failure to obtain such approval for all of the indications and labeling claims we deem desirable could reduce our potential revenues.

The results of pre-clinical studies and completed clinical trials are not necessarily predictive of future results, and our current product
candidates may not have favorable results in later studies or trials.

Pre-clinical studies and Phase 1 and Phase 2 clinical trials are not primarily designed to test the efficacy of a product candidate in the
general population, but rather to test initial safety, to study pharmacokinetics and pharmacodynamics, to study limited efficacy in a small
number of study patients in a selected disease population, and to identify and attempt to understand the product candidate’s side effects at
various doses and dosing schedules. Success in pre-clinical studies or completed clinical trials does not ensure that later studies or trials,
including continuing pre-clinical studies and large-scale clinical trials, will be successful nor does it predict future results. Favorable results
in early studies or trials may not be repeated in later studies or trials, and product candidates in later stage trials may fail to show acceptable
safety and efficacy despite having progressed through earlier trials. In addition, the placebo rate in larger studies may be higher than
expected.

15

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
We may be required to demonstrate through large, long-term outcome trials that our product candidates are safe and effective for use in a
broad population prior to obtaining regulatory approval.

There  is  typically  a  high  rate  of  attrition  from  the  failure  of  product  candidates  proceeding  through  clinical  trials.  In  addition,  certain
subjects in our clinical trials may respond positively to placebo treatment - these subjects are commonly known as “placebo responders” -
making it more difficult to demonstrate efficacy of the test drug compared to placebo. This effect is likely to be observed in the treatment of
hemorrhoids.

If  any  of  our  product  candidates  fail  to  demonstrate  sufficient  safety  and  efficacy  in  any  clinical  trial,  we  will  experience  potentially
significant delays in, or may decide to abandon development of that product candidate. If we abandon or are delayed in our development
efforts related to any of our product candidates, we may not be able to generate any revenues, continue our operations and clinical studies,
or become profitable. Our reputation in the industry and in the investment community would likely be significantly damaged. Further, it
might not be possible for us to raise funds in the public or private markets, and our stock price would likely decrease significantly.

If we are unable to file for approval of Mino-Lok or Hydro-Lido under Section 505(b)(2) of the Federal Food, Drug and Cosmetic Act
or if we are required to generate additional data related to safety and efficacy in order to obtain approval of Mino-Lok under Section
505(b)(2), we may be unable to meet our anticipated development and commercialization timelines.

Our current plans for filing additional NDAs for our product candidates include efforts to minimize the data we will be required to generate
in order to obtain marketing approval for our additional product candidates and therefore possibly reduce the time and cost of development
of a product candidate and obtain a shortened review period for the application. The timeline for filing and review of our planned NDA for
each of Mino-Lok and Hydro-Lido is based upon our plan to submit each such NDA under Section 505(b)(2) of the Federal Food, Drug
and Cosmetic Act, wherein we will rely in part on data in the public domain or elsewhere. Depending on the data that may be required by
the  FDA  for  approval,  some  of  the  data  may  be  related  to  products  already  approved  by  the  FDA.  If  the  data  relied  upon  is  related  to
products already approved by the FDA and covered by third-party patents we would be required to certify that we do not infringe the listed
patents  or  that  such  patents  are  invalid  or  unenforceable.  As  a  result  of  the  certification,  the  third  party  would  have  45  days  from
notification of our certification to initiate an action against us. In the event that an action is brought in response to such a certification, the
approval of our NDA could be subject to a stay of up to 30 months or more while we defend against such a suit. Approval of any product
candidate  under  Section  505(b)(2)  may  therefore  be  delayed  until  patent  exclusivity  expires  or  until  we  successfully  challenge  the
applicability of those patents applicable to our product candidates. Alternatively, we may elect to generate sufficient additional clinical data
so that we no longer rely on data which triggers a potential stay of the approval of any product candidate. Even if no exclusivity periods
apply to an application under Section 505(b)(2), the FDA has broad discretion to require us to generate additional data on the safety and
efficacy  of  our  product  candidates  to  supplement  third-party  data  on  which  we  may  be  permitted  to  rely.  In  either  event,  we  could  be
required, before obtaining marketing approval for such product candidate, to conduct substantial new research and development activities
beyond  those  we  currently  plan  to  engage  in  order  to  obtain  approval  of  that  product  candidate.  Such  additional  new  research  and
development activities would be costly and time consuming.

We may not be able to obtain shortened review of our applications where available, and in any event the FDA may not agree that any of our
product candidates qualify for marketing approval. If we are required to generate additional data to support approval, we may be unable to
meet our anticipated development and commercialization timelines, may be unable to generate the additional data at a reasonable cost, or at
all, and may be unable to obtain marketing approval of that product candidate. In addition, notwithstanding the approval of many products
by the FDA pursuant to Section 505(b)(2), over the last few years, some pharmaceutical companies and others have objected to the FDA’s
interpretation of Section 505(b)(2). If the FDA changes its interpretation of Section 505(b)(2), or if the FDA’s interpretation is successfully
challenged in court, this could delay or even prevent the FDA from approving any Section 505(b)(2) application that we submit.

16

 
 
 
 
 
 
 
 
Even if we receive regulatory approval to commercialize our product candidates, post-approval marketing and promotion of products is
highly regulated by the FDA, and marketing campaigns which violate FDA standards may  result  in  adverse  consequences  including
regulatory enforcement action by the FDA as well as follow-on actions filed by consumers and other end-payers, which could result in
substantial fines, sanctions and damage awards against us, any of which could harm our business.

Post-approval marketing and promotion of drugs, standards and regulations for direct-to-consumer advertising, dissemination of off-label
product  information,  industry-sponsored  scientific  and  educational  activities  and  promotional  activities  via  the  Internet  are  heavily
scrutinized and regulated by the FDA. Drugs may only be marketed for approved indications and in accordance with provisions of the FDA
approved labels. Failure to comply with such requirements may result in adverse publicity, warning letters issued by the FDA, and civil or
criminal penalties.

In the event the FDA discovers post-approval violations, we could face penalties in the future including the FDA’s issuance of a cease and
desist  order,  impounding  of  our  products,  and  civil  or  criminal  penalties. As  a  follow-on  to  such  governmental  enforcement  activities,
consumers and other end-payers of the product may initiate action against us claiming, among other things, fraudulent misrepresentation,
unfair competition, violation of various state consumer protection statues and unjust enrichment. If the plaintiffs in such follow-on actions
are successful, we could be subject to various damages, including compensatory damages, treble damages, punitive damages, restitution,
disgorgement, prejudgment and post-judgment interest on any monetary award, and the reimbursement of the plaintiff’s legal fees and costs,
any of which could have an adverse effect on our revenue, business, financial condition and prospects.

Even  if  we  receive  regulatory  approval  to  commercialize  a  product  candidate,  our  ability  to  generate  revenues  from  any  resulting
product will be subject to a variety of risks, many of which are out of our control.

Even if one of our product candidates obtain regulatory approval, the product may not gain market acceptance among physicians, patients,
healthcare  payers  or  the  medical  community.  The  indication  may  be  limited  to  a  subset  of  the  population  or  we  may  implement  a
distribution  system  and  patient  access  program  that  is  limited.  Coverage  and  reimbursement  of  our  product  candidates  by  third-party
payers,  including  government  payers,  generally  is  also  necessary  for  optimal  commercial  success.  We  believe  that  the  degree  of  market
acceptance  and  our  ability  to  generate  revenues  from  any  approved  produce  candidate  or  acquired  product  will  depend  on  a  number  of
factors, including:

● prevalence and severity of any side effects;

● results of any post-approval studies of the drug;

● potential or perceived advantages or disadvantages over alternative treatments including generics;

● the relative convenience and ease of administration and dosing schedule;

● availability of coverage and reimbursement from government and other third-party payers;

● the willingness of patients to pay out of pocket in the absence of government or third-party coverage;

● product labeling or product insert requirements of the FDA or other regulatory authorities;

● strength of sales, marketing and distribution support;

● price of any future drugs, if approved, both in absolute terms and relative to alternative treatments;

● the effectiveness of our or any future collaborators’ sales and marketing strategies;

● the effect of current and future healthcare laws on our product candidates;

● patient access programs that require patients to provide certain information prior to receiving new and refill prescriptions; and

● requirements for prescribing physicians to complete certain educational programs for prescribing drugs.

17

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
If approved, any product candidate may fail to achieve market acceptance or generate significant revenue to achieve or sustain profitability.
In  addition,  our  efforts  to  educate  the  medical  community  and  third-party  payers  on  the  benefits  of  any  product  candidate  may  require
significant resources and may never be successful.

Even if approved for marketing by applicable regulatory bodies, we will not be able to create a market for any of our products if we fail
to establish marketing, sales and distribution capabilities, or fail to enter into arrangements with third parties.

Our strategy with our product candidates is to outsource to third parties, all or most aspects of the product development process, as well as
marketing, sales and distribution activities. Currently, we do not have any sales, marketing or distribution capabilities. In order to generate
sales of any product candidates that receive regulatory approval, we must either acquire or develop an internal marketing and sales force
with technical expertise and with supporting distribution capabilities or make arrangements with third parties to perform these services for
us.  The  acquisition  or  development  of  a  sales  and  distribution  infrastructure  would  require  substantial  resources,  which  may  divert  the
attention of our management and key personnel and defer our product development efforts. To the extent that we enter into marketing and
sales arrangements with other companies, our revenues will depend on the efforts of others. These efforts may not be successful. If we fail
to develop sales, marketing and distribution channels, or enter into arrangements with third parties, we will experience delays in product
sales and incur increased costs.

The  markets  in  which  we  operate  are  highly  competitive  and  we  may  be  unable  to  compete  successfully  against  new  entrants  or
established companies.

Competition in the pharmaceutical and medical products industries is intense and is characterized by costly and extensive research efforts
and rapid technological progress. We are aware of several pharmaceutical companies also actively engaged in the development of therapies
for at least some of the same conditions we are targeting. Many of these companies have substantially greater research and development
capabilities  as  well  as  substantially  greater  marketing,  financial  and  human  resources  than  we  do.  In  addition,  many  of  these  companies
have  significantly  greater  experience  than  us  in  undertaking  pre-clinical  testing,  human  clinical  trials  and  other  regulatory  approval
procedures.  Our  competitors  may  develop  technologies  and  products  that  are  more  effective  than  those  we  are  currently  marketing  or
researching  and  developing.  Such  developments  could  render  our  product  candidates,  if  approved,  less  competitive  or  possibly  obsolete.
We are also competing with respect to marketing capabilities and manufacturing efficiency, areas in which we have no current capabilities
and  in  which  we  have  limited  experience.  Mergers,  acquisitions,  joint  ventures  and  similar  events  may  also  significantly  increase  the
competition we face. In addition, new developments, including the development of other drug technologies and methods of preventing the
incidence of disease, occur in the pharmaceutical and medical technology industries at a rapid pace. These developments may render our
products and product candidates obsolete or noncompetitive. Compared to us, many of our potential competitors have substantially greater:

● research and development resources, including personnel and technology;

● regulatory resources, experience and expertise;

● product candidate development and clinical trial resources and experience;

● product sourcing, sales and marketing resources and experience;

● experience and expertise in exploitation of intellectual property rights; and

● access to strategic partners and capital resources.

18

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
As  a  result  of  these  factors,  our  competitors  may  obtain  regulatory  approval  of  their  products  more  rapidly  than  we  can  or  may  obtain
patent  protection  or  other  intellectual  property  rights  that  limit  our  ability  to  develop  or  commercialize  our  product  candidates.  Our
competitors may also develop drugs or surgical approaches that are more effective, more useful and less costly than ours and may also be
more  successful  in  manufacturing  and  marketing  their  products.  In  addition,  our  competitors  may  be  more  effective  than  us  in
commercializing their products and as a result, our business and prospects might be materially harmed.

Physicians and patients might not accept and use any of our products for which regulatory approval is obtained.

Even if the FDA approves one of our product candidates, physicians and patients might not accept and use it. Acceptance and use of our
approved products will depend upon a number of factors, including:

● perceptions by members of the health care community, including physicians, about the safety and effectiveness of our products;

● cost-effectiveness of our product relative to competing products or therapies;

● availability of reimbursement for our product from government or other healthcare payers; and

● effective marketing and distribution efforts by us and/or our licensees and distributors, if any.

If our current product candidates are approved, we expect their sales to generate substantially all of our revenues for the foreseeable future,
and as a result, the failure of these products to find market acceptance would harm our business and would require us to seek additional
financing.

Our  two  product  candidates,  Mino-Lok  and  Hydro-Lido,  are  combination  products  consisting  of  components  that  have  each  been
separately  approved  by  the  FDA  for  other  indications  and  which  are  commercially  available  and  marketed  by  other  companies.  Our
approval under 505(b)(2), if received, would not preclude physicians, pharmacists and patients from obtaining individual drug products
and titrating the dosage of these drug products as close to our approved dose as possible.

Our Hydro-Lido product candidate for the treatment of hemorrhoids is a combination product consisting of two drugs, hydrocortisone and
lidocaine, that have each been separately approved by the FDA for other indications and which are commercially available and marketed
by other companies. Hydrocortisone creams are available from strengths ranging from 0.5% to 2.5% and lidocaine creams are also available
in strengths up to 5%. From our market analysis and discussions with a limited number of physicians, we know that patients sometimes
obtain two separate cream products and co-administer them as prescribed, giving them a combination treatment which could be very similar
to what we intend to study and seek approval for. As a branded, FDA-approved product with safety and efficacy data, we intend to price our
product  substantially  higher  than  the  generically  available  individual  creams.  We  will  then  have  to  convince  third-party  payers  and
pharmacy  benefit  managers  of  the  advantages  of  our  product  and  justify  our  premium  pricing.  We  may  encounter  resistance  from  these
entities and will then be dependent on patients’ willingness to pay the premium and not seek alternatives. In addition, pharmacists often
suggest lower cost prescription treatment alternatives to both physicians and patients. Our 505(b)(2) approval and the market exclusivity we
may  receive  will  not  guarantee  that  such  alternatives  will  not  exist,  that  substitution  will  not  occur,  or  that  there  will  be  immediate
acceptance to our pricing by payer formularies.

Our Mino-Lok solution contains minocycline, disodium ethylenediaminetetraacetic acid (edetate), and ethyl alcohol, all of which have been
separately approved by the FDA for other indications, or are used as excipients in other parenteral products.

19

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Our ability to generate product revenues will be diminished if any of our approved products sell for inadequate prices or patients are
unable to obtain adequate levels of reimbursement.

Our ability to commercialize our product candidates, alone or with collaborators, will depend in part on the extent to which reimbursement
will be available from:

● government and health administration authorities;

● private health maintenance organizations and health insurers; and

● other healthcare payers.

Significant uncertainty exists as to the reimbursement status of newly approved healthcare products. Healthcare payers, including Medicare,
are  challenging  the  prices  charged  for  medical  products  and  services.  Government  and  other  healthcare  payers  increasingly  attempt  to
contain healthcare costs by limiting both coverage and the level of reimbursement for drugs. Even if our product candidates are approved
by  the  FDA,  insurance  coverage  might  not  be  available,  and  reimbursement  levels  might  be  inadequate,  to  cover  our  products.  If
government  and  other  healthcare  payers  do  not  provide  adequate  coverage  and  reimbursement  levels  for  our  products,  once  approved,
market acceptance of such products could be reduced. Proposals to modify the current health care system in the U.S. to improve access to
health care and control its costs are continually being considered by the federal and state governments. In March 2010, the U.S. Congress
passed  landmark  healthcare  legislation.  Portions  of  this  legislation  have  been  repealed  recently  and  members  of  the  U.S.  Congress  and
some state legislatures continue to seek to overturn at least some remaining portions of the legislation and we expect they will continue to
review  and  assess  this  legislation  and  possibly  alternative  health  care  reform  proposals.  We  cannot  predict  what  impact  on  federal
reimbursement policies this legislation will have in general or on our business specifically. We cannot predict whether new proposals will
be made or adopted, when they may be adopted or what impact they may have on us if they are adopted.

Health administration authorities in countries other than the U.S. may not provide reimbursement for our products at rates sufficient for us
to achieve profitability, or at all. Like the U.S., these countries have considered health care reform proposals and could materially alter their
government-sponsored  health  care  programs  by  reducing  reimbursement  rates. Any  reduction  in  reimbursement  rates  under  Medicare  or
foreign health care programs could negatively affect the pricing of our products. If we are not able to charge a sufficient amount for our
products, then our margins and our profitability will be adversely affected.

We rely exclusively on third parties to formulate and manufacture our product candidates.

We do not have and do not intend to establish our own manufacturing facilities. Consequently, we lack the physical plant to formulate and
manufacture our own product candidates, which are currently being manufactured entirely by a commercial third party. If any additional
product candidate we might develop or acquire in the future receives FDA approval, we will rely on one or more third-party contractors to
manufacture  our  products.  If,  for  any  reason,  we  become  unable  to  rely  on  our  current  source  or  any  future  source  to  manufacture  our
product candidates, either for clinical trials or, for commercial quantities, then we would need to identify and contract with additional or
replacement  third-party  manufacturers  to  manufacture  compounds  for  preclinical,  clinical  and  commercial  purposes.  We  might  not  be
successful  in  identifying  additional  or  replacement  third-party  manufacturers,  or  in  negotiating  acceptable  terms  with  any  that  we  do
identify. If we are unable to secure and maintain third-party manufacturing capacity, the development and sales of our products and our
financial performance might be materially affected.

In addition, before any of our collaborators can begin to commercially manufacture our product candidates, each must obtain regulatory
approval  of  the  manufacturing  facility  and  process.  Manufacturing  of  drugs  for  clinical  and  commercial  purposes  must  comply  with  the
FDA’s  Current  Good  Manufacturing  Practices,  or  cGMP,  and  applicable  non-U.S.  regulatory  requirements.  The  cGMP  requirements
govern  quality  control  and  documentation  policies  and  procedures.  Complying  with  cGMP  and  non-U.S.  regulatory  requirements  will
require that we expend time, money, and effort in production, recordkeeping, and quality control to assure that the product meets applicable
specifications  and  other  requirements.  Our  contracted  manufacturing  facilities  must  also  pass  a  pre-approval  inspection  prior  to  FDA
approval. Failure to pass a pre- approval inspection might significantly delay FDA approval of our products. If any of our collaborators fails
to comply with these requirements, we would be subject to possible regulatory action which could limit the jurisdictions in which we are
permitted to sell our products. As a result, our business, financial condition, and results of operations might be materially harmed.

20

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Our reliance on a limited number of third-party manufacturers exposes us to the following risks:

● We might be unable to identify manufacturers for commercial supply on acceptable terms or at all because the number of potential
manufacturers is limited and the FDA must approve any replacement contractor. This approval would generally require compliance
inspections.  In  addition,  a  new  manufacturer  would  have  to  be  educated  in,  or  develop  substantially  equivalent  processes  for,
production of our products after receipt of FDA approval, if any;

● Our third-party manufacturers might be unable to formulate and manufacture our products in the volume and of the quality required

to meet our clinical and commercial needs, if any;

● Our contract manufacturers might not perform as agreed or might not remain in the contract manufacturing business for the time

required to supply our clinical trials or to successfully produce, store and distribute our products;

● Currently, our contract manufacturer for our clinical supplies is foreign, which increases the risk of shipping delays and adds the

risk of import restrictions;

● Drug manufacturers are subject to ongoing periodic unannounced inspection by the FDA and corresponding state agencies to ensure
strict  compliance  with  cGMP  and  other  government  regulations  and  corresponding  foreign  standards.  We  do  not  have  complete
control over third-party manufacturers’ compliance with these regulations and standards;

● If any third-party manufacturer makes improvements in the manufacturing process for our products, we might not own, or might

have to share, the intellectual property rights to the innovation with our licensors;

● Operations of our third-party manufacturers or suppliers could be disrupted by conditions unrelated to our business or operations,

including a bankruptcy of the manufacturer or supplier; and

● We might compete with other companies for access to these manufacturers’ facilities and might be subject to manufacturing  delays

if the manufacturers give other clients higher priority than us.

Each of these risks could delay our clinical trials or the approval, if any, of our product candidates by the FDA or any foreign regulatory
agency or the commercialization of our product candidates and could result in higher costs or deprive us of potential product revenues. As
a result, our business, financial condition, and results of operations might be materially harmed.

We are and will be dependent on third-party contract research organizations to conduct all of our future human trials.

We  are  and  will  be  dependent  on  third-party  research  organizations  to  conduct  all  of  our  human  trials  with  respect  to  our  product
candidates,  including  those  that  we  may  develop  in  the  future.  If  we  are  unable  to  obtain  any  necessary  testing  services  on  acceptable
terms, we may not complete our product development efforts in a timely manner. If we rely on third parties for human trials, we may lose
some control over these activities and become too dependent upon these parties. These third parties may not complete testing activities on
schedule or when we so request. We may not be able to secure and maintain suitable research organizations to conduct our human trials.
We are responsible for confirming that each of our clinical trials is conducted in accordance with our general plan and protocol. Moreover,
the  FDA  and  foreign  regulatory  agencies  require  us  to  comply  with  regulations  and  standards,  commonly  referred  to  as  good  clinical
practices,  for  conducting,  recording  and  reporting  the  results  of  clinical  trials  to  assure  that  data  and  reported  results  are  credible  and
accurate and that the trial participants are adequately protected. Our reliance on third parties does not relieve us of these responsibilities
and  requirements.  If  these  third  parties  do  not  successfully  carry  out  their  contractual  duties  or  regulatory  obligations  or  meet  expected
deadlines, if the third parties need to be replaced or if the quality or accuracy of the data they obtain is compromised due to the failure to
adhere to our clinical protocols or regulatory requirements or for other reasons, our preclinical development activities or clinical trials may
be extended, delayed, suspended or terminated, and we may not be able to obtain regulatory approval for our future product candidates.

21

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Any termination or breach by or conflict with our strategic partners or licensees could harm our business.

If we or any of our collaborators or licensees fail to renew or terminate any of our collaboration or license agreements or if either party fails
to  satisfy  its  obligations  under  any  of  our  collaboration  or  license  agreements  or  complete  them  in  a  timely  manner,  we  could  lose
significant sources of revenue, which could result in volatility in our future revenue. In addition, our agreements with our collaborators and
licensees  may  have  provisions  that  give  rise  to  disputes  regarding  the  rights  and  obligations  of  the  parties.  These  and  other  possible
disagreements could lead to termination of the agreement or delays in collaborative research, development, supply or commercialization of
certain products, or could require or result in litigation or arbitration. Any such conflicts with our collaborators could reduce our ability to
obtain  future  collaboration  agreements  and  could  have  a  negative  impact  on  our  relationship  with  existing  collaborators,  adversely
affecting our business and revenues. Finally, any of our collaborations or license agreements may prove to be unsuccessful.

We might seek to grow and develop our business through acquisitions of or investment in new or complementary businesses, products
or technologies, and the failure to manage these acquisitions or investments, or the failure to integrate them with our existing business,
could have a material adverse effect on us.

We might consider opportunities to acquire or invest in other technologies, products and businesses that might enhance our capabilities or
complement  our  current  product  candidates.  Potential  and  completed  acquisitions  and  strategic  investments  involve  numerous  risks,
including potential problems or issues associated with the following:

● assimilating the purchased technologies, products or business operations;

● maintaining uniform standards, procedures, controls and policies;

● unanticipated costs associated with the acquisition or investment;

● diversion of our management’s attention from our preexisting business;

● maintaining or obtaining the necessary regulatory approvals or complying with regulatory standards; and

● adverse effects on existing business operations.

We have no current commitments with respect to any acquisition or investment in other technologies or businesses. We do not know if we
will  identify  suitable  acquisitions,  whether  we  will  be  able  to  successfully  complete  any  acquisitions,  or  whether  we  will  be  able  to
successfully integrate any acquired product, technology or business into our business or retain key personnel, suppliers or collaborators.

Our  ability  to  successfully  develop  our  business  through  acquisitions  would  depend  on  our  ability  to  identify,  negotiate,  complete  and
integrate  suitable  target  businesses  or  technologies  and  obtain  any  necessary  financing.  These  efforts  could  be  expensive  and  time
consuming and might disrupt our ongoing operations. If we are unable to efficiently integrate any acquired business, technology or product
into our business, our business and financial condition might be adversely affected.

If we are unable to retain or hire additional qualified personnel, our ability to grow our business might be harmed.

We utilize the services of a clinical management team on part-time basis to assist us in managing our ongoing Phase 2 and Phase 3 trials
and intend to do so for future trials. While we believe this will provide us with sufficient staffing for our current and future development
efforts, we will need to hire or contract with additional qualified personnel with expertise in preclinical testing, clinical research and testing,
government regulation, formulation and manufacturing and sales and marketing in connection with the continued development, regulatory
approval  and  commercialization  of  our  product  candidates.  We  compete  for  qualified  individuals  with  numerous  pharmaceutical  and
biopharmaceutical companies, universities and other research institutions. Competition for these individuals is intense, and we cannot be
certain that our search for such personnel will be successful. Attracting and retaining qualified personnel will be critical to our success. In
addition, we may be unable to attract and retain those qualified officers, directors and members of board committees required to provide for
effective management. If we are unable to attract and retain qualified employees, officers and directors, the management and operation of
our business could be adversely affected.

22

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
We expect to need to increase the size of our organization to further develop our product candidates, and we may experience difficulties
in managing growth.

We will need to manage our anticipated growth and increased operational activity. Our personnel, systems and facilities currently in place
may not be adequate to support this future growth. Our need to effectively execute our growth strategy will require that we:

● manage our regulatory trials effectively;

● attract and motivate sufficient numbers of talented employees;

● manage our  internal  development  efforts  effectively  while  complying  with  our  contractual  obligations  to  licensors,  licensees,

contractors, collaborators and other third parties;

● develop internal sales and marketing capabilities or establish collaborations with third parties with such capabilities;

● commercialize our product candidates; and

● improve our operational, financial and management controls, reporting systems and procedures.

This planned future growth could place a strain on our administrative and operational infrastructure and may require our management to
divert  a  disproportionate  amount  of  its  attention  away  from  our  day-to-day  activities.  We  may  not  be  able  to  effectively  manage  the
expansion of our operations or recruit and train additional qualified personnel, which may result in weaknesses in our infrastructure, and
give rise to operational mistakes, loss of business opportunities, loss of employees and reduced productivity among remaining employees.
We may not be able to make improvements to our management information and control systems in an efficient or timely manner and may
discover  deficiencies  in  existing  systems  and  controls.  If  our  management  is  unable  to  effectively  manage  our  expected  growth,  our
expenses may increase more than expected, our ability to generate or increase our revenues could be reduced and we may not be able to
implement our business strategy. Our future financial performance and our ability to compete effectively will depend, in part, on our ability
to effectively manage any future growth.

We are subject to extensive and costly government regulation.

