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CytRX Corporation

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FY2009 Annual Report · CytRX Corporation
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UNITED STATES SECURITIES AND EXCHANGE COMMISSION 
Washington, D.C. 20549 

Form 10-K 

(Mark One) 
(cid:53) 

ANNUAL REPORT PURSUANT TO SECTION 13 OR 15(d) OF THE SECURITIES EXCHANGE ACT OF 1934 

For the fiscal year ended December 31, 2009 

or 

(cid:133) 

TRANSITION REPORT PURSUANT TO SECTION 13 OR 15(d) OF SECURITIES EXCHANGE ACT OF 1934 

For the transition period from __________________ to __________________ 

Commission file number 0-15327 

CytRx Corporation 

(Exact name of Registrant as specified in its charter) 

Delaware 
(State or other jurisdiction of incorporation or organization) 

58-1642740 
(I.R.S. Employer Identification No.) 

11726 San Vicente Blvd, Suite 650, 
Los Angeles, California 
(Address of principal executive offices) 

90049 
(Zip Code) 

Registrant’s telephone number, including area code: (310) 826-5648 

____________________________ 

Securities registered pursuant to Section 12(b) of the Act: 

Title of each class 
Common Stock, $0.001 par value per share 
Series A Junior Participating Preferred Stock Purchase Rights

Name of exchange on which registered
The NASDAQ Capital Market

Securities Registered Pursuant to Section 12(g) of the Act: 

None 

Indicate by check mark if the Registrant is a well-known seasoned issuer (as defined in Securities Act Rule 405). Yes (cid:133) No (cid:53) 

Indicate by check mark if the Registrant is not required to file reports pursuant to Section 13 or Section 15(d) of the Securities Exchange Act of 1934. 
Yes (cid:133) No (cid:53) 

Indicate by check mark whether the Registrant (1) has filed all reports required to be filed by Section 13 or 15(d) of the Securities Exchange Act 

of 1934 during the preceding 12 months and (2) has been subject to such filing requirements for the past 90 days. Yes (cid:53) No (cid:133) 

Indicate by check mark whether the registrant has submitted electronically and posted on its corporate website, if any, every Interactive Data 
File required to be submitted and posted pursuant to Rule 405 of Regulation S-T (§ 232.405 of this chapter) during the preceding 12 months (or for 
such shorter period that the registrant was required to submit and post such files). Yes (cid:133) No (cid:133) 

Indicate  by  check  mark  if  disclosure  of  delinquent  filers  pursuant  to  Item  405  of  Regulation  S-K  is  not  contained  herein,  and  will  not  be 
contained, to the best of the Registrant’s knowledge, in definitive proxy or information statements incorporated by reference in Part III of this Form 
10-K or any amendment to this Form 10-K. (cid:53) 

Indicate by check mark whether the registrant is a large accelerated filer, an accelerated filer, a non-accelerated filer, or a smaller reporting company. 

See the definitions of “large accelerated filer,” “accelerated filer” and “smaller reporting company” in Rule 12b-2 of the Exchange Act. (Check one): 

Large accelerated filer (cid:133) 

Accelerated filer (cid:53) 

Non-accelerated filer (cid:133) 

Smaller reporting company (cid:133) 

(Do not check if a smaller reporting company) 

Indicate by check mark whether the Registrant is a shell company (as defined in Rule 12b-2 of the Act). Yes (cid:133) No (cid:53) 

Based on the closing price as reported on The Nasdaq Capital Market, the aggregate market value of the Registrant's common stock held by non-
affiliates on June 30, 2009 (the last business day of the Registrant's most recently completed second fiscal quarter) was approximately $102.0 million. 
Shares of common stock held by directors and executive officers and their respective affiliates have been excluded from this calculation, because 
such stockholders may be deemed to be “affiliates” of the Registrant. This is not necessarily determinative of affiliate status for other purposes. The 
number of outstanding shares of the Registrant's common stock as of March 12, 2010 was 108,908,105, exclusive of treasury shares. 

 
 
 
 
 
 
 
 
 
  
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
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CYTRX CORPORATION 
2009 ANNUAL REPORT ON FORM 10-K 

TABLE OF CONTENTS 

“SAFE HARBOR” STATEMENT . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .
PART I 

Item 1. BUSINESS . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .
Item 1A. RISK FACTORS . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .
Item 2. PROPERTIES . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .
Item 3. LEGAL PROCEEDINGS . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .

PART II 

Item 5. MARKET FOR REGISTRANT’S COMMON EQUITY, RELATED STOCKHOLDER MATTERS AND 

ISSUER PURCHASES OF EQUITY SECURITIES . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .
Item 6. SELECTED FINANCIAL DATA . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .
Item 7. MANAGEMENT’S DISCUSSION AND ANALYSIS OF FINANCIAL CONDITION AND RESULTS OF 

OPERATIONS . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .
Item 7A. QUANTITATIVE AND QUALITATIVE DISCLOSURES ABOUT MARKET RISK . . . . . . . . . . . . . . . . . . . . . .
Item 8. FINANCIAL STATEMENTS AND SUPPLEMENTARY DATA. . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .
Item 9. CHANGES IN AND DISAGREEMENTS WITH ACCOUNTAINS ON ACCOUNTING AND FINANCIAL 

DISCLOSURE . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .
Item 9A. CONTROLS AND PROCEDURES . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .
Item 9B. OTHER INFORMATION . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .

PART III 

Item 10. DIRECTORS, EXECUTIVE OFFICERS AND CORPORATE GOVERNANCE . . . . . . . . . . . . . . . . . . . . . . . . . . . .
Item 11. EXECUTIVE COMPENSATION . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .
Item 12. SECURITY OWNERSHIP OF CERTAIN BENEFICIAL OWNERS AND MANAGEMENT AND 

RELATED STOCKHOLDER MATTERS . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .
Item 13. CERTAIN RELATIONSHIPS AND RELATED TRANSACTIONS, AND DIRECTOR INDEPENDENCE. . .
Item 14. PRINCIPAL ACCOUNTANT FEES AND SERVICES . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .

PART IV 

Item 15. EXHIBITS AND FINANCIAL STATEMENT SCHEDULES . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .
SIGNATURES . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .

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“SAFE HARBOR” STATEMENT 

Some of the information contained in this Annual Report may include forward-looking statements within the meaning of Section 
27A of the Securities Act of 1933, as amended, or the Securities Act, and Section 21E of the Securities Exchange Act of 1934, as 
amended,  or  the  Exchange  Act.  We  base  these  forward-looking  statements  on  our  current  views  with  respect  to  our  research  and 
development activities, business strategy, business plan, financial performance and other matters, both with respect to us, specifically, 
and  the  biotechnology  sector,  in  general.  Statements  that  include  the  words  “expect,”  “intend,”  “plan,”  “believe,”  “project,” 
“estimate,”  “may,”  “should,”  “anticipate,”  “will”  and  similar  statements  of  a  future  or  forward-looking  nature  identify  forward-
looking statements for purposes of the federal securities laws or otherwise, but the absence of these words does not necessarily mean 
that a statement is not forward-looking. 

All forward-looking statements involve inherent risks and uncertainties, and there are or will be important factors that could cause 
actual results to differ materially from those indicated in these statements. We believe that these factors include, but are not limited to, 
those  factors  set  forth  in  the  sections  entitled  “Business,”  “Risk  Factors,”  “Legal  Proceedings,”  “Management’s  Discussion  and 
Analysis  of  Financial  Condition  and  Results  of  Operations,”  “Quantitative  and  Qualitative  Disclosures  About  Market  Risk”  and 
“Controls  and  Procedures”  in  this  Annual  Report,  all  of  which  you  should  review  carefully.  Please  consider  our  forward-looking 
statements  in  light  of  those  risks  as  you  read  this  Annual  Report.  We  undertake  no  obligation  to  publicly  update  or  review  any 
forward-looking statement, whether as a result of new information, future developments or otherwise, except as required by law. 

If one or more of these or other risks or uncertainties materializes, or if our underlying assumptions prove to be incorrect, actual 
results may vary materially from what we anticipate. All subsequent written and oral forward-looking statements attributable to us or 
individuals  acting  on  our  behalf  are  expressly  qualified  in  their  entirety  by  the  cautionary  language  above.  You  should  consider 
carefully all of the factors set forth or referred to in this Annual Report that could cause actual results to differ. 

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Item 1. BUSINESS 

PART I 

In  this  Annual  Report,  we  sometimes  refer  to  CytRx  Corporation  as  “CytRx,”  to  our  former  subsidiary,  RXi  Pharmaceuticals 
Corporation, as “RXi,” and to Innovive Pharmaceuticals, Inc., which we acquired in September 2008, as “Innovive.” References in 
this Annual Report to the “company,” “we,” “us” or “our” refer to CytRx, alone, unless otherwise indicated. 

COMPANY OVERVIEW 

We are a biopharmaceutical research and development company engaged in the development of high-value human therapeutics, 
specializing  in  oncology.  Our  drug  development  pipeline  includes  clinical  development  of  three  product  candidates  for  cancer 
indications, including three planned Phase 2 clinical trials for INNO-206 as a treatment for pancreatic cancer, gastric (stomach) cancer 
and  soft  tissue  sarcomas,  two  Phase  2  proof-of-concept  clinical  trials  with  bafetinib  in  patients  with  high-risk  B-cell  chronic 
lymphocytic  leukemia,  or  B-CLL,  and  patients  with  glioblastoma  multiforme,  and  a  registration  study  of  tamibarotene  for  the 
treatment  of  acute  promyelocytic  leukemia,  or  APL.  In  addition  to  our  core  oncology  programs,  we  are  developing  two  drug 
candidates  based  on  our  molecular  chaperone  regulation  technology.  Our  current  business  strategy  for  our  molecular  chaperone 
regulation  technology  is  to  seek  one  or  more  strategic  partnerships,  or  a  possible  spin-out  transaction.  Apart  from  our  drug 
development programs, we currently maintain a 36% equity interest in our former subsidiary, RXi. 

We are a Delaware corporation, incorporated in 1985. Our corporate offices are located at 11726 San Vicente Boulevard, Suite 

650, Los Angeles, California 90049, and our telephone number is (310) 826-5648. 

OUR PRODUCT CANDIDATE PIPELINE 

The following tables summarize our product candidates and their current or planned stage of development: 

Technology 

Product Candidate

Indication(s)

Stage of Development

Doxorubicin prodrug . . . . . . . . . . . . . . . . .   INNO-2006 

Tyrosine kinase inhibitor . . . . . . . . . . . . .   Bafetinib 

Synthetic retinoid . . . . . . . . . . . . . . . . . . . .   Tamibarotene 
Molecular chaperone regulation . . . . . . .   Arimoclomol 

Molecular chaperone regulation . . . . . . .   Iroxanadine 

OUR CLINICAL DEVELOPMENT PROGRAMS 

Pancreatic cancer 
Gastric (stomach) cancer 
Soft tissue sarcomas 
B-CLL 
Glioblastoma Multiforme 
APL (acute promyelocytic leukemia) 
ALS (amyotrophic lateral sclerosis, or Lou 
Gehrig’s disease) 
Several potential indications 

Phase II (1H10) 
Phase II (2H10) 
Phase II (2H10) 
Phase II (1H10) 
Phase II (2H10) 
Pivotal Phase II 
Phase II 

Phase I 

Our current clinical development programs consist of our efforts to develop INNO-206 for gastric (stomach) cancer, pancreatic 
cancer  and  soft  tissue  sarcomas,  bafetinib  for  B-CLL  and  glioblastoma  multiforme,  tamibarotene  for  APL,  and  our  molecular 
chaperone regulation program, which includes a planned Phase II clinical study of arimoclomol in ALS. 

INNO-206. INNO-206 (formerly DOXO-EMCH) is a prodrug of the commonly prescribed chemotherapeutic agent doxorubicin. 
Specifically, it is the (6-Maleimidocaproyl) hydrazone of doxorubicin. Essentially, this chemical is doxorubicin (DOXO) attached to 
an acid sensitive linker (EMCH). 

INNO-206 for the Treatment of Cancer. Anthracyclines are a class of drugs that are among the most commonly used agents in the 
treatment of cancer. Doxorubicin, the first anthracycline to gain FDA approval, has demonstrated efficacy in a wide variety of cancers 
including breast cancer, lung cancer, sarcomas, and lymphomas. However, due to the uptake of doxorubicin by various parts of the 
body, it is associated with side effects such as cumulative cardiotoxicity, myelosuppression (decreased production of blood cells by 
bone marrow), gastrointestinal disorders, mucositis (inflammation of the mucous membranes lining the digestive tract, including the 
mouth), stomatitis (inflammation of the mouth’s soft tissue), and extravasation (the leakage of intravenous drugs from the vein into the 
surrounding tissue). 

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We believe INNO-206 has attributes that improve on native doxorubicin, including reduction of adverse events, improvement in 

efficacy and the ability to reach the tumor more quickly. 

Our anticipated mechanism of action for INNO-206 is as follows: 

• 

• 

• 

• 

after administration, INNO-206 rapidly binds circulating albumin through the EMCH linker; 

circulating  albumin  preferentially  accumulates  in  tumors,  bypassing  uptake  by  other  non-tumor  sites,  including  the  heart, 
bone marrow and the gastrointestinal tract; 

once albumin-bound INNO-206 reaches the tumor, the acidic environment of the tumor causes cleavage of the acid sensitive 
linker; and 

free doxorubicin is released at the site of the tumor and is taken up by the cancer cells. 

Pre-clinical  data.  In  a  variety  of  preclinical  models,  INNO-206  was  superior  to  doxorubicin  in  its  ability  to  increase  the  total 
doxorubicin  dose,  antitumor  efficacy,  and  safety,  including  a  reduction  in  cardiotoxicity.  Animal  studies  conducted  by  INNO-206 
inventor Dr. Felix Kratz, Department of Medical Oncology, Clinical Research, at the Tumor Biology Center in Freiburg, Germany, 
demonstrated  statistically  significant  efficacy  against  breast,  ovarian,  pancreatic  and  small  cell  lung  cancers  growing  in 
immunodeficient mice. 

Clinical data. A Phase I study of INNO-206 that demonstrated safety and objective clinical responses in a variety of tumor types 
was  completed  in  2005  and  presented  at  the  March  2006  Krebskongress  meeting  in  Berlin.  In  this  study,  single  doses  were 
administered  every  3  weeks  at  up  to  six  times  the  standard  dosing  of  doxorubicin  without  an  increase  in  side  effects  over  those 
historically  observed  with  doxorubicin.  Twenty-three  of  35  evaluable  patients  had  either  an  objective  clinical  (partial)  response  or 
stable disease. Objective clinical responses were observed in patients with sarcoma, breast, and lung cancers. 

Development Plan. Based on the objective clinical responses seen in the Phase I study, and preclinical data, we intend to initiate 

three Phase 2 clinical trials in 2010 of INNO-206 in patients with pancreatic cancer, gastric cancer and soft tissue sarcomas. 

Bafetinib. Bafetinib (formerly INNO-406) is a novel drug developed by the Japanese pharmaceutical company Nippon Shinyaku, 
to overcome the limitations of Gleevec and second-line tyrosine kinase inhibitors in resistant chronic myelogenous leukemia, or CML. 
We  have  announced  plans  to  develop  bafetinib  as  a  treatment  for  B-cell  chronic  lymphocytic  leukemia  (B-CLL)  and  glioblastoma 
multiforme (GBM), due to the potent and specific inhibitory properties of bafetinib against Lyn kinase, which is overexpressed in both 
B-CLL and GBM. 

Bafetinib for the Treatment of B-CLL. B-CLL is the most common form of leukemia in adults in Western countries. More than 
17,000 new cases of B-CLL are reported in the United States each year; however up to an estimated 40% of cases may not be reported 
due to under-diagnosis and lack of placement in cancer registries. Virtually all patients are older than 55 years at presentation, with an 
average age of 70 years. Patients in the high-risk B-CLL classification have a median overall survival of one to five years. 

Pre-clinical Data. In mice-leukemia models, bafetinib has been shown to markedly extend the survival of animals implanted with 
Gleevec-resistant leukemic cells. In toxicology studies done in mice, rats, and dogs, bafetinib appeared to be safe and well-tolerated. A 
dose described in dogs at which no side effects were seen was used to calculate the starting dose in humans for our recently completed 
clinical trial. 

Phase I Study. In November 2008, we announced that bafetinib demonstrated clinical responses in patients with CML in a Phase I 
clinical trial conducted in patients with CML and other leukemias that have a certain mutation called the Philadelphia Chromosome 
(Ph+)  and  are  intolerant  of  or  resistant  to  Gleevec  and,  in  some  cases,  second-line  tyrosine  kinase  inhibitors  such  as  dasatinib 
(Sprycel®)  and  nilotinib  (Tasigna®)).  The  clinical  trial  was  designed  to  identify  the  optimal  dose  for  possible  future  studies  by 
escalating doses from 30 mg once per day to up to 480 mg twice per day in a total of 56 patients with Ph+ leukemias. Of the patients, 
31 had CML in chronic phase (CML-CP), nine were in accelerated phase (CML-AP), seven were in blast phase (CML-BP), and nine 
had  Ph+  acute  lymphocytic  leukemia.  The  clinical  trial  was  conducted  at  seven  clinical  sites  in  the  US,  Germany,  and  Israel,  with 
Hagop Kantarjian, M.D., Professor & Chairman, Department of Leukemia, The University of Texas, M.D. Anderson Cancer Center, 
serving as the Principal Investigator. A positive, dramatic decrease in the number of leukemia cells in the bone marrow was seen in 
35% of the patients that were randomly chosen to begin their treatment with the optimal bafetinib dose of 240 mg twice per day.

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The maximum tolerated dose was determined to be 240 mg given twice per day, based on evidence of increasing potential liver 
toxicity at higher doses. Common adverse events (observed in greater than 20% of patients in the 240 mg twice per day dose group) 
were  gastrointestinal  toxicity,  swelling,  and  fatigue.  There  was  no  evidence  of  fluid  accumulating  around  the  lungs,  or  significant 
changes  in  a  certain  heart  rhythm  called  QTc  prolongation,  which  are  serious  side  effects  known  to  occur  in  patients  treated  with 
approved  drugs  for  this  indication.  Approximately  13%  of  patients  across  all  dose  groups  discontinued  dosing  due  to  unacceptable 
toxicity. 

Development Plan. We recently announced plans to initiate in the first half of 2010 a Phase 2 proof-of-concept clinical trial to 
evaluate the efficacy and safety of bafetinib in patients with B-CLL. In the planned Phase 2 trial, approximately 20 patients who have 
failed  treatment  with  first-line  agents  will  be  administered  daily  oral  doses  of  bafetinib.  Patients  will  be  monitored  for  clinical 
response,  time  to  disease  progression  and  cancer  progression-free  survival.  Based  on  trial  results,  we  plan  to  conduct  a  larger 
comparative trial to further determine efficacy of this agent. We also plan to initiate a clinical Phase 2 proof of concept clinical trial 
with bafetinib as a treatment for glioblastoma multiforme, a common and aggressive type of primary brain tumor, in the second half of 
2010. 

Tamibarotene. Tamibarotene is an orally available, synthetic retinoid rationally designed to overcome resistance and avoid toxic 

side effects of differentiation therapy with all-trans retinoic acid, or ATRA, a component of the current first-line treatment for APL. 

Tamibarotene  for  the  treatment  of  APL.  Acute  promyelocytic  leukemia,  or  APL,  is  a  specific  type  of  acute  myeloid  leukemia 
characterized by the t(15;17) translocation, which fuses the promyelocytic leukemia, or PML, gene on chromosome 15 to the retinoic 
acid receptor, or RARα gene on chromosome 17. This fusion causes abnormal cell growth. 

Differentiation therapy with ATRA, is the basis for the treatment of APL. Differentiation therapy causes leukemic promyelocytes 
to mature and undergo cell death. Patients typically receive ATRA in combination with chemotherapy as the initial therapy, followed 
by  anthracyline-based  consolidation  therapy  designed  to  produce  complete  remission.  The  majority  of  patients  treated  this  way 
generally experience a complete remission of disease. Current National Comprehensive Cancer Network guidelines recommend that 
patients then undergo one to two years of maintenance therapy with ATRA to prevent a recurrence. ATRA therapy is associated with 
several toxicities, the most serious of which, retinoic acid syndrome, or RAS. RAS, which occurs in up to 25% of patients treated with 
ATRA, is a serious and potentially fatal complication characterized by fever, dyspnea (breathing difficulties), weight gain, pulmonary 
infiltrates (abnormal accumulation in the lungs), and pleural or pericardial effusions (excess fluid around the lungs or heart). 

Patients that initially respond to front-line therapy with ATRA plus chemotherapy sometimes relapse, and some of these patients 
fail to respond to a second course of treatment with ATRA. Currently, patients who fail ATRA-based therapy are treated with arsenic 
trioxide,  a  compound  administered  intravenously  and  associated  with  significant  toxicity,  including  irregular  heartbeat.  There 
currently  is  no  standard  of  care  for  patients  who  do  not  respond  to  ATRA  and  arsenic  trioxide,  or  who  respond  but  subsequently 
relapse. In 2007, the FDA granted Orphan Drug Designation and Fast Track Designation for the use of tamibarotene in patients with 
relapsed or refractory APL following treatment with ATRA and arsenic trioxide. 

Tamibarotene was developed to overcome resistance to ATRA. In vitro, tamibarotene is approximately ten times more potent than 
ATRA at causing APL cells to differentiate and die. In addition, tamibarotene has a lower affinity for cellular retinoic acid binding 
protein,  or  CRABP,  which  we  believe  should  allow  for  sustained  plasma  levels  during  administration.  This  may  enhance 
tamibarotene’s  potential  efficacy,  because  patients  may  be  able  to  experience  benefits  from  the  drug  over  a  longer  period  of  time. 
Tamibarotene does not bind the RAR-γ receptor, the major retinoic acid receptor in the dermal epithelium, which should lessen the 
occurrence of skin toxicities. 

Pre-clinical data. In preclinical models, tamibarotene was superior to ATRA in its ability to cause APL cells to differentiate and 
die. In the clinical setting, in vitro response to tamibarotene appeared predictive of clinical response, including activity in patients who 
had a poor response to ATRA. 

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Clinical  data.  Tamibarotene  is  approved  in  Japan  under  the  brand  name  Amnolake  for  use  in  relapsed  or  refractory  APL.  The 
approval  was  based  on  data  from  two  studies  in  Japanese  patients.  In  the  pivotal  study,  the  effectiveness  of  orally  administered 
tamibarotene was administered to 42 patients with APL, 39 of whom were evaluable for response. Patients included individuals who 
had  never  received  treatment  for  APL  and  patients  who  had  been  previously  treated  with  ATRA.  Tamibarotene  was  administered 
orally at a dose of 6 mg/m2/day for eight weeks. The overall complete response rate in these patients was 61.5%. In patients who had a 
recurrence of APL following ATRA therapy, the response rate was 81%. RAS was reported in three patients, or 7.3% of the patient 
group. 

Development  Plan.  There  is  currently  a  Special  Protocol  Assessment  (SPA)  in  place  with  the  FDA  for  a  Phase  2  registration 
clinical trial, known as STAR-1, which is evaluating the efficacy and safety of tamibarotene as a third-line treatment for APL. The 
STAR-1 trial is ongoing and currently includes six clinical sites in the U.S. We recently reported that, of the 11 patients enrolled in the 
STAR-1  trial  to  date,  three  (27%)  achieved  a  hematologic  complete  response,  and  four  (36%)  a  morphologic  leukemia-free  state. 
Depending on the trial’s outcome, this study, in combination with the data from the two Japanese studies, could form the basis of a 
new drug application, or NDA. 

In addition, we have announced plans to develop tamibarotene, in combination with chemotherapy or arsenic trioxide (ATO), as a 
first-line treatment for APL. We have received favorable reviews on tamibarotene as a potential treatment for APL from key opinion 
leaders and have been working with notable clinicians in this field on trial design. 

Among other preparatory activities, in September 2009, we initiated a dose escalation clinical trial with tamibarotene combined 
with TRISENOX® (arsenic trioxide) injection (marketed by Cephalon, Inc.) in patients with relapsed APL. An objective of this trial is 
to determine the appropriate combination therapy dose for evaluation as a potential first-line treatment for APL. 

Arimoclomol. Arimoclomol is an orally-administered small-molecule product candidate that we believe functions by stimulating a 

normal cellular protein repair pathway by amplifying molecular chaperone proteins implicated in neurological disorders. 

Arimoclomol for the treatment of ALS. ALS, or Lou Gehrig’s disease, is a debilitating and ultimately deadly disease involving the 
progressive degeneration of motor neurons believed to be caused by toxic mis-folding of proteins. According to the ALS Association, 
approximately 30,000 people in the U.S. are living with ALS and 5,600 new cases are diagnosed each year. Worldwide, an estimated 
120,000 people are living with ALS. According to the ALS Survival Guide, 50% of ALS patients die within 18 months of diagnosis 
and 80% die within five years of diagnosis. 

The following is a summary of our clinical development of arimoclomol for treating ALS: 

• 

• 

• 

• 

in July 2006, we completed an 84-patient, multi-center, double-blind, placebo-controlled, multi-dose Phase IIa clinical trial of 
safety and tolerability of arimoclomol in volunteers with ALS, which we refer to as the Phase IIa trial; 

in May 2007, we completed an open-label extension of the Phase IIa trial in approximately 70 ALS patients from the trial 
who  were  administered  the  highest  investigational  dose  (100  mg  three  times  daily)  of  arimoclomol  for  an  additional  six 
months; 

in June 2007, we completed a multiple ascending-dose clinical trial of safety and tolerability involving 40 healthy volunteers; 
and 

in November 2007, we completed a 28-day safety clinical trial with 400 mg of arimoclomol three times daily involving 16 
healthy volunteers. 

Phase IIa clinical trial. Participants in the Phase IIa clinical trial of arimoclomol were administered either a placebo capsule, or 
one of three dosage levels of arimoclomol capsules, three times daily for a period of 12 weeks, immediately followed by a one-month 
period  without  the  drug.  The  primary  endpoints  of  the  Phase  IIa  trial  were  safety  and  tolerability.  Secondary  endpoints  included  a 
preliminary  evaluation  of  efficacy  using  two  widely  accepted  disease-progression  markers.  The  first  marker,  the  revised  ALS 
Functional Rating Scale, or ALSFRS-R, is used to determine patients’ overall functional capacity and independence in 13 activities. 
The  second  marker  measures  vital  capacity,  an  assessment  of  lung  capacity,  which  is  an  important  disease  indicator  since  ALS 
sufferers eventually lose the ability to breathe on their own. The trial was designed to be able to detect only extreme responses in these 
two markers. 

7 

  
  
  
  
  
  
  
  
  
  
  
 
 
The results from our Phase IIa trial and open-label extension clinical trial indicated that arimoclomol was safe and well tolerated 
in  ALS  volunteers,  even  at  the  highest  administered  dose.  Arimoclomol  was  detected  in  participants’  cerebral  spinal  fluid, 
demonstrating  that  it  passed  the  so-called  blood:brain  barrier,  and  participants  treated  with  arimoclomol  experienced  a  statistically 
significant decrease in adverse events of weakness compared with the placebo group. 

Phase IIb efficacy trial. In December 2009, the FDA accepted a revised protocol for an ascending dose efficacy trial to evaluate 
the safety and efficacy in ALS patients at up to 400 mg administered orally three times daily. The clinical trial protocol accepted by 
the  FDA  is  a  tiered,  placebo-controlled,  double-blind  ascending  dose  study.  The  study  is  designed  to  test  progressive  groups,  each 
with  between  20  and  30  ALS  patients  over  a  three-month  treatment  period.  Fifteen  patients  would  receive  a  combination  of 
arimoclomol at various dose levels and riluzole at a fixed dose of 50 mg twice daily, with between five and 15 ALS patients receiving 
placebo and riluzole at the same fixed dose. The first group would receive arimoclomol 100 mg capsules three times daily. Every four 
weeks,  another  group  of  ALS  patients  would  begin  three-month  testing  with  six  patients  receiving  arimoclomol  dosing  three  times 
daily at a 75 mg per dose increase from the prior group. The maximum dose in the protocol allows for testing arimoclomol at 400 mg 
three times daily. An independent safety monitoring board would review safety results prior to initiating each consecutive increase in 
dosage level. 

Other Clinical Development. In February 2009, a Phase II/III adaptive clinical trial commenced to study arimoclomol in a subset 
of patients with the inherited or familial form ALS. Patients with familial ALS (fALS) who harbor certain mutations in the superoxide 
dismutase-1 (SOD1) gene suffer from a rapidly progressing form of the disease. The clinical trial is being financially supported by 
grants  from  the  ALS  Association  and  the  U.S.  Food  and  Drug  Administration’s  (FDA’s)  Office  of  Orphan  Products  Development 
(OOPD),  and  we  are  supplying  the  drug  and  allowing  the  sponsor  to  reference  our  Investigational  New  Drug  Application  for 
regulatory purposes. 

Arimoclomol for recovery from stroke. Stroke results from an acute loss of normal blood flow to the brain caused most often by a 
blockage  in  a  blood  vessel  (ischemic)  or  due  to  leaking  of  blood  from  a  vessel  (hemorrhagic).  According  to  the  American  Heart 
Association: stroke is the third leading cause of death and the number one cause of long-term disability in the U.S.; between 50% and 
70%  of  stroke  survivors  regain  functional  independence,  but  between  15%  and  30%  are  permanently  disabled  and  20%  require 
institutional care within three months after stroke; and the direct and indirect stroke cost in the U.S. totaled approximately $58 billion 
in 2006. 

After the normal flow of blood is restored to the brain, post-stroke neurological function continues to decline. We believe that this 
continuing  decline  in  neurological  function  is  the  consequence  of  mis-folded  protein  aggregates  generated  as  a  result  of  oxygen 
deprivation  during  the  original  event.  Preclinical  efficacy  studies  completed  by  us  in  April  2007  indicated  that  arimoclomol 
accelerated the time to recovery, and improved recovery, in experimental animal models of stroke. These results were obtained even 
when arimoclomol was administered as long as 48 hours after onset. 

Arimoclomol  for  the  treatment  of  cancer.  Through  research  conducted  in  our  former  San  Diego  laboratory,  we  have  identified 
preclinical  pipeline  compounds  that  inhibit,  rather  than  amplify,  molecular  chaperone  proteins.  These  early  stage  compounds  are 
potential oncology therapeutics because cancer cells by their very nature generate large amounts of toxic, misfolded proteins and are 
far  more  dependent  upon  the  activity  of  molecular  chaperone  proteins  for  survival  than  are  normal  cells.  Because  several  of  these 
compounds have already been shown to selectively kill cancer cells and spare normal cells in tissue culture, they represent a novel 
approach to cancer therapeutics with the potential of having relatively large therapeutic indices. 

Iroxanadine. Iroxanadine also is an orally-administered small-molecule product candidate. We believe it functions by stimulating 
the  molecular  chaperone  protein  response  in  the  endothelium,  the  thin  layer  of  cells  that  line  the  interior  surface  of  human  blood 
vessels. 

Iroxanadine  for  the  treatment  of  diabetic  ulcers.  Type  2  diabetes  is  a  major  health  problem  with  significant  secondary 
complications. The American Diabetes Association estimates that there are 21 million type 2 diabetes sufferers in the U.S. The World 
Health Organization estimates that there are more than 162 million cases of type 2 diabetes worldwide. According to the American 
Diabetes Association, 15% of all diabetics will develop a foot ulcer during their lifetime, and over 82,000 non-traumatic lower-limb 
amputations were performed on diabetics in the U.S. in 2002 due to ulcers and other complications. We believe there are reasonable 
data  in  the  scientific  literature  supporting  the  concept  that  diabetic  foot  ulcers  fail  to  heal  efficiently  due  to  the  dysfunction  of 
endothelial cells lining the blood vessels caused by protein mis-folding. 

8 

  
  
  
  
  
  
  
 
 
Animal studies completed by us in May 2007 indicated that iroxanadine significantly decreased the time it took for wounds to 
heal in diabetic mice without affecting healing in healthy mice. Wound healing in the diabetic mice, which normally required twice 
the  time  to  heal  as  healthy  mice,  was  accelerated  to  the  extent  that  healing  time  of  diabetic  mice  treated  with  iroxanadine  was 
indistinguishable from that in untreated healthy mice. 

In Phase I clinical trials in healthy volunteers and Phase II clinical trials in patients with chronic high blood pressure conducted 
prior  to  our  acquisition  of  iroxanadine,  the  drug  candidate  was  shown  to  be  safe  and  well-tolerated  and  demonstrated  significant 
improvement in the function of endothelial cells in the brachial artery, a major blood vessel of the upper arm. 

Strategic  Plans  for  Molecular  Chaperone  Assets.  We  intend  to  seek  a  partner  for  the  development  of  arimoclomol  and 
iroxanadine for all indications on a worldwide basis. We are also exploring the possibility of a spin-out transaction to accelerate the 
development of our molecular chaperone assets. 

Other Technologies 

Our  other  current  technologies  are  CRL-5861,  an  intravenous  agent  for  treatment  of  sickle  cell  disease  and  other  acute  vaso-
occlusive  disorders,  and  TranzFect,  a  delivery  technology  for  DNA-based  and  conventional  vaccines  and  other  potential  uses.  We 
currently have no plans for development of these technologies. 

Our Separation from RXi Pharmaceuticals Corporation 

Until early 2008, we owned approximately 85% of the outstanding shares of common stock of RXi and our financial statements, 
including our financial statements as of and for the year ended December 31, 2007, included the consolidated financial condition and 
results of operations of RXi. On February 14, 2008, our board of directors declared a dividend of one share of RXi common stock for 
each  approximately  20.05  outstanding  shares  of  our  common  stock,  which  was  paid  on  March  11,  2008  and  which  reduced  our 
ownership  of  RXi  shares  to  less  than  50%.  As  a  result,  our  financial  statements  since  March  11,  2008  no  longer  consolidate  the 
financial condition and results of operation of RXi, but instead reflect our ongoing investment in RXi based on the equity method of 
accounting. As of March 12, 2010, we owned approximately 36% of the outstanding shares of RXi common stock. 

We are party to a letter agreement with RXi and some of RXi’s current stockholders under which we are entitled to preemptive 
rights  to  acquire  any  “new  securities”  (as  defined)  that  RXi  proposes  to  sell  or  issue,  so  that  we  may  maintain  our  percentage 
ownership in RXi. Our preemptive rights will expire on January 8, 2012 or such earlier time at which we own less than 10% of RXi’s 
outstanding common stock. 

Under the letter agreement with RXi, we agreed to vote our RXi shares for the election of RXi directors and take other actions to 
ensure that a majority of the board of directors of RXi are independent of us. We further agreed to approve of actions that may be 
adopted and recommended by the RXi board of directors to facilitate any future financing by RXi. 

Manufacturing 

We have no capability to manufacture supplies of any of our products, and rely on third-party manufacturers to produce materials 
needed  for  research  and  clinical  trials.  We  have  contracted  with  various  contract  manufacturing  facilities  for  supply  of  our  active 
pharmaceutical ingredient, or API, for our product candidates. Pursuant to our license with TMRC Co., Ltd., or TMRC, relating to 
tamibarotene, TMRC will provide us with tamibarotene at a fixed price and in a quantity and quality sufficient to meet our clinical and 
commercial needs. 

To  be  commercialized,  our  products  also  must  be  capable  of  being  manufactured  in  commercial  quantities  in  compliance  with 
stringent  regulatory  requirements  and  at  an  acceptable  cost. We  intend  to  rely  on  third-party  manufacturers  to  produce  commercial 
quantities of any products for which we are able to obtain marketing approval. We have not commercialized any product, and so we 
also  have  not  demonstrated  that  any  of  our  product  candidates  can  be  manufactured  in  commercial  quantities  in  accordance  with 
regulatory requirements or at an acceptable cost. 

If our product candidates cannot be manufactured in suitable quantities and in accordance with regulatory standards, our clinical 
trials,  regulatory  approvals,  and  marketing  efforts  for  such  products  may  be  delayed.  Such  delays  could  adversely  affect  our 
competitive position and our chances of generating significant recurring revenues. If our products are not able to be manufactured at 
an acceptable cost, the commercial success of our products may be adversely affected. 

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Marketing 

Our  tentative  plan  is  to  establish  our  own  sales  force  and  marketing  capability  in  order  to  commercialize  our  oncology  drug 
candidates,  including  INNO-206,  bafetinib  and  tamibarotene,  in  the  U.S.  and  to  seek  a  marketing  partner  for  commercialization  in 
other territories. 

Patents and Proprietary Technology 

We actively seek patent protection for our technologies, processes, uses, and ongoing improvements and consider our patents and 
other intellectual property to be critical to our business. We acquired patents and patent applications, and have filed several new patent 
applications, in connection with our molecular chaperone program. 

We regularly evaluate the patentability of new inventions and improvements developed by us or our collaborators, and, whenever 
appropriate,  will  endeavor  to  file  U.S.  and  international  patent  applications  to  protect  these  new  inventions  and  improvements.  We 
cannot be certain that any of the current pending patent applications we have filed or licensed, or any new patent applications we may 
file or license, will ever be issued in the U.S. or any other country. There also is no assurance that any issued patents will be effective 
to  prevent  others  from  using  our  products  or  processes.  It  is  also  possible  that  any  patents  issued  to  us,  as  well  as  those  we  have 
licensed or may license in the future, may be held invalid or unenforceable by a court, or third parties could obtain patents that we 
would need to either license or to design around, which we may be unable to do. Current and future competitors may have licensed or 
filed patent applications or received patents, and may acquire additional patents and proprietary rights relating to molecular chaperone 
amplification and other small molecule technology or other compounds, products or processes that may be competitive with ours. 

In  addition  to  patent  protection,  we  attempt  to  protect  our  proprietary  products,  processes  and  other  information  by  relying  on 
trade  secrets  and  non-disclosure  agreements  with  our  employees,  consultants  and  certain  other  persons  who  have  access  to  such 
products,  processes  and  information.  Under  the  agreements,  all  inventions  conceived  by  employees  are  our  exclusive  property,  but 
there is no assurance that these agreements will afford significant protection against misappropriation or unauthorized disclosure of 
our trade secrets and confidential information. 

LICENSE AGREEMENTS 

INNO-206 

We succeeded to Innovive’s agreement with KTB Tumorforschungs GmbH, or KTB, for the license of patent rights held by KTB 
for the worldwide development and commercialization of INNO-206. The license is exclusive and worldwide, applies to all product 
that  may  be  subject  to  the  licensed  intellectual  property  and  may  be  used  in  all  fields  of  use.  We  may  sublicense  the  intellectual 
property in our sole discretion. The agreement also grants us an option to include within the license any technology that is claimed or 
disclosed in the licensed patents and patent applications for use in the field of oncology and the right of first refusal on any license that 
KTB  wishes  to  make  to  a  third  party  regarding  any  technology  that  is  claimed  or  disclosed  in  the  licensed  patents  and  patent 
applications for use in the field of oncology. 

Under  the  agreement,  we  must  make  payments  to  KTB  in  the  aggregate  of  $7.5  million  upon  meeting  clinical  and  regulatory 

milestones up to and including the product’s second final marketing approval. We also agreed to pay: 

• 

• 

commercially reasonable royalties based on a percentage of net sales (as defined in the agreement); 

a percentage of non-royalty sub-licensing income (as defined in the agreement); and 

•  milestones of $1 million for each additional final marketing approval that we might obtain. 

In the event that we must pay a third party in order to exercise our rights to the intellectual property under the agreement, we will 
deduct a percentage of those payments from the royalties due KTB, up to an agreed upon cap. This deduction includes a percentage of 
any payments that might be required to be made by us to Bristol-Myers Squibb. Bristol-Myers Squibb holds a patent on technology 
that might be considered to block the patents and patent applications that are the subject of the agreement with KTB. 

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Under the agreement with KTB, we must use commercially reasonable efforts to conduct the research and development activities 
we determine are necessary to obtain regulatory approval to market the product in those countries that we determine are commercially 
feasible. Under the agreement, KTB is to use its commercially reasonable efforts to provide us with access to suppliers of the API of 
the product on the same terms and conditions as may be provided to KTB by those suppliers. 

The agreement will expire on a product-by-product basis upon the expiration of the subject patent rights. We have the right to 
terminate the agreement on 30 days notice, provided we pay a cash penalty to KTB. KTB may terminate the agreement if we are in 
breach and the breach is not cured within a specified cure period or if we fail to use diligent and commercial efforts to meet specified 
clinical milestones. 

Bafetinib 

We likewise succeeded to Innovive’s exclusive, worldwide (with the exception of Japan) royalty-bearing license agreement with 
Nippon Shinyaku, including the right to grant sublicenses, for the intellectual property relating to bafetinib in all fields. The license 
agreement will expire on a country-by-country basis upon the expiration of the subject patent rights. The bafetinib license covers two 
Patent Cooperation Treaty, or PTC, applications filed in 2003 and 2004, respectively. 

Under  the  agreement,  we  are  obliged  to  pay  Nippon  Shinyaku  an  aggregate  of  $13.35  million  (including  $5  million  upon  the 
product’s initial final marketing approval) upon the achievement of clinical and regulatory milestones up to and including approvals in 
the U.S. and Europe. We also will be obliged to pay: 

• 

• 

• 

commercially reasonable royalties based on a percentage of net sales (as defined in the Nippon Shinyaku license agreement), 
dependent on reaching certain revenue thresholds; 

annual minimum payments if sales of bafetinib do not meet specified levels; and 

a percentage of non-royalty sub-licensing income (as defined in the license agreement). 

The  agreement  includes  covenants  that  require  us  to,  among  other  things,  file  an  NDA  by  a  specific  date  and  use  our 
commercially  reasonable  efforts  to  bring  a  licensed  product  to  market.  In  the  event  that  we  breach  a  material  term  of  the  Nippon 
Shinyaku  license  agreement,  Nippon  Shinyaku  has  the  option  to  terminate  the  agreement  following  the  giving  of  notice  and  an 
opportunity to cure any such breach. 

Tamibarotene 

We also succeeded to Innovive’s agreement with TMRC for the license of patent rights held by TMRC for the North American 
development  and  commercialization  of  tamibarotene.  The  license  is  exclusive,  applies  to  all  products  that  may  be  subject  to  the 
licensed  intellectual  property  and  may  be  used  in  the  treatment  of  APL.  We  may  sublicense  the  intellectual  property  in  our  sole 
discretion.  The  agreement  also  grants  us  an  option  to  include  within  the  license  the  use  of  the  drug  in  other  fields  in  oncology 
including multiple myeloma, myelodysplastic syndrome, and solid tumors. 

Under the agreement, we must pay TMRC royalties based on net sales and make payments to TMRC in the aggregate of $4.165 
million  upon meeting  clinical,  regulatory, and sales  milestones up  to  and  including  the  first  commercial  sale  of  the  product  for  the 
treatment of APL. 

Under  the  agreement,  we  must  use  commercially  reasonable  efforts  to  conduct  the  research  and  development  activities  we 
determine are necessary to obtain regulatory approval to market the product in those countries in North America that we determine are 
commercially feasible. 

The agreement will expire upon the expiration of the subject patent rights, or 15 years from the date of first commercial sale of 
product in North America, whichever is later. The agreement may be terminated if either party is in breach and the breach is not cured 
within a required amount of time. We may also terminate the agreement in the event of a material change in the safety profile of the 
technology that makes continued development impossible. 

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Under the merger agreement by which we acquired Innovive, we agreed to pay the former Innovive stockholders up to $1.01 per 
Innovive share of future earnout merger consideration, subject to our achievement of specified net sales under the Innovive license 
agreements. The earnout merger consideration, if any, will be payable in shares of our common stock, subject to specified conditions, 
or,  at  our  election,  in  cash  or  by  a  combination  of  shares  of  our  common  stock  and  cash.  Our  common  stock  will  be  valued  for 
purposes of any future earnout merger consideration based upon the trading price of our common stock at the time the earnout merger 
consideration is paid. 

Competition 

INNO-206  is  a  prodrug  of  doxorubicin,  a  widely  used  anti-cancer  drug.  Doxorubicin  is  part  of  the  anthracycline  class  of 
chemotherapy agents. Anthracyclines, many of which are generic including doxorubicin, have been used throughout the world to treat 
various cancers for several decades. Due to their track record of broad anti-cancer activity, new types of anthracyclines and modified 
or reformulated versions continue to be developed to overcome toxicities which limit the use of these drugs. 

INNO-206  is  a  chemically  modified  version  of  doxorubicin  that  incorporates  an  acid  sensitive  linker  technology  to  improve 
targeting to the tumor. We believe that the albumin-binding ability of INNO-206 will allow the compound to overcome many of the 
side  effect  issues  typically  associated  with  anthracyclines.  We  also  believe  that  using  albumin  as  a  targeted  carrier  will  allow  for 
higher dosing and greater efficacy. 

Soft tissue sarcoma patients are typically treated with surgery followed by radiation therapy. Doxorubicin is the only approved 
drug for treating soft tissue sarcoma and is often used in combination with radiation. The National Comprehensive Cancer Network 
also  includes  the  use  of  ifosfamide,  epirubicin,  Eli  Lilly’s  Gemzar,  dacarbazine  and  liposomal  doxorubicin  marketed  in  the  US  as 
Doxil  by  Johnson  &  Johnson.  For  patients  ineligible  for  surgery,  radiation  and/or  chemotherapy  is  the  only  option.  Based  on  both 
human  and  animal  data,  we  believe  we  can  give  5-8  times  the  amount  of  doxorubicin  with  administration  of  INNO-206.  Other 
approaches  to  treating  soft  tissue  sarcoma  are  in  late  stage  clinical  development.  These  include  ridaforolimus  being  developed  by 
Ariad  Pharmaceuticals  and  Merck  &  Co.,  GlaxoSmithKline’s  pazopanib,  Sanofi-Aventis’  AVE8062,  Threshhold  Pharmaceuticals’s 
TH-302, and trabectedin being co-developed by Johnson and Johnson and PharmaMar. 

Advanced gastric cancer patients are those that have failed both surgery and prior chemotherapy. They may or may not be suitable 
candidates for chemoradiation. These patients are typically treated with a variety of combination of approved drugs such as cisplatin, 
docetaxel,  5-FU,  oxaliplatin,  iriniotecan  and  paclitaxel.  Epirubicin,  an  anthracycline,  is  part  of  several  gastric  cancer  treatment 
regimens. We believe INNO-206 could be a potentially more effective anthracycline and potentially more effective in this setting. 

Pancreatic  cancer  is  one  of  the  most  lethal  types  of  cancer  and  current  treatment  options  have  limited  benefit  due  to  the  rapid 
progression  of  this  cancer.  Patients  are  typically  treated  with  surgery,  radiation  and  chemotherapy.  Eli  Lilly’s  Gemzar  is  currently 
approved for the first line treatment of locally advanced or metastatic pancreatic cancer. It is also indicated for the use in patients who 
have  received  prior  treatment  with  5-FU.  OSI  Pharmaceuticals’  Tarceva  was  approved  in  2005  for  the  use  in  combination  with 
Gemzar. The NCCN believes the best management for these patients is in a clinical trial. Because of the tremendous unmet need for 
these  patients,  many  companies  are  developing  new  drugs  to  treat  pancreatic  cancer.  Late  stage  drugs  in  clinical  trials  include 
Abraxane by Abraxis BioScience, AGS-1C4D4 by Astellas Pharma Inc., TNFerade™ by GenVec, and S-1 by Sanofi-Aventis. 

There are currently three marketed competitors to bafetinib (formerly INNO-406) in the CML market, Gleevec®, Sprycel® and 
Tasigna®.  Gleevec  is  approved  for  treatment  of  newly  diagnosed  adult  patients  with  Philadelphia  chromosome–positive  chronic 
myeloid leukemia (Ph+ CML) in the chronic phase and patients with Ph+ CML in blast crisis (BC), accelerated phase (AP), or in the 
chronic  phase  (CP)  after  failure  of  interferon-alpha  therapy.  Sprycel®  and  Tasigna®  are  approved  for  Gleevec-resistant  CML. 
Because  of  the  highly  competitive  nature  of  the  CML  market  including  drug  candidates  in  development,  CytRx  plans  to  develop 
bafetinib  initially  in  cancers  other  than  CML.  CytRx  has  selected  B-cell  chronic  lymphocytic  leukemia  (B-CLL)  and  glioblastoma 
multiforme  due  to  the  potent  and  specific  inhibitory  properties  of  bafetinib  against  Lyn  kinase.  Lyn kinase  is  a  member  of  the Src 
family  of  kinases  which  are  known  to  be  involved  in  cell  growth.  Lyn  kinase  is  overexpressed  in  both  B-CLL  and  glioblastoma 
multiforme (GBM). 

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We are unaware of any compounds in development that target Lyn kinase. We plan to develop bafetinib as a treatment for B-CLL 
patients  that  have  failed  first-line  therapy.  There  are  several  drugs  approved  for  the  treatment  of  CLL.  First-line  therapy  for  CLL 
includes  a  variety  of  combination  therapies  including  fludarabine,  cyclophosphamide,  Rituxan®  and  Campath®.  Treatment  for 
relapsed or refractory CLL includes several chemotherapy regimens including CHOP, CFAR, hyperCFAD and OFAR in addition to 
single agents including GlaxoSmithKline’s ArzerraTM. Arzerra was approved in October 2009 for CLL patients who are refractory to 
treatment with fludarabine and Campath. 

Current therapy for glioblastoma  multiforme, the most common form of brain cancer, is surgery followed by radiation therapy 
and chemotherapy. Merck’s Temodar® is approved for treating newly diagnosed GBM concomitantly with radiotherapy and then as a 
maintenance  treatment.  Roche’s  Avastin  was  approved  in  May  2009  for  treatment  of  recurrent  GBM.  We  believe  that  bafetinib’s 
ability  to  selectively  inhibit  Lyn  kinase  and  to  penetrate  the  brain  in  an  animal  model  of  cancer  will  be  an  effective  treatment  for 
second-line therapy in GBM. 

To our knowledge, there are no competitors in clinical development for refractory APL. Currently, treatment of APL is based on 
induction  and  maintenance  therapy  with  ATRA  and  chemotherapy  (typically  idarubicin).  ATRA  and  idarubicin  are  both  generic 
compounds. Arsenic trioxide, currently marketed by Cephalon, is approved for use in patients who have relapsed after ATRA-based 
therapy in APL. There are no FDA-approved therapies for patients who have failed arsenic trioxide. In practice, it appears that patients 
who fail arsenic trioxide are retreated with ATRA or receive Mylotarg, which is marketed by Pfizer Inc. 

We are aware of only one drug, rilutek, developed by Aventis Pharma AG, that has been approved by the FDA for the treatment of 
ALS.  Many  companies  are  working  to  develop  pharmaceuticals  to  treat  ALS,  including  Aeolus  Pharmaceuticals,  Mitsubishi  Tanabe 
Pharma  Corporation,  Ono  Pharmaceuticals,  Trophos  SA,  Knopp  Neurosciences  Inc.,  Faust  Pharmaceuticals  SA,  Oxford  BioMedica  plc, 
Phytopharm plc and Teva Pharmaceutical Industries Ltd., as well as RXi. ALS patients often take over-the-counter supplements, including 
vitamin  E,  creatine  and  coenzyme  Q10,  or  drugs  such  as  lithium  that  are  approved  for  other  indications.  ALS  belongs  to  a  family  of 
neurodegenerative diseases that includes Alzheimer’s, Parkinson’s and Huntington’s diseases. Due to similarities between these diseases, a 
new treatment for one such disease potentially could be useful for treating others. There are many companies producing and developing 
drugs used to treat neurodegenerative diseases other than ALS, including Amgen, Inc., Biogen Idec, Boehringer Ingelheim, Cephalon, 
Inc., Ceregene, Inc., Elan Pharmaceuticals, plc, Forest Laboratories, Inc., H. Lundbeck A/S, Phytopharm plc, UCB Group and Wyeth. 

Many  companies,  including  large  pharmaceutical  and  biotechnology  firms  with  financial  resources,  research  and  development 
staffs,  and  facilities  that  may  be  substantially  greater  than  those  of  ours  or  our  strategic  partners  or  licensees,  are  engaged  in  the 
research and development of pharmaceutical products that could compete with our potential products. To the extent that we seek to 
acquire, through license or otherwise, existing or potential new products, we will be competing with numerous other companies, many 
of which will have substantially greater financial resources, large acquisition and research and development staffs that may give those 
companies a competitive advantage over us in identifying and evaluating these drug acquisition opportunities. Any products that we 
acquire  will  be  competing  with  products  marketed  by  companies  that  in  many  cases  will  have  substantially  greater  marketing 
resources than we have. The industry is characterized by rapid  technological advances and competitors may develop their products 
more rapidly and such products may be more effective than those currently under development or that may be developed in the future 
by our strategic partners or licensees. Competitive products for a number of the disease indications that we have targeted are currently 
being marketed by other parties, and additional competitive products are under development and may also include products currently 
under development that we are not aware of or products that may be developed in the future. 

Government Regulation 

The U.S. and other developed countries extensively regulate the preclinical and clinical testing, manufacturing, labeling, storage, 
record-keeping,  advertising,  promotion,  export,  marketing  and  distribution  of  drugs  and  biologic  products.  The  FDA,  under  the 
Federal  Food,  Drug,  and  Cosmetic  Act,  the  Public  Health  Service  Act  and  other  federal  statutes  and  regulations,  regulates 
pharmaceutical and biologic products. 

To obtain approval of our product candidates from the FDA, we must, among other requirements, submit data supporting safety 
and efficacy for the intended indication as well as detailed information on the manufacture and composition of the product candidate. 
In most cases, this will require extensive laboratory tests and preclinical and clinical trials. The collection of these data, as well as the 
preparation of applications for review by the FDA involve significant time and expense. The FDA also may require post-marketing 
testing to monitor the safety and efficacy of approved products or place conditions on any approvals that could restrict the therapeutic 
claims and commercial applications of these products. Regulatory authorities may withdraw product approvals if we fail to comply 
with regulatory standards or if we encounter problems at any time following initial marketing of our products. 

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The  first  stage  of  the  FDA  approval  process  for  a  new  biologic  or  drug  involves  completion  of  preclinical  studies  and  the 
submission  of  the  results  of  these  studies  to  the  FDA.  These  data,  together  with  proposed  clinical  protocols,  manufacturing 
information,  analytical  data  and  other  information  submitted  to  the  FDA,  in  an  investigational  new  drug  application,  or  IND,  must 
become  effective  before  human  clinical  trials  may  commence.  Preclinical  studies  generally  involve  FDA  regulated  laboratory 
evaluation of product characteristics and animal studies to assess the efficacy and safety of the product candidate. 

After  the  IND  becomes  effective,  a  company  may  commence  human  clinical  trials.  These  are  typically  conducted  in  three 
sequential phases, but the phases may overlap. Phase I trials consist of testing of the product candidate in a small number of patients or 
healthy volunteers, primarily for safety at one or more doses. Phase II trials, in addition to safety, evaluate the efficacy of the product 
candidate in a patient population somewhat larger than Phase I trials. Phase III trials typically involve additional testing for safety and 
clinical efficacy in an expanded population at multiple test sites. A company must submit to the FDA a clinical protocol, accompanied 
by the approval of the Institutional Review Boards at the institutions participating in the trials, prior to commencement of each clinical 
trial. 

To  obtain  FDA  marketing  authorization,  a  company  must  submit  to  the  FDA  the  results  of  the  preclinical  and  clinical  testing, 
together with, among other things, detailed information on the manufacture and composition of the product candidate, in the form of a 
new drug application, or NDA. 

The  amount  of  time  taken  by  the  FDA  for  approval  of  an  NDA  will  depend  upon  a  number  of  factors,  including  whether  the 
product candidate has received priority review, the quality of the submission and studies presented, the potential contribution that the 
compound will make in improving the treatment of the disease in question, and the workload at the FDA. 

The FDA may, in some cases, confer upon an investigational product the status of a fast track product. A fast track product is 
defined as a new drug or biologic intended for the treatment of a serious or life-threatening condition that demonstrates the potential to 
address unmet  medical  needs  for  this  condition.  The  FDA  can base  approval  of an NDA for  a fast track product on  an  effect on  a 
surrogate endpoint, or on another endpoint that is reasonably likely to predict clinical benefit. If a preliminary review of clinical data 
suggests that a fast track product may be effective, the FDA may initiate review of entire sections of a marketing application for a fast 
track  product  before  the  sponsor  completes  the  application.  The  FDA  has  granted  fast  track  designation  and  orphan  drug  status  to 
arimoclomol for the treatment of ALS and to tamibarotene for the treatment of relapsed or refractory APL. 

We anticipate that our products will be manufactured by our strategic partners, licensees or other third parties. Before approving 
an  NDA,  the  FDA  will  inspect  the  facilities  at  which  the  product  is  manufactured  and  will  not  approve  the  product  unless  the 
manufacturing  facilities  are  in  compliance  with  the  FDA’s  cGMP,  which  are  regulations  that  govern  the  manufacture,  holding  and 
distribution  of  a  product.  Our  manufacturers  also  will  be  subject  to  regulation  under  the  Occupational  Safety  and  Health  Act,  the 
Environmental  Protection  Act,  the  Nuclear  Energy  and  Radiation  Control  Act,  the  Toxic  Substance  Control  Act  and  the  Resource 
Conservation  and  Recovery  Act.  Following  approval,  the  FDA  periodically  inspects  drug  and  biologic  manufacturing  facilities  to 
ensure continued compliance with the good manufacturing practices regulations. Our manufacturers will have to continue to comply 
with those requirements. Failure to comply with these requirements subjects the manufacturer to possible legal or regulatory action, 
such as suspension of manufacturing or recall or seizure of product. Adverse patient experiences with the product must be reported to 
the FDA and could result in the imposition of marketing restrictions through labeling changes or market removal. Product approvals 
may be withdrawn if compliance with regulatory requirements is not maintained or if problems concerning safety or efficacy of the 
product occur following approval. 

The labeling, advertising, promotion, marketing and distribution of a drug or biologic product also must be in compliance with 
FDA and Federal Trade Commission requirements which include, among others, standards and regulations for off-label promotion, 
industry  sponsored  scientific  and  educational  activities,  promotional  activities  involving  the  internet,  and  direct-to-consumer 
advertising.  We  also  will  be  subject  to  a  variety  of  federal,  state  and  local  regulations  relating  to  the  use,  handling,  storage  and 
disposal  of  hazardous  materials,  including  chemicals  and  radioactive  and  biological  materials.  In  addition,  we  will  be  subject  to 
various laws and regulations governing laboratory practices and the experimental use of animals. In each of these areas, as above, the 
FDA has broad regulatory and enforcement powers, including the ability to levy fines and civil penalties, suspend or delay issuance of 
product approvals, seize or recall products, and deny or withdraw approvals. 

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We will also be subject to a variety of regulations governing clinical trials and sales of our products outside the U.S. Whether or 
not FDA approval has been obtained, approval of a product candidate by the comparable regulatory authorities of foreign countries 
and regions must be obtained prior to the commencement of marketing the product in those countries. The approval process varies 
from one regulatory authority to another and the time may be longer or shorter than that required for FDA approval. In the European 
Union, Canada and Australia, regulatory requirements and approval processes are similar, in principle, to those in the U.S. 

Employees 

As of March 12, 2010, we had 15 employees, six of whom were engaged in clinical development activities and nine of whom 

were involved in management and administrative operations. 

Available Information 

We maintain a website at www.cytrx.com and make available there, free of charge, our periodic reports filed with the Securities 
and Exchange Commission, or SEC, as soon as is reasonably practicable after filing. The public may read and copy any materials we 
file  with  the  SEC  at  the  SEC’s  Public  Reference  Room  at  100  F  Street,  NE,  Washington,  DC  20549.  The  public  may  obtain 
information on the operation of the Public Reference Room by calling the SEC at 1-800-SEC-0330. The SEC maintains a website at 
http:/www.sec.gov that contains reports, proxy and information statements, and other information regarding issuers such as us that file 
electronically with the SEC. We post on our website our Code of Business Conduct and Ethics. 

Item 1A. RISK FACTORS 

An investment in our shares involves a high degree of risk. Prior to making a decision about purchasing our shares, you should 
carefully  consider  the  risks  and  uncertainties  and  all  other  information  contained  in  this  Annual  Report,  including  the  risks  and 
uncertainties discussed below, as well as any modification, replacement or update to these risks and uncertainties that are reflected in 
any  subsequent  filings  we  make  with  the  SEC.  These  risks  and  uncertainties  are  not  the  only  ones  facing  us.  Additional  risks  and 
uncertainties not presently known to us, or that we currently perceive as immaterial, may also harm our business. If any of these risks 
or  uncertainties  actually  occurs,  our  business,  results  of  operations  and  financial  condition  could  be  materially  and  adversely 
affected. In that case, the trading price of our common stock could decline, and you could lose all or part of your investment. 

Risks Associated With Our Business 

We have operated at a loss and will likely continue to operate at a loss for the foreseeable future. 

We  have  operated  at  a  loss  due  to  our  ongoing  expenditures  for  research  and  development  of  our  product  candidates  and  for 
general and administrative purposes and lack of significant recurring revenue. We incurred net losses of $4.8 million, $27.0 million, 
and  $21.9  million  for  the  years  ended  December  31,  2009,  2008  and  2007,  respectively.  We  had  an  accumulated  deficit  as  of 
December  31,  2009  of  approximately  $197.4  million.  We  are  likely  to  continue  to  incur  losses  unless  and  until  we  are  able  to 
commercialize  one  or  more  of  our  product  candidates.  These  losses,  among  other  things,  have  had  and  will  continue  to  have  an 
adverse effect on our stockholders’ equity and working capital. Because of the numerous risks and uncertainties associated with our 
product development efforts, we are unable to predict when we may become profitable, if at all. If we do not become profitable or are 
unable to maintain future profitability, the market value of our common stock will be adversely affected. 

Because we have no source of significant recurring revenue, we must depend on financing to sustain our operations. 

Developing products and conducting clinical trials require substantial amounts of capital. To date, we have relied primarily upon 
proceeds from sales of our equity securities, including securities of RXi, and the exercise of options and warrants to generate funds 
needed to finance our business and operations. We will need to raise additional capital to, among other things: 

• 

• 

• 

fund our clinical trials and pursue regulatory approval of our existing and possible future product candidates; 

expand our research and development activities; 

finance our general and administrative expenses; 

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• 

• 

• 

acquire or license new technologies; 

prepare, file, prosecute, maintain, enforce and defend our patent and other proprietary rights; and 

develop and implement sales, marketing and distribution capabilities to successfully commercialize any product for which we 
obtain marketing approval and choose to market ourselves. 

Our revenues were $9.5 million, $6.3 million and $7.5 million, respectively, for years ended December 31, 2009, 2008 and 2007, 
which included $9.4 million, $6.2 million and $7.2 million, respectively, of deferred revenue recognized from our sale in August 2006 
of a one-percent royalty interest in worldwide sales of arimoclomol for the treatment of ALS to the privately-funded ALS Charitable 
Remainder Trust, or ALSCRT. Pursuant to an amendment signed between us and the beneficiary of the ALSCRT on August 6, 2009, 
we were released from all restrictions on the use of any proceeds previously paid to us in connection with the arrangement. As a result, 
we  recognized  $6.7  million  as  service  revenue  in  the  third  quarter  of  2009,  which  represented  the  remaining  deferred  revenue  and 
previously  un-recognized  portion  of  the  value  received.  We  will  have  no  significant  recurring  revenue  unless  we  are  able  to 
commercialize one or more of our product candidates in development, which may require us to first enter into license or other strategic 
arrangements with third parties. 

At December 31, 2009, we had cash and cash equivalents of approximately $9.9 million, marketable securities of $22.8 million, 
and held 5,768,881 shares of restricted common stock of RXi with a market value of $26.4 million based upon the closing price of the 
RXi  common  stock  on  that  date  as  reported  on  The  NASDAQ  Capital  Market.  On  July  27,  2009,  we  raised  approximately  $18.3 
million, net of fees and expenses, in a registered direct offering, and on September 23, 2009, we raised approximately $1.2 million, net 
of fees, from the sale of 500,000 of our shares of common stock of RXi. Management believes that our current cash on hand, together 
with our marketable securities and proceeds from possible future sales of our securities or our shares of RXi common stock, will be 
sufficient to fund our operations for the foreseeable future. The estimate is based, in part, upon our currently projected expenditures 
for  2010  of  approximately  $18.0  million,  which  includes  approximately  $3.2  million  for  our  clinical  programs  for  INNO-206, 
approximately  $1.6  million  for  our  clinical  programs  for  bafetinib,  approximately  $2.5  million  for  our  clinical  program  for 
tamibarotene, approximately $1.4 million for our activities for arimoclomol, approximately $2.2 million for general operation of our 
clinical  programs,  and  approximately  $7.1  million  for  other  general  and  administrative  expenses.  These  projected  expenditures  are 
based upon numerous assumptions and subject to many uncertainties, and our actual expenditures may be significantly different from 
these projections. 

If we obtain marketing approval as currently planned and successfully commercialize our product candidates, we anticipate it will 
take  a  minimum  of  three  years,  and  possibly  longer,  for  us  to  generate  significant  recurring  revenue,  and we  will  be  dependent  on 
future  financing  until  such  time,  if  ever,  as  we  can  generate  significant  recurring  revenue.  Our  ability  to  raise  capital  has  been 
materially  and  adversely  affected  by  the  continuing  poor  economy.  Despite  the  recover  in  the  U.S.  financial  markets  in  2009,  the 
market remains severely depressed for private investment in public equities, or PIPEs, transactions on which we have relied for raising 
needed capital. These conditions also may materially and adversely affect the market for our RXi shares. We have no commitments 
from third parties to provide us with any additional financing, and we may not be able to obtain future financing on favorable terms, or 
at  all.  Failure  to  obtain  adequate  financing  would  adversely  affect  our  ability  to  operate  as  a  going  concern.  If  we  raise  additional 
funds by issuing equity securities, dilution to stockholders may result and new investors could have rights superior to holders of the 
shares  issued  in  this  offering.  In  addition,  debt  financing,  if  available,  may  include  restrictive  covenants.  If  adequate  funds  are  not 
available to us, we may have to liquidate some or all of our assets or to delay or reduce the scope of or eliminate some portion or all of 
our development programs or clinical trials. We also may have to license to other companies our product candidates or technologies 
that we would prefer to develop and commercialize ourselves. 

If we do not achieve our projected development goals in the time frames we estimate, the commercialization of our products 

may be delayed and our business prospects may suffer. Our financial projections also may prove to be materially inaccurate. 

From  time  to  time,  we  estimate  the  timing  of  the  accomplishment  of  various  scientific,  clinical,  regulatory  and  other  product 
development goals, which we sometimes refer to as milestones. These milestones may include the commencement or completion of 
scientific studies and clinical trials and the submission of regulatory filings. For example, we have stated in our most recent Annual 
Report incorporated by reference in this Annual Report supplement the expected timing of certain milestones relating to our INNO-
206, bafetinib, tamibarotene and arimoclomol clinical development programs. 

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We  also  may  disclose  projected  expenditures  or  other  forecasts  for  future  periods  such  as  the  statements  above  in  this  Annual 
Report supplement regarding our current projected expenditures for fiscal year 2010. These and other financial projections are based 
on  management’s  current  expectations  and  do  not  contain  any  margin  of  error  or  cushion  for  any  specific  uncertainties,  or  for  the 
uncertainties inherent in all financial forecasting. 

The  actual  timing  of  milestones  and  actual  expenditures  or  other  financial  results  can  vary  dramatically  compared  to  our 
estimates, in some cases for reasons beyond our control. If we do not meet milestones or financial projections as announced from time 
to  time,  the  development  and  commercialization  of  our  products  may  be  delayed  and  our  business  prospects  may  suffer.  The 
assumptions management has used to produce these projections may significantly change or prove to be inaccurate. Accordingly, you 
should not unduly rely on any of these financial projections. 

If our products are not successfully developed and approved by the FDA, we may be forced to reduce or curtail our operations. 

All  of  our  product  candidates  in  development  must  be  approved  by  the  U.S.  Food  and  Drug  Administration,  or  FDA,  or 
corresponding foreign governmental agencies before they can be marketed. The process for obtaining FDA and foreign government 
approvals is both time-consuming and costly, with no certainty of a successful outcome. This process typically includes the conduct of 
extensive  pre-clinical  and  clinical  testing,  including  post-approval  testing,  which  may  take  longer  or  cost  more  than  we  or  our 
licensees, if any, anticipate, and may prove unsuccessful due to numerous factors. Product candidates that may appear to be promising 
at early stages of development may not successfully reach the market for a number of reasons. The results of preclinical and initial 
clinical testing of these product candidates may not necessarily be predictive of the results that will be obtained from later or more 
extensive  testing.  Companies  in  the  pharmaceutical  and  biotechnology  industries  have  suffered  significant  setbacks  in  advanced 
clinical trials, even after obtaining promising results in earlier trials. 

Numerous factors could affect the timing, cost or outcome of our product development efforts, including the following: 

• 

• 

• 

• 

• 

• 

• 

• 

difficulty in securing centers to conduct trials; 

difficulty in enrolling patients in conformity with required protocols or projected timelines; 

requirements for clinical trial design imposed by the FDA; 

unexpected adverse reactions by patients in trials; 

difficulty in obtaining clinical supplies of the product; 

changes  in  or  our  inability  to  comply  with  FDA  or  foreign  governmental  product  testing,  manufacturing  or  marketing 
requirements; 

regulatory  inspections  of  clinical  trials  or  manufacturing  facilities,  which  may,  among  other  things,  require  us  or  our 
manufacturers or licensees to undertake corrective action or suspend or terminate the affected clinical trials if investigators 
find them not to be in compliance with applicable regulatory requirements; 

inability to generate statistically significant data confirming the safety and efficacy of the product being tested; 

•  modification of the product during testing; and 

• 

reallocation of our limited financial and other resources to other clinical programs. 

It is possible that none of the product candidates we develop will obtain the regulatory approvals necessary for us to begin selling 
them. The time required to obtain FDA and foreign governmental approvals is unpredictable, but often can take years following the 
commencement  of  clinical  trials,  depending  upon  the  complexity  of  the  product  candidate.  Any  analysis  we  perform  on  data  from 
clinical activities is subject to confirmation and interpretation by regulatory authorities, which could delay, limit or prevent regulatory 
approval. 

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Furthermore, even if we obtain regulatory approvals, our products and the manufacturing facilities used to produce them will be 
subject to continual review, including periodic inspections and mandatory post- approval clinical trials by the FDA and other U.S. and 
foreign  regulatory  authorities.  Any  delay  or  failure  in  obtaining  required  approvals  or  to  comply  with  post-approval  regulatory 
requirements could have a material adverse effect on our ability to generate revenue from the particular product candidate. The failure 
to comply with any post-approval regulatory requirements also could also result in the rescission of the related regulatory approvals or 
the suspension of sales of the offending product. 

Our current and planned clinical trials of our product candidates may fail to show that these product candidates are clinically 

safe and effective, or that they are better than alternative treatments. 

INNO-206 was no more toxic than free doxorubicin in a Phase I clinical trial and showed limited biological responses against 
certain  tumors.  However,  these  conclusions  may  not  be  reproducible  in  larger  clinical  trials,  including  the planned Phase 2 clinical 
trials of INNO-206 as a treatment for pancreatic cancer, gastric cancer and soft tissue sarcomas. 

Bafetinib demonstrated clinical responses in patients with CML in a Phase I clinical trial conducted in patients with CML and 
other leukemias that have a certain mutation called the Philadelphia Chromosome (Ph+) and are intolerant of or resistant to Gleevec 
and, in some cases, second-line tyrosine kinase inhibitors. However, bafetinib has never been tested in human clinical trials in patients 
with B-CLL or glioblastoma multiforme, and there are no assurances that it will be effective in those indications. 

Tamibarotene has been shown to be safe, well tolerated, and efficacious in the Japanese population. However, it is possible that 
the response to the drug may be different in American or European populations. Furthermore, the efficacy studies that led to approval 
in Japan occurred prior to the advent of the use of arsenic trioxide, or ATO, for second line therapy. It is possible that the current use 
of ATO could alter the safety or efficacy of tamibarotene. The FDA might not accept the Japanese studies as a database for safety in 
the US. The majority of patients treated with ATRA as a first-line therapy way generally experience a complete remission of disease. 
As a result of the limited population of patients requiring third-line treatment for APL, there is no assurance that we will be successful 
in recruiting a sufficient number of patients into our ongoing clinical trial of tamibarotene as a third-line treatment for APL in order to 
demonstrate efficacy. In part for that reason, we have announced plans to develop tamibarotene, in combination with chemotherapy or 
arsenic trioxide (ATO), as a first-line treatment for APL. There is no assurance, however, that the FDA will accept a commercially 
reasonable  strategy  for  first-line  development  with  the  FDA,  and  any  FDA-required  changes  to  our  clinical  development  strategy 
could delay or increase the cost of the trial, adversely affect our ability to demonstrate the efficacy of tamibarotene in the trial or cause 
us not to pursue clinical development of tamibarotene for one or more of these considerations. 

Our  Phase  IIa  clinical  trial  and  open-label  extension  clinical  trial  of  arimoclomol  for  the  treatment  of  ALS  indicated  that 
arimoclomol  was  safe  and  well-tolerated  in  patients,  but  the  results  of  the  open-label  extension  clinical  trial  indicated  only  a  non-
statistically significant trend of improvement in the revised ALS Functional Rating Scale, or ALSFRS-R, in the arimoclomol high-
dose  group  as compared with  reports of previous  studies of untreated  patients.  This  trial  did not have  a  concurrent  placebo  control 
group, so we could draw no definitive conclusions with respect to efficacy. Further development of arimoclomal for ALS, as well as 
clinical  development  of  iroxanadine  for  diabetic  foot  ulcers,  would  require  significant  additional  testing,  and  it  is  possible  that  the 
favorable safety data we observed in earlier trials may not be reproduced in any later trials. 

In December 2009, the FDA accepted our revised protocol for an ascending dose clinical trial of arimoclomol for the treatment of 
ALS. Although we are making preparations related to that clinical trial, while simultaneously seeking potential strategic partners to 
advance development and evaluating the potential for a spin-off transaction for our molecular chaperone assets, it is possible that we 
will  further  amend  the  clinical  trial  protocol,  or  elect  not  to  proceed  with  further  development  of  some  or  all  of  our  molecular 
chaperone assets, as a result of future business or market conditions, capital constraints, an inability to secure a partnership or other 
factors.  The  planned  clinical  trial  includes  the  administration  of  arimoclomol  at  ascending  doses,  but  there  are  no  assurances  that 
arimoclomol will prove safe at higher doses. 

Later  trials  also  may  not  yield  statistically  significant  data  indicating  that  these  product  candidates  are  clinically  effective. 
Accordingly, we, or any development partners, may ultimately be unable to provide the FDA with satisfactory data on clinical safety 
and  efficacy  sufficient  to  obtain  FDA  approval  of  INNO-206,  tamibarotene,  bafetinib,  arimoclomol  or  iroxanadine  for  these 
indications. 

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We will rely upon third parties for the manufacture of our clinical product supplies. 

We  do  not  have  the  facilities  or  expertise  to  manufacture  supplies  of  any  of  our  product  candidates.  Accordingly,  we  are 
dependent  upon  third-party  manufacturers,  or  potential  future  strategic  alliance  partners,  to  manufacture  these  supplies.  We  have 
manufacturing  supply  arrangements  in  place  with  respect  to  a  portion  of  the  clinical  supplies  needed  for  the  clinical  development 
programs for INNO-206, tamibarotene and arimoclomol. However, we have no supply arrangements for the commercial manufacture 
of these product candidates or any manufacturing supply arrangements for any other potential product candidates, and we may not be 
able to secure needed supply arrangements on attractive terms, or at all. Our failure to secure these arrangements as needed could have 
a materially adverse effect on our ability to complete the development of our products or to commercialize them. 

If our product candidates cannot be manufactured in suitable quantities and in accordance with regulatory standards, our clinical 
trials,  regulatory  approvals  and  marketing  efforts  for  such  products  may  be  delayed.  Such  delays  could  adversely  affect  our 
competitive  position  and  our  chances  of  generating  significant  recurring  revenues.  If  our  products  cannot  be  manufactured  at  an 
acceptable cost, the commercial success of our products may be adversely affected. 

We may rely upon third parties in connection with the commercialization of our products. 

The completion of the development of INNO-206, bafetinib and tamibarotene, and our molecular chaperone product candidates, 
as well as the marketing of these products, may require us to enter into strategic alliances, license agreements or other collaborative 
arrangements with other pharmaceutical companies under which those companies will be responsible for one or more aspects of the 
commercial development and eventual marketing of our products. 

Our  products  may  not  have  sufficient  potential  commercial  value  to  enable  us  to  secure  strategic  arrangements  with  suitable 
companies  on  attractive  terms,  or  at  all.  If  we  are  unable  to  enter  into  such  arrangements,  we  may  not  have  the  financial  or  other 
resources to complete the development of any of our products and may have to sell our rights in them to a third party or abandon their 
development altogether. 

To  the  extent  we  enter  into  collaborative  arrangements,  we  will  be  dependent  upon  the  timeliness  and  effectiveness  of  the 
development and marketing efforts of our contractual partners. If these companies do not allocate sufficient personnel and resources to 
these  efforts  or  encounter  difficulties  in  complying  with  applicable  FDA  and  other  regulatory  requirements,  we  may  not  obtain 
regulatory  approvals  as  planned,  if  at  all,  and  the  timing  of  receipt  or  the  amount  of  revenue  from  these  arrangements  may  be 
materially and adversely affected. By entering into these arrangements rather than completing the development and then marketing 
these products on our own, the profitability to us of these products may decline. 

We may be unable to protect our intellectual property rights, which could adversely affect our ability to compete effectively. 

We believe that obtaining and maintaining patent and other intellectual property rights for our technologies and potential products 
is critical to establishing and maintaining the value of our assets and our business. We will be able to protect our technologies from 
unauthorized use by third parties only to the extent that we have rights to valid and enforceable patents or other proprietary rights that 
cover them. Although we own or have rights to patents and patent applications directed to INNO-206, bafetinib and our molecular 
chaperone  amplification  technologies,  these  patents  and  applications  may  not  prevent  third  parties  from  developing  or 
commercializing similar or identical technologies. In addition, our patents may be held to be invalid if challenged by third parties, and 
our patent applications may not result in the issuance of patents. 

The  patent  positions  of  pharmaceutical  and  biotechnology  companies  can  be  highly  uncertain  and  involve  complex  legal  and 
factual questions for which important legal principles remain unresolved. No consistent policy regarding the breadth of claims allowed 
in biotechnology patents has emerged to date in the U.S. and in many foreign countries. The application and enforcement of patent 
laws and regulations in foreign countries is even more uncertain. Accordingly, we may not be able to effectively file, protect or defend 
our proprietary rights on a consistent basis. Many of the patents and patent applications on which we rely were issued or filed by third 
parties prior to the time we acquired rights to them. The validity, enforceability and ownership of those patents and patent applications 
may  be  challenged,  and  if  a  court  decides  that  our  patents  are  not  valid,  we  will  not  have  the  right  to  stop  others  from  using  our 
inventions. There is also the risk that, even if the validity of our patents is upheld, a court may refuse to stop others on the ground that 
their activities do not infringe our patents. 

19 

  
  
  
  
  
  
  
  
  
 
 
Any litigation brought by us to protect our intellectual property rights could be costly and have a material adverse effect on our 
operating results or financial condition, make it more difficult for us to enter into strategic alliances with third parties to develop our 
products,  or  discourage  our  existing  licensees  from  continuing  their  development  work  on  our  potential  products.  If  our  patent 
coverage is insufficient to prevent third parties from developing or commercializing similar or identical technologies, the value of our 
assets is likely to be materially and adversely affected. 

We also rely on certain proprietary trade secrets and know-how, especially where we believe patent protection is not appropriate 
or  obtainable.  However,  trade  secrets  and  know-how  are  difficult  to  protect.  Although  we  have  taken  measures  to  protect  our 
unpatented trade secrets and know-how, including the use of confidentiality and invention assignment agreements with our employees, 
consultants  and  some  of  our  contractors,  it  is  possible  that  these  persons  may  disclose  our  trade  secrets  or  know-how  or  that  our 
competitors may independently develop or otherwise discover our trade secrets and know-how. 

If  our  product  candidates  infringe  the  rights  of  others,  we  could  be  subject  to  expensive  litigation  or  be  required  to  obtain 

licenses from others to develop or market them. 