Risks Related to Our Regulatory and Legal Environment

Product  candidates  and  approved  products  such  as  ours  are  subject  to  extensive  and  rigorous  domestic  government  regulation  including
regulation  by  the  FDA,  the  Centers  for  Medicare  and  Medicaid  Services,  other  divisions  of  the  U.S.  Department  of  Health  and  Human
Services,  the  U.S.  Department  of  Justice,  state  and  local  governments,  and  their  respective  foreign  equivalents.  The  FDA  regulates  the
research,  development,  preclinical  and  clinical  testing,  manufacture,  safety,  effectiveness,  record  keeping,  reporting,  labeling,  storage,
approval,  advertising,  promotion,  sale,  distribution,  import,  and  export  of  pharmaceutical  products.  The  FDA  regulates  small  molecule
chemical entities, whether administered orally, topically or by injection, as drugs, subject to an NDA, under the Federal Food, Drug, and
Cosmetic  Act.  If  our  product  candidates  are  to  be  marketed  abroad,  they  will  also  be  subject  to  extensive  regulation  by  foreign
governments,  whether  or  not  they  have  obtained  FDA  approval.  Such  foreign  regulation  might  be  equally  or  more  demanding  than
corresponding U.S. regulation. Government regulation substantially increases the cost and risk of researching, developing, manufacturing,
and selling our products. The regulatory review and approval process, which includes preclinical testing and clinical trials of each product
candidate,  is  lengthy,  expensive,  and  uncertain.  Our  collaborators  or  we  must  obtain  and  maintain  regulatory  authorization  to  conduct
clinical trials and approval for each product we intend to market, and the manufacturing facilities used for the products must be inspected
and meet legal requirements. Securing regulatory approval requires submitting extensive preclinical and clinical data and other supporting
information  for  each  proposed  therapeutic  indication  in  order  to  establish  the  product’s  safety  and  efficacy  for  each  intended  use.  The
development and approval process might take many years, requires substantial resources, and might never lead to the approval of a product.
Even  if  we  are  able  to  obtain  regulatory  approval  for  a  particular  product,  the  approval  might  limit  the  indicated  medical  uses  for  the
product,  limit  our  ability  to  promote,  sell,  and  distribute  the  product,  require  that  we  conduct  costly  post-marketing  surveillance,  and/or
require  that  we  conduct  ongoing  post-marketing  studies.  Material  changes  to  an  approved  product,  such  as,  for  example,  manufacturing
changes  or  revised  labeling,  might  require  further  regulatory  review  and  approval.  Once  obtained,  any  approvals  might  be  withdrawn,
including, for example, if there is a later discovery of previously unknown problems with the product, such as a previously unknown safety
issue.

23

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
If  we,  our  collaborators,  or  our  contract  manufacturers  fail  to  comply  with  applicable  regulatory  requirements  at  any  stage  during  the
regulatory  process,  such  noncompliance  could  result  in,  among  other  things,  delays  in  the  approval  of  applications  or  supplements  to
approved applications; refusal of a regulatory authority, including the FDA, to review pending market approval applications or supplements
to  approved  applications;  warning  letters;  fines;  import  and  export  restrictions;  product  recalls  or  seizures;  injunctions;  total  or  partial
suspension of production; civil penalties; withdrawals of previously approved marketing applications or licenses; recommendations by the
FDA or other regulatory authorities against governmental contracts; and/or criminal prosecutions.

We might not obtain the necessary U.S. regulatory approvals to commercialize any product candidates.

We  cannot  assure  you  that  we  will  receive  the  approvals  necessary  to  commercialize  for  sale  any  product  candidates  we  are  currently
developing or that we may acquire or develop in the future. We will need FDA approval to commercialize our product candidates in the
U.S.  In  order  to  obtain  FDA  approval  of  any  product  candidate,  we  must  submit  to  the  FDA  an  NDA  demonstrating  that  the  product
candidate is safe for humans and effective for its intended use. This demonstration requires significant research, pre-clinical studies, and
clinical  trials.  Satisfaction  of  the  FDA’s  regulatory  requirements  typically  takes  many  years,  depends  upon  the  type,  complexity  and
novelty of the product candidate and requires substantial resources for research, development and testing. We cannot predict whether our
research  and  clinical  approaches  will  result  in  additional  drugs  that  the  FDA  considers  safe  for  humans  and  effective  for  their  indicated
uses. The FDA has substantial discretion in the product approval process and might require us to conduct additional pre-clinical and clinical
testing,  perform  post-marketing  studies  or  otherwise  limit  or  impose  conditions  on  any  additional  approvals  we  obtain.  The  approval
process might also be delayed by changes in government regulation, future legislation or administrative action or changes in FDA policy
that occur prior to or during our regulatory review. Delays in obtaining regulatory approvals might:

● delay commercialization of, and our ability to derive product revenues from, our product candidates;

● impose costly procedures on us; and

● diminish any competitive advantages that we might otherwise enjoy.

Even if we comply with all FDA requests, the FDA might ultimately reject one or more of our NDAs. We cannot be sure that we will ever
obtain regulatory clearance for our product candidates. Failure to obtain FDA approval of our product candidates will severely undermine
our  business  by  leaving  us  without  saleable  products,  and  therefore  without  any  potential  sources  of  revenues,  until  another  product
candidate could be developed or obtained. There is no guarantee that we will ever be able to develop or acquire any product candidate.

Following  any  regulatory  approval  of  any  product  candidates,  we  will  be  subject  to  ongoing  regulatory  obligations  and  restrictions,
which may result in significant expense and limit our ability to commercialize our potential drugs.

If one of our product candidates is approved by the FDA or by a foreign regulatory authority, we will be required to comply with extensive
regulations  for  product  manufacturing,  labeling,  packaging,  adverse  event  reporting,  storage,  distribution,  advertising,  promotion  and
record keeping. Regulatory approvals may also be subject to significant limitations on the indicated uses or marketing of the products or to
whom  and  how  we  may  distribute  our  products.  Even  if  U.S.  regulatory  approval  is  obtained,  the  FDA  may  still  impose  significant
restrictions  on  a  drug’s  indicated  uses  or  marketing  or  impose  ongoing  requirements  for  potentially  costly  post-approval  studies.  For
example,  the  label  ultimately  approved  for  our  products,  if  any,  may  include  restrictions  on  use,  including  restrictions  based  on  level  of
obesity  and  duration  of  treatment.  If  so,  we  may  be  subject  to  ongoing  regulatory  obligations  and  restrictions,  which  may  result  in
significant expense and limit our ability to commercialize our products. The FDA could also require a registry to track the patients utilizing
the  drug  or  implement  a  Risk  Evaluation  and  Mitigation  Strategy,  or  REMS,  that  could  restrict  access  to  the  drug,  reduce  our  revenues
and/or  increase  our  costs.  Potentially  costly  post-marketing  clinical  studies  may  be  required  as  a  condition  of  approval  to  further
substantiate safety or efficacy, or to investigate specific issues of interest to the regulatory authority.

24

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Manufacturers of pharmaceutical products and their facilities are subject to continual review and periodic inspections by the FDA and other
regulatory  authorities  for  compliance  with  current  good  manufacturing  practices,  or  cGMP,  regulations,  which  include  requirements
relating  to  quality  control  and  quality  assurance  as  well  as  the  corresponding  maintenance  of  records  and  documentation.  Further,
regulatory agencies must approve these manufacturing facilities before they can be used to manufacture our future approved products, if
any, and these facilities are subject to ongoing regulatory inspections. In addition, regulatory agencies subject a pharmaceutical product, its
manufacturer  and  the  manufacturer’s  facilities  to  continual  review  and  inspections.  The  subsequent  discovery  of  previously  unknown
problems with a product, including adverse events of unanticipated severity or frequency, or problems with the facility where the product is
manufactured, may result in restrictions on the marketing of that product, up to and including, withdrawal of the product from the market.
If the manufacturing facilities of our suppliers fail to comply with applicable regulatory requirements, it could result in regulatory action
and additional costs to us. Failure to comply with applicable FDA and other regulatory requirements may, either before or after product
approval, if any, subject our company to administrative or judicially imposed sanctions, including:

● issuance of Form 483 notices, warning letters and adverse publicity by the FDA or other regulatory agencies;

● imposition of fines and other civil penalties due to product liability or other issues;

● injunctions, suspensions or revocations of regulatory approvals;

● suspension of any ongoing clinical trials;

● total or partial suspension of manufacturing;

● delays in commercialization;

● refusal by the FDA to approve pending applications or supplements to approved applications filed by us or our collaborators;

● refusals to permit medical products to be imported into or exported from the U.S.;

● restrictions on operations, including costly new manufacturing requirements;

● product recalls or seizures; and

● criminal prosecutions.

In addition, the law or regulatory policies governing pharmaceutical products may change. New statutory requirements may be enacted or
additional regulations may be enacted that could prevent or delay regulatory approval of our product candidates. Contract manufacturing
organizations, or CMOs, and their vendors or suppliers may also face changes in regulatory requirements from governmental agencies in
the U.S. and other countries. We cannot predict the likelihood, nature, extent or effects of government regulation that may arise from future
legislation or administrative action, either in the U.S. or elsewhere. If we are not able to maintain regulatory compliance, we might not be
permitted to market any future approved products and our business could suffer.

25

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
We could be forced to pay substantial damage awards if product liability claims that may be brought against us are successful.

The use of any of our product candidates in clinical trials, and the sale of any approved products, may expose us to liability claims and
financial losses resulting from the use or sale of our products. We have obtained limited product liability insurance coverage for our clinical
trials of $2.0 million per occurrence and in the aggregate, subject to a deductible of $50,000 per occurrence. There can be no assurance that
our  existing  insurance  coverage  will  extend  to  any  other  products  in  the  future. Any  product  liability  insurance  coverage  may  not  be
sufficient  to  satisfy  all  liabilities  resulting  from  product  liability  claims. A  successful  claim  may  prevent  us  from  obtaining  adequate
product liability insurance in the future on commercially desirable terms, if at all. Even if a claim is not successful, defending such a claim
would  be  time  consuming  and  expensive,  may  damage  that  product’s  and  our  reputations  in  the  marketplace,  and  would  likely  divert
management’s attention, any of which could have a material adverse effect on our company.

Our business depends on protecting our intellectual property.

Risks Related to our Intellectual Property

If  we  do  not  obtain  protection  for  our  intellectual  property  rights,  our  competitors  might  be  able  to  take  advantage  of  our  research  and
development efforts to develop competing products. Our success, competitive position and future revenues, if any, depend in part on our
ability  and  the  abilities  of  our  licensors  to  obtain  and  maintain  patent  protection  for  our  products,  methods,  processes  and  other
technologies,  to  preserve  our  trade  secrets,  to  prevent  third  parties  from  infringing  on  our  proprietary  rights  and  to  operate  without
infringing the proprietary rights of third parties. We anticipate filing additional patent applications both in the U.S. and in other countries,
as appropriate. However, the patent process is subject to numerous risks and uncertainties, and there can be no assurance that we will be
successful in protecting our products by obtaining and defending patents. These risks and uncertainties include the following:

● Our patent rights might be challenged, invalidated, or circumvented, or otherwise might not provide any competitive advantage;

● Our competitors,  many  of  which  have  substantially  greater  resources  than  we  do  and  many  of  which  might  make  significant
investments in  competing  technologies,  might  seek,  or  might  already  have  obtained,  patents  that  will  limit,  interfere  with,  or
eliminate our ability to make, use, and sell our potential products either in the U.S. or in international markets;

● Countries other than the U.S. might have less restrictive patent laws than those upheld by U.S. courts, allowing foreign competitors

the ability to exploit these laws to create, develop, and market competing products; and

● As a matter of public policy regarding worldwide health concerns, there might be significant pressure on the U.S. government and
other  international  governmental  bodies  to  limit  the  scope  of  patent  protection  both  inside  and  outside  the  U.S.  for  disease
treatments that prove successful.

In  addition,  the  U.S.  Patent  and  Trademark  Office  and  patent  offices  in  other  jurisdictions  have  often  required  that  patent  applications
concerning  pharmaceutical  and/or  biotechnology-related  inventions  be  limited  or  narrowed  substantially  to  cover  only  the  specific
innovations exemplified in the patent application, thereby limiting the scope of protection against competitive challenges. Thus, even if we
or our licensors are able to obtain patents, the patents might be substantially narrower than anticipated.

Because the time period from filing a patent application to the issuance, if ever, of the patent is often more than three years and because any
regulatory approval and marketing for a pharmaceutical product often occurs several years after the related patent application is filed, the
resulting market exclusivity afforded by any patent on our drug candidates and technologies will likely be substantially less than 20 years.
In  the  United  States,  the  European  Union  and  some  other  jurisdictions,  patent  term  extensions  are  available  for  certain  delays  in  either
patent office proceedings or marketing and regulatory approval processes. However, due to the specific requirements for obtaining these
extensions,  there  is  no  assurance  that  our  patents  will  be  granted  extensions  even  if  we  encounter  significant  delays  in  patent  office
proceedings or marketing and regulatory approval.

26

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Patent and other intellectual property protection is crucial to the success of our business and prospects, and there is a substantial risk that
such protections will prove inadequate. Our business and prospects will be harmed if these protections prove insufficient.

We rely on trade secret protections through confidentiality agreements with our employees, customers and other parties, and the breach
of these agreements could adversely affect our business and prospects.

We  rely  on  trade  secrets,  which  we  seek  to  protect,  in  part,  through  confidentiality  and  non-disclosure  agreements  with  our  employees,
collaborators,  suppliers,  and  other  parties.  There  can  be  no  assurance  that  these  agreements  will  not  be  breached,  that  we  would  have
adequate remedies for any such breach or that our trade secrets will not otherwise become known to or independently developed by our
competitors.  We  might  be  involved  from  time  to  time  in  litigation  to  determine  the  enforceability,  scope  and  validity  of  our  proprietary
rights. Any such litigation could result in substantial cost and divert management’s attention from our operations.

If  we  infringe  the  rights  of  third  parties  we  might  have  to  forego  developing  and/or  selling  any  approved  products,  pay  damages,  or
defend against litigation.

If  our  product  candidates,  methods,  processes  and  other  technologies  infringe  the  proprietary  rights  of  other  parties,  we  could  incur
substantial costs and we might have to:

● obtain licenses, which might not be available on commercially reasonable terms, if at all;

● abandon an infringing product candidate;

● redesign our products or processes to avoid infringement;

● stop using the subject matter claimed in the patents held by others;

● pay damages; and/or

● defend litigation  or  administrative  proceedings  which  might  be  costly  whether  we  win  or  lose,  and  which  could  result  in  a

substantial diversion of our financial and management resources.

Any of these events could substantially harm our earnings, financial condition and operations.

Risks Related to Our Securities

Our failure to meet the continued listing requirements of Nasdaq could result in a delisting of our common stock and warrants.

Our common stock and warrants are currently listed on the Nasdaq Capital Market. If we fail to satisfy the continued listing requirements
of Nasdaq, such as the corporate governance requirements or the minimum closing bid price requirement, Nasdaq may take steps to delist
our common stock and warrants. Such a delisting would likely have a negative effect on the price of our common stock and warrants and
would impair your ability to sell or purchase our common stock and warrants when you wish to do so. In addition, we could face significant
material adverse consequences, including:

● a limited availability of market quotations for our securities;

● a limited amount of news and analyst coverage for us; and

● a decreased ability to issue additional securities or obtain additional financing in the future.

27

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
In  the  event  of  a  delisting,  we  would  take  actions  to  restore  our  compliance  with  Nasdaq’s  listing  requirements,  but  we  can  provide  no
assurance that any such action taken by us would allow our common stock to become listed again, stabilize the market price or improve the
liquidity  of  our  common  stock,  prevent  our  common  stock  from  dropping  below  the  Nasdaq  minimum  bid  price  requirement  or  prevent
future non-compliance with Nasdaq’s listing requirements.

If  our  common  stock  were  delisted  and  determined  to  be  a  “penny  stock,”  a  broker-dealer  may  find  it  more  difficult  to  trade  our
common stock and an investor may find it more difficult to acquire or dispose of our common stock in the secondary market.

If our common stock were removed from listing with Nasdaq, it may be subject to the so-called “penny stock” rules. The SEC has adopted
regulations  that  define  a  “penny  stock”  to  be  any  equity  security  that  has  a  market  price  per  share  of  less  than  $5.00,  subject  to  certain
exceptions, such as any securities listed on a national securities exchange. For any transaction involving a “penny stock,” unless exempt,
the rules impose additional sales practice requirements on broker-dealers, subject to certain exceptions. If our common stock were delisted
and determined to be a “penny stock,” a broker-dealer may find it more difficult to trade our common stock and an investor may find it
more difficult to acquire or dispose of our common stock on the secondary market.

If we fail to maintain an effective system of internal controls, we may not be able to accurately report our financial results or detect
fraud.  Consequently,  shareholders  could  lose  confidence  in  our  financial  reporting  and  this  may  decrease  the  trading  price  of  our
common stock.

We are subject to the reporting requirements of the Exchange Act, Sarbanes-Oxley Act of 2002, or SOX, and Nasdaq rules and regulations.
SOX  requires,  among  other  things,  that  we  maintain  effective  disclosure  controls  and  procedures  and  internal  control  over  financial
reporting. We perform system and process evaluation and testing of our internal control over financial reporting to allow management to
report  on  the  effectiveness  of  our  internal  controls  over  financial  reporting  in  our Annual  Report  on  Form  10-K  filing  for  that  year,  as
required by Section 404 of SOX.. We previously had identified material weaknesses in our internal control over financial reporting related
to ineffective separation of duties due to our limited finance staff, our reliance on consultants to assist with the financial reporting function
and a lack of documented policies and procedures, which weaknesses were reported in fiscal 2016 and 2017. While we remediated these
material  weaknesses  as  of  September  30,  2018,  such  that  management  has  determined  that  our  internal  controls  over  financial  reporting
were effective as of that date, we cannot assure that, in the future, a material weakness or significant deficiency will not exist or otherwise
be discovered. If that were to happen, it could harm our operating results and cause shareholders to lose confidence in our reported financial
information. Any such loss of confidence would have a negative effect on the trading price of our securities.

The price of our securities may become volatile, which could lead to losses by shareholders and costly securities litigation.

The trading price of our securities is likely to be highly volatile and could fluctuate in response to factors such as:

● actual or anticipated variations in our operating results;

● announcements of developments by us or our competitors;

● the completion and/or results of our clinical trials;

● regulatory actions regarding our product candidates or any approved products;

● announcements by us or our competitors of significant acquisitions, strategic partnerships, joint ventures or capital commitments;

● adoption of new accounting standards affecting our industry;

● additions or departures of key personnel;

● introduction of new products by us or our competitors;

● sales of our common stock or other securities in the open market or in private placements; and

● other events or factors, many of which are beyond our control.

The stock market is subject to significant price and volume fluctuations. In the past, following periods of volatility in the market price of a
company’s securities, securities class action litigation has often been initiated against such a company. Any such litigation initiated against
us,  whether  or  not  successful,  could  result  in  substantial  costs  and  diversion  of  our  management’s  attention  and  resources,  which  could
harm our business and financial condition.

28

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
You may experience dilution of your ownership interests because of the future issuance of additional shares of our common stock or
securities convertible into common stock.

In the future, to finance our operations, including possible acquisitions or strategic transactions, we may issue equity securities, resulting in
the dilution of the ownership interests of our present stockholders. We are currently authorized to issue an aggregate of 200,000,000 shares
of  common  stock  and  10,000,000  shares  of  preferred  stock. As  of  December  1,  2018,  there  were  17,798,791  shares  of  common  stock
outstanding, 15,193,192 shares underlying warrants with a weighted average exercise price of $2.21 per share (including 721,569 shares
underlying pre-funded warrants with an exercise price of $0.01), and 1,601,039 shares underlying options with a weighted average exercise
price  of  $4.35  per  share.  We  may  also  issue  additional  shares  of  our  common  stock  or  other  securities  that  are  convertible  into  or
exercisable for common stock in connection with hiring or retaining employees, or for other business purposes. The future issuance of any
such additional shares of common stock or common stock equivalents may create downward pressure on the trading price of our common
stock.

The common stock is controlled by insiders.

As  of  December  1,  2018,  our  executive  officers  and  directors  beneficially  owned  approximately  58.5%  of  our  outstanding  shares  of
common stock. Such concentrated control of our company may adversely affect the price of our common stock. If you acquire common
stock, you may have no effective voice in the management of our company. Sales by our directors and executive officers or their affiliates,
along with any other market transactions, could adversely affect the market price of our common stock.

We do not intend to pay dividends for the foreseeable future.

We have paid no dividends on our common stock to date and we do not anticipate that any dividends will be paid to holders of our common
stock in the foreseeable future. While our future dividend policy will be based on the operating results and capital needs of the business, it
is currently anticipated that any earnings will be retained to finance our future expansion and for the implementation of our business plan.
The lack of a dividend can further affect the market value of our stock, and could significantly affect the value of any investment in our
company.

Our Certificate of Incorporation allows for our Board of Directors to create new series of preferred stock without further approval by
our stockholders, which could adversely affect the rights of the holders of the common stock.

Our Board of Directors has the authority to issue up to 10,000,000 shares of preferred stock and to fix and determine the relative rights and
preferences  of  any  such  preferred  stock  without  further  stockholder  approval. As  a  result,  our  Board  of  Directors  could  authorize  the
issuance  of  a  series  of  preferred  stock  that  would  grant  preferential  rights  to  our  assets  upon  liquidation,  the  right  to  receive  dividend
payments before dividends are distributed to the holders of common stock and the right to the redemption of the preferred shares, together
with a premium, prior to the redemption of the common stock. In addition, our Board of Directors could authorize the issuance of a series
of preferred stock that has greater voting power than the common stock or that is convertible into our common stock, which could decrease
the relative voting power of the common stock or result in dilution to our existing stockholders.

29

 
 
 
 
 
 
 
 
 
 
There is not an active liquid trading market for our common stock.

While our common stock is listed on the Nasdaq National Market, there has not been a regular active trading market in our common stock,
and we cannot give any assurance that an active trading market will develop. If an active market for our common stock were to develop,
there is a significant risk that the stock price could fluctuate dramatically in the future in response to any of the following factors, some of
which are beyond our control:

● the results of our preclinical and clinical trials;

● announcements by  us  or  our  competitors  of  significant  contracts,  acquisitions,  strategic  partnerships,  joint  ventures  or  capital

commitments;

● general economic slowdowns;

● issuances by us or resales by others of large amounts of our common stock;

● variations in our quarterly operating results; and

● announcements that our revenue or income are below analysts’ expectations.

Sales of a substantial number of shares of our common stock in the public market, or the perception such sales may occur, could cause
the market price of shares of our common stock to fall.

Sales of a substantial number of shares of our common stock in the public market could occur at any time. These sales, or the perception in
the market of such sales or that the holders of a large number of shares intend to sell shares, could reduce the market price of our shares of
our common stock. As of December 1, 2018, we had 17,798,791 shares of common stock outstanding. This includes registered shares of
common  stock  as  well  as  4,903,645  shares  of  our  common  stock  which  are  available  for  resale  under  Rule  144  of  the  Securities Act  of
1933, as amended, or the Securities Act.

Item 1B. Unresolved Staff Comments

Not Applicable

Item 2. Properties

We lease our offices at 11 Commerce Drive, Cranford, New Jersey 07016. The lease runs until April 30, 2019. The annual rent is $26,000.

Item 3. Legal Proceedings

We are not involved in any litigation that we believe could have a material adverse effect on our financial position or results of operations.
There  is  no  action,  suit,  proceeding,  inquiry  or  investigation  before  or  by  any  court,  public  board,  government  agency,  self-regulatory
organization or body pending or, to the knowledge of our executive officers, threatened against or affecting our company or our officers or
directors in their capacities as such.

In the future, we might from time to time become involved in litigation relating to claims arising from our ordinary course of business.

Item 4. Mine Safety Disclosures

Not applicable.

30

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Item 5. Market for Registrant’s Common Equity, Related Stockholder Matters and Issuer Purchases of Equity Securities

PART II

Market Information

Our common stock trades on the Nasdaq Capital Market under the symbol “CTXR”.

Recent Sales of Unregistered Securities

None.

Issuer Purchases of Equity Securities

We did not make any purchases of our Common Stock during the three months ended September 30, 2018, which is the fourth quarter of
our fiscal year.

Item 6. Selected Financial Data

Not required.

Item 7. Management’s Discussion and Analysis of Financial Condition and Results of Operations

The  following  discussion  and  analysis  of  our  financial  condition  and  results  of  operations  should  be  read  together  with  our  financial
statements  and  related  notes  included  elsewhere  in  this  annual  report  on  Form  10-K.  Management’s  discussion  and  analysis  contains
forward-looking  statements,  such  as  statements  of  our  plans,  objectives,  expectations  and  intentions.  Any  statements  that  are  not
statements of historical fact are forward-looking statements. When used, the words “believe,” “plan,” “intend,” “anticipate,” “target,”
“estimate,” “expect” and the like, and/or future tense or conditional constructions (“will,” “may,” “could,” “should,” etc.), or similar
expressions, identify certain of these forward-looking statements. These forward-looking statements are subject to risks and uncertainties
including those under “Risk Factors” in Item 1A in this Form 10-K that could cause actual results or events to differ materially from those
expressed  or  implied  by  the  forward-looking  statements.  Our  actual  results  and  the  timing  of  events  could  differ  materially  from  those
anticipated in these forward-looking statements as a result of several factors. The Company does not undertake any obligation to update
forward-looking statements to reflect events or circumstances occurring after the filing date of this report.

Historical Background

Citius  Pharmaceuticals,  Inc.  (“Citius”  or  the  “Company”)  is  a  specialty  pharmaceutical  company  dedicated  to  the  development  and
commercialization  of  critical  care  products  targeting  unmet  needs  with  a  focus  on  anti-infectives,  cancer  care  and  unique  prescription
products. On September 12, 2014, we acquired Citius Pharmaceuticals, LLC as a wholly-owned subsidiary.

On March 30, 2016, the Company acquired all of the outstanding stock of Leonard-Meron Biosciences, Inc. (“LMB”) by issuing 1,942,456
shares of its common stock. As of March 30, 2016, the stockholders of LMB received approximately 41% of the issued and outstanding
common  stock  of  the  Company.  In  addition,  the  Company  converted  the  outstanding  common  stock  warrants  of  LMB  into  243,020
common stock warrants of the Company and converted the outstanding common stock options of LMB into 77,252 common stock options
of the Company. Management estimated the fair value of the purchase consideration to be $19,015,073.

In connection with the acquisition, the Company acquired net assets of $17,428,277, including identifiable intangible assets of $19,400,000
related to in-process research and development. The Company recorded goodwill of $1,586,796 for the excess of the purchase price over
the net assets acquired.

31

 
 
 
 
 
    
 
  
 
 
 
 
 
 
 
 
 
 
In-process research and development represents the value of LMB’s leading drug candidate, which is an antibiotic solution used to treat
catheter-related bloodstream infections.  Goodwill represents the value of LMB’s industry relationships and its assembled workforce. In-
process  research  and  development  is  expected  to  be  amortized  on  a  straight-line  basis  over  a  period  of  eight  years  commencing  upon
revenue generation. Goodwill will not be amortized, but will be tested at least annually for impairment.

Through  September  30,  2018,  the  Company  has  devoted  substantially  all  of  its  efforts  to  product  development,  raising  capital,  building
infrastructure  through  strategic  alliances  and  coordinating  activities  relating  to  its  proprietary  products.  On  July  1,  2016,  the  Company
announced  that  it  was  discontinuing  Suprenza,  its  first  commercial  product,  for  strategic  reasons  and  not  due  to  safety  or  regulatory
concerns, and was focusing on the Phase 3 development of Mino-Lok, an antibiotic lock solution used to treat patients with catheter-related
bloodstream infections, and the Phase 2b development of Hydro-Lido for hemorrhoids. The Company has not yet realized any revenues
from its operations. 