Our competitors or others may have patent rights that they choose to assert against us or our licensees, suppliers, customers or 
potential  collaborators.  Moreover,  we  may  not  know  about  patents  or  patent  applications  that  our  products  would  infringe.  For 
example, because patent applications can take many years to issue, there may be currently pending applications, unknown to us, that 
may later result in issued patents that our arimoclomol, iroxanadine or other product candidates would infringe. In addition, if third 
parties file patent applications or obtain patents claiming technology also claimed by us in issued patents or pending applications, we 
may have to participate in interference proceedings in the US Patent and Trademark Office to determine priority of invention. If third 
parties file oppositions in foreign countries, we may also have to participate in opposition proceedings in foreign tribunals to defend 
the patentability of our foreign patent applications. 

If a third party claims that we infringe its proprietary rights, any of the following may occur: 

•  we may become involved in time-consuming and expensive litigation, even if the claim is without merit; 

•  we  may  become  liable  for  substantial  damages  for  past  infringement  if  a  court  decides  that  our  technology  infringes  a 

competitor’s patent; 

• 

a  court  may  prohibit  us  from  selling  or  licensing  our  product  without  a  license  from  the  patent  holder,  which  may  not  be 
available  on  commercially  acceptable  terms,  if  at  all,  or  which  may  require  us  to  pay  substantial  royalties  or  grant  cross 
licenses to our patents; and 

•  we may have to redesign our product candidates or technology so that it does not infringe patent rights of others, which may 

not be possible or commercially feasible. 

If any of these events occurs, our business and prospects will suffer and the market price of our common stock will likely decline 

substantially. 

Any  drugs  we  develop  may  become  subject  to  unfavorable  pricing  regulations,  third-party  reimbursement  practices  or 

healthcare reform initiatives, which could have a material adverse effect on our business. 

We  intend  to  sell  our products  primarily  to  hospitals  which  receive  reimbursement  for the  health  care  services  they provide  to 
their patients from third-party payors, such as Medicare, Medicaid and other domestic and international government programs, private 
insurance  plans  and  managed  care  programs.  Most  third-party  payors  may  deny  reimbursement  if  they  determine  that  a  medical 
product was not used in accordance with cost-effective treatment methods, as determined by the third-party payor, or was used for an 
unapproved  indication.  Third-party  payors  also  may  refuse  to  reimburse  for  experimental  procedures  and  devices.  Furthermore, 
because our programs are in the early stages of development, we are unable at this time to determine their cost-effectiveness and the 
level  or  method  of  reimbursement.  Increasingly,  the  third-party  payors  who  reimburse  patients  are  requiring  that  drug  companies 
provide them with predetermined discounts from list prices, and are challenging the prices charged for medical products. If the price 
we are able to charge for any products we develop is inadequate in light of our development and other costs, our profitability could be 
adversely affected. 

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We currently expect that any drugs we develop may need to be administered under the supervision of a physician. Under currently 

applicable law, drugs that are not usually self-administered may be eligible for coverage by the Medicare program if: 

• 

• 

• 

• 

they are “incidental” to a physician’s services, 

they are “reasonable and necessary” for the diagnosis or treatment of the illness or injury for which they are administered 
according to accepted standard of medical practice, 

they are not excluded as immunizations, and 

they have been approved by the FDA. 

We are subject to intense competition, and we may not compete successfully. 

We and our strategic partners or licensees may be unable to compete successfully against our current or future competitors. The 
pharmaceutical,  biopharmaceutical  and  biotechnology  industries  are  characterized  by  intense  competition  and  rapid  and  significant 
technological advancements. Many companies, research institutions and universities are working in a number of areas similar to our 
primary fields of interest to develop new products. There also is intense competition among companies seeking to acquire products 
that  already  are  being  marketed.  Many  of  the  companies  with  which  we  compete  have  or  are  likely  to  have  substantially  greater 
research  and  product  development  capabilities  and  financial,  technical,  scientific,  manufacturing,  marketing,  distribution  and  other 
resources than us and at least some of our present or future strategic partners or licensees. 

As a result, these competitors may: 

• 

• 

• 

• 

• 

• 

• 

succeed in developing competitive products sooner than us or our strategic partners or licensees; 

obtain FDA or foreign governmental approvals for their products before we can obtain approval of any of our products; 

obtain patents that block or otherwise inhibit the development and commercialization of our product candidate candidates; 

develop products that are safer or more effective than our products; 

devote greater resources than us to marketing or selling products; 

introduce or adapt more quickly than us to new technologies and other scientific advances; 

introduce products that render our products obsolete; 

•  withstand price competition more successfully than us or our strategic partners or licensees; 

• 

• 

negotiate third-party strategic alliances or licensing arrangements more effectively than us; and 

take better advantage than us of other opportunities. 

Companies that currently sell generic and proprietary compounds for the treatment of cancer and related diseases include, but are 
not limited to, Abraxis BioScience, Amgen, Sanofi-Aventis, Bayer, Bristol-Myers Squibb, Celgene, Cephalon, Genentech, Eli Lilly, 
Johnson  &  Johnson  and  Novartis.  Alternative  technologies  are  being  developed  to  treat  cancer  and  related  diseases  by  numerous 
companies including Bristol-Myers Squibb, Eisai, Merck and Genentech, several of which are in advanced clinical trials. There also 
are  FDA  approved  cancer  therapies  that  are  in  the  late  stage  of  development  by  larger  established  companies  for  new  cancer 
indications: Alimta (Eli Lilly), Avastin (Genentech), Eloxatin (Sanofi-Aventis), Erbitux (Bristol-Myers Squibb and Imclone Systems) 
and Tarceva (Genentech). 

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Soft tissue sarcoma patients are typically treated with surgery followed by radiation therapy. Doxorubicin is the only approved 
drug for treating soft tissue sarcoma and is often used in combination with radiation. The National Comprehensive Cancer Network 
also  includes  the  use  of  ifosfamide,  epirubicin,  Eli  Lilly’s  Gemzar,  dacarbazine  and  liposomal  doxorubicin  marketed  in  the  US  as 
Doxil by Johnson & Johnson. For patients ineligible for surgery, radiation and/or chemotherapy is the only option. Other approaches 
to  treating  soft  tissue  sarcoma  are  in  late  stage  clinical  development.  These  include  ridaforolimus  being  developed  by  Ariad 
Pharmaceuticals and Merck & Co., GlaxoSmithKline’s pazopanib, Sanofi-Aventis’ AVE8062, Threshhold Pharmaceuticals’s TH-302, 
and trabectedin being co-developed by Johnson and Johnson and PharmaMar. 

Advanced  gastric  cancer  patients  are  typically  treated  with  a  variety  of  combination  of  approved  drugs  such  as  cisplatin, 
docetaxel,  5-FU,  oxaliplatin,  iriniotecan  and  paclitaxel.  Epirubicin,  an  anthracycline,  is  part  of  several  gastric  cancer  treatment 
regimens. We believe INNO-206 could be a potentially more effective anthracycline and potentially more effective in this setting. 

Pancreatic  cancer  patients  are  typically  treated  with  surgery,  radiation  and  chemotherapy.  Eli  Lilly’s  Gemzar  is  currently 
approved for the first line treatment of locally advanced or metastatic pancreatic cancer. It is also indicated for the use in patients who 
have  received  prior  treatment  with  5-FU.  OSI  Pharmaceuticals’  Tarceva  was  approved  in  2005  for  the  use  in  combination  with 
Gemzar. The NCCN believes the best management for these patients is in a clinical trial. Because of the tremendous unmet need for 
these  patients,  many  companies  are  developing  new  drugs  to  treat  pancreatic  cancer.  Late  stage  drugs  in  clinical  trials  include 
Abraxane by Abraxis BioScience, AGS-1C4D4 by Astellas Pharma Inc., TNFerade™ by GenVec, and S-1 by Sanofi-Aventis. 

To our knowledge, there are no competitors in clinical development for refractory APL. Currently, treatment of APL is based on 
induction  and  maintenance  therapy  with  ATRA  and  chemotherapy  (typically  idarubicin).  ATRA  and  idarubicin  are  both  generic 
compounds. Arsenic trioxide, currently marketed by Cephalon, is approved for use in patients who have relapsed after ATRA-based 
therapy in APL. There are no FDA-approved therapies for patients who have failed arsenic trioxide. In practice, it appears that patients 
who fail arsenic trioxide are retreated with ATRA or receive Mylotarg, which is marketed by Pfizer Inc. 

There are currently three marketed competitors to bafetinib (formerly INNO-406) in the CML market, Gleevec®, Sprycel® and 
Tasigna®.  Gleevec  is  approved  for  treatment  of  newly  diagnosed  adult  patients  with  Philadelphia  chromosome–positive  chronic 
myeloid leukemia (Ph+ CML) in the chronic phase and patients with Ph+ CML in blast crisis (BC), accelerated phase (AP), or in the 
chronic  phase  (CP)  after  failure  of  interferon-alpha  therapy.  Sprycel®  and  Tasigna®  are  approved  for  Gleevec-resistant  CML. 
Because  of  the  highly  competitive  nature  of  the  CML  market  including  drug  candidates  in  development,  CytRx  plans  to  develop 
bafetinib  initially  in  cancers  other  than  CML.  We  have  selected  B-cell  chronic  lymphocytic  leukemia  (B-CLL)  and  glioblastoma 
multiforme  due  to  the  potent  and  specific  inhibitory  properties  of  bafetinib  against  Lyn  kinase.  Lyn kinase  is  a  member  of  the Src 
family  of  kinases  which  are  known  to  be  involved  in  cell  growth.  Lyn  kinase  is  overexpressed  in  both  B-CLL  and  glioblastoma 
multiforme (GBM). 

There are several drugs approved for the treatment of CLL. First-line therapy for CLL includes a variety of combination therapies 
including  fludarabine,  cyclophosphamide,  Rituxan®  and  Campath®.  Treatment  for  relapsed  or  refractory  CLL  includes  several 
chemotherapy regimens including CHOP, CFAR, hyperCFAD and OFAR in addition to single agents including GlaxoSmithKline’s 
ArzerraTM. Arzerra was approved in October 2009 for CLL patients who are refractory to treatment with fludarabine and Campath. 

Current therapy for glioblastoma  multiforme, the most common form of brain cancer, is surgery followed by radiation therapy 
and chemotherapy. Merck’s Temodar® is approved for treating newly diagnosed GBM concomitantly with radiotherapy and then as a 
maintenance  treatment.  Roche’s  Avastin  was  approved  in  May  2009  for  treatment  of  recurrent  GBM.  We  believe  that  bafetinib’s 
ability  to  selectively  inhibit  Lyn  kinase  and  to  penetrate  the  brain  in  an  animal  model  of  cancer  will  be  an  effective  treatment  for 
second-line therapy in GBM. 

We are aware of only one drug, rilutek, developed by Aventis Pharma AG, that has been approved by the FDA for the treatment 
of ALS. Many companies are working to develop pharmaceuticals to treat ALS, including Aeolus Pharmaceuticals, Mitsubishi Tanabe 
Pharma  Corporation, Ono Pharmaceuticals,  Trophos  SA, Knopp  Neurosciences Inc., Faust  Pharmaceuticals  SA, Oxford  BioMedica 
plc, Phytopharm plc and Teva Pharmaceutical Industries Ltd., as well as RXi. ALS patients often take over-the-counter supplements, 
including vitamin E, creatine and coenzyme Q10, or drugs such as lithium that are approved for other indications. ALS belongs to a 
family of neurodegenerative diseases that includes Alzheimer’s, Parkinson’s and Huntington’s diseases. Due to similarities between 
these  diseases,  a  new  treatment  for  one  such  disease  potentially  could  be  useful  for  treating  others.  There  are  many  companies 
producing  and  developing  drugs  used  to  treat  neurodegenerative  diseases  other  than  ALS,  including  Amgen,  Inc.,  Biogen  Idec, 
Boehringer  Ingelheim,  Cephalon,  Inc.,  Ceregene,  Inc.,  Elan  Pharmaceuticals,  plc,  Forest  Laboratories,  Inc.,  H.  Lundbeck  A/S, 
Phytopharm plc, UCB Group and Wyeth. 

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Any of these competing therapies could prove to be more effective than INNO-206, bafetinib, tamibarotene, or any future therapy 
of  ours.  Most  of  our  competitors  have  substantially  greater  research  and  product  development  capabilities  and  financial,  technical, 
scientific, manufacturing, marketing, distribution and other resources than us. 

We will be required to pay substantial milestone and other payments relating to the commercialization of our products. 

The  agreement  relating  to  our  worldwide  rights  to  INNO-206  provides  for  our  payment  of  an  aggregate  of  $7.5  million  upon 
meeting specified clinical and regulatory milestones up to and including the product’s second final marketing approval. We also will 
be obliged to pay: 

• 

• 

commercially reasonable royalties based on a percentage of net sales (as defined in the agreement); 

a percentage of non-royalty sub-licensing income (as defined in the agreement); and 

•  milestones of $1,000,000 for each additional final marketing approval that we might obtain. 

Our agreement relating to our worldwide (except Japan) rights to bafetinib provides for our payment of an aggregate of $13.35 
million  (including  $5  million  upon  the  product’s  initial  final  marketing  approval)  upon  the  achievement  of  specified  clinical  and 
regulatory milestones up to and including approvals in the U.S. and Europe. We also will be obliged to pay: 

• 

• 

• 

commercially reasonable royalties based on a percentage of net sales (as defined in the agreement), dependent on reaching 
certain revenue thresholds; 

annual minimum payments if sales of bafetinib do not meet specified levels; and 

a percentage of non-royalty sub-licensing income (as defined in the agreement). 

The agreement under which we have North American rights to tamibarotene provides for our payment of royalties based on net 
sales of any products, as well as aggregate payments of $4.4 million upon meeting specified clinical, regulatory and sales milestones 
up to and including the first commercial sale of tamibarotene for the treatment of APL. 

If we are required to pay any third party in order to exercise our rights under the agreement, we will deduct a percentage of those 

payments from the royalties due under the agreement, up to an agreed-upon cap. 

Under the merger agreement by which we acquired Innovive, we agreed to pay the former Innovive stockholders a total of up to 
approximately  $18.3  million  of  future  earnout  merger  consideration,  subject  to  our  achievement  of  specified  net  sales  under  the 
Innovive  license  agreements.  The  earnout  merger  consideration,  if  any,  will  be  payable  in  shares  of  our  common  stock,  subject  to 
specified conditions, or, at our election, in cash or by a combination of shares of our common stock and cash. Our common stock will 
be valued for purposes of any future earnout merger consideration based upon the trading price of our common stock at the time the 
earnout merger consideration is paid. 

Our  agreement  by  which  we  acquired  rights  to  arimoclomol  and our  other  molecular  chaperone  amplification  product  candidates 
provides for milestone payments by us upon the occurrence of specified regulatory filings and approvals related to the acquired products. 
In  the  event  that  we  successfully  develop  arimoclomol  or  any  of  these  other  product  candidates,  these  milestone  payments  could 
aggregate as much as $3.7 million, with the most significant payments due upon the first commercialization of any of these products. In 
addition, our agreement with the ALS CRT requires us to pay a one-percent royalty interest on worldwide sales of arimoclomol for the 
treatment of ALS. Also, any future license, collaborative or other agreements we may enter into in connection with our development and 
commercialization activities may require us to pay significant milestone, license and other payments in the future. 

We are subject to potential liabilities from clinical testing and future product liability claims. 

If any of our products are alleged to be defective, they may expose us to claims for personal injury by patients in clinical trials of 
our  products  or,  if  we  obtain  marketing  approval  and  commercialize  our  products,  by  patients  using  our  commercially  marketed 
products. Even if the if one or more of our products is approved by the FDA, users may claim that such products caused unintended 
adverse  effects.  We  maintain  clinical  trial  insurance  for  our  clinical  trial  of  tamibarotene  for  APL,  and  we  plan  to  seek  to  obtain 
similar insurance for any other clinical trials that we conduct. We also would seek to obtain product liability insurance covering the 
commercial  marketing  of  our  product  candidates.  We  may  not  be  able  to  obtain  additional  insurance,  however,  and  any  insurance 
obtained by us may prove inadequate in the event of a claim against us. Any claims asserted against us also may divert management’s 
attention from our operations, and we may have to incur substantial costs to defend such claims even if they are unsuccessful.

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We  may  be  unable  to  successfully  acquire  additional  technologies  or  products.  If  we  require  additional  technologies  or 
products, our product development plans may change and the ownership interests of our shareholders, or our ownership interest in 
RXi, could be diluted. 

We may seek to acquire additional technologies by licensing or purchasing such technologies, or through a merger or acquisition 
of one or more companies that own such technologies. We have no current understanding or agreement to acquire any technologies, 
however,  and  we  may  not  be  able  to  identify  or  successfully  acquire  any  additional  technologies.  We  also  may  seek  to  acquire 
products  from  third  parties  that  already  are  being  marketed  or  have  been  approved  for  marketing,  although  we  have  not  currently 
identified any of these products. We do not have any prior experience in acquiring or marketing products approved for marketing and 
may need to find third parties to market any products that we might acquire. 

Following our acquisition of Innovive in September 2008, we refocused our product development efforts on our oncology drug 
candidates, which we believe has the greatest near-term revenue potential. If we acquire additional technologies or product candidates, 
we  may  determine  to  make  further  changes  to  our  product  development  plans  and  business  strategy  to  capitalize  on  opportunities 
presented by the new technologies and product candidates. 

We may determine to issue shares of our common stock, or to use shares of RXi common stock owned by us, or both, to acquire 
additional technologies or products or in connection with a  merger or acquisition of another company. To the extent we do so, the 
ownership interest of our stockholders, or our ownership interest in RXi, or both, will be diluted accordingly. 

Risks Associated With Our Investment in RXi 

We may sell or dispose of some of our RXi shares, and may not be able to do so on attractive terms. 

As of December 31, 2009, we held 5,768,881 shares of common stock of RXi, or approximately 36% of the outstanding shares of 
RXi  common stock.  RXi  shares  are  listed on  The NASDAQ  Capital  Market under  the  symbol  “RXi.”  During  the 12-month period 
ended December 31, 2009, the market prices for RXi shares as reported on The NASDAQ Capital Market fluctuated from a high of 
$7.57  per  share  to  a  low  of  $1.51  per  share,  and  the  market  price  of  RXi  shares  and  the  value  of  our  RXi  shares  may  continue  to 
experience significant volatility. 

We intend to look for favorable opportunities to sell or otherwise dispose of our RXi shares in one or more transactions in order to 
obtain funds to carry on our operations or in connection with our acquisition of new technologies or products. There is no assurance, 
however, whether, or on what terms, we might be able to sell or dispose of our RXi shares. In addition, any sales or other disposition 
of  RXi  shares  by  us,  or  the  possibility  of  such  sales  or  disposition,  could  adversely  affect  the  market  price  of  our  remaining  RXi 
shares. 

If RXi undertakes future financings, our ownership interest in RXi may be diluted. 

Under our agreement with RXi, with some exceptions, we will have preemptive rights to acquire a portion of any new securities 
sold or issued by RXi so as to maintain our percentage ownership of RXi. Depending upon the terms and provisions of any proposed 
sale of new securities by RXi, our financial condition and other factors, we may be unwilling or unable to exercise our preemptive 
rights. We agreed to waive our preemptive rights in connection with a private placement by RXi in June 2008, which resulted in a 
reduction in our percentage ownership of RXi from approximately 49% to approximately 45%. In September, 2009, we sold 500,000 
shares of RXi which reduced our percentage ownership further to approximately 36%. If RXi undertakes future issuances of equity 
securities, our percentage ownership interest in RXi may be diluted further. 

24 

  
  
  
  
  
  
  
  
  
 
 
We do not control RXi, and the officers, directors and other RXi stockholders may have interests that are different from ours. 

Although  we  currently  own  a  significant  portion  of  RXi’s  outstanding  common  stock,  we  do  not  control  its  management  or 
operations.  RXi  has  its  own  board  of  directors  and  management,  who  are  responsible  for  the  affairs  and  policies  of  RXi  and  its 
development plans. We have entered into letter agreements with RXi and certain of its stockholders under which we agree to vote our 
shares of RXi common stock for the election of directors of RXi and to take other actions to ensure that a majority of RXi’s board of 
directors are independent of us. The board of directors and other stockholders of RXi may have interests that are different from ours, 
and RXi may engage in actions in connection with its business and operations that we believe are not in our best interests. 

Risks Associated with Our Common Stock 

Our anti-takeover measures may make it more difficult to change our management, or may discourage others from acquiring 

us, and thereby adversely affect stockholder value. 

We  have  a  stockholder  rights  plan  and  provisions  in  our  bylaws  that  are  intended  to  protect  our  stockholders’  interests  by 
encouraging  anyone  seeking  control  of  our  company  to  negotiate  with  our  board  of  directors.  These  provisions  may  discourage  or 
prevent a person or group from acquiring us without the approval of our board of directors, even if the acquisition would be beneficial 
to our stockholders. 

We have a classified board of directors, which means that at least two stockholder meetings, instead of one, will be required to 
effect  a  change  in  the  majority  control  of  our  board  of  directors.  This  applies  to  every  election  of  directors,  not  just  an  election 
occurring after a change in control. The classification of our board increases the amount of time it takes to change majority control of 
our  board  of  directors  and  may  cause  potential  acquirers  to  lose  interest  in  a  potential  purchase  of  us,  regardless  of  whether  our 
purchase would be beneficial to us or our stockholders. The additional time and cost to change a majority of the members of our board 
of directors makes it more difficult and may discourage our existing stockholders from seeking to change our existing management in 
order to change the strategic direction or operational performance of our company. 

Our bylaws provide that directors may only be removed for cause by the affirmative vote of the holders of at least a majority of 
the outstanding shares of our capital stock then entitled to vote at an election of directors. This provision prevents stockholders from 
removing any incumbent director without cause. Our bylaws also provide that a stockholder must give us at least 120 days notice of a 
proposal  or  director  nomination  that  such  stockholder  desires  to  present  at  any  annual  meeting  or  special  meeting  of  stockholders. 
Such  provision  prevents  a  stockholder  from  making  a  proposal  or  director  nomination  at  a  stockholder  meeting  without  us  having 
advance notice of that proposal or director nomination. This could make a change in control more difficult by providing our directors 
with  more  time  to  prepare  an  opposition  to  a  proposed  change  in  control.  By  making  it  more  difficult  to  remove  or  install  new 
directors,  these  bylaw  provisions  may  also  make  our  existing  management  less  responsive  to  the  views  of  our  stockholders  with 
respect to our operations and other issues such as management selection and management compensation. 

We are subject to the anti-takeover provisions of Section 203 of the Delaware General Corporation Law, which may also prevent 

or delay a takeover of us that may be beneficial to you. 

Our  outstanding  options  and  warrants  and  the  availability  for  resale  of  our  shares  issued  in  our  private  financings  may 

adversely affect the trading price of our common stock. 

As of December 31, 2009, there were outstanding stock options and warrants to purchase approximately 24.4 million shares of 
our  common  stock  at  a  weighted-average  exercise  price  of  $1.42  per  share.  Our  outstanding  options  and  warrants  could  adversely 
affect  our  ability  to  obtain  future  financing  or  engage  in  certain  mergers  or  other  transactions,  since  the  holders  of  options  and 
warrants  can  be  expected  to  exercise  them  at  a  time  when  we  may  be  able  to  obtain  additional  capital  through  a  new  offering  of 
securities on terms more favorable to us than the terms of outstanding options and warrants. For the life of the options and warrants, 
the holders have the opportunity to profit from a rise in the market price of our common stock without assuming the risk of ownership. 
The issuance of shares upon the exercise of outstanding options and warrants will also dilute the ownership interests of our existing 
stockholders. Many of our outstanding warrants contain anti-dilution provisions pertaining to dividends with respect to our common 
stock. In the event that these anti-dilution provisions are triggered by us in the future, we would likewise be required to reduce the 
exercise price, and increase the number of shares underlying, those warrants, which would have a dilutive effect on our stockholders. 

25 

  
  
  
  
  
  
  
  
  
 
 
We have registered with the SEC the resale by the holders of all or substantially all shares of our common stock issuable upon 
exercise of our outstanding options and warrants. The availability of these shares for public resale, as well as actual resales of these 
shares, could adversely affect the trading price of our common stock. 

We may issue preferred stock in the future, and the terms of the preferred stock may reduce the value of our common stock. 

We are authorized to issue shares of preferred stock in one or more series. Our board of directors may determine the terms of 
future preferred stock offerings without further action by our stockholders. If we issue preferred stock, it could affect your rights or 
reduce  the  value  of  our  outstanding  common  stock.  In  particular,  specific  rights  granted  to  future  holders  of  preferred  stock  may 
include  voting  rights,  preferences  as  to  dividends  and  liquidation,  conversion  and  redemption  rights,  sinking  fund  provisions,  and 
restrictions on our ability to merge with or sell our assets to a third party. 

We may experience volatility in our stock price, which may adversely affect the trading price of our common stock. 

The market price of our common stock has ranged from $0.23 to $2.98 per share since January 1, 2008, and it may continue to 
experience  significant  volatility  from  time  to  time.  Our  ability  to  raise  capital  has  been  materially  and  adversely  affected  by  the 
continuing  poor  economy.  Despite  the  recovery  in  the  U.S.  financial  markets  in  2009,  the  market  remains  depressed  for  private 
investment in public equity, or PIPEs, transactions on which we have relied for raising needed capital. 

Other factors that may affect the market price of our common stock include the following: 

• 

• 

• 

• 

• 

• 

• 

• 

• 

• 

announcements of regulatory developments or technological innovations by us or our competitors; 

changes in our relationship with our licensors and other strategic partners; 

changes in our ownership of or other relationships with RXi; 

our quarterly operating results; 

litigation involving or affecting us; 

shortfalls in our actual financial results compared to our guidance or the forecasts of stock market analysts; 

developments in patent or other technology ownership rights; 

acquisitions or strategic alliances by us or our competitors; 

public concern regarding the safety of our products; and 

government regulation of drug pricing. 

We do not expect to pay any cash dividends on our common stock. 

We have not declared or paid any cash dividends on our common stock or other securities, and we currently do not anticipate 
paying any cash dividends in the foreseeable future. Because we do not anticipate paying cash dividends for the foreseeable future, our 
stockholders will not realize a return on their investment in our common stock except to the extent of any appreciation in the value of 
our common stock. Our common stock may not appreciate in value, or may decline in value. 

26 

  
  
  
  
  
  
  
  
  
  
  
  
  
  
  
  
  
 
 
Item 2. PROPERTIES 

We  lease  our  headquarters  in  Los  Angeles,  California.  The  lease  covers  approximately  5,700  square  feet  of  office  space  and 
expires in March 2015. This lease requires us to make monthly payments of approximately $23,243, subject to annual increases. We 
also lease approximately 10,000 square feet of office and laboratory space in San Diego, California, for $35,270 per month. The lease 
expires  in  October  2010.  In  May  2009,  we  substantially  completed  the  initial  phase  of  the  research  and  development  activities 
performed at the San Diego facility, and in November 2009, we signed sublease agreements with two parties to sublet the facility for 
the remainder of the term of the lease. Under those subleases, we are entitled to aggregate annual rent of approximately $16,900 per 
month. 

We also acquired a sublease to approximately 5,526 square feet of office space at 555 Madison Avenue, New York, New York, in 
connection  with  our  acquisition  of  Innovive  in  September  2008.  This  lease  currently  requires  us  to  make  annual  payments  of 
approximately $210,000, plus certain taxes and operating expenses, and it expires on August 30, 2012. On December 4, 2008, we sub-
subleased the space through August 29, 2012. Under the sub-sublease, we are entitled to base annual rent of approximately $350,000, 
plus certain taxes and operating expenses.  

Item 3. LEGAL PROCEEDINGS 

We are occasionally involved in claims arising in the normal course of business. As of March 12, 2010, there were no such claims 

that we expect, individually or in the aggregate, to have a material adverse affect on us. 

27 

  
  
  
  
 
 
PART II 

Item  5.  MARKET  FOR  REGISTRANT’S  COMMON  EQUITY,  RELATED  STOCKHOLDER  MATTERS  AND  ISSUER 
PURCHASES OF EQUITY SECURITIES 

Market Information 

Our common stock is traded on The NASDAQ Capital Market under the symbol “CYTR.” The following table sets forth the high 

and low sale prices for our common stock for the periods indicated as reported by The NASDAQ Capital Market: 

Fiscal Year 2009: 

Fourth Quarter . . . . . . . . . . . . . . . . . . . . . . . . .
Third Quarter . . . . . . . . . . . . . . . . . . . . . . . . . .
Second Quarter . . . . . . . . . . . . . . . . . . . . . . . .
First Quarter . . . . . . . . . . . . . . . . . . . . . . . . . . .

Fiscal Year 2008: 

Fourth Quarter . . . . . . . . . . . . . . . . . . . . . . . . .
Third Quarter . . . . . . . . . . . . . . . . . . . . . . . . . .
Second Quarter . . . . . . . . . . . . . . . . . . . . . . . .
First Quarter . . . . . . . . . . . . . . . . . . . . . . . . . . .

High

Low

$ 1.29 
$ 1.72 
$ 1.09 
$ 0.45 

$ 0.71 
$ 0.84 
$ 0.34 
$ 0.24 

$ 0.65 
$ 0.68 
$ 1.27 
$ 2.98 

$ 0.23 
$ 0.40 
$ 0.61 
$ 1.00 

Holders 

On March 12, 2010, there were approximately 750 holders of record of our common stock. The number of record holders does 

not reflect the number of beneficial owners of our common stock for whom shares are held by brokerage firms and other nominees. 

Dividends 

We have not paid any cash dividends since our inception and do not contemplate paying any cash dividends in the foreseeable 
future. On March 11, 2008, we distributed to holders of our common stock approximately 36% of the outstanding shares of RXi on an 
approximate 1-for-20 basis. 

Equity Compensation Plans 

The following table sets forth certain information as of December 31, 2009, regarding securities authorized for issuance under our 

equity compensation plans: 

 Plan Category  
Equity compensation plans approved by our security holders:      
2000 Long-Term Incentive Plan . . . . . . . . . . . . . . . . . . . . . . . . .    
2008 Stock Incentive Plan . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Equity compensation plans not approved by our security holders: 
Outstanding warrants (1) . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Total . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
____________ 

(a)
Number of Securities 
to be Issued Upon 
Exercise of Outstanding 
Options, Warrants and 
Rights

(b)
Weighted-Average 
Exercise Price of 
Outstanding 
Options, Warrants 
and Rights 

Number of Securities 
Remaining Available for 
Issuance Under Equity 
Compensation Plans 
(Excluding Securities 
Reflected in Column (a))

7,907,090    $
1,100,000     

15,418,178     
24,425,268    $

1.17      
0.83      

1.57      
1.58      

155,000 
8,900,000 

— 
9,055,000 

(1)  The warrants shown were issued in discreet transactions from time to time as compensation for services rendered by consultants, 
advisors  or  other  third  parties,  and  do  not  include  warrants  sold  in  private  placement  transactions.  The  material  terms  of  such 
warrants  were  determined  based  upon  arm’s-length  negotiations  with  the  service  providers.  The  warrant  exercise  prices 
approximated the market price of our common stock at or about the date of grant, and the warrant terms range from one to ten 
years from the grant date. The warrants contain customary anti-dilution adjustments in the event of a stock split, reverse stock 
split, reclassification or combination of our outstanding common stock and similar events and certain of the warrants contain anti-
dilution adjustments triggered by other corporate events, such as dividends and sales of equity below market price.

28 

  
  
  
  
  
  
  
  
  
  
  
  
  
 
   
    
 
      
      
 
     
      
 
 
Comparison of Cumulative Total Returns 

The following line graph presentation compares cumulative total stockholder returns of CytRx with The NASDAQ Stock Market 
Index and the NASDAQ Pharmaceutical Index (the “Peer Index”) for the five-year period from December 31, 2004 to December 31, 
2009. The graph and table assume that $100 was invested in each of CytRx’s common stock, the NASDAQ Stock Market Index and 
the Peer Index on December 31, 2004, and that all dividends were reinvested. This data was furnished by Zacks Investment Research. 

Comparison of Cumulative Total Returns 

CytRx Corporation . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .
NASDAQ Stock Market Index . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .
NASDAQ Pharmaceutical Index . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .

Recent Issuances of Unregistered Securities 

2005
73.57 
102.12 
110.13 

December 31, 
2007 
202.84 
124.73 
113.36 

2006 
136.42 
112.73 
107.79 

2008
31.11 
74.87 
105.46 

2009
116.16 
108.83 
118.52 

During  the  three-month  period  ended  December  31,  2009,  we  issued  50,000  shares  of  our  common  stock,  and  warrants  to 
purchase a total of 800,000 shares of our common stock at exercise prices ranging from $1.10 to $4.00 per share, in connection with a 
consulting arrangement. The issuance of stock and warrants was exempt from registration under the Securities Act of 1933 pursuant to 
Section 4(2) of the Securities Act of 1933 and Regulation D under the Act. 

Repurchase of Shares 

We did not repurchase any of our shares during the three-month period ended December 31, 2009. 

29 

  
  
 
 
 
 
 
 
  
  
  
 
 
Item 6. SELECTED FINANCIAL DATA 

General 

The following selected financial data are derived from our audited financial statements. Our financial statements for 2009, 2008 
and 2007 have been audited by BDO Seidman, LLP, our independent registered public accounting firm. These historical results do not 
necessarily  indicate  future  results.  When  you  read  this  data,  it  is  important  that  you  also  read  our  financial  statements  and  related 
notes, as well as the “Management’s Discussion and Analysis of Financial Condition and Results of Operations” and “Risk Factors” 
sections of this Annual Report. Financial information provided below has been rounded to the nearest thousand. 

2009

2008

2007

2006 

2005

Statement of Operations Data: 
Revenues 

Service revenue . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   $ 9,400,000    $ 6,166,000    $ 7,242,000    $  1,859,000    $
Licensing revenue . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
101,000     
Grant revenue . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
106,000     
Total revenues . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   $ 9,500,000    $ 6,266,000    $ 7,459,000    $  2,066,000    $

101,000      
116,000      

100,000     
—     

100,000     
—     

83,000 
101,000 
— 
184,000 

Deemed dividend for anti-dilution adjustments made 

to outstanding common stock warrants . . . . . . . . . . .    

(1,076,000)
Net loss applicable to common stockholders . . . . . . . .   $ (4,800,000)   $(27,803,000)   $(21,890,000)   $ (17,240,000)   $(16,169,000)
Basic and diluted loss per share applicable to 

(488,000)    

(757,000)    

—      

—     

common stock . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   $

(0.05)   $

(0.30)   $

(0.26)   $ 

(0.25)   $

(0.28)

Balance Sheet Data: 
Cash, cash equivalents and marketable securities . . . .   $ 9,894,000    $ 25,042,000    $ 60,450,000    $  30,381,000    $ 8,299,000 
Total assets . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   $ 35,277,000    $ 28,324,000    $ 64,146,000    $  31,636,000    $ 9,939,000 
Total stockholders’ equity . . . . . . . . . . . . . . . . . . . . . . . . .   $ 28,348,000    $ 15,698,000    $ 40,224,000    $  5,150,000    $ 7,208,000 

Factors Affecting Comparability 

On September 19, 2008, we purchased all of the common stock of Innovive Pharmaceuticals in a transaction that for accounting 
purposes is considered an asset acquisition. The fair value of Innovive’s assets and liabilities at September 19, 2008, in millions of 
dollars, are presented below: 

In-process research and development. . . . . . . . . . . . .   $
Leasehold interests . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Prepaid expenses . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Accounts payable . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Net assets acquired through issuance of common 

stock . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   $

8.0  
.1  
.3  
(6.1) 

2.3  

As a result of the March 11, 2008 distribution by us to our stockholders of approximately 36% of the outstanding shares of RXi, 
we deconsolidated that previously majority-owned subsidiary. As part of the transaction, we deconsolidated $3.7 million of total assets 
and $4.6 million of total liabilities of RXi. 

In connection with applicable antidilution adjustments to the price of certain outstanding warrants in March 2008, we recorded a 
deemed  dividend  of  approximately  $757,000.  The  deemed  dividend  was  recorded  as  a  charge  to  accumulated  deficit  and  a 
corresponding credit to additional paid-in capital. 

In July 2009, we completed a $20.0 million registered direct public offering of approximately 15.3 million shares of our common 
stock at a price of $1.31 per share and warrants to purchase an additional approximately 4.7 million shares of common stock at an 
exercise price of $1.70 per share. Net of investment banking commissions, advisory fees, legal, accounting and other fees related to 
the transaction, we received proceeds of approximately $18.3 million (without giving effect to any proceeds that we may receive upon 
future exercises of the warrants sold in the offering). 

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In April 2007, we completed a $37.0 million private equity financing in which we issued 8.6 million shares of our common stock 
at  $4.30  per  share.  Net  of  investment  banking  commissions,  legal,  accounting  and  other  expenses  related  to  the  transaction,  we 
received approximately $34.2 million of proceeds. 

In  August  2006,  we  received  approximately  $24.5  million  in  marketable  securities  (which  were  sold  by  us  for  approximately 
$24.3 million) from the privately-funded ALS Charitable Remainder Trust, or ALSCRT, in exchange for our commitment to continue 
research and development of arimoclomol and other potential treatments for ALS and a one percent royalty from worldwide sales of 
arimoclomol.  We  recorded  the  value  received  under  the  arrangement  as  deferred  service  revenue,  which.  we  recognize  using  the 
proportional performance method of revenue recognition. In August 2009, we were released from all restrictions on the use of any As 
a  result,  we recognized  in  the  third quarter  $6.7  million  of  service  revenue,  representing  all  of  the  remaining  deferred  revenue  and 
previously  un-recognized  portion  of  the  value  received  in  the  arrangement  with  ALSCRT.  During  2009  and  2008,  we  recognized 
approximately $9.4 million and $6.2 million, respectively, of service revenue related to this transaction, respectively. 

Our Statements of Operations as of and for the years ended December 31, 2009, 2008, 2007 and 2006 reflect the impact of ASC 
718 (previously SFAS No. 123(R), Share-Based Payment (“SFAS 123(R)”)). In accordance with the modified prospective transition 
method, our results of operations for prior periods have not been restated to reflect the impact of ASC 718. Share-based compensation 
expense recognized under ASC 718 for the years ended December 31, 2009, 2008, 2007 and 2006 were $2.6 million, $2.1 million, 
$2.7  million  and  $1.2  million,  respectively.  As  of  December  31,  2009,  there  was  $2.5  million  of  unrecognized  compensation  cost 
related  to  outstanding  options  granted  to  employees  that  is  expected  to  be  recognized  as  a  component  of  our  operating  expenses 
through 2011. Compensation costs will be adjusted for future changes in estimated forfeitures. 

Item 7. MANAGEMENT’S DISCUSSION AND ANALYSIS OF FINANCIAL CONDITION AND RESULTS OF OPERATIONS 

The  following  discussion  and  analysis  of  our  financial  condition  and  results  of  operations  should  be  read  together  with  the 
discussion under “Selected Financial Data” and our consolidated financial statements included in this Annual Report. This discussion 
contains forward-looking statements, based on current expectations and related to future events and our future financial performance, 
that  involve  risks  and  uncertainties.  Our  actual  results  may  differ  materially  from  those  anticipated  in  these  forward-looking 
statements  as  a  result  of  many  important  factors,  including  those  set  forth  under  the  caption  “Risk  Factors”  and  elsewhere  in  this 
Annual Report. 

Overview 

CytRx Corporation 

We are a biopharmaceutical research and development company engaged in the development of high-value human therapeutics, 
specializing  in  oncology.  Our  drug  development  pipeline  includes  clinical  development  of  three  product  candidates  for  cancer 
indications, including three planned Phase 2 clinical trials for INNO-206 as a treatment for pancreatic cancer, gastric (stomach) cancer 
and  soft  tissue  sarcomas,  two  Phase  2  proof-of-concept  clinical  trials  with  bafetinib  in  patients  with  high-risk  B-cell  chronic 
lymphocytic  leukemia,  or  B-CLL,  and  patients  with  glioblastoma  multiforme,  and  a  registration  study  of  tamibarotene  for  the 
treatment  of  acute  promyelocytic  leukemia,  or  APL.  In  addition  to  our  core  oncology  programs,  we  are  developing  two  drug 
candidates based on our molecular chaperone regulation technology, which aim  to repair or degrade mis-folded proteins associated 
with disease. Apart from our drug development programs, we currently maintain a 36% equity interest in our former subsidiary, RXi. 