Patent and Technology License Agreement

LMB has a patent and technology license agreement with Novel Anti-Infective Therapeutics, Inc., (“NAT”) to develop and commercialize
Mino-Lok on an exclusive worldwide sub licensable basis, as amended. Since May 2014, LMB has paid an annual maintenance fee, which
began  at  $30,000  and  that  increases  over  five  years  to  $90,000,  where  it  is  to  remain  until  commercial  sales  of  a  product  subject  to  the
license commence. LMB will also pay annual royalties on net sales of licensed products, with royalties ranging from the mid-single digits
to the low double digits. In limited circumstances in which the licensed product is not subject to a valid patent claim and a competitor is
selling  a  competing  product,  the  royalty  rate  is  in  the  low-single  digits. After  a  commercial  sale  is  obtained,  LMB  must  pay  minimum
aggregate annual royalties that increase in subsequent years. LMB must also pay NAT up to $1,390,000 upon achieving specified regulatory
and sales milestones. Finally, LMB must pay NAT a specified percentage of payments received from any sub licensees.

Results of Operations for Year Ended September 30, 2018 compared to Year Ended September 30, 2017

Revenues

Operating expenses:

Research and development
General and administrative
Stock-based compensation – general and administrative

Total operating expenses

Operating loss

Gain on extinguishment of liability
Other income
Gain on revaluation of derivative warrant liability
Interest expense

Net loss

Revenues

Year Ended 
September 30,
2018

Year Ended 
September 30,
2017

  $

-    $

- 

6,562,925     
6,446,517     
779,701     
13,789,143     
(13,789,143)    
450,000     
818,343     
-     
(15,838)    

2,936,252 
6,063,439 
986,620 
9,986,311 
(9,986,311)
- 
- 
452,147 
(850,789)
  $ (12,536,638)   $ (10,384,953)

We did not generate any revenues for the years ended September 30, 2018 and 2017.

Research and Development Expenses

For  the  year  ended  September  30,  2018,  research  and  development  expenses  were  $6,562,925  as  compared  to  $2,936,252  for  the  year
ended  September  30,  2017.  The  $3,626,673  increase  in  2018  was  primarily  due  to  the  ongoing  Phase  3  trial  of  Mino-Lok  which
commenced during the quarter ended March 31, 2018. Research and development costs for Mino-Lok were $6,121,150 for the year ended
September  30,  2018  as  compared  to  $2,688,937  for  the  year  ended  September  30,  2017,  an  increase  of  $3,432,213.  Research  and
development costs for our product candidate for the treatment of hemorrhoids were $441,775 for the year ended September 30, 2018 as
compared to $247,315 for the year ended September 30, 2017, an increase of $194,460. We expect that research and development expenses
will continue to increase as we continue to focus on and expand our Phase 3 trial of Mino-Lok. We are actively seeking additional capital in
order to fund our research and development efforts.

32

 
 
 
 
 
 
 
 
 
   
 
 
   
      
  
   
      
  
   
   
   
   
   
   
   
   
   
 
 
 
 
 
General and Administrative Expenses

For  the  year  ended  September  30,  2018,  general  and  administrative  expenses  were  $6,446,517  as  compared  to  $6,063,439  for  the  year
ended September 30, 2017. The increase of $383,078 in 2018 was primarily due to increased compensation costs, increased consulting fees
incurred  for  financing  activities  and  corporate  development  services,  and  increased  investor  relations  fees.  In  addition,  we  incurred
$357,400  in  settlement  costs  for  the  termination  of  the  right  of  first  refusal  agreement  with  the  underwriter  of  our  2017  Public  Offering
during the year ended September 30, 2018 compared to $475,885 in settlement costs and $104,138 in financial consulting expenses incurred
related to the issuance of a unit purchase option during the year ended September 30, 2017.

Stock-based Compensation Expense

For  the  year  ended  September  30,  2018,  stock-based  compensation  expense  was  $779,701  as  compared  to  $986,620  for  the  year  ended
September 30, 2017. Stock-based compensation expense includes the expense for options assumed in the March 30, 2016 acquisition of
LMB, as well as grants to employees, directors and consultants. Stock-based compensation expense decreased by $206,919 in comparison
to  the  prior  period  as  certain  options  have  been  fully  expensed.  At  September  30,  2018,  unrecognized  total  compensation  cost  of
$1,425,957 related to unvested awards is expected to be recognized over the next 2.3 years.

Other Income (Expense)

During  the  year  ended  September  30,  2018,  the  Company  recorded  a  $450,000  gain  on  the  extinguishment  of  a  liability.  The  Company
reversed an accrual for certain research and development expenses that was recorded in a prior year that will not be paid. In addition, during
the year ended September 30, 2018, the Company recorded as other income a refund receivable in the amount of $818,343 from the FDA
for  2016  product  and  establishment  fees.  The  fees  previously  paid  by  the  Company  exceeded  the  costs  of  the  FDA’s  review  of  the
associated Suprenza applications.

There was no gain on revaluation of derivative warrant liability for the year ended September 30, 2018 as there were no warrants classified
as  derivative  warrants  during  the  year.  Gain  on  revaluation  of  derivative  warrant  liability  for  the  year  ended  September  30,  2017  was
$452,147.  The  fair  value  of  the  derivative  warrant  liability  fluctuated  with  changes  in  our  stock  price,  volatility,  remaining  lives  of  the
warrants, and interest rates.

Interest expense for the year ended September 30, 2018 was $15,838 as borrowings from our Chairman were converted to common stock
on August  8,  2017.  Interest  expense  on  the  notes  payable  acquired  in  the  acquisition  of  LMB  and  borrowings  from  our  Chairman  was
$850,789 for the year ended September 30, 2017, and includes net non-cash interest expense of $762,078 due to the beneficial conversion
feature on the conversion price of $1,595,411 and the amortization of the previously recorded modification premium of $833,333.

Net Loss

For the year ended September 30, 2018, we incurred a net loss of $12,536,638 compared to a net loss of $10,384,953 for the year ended
September 30, 2017. The $2,151,685 increase in the net loss was primarily due to the $3,626,673 increase in research and development
expenses offset by the $1,651,147 increase in net other income (expense).

33

 
 
 
 
 
 
 
 
 
 
 
 
Results of Operations for Year Ended September 30, 2017 compared to Year Ended September 30, 2016

Revenues

Operating expenses:

Research and development
General and administrative
Stock-based compensation – general and administrative

Total operating expenses

Operating loss

Interest income
Gain (loss) on revaluation of derivative warrant liability
Interest expense

Net loss

Revenues

Year Ended 
September 30,
2017

Year Ended 
September 30,
2016

  $

-    $

- 

2,936,252     
6,063,439     
986,620     
9,986,311     
(9,986,311)    
-     
452,147     
(850,789)    
  $ (10,384,953)   $

2,933,199 
3,783,941 
732,151 
7,449,291 
(7,449,291)
806 
(838,219)
(8,994)
(8,295,698)

We did not generate any revenues for the years ended September 30, 2017 and 2016.

Research and Development Expenses

For the year ended September 30, 2017, research and development expenses were $2,936,252 as compared to $2,933,199 during the year
ended September 30, 2016. The $3,053 increase in 2017 was primarily due to an increase of $776,192 in costs incurred in the development
of Mino-Lok offset by a decrease of $773,139 in costs incurred in the development of our product for the treatment of hemorrhoids and
costs related to Suprenza, including $292,575 received in 2016 from Alpex as reimbursement for regulatory filing fees. We are actively
seeking to raise additional capital in order to fund our research and development efforts.

General and Administrative Expenses

For the year ended September 30, 2017, general and administrative expenses were $6,063,439 as compared to $3,783,941 during the year
ended  September  30,  2016.  The  $2,279,498  increase  in  2017  was  primarily  due  to  the  acquisition  of  LMB  on  March  30,  2016,  which
resulted  in  increased  compensation  costs,  increased  consulting  fees  incurred  for  financing  activities  and  corporate  development  services,
and increased investor relations fees. In addition, the year ended September 30, 2016 only includes six months of expenses for LMB as the
acquisition was completed on March 30, 2016.

Stock-based Compensation Expense

For  the  year  ended  September  30,  2017,  stock-based  compensation  expense  was  $986,620  as  compared  to  $732,151  for  the  year  ended
September 30, 2016. The $254,469 increase in expense includes the expense for unvested options assumed in the acquisition of LMB, as
well as new grants to directors, employees and consultants.

Other Income (Expense)

There was no interest income earned on our cash balances for the year ended September 30, 2017 and only $806 in interest income earned
for the year ended September 30, 2016.

Gain (loss) on revaluation of derivative warrant liability for the year ended September 30, 2017 was $452,147 compared to $(838,219) for
the year ended September 30, 2016. The fair value of the derivative warrant liability fluctuates with changes in our stock price, volatility,
remaining lives of the warrants, and interest rates. The gain for the year ended September 30, 2017 was primarily due to a decrease in the
fair value of our stock from $9.45 per share at September 30, 2016 to $4.125 per share at August 8, 2017 when the final derivative warrants
were  reclassified  to  equity.  The  loss  for  the  year  ended  September  30,  2016  was  primarily  due  to  an  increase  in  the  fair  value  of  our
common stock from $8.10 at September 30, 2015 to $9.45 at September 30, 2016. At September 30, 2017, the Company has no outstanding
warrants that are considered to be derivative instruments.

34

 
 
 
 
 
   
 
 
   
      
  
   
      
  
   
   
   
   
   
   
   
   
 
 
 
 
 
 
 
 
 
 
 
 
Interest expense on the notes payable acquired in the acquisition of LMB and recent borrowings from our Chairman was $850,789 for the
year  ended  September  30,  2017,  and  includes  net  non-cash  interest  expense  of  $762,078  due  to  the  beneficial  conversion  feature  on  the
conversion  price  of  $1,595,411  and  the  amortization  of  the  previously  recorded  modification  premium  of  $833,333. After  the August  8,
2017  conversions  of  debt  to  common  stock,  the  Company  has  $172,970  in  outstanding  notes  payable  at  September  30,  2017.  Interest
expense on the notes payable acquired in the acquisition of LMB was $8,994 for the year ended September 30, 2016.

Net Loss

For the year ended September 30, 2017, we incurred a net loss of $10,384,953 compared to a net loss for the year ended September 30,
2016  of  $8,295,698.  The  $2,089,255  increase  in  the  net  loss  was  primarily  due  to  the  $2,279,498  increase  in  general  and  administrative
expenses and the $841,795 increase in interest expense offset by the $1,290,366 change in the (gain) loss on revaluation of the derivative
warrant liability.

LIQUIDITY AND CAPITAL RESOURCES

Going Concern Uncertainty and Working Capital

Citius  has  incurred  losses  of  $12,536,638,  $10,384,953  and  $8,295,698  for  the  years  ended  September  30,  2018,  2017  and  2016,
respectively. At September 30, 2018, Citius had an accumulated deficit of $40,257,838. Citius’ net cash used in operations during the years
ended September 30, 2018, 2017 and 2016, was $11,318,138, $7,971,205 and $5,900,421, respectively.

Our  independent  registered  accountants  report  on  our  September  30,  2018  consolidated  financial  statements  contains  an  emphasis  of  a
matter regarding substantial doubt about our ability to continue as a going concern and that the consolidated financial statements have been
prepared  assuming  we  will  continue  as  a  going  concern  and  do  not  include  any  adjustments  to  reflect  the  possible  future  effects  on  the
recoverability and classification of assets, or the amounts and classification of liabilities that may result if we do not continue as a going
concern.

As of September 30, 2018, Citius had working capital of $6,875,238. Our limited working capital was attributable to the operating losses
incurred  by  the  Company  since  inception  offset  by  our  capital  raising  activities.  At  September  30,  2018,  Citius  had  cash  and  cash
equivalents  of  $9,184,003  available  to  fund  its  operations.  The  Company’s  only  source  of  cash  flow  since  inception  has  been  from
financing  activities.  During  the  years  ended  September  30,  2018,  2017  and  2016,  the  Company  received  net  proceeds  of  $17,298,033,
$6,673,088 and $5,427,688, respectively from the issuance of equity. We also received $4,210,000 from the issuance of notes payable to
our  Chairman  of  the  Board,  Mr.  Leonard  Mazur,  during  the  year  ended  September  30,  2017.  Mr.  Mazur  converted  the  notes  payable  to
common  stock  on August  8,  2017.  Our  primary  uses  of  operating  cash  were  for  product  development  and  commercialization  activities,
regulatory expenses, employee compensation, consulting fees, legal and accounting fees, and insurance and travel expenses.

Financing Activities

During the year ended September 30, 2016, the Company sold 290,000 units for a purchase price of $8.10 per unit and 17,778 units for a
purchase price of $9.00 per unit for gross proceeds of $2,509,000. Each unit consisted of one share of common stock and one five-year
warrant to purchase a share of common stock at an exercise price of $9.00.

On March 22, 2016, the Company sold 333,333 shares of Common Stock at $9.00 per share to its Chairman of the Board, Leonard Mazur,
for gross proceeds of $3,000,000.

The  Board  of  Directors  authorized  revolving  demand  promissory  notes  with  Leonard  Mazur  in  an  aggregate  principal  amount  of  up  to
$2,500,000  that  accrue  interest  at  the  prime  rate  plus  1%.  On  September  7,  2016,  the  Company  issued  a  $500,000  note.  The  Company
issued  $2,000,000  of  additional  notes  through  the  period  ended  May  10,  2017.  On  May  10,  2017,  the  notes  were  converted  into  a
$2,500,000  convertible  promissory  note  that  is  convertible  into  shares  of  common  stock,  at  the  sole  discretion  of  Mr.  Mazur,  at  a
conversion price equal to 75% of the price per share paid by investors in the Company’s 2017 registered public offering. In connection with
the modification of the note, the Company recorded a charge of $833,333 to additional paid-in capital and increased the carrying value of
the notes to $3,333,333 which is the fair value of the common stock issuable on conversion. On August 8, 2017, Leonard Mazur converted
the $2,500,000 principal balance and accrued interest of $63,174 into 828,500 shares of common stock.

35

 
 
 
 
 
 
 
 
 
 
 
 
 
 
On May 10, 2017 and June 23, 2017, the Company executed a $1,500,000 future advance convertible promissory note and a $1,000,000
future advance convertible promissory note, respectively, with Leonard Mazur that accrue interest at the prime rate plus 1%. The notes are
convertible into shares of common stock, at the sole discretion of Mr. Mazur, at a conversion price equal to 75% of the price per share paid
by investors in the Company’s 2017 registered public offering. On August 8, 2017, Leonard Mazur converted the outstanding $2,210,000
principal balances and accrued interest of $13,066 into 718,567 shares of common stock.

In February 2017, the Company sold 128,017 units at $6.00 per unit for gross proceeds of $768,100. Each unit consisted of one share of
common stock and a five-year warrant to purchase one share of common stock at an exercise price of $8.25 per share. On June 8, 2017, the
Company  entered  into  agreements  where  it  was  released  from  the  restrictions  included  in  the  purchase  agreements.  In  exchange,  the
Company agreed to reprice the sale of the units to $4.125 per unit and reprice the warrants to an exercise price of $4.125 per share. During
the year ended September 30, 2017, the Company issued an additional 58,191 shares of common stock to the investors.

On August 8, 2017, the Company closed an underwritten public offering of 1,648,484 shares of common stock and warrants to purchase
1,648,484 shares of common stock at an offering price of $4.125 per share and $0.01 per warrant. The warrants have a per share exercise
price of $4.125, are exercisable immediately and will expire five years from the date of issuance.  The gross proceeds to Citius from this
offering  were  $6,802,469,  before  deducting  underwriting  discounts  and  commissions  and  other  offering  expenses  of  $685,573.  The
Company  granted  the  underwriters  a  45-day  option  to  purchase  up  to  an  additional  247,272  shares  of  common  stock  and  warrants  to
purchase  247,272  shares  of  common  stock  to  cover  over-allotments,  if  any.  On August  8,  2017,  the  underwriters  partially  exercised  the
over-allotment to purchase an additional 247,272 warrants.

On December 19, 2017, the Company closed a registered direct offering for the sale of 1,280,360 shares of common stock at $4.6925 per
share  for  gross  proceeds  of  $6,008,089.  Simultaneously,  the  Company  privately  sold  and  issued  to  the  investors  640,180  immediately
exercisable five and a half year warrants with an exercise price of $4.63 per share. Net proceeds from the offering were $5,482,523.

On March 29, 2018, the Company closed a registered direct offering for the sale of 669,504 shares of common stock at $2.985 per share for
gross proceeds of $1,998,469. Simultaneously, the Company privately sold and issued to investors 669,504 immediately exercisable five
and a half year warrants with an exercise price of $2.86 per share. Net proceeds from the offering were $1,763,576.

On August 13, 2018, the Company closed an offering for the sale of (i) 5,521,569 units, each unit consisted of one share of common stock
and one immediately exercisable five-year warrant to purchase one share at $1.15 per share, and (ii) 2,321,569 pre-funded units, each pre-
funded unit consisted of one pre-funded warrant to purchase one share of common stock and one immediately exercisable five-year warrant
to purchase one share at $1.15 per share. The exercise price of the pre-funded warrant is $0.01 and the pre-funded warrants do not expire.
The offering price was $1.275 per unit and $1.265 per pre-funded unit. Net proceeds from the offering were $8,926,786.

During the year ended September 30, 2018, an aggregate of 272,767 of the August 2017 public offering warrants were exercised at $4.125
per share for net proceeds of $1,125,148.

We  expect  that  we  will  have  sufficient  capital  to  continue  our  operations  through  June  2019.  We  plan  to  raise  additional  capital  in  the
future  to  support  our  operations.  There  is  no  assurance,  however,  that  we  will  be  successful  in  raising  the  needed  capital  or  that  the
proceeds will be received in a timely manner to fully support our operations.

Inflation

Our management believes that inflation has not had a material effect on our results of operations.

36

 
 
 
 
 
 
 
 
 
 
 
 
Off Balance Sheet Arrangements

We do not have any off-balance sheet arrangements.

CRITICAL ACCOUNTING POLICIES

Our  discussion  and  analysis  of  our  financial  condition  and  results  of  operations  is  based  on  our  financial  statements,  which  have  been
prepared in accordance with accounting principles generally accepted in the United States. The  preparation  of  these  financial  statements
requires us to make estimates and judgments that affect the reported amounts of assets, liabilities and expenses and related disclosure of
contingent  assets  and  liabilities.  We  review  our  estimates  on  an  ongoing  basis.  We  base  our  estimates  on  historical  experience  and  on
various other factors that we believe to be reasonable under the circumstances. Actual results may differ from these estimates. We believe
the judgments and estimates required by the following accounting policies to be critical in the preparation of our financial statements.

Research and Development

Research and development costs, including upfront fees and milestones paid to collaborators who are performing research and development
activities under contractual agreement with us, are expensed as incurred. We defer and capitalize our nonrefundable advance payments that
are  for  research  and  development  activities  until  the  related  goods  are  delivered  or  the  related  services  are  performed.  When  we  are
reimbursed by a collaboration partner for work we perform, we record the costs incurred as research and development expenses and the
related  reimbursement  as  a  reduction  to  research  and  development  expenses  in  our  statement  of  operations.  Research  and  development
expenses  primarily  consist  of  clinical  and  non-clinical  studies,  materials  and  supplies,  third-party  costs  for  contracted  services,  and
payments related to external collaborations and other research and development related costs.

In-process Research and Development and Goodwill

In process research and development represents the value of LMB’s leading drug candidate, Mino-Lok, an antibiotic lock solution in phase
3  clinical  development,  which  if  approved,  would  be  used  to  assist  in  the  treatment  of  catheter  related  bloodstream  infections  and  is
expected to be amortized on a straight-line basis over 8 years upon revenue generation. Goodwill represents the value of LMB’s industry
relationships and its assembled workforce. Goodwill will not be amortized and will be tested at least annually for impairment.

The Company reviews intangible assets annually to determine if any adverse conditions exist or a change in circumstances has occurred
that would indicate impairment or a change in the remaining useful life of any intangible asset. If the carry value of an asset exceeds its
undiscounted cash flows, the Company writes down the carrying value of the intangible asset to its fair value for the period identified. No
triggering events occurred since the acquisition of LMB that would suggest a potential impairment may have occurred through September
30, 2018.

The Company evaluates the recoverability of goodwill annually or more frequently if events or changes in circumstances indicate that the
carrying  value  of  an  asset  may  be  impaired.  Goodwill  is  first  qualitatively  assessed  to  determine  whether  further  impairment  testing  is
necessary. Factors that management considers in the assessment include macroeconomic conditions, industry and market conditions, overall
financial  performance,  (both  current  and  projected),  changes  in  management  and  strategy  as  well  as  changes  in  the  composition  of  the
carrying amount of net assets. If this qualitative assessment indicates that it is more likely that not that the fair value of a reporting unit is
less than its carrying amount, a two-step process is then performed.

The  Company  performed  a  qualitative  assessment  for  its  2018  analysis  of  goodwill.  Based  on  this  assessment,  management  does  not
believe that it is more likely than not, that the carrying value of the reporting unit exceeds its fair value. Accordingly, no further testing was
performed as management believes that there are no impairment issues with respect to goodwill as of September 30, 2018.

Income Taxes

We  follow  accounting  guidance  regarding  the  recognition,  measurement,  presentation  and  disclosure  of  uncertain  tax  positions  in  the
financial statements. Tax positions taken or expected to be taken in the course of preparing our tax returns are required to be evaluated to
determine  whether  the  tax  positions  are  “more-likely-than-not”  of  being  sustained  by  the  applicable  tax  authorities.  Tax  positions  not
deemed to meet a more-likely-than-not threshold would be recorded in the financial statements.

We recognize deferred tax assets and liabilities based on differences between the financial reporting and tax basis of assets and liabilities
using the enacted tax rates and laws that are expected to be in effect when the differences are expected to reverse. We provide a valuation
allowance for deferred tax assets for which we do not consider realization of such assets to be more likely than not.

Item 7A. Quantitative and Qualitative Disclosures About Market Risk 

Not required.

37

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Item 8.  Financial Statements and Supplementary Data

CITIUS PHARMACEUTICALS, INC.
CONSOLIDATED FINANCIAL STATEMENTS

INDEX

Report of Independent Registered Public Accounting Firm
Consolidated Balance Sheets
Consolidated Statements of Operations
Consolidated Statements of Changes in Stockholders’ Equity (Deficit)
Consolidated Statements of Cash Flows
Notes to Consolidated Financial Statements

F-1

Page

F-2
F-3
F-4
F-5
F-6
F-7

 
 
 
 
 
 
 
 
   
 
 
 
 
 
 
 
REPORT OF INDEPENDENT REGISTERED PUBLIC ACCOUNTING FIRM

To the Stockholders and Board of Directors of Citius Pharmaceuticals, Inc.:

Opinion on the Financial Statements

We have audited the accompanying consolidated balance sheets of Citius Pharmaceuticals, Inc. (the “Company”) as of September 30, 2018
and 2017, and the related consolidated statements of operations, changes in stockholders’ equity (deficit) and cash flows for each of the
years in the three-year period ended September 30, 2018, and the related notes to the consolidated financial statements (collectively, the
“financial  statements”).  In  our  opinion,  the  financial  statements  present  fairly,  in  all  material  respects,  the  financial  position  of  the
Company as of September 30, 2018 and 2017, and the results of its operations and its cash flows for each of the years in the three-year
period ended September 30, 2018, in conformity with accounting principles generally accepted in the United States of America.

Emphasis of Matter – Ability to Continue as a Going Concern

The accompanying financial statements have been prepared assuming that the Company will continue as a going concern. As discussed in
Note 2 to the financial statements, the Company has suffered recurring losses from operations, has negative cash flows from operations and
a  significant  accumulated  deficit.  These  conditions  raise  substantial  doubt  about  the  Company’s  ability  to  continue  as  a  going  concern.
Management’s plans in regard to these matters are described in Note 2. The financial statements do not include any adjustments that might
result from the outcome of this uncertainty.

Basis for Opinion

These  financial  statements  are  the  responsibility  of  the  Company’s  management.  Our  responsibility  is  to  express  an  opinion  on  the
Company’s  financial  statements  based  on  our  audits.  We  are  a  public  accounting  firm  registered  with  the  Public  Company Accounting
Oversight Board (United States) (“PCAOB”) and are required to be independent with respect to the Company in accordance with the U.S.
federal securities laws and the applicable rules and regulations of the Securities and Exchange Commission and the PCAOB.

We conducted our audits in accordance with the standards of the PCAOB. Those standards require that we plan and perform the audit to
obtain reasonable assurance about whether the financial statements are free of material misstatement, whether due to error or fraud. The
Company is not required to have, nor were we engaged to perform, an audit of its internal control over financial reporting. As part of our
audits  we  are  required  to  obtain  an  understanding  of  internal  control  over  financial  reporting,  but  not  for  the  purpose  of  expressing  an
opinion on the effectiveness of the Company’s internal control over financial reporting. Accordingly, we express no such opinion.

Our audits included performing procedures to assess the risks of material misstatement of the financial statements, whether due to error or
fraud, and performing procedures that respond to those risks. Such procedures included examining, on a test basis, evidence regarding the
amounts  and  disclosures  in  the  financial  statements.  Our  audits  also  included  evaluating  the  accounting  principles  used  and  significant
estimates  made  by  management,  as  well  as  evaluating  the  overall  presentation  of  the  financial  statements.  We  believe  that  our  audits
provide a reasonable basis for our opinion.

/s/ Wolf & Company, P.C.

Boston, Massachusetts
December 11, 2018

We have served as the Company’s auditor since 2014.

F-2

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
CITIUS PHARMACEUTICALS, INC.
CONSOLIDATED BALANCE SHEETS
SEPTEMBER 30, 2018 AND 2017

ASSETS

Current Assets:
Cash and cash equivalents
Other receivables
Prepaid expenses

Total Current Assets

Property and equipment, net

Other Assets:
Deposits
In-process research and development
Goodwill

Total Other Assets

Total Assets

LIABILITIES AND STOCKHOLDERS’ EQUITY

Current Liabilities:
Accounts payable
Accrued expenses
Accrued compensation
Accrued interest – related parties
Notes payable – related parties
Due to related party

Total Current Liabilities

Commitments and Contingencies

Stockholders’ Equity:
Preferred stock - $0.001 par value; 10,000,000 shares authorized; no shares issued and outstanding
Common stock - $0.001 par value; 200,000,000 shares authorized; 16,198,791 and 8,345,844 shares issued

and outstanding at September 30, 2018 and 2017, respectively

Additional paid-in capital
Accumulated deficit
Total Stockholders’ Equity

Total Liabilities and Stockholders’ Equity

2018

2017

  $

9,184,003    $
818,343     
57,732     
10,060,078     

3,204,108 
— 
220,246 
3,424,354 

1,483     

3,236 

2,167     

2,167 
19,400,000      19,400,000 
1,586,796 
1,586,796     
20,988,963      20,988,963 

  $ 31,050,524    $ 24,416,553 

  $

1,573,444    $
181,657     
1,198,915     
57,854     
172,970     
—     
3,184,840     

602,431 
560,918 
1,063,000 
42,209 
172,970 
27,637 
2,469,165 

—     

— 

16,199     

8,346 
68,107,323      49,660,242 

(40,257,838)     (27,721,200)
27,865,684      21,947,388 

  $ 31,050,524    $ 24,416,553 

See accompanying report of independent registered public accounting firm and notes to the consolidated financial statements.