In  order  to  fund  our  business  and  operations,  we  have  relied  primarily  upon  sales  of  our  equity  securities,  including  proceeds 
received  upon  the  exercise  of  options  and  warrants,  and  sales  of  our  shares  of  RXi  common  stock.  We  also  have  received  limited 
payments from our strategic partners and licensees. 

31 

 
 
 
 
  
 
  
  
 
 
At December 31, 2009, we had cash and cash equivalents of approximately $9.9 million, marketable securities of $22.8 million and 
held 5,768,881 shares of restricted common stock of RXi with a market value of $26.4 million based upon the closing price of the RXi 
common stock on that date. On July 27, 2009, we raised approximately $18.3 million, net of fees and expenses, in a registered direct 
offering, and on September 23, 2009, we raised approximately $1.2 million, net of fees, from the sale of 500,000 shares of our common 
stock of RXi. Management believes that our current cash on hand, together with our marketable securities and proceeds from possible 
future sales of RXi common stock, will be sufficient to fund our operations for the foreseeable future. The estimate is based, in part, upon 
our  currently  projected  expenditures  for  2010  of  approximately  $18.0  million  (unaudited),  which  includes  approximately  $3.2  million 
(unaudited)  for  our  clinical  programs  for  INNO-206,  approximately  $1.6  million  (unaudited)  for  our  clinical  programs  for  bafetinib, 
approximately $2.5 million (unaudited) for our clinical program for tamibarotene, approximately $1.4 million (unaudited) for our activities 
for  arimoclomol,  approximately  $2.2  million  (unaudited)  for  general  operation  of  its  clinical  programs,  and  approximately  $7.1  million 
(unaudited) for other general and administrative expenses. These projected expenditures are also based upon numerous other assumptions 
and subject to many uncertainties, and actual expenditures may be significantly different from these projections. We will be required to 
obtain additional funding in order to execute our long-term business plans, although we do not currently have commitments from any third 
parties to provide us with capital. The fair value of common stock investment in RXi is subject to market fluctuations that could impact the 
amount  of  cash  we  generate  from  the  sale  of  RXi  shares  in  the  future.  We  cannot  assure  that  additional  funding  will  be  available  on 
favorable terms, or at all. If we fail to obtain additional funding when needed, we may not be able to execute our business plans and our 
business may suffer, which would have a material adverse effect on our financial position, results of operations and cash flows. 

Our Separation from RXi Pharmaceuticals Corporation 

RXi Pharmaceuticals Corporation was founded in April 2006 by us and four researchers in the field of RNAi, including Dr. Craig 
Mello, recipient of the 2006 Nobel Prize for Medicine for his co-discovery of RNAi. RNAi is a naturally occurring mechanism for the 
regulation  of  gene  expression  that  has  the  potential  to  selectively  inhibit  the  activity  of  any  human  gene.  In  January  2007,  we 
transferred to RXi substantially all of our RNAi-related technologies and assets, and RXi began operating on a stand-alone basis for 
the  purpose  of  accelerating  the  discovery  of  RNAi  therapeutics  previously  sponsored  by  us.  RXi’s  initial  focus  is  on  developing 
RNAi-based product candidates for treating neurological and metabolic disorders and cancer. 

Until early 2008, we owned approximately 85% of the outstanding shares of common stock of RXi and our financial statements, 
including our financial statements as of and for the year ended December 31, 2007, included the consolidated financial condition and 
results of operations of RXi. On February 14, 2008, our board of directors declared a dividend of one share of RXi common stock for 
each  approximately  20.05  shares  of  our  common  stock  held  by  such  stockholders,  which  was  paid  on  March  11,  2008  and  which 
reduced our ownership of RXi shares to less than 50%. 

For  periods beginning  with  the  first  quarter  of 2008, we began  to  account for  our  investment  in  RXi  using  the  equity  method, 
under which we record only our pro-rata share of the financial results of RXi as “equity in loss of unconsolidated subsidiary” on our 
statements of operations. Because a portion of RXi’s financial results for 2008 and all of RXi’s financial results for 2007 were not 
recorded by us under the equity method, our results of operations for the year ended December 31, 2009 are not directly comparable to 
results of operations for the same periods in prior years. 

Research and Development 

Expenditures for research and development activities related to continuing operations were $7.5 million, $10.5 million and $18.8 
million  for  the  years  ended  December  31,  2009,  2008  and  2007,  or  approximately  44%,  35%  and  55%,  respectively,  of  our  total 
expenses. 

Research and development expenses are further discussed below under “Critical Accounting Policies and Estimates” and “Results 

of Operations.” 

Our  currently  projected  expenditures  for  2010  include  approximately  $3.2  million  for  our  clinical  programs  for  INNO-206, 
approximately  $1.6  million  for  our  clinical  programs  for  bafetinib,  approximately  $2.5  million  for  our  clinical  program  for 
tamibarotene, approximately $1.4 million for our activities for arimoclomol, and approximately $2.2 million for general operation of 
our  clinical  programs.  The  actual  cost  of  our  clinical  programs  could  differ  significantly  from  our  current  projections  due  to  any 
additional requirements or delays imposed by the FDA in connection with our planned trials, or if actual costs are higher than current 
management  estimates  for  other  reasons,  including  complications  with  manufacturing.  In  the  event  that  actual  costs  of  our  clinical 
program, or any of our other ongoing research activities, are significantly higher than our current estimates, we may be required to 
significantly modify our planned level of operations. 

32 

  
  
  
  
  
  
  
  
 
There is a risk that any drug discovery and development program may not produce revenue because of the risks inherent in drug 
discovery and development. The successful development of any product candidate is highly uncertain. We cannot reasonably estimate 
or know the nature, timing and costs of the efforts necessary to complete the development of, or the period in which material net cash 
inflows  are  expected  to  commence  from  any  product  candidate,  due  to  the  numerous  risks  and  uncertainties  associated  with 
developing drugs, including the uncertainty of: 

• 

• 

• 

• 

• 

• 

• 

• 

• 

• 

our ability to advance product candidates into pre-clinical and clinical trials; 

the scope, rate and progress of our pre-clinical trials and other research and development activities; 

the scope, rate of progress and cost of any clinical trials we commence; 

the cost of filing, prosecuting, defending and enforcing any patent claims and other intellectual property rights; 

future clinical trial results; 

the terms and timing of any collaborative, licensing and other arrangements that we may establish; 

the cost and timing of regulatory approvals; 

the cost and timing of establishing sales, marketing and distribution capabilities; 

the cost of establishing clinical and commercial supplies of our product candidates and any products that we may develop; 
and 

the effect of competing technological and market developments. 

Any failure to complete any stage of the development of our products in a timely manner could have a material adverse effect on 
our operations, financial position and liquidity. A discussion of the risks and uncertainties associated with our business is set forth in 
the “Risk Factors” section of this Annual Report. 

Critical Accounting Policies and Estimates 

Management’s discussion and analysis of our financial condition and results of operations are based on our consolidated financial 
statements, which have been prepared in accordance with accounting principles generally accepted in the United States of America. 
The preparation of these financial statements requires management to make estimates and judgments that affect the reported amounts 
of  assets,  liabilities,  revenues  and  expenses,  and  related  disclosure  of  contingent  assets  and  liabilities.  On  an  ongoing  basis, 
management  evaluates  its  estimates,  including  those  related  to  revenue  recognition,  stock  options,  impairment  of  long-lived  assets, 
including finite lived intangible assets, accrued liabilities and certain expenses. We base our estimates on historical experience and on 
various other assumptions that are believed to be reasonable under the circumstances, the results of which form the basis for making 
judgments about the carrying values of assets and liabilities that are not readily apparent from other sources. Actual results may differ 
materially from these estimates under different assumptions or conditions. 

Our  significant  accounting  policies  are  summarized  in  Note  2  of  the  Notes  to  Financial  Statements  included  in  this  Annual 
Report. We believe the following critical accounting policies are affected by our more significant judgments and estimates used in the 
preparation of our consolidated financial statements: 

Revenue Recognition 

Revenue consists of license fees from strategic alliances with pharmaceutical companies as well as service and grant revenues. 

Service revenue consists of contract research and laboratory consulting. Grant revenues consist of government and private grants. 

33 

 
 
 
 
 
 
 
 
 
 
 
  
  
  
  
  
 
 
Monies  received  for  license  fees  are  deferred  and  recognized  ratably  over  the  performance  period  in  accordance  with  Staff 
Accounting  Bulletin  (“SAB”)  No.  104,  Revenue  Recognition.  Milestone  payments  will  be  recognized  upon  achievement  of 
themilestone as long as the milestone is deemed substantive and we have no other performance obligations related to the milestone 
and  collectability  is  reasonably  assured,  which  is  generally  upon  receipt,  or  recognized  upon  termination  of  the  agreement  and  all 
related obligations. Deferred revenue represents amounts received prior to revenue recognition. 

Revenues from contract research, government grants, and consulting fees are recognized over the respective contract periods as 
the services are performed, provided there is persuasive evidence or an arrangement, the fee is fixed or determinable and collection of 
the  related  receivable  is  reasonably  assured.  Once  all  conditions of  the  grant  are  met  and no  contingencies remain  outstanding,  the 
revenue is recognized as grant fee revenue and an earned but unbilled revenue receivable is recorded. 

In August 2006, we received approximately $24.3 million in proceeds from the privately-funded ALS Charitable Remainder Trust 
(“ALSCRT”) in exchange for the commitment to continue research and development of arimoclomol and other potential treatments 
for  ALS  and  a  one  percent  royalty  in  the  worldwide  sales  of  arimoclomol.  We  accounted  for  the  transaction  under  ASC  730-20 
(previously  Statement  of  Financial  Accounting  Standards  No.  68,  Research  and  Development  Arrangements).  Accordingly,  we 
recorded the value received under the arrangement as deferred service revenue and recognize service revenue, using the proportional 
performance  method  of  revenue  recognition,  on  a  dollar-for-dollar  basis  for  each  dollar  of  expense  incurred  for  the  research  and 
development of arimoclomol and other potential ALS treatments. In August 2009, we were released from all restrictions on the use of 
any proceeds previously paid to us in connection with the arrangement. As a result, we recognized in the third quarter $6.7 million of 
service  revenue  representing  the  remaining  deferred  revenue  and  previously  un-recognized  portion  of  the  value  received  in  the 
transaction  with  ALSCRT.  For  the  years  ended  December  31,  2009  and  2008,  we  recognized  approximately  $9.4  million  and  $6.2 
million, respectively, of service revenue related to this transaction. 

Research and Development Expenses 

Research and development expenses consist of costs incurred for direct and overhead-related research expenses and are expensed 
as  incurred.  Costs  to  acquire  technologies,  including  licenses,  that  are  utilized  in  research  and  development  and  that  have  no 
alternative  future  use  are  expensed  when  incurred.  Technology  developed  for  use  in  its  products  is  expensed  as  incurred  until 
technological feasibility has been established. 

Clinical Trial Expenses 

Clinical trial expenses, which are included in research and development expenses, include obligations resulting from the Company’s 
contracts  with  various  clinical  research  organizations  in  connection  with  conducting  clinical  trials  for  its  product  candidates.  We 
recognize expenses for these  activities based on a variety of factors,  including actual  and estimated  labor hours, clinical  site initiation 
activities,  patient  enrollment  rates,  estimates  of  external  costs  and  other  activity-based  factors.  We  believe  that  this  method  best 
approximates the efforts expended on a clinical trial with the expenses we record. We adjust our rate of clinical expense recognition if 
actual results differ from our estimates. If our estimates are incorrect, clinical trial expenses recorded in any particular period could vary. 

Stock-based Compensation 

Our  stock-based  employee  compensation  plans  are  described  in  Note  15  of  the  Notes  to  our  Financial  Statements.  We  have 
adopted  the  provisions  of  ASC  718  (previously  SFAS  No.  123(R),  Share-Based  Payment  (“SFAS  123(R)”)),  which  requires  the 
measurement and recognition of compensation expense for all stock-based awards made to employees and non-employees. 

For stock options and stock warrants paid in consideration of services rendered by non-employees, we recognize compensation 
expense in accordance with the requirements of ASC 718 (previously SFAS No. 123(R)), ASC 505-50 (previously Emerging Issues 
Task  Force  Issue  No.  96-18  (“EITF  96-18”)),  Accounting  for  Equity  Instruments  that  are  Issued  to  other  than  Employees  for 
Acquiring,  or  in  Conjunction  with  Selling  Goods  or  Services  and  ASC  505  (previously  EITF  00-18,  Accounting  Recognition  for 
Certain Transactions involving Equity Instruments Granted to Other Than Employees), as amended. 

Non-employee option grants that do not vest immediately upon grant are recorded as an expense over the vesting period. At the 
end of each financial reporting period prior to performance, the value of these options, as calculated using the Black-Scholes option-
pricing model, is determined, and compensation expense recognized or recovered during the period is adjusted accordingly. Since the 
fair  market  value  of  options  granted  to  non-employees  is  subject  to  change  in  the  future,  the  amount  of  the  future  compensation 
expense is subject to adjustment until the common stock options or warrants are fully vested. 

34 

  
  
  
  
  
  
  
  
  
  
 
Impairment of Long-Lived Assets 

We review long-lived assets, including finite lived intangible assets, for impairment on an annual basis, as of December 31, or on 
an  interim  basis  if  an  event occurs  that  might reduce  the  fair value of such  assets below  their  carrying  values. An impairment loss 
would  be  recognized  based  on  the  difference  between  the  carrying  value  of  the  asset  and  its  estimated  fair  value,  which  would  be 
determined  based  on  either  discounted  future  cash  flows  or  other  appropriate  fair  value  methods.  If  our  estimates  used  in  the 
determination of either discounted future cash flows or other appropriate fair value methods are not accurate as compared to actual 
future results, we may be required to record an impairment charge. The fixed assets, from our San Diego laboratory and our molecular 
library, available for sale were re-allocated from Equipment and Furnishings to Assets Held for Sale and were written down to their 
estimated net realizable value as of September 30, 2009. 

Net Income (Loss) Per Share 

Basic  net  income  (loss)  per  common  share  is  computed  using  the  weighted-average  number  of  common  shares  outstanding. 
Diluted net income (loss) per common share is computed using the weighted-average number of common share and common share 
equivalents outstanding. Common share equivalents that could potentially dilute basic earnings per share in the future, and that were 
excluded  from  the  computation  of  diluted  loss  per  share,  totaled  approximately  24.4  million  shares,  15.2  million  shares  and  17.1 
million shares at December 31, 2009, 2008 and 2007, respectively. 

As a result of our March 11, 2008 distribution by our stockholders of approximately 36% of the outstanding shares of RXi, we 
recorded a deemed dividend of approximately $757,000. The deemed dividend was reflected as an adjustment to net loss for the first 
quarter of 2008 to arrive at net loss applicable to common stockholders on the consolidated statement of operations and for purposes 
of calculating basic and diluted earnings per shares. 

Quarterly Financial Data 

The following table sets forth unaudited consolidated statements of operations data for each quarter during our most recent two fiscal 
years.  This  quarterly  information  has  been  derived  from  our  unaudited  consolidated  financial  statements  and,  in  the  opinion  of 
management,  includes  all  adjustments,  consisting  only  of  normal  recurring  adjustments,  necessary  for  a  fair  presentation  of  the 
information for the periods covered. The quarterly financial data should be read in conjunction with our consolidated financial statements 
and related notes. The operating results for any quarter are not necessarily indicative of the operating results for any future period. 

Quarters Ended 

  March 31    

June 30 

     September 30     December 31  

(In thousands, except per share data)

2009 
Total revenues . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .  $
Net income (loss) . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   
Net income (loss) applicable to common stockholders . . . . . . . . . . . . . . . . . .  $
Basic and diluted (income) loss per share applicable to common stock   $

1,483    $
(3,973)    
(3,973)   $
(0.04)   $

1,000    $ 
(2,226)     
(2,226)   $ 
(0.02)   $ 

6,954    $
3,863     
3,863    $
0.04    $

2008 
Total revenues . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .  $
Net loss . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   
Deemed dividend for anti-dilution adjustments made to outstanding 

common stock warrants . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   
Net loss applicable to common stockholders . . . . . . . . . . . . . . . . . . . . . . . . . . .  $
Basic and diluted loss per share applicable to common stock . . . . . . . . . .  $

2,181    $
(5,374)    

1,740    $ 
(5,826)     

917    $
(12,316)    

(757)    
(6,131)   $
(0.07)   $

—      
(5,826)   $ 
(0.06)   $ 

—     
(12,316)   $
(0.14)   $

100 
(2,464)
(2,464)
(0.03)

1,427 
(3,530)

— 
(3,530)
(0.03)

Quarterly  and  yearly  loss  per  share  amounts  are  computed  independently  of  each  other.  Therefore,  the  sum  of  the  per  share 
amounts  for  the  quarters  may  not  equal  the  per  share  amounts  for  the  year.  In  2009  and  2008  we  incurred  $2.3  million  and  $2.1 
million, respectively, in employee non-cash compensation expenses. 

In connection with our adjustment to the exercise terms of certain outstanding warrants to purchase common stock on March 11, 
2008,  we  recorded  deemed  dividends  of  $757,000.  These  deemed  dividends  are  reflected  as  an  adjustment  to  net  loss  for  the  first 
quarter of 2008 to arrive at net loss applicable to common stockholders on the consolidated statement of operations and for purposes 
of calculating basic and diluted earnings per shares. 

35 

  
  
  
  
  
  
  
 
 
  
 
 
    
      
      
      
 
  
  
  
  
  
  
  
  
  
  
  
  
   
     
      
     
 
 
  
 
Liquidity and Capital Resources 

General 

In  order  to  fund  our  business  and  operations,  we  have  relied  primarily  upon  sales  of  our  equity  securities,  including  proceeds 
received  upon  the  exercise  of  options  and  warrants,  and  sales  of  our  shares  of  RXi  common  stock.  We  also  have  received  limited 
payments from our strategic partners and licensees. 

At December 31, 2009, we had cash and cash equivalents of approximately $9.9 million, marketable securities of $22.8 million 
and held 5,768,881 shares of restricted common stock of RXi with a market value of $26.4 million based upon the closing price of the 
RXi common stock on that date. On July 27, 2009, we raised approximately $18.3 million, net of fees and expenses, in a registered 
direct offering, and on September 23, 2009, we raised approximately $1.2 million, net of fees, from the sale of 500,000 shares of our 
common stock of RXi. Management believes that our current cash on hand, together with our marketable securities and proceeds from 
possible future sales of RXi common stock, will be sufficient to fund our operations for the foreseeable future. The estimate is based, 
in part, upon our currently projected expenditures for 2010 of approximately $18.0 million (unaudited), which includes approximately 
$3.2 million (unaudited) for our clinical programs for INNO-206, approximately $1.6 million (unaudited) for our clinical programs for 
bafetinib, approximately $2.5 million (unaudited) for our clinical program for tamibarotene, approximately $1.4 million (unaudited) 
for  our  activities  for  arimoclomol,  approximately  $2.2  million  (unaudited)  for  general  operation  of  its  clinical  programs,  and 
approximately  $7.1  million  (unaudited)  for  other  general  and  administrative  expenses.  These  projected  expenditures  are  also  based 
upon numerous other assumptions and subject to many uncertainties, and actual expenditures may be significantly different from these 
projections. We will be required to obtain additional funding in order to execute our long-term business plans, although we do not 
currently have commitments from any third parties to provide us with capital. The fair value of common stock investment in RXi is 
subject to market fluctuations that could impact the amount of cash we generate from the sale of RXi shares in the future. We cannot 
assure that additional funding will be available on favorable terms, or at all. If we fail to obtain additional funding when needed, we 
may  not  be  able  to  execute  our  business  plans  and  our  business  may  suffer,  which  would  have  a  material  adverse  effect  on  our 
financial position, results of operations and cash flows. 

If we obtain marketing approval as currently planned and successfully commercialize our product candidates, we anticipate it will 
take  a  minimum  of  three  years,  and  possibly  longer,  for  us  to  generate  significant  recurring  revenue,  and we  will  be  dependent  on 
future  financing  until  such  time,  if  ever,  as  we  can  generate  significant  recurring  revenue.  Our  ability  to  raise  capital  has  been 
materially  and  adversely  affected  by  the  continuing poor economy.  Despite  the  recovery  in  the  U.S. financial  markets  in  2009,  the 
market remains severely depressed for private investment in public equities, or PIPEs, transactions on which we have relied for raising 
needed capital. These conditions also may materially and adversely affect the market for our RXi shares. We have no commitments 
from third parties to provide us with any additional financing, and we may not be able to obtain future financing on favorable terms, or 
at  all.  Failure  to  obtain  adequate  financing  would  adversely  affect  our  ability  to  operate  as  a  going  concern.  If  we  raise  additional 
funds by issuing equity securities, dilution to stockholders may result and new investors could have rights superior to holders of the 
shares  issued  in  this  offering.  In  addition,  debt  financing,  if  available,  may  include  restrictive  covenants.  If  adequate  funds  are  not 
available to us, we may have to liquidate some or all of our assets or to delay or reduce the scope of or eliminate some portion or all of 
our development programs or clinical trials. We also may have to license to other companies our product candidates or technologies 
that we would prefer to develop and commercialize ourselves. 

Discussion of Operating, Investing and Financing Activities 

Net loss for the year ended December 31, 2009 was $4.8 million, and cash used for operating activities for that period was $12.1 
million.  The  net  loss  for  the  year  reflects  $9.4  million  of  revenue  recognized  under  the  2006  agreement  with  ALSCRT,  and  $2.8 
million for stock option and warrant expense. 

Net loss for the year ended December 31, 2008 was $27.0 million, and cash used for operating activities for that period was $19.4 
million. The net loss for the year reflects $6.2 million of revenue recognized under the 2006 agreement with ALSCRT, a expense of 
$8.0 million related to the acquisition of Innovive’s in-process research and development, a loss of $3.9 million in our equity in RXi, 
and $2.1 million for stock option and warrant expense. 

36 

  
  
  
  
  
  
  
 
 
Net loss for the year ended December 31, 2007 was $21.9 million, and cash used for operating activities for that period was $22.4 
million.  The  net  loss  for  the  year  reflects  $7.2  million  of  revenue  recognized  under  the  2006  agreement  with  ALSCRT  and  $3.5 
million for stock option and warrant expense. 

For  the  year  ended  December  31,  2009,  $21.6  million  was  used  in  investing  activities.  This  included  $22.8  million  used  to 
purchase  marketable  securities,  which  was  partially  offset  by  proceeds  of  $1.2  million  from  the  sale  of  500,000  of  our  shares  of 
common stock RXi. 

For  the  year  ended  December  31,  2008,  $7.0  million  was  used  in  investing  activities  including  $10.0  million  of  RXi  funds 
resulting from converting marketable securities to cash equivalents that is not available to us due to the deconsolidation. The total cash 
outlay to acquire Innovive totaled $5.7 million, which related primarily to the payment of Innovive’s accounts payable. The other $0.9 
million was used for the purchase of equipment and furnishings, primarily associated with equipping the San Diego laboratory. 

For the year ended December 31, 2007, $11.0 million was used in investing activities. Of this amount, $9.8 million was used by 
RXi  for  the  purchase  of  marketable  securities.  The  other  $1.3  million  was  used  for  the  purchase  of  equipment  and  furnishings 
primarily associated with equipping our San Diego laboratory. 

Cash provided by financing activities for the year ended December 31, 2009 was $18.6 million. During 2009, we raised $18.3 
million in a private placement of our common stock and an additional $0.3 million from the exercise of previously outstanding stock 
options and warrants. 

Cash provided by financing activities for the year ended December 31, 2008 was $1.0 million. During 2008, we received $1.0 

million from the exercise of stock options and warrants. 

Cash provided by financing activities for the year ended December 31, 2007 was $53.5 million. During 2007, we raised $34.2 
million in a private placement of our common stock and an additional $18.8 million from the exercise of previously outstanding stock 
options and warrants. 

Off-Balance Sheet Arrangements 

We  have  no  off-balance  sheet  arrangements  that  have  a  material  current  effect  or  that  are  reasonably  likely  to  have  a  material 
future effect on our financial condition, changes in financial condition, revenues or expenses, results of operations, liquidity, capital 
expenditures, or capital resources. 

Contractual Obligations 

We acquire assets still in development and enter into research and development arrangements with third parties that often require 
milestone and royalty payments to the third party contingent upon the occurrence of certain future events linked to the success of the 
asset in development. Milestone payments may be required, contingent upon the successful achievement of an important point in the 
development life-cycle of the pharmaceutical product (e.g., approval of the product for marketing by a regulatory agency). If required 
by the arrangement, we may have to make royalty payments based upon a percentage of the sales of the pharmaceutical product in the 
event that regulatory approval for marketing is obtained. Because of the contingent nature of these payments, they are not included in 
the table of contractual obligations. 

These  arrangements  may  be  material  individually,  and  in  the  event  that  milestones  for  multiple  products  covered  by  these 
arrangements were reached in the same period, the aggregate charge to expense could be material to the results of operations in any 
one period. In addition, these arrangements often give us the discretion to unilaterally terminate development of the product, which 
would  allow  us  to  avoid  making  the  contingent  payments;  however,  we  are  unlikely  to  cease  development  if  the  compound 
successfully achieves clinical testing objectives. 

37 

  
  
  
  
  
  
  
  
  
  
  
 
 
Our current contractual obligations that will require future cash payments are as follows (in thousands): 

2010 . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   $
2011 . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
2012 . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
2013 . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
2014 and thereafter . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Total . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   $
____________ 

Operating
Leases (1)(2)     

Employment
Agreements (3)    

Subtotal

Research and 
Development (4)    

Total

873    $
536     
459     
318     
372     
2,558    $

2,210    $
—     
—     
—     
—     
2,210    $

3,083    $ 
536      
459      
318      
372      
4,768    $ 

3,018    $
49     
149     
149     
383     
3,748    $

6,101 
585 
608 
467 
755 
8,516 

(1)  Operating  leases  are  primarily  facility  lease  related  obligations,  as well  as  equipment  and  software  lease  obligations  with  third 

party vendors. 

(2)  We  are  entitled  to  receive  future  rental  income  under  subleases  in  place  which  would  be  offset  against  future  operating  lease 

obligations as follows: $519,000 in 2010, $350,000 in 2011 and $235,000 in 2012. 

(3)  Employment agreements include management contracts, which have been revised from time to time, provide for minimum salary 
levels, adjusted annually at the discretion of our Compensation Committee, as well as for minimum bonuses that are payable. 

(4)  Research and development obligations relate primarily to clinical trials. Most of these purchase obligations are cancelable. 

We  apply  the  disclosure  provisions  of  ASC  460  (formerly  FASB  Interpretation  No.  (“FIN”)  45,  Guarantor’s  Accounting  and 
Disclosure Requirements for Guarantees, Including Indirect Guarantees of Indebtedness of Other), to our contractual guarantees and 
Indemnities. We have provided contractual indemnities to investors and other parties against possible losses suffered or incurred by 
the  indemnified  parties  in  connection  with  various  types  of  third-party  claims,  as  well  as  indemnities  to  our  officers  and  directors 
against third party claims arising from the services they provide to us. To date, we have not incurred material costs as a result of these 
indemnities, and we do not expect to incur material costs in the future; further, we maintain insurance to cover certain losses arising 
from  these  indemnities.  Accordingly,  we  have  not  accrued  any  liabilities  in  our  consolidated  financial  statements  related  to  these 
indemnities. 

Net Operating Loss Carryforwards 

At  December  31,  2009,  we  had  United  States  federal  and  state  net  operating  loss  carryforwards  of  $91.6  million  and  $81.9 
million,  respectively,  available  to  offset  against  future  taxable  income,  which  expire  in  2011  through  2029.  Approximately  $34.7 
million of our federal net operating loss carryforwards are limited in their availability to $0.3 million annually. Management currently 
believes that the remaining $56.9 million in federal net operating loss carryforwards, and the $57.6 million in state net operating loss 
carryforwards  as  of  December  31,  2009,  are  unrestricted.  However,  management  is  reviewing  its  recent  equity  transactions  to 
determine if they may have resulted in any further restrictions on the Company’s net operating loss carryforwards. As of December 
31, 2009, we also had research and development and alternative minimum tax credits for federal and state purposes of approximately 
$8.9 million and $0, respectively, available for offset against future income taxes, which expire in 2022 through 2029. Based on an 
assessment  of  all  available  evidence  including,  but  not  limited  to,  our  limited  operating  history  in  our  core  business  and  lack  of 
profitability, uncertainties of the commercial viability of its technology, the impact of government regulation and healthcare reform 
initiatives, and other risks normally associated with biotechnology companies, we have concluded that it is more likely than not that 
these net operating loss carryforwards and credits will not be realized and, as a result, a 100% deferred tax valuation allowance has 
been recorded against these assets. 

Results of Operations 

We incurred a net loss of $4.8 million, $27.0 million and $21.9 million for the years ended December 31, 2009, 2008 and 2007, 

respectively. 

38 

  
  
 
     
 
 
  
  
 
 
  
  
  
  
 
 
During fiscal 2009, we recognized $9.4 million in service revenues relating to our $24.3 million sale to the ALSCRT of a one-
percent  royalty  interest  in  the  worldwide  sales  of  arimoclomol  in  August  2006.  Pursuant  to  an  amendment  signed  between  us  and 
thebeneficiary of the ALSCRT on August 6, 2009, we were released from all restrictions on the use of any proceeds previously paid to 
us in connection with the arrangement. As a result, we recognized $6.7 million as service revenue in the third quarter of 2009, which 
represented the remaining deferred revenue and previously un-recognized portion of the value received. In the years ended December 
31, 2008 and 2007, we recognized $6.2 million and $7.2 million in service revenues, respectively. 

During 2009, 2008 and 2007, we earned an immaterial amount of license fees and grant revenue. All future licensing fees under 
our current licensing agreements are dependent upon successful development milestones being achieved by the licensor. During fiscal 
2010, we are not anticipating the receipt of any significant service or licensing fees. 

Our  net  loss  may  increase  from  current  levels  primarily  due  to  expenses  related  to  our  ongoing  and  planned  clinical  trials, 
research and development programs, possible technology acquisitions, and other general corporate activities. We anticipate, therefore, 
that  our  operating  results  will  fluctuate  for  the  foreseeable  future  and  period-to-period  comparisons  should  not  be  relied  upon  as 
predictive of the results in future periods. 

Research and Development 

Research and development expenses . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   $
Non-cash research and development expenses . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Impairment loss on fixed assets . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .
Employee stock option expense . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
  $

2009

Years Ended December 31,
2008 
(In thousands)

2007

5,621    $ 
62      
1,187      
672      
7,542    $ 

9,913    $
(224)    
—     
777     
10,466    $

14,454 
3,778 
— 
592 
18,824 

Research  expenses  are  expenses  incurred  by  us  in  the  discovery  of  new  information  that  will  assist  us  in  the  creation  and  the 
development  of  new  drugs  or  treatments.  Development  expenses  are  expenses  incurred  by  us  in  our  efforts  to  commercialize  the 
findings generated through our research efforts. 

Research and development expenses incurred during 2009, 2008 and 2007 relate to our various development programs. In 2009, 
we substantially completed the initial phase of our new-drug discovery research in our laboratory facility in San Diego, California, 
which account for the significant decrease in research and development expenses from 2008. In 2008, only the months of January and 
February included RXi-related expenses (totaling approximately $0.6 million), which accounts for the significant decrease in research 
and  development  expenses,  and  non-cash  research  and  development  expenses.  In  2009,  our  development  costs  associated  included 
approximately  $0.8  million  for  our  clinical  programs  for  INNO-206,  approximately  $0.25  million  for  our  clinical  programs  for 
bafetinib,  $0.8  million  for  our  clinical  program  for  tamibarotene,  approximately  $0.4  million  for  our  activities  for  arimoclomol, 
approximately  $0.4  million  for  general  operation  of  our  clinical  programs,  and  approximately  $3.0  million  for  other  general  and 
administrative expenses. None of our research and development costs have ever been capitalized. 

As  compensation  to  scientific  advisory  board  (“SAB”)  members  and  consultants,  and  in  connection  with  the  acquisition  of 
technology, we and RXi sometimes issue shares of common stock, stock options and warrants to purchase shares of common stock. 
For financial statement purposes, we value these shares of common stock, stock options, and warrants at the fair value of the common 
stock,  stock  options  or  warrants  granted,  or  the  services  received,  whichever  is  more  reliably  measurable.  We  recorded  charges 
(recovery) of $0.0 million, $(0.2 million) and $3.8 million in this regard during 2009, 2008 and 2007, respectively. Included in the 
research  and  development  charges  for  2007  were  $2.3  million  of  expense  related  to  RXi’s  issuance  of  462,112  shares  of  common 
stock to UMMS for certain license agreement rights and a new invention disclosure agreement and $1.0 million for non-qualifying 
stock  options  to  SAB  members  of  RXi.  In  2009,  we  recorded  $0.7  million  of  employee  stock  option  expense  as  compared  to  $0.8 
million in 2008 and $0.6 million in 2007. 

We  also  incurred  an  expenditure  of  $8.0  million  in  2008  related  to  the  acquisition  of  Innovive’s  in-process  research  and 

development, which has been reflected as a separate line item on our Consolidated Statements of Operations. 

In  2010,  we  expect  our  research  and  development  expenses  to  increase  as  a  result  of  our  clinical  programs  with  INNO-206, 

bafetinib and tamibarotene. 

39 

  
  
  
  
  
 
 
  
 
     
   
 
 
 
 
 
  
  
  
  
 
General and administrative expenses 

General and administrative expenses . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   $
Stock, stock option and warrant expenses to non-employees and consultants . . . . . . . . .    
Employee stock option expense . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
  $

2009

Year Ended December 31,
2008 
(In thousands)

2007

7,128    $ 
421      
1,579      
9,128    $ 

9,134    $
189     
1,610     
10,933    $

12,666 
2 
2,154 
14,822 

General and administrative expenses include all administrative salaries and general corporate expenses, including legal expenses 
associated with the prosecution of our intellectual property. Our general and administrative expenses, excluding common stock, stock 
options and warrants issued, and excluding depreciation expense, were $7.1 million in 2009, $9.1 million in 2008 and $12.7 million, 
respectively,  in  2007.  General  and  administrative  expenses  in  2007  included  $4.6  million  of  RXi-related  expenses.  In  2008,  we 
recognized RXi-related expenses for January and February only of $1.3 million. No RXi-related expenses were recognized in 2009. 
General and administrative expenses in 2009 decreased by $2.0 million as compared to 2008, due primarily to the $1.3 million of RXi-
related  expenses  recognized  in  2008.  In  2009,  legal  and  accounting/auditing  expenses  decreased  by  approximately  $302,000  and 
$304,000, respectively, primarily due to the higher expenses incurred in 2008 in connection with our acquisition of Innovive, as well 
as efficiencies in the administrative area. 

From  time  to  time,  we  issue  shares  of  our  common  stock  or  warrants  or  options  to  purchase  shares  of  our  common  stock  to 
consultants and other service providers in exchange for services. For financial statement purposes, we value these shares of common 
stock, stock options, and warrants at the fair value of the common stock, stock options or warrants granted, or the services received, 
whichever we can measure more reliably. 

We recorded employee stock option expense of $1.6 million in 2009, $1.6 million in fiscal 2008 and $2.2 million in fiscal 2007. 
The greater amount in 2007 primarily related to stock options granted by RXi to recruit and retain directors, officers and additional 
employees. 

Depreciation and amortization 

Depreciation and amortization expenses for the years ended December 31, 2009, 2008 and 2007 were $475,000, $625,000 and 
$272,000, respectively. The depreciation expense reflects the depreciation of our fixed assets and the amortization expenses related to 
our molecular library. The decrease in 2009 relates to a lower depreciation base due to the re-class of fixed assets to Assets-held-for-
sale and the value of the molecular library related to the closure of the San Diego lab in the third quarter of 2009. 

Other Income 

In 2009, we recognized a gain of $0.7 million on the valuation of our warrant derivative liability related to warrants issued in July 
2009. In  July 2009, we recognized  a  gain of  $1.2  million on  the  sale of  RXi  shares.  In  March 2008, we recognized  a  gain of  $0.2 
million on the transfer of some RXi common stock to certain employees. In June 2007, we recognized $1.5 million of income arising 
from  a  fee  received  pursuant  to  a  change-in-control  provision  included  in  the  purchase  agreement  for  our  1998  sale  of  our  animal 
pharmaceutical unit. 

Interest income 

Interest income was $0.3 million in 2009, $1.2 million in 2008 and $2.7 million in 2007. The variances between years are attributable 

primarily to the amount of funds available for investment each year and, to a lesser extent, changes in prevailing market rates. 

Noncontrolling Interest in RXi 

We offset $88,000 of losses in noncontrolling interest in RXi against our net loss for the months of January and February 2008. 
For the remainder of the year, and for 2009, RXi’s gain and losses were accounted for under the equity method, because we owned 
less than 50% of RXi following our March 11, 2008 distribution to our stockholders of RXi shares. We offset $449,000 of minority 
interest in losses of RXi against our net loss for the year ended December 31, 2007. 

40 

  
  
 
 
  
 
     
   
 
 
 
 
  
  
  
  
  
  
  
  
  
  
 
Recent Accounting Pronouncements 

In  December  2007,  the  FASB  issued  guidance  which  is  now  part  of  ASC  810-10,  Noncontrolling  Interests  in  Consolidated 
Financial  Statements,  an  Amendment  of  Accounting  Research  Bulletin  No.  51  “  (formerly  Statement  of  Financial  Accounting 
Standards  (SFAS)  160,  Noncontrolling  Interests  in  Consolidated  Financial  Statements—an  amendment  of  ARB  No.  51  ).  This 
guidance establishes accounting and reporting standards for ownership interests in subsidiaries held by parties other than the parent, 
changes in a parent’s ownership of a noncontrolling interest, calculation and disclosure of the consolidated net income attributable to 
the parent  and  the noncontrolling  interest, changes  in  a parent’s ownership  interest while  the parent  retains  its  controlling  financial 
interest  and  fair  value  measurement  of  any  retained  noncontrolling  equity  investment.  The  new  guidance  is  effective  for  financial 
statements issued for fiscal years beginning after December 15, 2008, and interim periods within those fiscal years. Early adoption is 
prohibited.  We  adopted  this  guidance  on  January  1,  2009,  the  beginning  of  its  2009  fiscal  year,  which  resulted  in  certain 
reclassifications related to the noncontrolling interest in the consolidated financial statements. 

In  March  2008,  the  FASB  issued  guidance  ASC  815-10  (formerly  Statement  of  Financial  Accounting  Standards  No.  161, 
Disclosures about Derivative Instruments and Hedging Activities (“SFAS No. 161”). The new standard amends Statement of Financial 
Accounting Standards No. 133, Accounting for Derivative Instruments and Hedging Activities (“SFAS 133”), and seeks to enhance 
disclosure about how and why a company uses derivatives; how derivative instruments are accounted for under SFAS 133 (and the 
interpretations  of  that  standard);  and  how  derivatives  affect  a  company’s  financial  position,  financial  performance  and  cash  flows. 
SFAS 161 will be effective for financial statements issued for fiscal years and interim periods beginning after November 15, 2008. 
Early application of the standard is encouraged, as well as comparative disclosures for earlier periods at initial adoption. The adoption 
of ASC 815-10 did not have a material impact on our consolidated financial statements. 

In April 2008, the FASB issued revised guidance on determining the useful life of intangible assets. The revised guidance, which 
is now part of ASC 350-30 General Intangibles Other than Goodwill (previously Staff Position No. FAS 142-3, Determination of the 
Useful Life of Intangible Assets), amends the factors that should be considered in developing renewal or extension assumptions used to 
determine the useful life of a recognized intangible asset. The Position is effective for fiscal years beginning after December 15, 2008 
and applies prospectively to intangible assets acquired after the effective date. Early adoption is not permitted. The adoption of SFAS 
No. ASC 350-30 did not have a material impact on our consolidated financial statements. 