F-3

 
 
 
 
 
   
 
 
 
     
 
 
   
     
 
   
     
 
   
   
   
 
   
      
  
   
 
   
      
  
   
      
  
   
   
   
   
 
   
      
  
 
   
      
  
   
      
  
 
   
      
  
   
      
  
   
   
   
   
   
   
 
   
      
  
   
      
  
 
   
      
  
   
      
  
   
   
   
   
   
 
   
      
  
 
 
CITIUS PHARMACEUTICALS, INC.
CONSOLIDATED STATEMENTS OF OPERATIONS
FOR THE YEARS ENDED SEPTEMBER 30, 2018, 2017 AND 2016

Revenues

Operating Expenses:

Research and development
General and administrative
Stock-based compensation – general and administrative

Total Operating Expenses

Operating Loss

Other Income (Expense), Net:

Interest income
Gain on extinguishment of liability
Other income
Gain (loss) on revaluation of derivative warrant liability
Interest expense

Total Other Income (Expense), Net

Loss before Income Taxes

Income tax benefit

Net Loss

2018

2017

2016

  $

—    $

—    $

— 

6,562,925     
6,446,517     
779,701     
13,789,143     

2,936,252     
6,063,439     
986,620     
9,986,311     

2,933,199 
3,783,941 
732,151 
7,449,291 

(13,789,143)    

(9,986,311)    

(7,449,291)

—     
450,000     
818,343     
—     
(15,838)    
1,252,505     

—     
—     
—     
452,147     
(850,789)    
(398,642)    

806 
— 
— 
(838,219)
(8,994)
(846,407)

(12,536,638)    
—     

(10,384,953)    
—     

(8,295,698)
— 

  $ (12,536,638)   $ (10,384,953)   $ (8,295,698)

Net Loss Per Share - Basic and Diluted

  $

(1.17)   $

(1.89)   $

(2.29)

Weighted Average Common Shares Outstanding

Basic and diluted

10,731,875     

5,482,494     

3,623,208 

See accompanying report of independent registered public accounting firm and notes to the consolidated financial statements.

F-4

 
 
 
 
 
   
   
 
 
   
     
   
 
 
 
   
      
      
  
 
   
      
      
  
   
      
      
  
   
   
   
   
 
   
      
      
  
   
 
   
      
      
  
   
      
      
  
   
   
   
   
   
   
 
   
      
      
  
   
   
 
   
      
      
  
 
   
      
      
  
 
   
      
      
  
   
      
      
  
   
 
 
CITIUS PHARMACEUTICALS, INC.
CONSOLIDATED STATEMENTS OF CHANGES IN STOCKHOLDERS’ EQUITY (DEFICIT)
FOR THE YEARS ENDED SEPTEMBER 30, 2018, 2017 AND 2016  

Preferred    

Common Stock

Stock

Shares

    Amount

    Additional      
Paid-In
Capital

    Accumulated   
Deficit

Total
    Stockholders’ 
Equity
(Deficit)

Balance, September 30, 2015
Issuance of common stock in private

  $

placement, net of costs

Issuance of common stock for services    
Issuance of common stock, warrants
and stock options for acquisition

Issuance of warrants for services
Reclassification of derivative warrant

liability to additional paid-in capital    

Stock-based compensation
Net loss

Balance, September 30, 2016
Issuance of common stock in private

placement, net of costs

Issuance of common stock in public

offering, net of costs

Issuance of common stock for services

and release agreements

Issuance of fractional shares for 1-for-

15 reverse stock split
Stock options exercised
Conversion of convertible promissory
notes – related party to common
stock

Beneficial conversion feature on
convertible promissory notes –
related party

Premium on convertible promissory

notes – related party

Issuance of unit purchase options
Issuance of warrants in settlement of

liabilities

Reclassification of derivative warrant

liability to additional paid-in capital,
net

Stock-based compensation
Net loss

Balance, September 30, 2017
Issuance of common stock in registered

direct offering, net of costs of
$760,459

Issuance of common stock, net of
issuance costs and underwriting
discount of $1,049,999

Issuance of common stock upon

exercise of warrants

Issuance of common stock for services

and release agreement

—     

2,274,526    $

2,275    $

8,403,061    $ (9,040,549)   $

(635,213)

—     
—     

641,111     
17,778     

641     
18     

4,228,483     
149,982     

—     
—     

4,229,124 
150,000 

—     
—     

1,942,456     
—     

1,942      19,013,131     
477,181     

—     

—     
—     

19,015,073 
477,181 

—     
—     
—     

—     
—     
—     

—     
—     
—     

1,093,765     
732,151     
—     

—     
—     
(8,295,698)    

1,093,765 
732,151 
(8,295,698)

—     

4,875,871     

4,876      34,097,754      (17,336,247)    

16,766,383 

—     

128,016     

128     

491,223     

—     

491,351 

—     

1,648,484     

1,648     

6,115,248     

6,116,896 

—     

140,843     

141     

703,878     

—     

704,019 

—     
—     

734     
4,829     

1     
5     

(1)    
35     

—     
—     

— 
40 

1,547,067     

1,547     

4,784,693     

—     

4,786,240 

—     

—     
—     

—     

—     
—     
—     

—     

—     
—     

—     

—     
—     
—     

—     

1,595,411     

—     

1,595,411 

—     
—     

(833,333)    
297,998     

—     
—     

(833,333)
297,998 

—     

190,890     

—     

190,890 

—     
—     
—     

1,229,826     
986,620     

—     
—     
—      (10,384,953)    

1,229,826 
986,620 
(10,384,953)

—     

8,345,844     

8,346      49,660,242      (27,721,200)    

21,947,388 

—     

1,949,864     

1,949     

7,244,150     

—     

7,246,099 

—     

5,521,569     

5,522     

8,921,264     

—     

8,926,786 

—     

289,314     

290     

1,124,858     

—     

1,125,148 

—     

92,200     

92     

377,108     

—     

377,200 

Stock-based compensation expense
Net loss

—     

—     

—     

779,701     

—     
—      (12,536,638)    

779,701 
(12,536,638)

Balance, September 30, 2018

—      16,198,791    $

16,199    $ 68,107,323    $ (40,257,838)   $ 27,865,684 

See accompanying report of independent registered public accounting firm and notes to the consolidated financial statements.

 
 
 
 
   
     
   
 
     
   
 
 
   
     
 
 
   
 
 
 
   
   
   
   
 
 
   
      
      
      
      
      
  
   
   
   
   
   
 
   
      
      
      
      
      
  
   
   
   
      
   
   
   
   
      
   
   
   
   
   
   
   
 
   
      
      
      
      
      
  
   
   
   
   
   
 
   
      
      
      
      
      
  
   
      
      
      
   
 
   
      
      
      
      
      
  
   
 
 
F-5

CITIUS PHARMACEUTICALS, INC.
CONSOLIDATED STATEMENTS OF CASH FLOWS
FOR THE YEARS ENDED SEPTEMBER 30, 2018, 2017 AND 2016

Cash Flows From Operating Activities:
Net loss
Adjustments to reconcile net loss to net cash used in operating activities:

Stock-based compensation
(Gain) loss on revaluation of derivative warrant liability
Gain on extinguishment of liability
Issuance of common stock for services and release agreements
Fair value of options issued to purchase units of common stock
Warrants issued and repriced in settlement agreements
Non-cash interest expense
Depreciation
Write-off of abandoned trademarks
Changes in operating assets and liabilities:

Other receivables
Prepaid expenses
Accounts payable
Accrued expenses
Accrued compensation
Accrued interest – related parties
Due to related party

Net Cash Used In Operating Activities

Cash Flows From Investing Activities:

Cash acquired in acquisition
Purchase of property and equipment

Net Cash Provided By (Used In) Investing Activities

Cash Flows From Financing Activities:

Proceeds from notes payable – related parties
Repayment of notes payable – related parties
Proceeds from common stock warrant exercises
Proceeds from stock option exercise
Net proceeds from common stock and warrants in August 2018 offering
Net proceeds from registered direct offering
Net proceeds from private placement
Net proceeds from public offering
Deferred offering costs

Net Cash Provided By Financing Activities

Increase (Decrease) in Cash and Cash Equivalents
Cash and Cash Equivalents – Beginning of Year

2018

2017

2016

  $ (12,536,638)   $ (10,384,953)   $ (8,295,698)

779,701     
—     
(450,000)    
377,200     
—     
—     
—     
1,753     
—     

986,620     
(452,147)    
—     
704,019     
104,138     
190,890     
762,078     
2,632     
—     

732,151 
838,219 
— 
150,000 
— 
— 
— 
1,343 
5,401 

(818,343)    
162,514     
971,013     
70,739     
135,915     
15,645     
(27,637)    
(11,318,138)    

—     
572,098     
(306,725)    
(397,183)    
159,750     
87,578     
—     
(7,971,205)    

— 
(40,759)
105,230 
351,182 
288,250 
7,009 
(42,749)
(5,900,421)

—     

—     
—     

—     

255,748 

(2,126)    
(2,126)    

— 
255,748 

—     
—     
1,125,148     
—     
8,926,786     
7,246,099     
—     
—     
—     
17,298,033     

4,210,000     
—     
—     
40     
—     
—     
556,152     
6,116,896     
—     
10,883,088     

500,000 
(600,000)
— 
— 
— 
— 
5,427,688 
— 
(64,801)
5,262,887 

5,979,895     
3,204,108     

2,909,757     
294,351     

(381,786)
676,137 

Cash and Cash Equivalents – End of Year

  $

9,184,003    $

3,204,108    $

294,351 

Supplemental Disclosures of Cash Flow Information and Non-cash Transactions:
Interest paid

Premium on convertible promissory notes – related party
Fair value of unit purchase option issued for future services

Fair value of warrants recorded as derivative warrant liability

Fair value of warrants issued for future services
Reclassification of derivative warrant liability to additional paid-in capital
Beneficial conversion feature on convertible promissory notes – related party

Conversion of convertible promissory notes – related party and related accrued interest

into common stock

Par value of common stock issued upon cashless exercise of warrants

  $
  $
  $
  $
  $
  $
  $

  $
  $

193    $
—    $
—    $
—    $
—    $
—    $
—    $

1,133    $
833,333    $
193,860    $
641,385    $
—     
1,229,826    $
1,595,411    $

1,985 
— 
— 
1,198,564 
477,181 
1,093,765 
— 

—    $
17    $

4,786,240    $
—    $

— 
— 

See accompanying report of independent registered public accounting firm and notes to the consolidated financial statements.

 
 
 
 
 
   
   
 
 
   
     
     
 
   
      
      
  
   
      
      
  
   
   
   
   
   
   
   
   
   
   
      
      
  
   
   
   
   
   
   
   
   
 
   
      
      
  
   
      
      
  
   
   
   
 
   
      
      
  
   
      
      
  
   
   
   
   
   
   
   
   
   
   
 
   
      
      
  
   
   
 
   
      
      
  
 
   
      
      
  
   
      
      
  
 
 
F-6

CITIUS PHARMACEUTICALS, INC.
NOTES TO CONSOLIDATED FINANCIAL STATEMENTS
FOR THE YEARS ENDED SEPTEMBER 30, 2018, 2017 AND 2016

1. NATURE OF OPERATIONS AND BASIS OF PRESENTATION

Business

Citius  Pharmaceuticals,  Inc.  (“Citius”  or  the  “Company”)  is  a  specialty  pharmaceutical  company  dedicated  to  the  development  and
commercialization  of  critical  care  products  targeting  unmet  needs  with  a  focus  on  anti-infectives,  cancer  care  and  unique  prescription
products.

On  March  30,  2016,  Citius  acquired  Leonard-Meron  Biosciences,  Inc.  (“LMB”)  as  a  wholly-owned  subsidiary  (see  “Acquisition  of
Leonard-Meron Biosciences, Inc.” below). Since its inception, the Company has devoted substantially all of its efforts to business planning,
research and development, recruiting management and technical staff, and raising capital.

Citius is subject to a number of risks common to companies in the pharmaceutical industry including, but not limited to, risks related to the
development by Citius or its competitors of research and development stage products, market acceptance of its products, competition from
larger  companies,  dependence  on  key  personnel,  dependence  on  key  suppliers  and  strategic  partners,  the  Company’s  ability  to  obtain
additional financing and the Company’s compliance with governmental and other regulations.

Acquisition of Leonard-Meron Biosciences, Inc.

On March 30, 2016, the Company acquired all of the outstanding stock of LMB by issuing 1,942,456 shares of Company common stock.
As  of  March  30,  2016,  the  stockholders  of  LMB  received  approximately  41%  of  the  issued  and  outstanding  common  stock  of  the
Company. In addition, the Company converted the outstanding common stock warrants of LMB into 243,020 common stock warrants of
the Company and converted the outstanding common stock options of LMB into 77,252 common stock options of the Company.

The Company recorded goodwill of $1,586,796 for the excess of the purchase price over the net assets acquired.

See report of independent accounting firm

F-7

 
 
  
 
 
 
 
 
 
 
 
Unaudited  pro  forma  operating  results  for  the  year  ended  September  30,  2016,  assuming  the  acquisition  of  LMB  had  been  made  as  of
October 1, 2015, are as follows:

Revenues

Net loss
Net loss per share – basic and diluted

Basis of Presentation

  $
— 
  $ (11,548,647)
(2.52)
  $

The  accompanying  consolidated  financial  statements  include  the  operations  of  Citius  Pharmaceuticals,  Inc.,  and  its  wholly-owned
subsidiaries,  Citius  Pharmaceuticals,  LLC  and  LMB  since  the  March  30,  2016  acquisition. All  significant  inter-company  balances  and
transactions have been eliminated in consolidation.

2. GOING CONCERN UNCERTAINTY AND MANAGEMENT’S PLAN

The accompanying consolidated financial statements have been prepared on a going concern basis, which contemplates the realization of
assets and the satisfaction of liabilities in the normal course of business. The Company experienced negative cash flows from operations of
$11,318,138,  $7,971,205  and  $5,900,421,  for  the  years  ended  September  30,  2018,  2017  and  2016,  respectively.  The  Company  has  no
revenue and has relied on proceeds from equity transactions and debt to finance its operations. At September 30, 2018, the Company had
limited capital to fund its operations. This raises substantial doubt about the Company’s ability to continue as a going concern within one
year after the date that the accompanying consolidated financial statements are issued.

The  Company  plans  to  raise  capital  through  equity  financings  from  outside  investors  as  well  as  raise  additional  funds  from  existing
investors. There is no assurance, however, that the Company will be successful in raising the needed capital and, if funding is available, that
it  will  be  available  on  terms  acceptable  to  the  Company.  The  accompanying  consolidated  financial  statements  do  not  include  any
adjustments that might result from the outcome of the above uncertainty.

3. PATENT AND TECHNOLOGY LICENSE AGREEMENT

LMB has a patent and technology license agreement with Novel Anti-Infective Therapeutics, Inc., (“NAT”) to develop and commercialize
Mino-Lok on an exclusive, worldwide sub licensable basis, as amended. LMB pays an annual maintenance fee in June until commercial
sales of a product subject to the license commence. The Company recorded maintenance fee expense of $75,000, $50,000 and $45,000 in
2018, 2017 and 2016, respectively under the terms of this agreement.

LMB will also pay annual royalties on net sales of licensed products, with royalties ranging from the mid-single digits to the low double
digits. In limited circumstances in which the licensed product is not subject to a valid patent claim and a competitor is selling a competing
product,  the  royalty  rate  is  in  the  low-single  digits.  After  a  commercial  sale  is  obtained,  LMB  must  pay  minimum  aggregate  annual
royalties  of  $100,000  in  the  first  commercial  year  which  is  prorated  for  a  less  than  12-month  period,  increasing  $25,000  per  year  to  a
maximum  of  $150,000  annually.  LMB  must  also  pay  NAT  up  to  $1,390,000  upon  achieving  specified  regulatory  and  sales  milestones.
Finally, LMB must pay NAT a specified percentage of payments received from any sub licensees.

Unless earlier terminated by NAT, based on the failure to achieve certain development and commercial milestones, the license agreement
remains in effect until the date that all patents licensed under the agreement have expired and all patent applications within the licensed
patent rights have been cancelled, withdrawn or expressly abandoned.

See report of independent accounting firm

F-8

 
 
 
 
 
 
 
 
 
 
 
 
 
4. SUMMARY OF SIGNIFICANT ACCOUNTING POLICIES

A summary of the significant accounting policies followed by the Company in the preparation of the consolidated financial statements is
as follows: 

Use of Estimates

The process of preparing financial statements in conformity with accounting principles generally accepted in the United States of America
(“GAAP”) requires management to make estimates and assumptions that affect the reported amounts of assets and liabilities and disclosure
of  contingent  assets  and  liabilities  at  the  date  of  financial  statements  and  the  reported  amounts  of  revenues  and  expenses  during  the
reporting period.

Cash and Cash Equivalents

The  Company  considers  all  highly  liquid  instruments  with  maturities  of  less  than  three  months  at  the  time  of  purchase  to  be  cash
equivalents. From time to time, the Company may have cash balances in financial institutions in excess of insurance limits. The Company
has never experienced any losses related to these balances.

Property and Equipment

Property  and  equipment  are  valued  at  cost  and  are  being  depreciated  over  their  useful  lives  using  the  straight-line  method  for  financial
reporting purposes. Routine maintenance and repairs are charged to expense as incurred. Expenditures which materially increase the value
or extend useful lives are capitalized. Property and equipment are depreciated over estimated useful lives of three to five years.

Research and Development

Research and development costs, including upfront fees and milestones paid to collaborators who are performing research and development
activities under contractual agreement with the Company, are expensed as incurred. The Company defers and capitalizes its nonrefundable
advance  payments  that  are  for  research  and  development  activities  until  the  related  goods  are  delivered  or  the  related  services  are
performed. When the Company is reimbursed by a collaboration partner for work the Company performs, it records the costs incurred as
research and development expenses and the related reimbursement as a reduction to research and development expenses in its consolidated
statement of operations. Research and development expenses primarily consist of clinical and non-clinical studies, materials and supplies,
third-party costs for contracted services, and payments related to external collaborations and other research and development related costs.

See report of independent accounting firm

F-9

 
 
 
 
 
 
 
 
 
 
 
 
In-process Research and Development and Goodwill

In-process  research  and  development  represents  the  value  of  LMB’s  leading  drug  candidate  which  is  an  antibiotic  solution  used  to  treat
catheter-related  bloodstream  infections  (Mino-Lok)  and  is  expected  to  be  amortized  on  a  straight-line  basis  over  a  period  of  eight  years
commencing  upon  revenue  generation.    Goodwill  represents  the  value  of  LMB’s  industry  relationships  and  its  assembled  workforce.
Goodwill will not be amortized but will be tested at least annually for impairment.

The Company reviews intangible assets annually to determine if any adverse conditions exist or a change in circumstances has occurred
that would indicate impairment or a change in the remaining useful life of any intangible asset. If the carrying value of an asset exceeds its
undiscounted cash flows, the Company writes down the carrying value of the intangible asset to its fair value in the period identified. No
triggering  events  occurred  since  the  acquisition  of  LMB  that  would  suggest  that  a  potential  impairment  may  have  occurred  through
September 30, 2018.

The Company evaluates the recoverability of goodwill annually or more frequently if events or changes in circumstances indicate that the
carrying  value  of  an  asset  might  be  impaired.  Goodwill  is  first  qualitatively  assessed  to  determine  whether  further  impairment  testing  is
necessary. Factors that management considers in this assessment include macroeconomic conditions, industry and market considerations,
overall financial performance (both current and projected), changes in management and strategy and changes in the composition or carrying
amount of net assets. If this qualitative assessment indicates that it is more likely than not that the fair value of a reporting unit is less than
its carrying amount, a two-step process is then performed. The two-step test first compares the fair value of the reporting unit to its carrying
value.  If the fair value exceeds the carrying value, no impairment exists, and the second step is not performed.  If the fair value of the
reporting  unit  is  less  than  its  carrying  value,  an  impairment  loss  is  recorded  as  part  of  the  second  step  of  the  test,  to  the  extent  that  the
implied fair value of the reporting unit goodwill is less than the carrying value.

The  Company  performed  a  qualitative  assessment  for  our  2018  analysis  of  goodwill.  Based  on  this  assessment,  management  does  not
believe that it is more likely than not that the carrying value of the reporting unit exceeds its fair value. Accordingly, no further testing was
performed as management believes that there are no impairment issues in regards to goodwill as of September 30, 2018.

Patents and Trademarks

Certain costs of outside legal counsel related to obtaining trademarks for the Company are capitalized. Patent costs are amortized over the
legal life of the patents, generally twenty years, starting at the patent issuance date. There are no capitalized patents and trademarks as of
September 30, 2018.

The  costs  of  unsuccessful  and  abandoned  applications  are  expensed  when  abandoned.  The  cost  of  maintaining  existing  patents  are
expensed as incurred.

Stock-Based Compensation

The Company recognizes compensation costs resulting from the issuance of stock-based awards to employees and directors as an expense
in the consolidated statement of operations over the requisite service period based on the fair value for each stock award on the grant date,
net  of  actual  forfeitures.  The  fair  value  of  each  option  grant  is  estimated  as  of  the  date  of  grant  using  the  Black-Scholes  option  pricing
model. Due to its limited operating history, limited number of sales of its common stock and limited history of its shares being publicly
traded,  the  Company  estimates  its  volatility  in  consideration  of  a  number  of  factors  including  the  volatility  of  comparable  public
companies. Because our stock options have characteristics significantly different from those of traded options, and because changes in the
input assumptions can materially affect the fair value estimate, the existing model may not necessarily provide a reliable single measure of
fair value of our stock options.

The  Company  recognizes  compensation  costs  resulting  from  the  issuance  of  stock-based  awards  to  non-employees  as  an  expense  in  the
consolidated statement of operations over the service period based on the measurement of fair value for each stock award.

See report of independent accounting firm

F-10

 
 
 
 
 
 
 
 
 
 
 
 
 
Derivative Instruments

The Company generally does not use derivative instruments to hedge exposures to cash-flow or market risks; however, certain warrants to
purchase common stock that did not meet the requirements for classification as equity were classified as liabilities. In such instances, net-
cash settlement was assumed for financial reporting purposes, even when the terms of the underlying contracts do not provide for a net-
cash settlement. Such financial instruments were initially recorded at fair value with subsequent changes in fair value charged (credited) to
operations in each reporting period. When these instruments subsequently met the requirements for classification as equity, the Company
reclassified the fair value to equity.

Income Taxes

The Company follows accounting guidance regarding the recognition, measurement, presentation and disclosure of uncertain tax positions
in the consolidated financial statements. Tax positions taken or expected to be taken in the course of preparing our tax returns are required
to be evaluated to determine whether the tax positions are “more-likely-than-not” of being sustained by the applicable tax authorities. Tax
positions  not  deemed  to  meet  a  more-likely-than-not  threshold  would  be  recorded  in  the  consolidated  financial  statements.  There  are  no
uncertain tax positions that require accrual or disclosure as of September 30, 2018.

Any  interest  or  penalties  are  charged  to  expense.  During  the  years  ended  September  30,  2018,  2017  and  2016,  the  Company  did  not
recognize  any  interest  and  penalties.  Tax  years  subsequent  to  September  30,  2014  are  subject  to  examination  by  federal  and  state
authorities.

We recognize deferred tax assets and liabilities based on differences between the financial reporting and tax basis of assets and liabilities,
and operating loss and tax credit carry forwards. Deferred tax assets and liabilities are measured using the enacted tax rates and laws that
are expected to be in effect when the differences are expected to reverse. We provide a valuation allowance, if necessary, for deferred tax
assets  for  which  we  do  not  consider  realization  of  such  assets  to  be  “more-likely-than-not”.  The  deferred  tax  benefit  or  expense  for  the
period represents the change in the deferred tax asset or liability from the beginning to the end of the period.

Basic and Diluted Net Loss per Common Share

Basic and diluted net loss per common share is computed by dividing net loss in each period by the weighted average number of shares of
common stock outstanding during such period. For the periods presented, common stock equivalents, consisting of options, warrants and
convertible securities were not included in the calculation of the diluted loss per share because they were anti-dilutive.

Fair Value of Financial Instruments

The financial statements include various estimated fair value information.  Financial instruments are initially recorded at historical cost. If
subsequent circumstances indicate that a decline in the fair value of a financial asset is other than temporary, the financial asset is written
down to its fair value.

Unless  otherwise  indicated,  the  fair  values  of  financial  instruments  approximate  their  carrying  amounts.  By  their  nature,  all  financial
instruments  involve  risk,  including  credit  risk  for  non-performance  by  counterparties.  The  fair  values  of  cash  and  cash  equivalents,
accounts payable, accrued interest, accrued expenses, notes payable and due to related party approximate their recorded amounts because of
their relatively short settlement terms.

See report of independent accounting firm

F-11

 
 
 
 
 
 
 
 
 
 
 
 
 
The Company groups its assets and liabilities measured at fair value in three levels, based on the markets in which the assets and liabilities
are traded and the reliability of the assumptions used to determine fair value.

Level 1: Valuation is  based  on  quoted  prices  in  active  markets  for  identical  assets  or  liabilities.  Level  1  assets  and  liabilities  generally
include debt and equity securities that are traded in an active exchange market. Valuations are obtained from readily available
pricing sources for market transactions involving identical assets or liabilities.

Level 2: Valuation is based on observable inputs other than Level 1 prices, such as quoted prices for similar assets or liabilities; quoted
prices in  markets  that  are  not  active;  or  other  inputs  that  are  observable  or  can  be  corroborated  by  observable  market  data  for
substantially the full term of the assets or liabilities. For example, Level 2 assets and liabilities may include debt securities with
quoted prices that are traded less frequently than exchange-traded instruments.

Level 3: Valuation is  based  on  unobservable  inputs  that  are  supported  by  little  or  no  market  activity  and  that  are  significant  to  the  fair
value of  the  assets  or  liabilities.  Level  3  assets  and  liabilities  include  financial  instruments  whose  value  is  determined  using
pricing models, discounted cash flow methodologies, or similar techniques, as well as instruments for which the determination of
fair  value  requires  significant  management  judgment  or  estimation.  This  category  generally  includes  certain  private  equity
investments and long-term derivative contracts.

The  Company’s  financial  liabilities  measured  at  fair  value  as  of  September  30,  2016  consisted  solely  of  the  derivative  warrant  liability
which  was  classified  as  Level  3  in  fair  value  hierarchy  (see  Note  6).  The  Company  used  a  valuation  method,  the  Black-Scholes  option
pricing  model,  and  the  requisite  assumptions  in  estimating  the  fair  value  for  the  warrants  considered  to  be  derivative  instruments.  The
Company has no financial assets measured at fair value as of September 30, 2018 and September 30, 2017.

The Company may also be required, from time to time, to measure certain other financial assets at fair value on a nonrecurring basis. These
adjustments to fair value usually result from application of lower-of-cost-or-market accounting or write-downs of individual assets. There
were no such adjustments in the years ended September 30, 2018, 2017 and 2016.

Segment Reporting

The Company currently operates as a single segment.

Concentrations of Credit Risk

The Company has no significant off-balance-sheet concentration of credit risk such as foreign exchange contracts, option contracts or other
hedging arrangements.

Recently Issued Accounting Standards

In June 2018, the Financial Accounting Standards Board (“FASB”) issued Accounting Standards Update (“ASU”) 2018-07, Compensation
– Stock Compensation (Topic 718): Improvements to Non-employee Share-Based Payment Accounting. ASU 2018-07 expands the scope
of Topic 718 to include share-based payment transactions for acquiring goods and services from nonemployees. An entity should apply the
requirements of Topic 718 to non-employees awards except for specific guidance on inputs to an option pricing model and the attribution of
cost.  The  amendments  in  this ASU  are  effective  for  public  business  entities  for  fiscal  years,  and  for  interim  periods  within  those  fiscal
years,  beginning  after  December  15,  2018.  Early  adoption  is  permitted.  The  Company  is  in  the  process  of  evaluating  the  impact  of  this
ASU on its consolidated results of operations, financial position or disclosures.