In May 2008, the FASB issued revised guidance on Convertible Debt Instruments. The revised guidance which is now part of 
ASC 470-20 (formerly Staff Position No. Accounting Principles Board 14-1, Accounting for Convertible Debt Instruments That May 
Be  Settled  in  Cash  upon  Conversion  (Including  Partial  Cash  Settlement)  (“FSP  No.  APB  14-1”)).  ASC  470-20  requires  that  the 
liability and equity components of convertible debt instruments that may be settled in cash upon conversion (including partial cash 
settlement)  be  separately  accounted  for  in  a  manner  that  reflects  an  issuer’s  nonconvertible  debt  borrowing  rate.  ASC  470-20  is 
effective for us as of January 1, 2009. The adoption of ASCO 470-20 did not have an impact on our consolidated financial statements. 

In June 2008, the FASB ratified guidance which is now part of ASC 815-40, Contracts in Entity’s Own Equity (formerly EITF 
(Emerging  Issues  Task  Force)  07-05),  Determining  Whether  an  Instrument  (or  Embedded  Feature)  Is  Indexed  to  an  Entity’s  Own 
Stock. The objective of this issue is to provide guidance for determining whether an equity-linked financial instrument (or embedded 
feature) is indexed to an entity’s own stock. This issue applies to any freestanding financial instrument or embedded feature that has 
all the characteristics of a derivative instrument or an instrument which may be potentially settled in an entity’s own stock regardless 
of  whether  the  instrument  possess  derivative  characteristics.  This  issue  provides  a  two-step  approach  to  assist  in  making  these 
determinations and is effective for financial statements issued for fiscal years beginning after December 15, 2008. The adoption of 
ASC 815-40 did not have a material impact on our consolidated financial statements. 

In  April  2009,  the  FASB  issued  guidance  which  is  now  part  of  ASC  825-10  Financial  Instruments  (formerly  Financial  Staff 
Position SFAS 107-1 and Accounting Principles Board (APB) Opinion No. 28-1, Interim Disclosures about Fair Value of Financial 
Instruments  (SFAS  107-1  and  APB  28-1).  This  statement  amends  FASB  Statement  No.  107,  Disclosures  about  Fair  Values  of 
Financial  Instruments,  to  require  disclosures  about  fair  value  of  financial  instruments  in  interim  financial  statements  as  well  as  in 
annual  financial  statements.  The  statement  also  amends  APB  Opinion  No.  28,  “Interim  Financial  Reporting,”  to  require  those 
disclosures in all interim financial statements. This statement is effective for interim periods ending after June 15, 2009. The adoption 
of ASC 825-10 did not have an impact on our financial statements. 

41 

  
  
  
  
  
  
 
 
In May 2009 and February 2010, the FASB issued new guidance for accounting for subsequent events. The new guidance, which is 
now part of ASC 855-10, Subsequent Events (formerly, SFAS No. 165, Subsequent Events) is consistent with existing auditing standards 
in defining subsequent events as events or transactions that occur after the balance sheet date but before the financialstatements are issued 
or  are  available  to  be  issued.  The  new  guidance  defines  two  types  of  subsequent  events:  “recognized  subsequent  events”  and  “non-
recognized subsequent events.” Recognized subsequent events provide additional evidence about conditions that existed at the balance 
sheet  date  and  must  be  reflected  in  the  company’s  financial  statements.  Non-recognized  subsequent  events  provide  evidence  about 
conditions that arose after the balance sheet date and are not reflected in the financial statements of a company. Certain non-recognized 
subsequent events may require disclosure to prevent the financial statements from being misleading. The new guidance was effective on a 
prospective basis for interim or annual periods ending after June 15, 2009. We adopted the provisions of ASC 855-10 as required. 

In  June  2009,  the  FASB  amended  ASC  860,  (formerly  SFAS  No.  166,  Accounting  for  Transfers  of  Financial  Assets,  an 
amendment to SFAS No. 140). ASC 860 eliminates the concept of a “qualifying special-purpose entity,” changes the requirements for 
derecognizing  financial  assets,  and  requires  additional  disclosures  in  order  to  enhance  information  reported  to  users  of  financial 
statements by providing greater transparency about transfers of financial assets, including securitization transactions, and an entity’s 
continuing  involvement  in  and  exposure  to  the  risks  related  to  transferred  financial  assets.  ASC  860  is  effective  for  fiscal  years 
beginning after November 15, 2009. The Company will adopt ASC 860 in fiscal 2010. We do not expect that the adoption of ASC 860 
will have a material impact on our financial statements. 

In  June  2009,  the  FASB  amended  ASC  810  (formerly  SFAS  No.167,  Amendments  to  FASB  Interpretation  No.  46).  The 
amendments include: (1) the elimination of the exemption for qualifying special purpose entities, (2) a new approach for determining 
who  should  consolidate  a  variable-interest  entity,  and  (3)  changes  to  when  it  is  necessary  to  reassess  who  should  consolidate  a 
variable-interest entity. ASC 810 is effective for the first annual reporting period beginning after November 15, 2009 and for interim 
periods within that first annual reporting period. We will adopt ASC 810 in fiscal 2010. We do not expect that the adoption of ASC 
810 will have a material impact on our financial statements. 

In  June  2009,  the  FASB  issued  new guidance  which  is  now  part  of  ASC  105-10  (formerly  Statement  of  Financial Accounting 
Standards No. 168, The FASB Accounting Standards Codification and the Hierarchy of Generally Accepted Accounting Principles ). 
ASC 105-10 replaces FASB Statement No. 162, “The Hierarchy of Generally Accepted Accounting Principles”, and establishes the 
FASB Accounting Standards Codification as the source of authoritative accounting principles recognized by the FASB to be applied 
by nongovernmental entities in the preparation of financial statements in conformity  with generally accepted accounting principles. 
ASC 105-10 is effective for interim and annual periods ending after September 15, 2009. The adoption of ASC 105-10 did not have a 
material impact on our financial statements. 

In January, 2010, the FASB issued ASU 2010-06, Improving Disclosures about Fair Value Measurements. The standard amends 
ASC Topic 820, Fair Value Measurements and Disclosures to require additional disclosures related to transfers between levels in the 
hierarchy of fair value measurement. The standard does not change how fair values are measured. The standard is effective for interim 
and annual reporting periods beginning after December 15, 2009. As a result, it is effective for us in the first quarter of fiscal year 
2010. We do not believe that the adoption of ASU 2010-06 will have a material impact on consolidated our financial statements. 

Item 7A. QUANTITATIVE AND QUALITATIVE DISCLOSURES ABOUT MARKET RISK 

Our exposure to market risk is limited primarily to interest income sensitivity, which is affected by changes in the general level of 
U.S.  interest  rates,  particularly  because  a significant  portion  of our  investments  are in short-term  debt securities  issued  by  the  U.S. 
government and institutional money market funds. The primary objective of our investment activities is to preserve principal. Due to 
the nature of our marketable securities, we believe that we are not exposed to any material market risk. We do not have any derivative 
financial  instruments  or  foreign  currency  instruments.  If  interest  rates  had  varied  by  10%  in  the  year  ended  December  31,  2009,  it 
would not have had a material effect on our results of operations or cash flows for that period. 

Item 8. FINANCIAL STATEMENTS AND SUPPLEMENTARY DATA 

Our consolidated financial statements and supplemental schedule and notes thereto as of December 31, 2009 and 2008, and for 
each of the three years in the period ended December 31, 2009, together with the reports thereon of our independent registered public 
accounting firms, are set forth on pages F-1 to F-26 of this Annual Report. 

Item  9.  CHANGES  IN  AND  DISAGREEMENTS  WITH  ACCOUNTANTS  ON  ACCOUNTING  AND  FINANCIAL 
DISCLOSURE 

None. 

42 

 
  
  
  
  
  
  
  
  
 
 
Item 9A. CONTROLS AND PROCEDURES 

Disclosure Controls and Procedures 

We maintain disclosure controls and procedures that are designed to ensure that the information disclosed in the reports we file 
with the Securities and Exchange Commission under the Exchange Act is recorded, processed, summarized and reported within the 
time periods specified in the Securities and Exchange Commission’s rules and forms, and that such information is accumulated and 
communicated to our management, including our Chief Executive Officer and Chief Financial Officer, as appropriate, to allow timely 
decisions regarding required disclosure. 

Our management, with the participation of our Chief Executive Officer and Chief Financial Officer, performed an evaluation of 
the effectiveness of the design and operation of our disclosure controls and procedures (as defined in Securities Exchange Act Rule 
13a-15(e)) as of the end of the period covered by this Annual Report. Based on that evaluation, our Chief Executive Officer and Chief 
Financial  Officer  have  concluded  that  our  disclosure  controls  and  procedures  were  effective  as  of  December  31,  2009  to  provide 
reasonable assurance that information required to be disclosed by us in reports that we file or submit under the Securities Exchange 
Act  of  1934  is  recorded,  processed,  summarized  and  reported  within  the  time  periods  specified  in  the  Securities  and  Exchange 
Commission’s rules and forms. 

There was no change in our internal control over financial reporting that occurred during the quarter ended December 31, 2009 

that materially affected, or is reasonably likely to materially affect, our internal control over financial reporting. 

Management’s Report on Internal Control Over Financial Reporting 

Our management is responsible for establishing and maintaining adequate internal control over financial reporting, as such term is 

defined in Exchange Act Rule 13a-15(f). 

Under  the  supervision  and  with  the  participation  of  our  management,  including  our  principal  executive  and  principal  financial 
officers,  we  assessed  the  effectiveness  of  our  internal  control  over  financial  reporting  as  of  December  31,  2009.  In  making  this 
assessment,  management  used  the  criteria  set  forth  by  the  Committee  of  Sponsoring  Organizations  of  the  Treadway  Commission 
(“COSO”) in Internal Control-Integrated Framework. Based upon management’s assessment using the criteria contained in COSO, 
our management has concluded that, as of December 31, 2009, our internal control over financial reporting was effective. 

Our internal control over financial reporting as of December 31, 2009 has been audited by BDO Seidman, LLP, an independent 

registered public accounting firm, as stated in their report thereon set forth on pages F-25, which is incorporated herein by reference. 

Item 9B. OTHER INFORMATION 

None. 

43 

  
  
  
  
  
  
  
  
  
 
 
 
Item 10. DIRECTORS, EXECUTIVE OFFICERS AND CORPORATE GOVERNANCE 

The following table sets forth information concerning our directors and executive officers: 

PART III 

Name 
Max Link, Ph.D. . . . . . . . . . . . .   
Steven A. Kriegsman . . . . . . .   
Marvin R. Selter . . . . . . . . . . . .   
Louis Ignarro, Ph.D. . . . . . . . .   
Joseph Rubinfeld, Ph.D. . . . . .   
Richard L. Wennekamp . . . . .   
John Caloz . . . . . . . . . . . . . . . . .   
Daniel Levitt, M.D., Ph.D. . .   
D. Scott Geyer . . . . . . . . . . . . .   
D. Scott Wieland . . . . . . . . . . .   
Benjamin S. Levin . . . . . . . . . .   
David J. Haen . . . . . . . . . . . . . .   
____________ 

Age
69 
68 
82 
68 
77 
67 
58 
62 
55 
50 
33 
31 

Class of 
Director(1)
III 
II 
II 
I 
I 
II 
— 
— 
— 
— 
— 
— 

Position 
Director, Chairman of the Board (2) (3) (4) 
Director, Chief Executive Officer, President 
Director, Vice Chairman of the Board (2) (3) (4) 
Director 
Director 
Director (2) (3) (4) 
Chief Financial Officer 
Chief Medical Officer 
Sr. Vice President-Manufacturing 
Sr. Vice President-Drug Development 
General Counsel, Vice President — Legal Affairs and Corporate Secretary 
Vice President – Business Development 

(1)  Our  Class  I  directors  serve  until  the  2010  annual  meeting  of  stockholders,  our  Class  II  directors  serve  until  the  2011  annual 

meeting of stockholders, and our Class III director serves until the 2012 annual meeting of stockholders. 

(2)  Members of our Audit Committee. Mr. Selter is the Chairman of the Committee. 

(3)  Members of our Nominating and Corporate Governance Committee. Mr. Wennekamp is Chairman of the Committee. 

(4)  Members of our Compensation Committee. Mr. Wennekamp is Chairman of the committee. 

Max Link, Ph.D has been a director since 1996. Dr. Link has been retired from business since 2003. From March 2002 until its 
acquisition by Zimmer Holdings, Dr. Link served as Chairman and CEO of Centerpulse, Ltd. From May 1993 to June 1994, Dr. Link 
served  as  the  Chief  Executive  Officer  of  Corange  Ltd.  (the  holding  company  for  Boehringer  Mannheim  Therapeutics,  Boehringer 
Mannheim Diagnostics and DePuy International). From 1992 to 1993, Dr. Link was Chairman of Sandoz Pharma, Ltd. From 1987 to 
1992, Dr. Link was the Chief Executive Officer of Sandoz Pharma and a member of the Executive Board of Sandoz, Ltd., Basel. Prior 
to 1987, Dr. Link served in various capacities with the United States operations of Sandoz, including President and Chief Executive 
Officer. Dr.  Link  also  serves  as  a  director of Alexion Pharmaceuticals,  Inc.,  Celsion Corporation,  Inc.  and Discovery  Laboratories, 
Inc.,  and  in  the  past  five  years,  also  served  as  a  director  of  Access  Pharmaceuticals,  Inc.,  Cell  Therapeutics,  Inc.,  Columbia 
Laboratories, Inc., Human Genome Sciences, Inc. and Protein Design Laboratories, Inc. 

Dr. Link has extensive executive-level experience with a number of large pharmaceutical companies, including Sandoz Pharma, 
Ltd.  In  these  positions,  he  was  responsible  for  major  strategic  and  other  business  initiatives,  including  new  drug  development, 
acquisitions and dispositions of new drug candidates and other technology, licensing, marketing and distribution agreements and other 
key contractual strategic arrangements that affect, or are likely to affect, our company’s own business efforts. As an executive officer 
and board member of these other companies, he has experience with the regulatory schemes in foreign jurisdictions and also has been 
exposed to different approaches to corporate governance matters, potential conflicts of interest, and similar matters, which enables him 
to offer importance guidance to our Board of Directors. 

Steven A. Kriegsman has been CytRx’s President and Chief Executive Officer and a director since July 2002. He also serves as a 
director of CytRx’s 36% owned affiliate, RXi Pharmaceuticals Corporation. He previously served as Director and Chairman of Global 
Genomics  from  June  2000.  Mr.  Kriegsman  is  an  inactive  Chairman  and  Founder  of  Kriegsman  Capital  Group  LLC,  a  financial 
advisory firm specializing in the development of alternative sources of equity capital for emerging growth companies in the healthcare 
industry.  He  has  advised  such  companies  as  SuperGen  Inc.,  Closure  Medical  Corporation,  Novoste  Corporation,  Miravant  Medical 
Technologies, and Maxim Pharmaceuticals. In the past five years, Mr. Kriegsman has also served on the Board of Directors of Bradley 
Pharmaceuticals, Inc. and Hythiam, Inc. Mr. Kriegsman has a BS degree with honors from New York University in Accounting and 

44 

 
  
  
 
 
 
 
 
  
  
completed the Executive Program in Mergers and Acquisitions at New York University, The Management Institute. Mr. Kriegsman is 
a graduate of the Stanford Law School Directors’ College. Mr. Kriegsman was formerly a Certified Public Accountant with KPMG in 
New  York  City.  In  February  2006,  Mr.  Kriegsman  received  the  Corporate  Philanthropist  of  the  Year  Award  from  the  Greater  Los 
Angeles  Chapter  of  the  ALS  Association  and  in  October  2006,  he  received  the  Lou  Gehrig  Memorial  Corporate  Award  from  the 
Muscular  Dystrophy  Association.  Mr.  Kriegsman  has  been  a  guest  speaker  and  lecturer  at  various  universities  including  California 
Institute of Technology (Caltech), Brown University, and New York University. Mr. Kriegsman has been active in various charitable 
organizations  including  the  Biotechnology  Industry  Organization,  the  ALS  Association,  the  Los  Angeles  Venture  Association,  the 
Southern California Biomedical Council, and the Palisades-Malibu YMCA. 

Marvin R. Selter has been a director since October 2003. He has been President and Chief Executive Officer of CMS, Inc. since 
he  founded  that  firm  in  1968.  CMS,  Inc.  is  a  national  management  consulting  firm.  In  1972,  Mr.  Selter  originated  the  concept  of 
employee leasing. He served as a member of the Business Tax Advisory Committee—City of Los Angeles, Small Business Board—
State of California and the Small Business Advisory Commission—State of California. Mr. Selter also serves on the Valley Economic 
Development Center as past Chairman and Audit Committee Chairman, the Board of Valley Industry and Commerce Association as 
past Chairman, the Advisory Board of the San Fernando Economic Alliance and the California State University—Northridge as Past 
Chairman of the Economic Research Center and President of the Olive View UCLA Medical Center Foundation. He has served, and 
continues  to  serve,  as  a  member  of  boards  of  directors  of  various  hospitals,  universities,  private  medical  companies  and  other 
organizations. Mr. Selter attended Rutgers—The State University, majoring in Accounting and Business Administration. He was an 
LPA  having  served  as  Controller,  Financial  Vice  President  and  Treasurer  at  distribution,  manufacturing  and  service  firms.  He  has 
lectured extensively on finance, corporate structure and budgeting for the American Management Association and other professional 
teaching associations. 

Mr. Selter has founded, operated, and grown his own successful businesses, which gives him a valuable insight into the financial 
constraints  and  operational  challenges  facing  companies  in  the  development  stage  and  as  they  mature.  He  also  has  many  years  of 
involvement  in  various  governmental  agencies  and  charitable  organizations,  which  affords  him  an  important  perspective  on  the 
business regulatory process and capital-raising activities. In addition, he has significant education and work experience in accounting 
and financial matters that he is able to utilize as the named financial expert on our Audit Committee. 

Louis Ignarro, Ph.D. has been a director since July 2002. He previously served as a director of Global Genomics since November 
20, 2000. Dr. Ignarro serves as the Jerome J. Belzer, M.D. Distinguished Professor of Pharmacology in the Department of Molecular 
and Medical Pharmacology at the UCLA School of Medicine. Dr. Ignarro has been at the UCLA School of Medicine since 1985 as a 
professor, acting chairman and assistant dean. Dr. Ignarro received the Nobel Prize for Medicine in 1998. Dr. Ignarro received a B.S. 
in  pharmacy  from  Columbia  University  and  his  Ph.D.  in  Pharmacology  from  the  University  of  Minnesota.  Dr.  Ignarro  is  a  Nobel 
Laureate and an esteemed medical researcher whose experience enables him to offer importance scientific guidance to our Board of 
Directors. 

Joseph Rubinfeld, Ph.D. has been a director since July 2002. He co-founded SuperGen, Inc. in 1991 and has served as its Chief 
Executive Officer and President and as a director since its inception until December 31, 2003. He resigned as Chairman Emeritus of 
SuperGen, Inc. on February 8, 2005. Dr. Rubinfeld was also Chief Scientific Officer of SuperGen from 1991 until September 1997. 
Dr. Rubinfeld is also a founder of JJ Pharma. Dr. Rubinfeld was one of the four initial founders of Amgen, Inc. in 1980 and served as 
a  Vice  President  and  its  Chief  of  Operations  until  1983.  From  1987  until  1990,  Dr.  Rubinfeld  was  a  Senior  Director  at  Cetus 
Corporation and from 1968 to 1980, Dr. Rubinfeld was employed at Bristol-Myers Company, International Division in a variety of 
positions.  Dr.  Rubinfeld  received  a  B.S.  degree  in  chemistry  from  C.C.N.Y.  and  an  M.A.  and  Ph.D.  in  chemistry  from  Columbia 
University. 

Dr.  Rubinfeld  served  as  a  senior  executive  of  several  large  pharmaceutical  companies  before  leaving  to  co-found  and  serve  as 
Chief Executive Officer or in other senior executive capacities with highly successful companies. Dr. Rubenfeld’s academic training 
and business experience enhances the breadth and scope of our Board’s oversight of our company’s management, business, strategic 
relationships, and other activities, while his vision adds to the long-range planning of our Board of Directors and management. 

Richard L. Wennekamp has been a director since October 2003. He retired from Community Bank in June 2008 where he was the 
Senior Vice President-Credit Administration since October 2002. From September 1998 to July 2002, Mr. Wennekamp was an executive 
officer of Bank of America Corporation, holding various positions, including Managing Director-Credit Product Executive for the last 
four years of his 22-year term with the bank. From 1977 through 1980, Mr. Wennekamp was a Special Assistant to former President of 
the United States, Gerald R. Ford, and the Executive Director of the Ford Transition Office. Prior thereto, he served as Staff Assistant to 
the President of the United States for one year, and as the Special Assistant to the Assistant Secretary of Commerce of the U.S.

45 

  
  
  
  
  
  
Mr.  Wennekamp’s  senior  executive  experience  in  the  banking  and  financial  services  industry  sets  him  apart  from  our  other 
directors and adds unique capabilities and a different perspective to the deliberations of our Board of Directors. As a former  Chief 
Credit  Officer at  Bank  of America  and  Community  Bank,  he  understands  the  credit  needs, financing  requirements,  and operational 
constraints of development-stage and mature businesses. 

Daniel Levitt, M.D., Ph.D. joined us in October 2009 as our Chief Medical Officer. Dr. Levitt brings more than 24 years of senior 
management  experience,  having  spearheaded  numerous  drug  development  programs  to  commercialization  at  leading  biotechnology 
and  pharmaceutical  companies.  Prior  to  joining  CytRx,  Dr.  Levitt  served  from  January  2007  to  February  2009  as  Executive  Vice 
President, Research and Development at Cerimon Pharmaceuticals, Inc. Prior to that, from August 2003 to April 2006, he was Chief 
Medical Officer and Head of Clinical and Regulatory Affairs at Dynavax Technologies Corporation, managing clinical trials for four 
programs and overseeing multi-country regulatory strategies. From August 2002 to July 2003, Dr. Levitt was Chief Operating Officer 
and Head of Research and Development at Affymax, Inc., and prior to that he spent six years at Protein Design Labs, Inc., completing 
his tenure as that firm’s President and Head of Research and Development. Dr. Levitt’s past experience includes a position as Head of 
Drug  Development  at  Geron  Corporation,  and  Head  of  the  Cytokine  Development  Unit  and  Global  Clinical  Oncology  at  Sandoz 
Pharmaceuticals Ltd., and as Director, Clinical Oncology and Immunology at Hoffmann-LaRoche, Inc. Dr. Levitt graduated Magna 
Cum Laude and Phi Beta Kappa with a Bachelor of Arts degree from Brandeis University. He earned both his M.D. and his Ph.D. in 
Biology from the University of Chicago Pritzker School of Medicine. Dr. Levitt has received 10 major research awards and authored 
or co-authored nearly 200 papers and abstracts. 

John  Y.  Caloz  joined  us  in  October  2007  as  our  Chief  Accounting  Officer.  In  January  of  2009  Mr.  Caloz  was  named  Chief 
Financial Officer. He has a history of providing senior financial leadership in the life sciences sector, as Chief Financial Officer of 
Occulogix,  Inc,  a  NASDAQ  listed,  a  medical  therapy  company.  Prior  to  that,  Mr.  Caloz  served  as  Chief  Financial  Officer  of  IRIS 
International Inc., a Chatsworth, CA based medical device manufacturer. He served as Chief Financial Officer of San Francisco-based 
Synarc, Inc., a medical imaging company, and from 1993 to 1999 he was Senior Vice President, Finance and Chief Financial Officer 
of Phoenix International Life Sciences Inc. of Montreal, Canada, which was acquired by MDS Inc. in 1999. Mr. Caloz was a partner at 
Rooney,  Greig,  Whitrod,  Filion  &  Associates  of  Saint  Laurent,  Quebec,  Canada,  a  firm  of  Chartered  Accountants  specializing  in 
research  and  development  and  high  tech  companies,  from  1983  to  1993.  Mr.  Caloz,  a  Chartered  Accountant,  holds  a  degree  in 
Accounting from York University, Toronto, Canada. 

Scott  Wieland,  Ph.D,  joined  CytRx  in  2005  as  the  Vice  President,  Clinical  and  Regulatory  Affairs  and  was  promoted  to  the 
position of Senior Vice President, Drug Development in December 2008. Prior to that, he served in senior level positions in the areas 
of Drug Development, Clinical and Regulatory Affairs at various biotech firms. He spent five years at NeoTherapeutics, Inc. serving 
as the Director of Product Development and was later promoted to Vice President of Product Development. From 1990 to 1997, he 
served  as Director of  Regulatory Affairs  at  CoCensys, Inc.  Dr. Wieland  has  a  Ph.D.  in  Biopsychology  and  an  M.A.  in  Psychology 
from the University of Arizona. He has an MBA from Webster University. Dr. Wieland received his B.S. in Physiological Psychology 
from the University of California, Santa Barbara. 

Scott  Geyer  joined  CytRx  in  November  2009  as  our  Senior  Vice  President,  Manufacturing.  Prior  to  joining  CytRx,  he  served 
since  May  2009,  and  also  from  May  2007  through  November  2008,  as  Vice  President,  Technical  Operations  at  Cerimon 
Pharmaceuticals, Inc. He previously served from December 2008 through April 2009 as Senior Vice President, Technical Operations 
&  Product  Development  at  TRF  Pharma,  Inc.,  from  October  2004  through  April  2007  as  Vice  President,  Technical  Operation  at 
Xencor, Inc., and from October 2003 through February 2004 as Vice President, Manufacturing and Process Development at BioMarin 
Pharmaceuticals Inc. Mr. Geyer's past experience includes holding senior positions at Onyx Pharmaceuticals and Protein Design Labs, 
Inc.,  as  well  as  positions  at  Ares-Sorono  Group  and  SmithKline  Beckman,  among  others.  Mr.  Geyer  has  co-authored  numerous 
publications  in  peer-reviewed  journals.  He  holds  an  M.S.  in  veterinary  microbiology  from  Texas  A&M  University  and  a  B.S.  in 
microbiology from the University of Southwestern Louisiana 

Benjamin S. Levin, has been our General Counsel, Vice President — Legal Affairs and Corporate Secretary since July 2004. From 
November 1999 to June 2004, Mr. Levin was an associate in the transactions department of the Los Angeles office of O’Melveny & 
Myers LLP. Mr. Levin received his S.B. in Economics from the Massachusetts Institute of Technology, and a J.D. from Stanford Law 
School. 

David  J.  Haen  joined  CytRx  in  October  2003  as  Director  of  Business  Development  and  was  promoted  to  Vice  President  of 
Business Development in December 2007. From 1999 to 2003, Mr. Haen worked as an associate for Kriegsman Capital Group LLC, a 
financial advisory firm focused on emerging companies in the life sciences field. Mr. Haen received a B.A. in Communications and 
Business from Loyola Marymount University. 

46 

  
  
  
  
  
  
 
Diversity 

Our board of directors, acting through the Nomination and Governance Committee, is responsible for assembling for shareholder 
consideration a group of director-nominees that, taken together, have the experience, qualifications, attributes, and skills appropriate 
for functioning effectively as a board. The Nomination and Governance Committee periodically reviews the composition of the board 
of directors in light of the company’s changing requirements, its assessment of the board of directors’ performance, and the input of 
shareholders and other key constituencies. The Nomination and Governance Committee looks for certain characteristics common to 
all board members, including integrity, strong professional reputation and record of achievement, constructive and collegial personal 
attributes,  and  the  ability  and  commitment  to  devote  sufficient  time  and  energy  to  board  service.  In  addition,  the  Nomination  and 
Governance Committee seeks to include on the board of directors a complementary mix of individuals with diverse backgrounds and 
skills reflecting the broad set of challenges that the board of directors confronts. These individual qualities can include matters such as 
experience  in  the  company’s  industry,  technical  experience  (i.e.,  medical  or  research  expertise),  experience  gained  in  situations 
comparable to the company’s, leadership experience, and relevant geographical diversity. 

Committees 

Our business, property and affairs are managed by or under the direction of the board of directors. Members of the board are kept 
informed of our business through discussion with the chief executive and financial officers and other officers, by reviewing materials 
provided to them and by participating at meetings of the board and its committees. 

Our  board  of  directors  currently  has  three  committees.  The  Audit  Committee,  Compensation  Committee,  and  Nomination  and 
Governance Committee consist of Messrs. Selter, Link, and Wennekamp. Such committees operate under a formal charter, copies of 
which are available on our website at www.cytrx.com, that governs their duties and conduct. 

Our board of directors has determined that Mr. Selter, one of the independent directors serving on our Audit Committee, is an 
“audit committee financial expert” as defined by the SEC’s rules. Our board of directors has determined that Messrs. Link, Selter and 
Wennekamp are “independent” under the current independence standards of both The NASDAQ Capital Market and the SEC. 

Section 16(a) Beneficial Ownership Reporting Compliance 

Our executive officers and directors and any person who owns more than 10% of our outstanding shares of common stock are 
required under Section 16(a) of the Securities Exchange Act to file with the SEC initial reports of ownership and reports of changes in 
ownership of our common stock and to furnish us with copies of those reports. Based solely on our review of copies of reports we 
have  received  and  written  representations  from  certain  reporting  persons,  we  believe  that  our  directors  and  executive  officers  and 
greater than 10% shareholders for 2009 complied with all applicable Section 16(a) filing requirements. 

Code of Ethics 

We  have  adopted  a  Code  of  Ethics  applicable  to  all  employees,  including  our  principal  executive  officer,  principal  financial 
officer, and principal accounting officer or controller, a copy of which is available on our website at www.cytrx.com. We will furnish, 
without charge, a copy of our Code of Ethics upon request. Such requests should be directed to Attention: Corporate Secretary, 11726 
San Vicente Boulevard, Suite 650, Los Angeles, California, or by telephone at 310-826-5648. 

Board Leadership Structure 

Our Board has placed the responsibilities of Chairman with an independent nonexecutive member of the Board, which we believe 
provides  better  accountability  between  the  Board  and  our  management  team.  We  believe  it  is  beneficial  to  have  an  independent 
Chairman  whose  sole  responsibility  to  us  is  guiding  our  Board  members  as  they  provide  leadership  to  our  executive  team.  Our 
Chairman is responsible for communication among the directors; setting the Board meeting agendas in consultation with the President 
and Chief Executive Officer; and presiding at Board meetings, executive sessions and stockholder meetings. This delineation of duties 
allows  the  President  and  Chief  Executive  Officer  to  focus  his  attention  on  managing  the  day-to-day  business  of  the  company.  We 
believe  this  structure  provides  strong  leadership  for  our  Board,  while  positioning  our  President  and  Chief  Executive  Officer  as  the 
leader of the company in the eyes of our employees and other stakeholders. 

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Board of Directors Role in Risk Oversight 

In connection with its oversight responsibilities, our board of directors, including the Audit Committee, periodically assesses the 
significant risks that we face. These risks include, but are not limited to, financial, technological, competitive, and operational risks. 
Our board of directors administers its risk oversight responsibilities through our Chief Executive Officer and Chief Financial Officer, 
who review and assess the operations of our business as well as operating management’s identification, assessment and mitigation of 
the material risks affecting our operations. 

Item 11. EXECUTIVE COMPENSATION 

Compensation Discussion and Analysis 

Overview of Executive Compensation Program 

The  Compensation  Committee  of  our  board  of  directors  has  responsibility  for  establishing,  implementing  and  monitoring  our 
executive compensation program philosophy and practices. The Compensation Committee seeks to ensure that the total compensation 
paid to our named executive officers is fair, reasonable and competitive. Generally, the types of compensation and benefits provided to 
the named executive officers are similar to those provided to our other officers. 

Throughout this Annual Report, the individuals included in the Summary Compensation Table on page 53 are referred to as the 

“named executive officers.” 

Compensation Philosophy and Objectives 

The  components  of  our  executive  compensation  consist  of  salary,  annual  cash  bonuses  awarded  based  on  the  Compensation 
Committee’s  subjective  assessment  of  each  individual  executive’s  job  performance,  including  evaluations  of,  during  the  past  year, 
stock option grants to provide executives with longer-term incentives, and occasional special compensation awards (either cash, stock 
or stock options) to reward extraordinary efforts or results. 

The  Compensation  Committee  believes  that  an  effective  executive  compensation  program  should  provide  base  annual 
compensation that is reasonable in relation to individual executive’s job responsibilities and reward the achievement of both annual 
and long-term strategic goals of our company. The Compensation Committee uses annual and other periodic cash bonuses to reward 
an  officer’s  achievement  of  specific  goals,  including  goals  related  to  the  development  of  the  product’s  drug  candidates  and 
management  of  working  capital,  and  employee  stock  options  as  a  retention  tool  and  as  a  means  to  align  the  executive’s  long-term 
interests with those of our stockholders, with the ultimate objective of affording our executives an appropriate incentive to improve 
stockholder value. The Compensation Committee evaluates both performance and compensation to maintain our company’s ability to 
attract  and  retain  excellent  employees  in  key  positions  and  to  assure  that  compensation  provided  to  key  employees  remains 
competitive  relative  to  the  compensation  paid  to  similarly  situated  executives  of  comparable  companies.  To  that  end,  the 
Compensation Committee believes executive compensation packages provided by us to our named executive officers should include 
both cash compensation and stock options. 

Because  of  the  size  of  our  company,  the  small  number  of  executive  officers  in  our  company,  and  our  company’s  financial 
priorities,  the  Compensation  Committee  has  not  implemented  any  pension  benefits,  deferred  compensation  plans,  or  other  similar 
plans for our named executive officers. 

As a biopharmaceutical company engaged in developing potential products that, to date, have not generated significant revenues 
and  are  not  expected  to  generate  significant  revenues  or  profits  for  several  years,  the  Compensation  Committee  also  takes  the 
company’s  financial  and  working  capital  condition  into  account  in  its  compensation  decisions.  Accordingly,  the  Compensation 
Committee  recently  has  weighted  bonuses  more  heavily  with  stock  options  rather  than  cash.  The  Compensation  Committee  may 
periodically reassess the proper weighting of equity and cash compensation in light of the company’s working capital situation from 
time to time. 

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Role of Executive Officers in Compensation Decisions 

The  Compensation  Committee  makes  all  compensation  decisions  for 

the  named  executive  officers  and  approves 
recommendations  made  by  our  President  and  Chief  Executive  Officer  regarding  equity  awards  to  our  other  officers.  Decisions 
regarding the non-equity compensation of our other officers are made by our President and Chief Executive Officer. 

The  Compensation  Committee  and  the  President  and  Chief  Executive  Officer  annually  review  the  performance  of  each  named 
executive officer (other than the President and Chief Executive Officer, whose performance is reviewed only by the Compensation 
Committee). The conclusions reached and recommendations based on these reviews, including with respect to salary adjustments and 
annual  award amounts,  are presented  to  the  Compensation  Committee.  The  Compensation  Committee  can  exercise  its  discretion  in 
modifying or declining any recommended adjustments or awards to executives. 

Setting Executive Compensation 

Based on the foregoing objectives, the Compensation Committee has structured the company’s annual cash and incentive-based cash 
and non-cash executive compensation to seek to motivate our named executives to achieve the company’s business goals, including goals 
related to the development of the our drug candidates and management of working capital, to reward the executives for achieving such 
goals,  and  to  retain  the  executives.  In  doing  so,  the  Compensation  Committee  historically  has  not  employed  outside  compensation 
consultants. However, during 2009, the Compensation Committee obtained two third-party industry compensation surveys and used them 
in  its  compensation  deliberations  regarding  cash  and  equity  compensation  for  our  executive  officers.  The  Compensation  Committee 
utilized this data to set compensation for our executive officers at levels targeted at or around the third quartile of compensation amounts 
provided to executives at comparable companies considering each individual’s individual experience level related to their position with 
us. There is no pre-established policy or target for the allocation between either cash and non-cash incentive compensation. 

2009 Executive Compensation Components 

For 2009, the principal components of compensation for the named executive officers were: 

• 

• 

• 

base salary; 

annual and special bonuses; and 

equity incentive compensation. 

Base Salary 

The Company provides named executive officers and other employees with base salary to compensate them for services rendered 
during the year. Base salary ranges for the named executive officers are determined for each named executive officer based on his 
position and responsibility. 

During its review of base salaries for executives, the Compensation Committee primarily considers: 

• 

• 

• 

• 

the negotiated terms of each executive’s employment agreement, if any; 

an internal review of the executive’s compensation, both individually and relative to other named executive officers; 

each executive’s individual performance; and 

base salaries paid by comparable companies. 

Salary levels are typically considered annually as part of the company’s performance review process, as well as upon a change in 
job  responsibility.  Merit-based  increases  to  salaries  are  based  on  the  company’s  available  resources  and  the  Compensation 
Committee’s assessment of the individual’s performance. Both assessments are based upon written evaluations of such criteria as job 
knowledge, communication, problem solving, initiative, goal-setting, and expense management. Base salaries for the named executive 
officers  in  2009  were  increased  from  the  base  salaries  in  effect  during  the  prior  year  by  amounts  ranging  from  15%  for  our  Vice 
President – Legal Affairs and our Senior Vice President – Drug Development, to 18% for our President and Chief Executive Officer 
and our Chief Financial Officer. 

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Annual and Special Bonuses 

The Compensation Committee has not established an incentive compensation program with fixed performance targets. Because 
we  do  not  generate  significant  revenues  and  have  not  commercially  released  any  products,  the  Compensation  Committee  bases  its 
discretionary compensation awards on the achievement of product development targets and milestones, efforts related to extraordinary 
transactions, effective fund-raising efforts, and effective management of personnel and capital resources, among other criteria. During 
2009, the Compensation Committee granted Mr. Kriegsman an annual cash bonus of $450,000, and granted cash bonuses to the other 
named executive officers ranging from $0 to $80,000, principally based on their efforts in helping us advance the development of our 
products and raise capital. 

Equity Incentive Compensation 

As indicated above, the Compensation Committee also aims to encourage the company’s executive officers to focus on long-term 
company  performance  by  allocating  to  them  stock  options  that  vest  over  a  period  of  several  years.  In  2009,  the  Compensation 
Committee granted to Mr. Kriegsman nonqualified options to purchase 750,000 shares of our common stock at a price of $1.05 per 
share,  which  equaled  the  closing  market  price  on  the  date  of  grant.  The  option  vests  monthly  over  three  years,  provided  that  Mr. 
Kriegsman continues in our employ through such monthly vesting periods. In addition, in connection with the annual review of our 
other  named  executive  officers,  the  Compensation  Committee  also  granted  stock  options  to  those  named  executive  officers.  All  of 
these other stock options had an exercise price equal to the closing market price on the date of grant, and also vest monthly over three 
years, provided that such executives remain in our employ through such monthly vesting periods. 

Retirement Plans, Perquisites and Other Personal Benefits 

We have adopted a tax-qualified employee savings and retirement plan, the 401(k) Plan, for eligible U.S. employees, including 
our named executive officers. Eligible employees may elect to defer a percentage of their eligible compensation in the 401(k) Plan, 
subject to the statutorily prescribed annual limit. We may make matching contributions on behalf of all participants in the 401(k) Plan 
in  an  amount  determined  by  our  board  of  directors.  We  did  not  make  any  matching  contribution  to  the  401(k)  Plan  for  2009.  
Matching and profit-sharing contributions, if any, are subject to a vesting schedule; all other contributions are at all times fully vested. 
We intend the 401(k) Plan, and the accompanying trust, to qualify under Sections 401(k) and 501 of the Internal Revenue Code so that 
contributions by employees to the 401(k) Plan, and income earned (if any) on plan contributions, are not taxable to employees until 
withdrawn from the 401(k) Plan, and so that we will be able to deduct our contributions, if any, when made. The trustee under the 
401(k) Plan, at the direction of each participant, may invest the assets of the 401(k) Plan in any of a number of investment options. 

We  do  not  provide  any  of  our  executive  officers  with  any  other  perquisites  or  personal  benefits,  other  than  benefits  to  Mr. 
Kriegsman  provided  for  in  his  employment  agreement.  As  required  by  his  employment  agreement,  during  2009  we  paid  insurance 
premiums  with  respect  to  a  life  insurance  policy  for  Mr.  Kriegsman  which  had  a  face  value  of  approximately  $1.4  million  as  of 
December 31, 2009 and under which Mr. Kriegsman’s designee is the beneficiary. 

Employment Agreements and Severance Arrangements 

We  have  entered  into  written  employment  agreements  with  each  of  our  named  executive  officers.  The  main  purpose  of  these 
agreements is to protect the company from business risks such  as competition for the executives’ service, loss of confidentiality  or 
trade  secrets,  and  solicitation  of  our  other  employees,  and  to  define  our  right  to  terminate  the  employment  relationship.  The 
employment  agreements  also  protect  the  executive  from  termination  without  “cause”  (as  defined)  and,  in  Mr.  Kriegsman’s  case, 
entitles  him  to  resign  for  “good  reason”  (as  defined).  Each  employment  agreement  was  individually  negotiated,  so  there  are  some 
minor  variations  in  the  terms  among  executive  officers.  Generally  speaking,  however,  the  employment  agreements  provide  for 
termination  and  severance  benefits  that  the  Compensation  Committee  believes  are  consistent  with  industry  practices  for  similarly 
situated executives. The Compensation Committee believes that the termination and severance benefits help the company retain the 
named executive officers by providing them with a competitive employment arrangement and protection against unknowns such as 
termination without “cause” that go along with the position. 

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In  the  event of  termination  without  “cause,”  the named  executive officers  will be  entitled  to  a  lump-sum  payment  equal  to six 
months  of  base  salary  (24  months  in  the  case  of  Mr.  Kriegsman).  Mr.  Kriegsman’s  employment  agreement  also  provides  for  our 
continuation  of  Mr.  Kriegsman’s  life  insurance  and  medical  benefits  during  his  24-month  severance  period.  If  Mr.  Kriegsman’s 
employment is terminated by us without “cause,” or by Mr. Kriegsman for “good reason,” within two years following a change of 
control of CytRx, he also would be entitled under his employment agreement to receive a “gross-up” payment equal to the sum of any 
excise tax on his termination benefits (including any accelerated vesting of his options under our Plans as described below) plus any 
penalties and interest. 

Change of Control Arrangements 

The company’s 2000 Long-Term Incentive Plan and 2008 Stock Incentive Plan provide generally that, upon a change of control 
of CytRx, all unvested stock options and awards under the Plans held by plan participants, including the named executive officers, will 
become immediately vested and exercisable immediately prior to the effective date of the transaction. The Compensation Committee 
believes  that  such  “single  trigger”  change  of  control  policy  is  consistent  with  the  objective  of  aligning  the  interests  of  the  named 
executive officer’s and of the company’s stockholders by allowing the executives to participate equally with stockholders in the event 
of a change of control transaction. 

The foregoing severance and change of control arrangements, including the quantification of the payment and benefits provided 
under these arrangements, are described in more detail elsewhere in this Annual Report under the heading “Executive Compensation – 
Potential Payments Upon Termination or Change of Control.” 

Ownership Guidelines 

The Compensation Committee has no requirement that each named executive officer maintain a minimum ownership interest in 

our company. 

Our  long-term  incentive  compensation  consists  solely  of  periodic  grants of  stock options  to our named  executive officers.  The 

stock option program: 

• 

• 

• 

links the creation of stockholder value with executive compensation; 

provides increased equity ownership by executives; 

functions as a retention tool, because of the vesting features included in all options granted by the Compensation Committee; 
and 

•  maintains competitive levels of total compensation. 

We normally grant stock options to new executive officers when they join our company based upon their position with us and 
their relevant prior experience. The options granted by the Compensation Committee generally vest monthly over the first three years 
of the ten-year option term. Vesting and exercise rights cease upon termination of employment (or, in the case of exercise rights, 90 
days  thereafter),  except  in  the  case  of  death  (subject  to  a  one-year  limitation),  disability  or  retirement.  Prior  to  the  exercise  of  an 
option, the holder has no rights as a stockholder with respect to the shares subject to such option, including voting rights and the right 
to  receive  dividends  or  dividend  equivalents.  In  addition  to  the  initial  option  grants,  our  Compensation  Committee  may  grant 
additional  options  to  retain  our  executives  and  reward,  or  provide  incentive  for,  the  achievement  of  corporate  goals  and  strong 
individual  performance.  Our  board  of  directors  has  granted  our  President  and  Chief  Executive  Officer  discretion  to  grant  up  to 
100,000 options to employees upon joining our company, and to make grants from an additional “discretionary pool” of up to 100,000 
options  during  each  annual  employee  review  cycle.  Options  are  granted  based  on  a  combination  of  individual  contributions  to  our 
company  and  on  general  corporate  achievements,  which  may  include  the  attainment  of  product  development  milestones  (such  as 
commencement and completion of clinical trials) and attaining other annual corporate goals and objectives. On an annual basis, the 
Compensation Committee assesses the appropriate individual and corporate goals for our executives and provides additional option 
grants based upon the achievement by the new executives of both individual and corporate goals. We expect that we will continue to 
provide new employees with initial option grants in the future to provide long-term compensation incentives and will continue to rely 
on  performance-based  and  retention  grants  to  provide  additional  incentives  for  current  employees.  Additionally,  in  the  future,  the 
Compensation Committee may consider awarding additional or alternative forms of equity incentives, such as grants of bonus stock, 
restricted stock and restricted stock units. 

51 

  
  
  
  
  
  
  
  
  
  
  
 
It is our policy to award stock options at an exercise price equal to The NASDAQ Capital Market’s closing price of our common 
stock on the date of the grant. In certain limited circumstances, the Compensation Committee may grant options to an executive at an 
exercise price in excess of the closing price of the common stock on the grant date. The Compensation Committee has never granted 
options  with  an  exercise  price  that  is  less  than  the  closing price  of our common  stock  on  the grant date, nor  has  it  granted options 
which are priced on a date other than the grant date. For purposes of determining the exercise price of stock options, the grant date is 
deemed to be the first day of employment for newly hired employees, or the date on which the Compensation Committee or the Chief 
Executive Officer, as applicable, approves the stock option grant to existing employees. 

We  have  no  program,  practice  or  plan  to  grant  stock  options  to  our  executive  officers,  including  new  executive  officers,  in 
coordination with the release of material nonpublic information. We also have not timed the release of material nonpublic information 
for the purpose of affecting the value of stock options or other compensation to our executive officers, and we have no plan to do so. 
We have no policy regarding the adjustment or recovery of stock option awards in connection with the restatement of our financial 
statements, as our stock option awards have not been tied to the achievement of specific financial goals. 

Tax and Accounting Implications 

Deductibility of Executive Compensation 

As part of its role, the Compensation Committee reviews and considers the deductibility of executive compensation under Section 
162(m) of the Internal Revenue Code, which provides that corporations may not deduct compensation of more than $1,000,000 that is 
paid  to  certain  individuals.  We  believe  that  compensation  paid  to  our  executive  officers  generally  is  fully  deductible  for  federal 
income tax purposes. 

Accounting for Share-Based Compensation 

Beginning on January 1, 2006, we began accounting for share-based compensation in accordance with the requirements of FASB 
Statement 123(R), Share-Based Payment. This accounting treatment has not significantly affected our compensation decisions. The 
Compensation  Committee  takes  into  consideration  the  tax  consequences  of  compensation  to  the  named  executive  officers,  but  tax 
considerations are not a significant part of the company’s compensation policy. 

Benchmarking 

The Compensation Committee does not attempt to establish or measure executive compensation against any benchmarks. With 
certain exceptions, our company’s compensation policies are not related specifically to our company’s performance, which is just one 
of  the  factors  considered  by  us  and  our  Compensation  Committee  in  establishing  base  salaries  and  awarding  discretionary 
compensation. We have not established any policy regarding recoupment, or “clawback,” of any performance-based compensation in 
the  event  our  company’s  historical  performance  is  subsequently  revised  or  restated  in  a  way  that  would  have  produced  a  lower 
compensation amount. We also have not relied upon wealth accumulation analyses, or “tally sheets,” or internal pay equity analyses in 
making executive compensation decisions. 

Compensation Committee Interlocks and Insider Participation in Compensation Decisions 

There are no “interlocks,” as defined by the SEC, with respect to any member of the Compensation Committee. Max Link, Ph.D., 

Marvin R. Selter and Richard L. Wennekamp all served as members of the Compensation Committee during 2009. 

Compensation Committee Report 

The  Compensation  Committee  has  reviewed  and  discussed  with  management  the  “Compensation  Discussion  and  Analysis” 
required by Item 402(b) of Regulation S-K and, based on such review and discussions, has recommended to our board of directors that 
the foregoing “Compensation Discussion and Analysis” be included in this Annual Report. 

Richard L. Wennekamp, Chairman 

Marvin R. Selter 

Dr. Max Link

52 

  
  
  
  
  
  
  
  
  
  
  
  
  
 
 
 
Summary Compensation Table 

The following table presents summary information concerning all compensation paid or accrued by us for services rendered in all 
capacities during 2009, 2008 and 2007 by Steven A. Kriegsman and John Y. Caloz, who are the only individuals who served as our 
principal  executive  and  financial  officers  during  the  year  ended  December  31,  2009,  and  our  three  other  most  highly  compensated 
executive officers who were serving as executive officers as of December 31, 2009: 

Name and Principal Position 
Steven A. Kriegsman 

President and Chief Executive 

Officer . . . . . . . . . . . . . . . . . . . .   

John Y. Caloz 

Chief Financial Officer and 

Treasurer . . . . . . . . . . . . . . . . . .   

Daniel Levitt, M.D., M.D., Ph.D. 

Chief Medical Officer . . . . . . . . .   

Benjamin S. Levin General 

Counsel, 
General Counsel, Vice President 
— Legal . . . . . . . . . . . . . . . . . . .   
Affairs and Secretary . . . . . . . . . . .   

Scott Wieland, Ph.D. 

Senior Vice President – Drug 

Development . . . . . . . . . . . . . . .   

____________ 

Summary Compensation Table 

Year 

Salary ($)

Bonus 
($)(1)

Option
Awards 
($) (2)

All Other
Compensation 
($)(3) 

Total 
($)

2009 
2008 
2007 

550,000     
551,000     
524,767     

450,000     
150,000     
300,000     

906,000      
517,800      
1,328,600      

10,000     
10,000     
—     

1,916,000 
1,228,800 
2,153,367 

2009 

275,000     

80,000     

137,750      

—     

492,750 

2009 

83,894     

—     

405,000      

—     

488,894 

2009 
2008 
2007 

2009 
2008 
2007 

276,000     
276,000     
250,000     

75,000     
55,000     
100,000     

119,100      
125,300      
407,000      

275,000     
255,500     
134,000     

75,000     
73,250     
35,000     

105,750      
28,580      
447,925      

—     
—     
—     

—     
—     
—     

470,100 
456,300 
730,000 

455,750 
372,480 
587,750 

(1)  Bonuses  to  the  named  executive  officers  reported  above  relating  to  2009  were  paid  in  December  2009.  Bonuses  to  the  named 
executive officers reported above relating to 2008 were paid in December 2008. Bonuses to the named executive officers reported 
above relating to 2007 were paid in April 2008. 

(2)  The values shown in this column represent the aggregate grant date fair value of equity-based awards granted during the fiscal 
year, in accordance with ASC 718, “Share Based-Payment”. At the 2009 Annual Meeting of Stockholders held on July 1, 2009, 
the Company’s stockholders approved an amendment to the Company’s 2000 Long-Term Incentive Plan to allow for a one-time 
stock option re-pricing program for employees and officers. Pursuant to the re-pricing program, 3,265,500 eligible stock options 
held by ten eligible employees and officers were amended to reduce the exercise prices of the options to $1.15 per share, which 
was the closing sale price of CytRx’s common stock as reported on The NASDAQ Capital Market on the July 1, 2009 completion 
date of the re-pricing program, and to impose a new option vesting schedule. The values in this column include the incremental 
increase in the fair value of the re-priced options over the fair value of the original award. The fair value of the stock options at 
the date of grant was estimated using the Black-Scholes option-pricing model, based on the assumptions described in Note 15 of 
the Notes to Financial Statements included in this Annual Report. 

(3)  This amount represents life insurance premiums. 

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2009 Grants of Plan-Based Awards 

In  2009,  we  granted  stock  options  to  our  named  executive  officers  under  our  2000  Long-Term  Incentive  Plan  and  2008  Stock 

Incentive Plan as follows: 

2008 Grants of Plan-Based Awards 

 Name   
Steven A. Kriegsman . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .  

President and Chief Executive Officer 

All Other 
Option Awards 
(# of CytRx 
Shares)

Exercise Price 
of 
Option Awards
($/Share)

Grant Date

12/10/2009   

750,000    $ 

1.05    $

Grant Date
Fair Value of
Option Awards
($)
609,000 

John Y. Caloz . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .  
Chief Financial Officer and Treasurer . . . . . . . . . . . . . . . .  

12/10/2009   
1/2/2009   

125,000    $ 
50,000      

1.05    $
0.30     

101,500 
11,750 

Daniel Levitt, M.D., Ph.D. . . . . . . . . . . . . . . . . . . . . . . . . . . . .  

10/12/2009   

500,000    $ 

1.06    $

405,000 

Chief Medical Officer 

Benjamin S. Levin . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .  
General Counsel, Vice President — Legal Affairs and 

Secretary 

Scott Wieland, Ph.D. . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .  

Senior Vice President – Drug Development 

____________ 

2000 Long-Term Incentive Plan and 2008 Stock Incentive Plan 

12/10/2009   

100,000    $ 

1.05    $

81,200 

12/10/2009   

100,000    $ 

1.05    $

81,200 

The purpose of our 2000 Long-Term Incentive Plan, or 2000 Plan, and our 2008 Stock Incentive Plan, or 2008 Plan, is to promote 
our success and enhance our value by linking the personal interests of our employees, officers, consultants and directors to those of 
our stockholders. The 2000 Plan was originally adopted by our Board of Directors on August 24, 2000 and by our stockholders on 
June 7, 2001, with certain amendments to the Plan having been subsequently approved by our Board of Directors and stockholders. 
On May 11, 2009, our Board of Directors approved an amendment to the 2000 Plan to allow for a one-time stock option re-pricing 
program for our employees. The 2008 Plan was adopted by our Board of Directors on November 21, 2008 and by our stockholders on 
July 1, 2009. 

2000 Plan and 2008 Plan Descriptions 

The 2000 Plan and the 2008 Plan, or the Plans, are administered by the Compensation Committee of our Board of Directors. The 

Compensation Committee has the power, authority and discretion to: 

• 

• 

• 

designate participants; 

determine the types of awards to grant to each participant and the number, terms and conditions of any award; 

establish, adopt or revise any rules and regulations as it may deem necessary or advisable to administer the Plan; and 

•  make all other decisions and determinations that may be required under, or as the Compensation Committee deems necessary 

or advisable to administer, the Plan. 

Awards 

The following is summary description of financial instruments that may be granted to participants by the Compensation Committee 

of our Board of Directors. The Compensation Committee to date has only granted stock options to participants in the Plans.

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Stock Options. The Compensation Committee is authorized to grant both incentive stock options and non-qualified stock options. 
The terms of any incentive stock option must meet the requirements of Section 422 of the Internal Revenue Code. The exercise price 
of an option may not be less than the fair market value of the underlying stock on the date of grant, and no option may have a term of 
more than 10 years from the grant date. 

Stock Appreciation Rights. The Compensation Committee may grant stock appreciation rights to participants. Upon the exercise 
of a stock appreciation right, the participant has the right to receive the excess, if any, of (1) the fair  market value of one share of 
common  stock  on  the  date  of  exercise,  over  (2)  the  grant  price  of  the  stock  appreciation  right  as  determined  by  the  Compensation 
Committee, which will not be less than the fair market value of one share of common stock on the date of grant. 

Restricted Stock. The Compensation Committee may make awards of restricted stock, which will be subject to such restrictions 
on  transferability  and  other  restrictions  as  the  Compensation  Committee  may  impose  (including  limitations  on  the  right  to  vote 
restricted stock or the right to receive dividends, if any, on the restricted stock). 

Performance  Units.  The  Compensation  Committee  may  grant  under  the  2000  Plan  performance  units  on  such  terms  and 
conditions as may be selected by the Compensation Committee. The Compensation Committee will have the complete discretion to 
determine the number of performance units granted to each participant and to set performance goals and other terms or conditions to 
payment  of  the  performance  units  which,  depending  on  the  extent  to  which  they  are  met,  will  determine  the  number  and  value  of 
performance units that will be paid to the participant. 

Dividend  Equivalents.  The  Compensation  Committee  is  authorized  to  grant  under  the  2000  Plan  dividend  equivalents  to 
participants subject to such terms and conditions as may be selected by the Compensation Committee. Dividend equivalents entitle the 
participant to receive payments equal to dividends with respect to all or a portion of the number of shares of common stock subject to 
an option or other award, as determined by the Compensation Committee. The Compensation Committee may provide that dividend 
equivalents  be  paid  or  distributed  when  accrued  or  be  deemed  to  have  been  reinvested  in  additional  shares  of  common  stock,  or 
otherwise reinvested. 

Other  Stock-Based  Awards.  The  Compensation  Committee  may  grant  other  awards  under  the  2000  Plan  that  are  payable  in, 
valued  in  whole  or  in  part  by  reference  to,  or  otherwise  based  on  or  related  to  shares  of  common  stock,  as  deemed  by  the 
Compensation  Committee  to  be  consistent  with  the  purposes  of  the  2000  Plan.  These  stock-based  awards  may  include  shares  of 
common stock awarded as a bonus and not subject to any restrictions or conditions, convertible or exchangeable debt securities, other 
rights convertible or exchangeable into shares of common stock, and awards valued by reference to book value of shares of common 
stock or the value of securities of or the performance of our subsidiaries. The Compensation Committee will determine the terms and 
conditions of any such awards. 

Performance Goals. The Compensation Committee in its discretion may determine awards under the 2000 Plan based on: 

• 

the achievement by CytRx or a parent or subsidiary of a specific financial target; 

•  CytRx’s stock price; 

• 

• 

• 

the achievement by an individual or a business unit of CytRx or a subsidiary of a specific financial target; 

the achievement of specific goals with respect to (i) product development milestones, (ii) corporate financings, (iii) merger 
and acquisition activities, (iv) licensing transactions, (v) development of strategic partnerships or alliances, or (vi) acquisition 
or development of new technologies; and 

any combination of the goals set forth above. 

The Compensation Committee has the right for any reason to reduce (but not increase) any award, even if a specific goal has been 
achieved. If an award is made on the basis of the achievement of a goal, the Compensation Committee must have established the goal 
before the beginning of the period for which the performance goal relates (or a later date as may be permitted under Internal Revenue 
Code  Section  162(m)).  Any  payment  of  an  award  for  achieving  a  goal  will  be  conditioned  on  the  written  certification  of  the 
Compensation Committee in each case that the goals and any other material conditions were satisfied. 

55 

  
  
  
  
  
  
  
  
  
  
  
  
 
 
Limitations on Transfer; Beneficiaries. Awards under the Plans may not be transferred or assigned by participants other than by 
will or the laws of descent and distribution and, in the case of an incentive stock option, pursuant to a qualified domestic relations 
order,  provided  that  the  Compensation  Committee  may  (but  need  not)  permit  other  transfers  where  the  Compensation  Committee 
concludes that such transferability (1) does not result in accelerated taxation, (2) does not cause any option intended to be an incentive 
stock option to fail to qualify as such, and (3) is otherwise appropriate and desirable, taking into account any factors deemed relevant, 
including any state or federal tax or securities laws or regulations applicable to transferable awards. A participant may, in the manner 
determined by the Compensation Committee, designate a beneficiary to exercise the participant’s rights and to receive any distribution 
with respect to any award upon the participant’s death. 

Acceleration  Upon  Certain  Events.  In  the  event  of  a  “Change  in  Control”  of  CytRx,  which  is  a  term  defined  in  the  Plans,  all 
outstanding options and other awards in the nature of rights that may be exercised will become fully vested and exercisable and all 
restrictions  on  all  outstanding  awards  will  lapse.  The  Compensation  Committee  may,  however,  in  its  sole  discretion  declare  all 
outstanding options, stock appreciation rights and other awards in the nature of rights that may be exercised to become fully vested 
and exercisable, and all restrictions on all outstanding awards to lapse, in each case as of such date as the Compensation Committee 
may, in its sole discretion, declare. The Compensation Committee may discriminate among participants or among awards in exercising 
such discretion. 

Termination and Amendment 

Our Board of Directors or the Compensation Committee may, at any time and from time to time, terminate or amend the Plans 
without stockholder approval; provided, however, that our board or the Compensation Committee may condition any amendment on 
the approval of our stockholders if such approval is necessary or deemed advisable with respect to tax, securities or other applicable 
laws, policies or regulations. No termination or amendment of the Plans may adversely affect any award previously granted without 
the  written  consent  of  the  participants  affected.  The  Compensation  Committee  may  amend  any  outstanding  award  without  the 
approval of the participants affected, except that no such amendment may diminish the value of an award determined as if it has been 
exercised, vested, cashed in or otherwise settled on the date of such amendment, and, except as otherwise permitted in the Plan, the 
exercise price of any option may not be reduced and the original term of any option may not be extended. 

56 

  
  
  
 
 
Holdings of Previously Awarded Equity 

Equity awards held as of December 31, 2009 by each of our named executive officers were issued under our 2000 Plan, except for 
the most recent equity award to Mr. Kriegsman, which was issued under our 2008 Plan. The following table sets forth outstanding 
equity awards held by our named executive officers as of December 31, 2009: 

2009 Outstanding Equity Awards at Fiscal Year-End 

Option Awards 

Number of Securities
Underlying Unexercised Options (#)

Option Exercis 
Price (3) 
($) 

Option Expiration

Date

Name  
Steven A. Kriegsman . . . . . . . . . . . . . . . . . . . . . . .       
President and Chief Executive Officer . . . . . .       

   Exercisable

—     
99,972     
250,056     
252,805     
200,000     
300,000     
250,000     
750,000     

—     
15,288     
8,335     
8,335     
25,005     

Unexercisable
(1)    
(1)    
(1)    
(1)    
(1)    
(1)    
(2)    
(2)    

(1)    
(1)    
(2)    
(2)    
(2)    

750,000     
200,028     
199,944     
97,195     
—     
—     
—     
—     

125,000     
34,713     
16,665     
16,665     
49,995     

John Y. Caloz . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .       
Chief Financial Officer and Treasurer . . . . . .       

Daniel Levitt, M.D., Ph.D. . . . . . . . . . . . . . . . . . .       

27,910     

(1)    

472,090     

Chief Medical Officer 

Benjamin S. Levin . . . . . . . . . . . . . . . . . . . . . . . . . .       
General Counsel, Vice President — Legal . .       
Affairs and Secretary . . . . . . . . . . . . . . . . . . . . .       

Scott Wieland, Ph.D. . . . . . . . . . . . . . . . . . . . . . . . .       
Senior Vice President – Drug Development .       

____________ 

—     
36,100     
30,575     
72,230     
90,000     
150,000     
160,000     

—     
8,335     
8,335     
50,000     

(1)    
(1)    
(1)    
(1)    
(1)    
(1)    
(2)    

(1)    
(2)    
(2)    
(2)    

100,000     
63,900     
69,425     
27,770     
—     
—     
—     

100,000     
16,665     
16,665     
25,000     

1.05  
0.37  
1.15  
1.15  
1.15  
0.79  
1.15  
1.15  

1.05  
0.30  
1.15  
1.15  
1.15  

1.06  

1.05  
0.37  
1.15  
1.15  
1.15  
0.79  
1.15  

1.05  
1.15  
1.15  
1.15  

12/10/19
11/21/18
4/07/18
4/18/17
6/16/16
5/17/15
6/19/13
6/20/13

12/10/19
01/02/19
04/07/18
12/06/17
10/26/17

11/21/18

12/10/19
11/21/18
4/07/18
4/18/17
6/16/16
5/17/15
7/15/14

12/10/19
11/21/18
12/06/17
4/30/17

(1)  These options vest in 36 equal monthly installments, subject to the option holder’s remaining in our continuous employ through 

such dates. 

(2)  These options vest in three annual installments, subject to the option holder’s remaining in our continuous employ through such 

dates. 

(3)  The reported options with prices of $1.15 were re-priced to that exercise price on July 1, 2009 at $1.15. 

Option Exercises and Stock Vested 

There were no exercises of stock options by any of our named executive officers during 2009. 

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Employment Agreements and Potential Payment upon Termination or Change in Control 

Employment Agreement with Steven A. Kriegsman 

Mr.  Kriegsman  is  employed  as  our  Chief  Executive  Officer  and  President  pursuant  to  an  employment  agreement  that  was 
amended as of May 2009 to continue through December 31, 2012. The employment agreement will automatically renew in December 
2012 for an additional one-year period, unless either Mr. Kriegsman or we elect not to renew it. 

Under his employment agreement as amended, Mr. Kriegsman is entitled to receive an annual base salary of $650,000. Our board 
of directors (or its Compensation Committee) will review the base salary annually and may increase (but not decrease) it in its sole 
discretion.  In  addition  to  his  annual  salary,  Mr.  Kriegsman  is  eligible  to  receive  an  annual  bonus  as  determined  by  our  board  of 
directors  (or  its  Compensation  Committee)  in  its  sole  discretion,  but  not  to  be  less  than  $150,000.  Pursuant  to  his  employment 
agreement with us, we have agreed that he shall serve on a full-time basis as our Chief Executive Officer and President and that he 
may continue to serve as Chairman of the Kriegsman Group only so long as necessary to complete certain current assignments. 

Mr. Kriegsman is eligible to receive grants of options to purchase shares of our common stock. The number and terms of those options, 

including the vesting schedule, will be determined by our board of directors (or its Compensation Committee) in its sole discretion. 

Under Mr. Kriegsman’s employment agreement, we have agreed that, if he is made a party, or threatened to be made a party, to a 
suit or proceeding by reason of his service to us, we will indemnify and hold him harmless from all costs and expenses to the fullest 
extent permitted or authorized by our certificate of incorporation or bylaws, or any resolution of our board of directors, to the extent 
not inconsistent with Delaware law. We also have agreed to advance to Mr. Kriegsman such costs and expenses upon his request if he 
undertakes  to repay such  advances  if  it  ultimately  is  determined  that he  is  not  entitled  to  indemnification with respect  to  the  same. 
These  employment  agreement  provisions  are  not  exclusive  of  any  other  rights  to  indemnification  to  which  Mr.  Kriegsman  may  be 
entitled and are in addition to any rights he may have under any policy of insurance maintained by us. 

In  the  event  we  terminate  Mr.  Kriegsman’s  employment  without  “cause”  (as  defined),  or  if  Mr.  Kriegsman  terminates  his 
employment with “good reason” (as defined), (i) we have agreed to pay Mr. Kriegsman a lump-sum equal to his salary and prorated 
minimum annual bonus through to his date of termination, plus his salary and minimum annual bonus for a period of two years after 
his  termination  date,  or  until  the  expiration  of  the  amended  and  restated  employment  agreement,  whichever  is  later,  (ii)  he  will  be 
entitled to immediate vesting of all stock options or other awards based on our equity securities, and (iii) he will also be entitled to 
continuation of his life insurance premium payments and continued participation in any of our health plans through to the later of the 
expiration of the amended and restated employment agreement or 24 months following his termination date. Mr. Kriegsman will have 
no obligation in such events to seek new employment or offset the severance payments to him by any compensation received from any 
subsequent reemployment by another employer. 

Under Mr. Kriegsman’s employment agreement, he and his affiliated company, The Kriegsman Group, are to provide us during 
the term of his employment with the first opportunity to conduct or take action with respect to any acquisition opportunity or any other 
potential transaction identified by them within the biotech, pharmaceutical or health care industries and that is within the scope of the 
business  plan  adopted  by  our  board  of  directors.  Mr.  Kriegsman’s  employment  agreement  also  contains  confidentiality  provisions 
relating  to  our  trade  secrets  and  any  other  proprietary  or  confidential  information,  which  provisions  shall  remain  in  effect  for  five 
years after the expiration of the employment agreement with respect to proprietary or confidential information and for so long as our 
trade secrets remain trade secrets. 

Potential Payment upon Termination or Change in Control for Steven A. Kriegsman 

Mr. Kriegsman’s employment agreement contains no provision for payment to him in the event of a change in control of CytRx. 
If,  however,  a  change  in  control  (as  defined  in  our  2000  Long-Term  Incentive  Plan)  occurs  during  the  term  of  the  employment 
agreement,  and  if,  during  the  term  and  within  two  years  after  the  date  on  which  the  change  in  control  occurs,  Mr.  Kriegsman’s 
employment is terminated by us without cause or by him for good reason (each as defined in his employment agreement), then, in 
addition to the severance benefits described above, to the extent that any payment or distribution of any type by us to or for the benefit 
of Mr. Kriegsman resulting from the termination of his employment is or will be subject to the excise tax imposed under Section 4999 
of the Internal Revenue Code of 1986, as amended, we have agreed to pay Mr. Kriegsman, prior to the time the excise tax is payable 
with respect to any such payment (through withholding or otherwise), an additional amount that, after the imposition of all income, 
employment, excise and other taxes, penalties and interest thereon, is equal to the sum of (i) the excise tax on such payments plus (ii) 
any penalty and interest assessments associated with such excise tax. 

58 

  
  
  
  
  
  
  
  
  
 
Employment Agreement with Daniel Levitt, M.D., Ph.D. 

Daniel Levitt is employed as our Chief Medical Officer pursuant to an employment agreement dated as of October 12, 2009 that 
expires on December 31, 2010. Dr. Levitt is entitled under his employment agreement to receive an annual base salary of $375,000 
and  is  eligible  to  receive  an  annual  bonus  as  determined  by  our  board  of  directors  (or  our  Compensation  Committee)  in  its  sole 
discretion, but not to be less than 25% of his 2010 base salary. As an incentive to enter into his employment agreement, we granted 
Dr. Levitt a ten-year non-qualified stock option under our 2000 Long-Term Incentive Plan to purchase up to 500,000 shares of our 
common stock at an exercise price of $1.06 per share, which equaled the market price of our common stock on October 12, 2009 as 
reported  in  The  NASDAQ  Capital  Market.  The  option  will  vest  ratably  in  36  equal  monthly  installments  commencing  on  the  first 
monthly  anniversary  of  the  grant  date  and  continuing  on  each  successive  monthly  anniversary  of  the  grant  date  until  the  option 
becomes fully vested, subject to Mr. Geyer remaining in our continuous employ through such monthly vesting periods. 

In the event we terminate Dr. Levitt’s employment without cause (as defined), we have agreed to pay him a lump-sum equal to 

his accrued but unpaid salary and vacation, plus an amount equal to six months’ salary under his employment agreement. 

Employment Agreement with John Y. Caloz 

John  Y.  Caloz  is  employed  as  our  Chief  Financial  Officer  and  Treasurer  pursuant  to  an  employment  agreement  dated  as  of 
January 1, 2010 that expires on December 31, 2010. Mr. Caloz is entitled under his employment agreement to receive an annual base 
salary  of  $325,000  and  is  eligible  to  receive  an  annual  bonus  as  determined  by  our  board  of  directors  (or  our  Compensation 
Committee) in its sole discretion. 

In the event we terminate Mr. Caloz’s employment without cause (as defined), we have agreed to pay him a lump-sum equal to 

his accrued but unpaid salary and vacation, plus an amount equal to six months’ salary under his employment agreement. 

Employment Agreement with Scott Wieland, Ph.D. 

Scott Wieland is employed as our Senior Vice President — Drug Development pursuant to an employment agreement dated as of 
January 1, 2010 that expires on December 31, 2010. Dr. Wieland is paid an annual base salary of $315,000 and is eligible to receive 
an annual bonus as determined by our board of directors (or our Compensation Committee) in its sole discretion. 

In the event we terminate Dr. Wieland’s employment without “cause” (as defined), we have agreed to pay him a lump-sum equal 

to his accrued but unpaid salary and vacation, plus an amount equal to six months’ base salary. 

Employment Agreement with Benjamin S. Levin 

Benjamin  S.  Levin  is  employed  as  our  Vice  President  —  Legal  Affairs,  General  Counsel  and  Secretary  pursuant  to  an 
employment agreement dated as of January 1, 2010 that expires on December 31, 2010. Mr. Levin is paid an annual base salary of 
$315,000 and is eligible to receive an annual bonus as determined by our board of directors (or our Compensation Committee) in its 
sole discretion. 

In the event we terminate Mr. Levin’s employment without “cause” (as defined), we have agreed to pay him a lump-sum equal to 

his accrued but unpaid salary and vacation, plus an amount equal to six months’ base salary. 

Employment Agreement with Scott Geyer 

Scott  Geyer  is  employed  as  our  Senior  Vice  President  —  Manufacturing  pursuant  to  an  employment  agreement  dated  as  of 
November 30, 2009 that expires on December 31, 2010. Mr. Geyer is paid an annual base salary of $290,000 and is eligible to receive 
an annual bonus as determined by our board of directors (or our Compensation Committee) in its sole discretion. As an incentive to 
enter  into  his  employment  agreement,  we  granted  Mr.  Geyer  a  ten-year  non-qualified  stock  option  under  our  2000  Long-Term 
Incentive  Plan  to  purchase  up  to  150,000  shares  of  our  common  stock  at  an  exercise  price  of  $0.96  per  share,  which  equaled  the 
market price of our common stock on November 30, 2009 as reported in The NASDAQ Stock Market. The option will vest ratably 
in36  equal  monthly  installments  commencing  on  the  first  monthly  anniversary  of  the grant  date  and  continuing  on  each  successive 
monthly anniversary of the grant date until the option becomes fully vested, subject to Mr. Geyer remaining in our continuous employ 
through such monthly vesting periods. 

59 

  
  
  
  
  
  
  
  
  
  
  
  
  
 
 
In the event we terminate Mr. Geyer’s employment without cause (as defined), we have agreed to pay him a lump-sum equal to 

his accrued but unpaid salary and vacation, plus an amount equal to six months’ salary under his employment agreement. 

Quantification of Termination Payments and Benefits 

The table below reflects the amount of compensation to each of our named executive officers in the event of termination of such 
executive’s  employment  without  “cause”  or  his  resignation  for  “good  reason,”  termination  following  a  change  in  control  and 
termination upon the executive’s death of permanent disability. The named executive officers are not entitled to any payments other 
than accrued compensation and benefits in the event of their voluntary resignation. The amounts shown in the table below assume that 
such termination was effective as of December 31, 2009, and thus includes amounts earned through such time, and are estimates only 
of the amounts that would be payable to the executives. The actual amounts to be paid will be determined upon the occurrence of the 
events indicated. 

Termination Payments and Benefits 

Termination w/o Cause or
for Good Reason

Name  
Steven A. Kriegsman . . . . . .   Severance Payment(4)     

Benefit 

President and Chief . . . . . .   Stock Options (1) 

Executive Officer  . . . . .   Health Insurance (2) 

Life Insurance 
Bonus 
Tax Gross Up (3) 

John Y. Caloz . . . . . . . . . . . . .   Severance Payment(4)     

Chief Financial Officer  . .   Stock Options (1) 

Daniel Levitt, M.D., Ph.D. .   Severance Payment(4)     

Chief Medical Officer . . . .   Stock Options (1) 
Benjamin S. Levin . . . . . . . . .   Severance Payment 
General Counsel, Vice . . .   Stock Options (1) 

Before Change 
in Control ($)    

After Change 
in Control ($)    

1,100,000     
—     
87,420     
10,000     
300,000     
—     
137,500     
—     
187,500     
—     
137,500     
—     

1,100,000     
—     
87,420     
10,000     
300,000     
0     
137,500     
—     
187,500     
—     
137,500     
—     

      Disability ($)    

Death ($) 
1,100,000       1,100,000     
—     
87,420     
10,000     
300,000     
—     
—     
—     
—     
—     
—     
—     

—      
—      
—      
300,000      
—      
—      
—      
—      
—      
—      
—      

Change in
Control ($)

— 
— 
87,420 
— 
— 
— 
— 
— 
— 
— 
— 
— 

President — Legal 
Affairs and Secretary 

Scott Wieland, Ph.D. . . . . . . .   Severance Payment(4)     

Senior Vice President – . .   Stock Options (1) 

137,500     
—     

137,500     
—     

—      
—      

—     
—     

— 
— 

Drug Development 

____________ 

(1)  Represents the aggregate value of stock options that vest and become exercisable immediately upon each of the triggering events 
listed as if such events took place on December 31, 2009, determined by the aggregate difference between the stock price as of 
December 31, 2009 and the exercise prices of the underlying options. 

(2)  Represents the cost as of December 31, 2009 for the family health benefits provided to Mr. Kriegsman for a period of two years. 

(3)  Mr.  Kriegsman’s  employment  agreement  provides  that  if  a  change  in  control  (as  defined  in  our 2000  Long-Term  Incentive  Plan) 
occurs during the term of the employment agreement, and if, during the term and within two years after the date on which the change 
in control occurs, Mr. Kriegsman’s employment is terminated by us without “cause” or by him for “good reason” (each as defined in 
his  employment  agreement),  then,  to  the  extent  that  any  payment  or  distribution  of  any  type  by  us  to  or  for  the  benefit  of  Mr. 
Kriegsman resulting from the termination of his employment is or will be subject to the excise tax imposed under Section 4999 of the 
Internal Revenue Code of 1986, as amended, we will pay Mr. Kriegsman, prior to the time the excise tax is payable with respect to 
any such payment (through withholding or otherwise), an additional amount that, after the imposition of all income, employment, 
excise and other taxes, penalties and interest thereon, is equal to the sum of (i) the excise tax on such payments plus (ii) any penalty 
and interest assessments associated with such excise tax. Based on Mr. Kriegsman’s past compensation and the estimated payment 
that would result from a termination of his employment following a change in control, we have estimated that a gross-up payment 
would  not  be  required.  “Good  reason”  as  defined  in  Mr.  Kriegsman’s  employment  agreement  includes  any  change  in  Mr. 
Kriegsman’s duties or title that are inconsistent with his position as Chief Executive Officer. 

(4)  Severance payments are prescribed by our employment agreements with the named executive officers and represent a factor of 

their annual base compensation ranging from six months to two years. 

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Compensation of Directors 

The following table sets forth the compensation paid to our directors other than our Chief Executive Officer for 2009: 

Director Compensation Table 

Name (1)  
Max Link, Ph.D. . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    

Fees Earned or 
Paid in Cash 
($) (2)
132,250      

Option Awards
($) (3) 

Total ($)

44,400     

176,650 

Chairman 

Marvin R. Selter . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    

Vice Chairman 

Louis Ignarro, Ph.D. . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    

Director 

Joseph Rubinfeld, Ph.D. . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    

Director 

Richard L. Wennekamp . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    

112,250      

44,400     

156,650 

37,500      

44,400     

81,900 

79,000      

44,400     

123,400 

112,250      

44,400     

156,650 

Director 
____________ 

(1)  Steven  A.  Kriegsman  does  not  receive  additional  compensation  for  his  role  as  a  Director.  For  information  relating  to  Mr. 

Kriegsman’s compensation as President and Chief Executive Officer, see the Summary Compensation Table above. 

(2)  The  amounts  in  this  column  represent  cash  payments  made  to  Non-Employee  Directors  for  attendance  at  meetings  during  the 

year. 

(3)  In July 2009, we granted stock options to purchase 50,000 shares of our common stock at an exercise price equal to the current 
market  value  of  our  common  stock  to  each  non-employee  director,  which  had  a  grant  date  fair  value  of  $44,400  calculated  in 
accordance with FASB ASC Topic 718, excluding the effect of estimated forfeitures related to service-based vesting conditions. 
The amount recognized for these awards was calculated using the Black Scholes option-pricing model, and reflect grants from our 
2000 Long-Term Incentive Plan, which is described in Note 15 of the Notes to Consolidated Financial Statements. 

We use a combination of cash and stock-based compensation to attract and retain qualified candidates to serve on our board of 
directors.  Directors  who  also  are  employees  of  our  company  currently  receive  no  compensation  for  their  service  as  directors  or  as 
members of board committees. In setting director compensation, we consider the significant amount of time that directors dedicate to 
the fulfillment of their director responsibilities, as well as the competency and skills required of members of our board. The directors’ 
current compensation schedule has been in place since May 2009. The directors’ annual compensation year begins with the annual 
election of directors at the annual meeting of stockholders. The annual retainer year period has been in place for directors since 2003. 
Periodically, our board of directors reviews our director compensation policies and, from time to time, makes changes to such policies 
based on various criteria the board deems relevant. 