5. NOTES PAYABLE 

A summary of notes payable outstanding as of September 30, 2018 and 2017 is as follows:

Demand notes payable – Leonard Mazur
Demand notes payable – Myron Holubiak
Notes payable

2018

2017

160,470    $
12,500     
172,970    $

160,470 
12,500 
172,970 

  $

  $

See report of independent accounting firm

F-12

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
 
   
 
Notes Payable - Related Parties

On  March  30,  2016,  the  Company  assumed  $772,970  of  demand  notes  payable  in  the  acquisition  of  LMB,  including  $760,470  to  our
Chairman,  Leonard  Mazur,  and  $12,500  to  our  Chief  Executive  Officer,  Myron  Holubiak.  Notes  with  a  principal  balance  of  $704,000
accrue interest at the “Prime Rate”, as published in the Wall Street Journal on the last day of each month plus 1% and notes with a principal
balance of $68,970 accrue interest at 12% per annum. In April 2016, $600,000 of the “Prime Rate” plus 1% demand notes payable and
accrued interest of $1,985 was repaid to Leonard Mazur.

The  Board  of  Directors  authorized  revolving  demand  promissory  notes  with  Leonard  Mazur  in  an  aggregate  principal  amount  of  up  to
$2,500,000 that accrued interest at the prime rate plus 1%. On September 7, 2016, the Company issued a $500,000 note. The Company
issued  $2,000,000  of  additional  notes  through  the  period  ended  May  10,  2017.  On  May  10,  2017,  the  notes  were  converted  into  a
$2,500,000 convertible promissory note. The note was convertible into shares of common stock, at the sole discretion of Mr. Mazur, at a
conversion price equal to 75% of the price per share paid by investors in the Company’s 2017 registered public offering. In connection with
the modification of the note, in 2017 the Company recorded a charge of $833,333 to additional paid-in capital and increased the carrying
value of the notes to $3,333,333 which was the fair value of the common stock issuable on conversion. On August 8, 2017, Leonard Mazur
converted the $2,500,000 principal balance and accrued interest of $63,174 into 828,500 shares of common stock.

On May 10, 2017 and June 23, 2017, the Company executed future advance convertible promissory notes with Leonard Mazur that were
scheduled  to  mature  on  December  31,  2017  and  accrue  interest  at  the  prime  rate  plus  1%.  The  notes  were  convertible  into  shares  of
common  stock,  at  the  sole  discretion  of  Mr.  Mazur,  at  a  conversion  price  equal  to  75%  of  the  price  per  share  paid  by  investors  in  the
Company’s 2017 registered public offering. On August 8, 2017, Leonard Mazur converted the outstanding $2,210,000 principal balances
and accrued interest of $13,066 into 718,567 shares of common stock.

In  connection  with  the  conversions,  the  Company  recorded  net  non-cash  interest  expense  of  $762,078  due  to  the  beneficial  conversion
feature on the conversion price of $1,595,411 and the amortization of the previously recorded modification premium of $833,333.

The  Company  evaluated  all  terms  of  the  future  advance  convertible  promissory  notes,  including  the  Change  in  Control  provision,  to
identify any embedded features that required bifurcation and recording as derivative instruments. The Company determined that there were
no such features requiring separate accounting.

Interest Expense

Interest expense on notes payable for the years ended September 30, 2018, 2017 and 2016 was $15,645, $850,789 and $8,994, respectively.

6. DERIVATIVE WARRANT LIABILITY

Derivative financial instruments are recognized as a liability on the consolidated balance sheet and measured at fair value.

The Company performed valuations of the warrants using a probability weighted Black-Scholes option pricing model which value was also
compared to a Binomial Option Pricing Model for reasonableness. This model requires input of assumptions including the risk-free interest
rates,  volatility,  expected  life  and  dividend  rates,  and  has  also  considered  the  likelihood  of  “down-round”  financings.  Selection  of  these
inputs involves management’s judgment and may impact net income. Due to our limited operating history and limited number of sales of
our  common  stock,  we  estimate  our  volatility  based  on  a  number  of  factors  including  the  volatility  of  comparable  publicly  traded
pharmaceutical  companies.  The  volatility  factor  used  in  the  Black-Scholes  option  pricing  model  has  a  significant  effect  on  the  resulting
valuation of the derivative liabilities on our balance sheet.

See report of independent accounting firm

F-13

 
 
 
 
 
 
 
 
 
 
 
 
 
The  table  below  presents  the  changes  in  the  derivative  warrant  liability  for  the  years  ended  September  30,  2017  and  2016,  which  were
measured at fair value on a recurring basis and classified as Level 3 in the fair value hierarchy (see Note 4). No warrants are classified as
derivative warrant liabilities as of September 30, 2018 and 2017:

Derivative warrant liability, beginning of year

Fair value of warrants issued
Total realized/unrealized losses (gains) included in net loss
Reclassification of liability to additional paid-in capital

Derivative warrant liability, end of year

7. COMMON STOCK, STOCK OPTIONS AND WARRANTS

Private Offerings and Common Stock Issued for Services and Release Agreements

2017
1,681,973    $
641,385     
(452,147)    
(1,871,211)    
-    $

2016

738,955 
1,198,564 
838,219 
(1,093,765)
1,681,973 

  $

  $

During the year ended September 30, 2016, the Company sold 290,000 Units for a purchase price of $8.10 per Unit and 17,778 Units for a
purchase price of $9.00 per Unit for gross proceeds of $2,509,000. There was no placement agent for these private placements and other
cash  expenses  related  to  the  placements  were  $81,312.  In  connection  with  these  placements,  the  Company  credited  $1,229,124  to
stockholders’ equity and $1,198,564 to derivative warrant liability.

On March 22, 2016, the Company sold 333,333 shares of common stock at $9.00 per share to its Chairman of the Board, Leonard Mazur,
for gross proceeds of $3,000,000. There were no expenses related to this placement.

In  February  2017,  the  Company  completed  its  2016  Offering.  The  Company  sold  128,017  units  at  $6.00  per  unit  for  gross  proceeds  of
$768,100. Each unit consisted of (i) one share of common stock and (ii) a five-year warrant to purchase one share of common stock at an
exercise price of $8.25 per share. The placement agent received a 10% cash commission on the gross proceeds, an expense allowance equal
to 3% of the proceeds, and warrants to purchase 12,802 shares of common stock at an exercise price of $8.25 per share. The estimated fair
value  of  the  128,017  warrants  issued  to  the  investors  was  $587,592  and  the  estimated  fair  value  of  the  12,802  warrants  issued  to  the
placement agent was $58,759. The placement agent commissions and expense allowance was $99,853. Other costs of the placement were
$176,896.

See report of independent accounting firm

F-14

 
 
 
 
 
   
 
   
   
   
 
 
 
 
 
 
During January 2017, the Company issued 29,729 shares of its common stock for investor relations services. The $298,774 fair value of the
common stock was expensed during the year ended September 30, 2017.

On May 5, 2017, the Company issued 11,400 shares of common stock valued at $77,748 in connection with a settlement agreement and
release  with  a  consultant  that  had  an  agreement  with  Leonard-Meron  Biosciences.  The  Company  expensed  the  $77,748  as  a  settlement
expense during the year ended September 30, 2017.

On  June  7,  2017,  the  Company  entered  into  a  release  agreement  with  the  placement  agent  for  the  2016  Offering.  The  placement  agent
consented to future financings and waived certain covenants contained in the 2016 Offering agreements. As consideration for the release,
the Company issued 6,668 shares of common stock valued at $45,476 to the placement agent. The Company expensed the $45,476 as a
settlement expense during the year ended September 30, 2017.

On June 8, 2017, the Company entered into release agreements with the investors in the 2016 Offering where each investor released the
Company  from  the  restrictions  included  in  the  unit  purchase  agreements.  In  exchange,  the  Company  agreed  that  (i)  in  the  event  that  a
financing is conducted at a price per share or price per unit lower than $6.00, then the Company will issue additional shares to each investor
sufficient to effectively reprice the sale of the 2016 Offering units to the lower price; (ii) in the event that the financing is conducted at a
price per share or price per unit less than the $8.25 exercise price of the warrants issued in the 2016 Offering then the exercise price of the
warrants shall be reduced to the lower price; and (iii) the Company will give each investor no less than 6 hours of notice before the closing
of any subsequent financing, through and including the Company’s 2017 registered public offering, and each investor shall have a 6-hour
option  to  purchase  up  to  20%  of  the  securities  sold  in  such  offering.  In  connection  with  these  agreements  the  Company  reclassified  the
$641,385 fair value of the 140,819 warrants issued in the 2016 Offering to derivative warrant liability on June 8, 2017 (see Note 6). On
August 8, 2017, the Company completed the 2017 public offering and issued 58,191 shares of common stock to the investors in the 2016
Offering to reprice the sale of the 2016 Offering units to $4.125 per unit and repriced the 2016 Offering Warrants to an exercise price of
$4.125 per share. During the year ended September 30, 2017, the Company recorded a settlement expense of $161,771 in connection with
the issuance of the additional 58,191 shares of common stock and reclassified the current fair value of the warrants to additional paid-in
capital.

On  February  7,  2018,  the  Company  issued  22,200  shares  of  common  stock  for  services  provided  by  two  consultants  and  expensed  the
$88,800 fair value of the common stock issued.

On April 1, 2018, the Company issued 10,000 shares of common stock for services provided by a consultant and expensed the $31,000 fair
value of the common stock issued.

2017 Public Offering and Release Agreement

On August 8, 2017, the Company closed an underwritten public offering of 1,648,484 shares of common stock and warrants to purchase
1,648,484 shares of common stock at an offering price of $4.125 per share and $0.01 per warrant. The warrants have a per share exercise
price of $4.125, are exercisable immediately and will expire five years from the date of issuance.  Gross proceeds were $6,802,469, before
deducting  underwriting  discounts  and  commissions  and  other  estimated  offering  expenses  of  $685,573.  The  Company  granted  the
underwriters a 45-day option to purchase up to an additional 247,272 shares of common stock and warrants to purchase 247,272 shares of
common stock to cover over-allotments, if any. On August 8, 2017, the underwriters partially exercised the over-allotment to purchase an
additional 247,272 warrants. The estimated fair value of the 1,895,756 warrants issued to the investors was $4,160,195 and the estimated
fair value of the 65,940 warrants issued to the underwriters was $142,419.

On November 7, 2017, the Company entered into a release agreement with the underwriter. The Company had previously granted a right of
first  refusal  to  underwrite  all  equity  and  debt  offerings  for  a  period  of  twelve  months  following  completion  of  the  2017  public  offering
(“Right  of  First  Refusal”).  Under  the  release,  the  Company  agreed  to  pay  the  underwriter  $100,000  in  cash  and  issue  60,000  shares  of
restricted  common  stock  with  a  fair  value  of  $257,400  in  exchange  for  a  full  release  from  all  obligations  related  to  the  Right  of  First
Refusal. The Company expensed the $357,400 cost of the release agreement in November 2017.

See report of independent accounting firm

F-15

 
 
 
 
 
 
 
 
 
 
 
Registered Direct/Private Placement Offerings

On December 19, 2017, the Company closed a registered direct offering with several institutional and accredited investors for the sale of
1,280,360 shares of common stock at $4.6925 per share for gross proceeds of $6,008,089. Simultaneously, the Company sold the investors
640,180 immediately exercisable five and a half year warrants at $4.63 per share. The Company paid the placement agent for the offering a
fee  of  7%  of  the  gross  proceeds  totaling  $420,566  and  issued  the  placement  agent  89,625  immediately  exercisable  five-year  warrants  at
$5.8656 per share. The Company also reimbursed the placement agent for $85,000 in expenses and incurred $20,000 in other expenses. Net
proceeds from the offering were $5,482,523. The estimated fair value of the 640,180 warrants issued to the investors was $2,407,276 and
the estimated fair value of the 89,625 warrants issued to the placement agent was $316,071.

On March 29, 2018, the Company closed a registered direct offering with an institutional and an accredited investor for the sale of 669,504
shares of common stock at $2.985 per share for gross proceeds of $1,998,469. Simultaneously, the Company sold to the investors 669,504
immediately exercisable five and a half year warrants at $2.86 per share. The Company paid the placement agent for the offering a fee of
7% of the gross proceeds totaling $139,893 and issued the placement agent 46,866 immediately exercisable five-year warrants at $3.73125
per  share.  The  Company  also  reimbursed  the  placement  agent  for  $85,000  in  expenses  and  incurred  $10,000  in  other  expenses.  Net
proceeds from the offering were $1,763,576. The estimated fair value of the 669,504 warrants issued to the investors was $1,679,482 and
the estimated fair value of the 46,866 warrants issued to the placement agent was $110,511.

August 2018 Offering

On August 13, 2018, Citius closed an underwritten offering of (i) 5,521,569 units, each unit consisting of one share of common stock and
one  immediately  exercisable  five-year  warrant  to  purchase  one  share  at  $1.15  per  share,  and  (ii)  2,321,569  pre-funded  units,  each  pre-
funded unit consists of one pre-funded warrant to purchase one share and one immediately exercisable five-year warrant to purchase one
share at $1.15 per share. The pre-funded warrants included in the pre-funded units are immediately exercisable at a price of $0.01 per share
and  do  not  expire.  The  offering  price  was  $1.275  per  unit  and  $1.265  per  pre-funded  unit.  The  net  proceeds  of  the  offering  were
$8,926,786. The Company issued underwriter warrants to purchase up to 549,020 shares at $1.59375 per share with an estimated fair value
of $491,737. The underwriter warrants are exercisable following February 8, 2019 and expire on August 8, 2023. The estimated fair value
of the 2,321,569 pre-funded warrants was $2,630,072, and the estimated fair value of the 7,843,138 warrants included in the units and the
pre-funded units issued to the investors was $7,311,727.

Unit Purchase Options

On April 7, 2017, the Company issued a three-year Unit Purchase Option Agreement to a consultant for 38,000 units at a purchase price of
$9.00 per unit. Each unit consists of one share of common stock and a warrant to purchase one share of common stock at an exercise price
of $9.00 per share which expires on the earlier of three years after exercise of the Unit Purchase Option Agreement or April 7, 2023. The
consultant  provided  the  Company  with  business  development  and  financing  assistance  for  the  three  months  ended  June  30,  2017.  The
Company estimated the fair value of the unit purchase option agreement at $104,138 and expensed it during the year ended September 30,
2017.

On June 29, 2017, the Company issued a three-year Unit Purchase Option Agreement to a consultant for 62,667 units at a purchase price of
$9.00 per unit. Each unit consists of one share of common stock and a warrant to purchase one share of common stock at an exercise price
of $9.00 per share which expires on the earlier of three years after exercise of the Unit Purchase Option Agreement or June 29, 2022. The
consultant  will  provide  the  Company  with  business  development  and  financing  assistance  through  December  31,  2017.  The  Company
estimated the fair value of the unit purchase option agreement at $193,860 and recorded it as a prepaid expense. The Company recorded an
expense of $96,930 for this agreement during the year ended September 30, 2017 and expensed the remaining balance of $96,930 during
the year ended September 30, 2018.

See report of independent accounting firm

F-16

 
 
 
 
 
 
 
 
 
 
Stock Option Plans

On September 12, 2014, the Board of Directors adopted the 2014 Stock Incentive Plan (the “2014 Plan”) and reserved 866,667 shares of
common stock for issuance to employees, directors and consultants. On September 12, 2014, our stockholders approved the plan. Pursuant
to  the  2014  Plan,  the  Board  of  Directors  (or  committees  and/or  executive  officers  delegated  by  the  Board  of  Directors)  may  grant  stock
options, stock appreciation rights, restricted stock, restricted stock units, other stock-based awards and cash-based awards. As of September
30, 2018, there were options to purchase 856,039 shares outstanding under the 2014 Plan, options to purchase 4,829 shares were exercised,
and 5,799 shares were available for future grants.

On  February  7,  2018,  our  stockholders  approved  the  2018  Omnibus  Stock  Incentive  Plan  (the  “2018  Plan”)  and  the  Company  reserved
2,000,000 shares of common stock for issuance to employees, directors and consultants. Pursuant to the 2018 Plan, the Board of Directors
(or committees and/or executive officers delegated by the Board of Directors) may grant stock options, stock appreciation rights, restricted
stock, restricted stock units, other stock-based awards and cash-based awards. As of September 30, 2018, there were options to purchase
745,000 shares outstanding under the 2018 Plan and 1,255,000 shares were available for future grants.

The fair value of each stock option award is estimated on the date of grant using the Black-Scholes option pricing model. Due to its limited
operating history and limited number of sales of its common stock, the Company estimated its volatility in consideration of a number of
factors  including  the  volatility  of  comparable  public  companies.  The  risk-free  interest  rate  is  based  on  the  U.S.  Treasury  yield  curve  in
effect at the time of grant commensurate with the expected term assumption. The expected term of stock options granted to employees and
directors, all of which qualify as “plain vanilla,” is based on the average of the contractual term (generally 10 years) and the vesting period.
For non-employee options, the expected term is the contractual term.

The following assumptions were used in determining the fair value of stock option grants for the years ended September 30, 2018, 2017
and 2016:

2018

2017

2016

Risk-free interest rate
Expected dividend yield
Expected term
Expected volatility

2.78 – 2.99 %   
%   

0
    6.50 – 10 years 
116

%   

1.79 – 1.90 %    0.95 – 1.40 %
%

%   

0
    4.75 – 9 years 

0
    6.50 – 10 years 

85 – 108 %   

57 – 74 %

A summary of option activity under the 2014 Plan and 2018 Plan is presented below:

Outstanding at September 30, 2017
Granted
Exercised
Forfeited or expired
Outstanding at September 30, 2018
Exercisable at September 30, 2018

Weighted-
Average
Exercise
Price

Weighted-
Average
Remaining
Contractual

Term    

Aggregate
Intrinsic
Value

6.69     
1.63     
—     
3.45     
4.35     
7.15     

8.56 years    $
7.10 years    $

173,291 
112,541 

Shares

861,039    $
745,000     
—     
(5,000)    
1,601,039    $
729,675    $

See report of independent accounting firm

F-17

 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
   
   
 
 
 
 
   
   
 
   
      
  
   
      
  
   
      
  
   
      
  
   
   
 
On March 30, 2016, the Company assumed stock options to purchase 77,252 shares of common stock in connection with the acquisition of
LMB. The LMB option holders received stock options to purchase 71,217 shares at an exercise price of $0.01 per share and 6,035 shares at
an exercise price of $13.65 per share. Pursuant to the original grants, options to purchase 4,829 shares were immediately vested and options
to purchase 72,423 shares vest over three years. These options all had original terms of 10 years.

On  June  23,  2016,  the  Board  of  Directors  granted  stock  options  to  four  directors.  Each  director  received  an  option  to  purchase  13,333
shares of common stock at an exercise price of $12.00 per share in consideration for their services. These options vest in full on June 23,
2017 and have a term of 10 years.

In July 2016, the Board of Directors granted stock options to purchase a total of 138,267 shares to three employees at prices ranging from
$10.50 to $13.50 per share. These options vest over terms of 19 to 36 months and have a term of 10 years.

On January 1, 2017, the Board of Directors granted stock options to purchase a total of 8,669 shares to four consultants at $10.05 per share.
These options vest over terms of 12 to 36 months and have a term of 10 years.

In September 2017, the Board of Directors granted stock options to purchase a total of 225,000 shares to 12 employees and 50,000 options
to two consultants at $3.45 per share. These options vest over terms of 12 to 36 months and have a term of 10 years.

In September 2018, the Board of Directors granted stock options to purchase a total of 520,000 shares to six employees, 75,000 options to
five directors, and 80,000 options to three consultants at $1.62 per share. In addition, the Board granted stock options to purchase 70,000
shares to a financial consultant at $1.75 per share. These options vest over terms of 12 to 36 months and have a term of 10 years.

Stock-based  compensation  expense  for  the  years  ended  September  30,  2018,  2017  and  2016  was  $779,701,  $986,620  and  $732,151,
respectively.

At September 30, 2018, unrecognized total compensation cost related to unvested awards of $1,425,957 is expected to be recognized over a
weighted average period of 2.3 years.

See report of independent accounting firm

F-18

 
 
 
 
 
 
 
 
 
 
Warrants

The Company has reserved 15,193,192 shares of common stock for the exercise of outstanding warrants. The following table summarizes
the warrants outstanding at September 30, 2018:

Investor and Placement Agent Warrants
Investor Warrants
Investor Warrants
LMB Warrants
LMB Warrants
LMB Warrants
LMB Warrants
LMB Warrants
Financial Advisor Warrants
2016 Offering Warrants
Convertible Note Warrants
2017 Public Offering Warrants
2017 Public Offering Underwriter Warrants
December 2017 Registered Direct/Private
Placement Offering Investor Warrants
December 2017 Registered Direct/Private

Placement Offering Agent Warrants

March 2018 Registered Direct/Private Placement
Offering Investor Warrants
March 2018 Registered Direct/Private Placement
Offering Agent Warrants
August 2018 Offering Investor Warrants
August 2018 Offering Pre-Funded Unit Warrants
August 2018 Offering Agent Warrants

  $

Exercise
price

    Number

9.00     
9.00     
9.00     
6.15     
9.90     
20.70     
7.50     
7.50     
3.00     
4.13     
9.75     
4.13     
4.54     

384,006   
202,469   
307,778   
90,151   
8,155   
17,721   
73,883   
53,110   
25,833   
140,819   
40,436   
1,622,989   
65,940   

Expiration Dates
September 12, 2019
March 19, 2020 – September 14, 2020
November 5, 2020 – April 25, 2021
June 12, 2019 – March 2, 2021
September 30, 2019 – January 8, 2020
November 3, 2019 – March 6, 2020
August 18, 2020 – March 14, 2021
March 24, 2022 – April 29, 2022
August 15, 2021
November 23, 2021 – February 27, 2022
September 12, 2019
August 2, 2022
February 2, 2023

4.63     

640,180   

June 19, 2023

5.87     

89,625   

December 19, 2022

2.86     

669,504   

October 2, 2023

3.73     
1.15     
0.01     
1.59     

46,866   
7,843,138   
2,321,569   
549,020   

       15,193,192     

March 28, 2023
August 14, 2023
No expiration date
August 8, 2023

On  March  30,  2016,  the  Company  granted  warrants  to  purchase  243,020  shares  of  common  stock  in  connection  with  the  acquisition  of
LMB. The warrants have exercise prices between $6.15 and $20.70 per share. All warrants were vested at March 30, 2016. The fair value
of the warrants was estimated at $1,071,172 and has been included in the purchase price of LMB.

On August 16, 2016, the Company granted warrants to purchase 66,667 shares of common stock in connection with a one-year financial
advisory  agreement.  The  warrants  were  vested  on  issuance,  have  an  exercise  price  of  $3.00  per  share  and  are  exercisable  on  a  cash  or
cashless basis. The fair value of the warrants was estimated at $477,181 and recorded as a prepaid expense on the issuance date. During the
years ended September 30, 2017 and 2016, the Company expensed $417,181 and $60,000, respectively, in connection with the agreement.
During the year ended September 30, 2018, 40,834 warrants were exercised on a cashless basis resulting in the issuance of 16,547 shares of
common stock.

During the year ended September 30, 2017, the Company sold 128,017 2016 Offering Units, at a price of $6.00 per Unit, consisting of (i)
one share of common stock and (ii) a warrant to purchase one share of common stock. Each 2016 Offering Warrant had an exercise price of
$8.25 and is exercisable for five years from the date of issuance. Additionally, warrants to purchase 12,802 shares of common stock were
granted to the Placement Agent pursuant to the above pricing terms. On June 8, 2017, the Company entered into release agreements with
the investors and as a result the Company repriced the 2016 Offering Warrants to an exercise price of $4.125 per share on August 8, 2017.

On  June  7,  2017,  the  Company  issued  a  warrant  to  purchase  40,436  shares  of  common  stock  at  $9.75  per  share  in  settlement  of  issues
related to the July 31, 2014 conversion of a subordinated convertible promissory note. The Company charged the $119,402 estimated fair
value of the warrant to settlement expenses during the year ended September 30, 2017.

Effective  June  16,  2017,  the  Company  amended  warrants  associated  with  the  Leonard-Meron  Biosciences,  Inc.  2015  private  placement
offering.  The  warrant  amendments  removed  the  exercise  price  reset  provisions,  adjusted  the  exercise  price  of  the  warrants  to  $7.50  per
share and extended the term of the warrants by three years. The estimated fair value of the warrants on June 16, 2017 after the amendments
was $250,733. As a result of the amendment, the Company recorded an incremental cost of $71,488 as a settlement expense during the year
ended September 30, 2017.

See report of independent accounting firm

F-19

 
 
 
 
 
 
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
 
   
      
    
 
 
   
 
 
 
 
 
 
See  Note  7  above  for  descriptions  of  the  warrants  issued  in  the  2017  public  offering,  the  December  2017  and  March  2018  registered
direct/private placement offerings, and the August 2018 offering. During the year ended September 30, 2018, 272,767 of the 2017 public
offering warrants were exercised at $4.25 per share for net proceeds of $1,125,148.

At September 30, 2018, the weighted average remaining life of all of the outstanding warrants is 3.89 years, all warrants are exercisable,
and the aggregate intrinsic value for the warrants outstanding was $8,402,648. 

Common Stock Reserved 

A summary of common stock reserved for future issuances as of September 30, 2018 is as follows:

Stock plan options outstanding
Stock plan shares available for future grants
Warrants
Unit purchase options
Total

8. RELATED PARTY TRANSACTIONS

1,601,039 
1,260,799 
    15,193,192 
201,334 
    18,256,364 

The  Company’s  headquarters  were  previously  located  in  Maynard,  MA  in  the  office  space  of  a  company  affiliated  through  common
ownership. In connection with the March 30, 2016 acquisition of LMB, the Company moved its principal executive offices to Cranford,
NJ.  The  Company  did  not  record  any  revenue  or  expense  related  to  the  use  of  the  Maynard,  MA  office  space  as  management  has
determined the usage to be immaterial and the affiliate has not charged for the usage.

As  of  September  30,  2018  and  2017,  the  Company  owed  $0  and  $27,637  to  a  company  affiliated  through  common  ownership  for  the
expenses the related party paid on the Company’s behalf and services performed by the related party.

Our  Chairman  of  the  Board,  Leonard  Mazur,  is  the  cofounder  and  Vice  Chairman  of Akrimax  Pharmaceuticals,  LLC  (“Akrimax”),  a
privately held pharmaceutical company specializing in producing cardiovascular and general pharmaceutical products. The Company leases
office space from Akrimax (see Note 9).

Our  Chairman  of  the  Board,  Leonard  Mazur,  and  our  Chief  Executive  Officer,  Myron  Holubiak,  are  co-founders  and  were  significant
shareholders in LMB. In connection with the acquisition of LMB, our Chairman purchased an additional 333,333 shares of the Company.
See Note 5 for a description of related party debt transactions.

In connection with the 2017 Public Offering, Mr. Mazur purchased 421,400 units consisting of 421,400 shares of common stock at $4.125
per share and 421,400 warrants at $0.01 per warrant and converted certain notes payable to common stock (See Note 5).

In  connection  with  the  December  2017  Registered  Direct/Private  Placement  Offering,  Mr.  Mazur  purchased  213,106  shares  of  common
stock at $4.6925 per share and received 106,553 warrants exercisable at $4.63 per share. In connection with the March 2018 Registered
Direct/Private  Placement  Offering,  Mr.  Mazur  purchased  167,504  shares  of  common  stock  at  $2.985  per  share  and  received  167,504
warrants exercisable at $2.86 per share. The purchases were made on the same terms as for all other investors.