Our  non-employee  directors  receive  a  quarterly  retainer  of  $6,000  (plus  an  additional  $12,500  for  the  Chairman  of  the  Board, 
$5,000 for the Chairman of the Audit Committee, and $1,500 for the Chairmen of the Nomination and Governance Committee and the 
Compensation  Committee),  a  fee  of  $3,000  for  each  board  meeting  attended  ($750  for  board  actions  taken  by  unanimous  written 
consent),  $2,000  for  each  meeting  of  the Audit  Committee  attended,  and  $1,000  for  each  other  committee  meeting  attended.  Non-
employee directors who serve as the chairman of a board committee receive an additional $2,000 for each meeting of the Nomination 
and Governance Committee or the Compensation Committee attended and an additional $2,500 for each meeting attended of the audit 
committee. In July 2009, we granted stock options to purchase 50,000 shares of our common stock at an exercise price equal to the 
current market value of our common stock to each non-employee director. The options were vested, in full, upon grant. 

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Joseph Rubinfeld, Ph.D. Consulting Agreement 

On December 2, 2008, we entered into a written consulting agreement with Joseph Rubinfeld, Ph.D., under which Dr. Rubinfeld 
agrees to serve as our Chief Scientific Advisor. In exchange, we granted to Dr. Rubinfeld under our 2008 Stock Incentive Plan a ten-
year stock option to purchase up to 350,000 shares of our common stock at an exercise price of $0.35 per share, which equaled the 
market price of our common stock as of the grant date. The stock option vested immediately upon grant as to 50,000 of the option 
shares  and  will  vest  as  to  the  remaining  option  shares  in  36  equal  monthly  installments,  subject  in  each  case  to  Dr.  Rubinfeld 
remaining in our service through such dates. We also agree in the consulting agreement to pay Dr. Rubinfeld a monthly fee of $1,000. 
The consulting agreement is terminable at any time by either party upon notice to the other party. 

Item  12.  SECURITY  OWNERSHIP  OF  CERTAIN  BENEFICIAL  OWNERS  AND  MANAGEMENT  AND  RELATED 
STOCKHOLDER MATTERS 

Based  solely  upon  information  made  available  to  us,  the  following  table  sets  forth  information  with  respect  to  the  beneficial 
ownership of our common stock as of March 12, 2010 by (1) each person who is known by us to beneficially own more than five 
percent of our common stock; (2) each of our directors; (3) the named executive officers listed in the Summary Compensation Table 
under Item 11; and (4) all of our executive officers and directors as a group. Beneficial ownership is determined in accordance with 
the SEC rules. Shares of common stock subject to any warrants or options that are presently exercisable, or exercisable within 60 days 
of March 12, 2010 (which are indicated by footnote) are deemed outstanding for the purpose of computing the percentage ownership 
of  the  person  holding  the  warrants  or  options,  but  are  not  treated  as  outstanding  for  the  purpose  of  computing  the  percentage 
ownership of any other person. The percentage ownership reflected in the table is based on 108,908,105 shares of our common stock 
outstanding as of March 12, 2010, excluding treasury shares. Except as otherwise indicated, the holders listed below have sole voting 
and investment power with respect to all shares of common stock shown, subject to applicable community property laws. An asterisk 
represents beneficial ownership of less than 1%. 

Shares of Common Stock

Name of Beneficial Owner  
Louis Ignarro, Ph.D.(1) . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .       
618,916     
Steven A. Kriegsman(2) . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .        6,305,808     
Max Link, Ph.D.(3) . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .       
239,519     
Joseph Rubinfeld, Ph.D.(4) . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .       
177,000     
Marvin R. Selter(5) . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .       
522,451     
Richard L. Wennekamp(6) . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .       
170,000     
Dan Levitt, M.D., Ph.D.(7) . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .       
83,334     
John Y. Caloz (8) . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .       
113,197     
Scott Wieland, Ph.D.(9) . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .       
122,502     
Benjamin S. Levin(10) . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .       
608,350     
All executive officers and directors as a group (eleven persons)(11). . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .        8,981,912     
____________ 

Number

Percent

*  
5.7%
*  
*  
*  
*  
*  
*  
*  
*  
7.9%

(1)  Includes 527,000 shares subject to options or warrants. 

(2)  Includes 2,284,708 shares subject to options or warrants. Mr. Kriegsman’s address is c/o CytRx Corporation, 11726 San Vicente 

Boulevard, Suite 650, Los Angeles, CA 90049. 

(3)  Includes 184,543 shares subject to options or warrants. 

(4)  Includes 177,000 shares subject to options or warrants. 

(5)  The shares shown are owned, of record, by the Selter Family Trust or Selter IRA Rollover. Includes 165,000 shares subject to 

options or warrants owned by Mr. Selter. 

(6)  Includes 165,000 shares subject to options or warrants. 

(7)  Includes 83,334 shares subject to options or warrants. 

(8)  Includes 113,197 shares subject to options or warrants. 

62 

  
  
  
  
   
  
  
  
   
  
 
 
 
 
 
 
 
 
 
(9)  Includes 122,502 shares subject to options or warrants. 

(10) Includes 608,350 shares subject to options or warrants. 

(11) Includes 4,451,469 shares subject to options or warrants. 

Item 13. CERTAIN RELATIONSHIPS AND RELATED TRANSACTIONS 

Director Independence 

Our  board  of  directors  has  determined  that  Messrs.  Link,  Selter,  Ignarro  and  Wennekamp  are  “independent”  under  the  current 
independence standards of both The NASDAQ Capital Market and the SEC, and have no material relationships with us (either directly 
or as a partner, shareholder or officer of any entity) which could be inconsistent with a finding of their independence as members of 
our board of directors or as the members of our Audit Committee. In making these determinations, our board of directors has broadly 
considered all relevant facts and circumstances, recognizing that material relationships can include commercial, banking, consulting, 
legal, accounting, and familial relationships, among others. 

Transactions with Related Persons 

General 

Our  Audit  Committee  is  responsible  for  reviewing  and  approving,  as  appropriate,  all  transactions  with  related  persons,  in 

accordance with its Charter and NASDAQ Marketplace Rules. 

Transactions between us and one or more related persons may present risks or conflicts of interest or the appearance of conflicts 
of interest. Our Code of Ethics requires all employees, officers and directors to avoid activities or relationships that conflict, or may be 
perceived  to  conflict,  with  our  interests  or  adversely  affect  our  reputation.  It  is  understood,  however,  that  certain  relationships  or 
transactions may arise that would be deemed acceptable and appropriate so long as there is full disclosure of the interest of the related 
parties  in  the  transaction  and  review  and  approval  by  disinterested  directors  to  ensure  there  is  a  legitimate  business  reason  for  the 
transaction and that the transaction is fair to us and our stockholders. 

As a result, the procedures followed by the Audit Committee to evaluate transactions with related persons require: 

• 

• 

that all related person transactions, all material terms of the transactions, and all the material facts as to the related person’s 
direct or indirect interest in, or relationship to, the related person transaction must be communicated to the Audit Committee; 
and 

that  all  related  person  transactions,  and  any  material  amendment  or  modification  to  any  related  person  transaction,  be 
reviewed and approved or ratified by the Audit Committee, as required by NASDAQ Marketplace Rules. 

Our Audit Committee will evaluate related person transactions based on: 

• 

• 

• 

• 

information  provided  by  members  of  our  board  of  directors  in  connection  with  the  required  annual  evaluation  of  director 
independence; 

pertinent  responses  to  the  Directors’  and  Officers’  Questionnaires  submitted  periodically  by  our  officers  and  directors  and 
provided to the Audit Committee by our management; 

background information on nominees for director provided by the Nominating and Corporate Governance Committee of our 
board of directors; and 

any other relevant information provided by any of our directors or officers. 

63 

 
 
 
  
  
  
  
  
  
  
  
  
  
  
  
  
  
 
 
In connection with its review and approval or ratification, if appropriate, of any related person transaction, our Audit Committee 
is  to  consider whether  the  transaction will  compromise  standards  included  in our  Code  of  Ethics. In  the  case of  any  related person 
transaction involving an outside director or nominee for director, the Audit Committee also is to consider whether the transaction will 
compromise the director’s status as an independent director as prescribed in the NASDAQ Marketplace Rules. 

Exemption Clause 

Item  404(a)(7)(a)  of  Securities  and  Exchange  Commission  Regulation  S-K  states  that:  Disclosure  need  not  be  provided  if  the 
transaction is one where the rates or charges involved in the transaction are determined by competitive bid, or the transaction involves 
rendering  of  services  as  a  common  or  contract  carrier,  or  public  utility,  at  rates  or  charges  fixed  in  conformity  with  law  or 
governmental authority. 

Applicable Definitions 

For purposes of our Audit Committee’s review: 

• 

• 

“related person” has the meaning given to such term in Item 404(a) of Securities and Exchange Commission Regulation S-K 
(“Item 404(a)”); and 

“related person transaction” means any transaction for which disclosure is required under the terms of Item 404(a) involving 
the Company and any related persons. 

Item 14. PRINCIPAL ACCOUNTANT FEES AND SERVICES 

BDO Seidman, LLP, or BDO, serves as our independent registered public accounting firm and audited our financial statements 

for the years ended December 31, 2009, 2008 and 2007. 

Audit Fees 

The  fees  for  2009  and  2008  billed  to  us  by  BDO  for  professional  services  rendered  for  the  audit  of  our  annual  consolidated 

financial statements and internal controls over financial reporting were $383,500 and $350,311, respectively. 

Audit-Related Fees 

BDO rendered $25,175 of assurance and other related services in 2009, and $152,262 of assurance and other related services in 

2008, which included services relating to our shelf registration with the SEC and the Innovive acquisition. 

Tax Fees 

The aggregate fees billed by BDO for professional services for tax compliance, tax advice and tax planning were $33,260 and 

$39,000 for 2009 and 2008, respectively. 

All Other Fees 

No other services were rendered by BDO for 2009 or 2008. 

Pre-Approval Policies and Procedures 

It  is  the  policy  of  our  Audit  Committee  that  all  services  to  be  provided  by  our  independent  registered  public  accounting  firm, 
including audit services and permitted audit-related and non-audit services, must be pre-approved by our Audit Committee. Our Audit 
Committee pre-approved all services, audit and non-audit, provided to us by BDO for 2009 and 2008. 

64 

  
  
  
  
  
  
  
  
  
  
  
  
  
  
  
  
  
  
 
 
PART IV 

Item 15. EXHIBITS AND FINANCIAL STATEMENT SCHEDULES 

(a) The following documents are filed as part of this 10-K: 

(1) Financial Statements 

Our consolidated financial statements and the related report of the independent registered public accounting firm thereon are set 

forth on pages F-1 to F-26 of this Annual Report. These consolidated financial statements are as follows: 

Consolidated Balance Sheets as of December 31, 2009 and 2008 

Consolidated Statements of Operations for the Years Ended December 31, 2009, 2008 and 2007 

Consolidated Statements of Stockholders’ Equity for the Years Ended December 31, 2009, 2008 and 2007 

Consolidated Statements of Cash Flows for the Years Ended December 31, 2009, 2008 and 2007 

Notes to Consolidated Financial Statements 

Reports of Independent Registered Public Accounting Firms 

(2) Financial Statement Schedules 

The following financial statement schedule is set forth on page F-26 of this Annual Report. 

Schedule II — Valuation and Qualifying Accounts for the years ended December 31, 2009, 2008 and 2007 

All  other  schedules  are  omitted  because  they  are  not  required,  not  applicable,  or  the  information  is  provided  in  the  financial 

statements or notes thereto. 

(b) Exhibits 

See Exhibit Index on page 66 of this Annual Report, which is incorporated herein by reference. 

65 

 
 
  
  
  
  
  
  
  
  
  
  
  
  
  
  
 
 
Exhibit 
Number 
3.1 

 Description  
  Amended and Restated Certificate of Incorporation, as amended 

CytRx Corporation 
Form 10-K Exhibit Index 

  Restated By-Laws, as amended 

Footnote

  (a) 

  (a) 

  (z) 

  (c) 

  (d) 

  (e) 

  (g) 

  (g) 

  (h) 

  (h) 

  (y) 

  (f) 

  (h) 

  (h) 

  (s) 

  (t) 

  (t) 

  (t) 

3.2 

4.1 

4.2 

4.3 

4.4 

4.5 

4.6 

4.7 

4.8 

4.9 

10.1* 

10.2* 

10.3* 

10.4* 

10.5* 

10.6* 

10.7* 

10.8* 

10.9† 

10.11 

10.12 

10.13 

10.21 

10.22 

10.23 

10.24 

10.25 

10.26 

10.27 

10.28 

10.29 

10.30 

  Shareholder Protection Rights Agreement dated April 16, 1997 between CytRx Corporation and American Stock Transfer &Trust Company as Rights Agent    (b) 

  Amendment No. 1 to Shareholder Protection Rights Agreement 

  Amendment No. 2 to Shareholder Protection Rights Agreement 

  Warrant issued on May 10, 2004 to MBN Consulting, LLC 

  Form of Common Stock Purchase Warrant between CytRx Corporation and each of the investors in the October 4, 2004 private placement 

  Form of Common Stock Purchase Warrant between CytRx Corporation and each of the investors in the January 2005 private placement 

  Form of Common Stock Purchase Warrant between CytRx Corporation and each of the investors in the March 2006 private placement 

  (e) 

  (r) 

  (i) 

  (j) 

  (k) 

  (p) 

  Securities Purchase Agreement, dated July 24, 2009, by and among CytRx Corporation and the purchasers listed on the signature pages thereto    (z) 

  Form of Common Stock Purchase Warrant to be issued by CytRx Corporation to purchasers under the Securities Purchase Agreement 

  1994 Stock Option Plan, as amended and restated 

  1998 Long-Term Incentive Plan 

  2000 Long-Term Incentive Plan 

  Amendment No. 1 to 2000 Long-Term Incentive Plan 

  Amendment No. 2 to 2000 Long-Term Incentive Plan 

  Amendment No. 3 to 2000 Long-Term Incentive Plan 

  Amendment No. 4 to 2000 Long-Term Incentive Plan 

  2008 Stock Incentive Plan 

  License Agreement dated December 7, 2001 by and between CytRx Corporation and Vical Incorporated 

10.10† 

  Agreement between CytRx Corporation and Dr. Robert Hunter regarding SynthRx, Inc dated October 20, 2003 

  Office Lease between The Kriegsman Group and Douglas Emmett, dated April 13, 2000 

  Assignment to CytRx Corporation effective July 1, 2003 of Office Lease between The Kriegsman Group and Douglas Emmett, dated April 13, 2000   (h) 

  Asset Sale and Purchase Agreement dated October 4, 2004, by and among CytRx Corporation, Biorex Research & Development, RT and BRX 

Research and Development Company Ltd 

10.14 

  Sublease dated March 14, 2005 between Innovive Pharmaceuticals, Inc. and Friedman, Billings, Ramsey Group, Inc. 

10.15* 

  Amended and Restated Employment Agreement dated May 17, 2005 between CytRx Corporation and Steven A. Kriegsman 

10.16 

  First Amendment to Office Lease dated October 14, 2005, by and between CytRx Corporation and Douglas Emmett 1993, LLC 

10.17† 

  License Agreement dated December 28, 2005 between Innovive Pharmaceuticals, Inc. and Nippon Shinyaku Co., Ltd. 

10.18† 

  License Agreement dated April 17, 2006 between Innovive Pharmaceuticals, Inc. and KTB Tumorforschungs GmbH 

  (j) 

  (l) 

  (m) 

  (n) 

  (l) 

  (o) 

10.19 

  Royalty Agreement dated August 28, 2006 between CytRx Corporation and Kenneth Council, as Trustee of the ALS Charitable Remainder Trust 

  (q) 

10.20† 

  License Agreement dated December 6, 2006 between Innovive Pharmaceuticals, Inc. and TMRC Co., Ltd. 

  Contribution Agreement, dated as of January 8, 2007, between CytRx Corporation and RXi Pharmaceuticals Corporation 

  Voting agreement, dated as of January 10, 2007, between CytRx Corporation and the University of Massachusetts 

  Stockholders agreement, dated February 23, 2007, among CytRx Corporation, RXi Pharmaceuticals Corporation, Craig C. Mello, Ph.D., Tariq 

Rana, Ph.D., Gregory J. Hannon, Ph.D., and Michael P. Czech, Ph.D 

  Form of Purchase Agreement, dated as of April 17, 2007, by and between CytRx Corporation and each of the selling stockholders named therein 

  (u) 

  Contribution Agreement, dated as of April 30, 2007, between CytRx Corporation and RXi Pharmaceuticals Corporation 

  Lease dated July 20, 2007, between CytRx Corporation and BMR-3030 Bunker Hill Street LLC 

  (t) 

  (v) 

  Agreement and Plan of Merger, dated as of June 6, 2008, among CytRx Corporation, CytRx Merger Subsidiary, Inc., Innovive Pharmaceuticals, 

Inc., and Steven Kelly 

  Loan and Security Agreement, dated as of June 6, 2008, between CytRx Corporation and Innovive Pharmaceuticals, Inc. 

  Second Amendment to Office Lease dated June 30, 2008, by and between CytRx Corporation and Douglas Emmett 1993, LLC 

  Amendment to Contribution Agreement, dated July 28, 2008, between CytRx Corporation and RXi Pharmaceuticals Corporation 

  (w) 

  (w) 

  (y) 

  (x) 

66 

 
  
 
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
       
 
     
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
 
  
  
10.31 

  Amendment to Stockholders Agreement, dated July 28, 2008, among CytRx Corporation, RXi Pharmaceuticals Corporation, and Michael P. 

Czech, PhD., Gregory J. Hannon, Ph.D., Craig C. Mello, PhD., and Tariq M. Rana, Ph.D. 

10.32 

10.33 

  Sub-Sublease dated December 4, 2008, by and between CytRx Oncology Corporation and Red Pine Advisors LLC 

  Investment Banking Agreement, dated January 29, 2009, by and between CytRx Corporation and Legend Securities, Inc. 

10.34* 

  Employment Agreement dated October 12, 2009 between CytRx Corporation and Daniel Levitt, M.D., Ph.D. 

10.35* 

  Employment Agreement dated November 30, 2009, between CytRx Corporation and Scott Geyer 

  (x) 

  (y) 

  (y) 

  (aa) 

10.36 

  Third Amendment to Office Lease dated December 1, 2009, by and between CytRx Corporation and Douglas Emmett 1993, LLC 

  (bb) 

10.37* 

  Employment Agreement dated January 1, 2010, between CytRx Corporation and Benjamin S. Levin 

10.38* 

  Employment Agreement dated January 1, 2010, between CytRx Corporation and Scott Wieland 

10.39* 

  Employment Agreement dated January 1, 2010, between CytRx Corporation and John Y. Caloz 

23.1 

31.1 

31.2 

32.1 

  Consent of BDO Seidman, LLP 

  Certification of Chief Executive Officer Pursuant to 15 U.S.C. Section 7241, as adopted pursuant to Section 302 of the Sarbanes-Oxley Act of 2002  

  Certification of Chief Financial Officer Pursuant to 15 U.S.C. Section 7241, as adopted pursuant to Section 302 of the Sarbanes-Oxley Act of 2002 

  Certification of Chief Executive Officer Pursuant to 18 U.S.C. Section 1350, as adopted pursuant to Section 906 of the Sarbanes-Oxley Act of 2002  

  Certification of Chief Financial Officer Pursuant to 18 U.S.C. Section 1350, as adopted pursuant to Section 906 of the Sarbanes-Oxley Act of 2002 

32.2 
__________________ 
* 

Indicates a management contract or compensatory plan or arrangement. 

† 

Confidential  treatment  has  been  requested  or  granted for  certain  portions  which  have been  blanked out  in  the  copy  of  the  exhibit  filed  with  the Securities  and 
Exchange Commission. The omitted information has been filed separately with the Securities and Exchange Commission. 

(a) 

Incorporated by reference to the Registrant’s Form 10-K filed on April 1, 2008 

(b) 

Incorporated by reference to the Registrant’s 8-K filed on April 17, 1997 

(c) 

Incorporated by reference to the Registrant’s 10-Q filed on August 14, 1997 

(d) 

Incorporated by reference to the Registrant’s Proxy Statement filed on April 30, 1998 

(e) 

Incorporated by reference to the Registrant’s Form 10-K filed on March 27, 2001 

(f) 

Incorporated by reference to the Registrant’s Form 8-K filed on December 21, 2001 

(g) 

Incorporated by reference to the Registrant’s Proxy Statement filed June 11, 2002 

(h) 

Incorporated by reference to the Registrant’s 10-K filed on May 14, 2004 

(i) 

(j) 

Incorporated by reference to the Registrant’s 10-Q filed on August 16, 2004 

Incorporated by reference to the Registrant’s 8-K filed on October 5, 2004 

(k) 

Incorporated by reference to the Registrant’s 8-K filed on January 21, 2005 

(l) 

Incorporated by reference to the Innovive Pharmaceuticals Form 10 filed on April 20, 2006 

(m)  Incorporated by reference to the Registrant’s 10-Q filed on August 15, 2005 

(n) 

Incorporated by reference to the Registrant’s 8-K filed on October 20, 2005 

(o) 

Incorporated by reference to the Innovive Pharmaceuticals 10-Q filed on November 14, 2006 

(p) 

Incorporated by reference to the Registrant’s 8-K filed on March 3, 2006 

(q) 

Incorporated by reference to the Registrant’s 10-Q filed on November 13, 2006 

(r) 

Incorporated by reference to the Registrant’s 10-K filed on April 2, 2007 

(s) 

Incorporated by reference to the Innovive Pharmaceuticals 10-K filed on March 21, 2007 

(t) 

Incorporated by reference to the Registrant’s 10-Q filed on May 10, 2007 

(u) 

Incorporated by reference to the Registrant’s 8-K filed on April 18, 2007 

(v) 

Incorporated by reference to the Registrant’s 10-Q filed on August 9, 2007 

(w)  Incorporated by reference to the Registrant’s 8-K filed on June 9, 2008 

(x) 

Incorporated by reference to the Registrant’s 10-Q filed on August 11, 2008 

(y) 

Incorporated by reference to the Registrant’s 10-K filed on March 13, 2009 

(z) 

Incorporated by reference to the Registrant’s 8-K filed on July 27, 2009 

(aa)  Incorporated by reference to the Registrant’s 10-Q filed on November 9, 2009 

(bb 

Incorporated by reference to the Registrant’s 8-K filed on December 4, 2009 

67 

 
  
  
 
  
  
 
  
  
  
 
   
 
 
  
  
 
  
  
 
 
  
  
 
 
  
  
 
 
  
  
 
 
  
  
 
  
  
 
 
  
  
 
  
  
  
  
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Pursuant to the requirements of Section 13 or 15(d) of the Securities Exchange Act of 1934, the Registrant has duly caused this 

report to be signed on its behalf by the undersigned, thereunto duly authorized. 

SIGNATURES 

Date: March 12, 2010 

CYTRX CORPORATION

By: /s/ STEVEN A. KRIEGSMAN 

Steven A. Kriegsman 
President and Chief Executive Officer 

68 

  
 
 
 
 
 
  
 
 
 
 
 
 
 
 
 
 
  
INDEX TO FINANCIAL STATEMENTS 
AND FINANCIAL STATEMENT SCHEDULE 

CytRx Corporation 
Consolidated Balance Sheets . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . F-2 
Consolidated Statements of Operations . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . F-3 
Consolidated Statements of Stockholders’ Equity . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . F-4 
Consolidated Statements of Cash Flows . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . F-5 
Notes to Consolidated Financial Statements . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . F-7 
Reports of Independent Registered Public Accounting Firm . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . F-24 
Financial Statement Schedule II — Valuation and Qualifying Accounts . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . F-26

F-1 

 
 
 
CYTRX CORPORATION 
CONSOLIDATED BALANCE SHEETS 

ASSETS

December 31,

2009 

2008

Current assets: 

Cash and cash equivalents . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .      $
Marketable securities . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .         22,750,000    
Receivable . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .        
139,680    
Income taxes recoverable . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .        
519,158    
Interest receivable . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .        
130,779    
Assets held for sale . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .        
73,634    
Prepaid expenses and other current assets . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .        
1,088,074    
Total current assets . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .         34,594,915    
174,959    
—    
183,780    
323,235    

9,893,590   $ 25,041,772 
— 
127,280 
215,623 
— 
— 
486,609 
25,871,284 
1,835,052 
103,882 
183,780 
330,032 
Total assets . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .      $ 35,276,889   $ 28,324,030 

Equipment and furnishings, net . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .        
Molecular library, net . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .        
Goodwill . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .        
Other assets . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .        

LIABILITIES AND STOCKHOLDERS’ EQUITY

Current liabilities: 

Accounts payable . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .      $
Accrued expenses and other current liabilities . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .        
Warrant liability . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .        
Deferred revenue, current portion . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .        
Total current liabilities . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .        
Deferred revenue, non-current portion . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .        
Total liabilities . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .        

1,066,055   $
2,492,450    
3,370,701    
—    
6,929,206    
—    
6,929,206    

668,422 
2,556,904 
— 
1,817,600 
5,042,926 
7,582,797 
12,625,723 

Commitment and contingencies 

Stockholders’ equity: 

Preferred Stock, $.01 par value, 5,000,000 shares authorized, including 15,000 shares of Series A 

Junior Participating Preferred Stock; no shares issued and outstanding . . . . . . . . . . . . . . . . . . . . . . . .        

—    

— 

Common stock, $.001 par value, 175,000,000 shares authorized; 109,538,821 and 93,978,448 

shares issued and outstanding at December 31, 2009 and 2008, respectively . . . . . . . . . . . . . . . . . . .        

93,978 
Additional paid-in capital . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .         227,441,591     210,007,468 
Treasury stock, at cost (633,816 shares held, at December 31, 2009 and 2008, respectively). . . . . . .        
(2,279,238)
Accumulated deficit . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .        (196,924,209)    (192,123,901)
Total stockholders’ equity . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .         28,347,683    
15,698,307 
Total liabilities and stockholders’ equity . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .      $ 35,276,889   $ 28,324,030 

(2,279,238)   

109,539    

The accompanying notes are an integral part of these consolidated financial statements. 

F-2 

 
  
  
 
  
  
   
 
    
      
 
    
      
 
    
    
 
    
    
 
  
    
    
 
    
    
 
 
 
 
CYTRX CORPORATION 
CONSOLIDATED STATEMENTS OF OPERATIONS 

Years Ended December 31,
2008 

2007

2009

Revenue: 

Service revenue . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   $ 9,400,397    $  6,166,150    $ 7,241,920 
Licensing revenue . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
101,000 
Grant revenue . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
116,118 
7,459,038 

100,000     
—     
9,500,397       6,266,150     

100,000      
—      

Expenses: 

Research and development . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
General and administrative . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
In-process research and development . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .
Depreciation and amortization . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    

Loss before other income . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Other income: 

Interest and dividend income . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Other income, net . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Gain on warrant derivative liability . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Gain on sale of affiliate’s RXi Pharmaceutical shares . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Equity in loss of affiliate – RXi Pharmaceuticals . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    

Net loss before provision for income taxes . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Provision for income taxes . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Net loss . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Deemed dividend for anti-dilution adjustments made to outstanding common stock 

7,541,998       10,465,591      18,823,802 
9,127,845       10,932,522      14,822,142 
— 
   8,012,154     
272,229 
624,980     
    17,145,159       30,035,247      33,918,173 
(7,644,762)     (23,769,097)     (26,459,135)

475,316      

—  

93,950      
656,905      
1,224,951      

349,490       1,203,629     
219,489     
—     
—     
—       (3,915,514)    

2,663,542 
1,496,979 
— 
— 
— 

(5,319,466)     (26,261,493)     (22,298,614)
(40,000)
(4,800,308)     (27,134,496)     (22,338,614)

(873,003)    

519,158      

warrants . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Net loss . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Add: Loss of noncontrolling interest . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    

— 
(4,800,308)     (27,891,450)     (22,338,614)
448,671 
Net loss attributable to CytRx Corporation . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   $ (4,800,308)   $ (27,803,075)   $(21,889,943)
Basic and diluted loss per share . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   $
(0.26)
Basic and diluted weighted average shares outstanding. . . . . . . . . . . . . . . . . . . . . . . . . . . . .     99,978,124       91,383,934      84,006,728 

(756,954)    

88,375     

(0.05)   $ 

(0.30)   $

—      

—      

The accompanying notes are an integral part of these consolidated financial statements. 

F-3 

 
  
 
 
  
 
     
   
 
    
        
      
 
   
   
      
     
 
 
   
      
     
 
   
      
     
 
 
 
 
CYTRX CORPORATION 
CONSOLIDATED STATEMENTS OF STOCKHOLDERS’ EQUITY 

Balance at December 31, 2006 . . . . . . . .     70,788,586$ 70,789$ 146,961,657$ (140,139,915)$(2,279,238)  $ 

537,046   

Common Stock
 Shares Issued  Amount

Additional
Paid-In

Capital

Accumulated   Treasury 

Deficit

Stock 

   Noncontrolling     
Interest

Total
5,150,339 

Common stock and warrants issued 

in connection with private 
placements . . . . . . . . . . . . . . . . . . . . . .     8,615,000 

8,615  34,239,442 

—   

—     

    34,248,057 

Issuance of stock options/warrants 
for compensation, services and 
licenses . . . . . . . . . . . . . . . . . . . . . . . . .    

2,402,035 
Options and warrants exercised . . . . .     10,994,281  10,994  18,778,180 
Issuance of stock options by 

—   
—   

—     
—     

2,402,035 
    18,789,174 

subsidiary  . . . . . . . . . . . . . . . . . . . . . .    
Net loss . . . . . . . . . . . . . . . . . . . . . . . . . . .    

—     
—     
Balance at December 31, 2007 . . . . . . . .     90,397,867$ 90,398$ 203,905,691$ (161,492,812)$(2,279,238)  $ 

—   
(21,889,943) 

1,524,377 
— 

— 
— 

— 
— 

1,524,377 
(448,671)  (22,338,614)
(448,671)$ 40,312,414 

Issuance of stock options/warrants 
for compensation, services and 
licenses . . . . . . . . . . . . . . . . . . . . . . . . .    

— 
Options and warrants exercised . . . . .     1,006,402 
Common stock issued in connection 

with the acquisition of Innovive . .     2,574,179 

— 
1,006 

2,029,209 
975,782 

2,574 

2,339,832 

—   
—   

—   

—     
—     

—     

2,029,209 
976,788 

2,342,406 

Deemed dividend for anti-dilution 

adjustment . . . . . . . . . . . . . . . . . . . . . .    
Dividend of RXi stock . . . . . . . . . . . . .    
Net loss . . . . . . . . . . . . . . . . . . . . . . . . . . .    

—     
—     
—     
Balance at December 31, 2008 . . . . . . . .     93,978,448$ 93,978$ 210,007,468$ (192,123,901)$(2,279,238)  $ 

(756,954) 
(2,828,014) 
(27,046,121) 

756,954 
— 
— 

— 
— 
— 

— 
— 

— 
(2,828,014)
(88,375)  (27,134,496)
—  $ 15,698,307 

Common stock and warrants issued 

in connection with private 
placements . . . . . . . . . . . . . . . . . . . . . .     15,252,040  15,253  14,230,710 

—   

—     

    14,245,963 

Issuance of stock options/warrants 

for compensation and services . . . .    
Common stock issued for services . .    
Options and warrants exercised . . . . .    
Net loss . . . . . . . . . . . . . . . . . . . . . . . . . . .    

—     
—     
—     
—     
Balance at December 31, 2009 . . . . . . . .    109,538,821$109,539$ 227,441,591$ (196,924,209)$(2,279,238)  $ 

—   
—   
—   
(4,800,308) 

2, 867,638 
42,950 
292,825 
— 

— 
50,000 
258,333 
— 

— 
50 
258 
— 

2,867,638 
43,000 
293,083 
—   
(5,319,466)
—  $ 27,828,525 

The accompanying notes are an integral part of these consolidated financial statements. 

F-4 

 
   
  
    
     
    
 
 
 
 
   
 
 
 
 
   
   
   
   
   
 
   
   
   
   
   
 
 
 
CYTRX CORPORATION 
CONSOLIDATED STATEMENTS OF CASH FLOWS 

Years Ended December 31,
2008 

2007

2009

Cash flows from operating activities: 

Net loss attributable to CytRx Corporation . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   $ (4,800,308)   $  (27,046,121)   $ (21,889,943)
Adjustments to reconcile net loss to net cash provided by (used in) operating activities:     
Depreciation and amortization . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Retirement of fixed assets . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Interest receivable on marketable securities . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Loss of noncontrolling interest . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Fair value adjustment of warrant liability . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Impairment loss on fixed assets . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Equity in loss of affiliate . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Non-cash gain on transfer of RXi common stock . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Gain on sale of affiliate’s shares . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Non-cash expense on the acquisition of Innovive’s in-process research & development .    
Stock option and warrant expense . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Common stock issued for services . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Changes in assets and liabilities: 

475,316      
103,241      
—      
—      
(656,905)     
1,187,305      
—      
—      
(1,224,951)     
—      
2,734,247      
43,000      

624,980     
262     
(48,452)    
(88,375)    
—     
—     
3,915,515     
(226,579)    
—     
8,012,154     
2,103,752     
244,860     

272,229 
— 
(172,055)
(448,671)
— 
— 
— 
— 
— 
— 
3,511,541 
3,089,639 

Accounts receivable . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
4,713 
Interest receivable . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
— 
Income taxes recoverable . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
— 
Prepaid expenses and other current assets . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
(1,214,836)
Accounts payable . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
757,086 
Deferred revenue . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
(7,241,919)
Accrued expenses and other current liabilities . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
978,388 
Total adjustments . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
(463,885)
Net cash used in operating activities . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .     (12,114,264)      (19,409,944)     (22,353,828)

(12,400)     
(130,779)     
(303,535)     
(461,277)     
397,633      
(9,400,397)     
(64,454)     
(7,313,956)     

238,131     
—     
(215,623)    
478,965     
(1,181,116)    
(6,166,151)    
(56,146)    
7,636,177     

Cash flows from investing activities: 

Proceeds (Purchase) from sale of marketable securities . . . . . . . . . . . . . . . . . . . . . . . . . . . . .     (22,750,000)      10,000,000     
Proceeds from sale of fixed assets . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
—     
Deconsolidation of subsidiary . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
—       (10,359,278)    
Proceeds from sale of unconsolidated sub shares . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
1,224,951      
—     
Cash outlay in the acquisition of Innovive, relating to its accounts payable . . . . . . . . . . . .    
(5,669,749)    
—      
Purchases of equipment and furnishings . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
(994,326)    
(195,449)     
Net cash used in investing activities . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .     (21,600,569)     

(9,779,493)
— 
— 
— 
— 
(1,269,313)
(7,023,353)     (11,048,806)

119,929      

Cash flows from financing activities: 

Net proceeds from exercise of stock options and warrants. . . . . . . . . . . . . . . . . . . . . . . . . . .    
293,083      
Common stock issued in accordance with financing . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .     18,273,568      
Net proceeds from issuances of common stock . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
—      
Capital contributions from minority interest . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
—      
Net cash provided by financing activities . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .     18,566,651      

976,808      18,789,173 
— 
—     
—      34,248,058 
482,271 
—     
976,808      53,519,502 

Net increase (decrease) in cash and cash equivalents . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .     (15,148,182)      (25,456,489)     20,116,868 
Cash and cash equivalents at beginning of year . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .     25,041,772       50,498,261      30,381,393 
9,893,590    $  25,041,772    $ 50,498,261 

Cash and cash equivalents at end of year . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   $

Supplemental disclosure of cash flow information: 

Cash paid during the years for income taxes . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   $

Supplemental disclosures of non-cash investing and financing activities: 

Acquisition of property and equipment through accrued liabilities . . . . . . . . . . . . . . . . . . .   $
Warrants issued in connection with financing . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   $
Warrants issued for prepaid services . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   $

—    $  1,093,764    $

183,461 

—    $ 
4,027,606    $ 
133,391    $ 

130,955    $
—    $
—    $ 

233,974 
— 
 — 

The accompanying notes are an integral part of these consolidated financial statements. See supplemental information on the following page.

F-5 

 
 
 
  
 
     
   
 
    
      
      
 
      
     
 
   
      
     
 
     
        
        
  
   
      
     
 
     
        
        
  
   
      
     
 
     
        
        
  
     
        
        
  
   
      
     
 
   
      
     
 
 
Supplemental schedule of non-cash investing and financing activities: 

CytRx  purchased  all  of  the  common  stock  of  Innovive  Pharmaceuticals,  Inc.  in  a  transaction  that  for  accounting  purposes  is 
considered  an  asset  acquisition.  See  Note  20  below.  The  fair  values  of  Innovive’s  assets  and  liabilities  at  September  19,  2008,  in 
millions of dollars, are presented below: 

In-process research and development. . . . . . . . . . . . .   $
Leasehold interests . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Prepaid expenses . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Accounts payable . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Net assets acquired through issuance of common 

stock . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   $

8.0  
0.1  
0.3  
(6.1) 

2.3  

As a result of the March 11, 2008 distribution by CytRx Corporation (the “Company”) to its stockholders of approximately 36% 
of  the  outstanding  shares  of  RXi  Pharmaceuticals  Corporation,  the  Company  deconsolidated  that  previously  majority-owned 
subsidiary. As part of the transaction, the Company deconsolidated $3.7 million of total assets and $4.6 million of total liabilities. 

In connection with applicable antidilution adjustments to the price of certain outstanding warrants in March 2008, the Company 
recorded  a  deemed  dividend  of  approximately  $756,954  in  the  current  year.  The  deemed  dividend  was  recorded  as  a  charge  to 
accumulated deficit and a corresponding credit to additional paid-in capital. 

During 2007, the Company allocated $289,254 of additional paid in capital arising from subsidiary common stock options issued 

to minority interest. 

F-6 

 
  
  
  
  
 
 
CYTRX CORPORATION 

NOTES TO CONSOLIDATED FINANCIAL STATEMENTS 

1. Nature of Business 

CytRx  Corporation  (“CytRx”  or  the  “Company”)  is  a  biopharmaceutical  research  and  development  company  engaged  in  the 
development  of  high-value  human  therapeutics,  specializing  in  oncology.  CytRx’s  drug  development  pipeline  includes  clinical 
development  of  three  product  candidates  for  cancer  indications,  including  three  planned  Phase  2  clinical  trials  for  INNO-206  as  a 
treatment for pancreatic cancer, gastric (stomach) cancer and soft tissue sarcomas, two Phase 2 proof-of-concept clinical trials with 
bafetinib in patients with high-risk B-cell chronic lymphocytic leukemia, or B-CLL, and patients with glioblastoma multiforme, and a 
registration  study  of  tamibarotene  for  the  treatment  of  acute  promyelocytic  leukemia,  or  APL.  In  addition  to  its  core  oncology 
programs, CytRx is developing two drug candidates based on its molecular chaperone regulation technology, which aim to repair or 
degrade  mis-folded  proteins  associated  with  disease.  Apart  from  its  drug  development  programs,  CytRx  currently  maintain  a  36% 
equity  interest  in  its  former  subsidiary,  RXi.  The  Company’s  current  business  strategy  for  its  molecular  chaperone  regulation 
technology is to seek one or more strategic partnerships, or a possible spin-out transaction. 

At December 31, 2009, the Company had cash and cash equivalents of approximately $9.9 million, marketable securities of $22.8 
million and held 5,768,881 shares of restricted common stock of RXi Pharmaceuticals Corporation, or RXi, with a market value of 
$26.4  million  based  upon  the  closing  price  of  the  RXi  common  stock  on  that  date.  On  July  27,  2009,  the  Company  raised 
approximately $18.3 million, net of fees and expenses, in a registered direct offering, and on September 23, 2009, the Company raised 
approximately $1.2 million, net of fees, from the sale of 500,000 shares of its common stock of RXi. Management believes that the 
Company’s current cash on hand, together with its marketable securities and proceeds from possible future sale of RXi common stock, 
will  be  sufficient  to  fund  its  operations  for  the  foreseeable  future.  The  estimate  is  based,  in  part,  upon  the  Company’s  currently 
projected expenditures for 2010 of approximately $18.0 million (unaudited), which includes approximately $3.2 million (unaudited) 
for its clinical programs for INNO-206, approximately $1.6 million (unaudited) for its clinical programs for bafetinib, approximately 
$2.5  million  (unaudited)  for  its  clinical  program  for  tamibarotene,  approximately  $1.4  million  (unaudited)  for  its  activities  for 
arimoclomol, approximately $2.2 million (unaudited) for general operation of its clinical programs, and approximately $7.1 million 
(unaudited)  for  other  general  and  administrative  expenses.  These  projected  expenditures  are  also  based  upon  numerous  other 
assumptions  and  subject  to  many  uncertainties,  and  actual  expenditures  may  be  significantly  different  from  these  projections.  The 
Company will be required to obtain additional funding in order to execute its long-term business plans, although it does not currently 
have commitments from any third parties to provide it with capital. The fair value of common stock investment in RXi is subject to 
market  fluctuations  that  could  impact  the  amount  of  cash  the  Company  generates  from  the  sale  of  RXi  shares  in  the  future.  The 
Company cannot assure that additional funding will be available on favorable terms, or at all. If the Company fails to obtain additional 
funding  when  needed,  it  may  not  be  able  to  execute  its  business  plans  and  its  business  may  suffer,  which  would  have  a  material 
adverse effect on its financial position, results of operations and cash flows. 