In connection with the August 2018 offering, Mr. Mazur purchased 3,137,255 shares of common stock at $1.275 per share and received
3,137,255 warrants exercisable at $1.15 per share, and Mr. Holubiak purchased 784,314 shares of common stock at $1.275 per share and
received 784,314 warrants exercisable at $1.15 per share. The purchases were made on the same terms as for all other investors.

See report of independent accounting firm

F-20

 
 
 
 
 
 
   
   
   
 
 
 
 
 
 
 
 
 
9. EMPLOYMENT AND CONSULTING AGREEMENTS

Employment Agreements

On October 19, 2017, the Company and Mr. Mazur, entered into an amended employment agreement with a three-year term. Under the
terms  of  the  amended  agreement,  the  Company  is  required  to  pay  base  compensation  plus  incentives  over  the  employment  term  plus
severance benefits upon the occurrence of certain events as described in the agreement.

On March 30, 2016, in connection with the acquisition of LMB, the Company entered into a three-year employment agreement with Myron
Holubiak  to  serve  as  Chief  Executive  Officer.  Upon  expiration,  the  agreement  automatically  renews  for  successive  periods  of  one-year.
The agreement requires the Company to pay base compensation plus incentives over the employment term plus severance benefits upon the
occurrence of certain events as described in the agreement.

The  Company  has  employment  agreements  with  certain  other  employees  that  require  the  Company  to  pay  base  compensation  plus
incentives over the employment term plus severance benefits upon the occurrence of certain events as described in the agreement.

Consulting Agreements

Effective September 1, 2014, the Company entered into three consulting agreements. Two of the agreements are for financial consulting
services including accounting, preparation of financial statements and filings with the SEC. The third agreement is for financing activities,
product development strategies and corporate development. The agreements may be terminated by the Company or the consultant with 90
days written notice.

Consulting expense under the agreements for the years ended September 30, 2018, 2017 and 2016 was $422,000, $372,000, and $460,000,
respectively.  Consulting  expense  for  the  years  ended  September  30,  2018,  2017  and  2016  includes  $48,000,  $48,000  and  $48,000,
respectively, paid to a financial consultant who is a stockholder of the Company. In addition, one financial consulting services agreement
provides  for  the  grant  of  options  to  purchase  33,333  shares  of  common  stock  contingent  upon  approval  by  the  Board  of  Directors.  The
options were granted on June 1, 2015.

10. FDA REFUND

On August 29, 2018, the Company received notification from the Food and Drug Administration (“FDA”) that the Company was being
refunded $818,343 of 2016 product and establishment fees because the fees paid by the Company exceeded the costs of the FDA’s review
of the associated Suprenza applications. The Company recorded as other income in the statements of operations the $818,343 receivable
from the FDA as of September 30, 2018. The Company received the refund in full on October 1, 2018.

11. COMMITMENTS AND CONTINGENCIES

Operating Lease

The Company leases office space from Akrimax, a related party (see Note 8), in Cranford, New Jersey at a monthly rental rate of $2,167
pursuant to an agreement which currently expires on April 30, 2019. Rent expense for the years ended September 30, 2018, 2017 and 2016
was $26,000, $26,000 and $13,002. Future minimum rentals for the year ending September 30, 2019 are $15,167.

See report of independent accounting firm

F-21

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Legal Proceedings

The Company is not involved in any litigation that we believe could have a material adverse effect on our financial position or results of
operations.  There  is  no  action,  suit,  proceeding,  inquiry  or  investigation  before  or  by  any  court,  public  board,  government  agency,  self-
regulatory organization or body pending or, to the knowledge of our executive officers, threatened against or affecting our company or our
officers or directors in their capacities as such.

12.  INCOME TAXES

There was no provision for federal or state income taxes for the years ended September 30, 2018, 2017 and 2016 due to the Company’s
operating losses and a full valuation reserve on deferred tax assets.

On December 22, 2017, the Tax Cuts and Jobs Act (the “Act”), was signed into law by the President of the United States. The Act includes
a  number  of  changes,  including  the  lowering  of  the  U.S.  corporate  tax  rate  from  35%  to  21%,  effective  January  1,  2018,  and  the
establishment  of  a  territorial-style  system  for  taxing  foreign-source  income  of  domestic  multinational  corporations.  The  Company  has
recognized provisional tax impacts related to the revaluation of the Company’s deferred tax assets and the impact of revaluation of those
deferred tax assets on the Company’s valuation allowance and included those amounts in the consolidated financial statements for the year
ended September 30, 2018. The actual impact of the Act may differ from the Company’s estimates due to, among other things, changes in
interpretations and assumptions made and guidance that may be issued as a result of the Tax Act.

The income tax benefit differs from the amount of income tax determined by applying the U.S. federal income tax rate to pretax income for
the years ended September 30, 2018, 2017 and 2016 due to the following:

Computed “expected” tax benefit
Increase (decrease) in income taxes resulting from:
State taxes, net of federal benefit
Permanent differences
Increase in the valuation reserve

2018

2017

2016

(24.5%)   

(35.0%)   

(35.0%)

(6.0%)   
0.0%    
30.5%    
0.0%    

(5.2%)   
1.3%    
38.9%    
0.0%    

(5.2%)
4.2%
36.0%
0.0%

Deferred  income  taxes  reflect  the  net  tax  effects  of  temporary  differences  between  the  carrying  amounts  of  assets  and  liabilities  for
financial reporting purposes and the amounts used for income tax purposes. Significant components of the Company’s deferred tax assets
and liabilities are as follows:

Deferred tax assets:
Net operating loss carryforward
Stock-based compensation
Valuation allowance
Deferred tax assets

September 30,
2018

September 30,
2017

  $

  $

8,962,000    $
1,350,000     
(10,312,000)    
—    $

7,123,000 
1,425,000 
(8,548,000)
— 

The Company has recorded a valuation allowance against deferred tax assets as the utilization of the net operating loss carryforward and
other deferred tax assets is uncertain.  During the years ended September 30, 2018, 2017 and 2016, the valuation allowance increased by
$1,764,000, $4,044,000 and $2,989,000, respectively. The increase in the valuation allowance during the years ended September 30, 2018,
2017 and 2016 was primarily due to the Company’s net operating loss offset by the decrease in the effective U.S. federal income tax rate
from 35% to 21%. At September 30, 2018, the Company has a net operating loss carryforward of approximately $29,344,000 which begins
expiring in 2034.

13. SUBSEQUENT EVENTS

Exercise of Pre-Funded Unit Warrants

On October 3, 2018 the Company received a notice of exercise for the purchase of 1,600,000 shares of common stock at $0.01 per share
pursuant to its pre-funded unit warrants issued in the August 2018 offering. Proceeds from the exercise were $16,000.

See report of independent accounting firm

F-22

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
   
  
   
  
   
  
   
   
   
 
   
  
 
 
 
   
 
   
      
  
   
   
 
 
 
 
 
Item 9. Changes in and Disagreements with Accountants on Accounting and Financial Disclosure

None.

Item 9A. Controls and Procedures

Disclosure Controls and Procedures

We  maintain  disclosure  controls  and  procedures  designed  to  provide  reasonable  assurance  that  information  required  to  be  disclosed  in
reports  filed  under  the  Securities  Exchange Act  of  1934,  as  amended  (the  “Exchange Act”),  is  recorded,  processed,  summarized  and
reported  within  the  specified  time  periods  and  accumulated  and  communicated  to  our  management,  including  our  principal  executive
officer and principal financial officer, as appropriate to allow timely decisions regarding disclosure.

Our Chief Executive Officer (who is our principal executive officer) and Chief Financial Officer (who is our principal financial officer and
principal accounting officer), evaluated the effectiveness of our disclosure controls and procedures (as defined in Rules 13a-15(e) and 15d-
15(e) promulgated under the Exchange Act) as of September 30, 2018, the end of our fiscal year. In designing and evaluating disclosure
controls and procedures, we recognize that any disclosure controls and procedures, no matter how well designed and operated, can only
provide  reasonable  assurance  of  achieving  the  desired  control  objective. As  of  September  30,  2018,  based  on  the  evaluation  of  these
disclosure  controls  and  procedures,  our  Chief  Executive  Officer  and  Chief  Financial  Officer  concluded  that  our  disclosure  controls  and
procedures were effective in ensuring that information required to be disclosed by us in reports that we file or submit under the Exchange
Act is recorded, processed, summarized, and reported within the time periods specified in the SEC’s rules and forms.

Management’s Annual Report on Internal Control over Financial Reporting

Our management is responsible for establishing and maintaining effective internal control over financial reporting as defined in Rule 13a-
15(f)  under  the  Exchange Act.  Because  of  its  inherent  limitations,  internal  control  over  financial  reporting  is  not  intended  to  provide
absolute  assurance  that  a  misstatement  of  our  financial  statements  would  be  prevented  or  detected.  Under  the  supervision  of  our  Chief
Executive  Officer  and  Chief  Financial  Officer,  the  Company  conducted  an  evaluation  of  the  effectiveness  of  our  internal  control  over
financial  reporting  as  of  September  30,  2018  using  the  criteria  established  in  Internal  Control—Integrated  Framework  issued  by  the
Committee of Sponsoring Organizations of the Treadway Commission (“COSO”) (2013 Framework).

Based  on  this  evaluation,  management  has  concluded  that  our  internal  controls  were  effective  and  that  we  maintained  effective  controls
over our financial reporting as of September 30, 2018.

Because of its inherent limitations, internal control over financial reporting may not prevent or detect misstatements. Also, projections of
any  evaluation  of  effectiveness  to  future  periods  are  subject  to  the  risks  that  controls  may  become  inadequate  because  of  changes  in
conditions, or that the degree of compliance with the policies or procedures may deteriorate.

Changes in Internal Controls over Financial Reporting

In the fourth quarter of fiscal 2018, as part of our then ongoing efforts to remediate the material weaknesses in our internal controls over
financial  reporting,  we  completed  documenting  various  policies  and  procedures,  and  implemented  sufficient  separation  of  duties  by
developing  appropriate  review,  signoffs  and  grants  of  authority,  as  well  as  consolidating  key  financial  functions  which  are  administered
solely  by  employees  at  our  Company’s  Cranford,  New  Jersey  office. As  a  result  of  these  remedial  efforts,  our  management  was  able  to
determine that our internal controls over financial reporting were effective as of September 30, 2018.

Other than as described above, there were no other changes in our internal controls over financial reporting during the fourth quarter of
fiscal 2018 that materially affected, or are reasonably likely to materially affect, our internal control over financial reporting.

ITEM 9B. Other Information. 

None.

38

 
 
 
 
 
 
 
  
 
 
 
 
 
 
 
 
 
ITEM 10. DIRECTORS, EXECUTIVE OFFICERS AND CORPORATE GOVERNANCE

PART III

We have adopted a written Code of Ethics and  Business  Conduct  that  applies  to  our  directors,  officers  and  all  employees.  We  intend  to
disclose any amendments to, or waivers from, our code of ethics and business conduct that are required to be publicly disclosed pursuant to
rules of the SEC by filing such amendment or waiver with the SEC. This code of ethics and business conduct can be found in the “Investors
- Corporate Governance” section of our website, www.citiuspharma.com.

The  other  information  required  by  this  Item  concerning  our  directors  and  executive  officers  is  incorporated  by  reference  to  the  section
captioned “Proposal No. 1—Election of Directors” and “Corporate Governance” to be contained in our proxy statement related to the 2019
Annual Meeting of Stockholders (the “Proxy Statement”), which information is expected to be filed with the SEC within 120 days of the
end of our fiscal year pursuant to General Instruction G(3) of Form 10-K. The information required by this Item concerning compliance
with  Section  16(a)  of  the  Exchange Act  by  our  directors,  executive  officers  and  persons  who  own  more  than  10%  of  our  outstanding
common stock is incorporated by reference from the section captioned “Section 16(a) Beneficial Ownership Reporting Compliance” to be
contained in the Proxy Statement.

ITEM 11. EXECUTIVE COMPENSATION

The  information  required  by  this  Item  concerning  directors  and  executive  compensation  is  incorporated  by  reference  from  the  sections
captioned “Director Compensation” and “Executive Compensation”, respectively, to be contained in the Proxy Statement.

ITEM  12.  SECURITY  OWNERSHIP  OF  CERTAIN  BENEFICIAL  OWNERS  AND  MANAGEMENT  AND  RELATED
STOCKHOLDER MATTERS

The following table sets forth the indicated information as of September 30, 2018 with respect to our equity compensation plans: 

Plan Category
Equity compensation plans approved by security holders

2014 Stock Incentive Plan
2018 Omnibus Stock Incentive Plan

Total

Number of
securities to
be issued
upon
exercise of
outstanding
options,
warrants
and rights    

Weighted-
average
exercise price
of outstanding
options,
warrants and
rights

Number of
securities
remaining
available for
future
issuance
under equity
compensation
plans

856,039    $
745,000    $

6.71     
1.63     

5,799 
1,255,000 

1,601,039    $

4.35     

1,260,799 

Our equity compensation plans consist of the Citius Pharmaceuticals, Inc. 2018 Omnibus Stock Incentive Plan and 2014 Stock Incentive
Plan, which were both approved by our stockholders. We do not have any equity compensation plans or arrangements that have not been
approved by our stockholders.

The  other  information  required  by  this  Item  is  incorporated  by  reference  to  the  information  under  the  section  captioned  “Security
Ownership of Certain Beneficial Owners and Management” contained in the Proxy Statement.

ITEM 13. CERTAIN RELATIONSHIPS AND RELATED TRANSACTIONS, AND DIRECTOR INDEPENDENCE

The information required by this Item is incorporated by reference to the information under the section captioned “Certain Relationships
and Related Transactions” and “Proposal No. 1—Election of Directors” to be contained in the Proxy Statement.

ITEM 14. PRINCIPAL ACCOUNTING FEES AND SERVICES

The  information  required  by  this  Item  is  incorporated  by  reference  to  the  information  under  the  section  captioned  “Auditor  and Audit
Committee Matters” to be contained in the Proxy Statement.

39

 
 
 
 
 
 
 
 
 
 
 
   
 
   
      
      
  
   
   
 
   
      
      
  
   
 
 
 
 
 
 
 
PART IV

Item 15. Exhibits, Financial Statement Schedules

Exhibit
Number
2.1

Description of Document

  Share Exchange and Reorganization Agreement, among Citius

Pharmaceuticals, LLC, Trail One, Inc. and the beneficial holders of
the membership interests of Citius Pharmaceuticals, LLC identified
in the Agreement, dated as of September 12, 2014.

Registrant’s
Form
8-K

Dated
9/18/2014

Exhibit
Number  
2.1

Filed
Herewith

2.2

  Agreement and Plan of Merger among Citius LMB Acquisition

8-K

4/5/2016

3.1

3.2

Corporation, Leonard-Meron Biosciences, Inc. and Citius
Pharmaceuticals Holdings, Inc., dated March 30, 2016.
  Amended and Restated Articles of Incorporation of Citius

Pharmaceuticals, Inc.

  Certificate of Amendment to the Amended and Restated Articles of
Incorporation of Citius Pharmaceuticals, Inc., effective September
16, 2016.

8-K

8-K

9/18/2014

9/21/2016

3.3

  Certificate of Amendment to the Amended and Restated Articles of

8-K

6/8/2017

2.1

3.1

3.1

3.1

3.4
4.1

Incorporation of Citius Pharmaceuticals, Inc., effective June 9,
2017.

  Amended and Restated Bylaws of Citius Pharmaceuticals, Inc.
  Form of Registration Rights Agreement between the Purchasers
named therein and Citius Pharmaceuticals Holdings, Inc., dated
September 12, 2014.

8-K
8-K

2/9/2018
9/18/2014

3.1
10.2

4.2

  Placement Agent’s Unit Warrant in favor of Merriman Capital, Inc.,

S-1/A

12/29/2015

10.12

dated September 12, 2014.

4.3
4.4
4.5
4.6
4.7
4.8
4.9
4.10 
4.11

  Form of Investor Warrant, dated September 12, 2014.
  Form of Common Stock Purchase Warrant, dated May 10, 2017.
  Form of Representative’s Warrant, dated August 3, 2017.
  Form of Investor Warrant, dated December 15, 2017.
  Form of Placement Agent Warrant, dated December 15, 2017.
  Form of Investor Warrant, dated March 28, 2018.
  Form of Placement Agent Warrant, dated March 28, 2018.
  Form of Common Stock Purchase Warrant, dated August 13, 2018.
  Form of Pre-Funded Common Stock Purchase Warrant, dated

August 13, 2018.

4.12 

  Form of Underwriter’s Common Stock Purchase Warrant, dated

August 13, 2018.

8-K
10-Q
8-K
8-K
8-K
8-K
8-K
8-K
8-K

8-K

9/18/2014
5/15/2017
8/4/2017
  12/19/2017  
  12/19/2017  
3/29/2018
3/29/2018
8/13/2018
8/13/2018

8/13/2018

10.1

  Collaboration and License Agreement between Alpex Pharma S.A.

S-1/A

10/16/2015

and Citius Pharmaceuticals, LLC, dated June 12, 2008.

10.2

  Product Development and Pilot Lot Manufacturing Proposal

S-1/A

10/16/2015

Version 01 between IGI, Inc. and Citius Pharmaceuticals, Inc.,
dated July 21, 2010.

10.3

  Exclusive License Agreement between Prenzamax, LLC and Citius

S-1/A

10/16/2015

Pharmaceuticals, Inc., dated November 15, 2011.

10.4

  Amendment and Coordination Agreement among Prenzamax LLC,
Akrimax Pharmaceuticals, LLC, Citius Pharmaceuticals LLC and
Alpex Pharma S.A., dated November 15, 2011.

S-1/A

10/16/2015

10.3
10.4
4.2
4.1
4.2
4.1
4.2
4.1
4.2

4.3

10.6

10.9

10.8

10.5

 10.5

  Supply Agreement between Prenzamax, LLC and Alpex Pharma

S-1/A

10/16/2015

10.10

S.A., dated November 15, 2011.

10.6

  Technical and Quality Agreement among Citius Pharmaceuticals
LLC, Alpex Pharma S.A. and Akrimax Pharmaceuticals, LLC,
dated November 15, 2011.

S-1/A

10/16/2015

10.11

40

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
  
Exhibit
Number
10.7

  Description of Document
  Consultant Services Agreement between Neeta Wadekar and Citius

Pharmaceuticals, Inc., dated September 1, 2014.

10.8

  Employment Agreement between Leonard Mazur and Citius

Pharmaceuticals, Inc., dated September 12, 2014.

10.9
10.10

  Citius Pharmaceuticals, Inc. 2014 Stock Incentive Plan.
  Form of Citius Pharmaceuticals, Inc. 2014 Stock Incentive Plan

Nonqualified Stock Option.

10.11

  Employment Agreement between Myron Holubiak and Citius

Pharmaceuticals, Inc., executed March 30, 2016, effective March 1,
2016.

Registrant’s
Form
S-1/A

10-K

10-Q
10-Q

8-K

Dated
10/16/2015

12/29/2014

8/15/2016
8/15/2016

4/5/2016

Exhibit
Number  
10.7

Filed
Herewith

10.4

10.1
10.2

10.2

10.12

  Voting Agreement among Citius Pharmaceuticals, Inc., Leonard

8-K

4/5/2016

10.3

Mazur and certain other stockholders of the Company, dated March
30, 2016.

10.13

  Form of Unit Purchase Agreement, between each investor and

Citius Pharmaceuticals, Inc., dated September 27, 2016.

10.14

  Placement Agency Agreement between Garden State Securities, Inc.

10.15

and Citius Pharmaceuticals, Inc., dated September 27, 2016.

  Amendment to Placement Agency Agreement between Garden State
Securities, Inc. and Citius Pharmaceuticals, Inc., dated November
23, 2016.

10-Q

10-Q

10-Q

5/15/2017

5/15/2017

5/15/2017

10.5

10.6

10.7

10.16

  Second Amendment to the Patent and Technology License

10-Q

5/15/2017

10.8

Agreement between Novel Anti-Infective Technologies, LLC and
Leonard-Meron Biosciences, Inc., dated March 20, 2017.

10.17

  Future Advance Convertible Promissory Note between Leonard
Mazur and Citius Pharmaceuticals, Inc.,  dated May 10, 2017.

10.18

  Conversion Agreement between Leonard Mazur and Citius

Pharmaceuticals, Inc., dated May 10, 2017.

10.19

  Amended and Restated Demand Convertible Promissory Note

between Leonard Mazur and Citius Pharmaceuticals, Inc., dated
May 10, 2017.

10.20

  Release Agreement between Garden State Securities, Inc. and Citius

Pharmaceuticals, Inc., dated June 7, 2017.

10.21

  Form of Release Agreement between Citius Pharmaceuticals, Inc.

and each investor, dated June 8, 2017.

10.22

  Warrant Agent Agreement between VStock Transfer, LLC and

Citius Pharmaceuticals, Inc., dated August 3, 2017.

10.23

  Amended and Restated Employment Agreement between Leonard
Mazur and Citius Pharmaceuticals, Inc., dated October 19, 2017.

10-Q

10-Q

10-Q

8-K

8-K

8-K

--

5/15/2017

5/15/2017

5/15/2017

6/13/2017

6/13/2017

8/4/2017

--

10.24

  Release Agreement between Aegis Capital Corp. and Citius

10-Q

2/14/2018

Pharmaceuticals, Inc., dated November 7, 2017.

10.25

  Employment Agreement between Jaime Bartushak and Citius

Pharmaceuticals, Inc., dated November 27, 2017.

10.26

  Form of Securities Purchase Agreement between Citius

Pharmaceuticals, Inc. and the purchasers named therein, dated
December 15, 2017.

10.27 

  Engagement Letter between H.C. Wainwright & Co., LLC and

Citius Pharmaceuticals, Inc., dated December 15, 2017.

10.28
10.29

  Citius Pharmaceuticals, Inc. 2018 Omnibus Stock Incentive Plan
  Form of Securities Purchase Agreement between Citius

Pharmaceuticals, Inc. and the purchasers named therein, dated
March 28, 2018.

8-K

8-K

8-K 

10-Q
8-K

12/1/2017

12/19/2017

12/19/2017

2/14/2018
3/29/2018

10.1

10.2

10.3

10.1

10.2

4.1

--

10.1

10.1

10.1

10.2

10.2
10.1

10.30 

  Engagement Letter between H.C. Wainwright & Co., LLC and

8-K 

3/29/2018 

10.2

Citius Pharmaceuticals, Inc., dated March 28, 2018.

21
23.1
31.1

  Subsidiaries.
  Consent of Independent Registered Public Accounting Firm.
  Certification of the Chief Executive Officer pursuant to Exchange

Act Rule 13a-14(a).

10-K
--

--

  12/13/2017  
--

--

21
--

--

X

X

X

41

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
  
Exhibit
Number
31.2

  Description of Document
  Certification of the Chief Financial Officer pursuant to Exchange

Act Rule 13a-14(a).

32.1

  Certification of the Chief Executive Officer pursuant to 18 U.S.C.

1350, as adopted pursuant to Section 906 of the Sarbanes Oxley Act
of 2002.

32.2

  Certification of the Chief Financial Officer pursuant to 18 U.S.C.

1350, as adopted pursuant to Section 906 of the Sarbanes Oxley Act
of 2002.

EX-
101.INS*
EX-
101.SCH*
EX-
101.CAL*
EX-
101.DEF*
EX-
101.LAB*
EX-
101.PRE*

  XBRL INSTANCE DOCUMENT

  XBRL TAXONOMY EXTENSION SCHEMA DOCUMENT

  XBRL TAXONOMY EXTENSION CALCULATION LINKBASE  

  XBRL TAXONOMY EXTENSION DEFINITION LINKBASE

  XBRL TAXONOMY EXTENSION LABELS LINKBASE

  XBRL TAXONOMY EXTENSION PRESENTATION LINKBASE  

Registrant’s
Form

Dated

Exhibit
Number  

Filed
Herewith

--

--

--

--

--

--

--

--

--

--

--

--

--

--

--

--

--

--

--

--

--

--

--

--

--

--

--

X

X

X

X

X

X

X

X

X

*

Pursuant to Rule 406T of Regulation S-T, the Interactive Data Files in Exhibit 101 hereto are deemed not filed or part of a registration
statement or prospectus for purposes of Sections 11 or 12 of the Securities Act of 1933, as amended, are deemed not filed for purposes
of Section 18 of the Securities Exchange Act of 1934, as amended, and otherwise are not subject to liability under those sections.

42

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Pursuant to the requirements of the Securities Exchange Act of 1934, the registrant has duly caused this report to be signed on its behalf by
the undersigned, thereunto duly authorized.

Signatures

Date: December 11, 2018

CITIUS PHARMACEUTICALS, INC.

By: /s/ Myron Holubiak
  Myron Holubiak

President and Chief Executive Officer
(Principal Executive Officer)

In accordance with the Exchange Act, this Report has been signed below by the following persons on behalf of the Registrant and in the
capacities and on the dates indicated.

Signature

/s/ Leonard Mazur
Leonard Mazur

/s/ Myron Holubiak
Myron Holubiak

/s/ Jaime Bartushak
Jaime Bartushak

/s/ Suren Dutia
Suren Dutia

/s/ Carol Webb
Carol Webb

/s/ William Kane
William Kane

/s/ Howard Safir
Howard Safir

/s/ Eugene Holuka
Eugene Holuka

Title

Date

  Executive Chairman of the Board of Directors

December 11, 2018

  President and Chief Executive Officer and Director

December 11, 2018

(Principal Executive Officer)

  Chief Financial Officer and Chief Accounting Officer
  (Principal Financial Officer and Principal Accounting

December 11, 2018

Officer)

  Director

  Director

  Director

  Director

  Director

43

December 11, 2018

December 11, 2018

December 11, 2018

December 11, 2018

December 11, 2018

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
 
 
 
   
 
 
 
   
 
 
 
   
 
 
 
   
 
 
 
 
 
 
   
 
 
 
   
 
 
 
   
 
 
 
   
 
 
 
   
 
 
 
   
 
 
 
   
 
 
 
   
 
 
 
   
 
 
 
   
 
 
 
 
Exhibit 10.23

AMENDED AND RESTATED EMPLOYMENT AGREEMENT

This Employment Agreement (the “Agreement”) is made as of October 19, 2017 (the “Effective Date”), by and between Citius
Pharmaceuticals, Inc. (the “Employer”), and Leonard L. Mazur (the “Executive”). In consideration of the mutual covenants contained in
this Agreement, the Employer and the Executive agree as follows:

1. Employment. The Employer agrees to employ the Executive and the Executive agrees to be employed by the Employer on the

terms and conditions set forth in this Agreement.

2. Term. The initial term (the “Initial Term”) of this Agreement shall begin as of the Effective Date and shall continue for three (3)
years,  until  the  third  anniversary  of  the  Effective  Date,  unless  sooner  terminated  by  either  party  as  set  forth  below.  Effective  upon  the
expiration of the Initial Term and of each Renewal Term (as defined below), if any, the term of this Agreement shall automatically renew
for successive periods of one-year (each, a “Renewal Term”) unless the Employer gives written notice to the Executive at least ninety (90)
days prior to the end of the Initial Term or at least ninety (90) days prior to the end of any Renewal Term that the term of the Agreement
shall not be further extended. As used in this Agreement, the “Term” shall refer to the Initial Term and any Renewal Term.

3. Capacity. The Executive shall serve as Executive Chairman of the Employer’s Board (as defined below). The Executive shall
also  serve  the  Employer  in  such  other  or  additional  offices  as  the  Executive  and  Employer’s  Board  of  Directors  (the  “Board”)  mutually
may agree, provided that such other or additional offices are consistent with the Executive’s position and the terms of Section 6 below. In
such capacity or capacities, the Executive shall serve as chair of the board of directors, develop agendas for board meetings, participate in
the  Company’s  executive  meetings,  represent  the  Company  to  the  investor  community,  lead  capital  raise  efforts,  engage  in  strategic
business  opportunities  and  negotiations  for  the  Company,  and  perform  such  other  services  and  duties  in  connection  with  the  business,
affairs  and  operations  of  the  Employer  and  consistent  with  his  position(s)  and  the  terms  of  Section  6  below;  provided,  however,  it  is
understood and agreed that, in the event of a dispute between the Employer and Akrimax (as defined in Section 6 below and/or Prezamax
(as  defined  in  Section  6  below),  the  Executive  shall  not  be  required  to  provide  any  services  to  the  Employer  related  to  such  dispute.
Employer  shall  use  its  best  efforts  to  cause  the  Executive  to  be  elected  as  a  voting  member  of  its  Board  throughout  the  Term  and  shall
include him in the management slate for election as a director at every stockholders meeting during the Term at which his term as a director
would  otherwise  expire.  The  Executive  agrees  to  accept  election,  and  to  serve  during  the  Term,  as  a  member  of  the  Board  without  any
compensation therefore other than as specified in this Agreement.

4. Compensation and Benefits. The regular compensation and benefits payable to the Executive under this Agreement shall be as

follows:

(a) Salary.  For  all  services  rendered  by  the  Executive  under  this Agreement,  the  Employer  shall  pay  the  Executive  a
salary  (the  “Salary”)  at  the  annual  rate  of  two  hundred  and  fifty  thousand  dollars  ($250,000).  The  Salary  shall  be  payable  in  periodic
installments in accordance with the Employer’s usual practice for its senior executives.

 
 
 
 
 
 
 
 
 
(b) Annual  Milestone  Bonus.  Executive  will  receive  a  discretionary  bonus  on  each  anniversary  of  the  Effective  Date
during  the  Term  (the  “Annual  Milestone  Bonus”)  in  an  amount  up  to  fifty  percent  (50%)  of  his  then  current  Base  Salary  based  on  the
attainment by the Executive of certain financial, clinical development and business milestones (the “Milestones”) as established annually
by the Board (or a committee thereof), after consultation with the Executive. The Annual Milestone Bonus shall be payable as a lump-sum
payment by no later than March 15 of the year following the close of the year to which such bonus relates.

(c) Regular Benefits.  The  Executive  shall  also  be  entitled  to  participate  in  any  medical  insurance  plans,  life  insurance
plans,  disability  income  plans,  retirement  plans,  vacation  and  other  paid  time  off  plans  and  policies,  expense  reimbursement  plans  and
policies and other benefit plans and policies, which the Employer may from time to time establish and have in effect for all or most of its
senior  executives.  Such  participation  shall  be  subject  to  the  terms  of  the  applicable  plan  documents  and  policies,  and  applicable  law.
Nothing contained in this Agreement shall be construed to create any obligation on the part of the Employer to establish any such plan or to
maintain the effectiveness of any such plan which may be in effect from time to time. The Executive shall be entitled to four (4) weeks of
paid vacation each calendar year, which vacation shall be taken in accordance with the Employer’s vacation plans and policies.

(d) Equity Grants.

(i)  On  the  September  12,  2014,  the  Employer  granted  the  Executive  an  option  to  purchase  3,300,000  shares  of
common  stock  of  the  Employer,  at  an  exercise  price  of  $0.45  cents  per  share  (the  “Option”).  The  Company  executed  a  1  for  15
reverse stock split on June 9, 2017, the (“Split”). The impact of the split was such that the Option now consisted of 220,000 shares
of common stock at an exercise price of $6.75 per share The Option has fully vested as of September 12, 2017.

(ii) On the September 15, 2017, the Citius Board of Directors granted the Executive an option to purchase 40,000
shares of common stock of the Employer, at an exercise price of $3.45 cents per share (the “2017 Option”). The options will vest
1/3 on the one year anniversary of the Vesting Commencement Date, and then vest monthly at the end of each month for the next
two  years  in  equal  amounts  for  the  remaining  2/3  of  the  options,  provided  that  the  Optionee  provides  Continuous  Service  to  the
Company as of each such vesting date.

(iii)  If  application  of  the  vesting  percentages  causes  a  fractional  Share  or  Unit,  such  fractional  Share  shall  be
rounded down to the nearest whole Share or Unit for each vesting date except for the last vesting date, on which the Option shall
become exercisable for the full remainder of the Shares.

(iv)  Notwithstanding  anything  to  the  contrary,  upon  a  Change  of  Control  (as  defined  in  Section  8),  all  options
granted  to  the  Executive  by  the  Employer,  including,  but  not  limited  to  the  Option,  shall  immediately  accelerate  and  become
exercisable or non-forfeitable as of the consummation of such Change of Control.

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( v ) The  Option  was  granted  pursuant  to  and  subject  to  the  terms  and  conditions  established  in  the  Citius
Pharmaceuticals, Inc. 2014 Stock Incentive Plan, a copy of which is attached hereto as Exhibit A (“Stock Incentive Plan”) and the
award agreement (the “Option Award Agreement”) in the form attached hereto as Exhibit B.

(vi) Subject to the terms of this Section 4(d), the Executive shall also be entitled to any other rights and benefits
with respect to option awards, to the extent and  upon  the  terms  provided  in  the  employee  option  plan  or  any  agreement  or  other
instrument attendant thereto pursuant to which such options were granted.

(e) Taxation of Payments and Benefits . The Employer shall undertake to make deductions, withholdings and tax reports
with respect to payments and benefits under this Agreement to the extent that it reasonably and in good faith believes that it is required to
make  such  deductions,  withholdings  and  tax  reports.  Payments  under  this Agreement  shall  be  in  amounts  net  of  any  such  deductions  or
withholdings. Nothing in this Agreement shall be construed to require the Employer to make any payments to compensate the Executive for
any adverse tax effect associated with any payments or benefits or for any deduction or withholding from any payment or benefit.

provided under this Agreement, or as otherwise agreed between the Executive and the Employer.

(f) Exclusivity of Salary and Benefits. The Executive shall not be entitled to any payments or benefits other than those

5. Principal Place of Business. Executive shall perform services under this Agreement in the Employer’s office space located in
New  Jersey,  USA. At  all  times  during  the  Term  of  this Agreement,  Employer  shall  provide  Executive  with  appropriate  and  reasonable
administrative support for the performance of his services under this Agreement.

6. Extent of Service. During the Executive’s employment under this Agreement, the Executive shall, subject to the direction and
supervision  of  the  Board,  devote  the  Executive’s  best  efforts  and  business  judgment,  skill  and  knowledge  to  the  advancement  of  the
Employer’s interests and to the discharge of the Executive’s duties and responsibilities under this Agreement; provided, however, that the
Executive may engage in the Permitted Activities (as defined below) both during and outside of regular business hours, provided that such
Permitted Activities during regular business hours do not impair the Executive’s ability to fulfill the Executive’s duties and responsibilities
under this Agreement. “Permitted Activities” means (a) serving on the board of directors or similar governing body (and any committee
thereof)  of  IntelliCell  Biosciences  (“IntelliCell”),  Leonard  Meron  Biosciences  (“Meron”),  Akrimax  Pharmaceuticals  (“Akrimax”),
Prenzamax LLC (“Prenzamax”), Rouses Point Pharmaceuticals, LLC (“Rouses”), Novellus, Inc. (“Novellus”), their respective subsidiaries
and any of their respective successors and assigns (together, the “Excluded Businesses”), (b) serving as interim Chief Executive Officer of
Novellus, (c) continuing to have an equity interest in and/or investing in the Excluded Businesses, and (d) activities in connection with the
operations or affairs of the Excluded Businesses. During the Executive’s employment under this Agreement, the Executive shall not engage
in any other competing business activity, except for such other business activities as may be previously approved by the Board; provided,
however, for the avoidance of doubt, the Permitted Activities shall in no event be deemed a “competing business activity” In addition to the
express understanding that Executive may engage in the Permitted Activities, nothing in this Agreement shall be construed as preventing
the Executive from:

(a) investing the Executive’s assets in any company or other entity in a manner not prohibited by Section 9(d) and in such
form or manner as shall not require any activities on the Executive’s part in connection with the operations or affairs of the companies or
other  entities  in  which  such  investments  are  made  or  otherwise  impair  the  Executive’s  ability  to  fulfill  the  Executive’s  duties  and
responsibilities under this Agreement; or

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to fulfill the Executive’s duties and responsibilities under this Agreement.

(b) engaging in religious, charitable or other community or non-profit activities that do not impair the Executive’s ability

7. Termination. The Executive’s employment under this Agreement shall terminate under the following circumstances.

(a) Termination by the Employer for Cause. The Executive’s employment under this Agreement may be terminated for
Cause without further liability (other than to pay or provide the Accrued Benefits) on the part of the Employer effective immediately upon
a vote of the Board and written notice to the Executive. Only the following shall constitute “Cause” for such termination:

the Employer, as reasonably determined in good faith by the Board;

(i) any act of fraud, dishonesty or gross willful misconduct that is demonstrated to have caused material harm to

moral turpitude or fraud.

(ii) the indictment of the Executive for the Executive’s commission of a (x) felony or (y) misdemeanor involving

(iii)  failure  of  the  Executive  to  make  a  good  faith  effort  to  perform  the  Executive’s  material  duties  and
responsibilities  lawfully  assigned  or  delegated  by  the  Board  under  this  Agreement,  which  failure  continues  uncured  (in  the
reasonable judgment of the Board, acting in good faith) for more than thirty (30) days after written notice describing the particulars
of such alleged failure is given to the Executive by the Board; or

(iv)  a  material  and  willful  breach  by  the  Executive  of  any  of  the  Executive’s  material  obligations  under  this
Agreement, which breach continues uncured (in the reasonable judgment of the Board acting in good faith) for more than thirty (30)
days, after written notice describing the particulars of such alleged breach is given to the Executive by the Board.

For purposes of this definition of “Cause,” no act or failure to act, on the part of the Executive, shall be considered “willful” unless it is
done, or omitted to be done, by the Executive in bad faith or without reasonable belief that the Executive’s action or omission was in the
best interests of the Employer.

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(b) Termination by the Executive for Good Reason . Subject to the payment of Termination Benefits pursuant to Section
8(c)  or  Section  8(d),  as  applicable,  the  Executive’s  employment  under  this Agreement  may  be  terminated  by  the  Executive  for  Good
Reason, provided that the Executive first provides written notice (“Good Reason Notice”) to the Board not later than forty-five (45) days
following the initial occurrence of the act or failure to act that constitutes Good Reason setting forth the act or failure to act that constitutes
Good  Reason.  The  Employer  shall  have  a  period  of  thirty  (30)  days  in  which  it  may  correct  the  act  or  failure  to  act  that  constitutes  the
grounds for Good Reason as set forth in the Executive’s Good Reason Notice (the “Good Reason Cure Period”). If the Employer does not
correct the act or failure to act, the Executive must terminate his employment for Good Reason within thirty (30) days after the end of the
Good  Reason  Cure  Period,  in  order  for  the  termination  to  be  considered  a  Good  Reason  termination.  Good  Reason  shall  mean  the
occurrence of one or more of the following, without the Executive’s consent:

(i) a reduction of the Executive’s Salary, other than a reduction of the Executive’s Salary by a percentage that is
not greater than 10% in connection with a general reduction in base compensation that affects all of the Employer’s executives in
substantially the same proportions;

(ii) a material diminution in the Executive’s authority, responsibilities or duties;

(iii)  a  material  relocation  of  the  geographic  location  at  which  the  Executive  must  perform  services  for  the
Employer,  which,  for  purposes  of  this Agreement,  means  the  relocation  of  the  geographic  location  at  which  the  Executive  must
perform  services  for  the  Employer  to  a  location  more  than  fifty  (50)  miles  from  such  geographic  location  prior  to  the  relocation
(“Relocation”);

(iv) the Executive is not elected or re-elected, as applicable, to serve on the Board; or

(v) a material breach by the Employer of this Agreement, including, but not limited to Section 13 below.

(c) Termination by the Employer Without Cause. Subject to the payment of Termination Benefits pursuant to Section 8(c)
or Section 8(d), as applicable, the Executive’s employment under this Agreement may be terminated by the Employer without Cause upon
at least thirty (30) days advance written notice to the Executive.

the Executive voluntarily without Good Reason upon at least thirty (30) days advance written notice to the Employer.

(d) Voluntary Termination by the Executive without Good Reason . The Executive’s employment may be terminated by

(e) Death. The Executive’s employment with the Employer shall terminate upon his death.

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(f) Disability.  If  the  Executive  shall  incur  a  “Disability”  so  as  to  be  unable  to  perform  the  essential  functions  of  the
Executive’s then existing position or positions under this Agreement, with or without reasonable accommodation, the Board may relieve
him from any responsibilities during the period of such Disability. Notwithstanding any such removal or reassignment, the Executive shall
continue to receive the Executive’s full Salary (less any Disability pay or sick pay benefits to which the Executive may be entitled under the
Employer’s plans or policies) and benefits under Section 5 of this Agreement (except to the extent that the Executive may be ineligible for
one or more such benefits under applicable plan terms) for up to ninety (90) or more consecutive days or one hundred eighty (180) days in
the aggregate during any consecutive twelve (12) month period, and the Executive’s employment may be terminated by the Employer on
account of Disability at any time thereafter. For purposes of this Agreement, “Disability” shall mean the Executive is eligible to receive
long-term disability benefits under the Employer’s long-term disability plan, provided, however, that if the Employer does not maintain a
long-term  disability  plan,  “Disability”  shall  mean  a  medical  determination  by  physician(s)  selected  by  the  Employer  to  whom  the
Executive  or  the  Executive’s  guardian  has  no  reasonable  objections  that  due  to  the  Executive’s  illness  or  other  physical  or  mental
disability, the Executive was or will be unable to substantially perform the essential functions of the Executive’s employment under this
Agreement,  with  or  without  reasonable  accommodation,  for  a  period  of  ninety  (90)  or  more  consecutive  days  or  for  one  hundred  eighty
(180) days in the aggregate during any consecutive twelve (12) month period. Nothing in this Section 7(g) shall be construed to waive the
Executive’s rights, if any, under existing law including, without limitation, the Family and Medical Leave Act of 1993, 29 U.S.C. §2601  et
seq. and the Americans with Disabilities Act, 42 U.S.C. §12101 et seq.

8. Compensation Upon Termination.

(a) Termination Generally. If the Executive’s employment with the Employer is terminated for any reason, the Employer
shall pay or provide to the Executive (or to his authorized representative or estate) any earned but unpaid Salary (which earned, but unpaid
Salary shall be paid on or before the time required by law, but in no event more than sixty (60) days after the last day of the Executive’s
employment), unpaid expense reimbursements (which unpaid expense reimbursements shall be paid on or before the time required by law,
but in no event more than sixty (60) days after the last day of the Executive employment), accrued but unused vacation (which accrued but
unused  vacation  shall  be  paid  on  or  before  the  time  required  by  law,  but  in  no  event  more  than  sixty  (60)  days  after  the  last  day  of  the
Executive’s employment), any bonus Executive has earned under Section 4(b) of the Agreement (which bonus shall be paid according to
the time set forth in Section 4(b) above), and any vested benefits the Executive may have under any employee benefit plan of the Employer
(which benefits shall be paid and/or provided in accordance with the terms of the applicable plan) (the “Accrued Benefit”).

(b) Voluntary Termination without Good Reason. If the Executive elects voluntarily to terminate his employment without
Good  Reason  in  accordance  with  Section  7(b),  the  Employer  shall  have  no  further  obligation  to  the  Executive  other  than  to  pay  and/or
provide  his Accrued  Benefit  through  the  date  of  termination  (which Accrued  Benefit  will  be  paid  and/or  provided  in  accordance  with
Section 8(a) above).

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(c) Termination by the Employer Without Cause or by the Executive for Good Reason. In the event of a termination of
the Executive’s employment with the Employer by the Employer without Cause or by the Executive for Good Reason, and subject to the
Executive’s execution and non-revocation of a release of any and all legal claims in the form annexed hereto as Exhibit C (the “Release”),
in  addition  to  the  Accrued  Benefit,  the  Employer  shall  provide  to  the  Executive  the  following  termination  benefits  (“Termination
Benefits”):

preceding the date of termination;

(i)  continuation  of  the  Executive’s  Salary  at  the  highest  annual  rate  applicable  within  the  four  (4)  months

(ii) provided the Executive timely elects continued coverage under any of Employer’s group health, dental, vision
or prescription drug plan benefits in which he participates on the date of his termination of employment to the extent authorized by
and consistent with 29 U.S.C. § 1161 et seq. (commonly known as “COBRA”), monthly reimbursement for COBRA premiums paid
by the Executive for such continued coverage, less the amount that the Executive would be required to contribute for such coverage
if the Executive were an active employee of the Employer;

(iii) immediate vesting in any options that would have vested at the next immediate vesting event following the
date the Executive’s employment is terminated, provided, however, that the Executive must continue to comply with his obligations
under  this Agreement  to  be  eligible  for  such  vesting,  including,  without  limitation,  his  post-employment  obligations  set  forth  in
Section 9 below.

The  Termination  Benefits  set  forth  in  Sections  8(c)(i)  and  (ii)  above  shall  continue  effective  for  twelve  (12)  months  after  the  date  of
termination  (the  “Termination  Benefits  Period”).  The  Salary  continuation  payments  under  Section  8(c)(i)  will  be  paid  in  installments  in
accordance with the Employer’s regular payroll practices, commencing with the first regular payroll date on or following sixty (60) days
following the date of the Executive’s termination of employment, and the first payment will include any payments not yet paid during the
period between the date of termination of employment and the date of the first payment.

(d) Termination by the Employer Without Cause or by the Executive for Good Reason and Within Ninety (90) Days Prior
to a Change of Control or Within Two Years Following a Change of Control . Notwithstanding the foregoing, in the event of a termination
of  the  Executive’s  employment  with  the  Employer  by  the  Employer  without  Cause  or  by  the  Executive  for  Good  Reason  and  within
ninety  (90)  days  prior  to  a  Change  of  Control  or  within  two  (2)  years  following  a  Change  of  Control,  and  subject  to  the  Executive’s
execution  and  non-revocation  of  the  Release,  the  Executive  will  receive  (in  addition  to  the Accrued  Benefit)  all  of  the  payments  and
benefits  as  set  forth  in  Section  8(c),  except  that  the  Termination  Benefits  Period  shall  be  eighteen  (18)  months  instead  of  twelve  (12)
months, and any such options shall immediately vest and be exercisable in full and, in the event of a termination on or within two (2) years
following a Change of Control, the Salary continuation payments under Section 8(c)(i) shall be paid in a lump sum no later than sixty (60)
days following the termination of the Executive’s employment.

the Employer shall have no further obligation to the Executive other than payment of his Accrued Benefit.

(e) Termination by the Employer with Cause. If the Executive’s employment is terminated by the Employer with Cause,

-7-

 
 
 
 
 
 
 
 
 
(f) Additional Limitation.

(i) In the event that it shall be determined that any benefit or payment in the nature of compensation (within the
meaning of Section 280G(b)(2) of the Code) to or for the benefit of the Executive under this Agreement, or any other plan, arrangement, or
agreement with the Employer (the “Payments”) would constitute a “parachute payment” within the meaning of Section 280G of the Code
and  (but  for  this  sentence)  be  subject  to  the  tax  (the  “Excise  Tax”)  imposed  by  Section  4999  of  the  Code  (or  any  similar  tax  that  may
hereafter be imposed), the aggregate present value of the Payments under this Agreement, and such other plan, arrangement or agreement
with the Employer, shall be reduced (but not below zero) to the Reduced Amount. The “Reduced Amount” shall be either (A) the largest
portion of the Payments that would result in no portion of the Payments being subject to the Excise Tax or (B) the largest portion, up to
and  including  the  total,  of  the  Payments,  whichever  amount,  after  taking  into  account  all  applicable  federal,  state  and  local  employment
taxes,  income  taxes,  and  the  Excise  Tax,  results  in  the  Executive’s  receipt,  on  an  after-tax  basis,  of  the  greater  amount  of  the  Payments
notwithstanding  that  all  or  some  portion  of  the  Payments  may  be  subject  to  the  Excise  Tax.  If  a  reduction  in  payments  or  benefits
constituting “parachute payments” is necessary so that the Payments equal the Reduced Amount, the Employer shall reduce the Payments
by  first  reducing  or  eliminating  any  cash  payments  (with  the  Payments  to  be  made  furthest  in  the  future  being  reduced  first),  then  by
reducing or eliminating accelerated vesting of stock options or similar awards, and then by reducing or eliminating any other remaining
Payments,  provided  that  with  each  category  the  reduction  shall  be  done  on  a  basis  resulting  in  the  highest  amount  retained  by  the
Executive; and provided, further, that to the extent permitted by Section 409A of the Code and Sections 280G and 4999 of the Code, if a
different reduction procedure would be permitted without violating Section 409A of the Code or losing the benefit of the reduction under
Sections 280G and 4999 of the Code, the Executive may designate a different order of reduction.

(ii)  All  determinations  to  be  made  under  this  Section  8(f)  shall  be  made  by  an  independent  certified  public
accounting firm selected by the Employer and approved by the Executive (the “Accounting Firm”), which shall provide its determinations
and  any  supporting  calculations  both  to  the  Employer  and  the  Executive  within  ten  (10)  days  following  the  Change  of  Control.  For
purposes of this Section 8(f), the Accounting Firm shall take into account all applicable federal, state and local income and employment
taxes  and  the  Excise  Tax  (all  computed  at  the  Executive’s  actual  marginal  tax  rate).  Any  determinations  by  the  Accounting  Firm  in
accordance with this Section 8(f) shall be binding upon the Employer and the Executive. All of the fees and expenses of the Accounting
Firm in performing the determinations referred to in this Section 8(f) shall be borne solely by the Employer.

(iii) Notwithstanding anything herein to the contrary, for purposes of Section 409A of the Internal Revenue Code
of 1986, as amended (the “Code”), if the Executive is a “specified employee” of a publicly held corporation at his termination date, the
postponement  provisions  of  Section  409A  of  the  Code,  as  described  in  Section  18(a)  below,  shall  apply,  if  applicable.  Additionally,
notwithstanding  anything  herein  to  the  contrary,  in  no  event  shall  the  timing  of  the  Executive’s  execution  of  the  Release,  directly  or
indirectly, result in the Executive designating the calendar year of payment, and if a payment that is subject to execution of the Release
could  be  made  in  more  than  one  taxable  year,  payment  shall  be  made  in  the  later  taxable  year.  The  Employer’s  liability  for  Salary
continuation  pursuant  to  Section  8(c)(i)  shall  be  reduced  by  the  amount  of  any  severance  actually  paid  to  the  Executive  pursuant  to  any
severance pay plan of the Employer. Nothing in Section 8(c) or Section 8(d) shall be construed to affect the Executive’s right to receive
COBRA  continuation  entirely  at  the  Executive’s  own  cost  to  the  extent  that  the  Executive  may  continue  to  be  entitled  to  COBRA
continuation after the Executive’s right to reimbursements under Section 8(c)(ii) or Section 8(d) ceases.

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clause (A) below or (y) a change in the ownership of a substantial portion of the assets of the Employer under clause (B) below:

(iv) As used in this Agreement, “Change of Control” means (x) a change in ownership of the Employer under

(A) Change  in  the  Ownership  of  the  Employer. A  change  in  the  ownership  of  the  Employer
shall occur on the date that any one person, or more than one person acting as a group (as defined in clause (C)
below), acquires ownership of capital stock of the Employer that, together with capital stock held by such person
or group, constitutes more than 50 percent of the total fair market value or total voting power of the capital stock
of  the  Employer.  However,  if  any  one  person  or  more  than  one  person  acting  as  a  group,  is  considered  to  own
more than 50 percent of the total fair market value or total voting power of the capital stock of the Employer, the
acquisition of additional capital stock by the same person or persons shall not be considered to be a change in the
ownership of the Employer. An increase in the percentage of capital stock owned by any one person, or persons
acting  as  a  group,  as  a  result  of  a  transaction  in  which  the  Employer  acquires  capital  stock  in  the  Employer  in
exchange for property will be treated as an acquisition of stock for purposes of this paragraph.

(B) Change in the Ownership of a Substantial Portion of the Employer’s Assets. A change in the
ownership of a substantial portion of the Employer’s assets shall occur on the date that any one person, or more
than one person acting as a group (as defined in clause (C) below), acquires (or has acquired during the 12-month
period ending on the date of the most recent acquisition by such person or persons) assets from the Employer that
have a total gross fair market value equal to or more than 80 percent of the total gross fair market value of all of
the  assets  of  the  Employer  immediately  prior  to  such  acquisition  or  acquisitions.  For  this  purpose,  gross  fair
market  value  means  the  value  of  the  assets  of  the  Employer,  or  the  value  of  the  assets  being  disposed  of,
determined without regard to any liabilities associated with such assets. There is no Change of Control under this
clause (B) when there is a transfer to an entity that is controlled by the shareholders of the Employer immediately
after  the  transfer,  as  provided  below  in  this  clause  (B). A  transfer  of  assets  by  the  Employer  is  not  treated  as  a
change  in  the  ownership  of  such  assets  if  the  assets  are  transferred  to  (1)  a  shareholder  of  the  Employer
(immediately before the asset transfer) in exchange for or with respect to its capital stock, (2) an entity, 50 percent
or more of the total value or voting power of which is owned, directly or indirectly, by the Employer, (3) a person,
or more than one person acting as a group, that owns, directly or indirectly, 50 percent or more of the total value
or voting power of all the outstanding capital stock of the Employer, or (4) an entity, at least 50 percent of the
total value or voting power of which is owned, directly or indirectly, by a person described in clause (B)(3) of this
paragraph. For purposes of this clause (B), a person’s status is determined immediately  after  the  transfer  of  the
assets.

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(C) Persons Acting as a Group . For purposes of clauses (A) and (B) above, persons will not be
considered  to  be  acting  as  a  group  solely  because  they  purchase  or  own  capital  stock  or  purchase  assets  of  the
Employer at the same time. However, persons will be considered to be acting as a group if they are owners of a
corporation that enters into a merger, consolidation, purchase or acquisition of assets or capital stock, or similar
business transaction with the Employer. If a person, including an entity, owns stock in both corporations that enter
into  a  merger,  consolidation,  purchase  or  acquisition  of  assets  or  capital  stock,  or  similar  transaction,  such
shareholder is considered to be acting as a group with other shareholders in a corporation only with respect to the
ownership  in  that  corporation  before  the  transaction  giving  rise  to  the  change  and  not  with  respect  to  the
ownership interest in the other corporation. For purposes of this paragraph, the term “corporation” shall have the
meaning assigned such term under Treasury Regulation section 1.280G-1, Q&A-45.

(D) Each of clauses (A) through (C) above shall be construed and interpreted consistent with the
requirements  of  Section  409A  and  any  Treasury  Regulations  or  other  guidance  issued  thereunder.  For  the
avoidance  of  doubt,  the  Transaction  or  a  similar  financing  or  recapitalization,  including  a  financing  or
recapitalization  that  results  in  any  person  or  entity  acquiring  a  majority  interest  of  the  Employer’s  outstanding
equity, shall not be a “Change of Control” for purposes of this Agreement.

9. Confidential Information, Noncompetition and Cooperation.

(a) Confidential Information. As used in this Agreement, “Confidential Information” means information belonging to the
Employer which is of value to the Employer in the course of conducting its business and is maintained as confidential by the Employer and
the  disclosure  of  which  could  result  in  a  competitive  or  other  disadvantage  to  the  Employer.  Confidential  Information  includes,  without
limitation, financial information, reports, and forecasts; inventions, improvements and other intellectual property; trade secrets; know-how;
designs,  processes  or  formulae;  software;  market  or  sales  information  or  plans;  customer  lists;  and  business  plans,  prospects  and
opportunities  (such  as  possible  acquisitions  or  dispositions  of  businesses  or  facilities)  which  have  been  discussed  or  considered  by  the
management of the Employer. Confidential Information includes information developed by the Executive in the course of the Executive’s
employment  by  the  Employer,  as  well  as  other  information  to  which  the  Executive  may  have  access  in  connection  with  the  Executive’s
employment.  Confidential  Information  also  includes  the  confidential  information  of  others  with  which  the  Employer  has  a  business
relationship. Notwithstanding the foregoing, Confidential Information does not include: (i) information in the public domain unless due to
breach of the Executive’s duties under Section 9(b); (ii) information known to the Executive prior to such information being disclosed to
the Executive in connection with his employment hereunder; (iii) is disclosed to the Executive at any time other than in the course of the
Executive’s performance of his duties as an employee of Employer, by any third party not bound at the time of the disclosure directly or
indirectly, by any confidentiality agreement with Employer.

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(b) Confidentiality.  The  Executive  understands  and  agrees  that  the  Executive’s  employment  creates  a  relationship  of
confidence and trust between the Executive and the Employer with respect to all Confidential Information. At all times, both during the
Executive’s employment with the Employer and after its termination, the Executive will keep in confidence and trust all such Confidential
Information, and will not use or disclose any such Confidential Information without the written consent of the Employer, except (i) as may
be necessary in the ordinary course of performing the Executive’s duties to the Employer, (ii) to enforce any rights or defend any claims
hereunder or under any other agreement to which the Executive is a party, provided that such disclosure is relevant to the enforcement of
such rights or defense of such claims and is only disclosed to the extent necessary in the formal proceedings related thereto, or (iii) when
required to do so by a court of law, by any governmental agency having supervisory authority over the business of the Employer or by any
administrative  or  legislative  body  (including  a  committee  thereof)  with  jurisdiction  to  order  the  Executive  to  divulge,  disclose  or  make
accessible such information, provided that the Executive shall give prompt written notice to the Employer of such requirement, disclose no
more information than is so required, and reasonably cooperate with any attempt by the Employer to obtain a protective order or similar
treatment.

(c) Documents, Records, etc. All documents, records, data, apparatus, equipment and other physical property, whether or
not  pertaining  to  Confidential  Information,  which  are  furnished  to  the  Executive  by  the  Employer  or  are  produced  by  the  Executive  in
connection  with  the  Executive’s  employment  will  be  and  remain  the  sole  property  of  the  Employer.  The  Executive  will  return  to  the
Employer all such materials and property as and when requested by the Employer. In any event, the Executive will return all such materials
and  property  immediately  upon  termination  of  the  Executive’s  employment  for  any  reason.  The  Executive  will  not  retain  with  the
Executive any such material or property or any copies thereof after such termination.

(d) Noncompetition and Nonsolicitation.

(i)  During  the  term  of  the  Executive’s  employment  with  the  Employer  hereunder  and  for  nine  (9)  months
thereafter,  the  Executive  will  not,  directly  or  indirectly,  whether  as  owner,  partner,  shareholder,  consultant,  agent,  employee,  co-
venturer or otherwise, engage, participate, assist or invest in any Competing Business (as defined below in this Section 9(d) below).

(ii)  During  the  term  of  the  Executive’s  employment  with  the  Employer  and  for  two  (2)  years  thereafter,  the
Executive  will  not,  directly  or  indirectly,  whether  as  owner,  partner,  shareholder,  consultant,  agent,  employee,  co-venturer  or
otherwise;  (A)  attempt  to  employ,  recruit  or  otherwise  solicit,  induce  or  influence  any  person  to  leave  employment  with  the
Employer (other than terminations of employment of employees undertaken in the course of the Executive’s employment with the
Employer and/or in the Executive’s capacity as a member of the Board); and (B) solicit or encourage any customer or supplier to
terminate  or  otherwise  modify  adversely  its  business  relationship  with  the  Employer;  provided,  that  neither  (1)  the  general
advertisement for employees or service providers (i.e., not targeted toward any of the Employer’s employees) nor (2) the Executive
being named as an reference for an employee of the Employer and responding to ordinary course inquiries made of the Executive by
prospective  employers  or  service  recipients  of  such  employee  in  connection  with  such  reference  so  long  as  the  reference  is  for
employment  with  an  employer  that  does  not  engaging  a  Competing  Business  with  Employer,  shall  be  deemed  a  violation  of  this
Section 9(d)(ii). Further, for the avoidance of doubt, nothing in this Section 9(d)(ii) shall be deemed to prohibit senior level general
solicitations in connection with any activities that are not prohibited by Section 9(d)(i) above shall not be deemed a violation of this
Section 9(d)(ii).

-11-

 
 
 
 
 
 
 
The  Executive  understands  that  the  restrictions  set  forth  in  this  Section  9(d)  are  intended  to  protect  the
Employer’s interest in its Confidential Information and established employee, customer and supplier relationships and goodwill, and
agrees that such restrictions are reasonable and appropriate for this purpose. For purposes of this Agreement, the term “Competing
Business”  shall  mean  a  biopharmaceuticals  business  conducted  anywhere  in  the  United  States  which  is  focused  on  therapies  for
obesity, or topical therapies for hemorrhoids and/or other anal rectal diseases or disorders, or on other therapeutic categories to be
identified  and  added  to Addendum A  to  this Agreement  from  time  to  time  during  the  employment  of  the  Executive;  provided,
however, in no event shall any of the Excluded Businesses be deemed a Competing Business, and provided further, however, that
any other therapeutic categories identified and added to Addendum A of this Agreement shall relate to therapeutic categories with
respect  to  which  the  Employer  is  actively  conducting  business  or  which  are  actively  under  development  by  the  Employer.
Notwithstanding  the  foregoing,  the  Executive  may  own  up  to  one  percent  (1%)  of  the  outstanding  stock  of  a  publicly  held
corporation which constitutes or is affiliated with a Competing Business.

(e) Third-Party Agreements and Rights. The Executive hereby confirms that the Executive is not bound by the terms of
any non-competition and/or non-solicitation agreement with any previous employer, other current employer or other party which prohibits
or materially limits the performance by the Executive of his duties to Employer hereunder. The Executive represents to the Employer that
the  Executive’s  execution  of  this Agreement,  the  Executive’s  employment  with  the  Employer  and  the  performance  of  the  Executive’s
proposed  duties  for  the  Employer  will  not  violate  any  obligations  the  Executive  may  have  to  any  such  previous  employer,  other  current
employer  or  other  party.  In  the  Executive’s  work  for  the  Employer,  the  Executive  will  not  disclose  or  make  use  of  any  information  in
violation of any agreements with or rights of any such previous employer, current employer or other party, and the Executive will not bring
to the premises of the Employer any copies or other tangible embodiments of non-public information belonging to or obtained from any
such previous employment, concurrent employment or other party.

-12-

 
 
 
 
(f) Litigation and Regulatory Cooperation. During and after the Executive’s employment, the Executive shall reasonably
cooperate with the Employer in the defense or prosecution of any claims or actions now in existence or which may be brought in the future
against  or  on  behalf  of  the  Employer  which  relate  to  events  or  occurrences  that  transpired  while  the  Executive  was  employed  by  the
Employer.  The  Executive’s  cooperation  in  connection  with  such  claims  or  actions  shall  include,  but  not  be  limited  to,  being  reasonably
available to meet with counsel to prepare for discovery or trial and to act as a witness on behalf of the Employer at mutually convenient
times. During and after the Executive’s employment, the Executive also shall reasonably cooperate with the Employer in connection with
any  investigation  or  review  of  any  federal,  state  or  local  regulatory  authority  as  any  such  investigation  or  review  relates  to  events  or
occurrences  that  transpired  while  the  Executive  was  employed  by  the  Employer.  The  Employer  shall  reimburse  the  Executive  for  any
reasonable  out-of-pocket  expenses  incurred  in  connection  with  the  Executive’s  performance  of  obligations  pursuant  to  this  Section  9(f),
including  Executive’s  attorneys’  fees  to  the  extent  the  Executive  reasonably  determines  that  the  Executive  should  be  represented  by  his
own counsel.

(g) Injunction.  The  Executive  agrees  that  it  would  be  difficult  to  measure  any  damages  caused  to  the  Employer  which
might result from any breach by the Executive of the promises set forth in this Section 9, and that in any event money damages would be an
inadequate remedy for any such breach. Accordingly, subject to Section 10 of this Agreement, the Executive agrees that if the Executive
breaches, or proposes to breach, any portion of this Agreement, the Employer shall be entitled, in addition to all other remedies that it may
have, to seek an injunction or other appropriate equitable relief to restrain any such breach without showing or proving any actual damage
to the Employer.

10. Arbitration  of  Disputes.  Any  controversy  or  claim  arising  out  of  or  relating  to  this  Agreement  or  the  breach  thereof  or
otherwise arising out of the Executive’s employment or the termination of that employment (including, without limitation, any claims of
unlawful  employment  discrimination  whether  based  on  age  or  otherwise)  shall,  to  the  fullest  extent  permitted  by  law,  be  settled  by
arbitration in any forum and form agreed upon by the parties or, in the absence of such an agreement, under the auspices of the American
Arbitration Association  (“AAA”)  in  Boston,  Massachusetts  in  accordance  with  the  Employment  Dispute  Resolution  Rules  of  the AAA,
including, but not limited to, the rules and procedures applicable to the selection of arbitrators. In the event that any person or entity other
than  the  Executive  or  the  Employer  may  be  a  party  with  regard  to  any  such  controversy  or  claim,  such  controversy  or  claim  shall  be
submitted  to  arbitration  subject  to  such  other  person  or  entity’s  agreement.  Judgment  upon  the  award  rendered  by  the  arbitrator  may  be
entered  in  any  court  having  jurisdiction  thereof.  This  Section  10  shall  be  specifically  enforceable.  Notwithstanding  the  foregoing,  this
Section 10 shall not preclude either party from pursuing a court action for the sole purpose of obtaining a temporary restraining order or a
preliminary  injunction  in  circumstances  in  which  such  relief  is  appropriate,  provided  that  any  other  relief  shall  be  pursued  through  an
arbitration  proceeding  pursuant  to  this  Section  10.  The  Employer  shall  bear  the  cost  of  all  arbitration  fees,  but  each  party  shall  be
responsible for its own attorneys’ fees.

11. Consent  to  Jurisdiction.  To  the  extent  that  any  court  action  is  permitted  consistent  with  or  to  enforce  Section  10  of  this
Agreement, the parties hereby consent to the jurisdiction of the Superior Court of the State of New Jersey and the United States District
Court  for  the  District  of  New  Jersey.  Accordingly,  with  respect  to  any  such  court  action,  the  Executive  (a)  submits  to  the  personal
jurisdiction of such courts; (b) consents to service of process; and (c) waives any other requirement (whether imposed by statute, rule of
court, or otherwise) with respect to personal jurisdiction or service of process.

-13-

 
 
 
 
 
 
12. Integration.  This  Agreement,  the  Stock  Incentive  Plan  and  the  Option  Award  Agreement  constitute  the  entire  agreement
between  the  parties  with  respect  to  the  subject  matter  hereof  and  supersede  all  prior  agreements  between  the  parties  with  respect  to  any
related subject matter.

1 3 . Indemnification;  Liability  Insurance.  The  Employer  shall  indemnify  and  hold  Executive  harmless  to  the  fullest  extent
permitted by the laws of the Employer’s state of organization or incorporation in effect at the time against and in respect of any and all
actions, suits, proceedings, claims, demands, judgments, costs, expenses (including advancement of reasonable attorney’s fees), losses, and
damages  resulting  from  the  Executive’s  performance  of  the  Executive’s  duties  and  obligations  with  the  Employer.  Executive  will  be
entitled  to  be  covered,  both  during  and,  while  potential  liability  exists,  by  the  insurance  policies  the  Employer  may  elect  to  maintain
generally for the benefit of officers and directors of the Employer against all costs, charges and expenses incurred in connection with any
action, suit or proceeding to which the Executive may be made a party by reason of being an officer or director of the Employer in the same
amount and to the same extent as the Employer covers its other officers and directors. Without limitation of the foregoing, the Employer
agrees to continue and maintain a directors’ and officers’ liability insurance policy covering the Executive in an amount, and on terms and
conditions (including without limitation, with respect to scope, exclusions, sub-amounts and deductibles), no less favorable to him than (x)
the  coverage  the  Employer  provides  other  senior  executives  and  directors  from  time  to  time  or,  if  greater,  (y)  the  coverage  provided  to
senior executives and directors on the Effective Date. These obligations shall survive the termination of Executive’s employment with the
Employer.

14. Assignment;  Successors  and Assigns,  etc .  Except  as  otherwise  set  forth  in  this  Section  14,  neither  the  Employer  nor  the
Executive may make any assignment of this Agreement or any interest herein, by operation of law or otherwise, without the prior written
consent of the other party. Notwithstanding the foregoing, the Employer may assign its rights under this Agreement without the consent of
the  Executive  to  a  successor  in  the  event  that  the  Employer  shall  effect  a  reorganization,  consolidate  with  or  merge  into  any  other
corporation, partnership, organization or other entity, or transfer all of substantially all of its properties or assets to any other corporation,
partnership, organization or other entity and such successor shall assume and agree to perform this Agreement in the same manner and to
the  same  extent  that  the  Employer  would  be  required  to  perform  it  if  no  such  succession  had  taken  place. As  used  in  this Agreement,
“Employer”  shall  mean  the  Employer  and  any  such  successor  which  assumes  and  agrees  to  perform  the  duties  and  obligations  of  the
Employer under this Agreement by operation of law or otherwise. This Agreement shall inure to the benefit of and be binding upon the
Employer and the Executive, their respective successors, executors, administrators, heirs and permitted assigns.

15. Enforceability. If any portion or provision of this Agreement (including, without limitation, any portion or provision of any
section of this Agreement) shall to any extent be declared illegal or unenforceable by a court of competent jurisdiction, then the remainder
of this Agreement, or the application of such portion or provision in circumstances other than those as to which it is so declared illegal or
unenforceable, shall not be affected thereby, and each portion and provision of this Agreement shall be valid and enforceable to the fullest
extent permitted by law.

-14-

 
 
 
 
 
 
16. Waiver.  No  waiver  of  any  provision  hereof  shall  be  effective  unless  made  in  writing  and  signed  by  the  waiving  party.  The
failure of any party to require the performance of any term or obligation of this Agreement, or the waiver by any party of any breach of this
Agreement, shall not prevent any subsequent enforcement of such term or obligation or be deemed a waiver of any subsequent breach.

17. Notices. Any notices, requests, demands and other communications provided for by this Agreement  shall  be  sufficient  if  in
writing  and  delivered  in  person  or  sent  by  a  nationally  recognized  overnight  courier  service  or  by  registered  or  certified  mail,  postage
prepaid, return receipt requested, to the Executive at the last address the Executive has filed in writing with the Employer or, in the case of
the Employer, at its main offices, attention of the Board, and shall be effective on the date of delivery in person or by courier or three (3)
days after the date mailed.

18. Section 409A.

(a) This Agreement is intended to comply with Section 409A of the Code and its corresponding regulations, or an exemption, and
payments may only be made under this Agreement upon an event and in a manner permitted by Section 409A of the Code, to the extent
applicable. To the extent that any provision in this Agreement is ambiguous as to its compliance with Section 409A of the Code, or to the
extent any provision in this Agreement must be modified to comply with Section 409A of the Code, such provision shall be read in such a
manner so that no payment due to the Executive shall be subject to an “additional tax” within the meaning of Section 409A(a)(1)(B) of the
Code. Severance benefits under the Agreement are intended to be exempt from Section 409A of the Code under the “short-term deferral”
exception,  to  the  maximum  extent  applicable,  and  then  under  the  “separation  pay”  exception,  to  the  maximum  extent  applicable.
Notwithstanding  anything  in  this Agreement  to  the  contrary,  if  required  by  Section  409A  of  the  Code,  if  the  Executive  is  considered  a
“specified employee” for purposes of Section 409A of the  Code  and  if  payment  of  any  amounts  under  this Agreement  is  required  to  be
delayed for a period of six (6) months after separation from service pursuant to Section 409A of the Code, payment of such amounts shall
be delayed as required by Section 409A of the Code, and the accumulated amounts shall be paid in a lump sum payment within ten (10)
days after the end of the six (6) month period. If the Executive dies during the postponement period prior to the payment of benefits, the
amounts withheld on account of Section 409A of the Code shall be paid to the personal representative of the Executive’s estate within sixty
(60) days after the date of the Executive’s death.

(b) To the extent required to comply with Section 409A of the Code, any Termination Benefits or other payments to be made upon
a termination of employment under this Agreement may only be made upon a “separation from service” as defined under Section 409A of
the  Code.  For  purposes  of  Section  409A  of  the  Code,  each  payment  hereunder  shall  be  treated  as  a  separate  payment  and  the  right  to  a
series  of  installment  payments  under  this Agreement  shall  be  treated  as  a  right  to  a  series  of  separate  payments.  In  no  event  may  the
Executive,  directly  or  indirectly,  designate  the  calendar  year  of  a  payment. All  reimbursements  and  in-kind  benefits  provided  under  the
Agreement shall be made or provided in accordance with the requirements of Section 409A of the Code.

-15-

 
 
 
 
 
 
 
19. Amendment. This Agreement may be amended or modified only by a written instrument signed by the Executive and by a duly

authorized representative of the Employer.

20. Governing Law. This is a New Jersey contract and shall be construed under and be governed in all respects by the laws of the
state of New Jersey, without giving effect to the conflict of laws principles of such state. With respect to any disputes concerning federal
law,  such  disputes  shall  be  determined  in  accordance  with  the  law  as  it  would  be  interpreted  and  applied  by  the  United  States  Court  of
Appeals for the Third Circuit.

21. Counterparts. This Agreement may be executed in any number of counterparts, each of which when so executed and delivered

shall be taken to be an original; but such counterparts shall together constitute one and the same document.

IN  WITNESS  WHEREOF,  this Agreement  has  been  executed  as  a  sealed  instrument  by  the  Employer,  by  its  duly  authorized

member, and by the Executive, as of the Effective Date.

LEONARD MAZUR

/s/ Leonard Mazur

CITIUS PHARMACEUTICALS, INC.

/s/ Myron Holubiak
By: Myron Holubiak

-16-

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
CONSENT OF INDEPENDENT REGISTERED PUBLIC ACCOUNTING FIRM

We consent to the incorporation by reference in the Registration Statements on Forms S-1 (333-224386 and 333-226395) and on Form S-3
(File  No.  333-221492)  of  Citius  Pharmaceuticals,  Inc.  of  our  report  dated  December  11,  2018,  relating  to  the  consolidated  financial
statements of Citius Pharmaceuticals, Inc., appearing in the Annual Report on Form 10-K for the year ended September 30, 2018.

Exhibit 23.1

/s/ Wolf & Company, P.C.

Wolf & Company, P.C.
Boston, Massachusetts
December 11, 2018 

 
 
EXHIBIT 31.1

CERTIFICATION OF CHIEF EXECUTIVE OFFICER
PURSUANT TO SECTION 302 OF THE
SARBANES-OXLEY ACT OF 2002

I, Myron Holubiak, certify that:

1. I have reviewed this report on Form 10-K of Citius Pharmaceuticals, Inc.;

2.  Based  on  my  knowledge,  this  report  does  not  contain  any  untrue  statement  of  a  material  fact  or  omit  to  state  a  material  fact
necessary to make the statements made, in light of the circumstances under which such statements were made, not misleading with respect
to the period covered by this report;

3. Based on my knowledge, the financial statements, and other financial information included in this report, fairly present in all
material respects the financial condition, results of operations and cash flows of the registrant as of, and for, the periods presented in this
report;

4.  The  registrant’s  other  certifying  officer(s)  and  I  are  responsible  for  establishing  and  maintaining  disclosure  controls  and
procedures  (as  defined  in  Exchange  Act  Rules  13a-15(e)  and  15d-15(e))  and  internal  control  over  financial  reporting  (as  defined  in
Exchange Act Rules 13a-15(f) and 15d-15(f)) for the registrant and have:

a) designed such disclosure controls and procedures, or caused such disclosure controls and procedures to be designed under our
supervision, to ensure that material information relating to the registrant, including its consolidated subsidiaries, is made known
to us by others within those entities, particularly during the period in which this report is being prepared;

b) designed such internal control over financial reporting, or caused such internal control over financial reporting to be designed
under our  supervision,  to  provide  reasonable  assurance  regarding  the  reliability  of  financial  reporting  and  the  preparation  of
financial statements for external purposes in accordance with generally accepted accounting principles;

c)

evaluated the effectiveness of the registrant’s disclosure controls and procedures and presented in this report our conclusions
about the effectiveness of the disclosure controls and procedures, as of the end of the period covered by this report based on
such evaluation; and

d) disclosed in  this  report  any  change  in  the  registrant’s  internal  control  over  financial  reporting  that  occurred  during  the
registrant’s most recent fiscal quarter (the registrant's fourth fiscal quarter in the case of an annual report) that has materially
affected, or is reasonably likely to materially affect, the registrant’s internal control over financial reporting; and

5.  The  registrant’s  other  certifying  officer(s)  and  I  have  disclosed,  based  on  our  most  recent  evaluation  of  internal  control  over
financial  reporting,  to  the  registrant’s  auditors  and  the  audit  committee  of  the  registrant’s  board  of  directors  (or  persons  performing  the
equivalent functions):

a)

all significant deficiencies and material weaknesses in the design or operation of internal control over financial reporting which
are reasonably likely to adversely affect the registrant’s ability to record, process, summarize and report financial  information;
and

b)

any fraud, whether or not material, that involves management or other employees who have a significant role in the registrant’s
internal control over financial reporting.

December 11, 2018

By:

/s/ Myron Holubiak
Myron Holubiak
President and Chief Executive Officer
(Principal Executive Officer)

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
EXHIBIT 31.2

CERTIFICATION OF CHIEF FINANCIAL OFFICER
PURSUANT TO SECTION 302 OF THE
SARBANES-OXLEY ACT OF 2002

I, Jaime Bartushak, certify that:

1. I have reviewed this report on Form 10-K of Citius Pharmaceuticals, Inc.;

2.  Based  on  my  knowledge,  this  report  does  not  contain  any  untrue  statement  of  a  material  fact  or  omit  to  state  a  material  fact
necessary to make the statements made, in light of the circumstances under which such statements were made, not misleading with respect
to the period covered by this report;

3. Based on my knowledge, the financial statements, and other financial information included in this report, fairly present in all
material respects the financial condition, results of operations and cash flows of the registrant as of, and for, the periods presented in this
report;

4.  The  registrant’s  other  certifying  officer(s)  and  I  are  responsible  for  establishing  and  maintaining  disclosure  controls  and
procedures  (as  defined  in  Exchange  Act  Rules  13a-15(e)  and  15d-15(e))  and  internal  control  over  financial  reporting  (as  defined  in
Exchange Act Rules 13a-15(f) and 15d-15(f)) for the registrant and have:

a) designed such disclosure controls and procedures, or caused such disclosure controls and procedures to be designed under our
supervision, to ensure that material information relating to the registrant, including its consolidated subsidiaries, is made known
to us by others within those entities, particularly during the period in which this report is being prepared;

b) designed such internal control over financial reporting, or caused such internal control over financial reporting to be designed
under our  supervision,  to  provide  reasonable  assurance  regarding  the  reliability  of  financial  reporting  and  the  preparation  of
financial statements for external purposes in accordance with generally accepted accounting principles;

c)

evaluated the effectiveness of the registrant’s disclosure controls and procedures and presented in this report our conclusions
about the effectiveness of the disclosure controls and procedures, as of the end of the period covered by this report based on
such evaluation; and

d) disclosed in  this  report  any  change  in  the  registrant’s  internal  control  over  financial  reporting  that  occurred  during  the
registrant’s most recent fiscal quarter (the registrant's fourth fiscal quarter in the case of an annual report) that has materially
affected, or is reasonably likely to materially affect, the registrant’s internal control over financial reporting; and

5.  The  registrant’s  other  certifying  officer(s)  and  I  have  disclosed,  based  on  our  most  recent  evaluation  of  internal  control  over
financial  reporting,  to  the  registrant’s  auditors  and  the  audit  committee  of  the  registrant’s  board  of  directors  (or  persons  performing  the
equivalent functions):

a)

all significant deficiencies and material weaknesses in the design or operation of internal control over financial reporting which
are reasonably likely to adversely affect the registrant’s ability to record, process, summarize and report financial  information;
and

b)

any fraud, whether or not material, that involves management or other employees who have a significant role in the registrant’s
internal control over financial reporting.

December 11, 2018

By:

/s/ Jaime Bartushak
Jaime Bartushak
Chief Financial Officer
(Principal Financial Officer and 
Principal Accounting Officer)

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
  
 
CERTIFICATION OF CHIEF EXECUTIVE OFFICER
PURSUANT TO 18 U.S.C. SECTION 1350
AS ADOPTED PURSUANT TO
SECTION 906 OF THE SARBANES-OXLEY ACT OF 2002

Exhibit 32.1

In  connection  with  the  Annual  Report  of  Citius  Pharmaceuticals,  Inc.  (the  “Company”)  on  Form  10-K  for  the  year  ended
September 30, 2018 as filed with the Securities and Exchange Commission on the date hereof (the “Report”), I, Myron Holubiak, President
and  Chief  Executive  Officer  of  the  Company,  certify,  pursuant  to  18  U.S.C.  section  1350,  as  adopted  pursuant  to  Section  906  of  the
Sarbanes-Oxley Act of 2002, that:

(1) The Report fully complies with the requirements of section 13(a) or 15(d) of the Securities Exchange Act of 1934; and

(2) The information contained in the Report fairly presents, in all material respects, the financial condition and results of operations

of the Company.

Date: December 11, 2018

By:

/s/ Myron Holubiak
Myron Holubiak
President and Chief Executive Officer
(Principal Executive Officer, Principal Financial
Officer and Principal Accounting Officer)

 
 
 
 
 
 
 
 
 
 
 
 
 
CERTIFICATION OF CHIEF FINANCIAL OFFICER
PURSUANT TO 18 U.S.C. SECTION 1350
AS ADOPTED PURSUANT TO
SECTION 906 OF THE SARBANES-OXLEY ACT OF 2002

Exhibit 32.2

In  connection  with  the  Annual  Report  of  Citius  Pharmaceuticals,  Inc.  (the  “Company”)  on  Form  10-K  for  the  year  ended
September 30, 2018 as filed with the Securities and Exchange Commission on the date hereof (the “Report”), I, Jaime Bartushak, Chief
Financial Officer of the Company, certify, pursuant to 18 U.S.C. section 1350, as adopted pursuant to Section 906 of the Sarbanes-Oxley
Act of 2002, that:

(1) The Report fully complies with the requirements of section 13(a) or 15(d) of the Securities Exchange Act of 1934; and

(2) The information contained in the Report fairly presents, in all material respects, the financial condition and results of operations

of the Company.

Date: December 11, 2018

By:

/s/ Jaime Bartushak
Jaime Bartushak
Chief Financial Officer
(Principal Financial Officer and 
Principal Accounting Officer)