2. Summary of Significant Accounting Policies 

Basis  of  Presentation  and  Principles  of  Consolidation  —  Through  February  2008,  the  Company  owned  a  majority  of  the 
outstanding shares of common stock of RXi, which was founded in April 2006 by the Company and four researchers in the field of 
RNAi,  including  Dr.  Craig  Mello,  recipient  of  the  2006  Nobel  Prize  for  Medicine  for  his  co-discovery  of  RNAi.  While  RXi  was 
majority-owned, the Company’s consolidated financial statements reflected 100% of the assets and liabilities and results of operations 
of RXi, with the interests of the minority shareholders of RXi recorded as “noncontrolling interests.” In March 2008, the Company 
distributed to its stockholders approximately 36% of RXi’s outstanding shares, which reduced CytRx’s ownership to less than 50% of 
RXi. As a result of the reduced ownership, CytRx began to account for its investment in RXi using the equity method, under which 
CytRx  records  only  its  pro-rata  share  of  the  financial  results  of  RXi  as  “equity  in  loss  of  unconsolidated  subsidiary”  on  the 
consolidated  statements  of  operations  (see  Note  14  below).  Because  a  portion  of  RXi’s  financial  results  for  2008  and  all  of  RXi’s 
financial  results  for  2007  were  not  recorded  by  CytRx  under  the  equity  method,  the  Company’s  results  of  operations  for  the  year 
ended December 31, 2009 are not directly comparable to results of operations for the same periods in prior years. 

Revenue  Recognition  —  Revenue  consists  of  license  fees  from  strategic  alliances  with  pharmaceutical  companies  as  well  as 
service  and  grant  revenues.  Service  revenue  consists  of  contract  research  and  laboratory  consulting.  Grant  revenues  consist  of 
government and private grants. 

F-7 

  
  
  
  
  
  
  
 
 
Monies  received  for  license  fees  are  deferred  and  recognized  ratably  over  the  performance  period  in  accordance  with  Staff 
Accounting  Bulletin  (“SAB”)  No.  104,  Revenue  Recognition.  Milestone  payments  will  be  recognized  upon  achievement  of  the 
milestone as long as the milestone is deemed substantive and we have no other performance obligations related to the milestone and 
collectability is reasonably assured, which is generally upon receipt, or recognized upon termination of the agreement and all related 
obligations. Deferred revenue represents amounts received prior to revenue recognition. 

Revenues from contract research, government grants, and consulting fees are recognized over the respective contract periods as 
the services are performed, provided there is persuasive evidence or an arrangement, the fee is fixed or determinable and collection of 
the  related  receivable  is  reasonably  assured.  Once  all  conditions of  the  grant  are  met  and no  contingencies remain  outstanding,  the 
revenue is recognized as grant fee revenue and an earned but unbilled revenue receivable is recorded. 

In  August  2006,  the  Company  received  approximately  $24.3  million  in  proceeds  from  the  privately-funded  ALS  Charitable 
Remainder  Trust  (“ALSCRT”)  in  exchange  for  the  commitment  to  continue  research  and  development  of  arimoclomol  and  other 
potential treatments for ALS and a one percent royalty in the worldwide sales of arimoclomol. Under the arrangement, we retain the 
rights to any products or intellectual property funded by the arrangement and the proceeds of the transaction are non-refundable. The 
ALSCRT has no obligation to provide any further funding to the Company. The Company has concluded that due to the research and 
development  components  of the  transaction  that  it  is  properly  accounted  for  under  ASC  730-20  (previously  Statement  of  Financial 
Accounting  Standards  No.  68,  Research  and  Development  Arrangements).  Accordingly,  the  Company  recorded  the  value  received 
under  the  arrangement  as  deferred  service  revenue  and  recognized  service  revenue  using  the  proportional  performance  method  of 
revenue recognition, meaning that service revenue was recognized on a dollar-for-dollar basis for each dollar of expense incurred for 
the research and development of arimoclomol and other potential ALS treatments. CytRx believes that this method best approximates 
the efforts expended related to the services provided. The Company adjusted its estimates of expense incurred for this research and 
development on a quarterly basis. 

The amount of “deferred revenue, current portion” is the amount of deferred revenue that is expected to be recognized in the next 
twelve  months  and  is  subject  to  fluctuation  based  upon  management’s  estimates.  Management’s  estimates  include  an  evaluation of 
what pre-clinical and clinical trials are necessary, the timing of when trials will be performed and the estimated clinical trial expenses. 
These estimates are subject to changes and could have a significant effect on the amount and timing of when the deferred revenues are 
recognized. 

Pursuant to an amendment signed between the Company and the beneficiary of the ALSCRT on August 6, 2009, the Company 
was  released  from  all  restrictions  on  the  use  of  any  proceeds  previously  received  by  us  in  connection  with  the  arrangement.  As  a 
result, the Company recognized $6.7 million as service revenue in the third quarter of 2009, which represented the remaining deferred 
revenue and previously un-recognized portion of the value received. For the years ended December 31, 2009 and 2008, the Company 
recognized approximately $9.4 million and $6.2 million, respectively, of service revenue related to this transaction. 

Other Income — The Company realized a net gain of $0.1 million in 2009 on the sub-lease of its New York city rental property 
inherited on the acquisition of Innovive. In March 2008, the Company recognized a non-cash gain of $0.2 million on the transfer of some 
RXi  common  stock  to  certain  employees.  In  June  2007,  the  Company  recognized  $1.5  million  of  income  arising  from  a  fee  received 
pursuant to a change-in-control provision included in the purchase agreement for its 1998 sale of its animal pharmaceutical unit. 

Cash Equivalents — The Company considers all highly liquid debt instruments with an original maturity of 90 days or less to be 

cash equivalents. Cash equivalents consist primarily of amounts invested in money market accounts. 

Marketable securities — Investment securities held by the Company are classified as available for sale. 

Fair  Value  of  Financial  Instruments  —  The  carrying  amounts  reported  in  the  balance  sheet  for  cash  and  cash  equivalents  and 

marketable securities approximate their fair values. 

Equipment and Furnishings — Equipment and furnishings are stated at cost and depreciated using the straight-line method based 
on  the  estimated  useful  lives  (generally  three  to  five  years  for  equipment  and  furniture)  of  the  related  assets.  Whenever  there  is  a 
triggering event that might suggest an impairment, management evaluates the realizability of recorded long-lived assets to determine 
whether their carrying values have been impaired. The Company records impairment losses on long-lived assets used in operations 
when events and circumstances indicate that the assets might be impaired and the non-discounted cash flows estimated to be generated 
by those assets are less than the carrying amount of those assets. Any impairment loss is measured by comparing the fair value of the 
asset to its carrying amount. 

F-8 

  
  
  
  
  
  
  
  
  
 
Fair  Value  Measurements  —  The  Company  adopted  new  guidance  which  is  now  part  of  ASC  820-10  (formerly  Financial 
Accounting  Standards  Board  Statement  of  Financial  Accounting  Standards  No.  157),  Fair  Value  Measurements  (“FAS  157”), 
effective January  1,  2008.  SFAS 157  does not require  any  new  fair  value  measurements;  instead  it  defines fair value,  establishes  a 
framework  for  measuring  fair  value  in  accordance  with  existing  generally  accepted  accounting  principles  and  expands  disclosure 
about fair value measurements. The adoption of SFAS 157 for the Company’s financial assets and liabilities did not have an impact on 
its  financial  position  or  operating  results.  Beginning  January  1,  2008,  assets  and  liabilities  recorded  at  fair  value  in  consolidated 
balance  sheets  are  categorized  based  upon  the  level  of  judgment  associated  with  the  inputs  used  to  measure  the  fair  value.  Level 
inputs, as defined by SFAS 157, are as follows: 

•  Level 1 – quoted prices in active markets for identical assets or liabilities. 

•  Level  2  –  other  significant  observable  inputs  for  the  assets  or  liabilities  through  corroboration  with  market  data  at  the 

measurement date. 

•  Level 3 – significant unobservable inputs that reflect management’s best estimate of what market participants would use to 

price the assets or liabilities at the measurement date. 

The following table summarizes fair value measurements by level at December 31, 2009 for assets and liabilities measured at fair 

value on a recurring basis: 

(In thousands) 
Cash and cash equivalents . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . $
Marketable securities . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .
Warrant Liability . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .

Level I

Level II

Level III

Total

9,894  $
22,750 
—

— $ 
—
3,371

— $
—
—

9,894
22,750
3,371

The following table summarizes fair value measurements by level at December 31, 2008 for assets and liabilities measured at fair 

value on a recurring basis: 

(In thousands) 
Cash and cash equivalents . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . $

Level I

Level II

Level III

Total

25,042  $

— $ 

— $

25,042

Liabilities  measured  at  market  value  on  a  recurring  basis  include  warrant  liabilities  resulting  from  recent  debt  and  equity 
financing. In accordance with ASC 815-40 (formerly EITF 00-19, Accounting for Derivative Financial Instruments Indexed to, and 
Potentially  Settled  in,  a  Company’s  Own  Stock),  the  warrant  liabilities  are  being  marked  to  market  each  quarter-end  until  they  are 
completely  settled.  The  warrants  are  valued  using  the  Black-Scholes  method,  using  assumptions  consistent  with  the  Company’s 
application of ASC 505-50. See Warrant Liabilities below. 

The  Company  considers  carrying  amounts  of  accounts  receivable,  accounts  payable  and  accrued  expenses  to  approximate  fair 

value due to the short-term nature of these financial instruments.  

F-9 

  
 
 
 
 
 
 
 
  
 
 
The  Company’s  non-financial  assets,  such  as  assets  held  for  sale  are  measured  at  fair  value  when  there  is  an  indicator  of 
impairment and recorded at fair value only when an impairment charge is recognized. The following table summarizes the Company’s 
financial assets measured at fair value on a nonrecurring basis as of December 31, 2009: 

Carrying 
Amount as of 
December 31, 
2009

Level 1

Fair Value Measurements  
as of December 31, 2009  
Level 3 
Level 2

  Total Losses

(in thousands) 
Long-lived assets held for sale: 

Plant and equipment, net . . . . . . . . . . . . . . . . . . . . . . . . $
Asssets held for sale . . . . . . . . . . . . . . . . . . . . . . . . . . . . $

74
74

$
$

— $
— $

74
74

$ 
$ 

— $ 
— $ 

1,187 
1,187 

Impairment  of  Long-Lived  Assets  —  The  Company  reviews  long-lived  assets,  including  finite  lived  intangible  assets,  for 
impairment on an annual basis, as of December 31, or on an interim basis if an event occurs that might reduce the fair value of such 
assets below their carrying values. An impairment loss would be recognized based on the difference between the carrying value of the 
asset and its estimated fair value, which would be determined based on either discounted future cash flows or other appropriate fair 
value methods. If the Company’s estimates used in the determination of either discounted future cash flows or other appropriate fair 
value methods are not accurate as compared to actual future results, the Company may be required to record an impairment charge. 
The  fixed  assets,  from  the  Company’s  San  Diego  laboratory  and  its  molecular  library,  available  for  sale  were  re-allocated  from 
Equipment and Furnishings to Assets Held for Sale and were written down to their estimated net realizable value as of September 30, 
2009 (see Note7 below). 

Patents  and  Patent  Application  Costs  —  Although  the  Company  believes  that  its  patents  and  underlying  technology  have 
continuing  value,  the  amount  of  future  benefits  to  be  derived  from  the  patents  is  uncertain.  Patent  costs  are  therefore  expensed  as 
incurred. 

Net Income (Loss) Per Share — Basic net income (loss) per common share has computed using the weighted-average number of 
common shares outstanding. Diluted net income (loss) per common share computed using the weighted-average number of common 
share and common share equivalents outstanding. Common share equivalents which could potentially dilute basic earnings per share 
in the future, and which were excluded from the computation of diluted loss per share, totaled approximately 24.4 million shares, 15.2 
million shares and 17.1 million shares at December 31, 2009, 2008 and 2007, respectively. 

As a result of the March 11, 2008 distribution by CytRx to its stockholders of approximately 36% of the outstanding shares of 
RXi Pharmaceuticals Corporation, the Company recorded a deemed dividend of approximately $757,000. The deemed dividend was 
reflected  as  an  adjustment  to  net  loss  for  the  first  quarter  of  2008  to  arrive  at  net  loss  applicable  to  common  stockholders  on  the 
consolidated statement of operations and for purposes of calculating basic and diluted earnings per shares. 

Warrant  Liabilities  —  Liabilities  measured  at  market  value  on  a  recurring  basis  include  warrant  liabilities  resulting  from  our 
recent  equity  financing.  In  accordance  with  ASC  815-40  (formerly  EITF  (Emerging  Issues  Task  Force)  00-19,  Accounting  for 
Derivative  Financial  Instruments  Indexed  to  and  Potentially  Settled  in  a  Company’s  Own  Stock,  the  warrant  liabilities  are  being 
marked to market each quarter-end until they are completely settled. The warrants are valued using the Black-Scholes method. The 
gain  or  loss  resulting  from  the  marked  to  market  calculation  is  shown  on  the  Consolidated  Statements  of  Operations  as  Gain  on 
warrant derivative liability. 

Shares Reserved for Future Issuance — As of December 31, 2009, the Company has reserved approximately 9.1 million of its 
authorized but unissued shares of common stock for future issuance pursuant to its employee stock option plans issued to consultants 
and investors. 

Stock-based  Compensation  —  The  Company’s  stock-based  employee  compensation  plans  are  described  in  Note  15.  The 
Company  has  adopted  the  provisions  of  ASC  718  (previously  SFAS  No.  123(R),  Share-Based  Payment  (“SFAS  123(R)”)),  which 
requires  the  measurement  and  recognition  of  compensation  expense  for  all  stock-based  awards  made  to  employees  and  non-
employees. 

F-10 

 
 
 
  
  
  
  
        
 
 
  
  
  
  
  
  
 
 
For  stock  options  and  stock  warrants  paid  in  consideration  of  services  rendered  by  non-employees,  the  Company  recognizes 
compensation  expense  in  accordance  with  the  requirements  of  ASC  718  (previously  SFAS  No.  123(R)),  ASC  505-50  (previously 
Emerging  Issues  Task  Force  Issue  No.  96-18  (“EITF  96-18”)),  Accounting  for  Equity  Instruments  that  are  Issued  to  other  than 
Employees  for  Acquiring,  or  in  Conjunction  with  Selling  Goods  or  Services  and  ASC  505  (previously  EITF  00-18,  Accounting 
Recognition for Certain Transactions involving Equity Instruments Granted to Other Than Employees), as amended. 

Non-employee option grants that do not vest immediately upon grant are recorded as an expense over the vesting period. At the 
end of each financial reporting period prior to performance, the value of these options, as calculated using the Black-Scholes option-
pricing model, is determined, and compensation expense recognized or recovered during the period is adjusted accordingly. Since the 
fair  market  value  of  options  granted  to  non-employees  is  subject  to  change  in  the  future,  the  amount  of  the  future  compensation 
expense is subject to adjustment until the common stock options or warrants are fully vested. 

Research and Development Expenses — Research and development expenses consist of costs incurred for direct and overhead-
related research expenses and are expensed as incurred. Costs to acquire technologies, including licenses, that are utilized in research 
and development and that have no alternative future use are expensed when incurred. Technology developed for use in its products is 
expensed as incurred until technological feasibility has been established. 

Clinical Trial Expenses — Clinical trial expenses, which are included in research and development expenses, include obligations 
resulting from the Company’s contracts with various clinical research organizations in connection with conducting clinical trials for its 
product candidates. The Company recognize expenses for these activities based on a variety of factors, including actual and estimated 
labor hours, clinical site initiation activities, patient enrollment rates, estimates of external costs and other activity-based factors. The 
Company  believe  that  this  method  best  approximates  the  efforts  expended  on  a  clinical  trial  with  the  expenses  it  records.  The 
Company adjusts its rate of clinical expense recognition if actual results differ from its estimates. If its estimates are incorrect, clinical 
trial expenses recorded in any particular period could vary. 

Income Taxes — Income taxes are accounted for using an asset and liability approach that requires the recognition of deferred tax 
assets  and  liabilities  for  the  expected  future  tax  consequences  of  events  that  have  been  recognized  in  the  Company’s  financial 
statements or tax returns. A valuation allowance is established to reduce deferred tax assets if all, or some portion, of such assets will 
more  than  likely  not  be  realized.  Effective  January  1,  2007,  we  adopted  the  provisions  of  ASC  740-10  (formerly  FIN  48),  which 
contains a two-step process for recognizing and measuring uncertain tax positions. The first step is to determine whether or not a tax 
benefit  should  be  recognized.  A  tax benefit  will  be  recognized  if  the  weight  of  available  evidence  indicates  that  the  tax position  is 
more likely than not to be sustained upon examination by the relevant tax authorities. The recognition and measurement of benefits 
related to our tax positions requires significant judgment, as uncertainties often exist with respect to new laws, new interpretations of 
existing laws, and rulings by taxing authorities. Differences between actual results and our assumptions or changes in our assumptions 
in future periods are recorded in the period they become known. 

Concentrations of Risks — Financial instruments that potentially subject the Company to significant concentrations of credit risk 
consist  principally  of  cash,  cash  equivalents  and  marketable  securities.  The  Company  maintains  cash  and  cash  equivalents  in  large 
well-capitalized financial institutions and the Company’s investment policy disallows investment in any debt securities rated less than 
“investment-grade”  by  national  ratings  services.  The  Company  has  not  experienced  any  losses  on  its  deposits  of  cash  or  cash 
equivalent  or  its  marketable  securities.  The  Company  also  has  a  36%  investment  in  RXi,  the  shares  of  which  can  significantly 
fluctuate.  The  sale  of  these  common  shares  represents  a  future  source  of  cash  and  any  decline  in  the  share  price  can  impact  the 
Company. 

Use of Estimates — The preparation of the financial statements in conformity with accounting principles generally accepted in the 
United States of America requires management to make estimates and assumptions that affect the amounts reported in the financial 
statements and accompanying notes. Significant estimates include the accrual for research and development expenses, the basis for the 
classification of current deferred revenue, estimated income taxes and the estimate of expense arising from the common stock options 
granted to employees and non-employees. Actual results could materially differ from those estimates. 

Other  comprehensive  income/(loss)  —  The  Company  follows  the provisions of ASC  220, (formerly  SFAS No.  130,  Reporting 
Comprehensive Income), which requires separate representation of certain transactions, which are recorded directly as components of 
shareholders’ equity. The Company has no components of other comprehensive income (loss) and accordingly comprehensive loss is 
the same as net loss reported. 

F-11 

  
  
  
  
 
  
  
 
 
3. Recent Accounting Pronouncements 

In  December  2007,  the  FASB  issued  guidance  which  is  now  part  of  ASC  810-10,  Noncontrolling  Interests  in  Consolidated 
Financial  Statements,  an  Amendment  of  Accounting  Research  Bulletin  No.  51  “  (formerly  Statement  of  Financial  Accounting 
Standards  (SFAS)  160,  Noncontrolling  Interests  in  Consolidated  Financial  Statements—an  amendment  of  ARB  No.  51  ).  This 
guidance establishes accounting and reporting standards for ownership interests in subsidiaries held by parties other than the parent, 
changes in a parent’s ownership of a noncontrolling interest, calculation and disclosure of the consolidated net income attributable to 
the parent  and  the noncontrolling  interest, changes  in  a parent’s ownership  interest while  the parent  retains  its  controlling  financial 
interest  and  fair  value  measurement  of  any  retained  noncontrolling  equity  investment.  The  new  guidance  is  effective  for  financial 
statements issued for fiscal years beginning after December 15, 2008, and interim periods within those fiscal years. Early adoption is 
prohibited. The Company adopted this guidance on January 1, 2009, the beginning of its 2009 fiscal year, which resulted in certain 
reclassifications related to the noncontrolling interest in the consolidated financial statements. 

In  March  2008,  the  FASB  issued  guidance  ASC  815-10  (formerly  Statement  of  Financial  Accounting  Standards  No.  161, 
Disclosures about Derivative Instruments and Hedging Activities (“SFAS No. 161”). The new standard amends Statement of Financial 
Accounting Standards No. 133, Accounting for Derivative Instruments and Hedging Activities (“SFAS 133”), and seeks to enhance 
disclosure about how and why a company uses derivatives; how derivative instruments are accounted for under SFAS 133 (and the 
interpretations  of  that  standard);  and  how  derivatives  affect  a  company’s  financial  position,  financial  performance  and  cash  flows. 
SFAS 161 will be effective for financial statements issued for fiscal years and interim periods beginning after November 15, 2008. 
Early application of the standard is encouraged, as well as comparative disclosures for earlier periods at initial adoption. The adoption 
of ASC 815-10 did not have a material impact on the Company’s consolidated financial statements. 

In April 2008, the FASB issued revised guidance on determining the useful life of intangible assets. The revised guidance, which 
is now part of ASC 350-30 General Intangibles Other than Goodwill (previously Staff Position No. FAS 142-3, Determination of the 
Useful Life of Intangible Assets), amends the factors that should be considered in developing renewal or extension assumptions used to 
determine the useful life of a recognized intangible asset. The Position is effective for fiscal years beginning after December 15, 2008 
and applies prospectively to intangible assets acquired after the effective date. Early adoption is not permitted. The adoption of SFAS 
No. ASC 350-30 did not have a material impact on the Company’s consolidated financial statements. 

In May 2008, the FASB issued revised guidance on Convertible Debt Instruments. The revised guidance which is now part of 
ASC 470-20 (formerly Staff Position No. Accounting Principles Board 14-1, Accounting for Convertible Debt Instruments That May 
Be  Settled  in  Cash  upon  Conversion  (Including  Partial  Cash  Settlement)  (“FSP  No.  APB  14-1”)).  ASC  470-20  requires  that  the 
liability and equity components of convertible debt instruments that may be settled in cash upon conversion (including partial cash 
settlement)  be  separately  accounted  for  in  a  manner  that  reflects  an  issuer’s  nonconvertible  debt  borrowing  rate.  ASC  470-20  is 
effective for us as of January 1, 2009. The adoption of ASCO 470-20 did not have an impact on the Company’s consolidated financial 
statements. 

In June 2008, the FASB ratified guidance which is now part of ASC 815-40, Contracts in Entity’s Own Equity (formerly EITF 
(Emerging  Issues  Task  Force)  07-05),  Determining  Whether  an  Instrument  (or  Embedded  Feature)  Is  Indexed  to  an  Entity’s  Own 
Stock. The objective of this issue is to provide guidance for determining whether an equity-linked financial instrument (or embedded 
feature) is indexed to an entity’s own stock. This issue applies to any freestanding financial instrument or embedded feature that has 
all the characteristics of a derivative instrument or an instrument which may be potentially settled in an entity’s own stock regardless 
of  whether  the  instrument  possess  derivative  characteristics.  This  issue  provides  a  two-step  approach  to  assist  in  making  these 
determinations and is effective for financial statements issued for fiscal years beginning after December 15, 2008. The adoption of 
ASC 815-40 did not have a material impact on the Company’s consolidated financial statements. 

In  April  2009,  the  FASB  issued  guidance  which  is  now  part  of  ASC  825-10  Financial  Instruments  (formerly  Financial  Staff 
Position SFAS 107-1 and Accounting Principles Board (APB) Opinion No. 28-1, Interim Disclosures about Fair Value of Financial 
Instruments  (SFAS  107-1  and  APB  28-1).  This  statement  amends  FASB  Statement  No.  107,  Disclosures  about  Fair  Values  of 
Financial  Instruments,  to  require  disclosures  about  fair  value  of  financial  instruments  in  interim  financial  statements  as  well  as  in 
annual  financial  statements.  The  statement  also  amends  APB  Opinion  No.  28,  “Interim  Financial  Reporting,”  to  require  those 
disclosures in all interim financial statements. This statement is effective for interim periods ending after June 15, 2009. The adoption 
of ASC 825-10 did not have an impact on the Company’s financial statements. 

F-12 

  
  
  
  
  
  
 
 
In May 2009 and February 2010, the FASB issued new guidance for accounting for subsequent events. The new guidance, which 
is  now  part  of  ASC  855-10,  Subsequent  Events  (formerly,  SFAS  No.  165,  Subsequent  Events)  is  consistent  with  existing  auditing 
standards  in  defining  subsequent  events  as  events  or  transactions  that  occur  after  the  balance  sheet  date  but  before  the  financial 
statements are issued or are available to be issued. The new guidance defines two types of subsequent events: “recognized subsequent 
events”  and  “non-recognized  subsequent  events.”  Recognized  subsequent  events  provide  additional  evidence  about  conditions  that 
existed  at  the  balance  sheet  date  and  must  be  reflected  in  the  company’s  financial  statements.  Non-recognized  subsequent  events 
provide  evidence  about  conditions  that  arose  after  the  balance  sheet  date  and  are  not  reflected  in  the  financial  statements  of  a 
company. Certain non-recognized subsequent events may require disclosure to prevent the financial statements from being misleading. 
The  new  guidance  was  effective  on  a  prospective  basis  for  interim  or  annual  periods  ending  after  June  15,  2009.  The  Company 
adopted the provisions of ASC 855-10 as required. 

In  June  2009,  the  FASB  amended  ASC  860,  (formerly  SFAS  No.  166,  Accounting  for  Transfers  of  Financial  Assets,  an 
amendment to SFAS No. 140). ASC 860 eliminates the concept of a “qualifying special-purpose entity,” changes the requirements for 
derecognizing  financial  assets,  and  requires  additional  disclosures  in  order  to  enhance  information  reported  to  users  of  financial 
statements by providing greater transparency about transfers of financial assets, including securitization transactions, and an entity’s 
continuing  involvement  in  and  exposure  to  the  risks  related  to  transferred  financial  assets.  ASC  860  is  effective  for  fiscal  years 
beginning  after  November  15,  2009.  The  Company  will  adopt  ASC  860  in  fiscal  2010.  The  Company  does  not  expect  that  the 
adoption of ASC 860 will have a material impact on its financial statements. 

In  June  2009,  the  FASB  amended  ASC  810  (formerly  SFAS  No.167,  Amendments  to  FASB  Interpretation  No.  46).  The 
amendments include: (1) the elimination of the exemption for qualifying special purpose entities, (2) a new approach for determining 
who  should  consolidate  a  variable-interest  entity,  and  (3)  changes  to  when  it  is  necessary  to  reassess  who  should  consolidate  a 
variable-interest entity. ASC 810 is effective for the first annual reporting period beginning after November 15, 2009 and for interim 
periods within that first annual reporting period. The Company will adopt ASC 810 in fiscal 2010. The Company does not expect that 
the adoption of ASC 810 will have a material impact on its financial statements. 

In  June  2009,  the  FASB  issued  new guidance  which  is  now  part  of  ASC  105-10  (formerly  Statement  of  Financial Accounting 
Standards No. 168, The FASB Accounting Standards Codification and the Hierarchy of Generally Accepted Accounting Principles ). 
ASC 105-10 replaces FASB Statement No. 162, “The Hierarchy of Generally Accepted Accounting Principles”, and establishes the 
FASB Accounting Standards Codification as the source of authoritative accounting principles recognized by the FASB to be applied 
by nongovernmental entities in the preparation of financial statements in conformity  with generally accepted accounting principles. 
ASC 105-10 is effective for interim and annual periods ending after September 15, 2009. The adoption of ASC 105-10 did not have a 
material impact on the Company’s financial statements. 

In January, 2010, the FASB issued ASU 2010-06, Improving Disclosures about Fair Value Measurements. The standard amends 
ASC Topic 820, Fair Value Measurements and Disclosures to require additional disclosures related to transfers between levels in the 
hierarchy of fair value measurement. The standard does not change how fair values are measured. The standard is effective for interim 
and annual reporting periods beginning after December 15, 2009. As a result, it is effective for us in the first quarter of fiscal year 
2010. We do not believe that the adoption of ASU 2010-06 will have a material impact on consolidated our financial statements. 

4. Receivable 

At December 31, 2009 and 2008, the Company had a receivable of $139,680 and $127,280, respectively, primarily related to annual 

licensing fees due to the Company. Due to the certainty of the collectability of the accounts receivable, no allowance was recorded. 

5. Other Assets 

At  December  31,  2009  and  2008,  the  Company  had  $323,235  and  $330,032,  respectively,  of  non-current  other  assets,  which 

consist primarily of security deposits on contracts for research and development, prepaid insurance and leases for its facilities. 

6. Marketable securities 

The Company held $22.8 million of marketable securities at December 31, 2009. The Company has classified these investments 
as available for sale. These investments are comprised of federally insured certificates of deposit and these four accounts detailed as 
follows: $5.0 million with a maturity date of January 28, 2010; $8.8 million with a maturity date of April 1, 2010; $5 million with a 
maturity date of July 29, 2010; and $4 million with a maturity date of September 30, 2010. 

F-13 

 
  
  
  
  
  
  
  
  
  
 
7. Assets Held for Sale 

In May 2009, the Company substantially completed the initial phase of the closure of its drug discovery research at its laboratory 
facility in San Diego, California. The Company concluded that it will conduct its research and development activities through third 
parties  for  the  foreseeable  future.  The  Company  has  sublet  the  laboratory  facility,  sold  some  of  the  laboratory  equipment  and  is 
actively  searching  for  additional  buyers.  In  the  third  quarter  of  2009,  the  fixed  assets  related  to  the  San  Diego  laboratory  were  re-
allocated from Equipment and Furnishings to Assets Held for Sale and were written down to their estimated net realizable value as of 
September  30,  2009,  which resulted  in  a  charge of $1.2 million  for  that  quarter.  In November  2009,  the  Company  signed  sublease 
agreements  with  two  parties  to  sublet  the  facility  for  the  remainder  of  the  term  of  the  lease,  which  expires  in  October,  2010.  The 
Company recognized an onerous lease accrual of $254,000 as of September 2009. 

Assets held for sale consisted of the following: 

(in thousands) 
Long-lived assets held for sale: 

Plant and equipment, net . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .
Asssets held for sale . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .

December 31,

2009 

2008

$
$

74 
74 

$
$

—
—

As of December 31, 2009, the carrying amount approximates fair value. The costs associated with disposing of these assets held 

for sale are minimal. 

8. Equipment, Furnishings and Molecular Library, net 

Equipment, furnishings and molecular library, net, at December 31, 2009 and 2008 consist of the following (in thousands): 

Equipment and furnishings . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .     $ 
Less — accumulated depreciation . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .       
Equipment and furnishings, net . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .       

Molecular library . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .     $ 
Less — accumulated amortization  . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .       
Molecular library, net . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .     $ 

2009 

2008

334    $
(159)    
175     

0    $
0     
0    $

2,606 
(771)
1,835 

447 
(343)
104 

The molecular library was purchased in 2004 and placed in service by the Company in March 2005. In the third quarter of 2009, 

the molecular library was re-allocated to Assets Held for Sale and was written down to its estimated net realizable value. 

Depreciation  and  amortization  expense  for the  years  ended  December 31, 2009, 2008 and 2007 were  approximately  $475,000, 

$625,000 and $272,000, respectively. 

9. Accrued Expenses and Other Current Liabilities 

Accrued expenses and other current liabilities at December 31, 2009 and 2008 are summarized below (in thousands). 

Professional fees . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .     $ 
Research and development costs . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .       
Wages, bonuses and employee benefits . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .       
Income taxes . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .       
Other . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .       
Total . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .     $ 

423    $
1,255     
208     
—     
606     
2,492    $

531 
1,662 
196 
— 
168 
2,557 

2009 

2008

F-14 

  
  
  
 
 
  
  
 
  
  
  
  
  
  
   
 
    
     
 
 
  
  
  
  
  
  
   
 
 
 
 
10. Warrant Liabilities 

Liabilities  measured  at  market  value  on  a  recurring  basis  include  warrant  liabilities  resulting  from  the  Company’s  2009  equity 
financing. In accordance with the guidance which is now ASC 815-40 (formerly EITF (Emerging Issues Task Force) 00-19, Accounting 
for Derivative Financial Instruments Indexed and Potentially Settled in a Company’s Own Stock), the warrant liabilities are being marked 
to market each quarter-end until they are completely settled. The warrants are valued using the Black-Scholes method, using assumptions 
consistent  with  our  application  of  ASC  505-50.  The  gain  or  loss  resulting  from  the  marked  to  market  calculation  is  shown  on  the 
Consolidated Statements of Operations as Gain on warrant derivative liability. The Company recognized a gain of $657,000 during 2009. 

11. Commitments and Contingencies 

The Company acquires assets still in development and enters into research and development arrangements with third parties that 
often require milestone and royalty payments to the third party contingent upon the occurrence of certain future events linked to the 
success  of  the  asset  in  development.  Milestone  payments  may  be  required,  contingent  upon  the  successful  achievement  of  an 
important  point  in  the  development  life-cycle  of  the  pharmaceutical  product  (e.g.,  approval  of  the  product  for  marketing  by  a 
regulatory agency). If required by the arrangement, CytRx may have to make royalty payments based upon a percentage of the sales of 
the pharmaceutical product in the event that regulatory approval for marketing is obtained. Because of the contingent nature of these 
payments, they are not included in the table of contractual obligations. 

These arrangements may be material individually, and in the unlikely event that milestones for multiple products covered by these 
arrangements were reached in the same period, the aggregate charge to expense could be material to the results of operations in any 
one  period.  In  addition,  these  arrangements  often  give  CytRx  the  discretion  to  unilaterally  terminate  development  of  the  product, 
which  would  allow  CytRx  to  avoid  making  the  contingent  payments;  however,  CytRx  is  unlikely  to  cease  development  if  the 
compound successfully achieves clinical testing objectives. 

CytRx’s current contractual obligations that will require future cash payments are as follows (in thousands): 

Operating
Leases (1)(2)    

Employment
Agreements (3)   

Subtotal

Research and 
Development (4)    

Total

2010 . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .  $
2011 . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   
2012 . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   
2013 . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   
2014 and thereafter . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   
Total . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .  $
____________ 
(1)  Operating  leases  are  primarily  facility  lease  related  obligations,  as well  as  equipment  and  software  lease  obligations  with  third 

3,083    $ 
536      
459      
318      
372      
4,768    $ 

2,210    $
—     
—     
—     
—     
2,210    $

873    $
536     
459     
318     
372     
2,558    $

3,018    $
49     
149     
149     
383     
3,748    $

6,101 
585 
608 
467 
755 
8,516 

party vendors. 

(2)  The Company is entitled to receive future rental income under subleases in place which would be offset against future operating 

lease obligations as follows: $519,000 in 2010, $350,000 in 2011 and $235,000 in 2012. 

(3)  Employment agreements include management contracts, which have been revised from time to time, provide for minimum salary levels, 

adjusted annually at the discretion of the Company's Compensation Committee, as well as for minimum bonuses that are payable. 

(4)  Research and development obligations relate primarily to clinical trials. Most of these purchase obligations are cancelable. 

The Company applies the disclosure provisions of ASC 460 (formerly FASB Interpretation No. 45, Guarantor’s Accounting and 
Disclosure  Requirements  for  Guarantees,  Including  Indirect  Guarantees  of  Indebtedness  of  Others),  to  its  agreements  that  contain 
guarantee or indemnification clauses. The Company provides (i) indemnifications of varying scope and size to certain investors and 
other parties for certain losses suffered or incurred by the indemnified party in connection with various types of third-party claims; and 
(ii)  indemnifications  of  varying  scope  and  size  to  officers  and  directors  against  third  party  claims  arising  from  the  services  they 
provide to us. These indemnifications and guarantees give rise only to the disclosure provisions of ASC 460. To date, the Company 
has not incurred material costs as a result of these obligations and does not expect to incur material costs in the future; further, the 
Company maintains insurance to cover certain losses arising from these indemnifications. Accordingly, the Company has not accrued 
any liabilities in its consolidated financial statements related to these indemnifications or guarantees. 

F-15 

  
  
  
  
  
  
  
 
     
 
  
  
 
  
 
12. Equity Transactions 

On April 19, 2007, the Company completed a $37.0 million private equity financing in which it issued 8.6 million shares of its 
common  stock  at  $4.30  per  share.  Net  of  investment  banking  commissions,  legal,  accounting  and  other  expenses  related  to  the 
transaction, the Company received approximately $34.2 million of proceeds. 

On  March  11,  2008,  the  Company  paid  a  dividend  to  its  stockholders  of  approximately  36%  of  the  outstanding  shares  of  RXi 
common stock. In connection with that dividend, the Company adjusted the price of warrants to purchase approximately 10.6 million 
shares that had been issued in prior equity financings in October 2004, January 2005 and March 2006. The adjustments were made as 
a result of anti-dilution provisions in those warrants that were triggered by the Company’s distribution of a portion of its assets to its 
stockholders. The Company accounted for the anti-dilution adjustments as deemed dividends analogous with the guidance in ASC 470 
(previously Emerging Issues Task Force Issue (“EITF”) No. 98-5, Accounting for Convertible Securities with Beneficial Conversion 
Features  or  Contingently  Adjustable  Conversion  Ratio)s,  and  ASC  470  (previously  EITF  00-27,  Application  of  98-5  to  Certain 
Convertible  Instruments),  and  recorded  an  approximate  $757,000  charge  to  accumulated  deficit  and  a  corresponding  credit  to 
additional paid-in capital. 

On July 27, 2009, the Company completed a $20.0 million registered direct public offering in which it issued approximately 15.3 
million shares of its common stock at a price of $1.31 per share, and warrants to purchase an additional approximately 4.7 million 
shares  of  common  stock  at  an  exercise  price  of  $1.70  per  share.  Net  of  investment  banking  commissions,  advisory  fees,  legal, 
accounting and other fees related to the transaction, the Company received proceeds of approximately $18.3 million (without giving 
effect to any proceeds that may in the future be received by the Company upon exercise of warrants sold in the offering). Immediately 
after  the  sale,  the  Company  had  approximately  109.5  million  shares  of  common  stock  outstanding,  without  giving  effect  to  the 
possible exercise of the warrants sold in the offering or any of our other outstanding warrants or stock options. 

13. Noncontrolling Interest in RXi 

Through February 2008, the Company owned approximately 85% of the outstanding shares of common stock of RXi. While RXi 
was  majority-owned,  the  Company’s  consolidated  financial  statements  reflected  100%  of  the  assets  and  liabilities  and  results  of 
operations of RXi, with the interests of the minority shareholders of RXi recorded as “noncontrolling interests.” The Company offset 
$88,000 of loss in noncontrolling interest of RXi against its net loss for the months of January and February 2008. 

On  March  11,  2008,  the  Company  distributed  to  its  stockholders  approximately  4.5  million  shares  of  RXi  common  stock,  or 
approximately 36% of RXi’s outstanding shares, which reduced the Company’s ownership to less than 50% of RXi. As a result, the 
Company  began  to  account  for  its  investment  in  RXi  using  the  equity  method, under which  the  Company  records  only  its  pro-rata 
share of the financial results of RXi. Because only a portion of RXi’s financial results for 2008 were recorded by the Company under 
the  equity  method,  the  Company’s  results  of  operations  for  2008  are  not  directly  comparable  to  results  of  operations  for  the  same 
period in 2009. The future results of operations of the Company also will not be directly comparable to corresponding periods in prior 
years during which our financial statements reflected the consolidation of RXi. 

14. Equity Investment in RXi 

Management determined that the distribution of RXi common stock to stockholders of CytRx in March 2008 represented a partial 
spin-off of RXi and accounted for the distribution of the RXi common shares at cost. As a result of its reduced ownership in RXi, 
CytRx began to account for its investment in RXi using the equity method, under which CytRx records only its pro-rata share of the 
financial results of RXi. The investment balance in RXi has been reduced to zero and the Company has not made any advances or 
guarantees to RXi. Therefore the Company has stopped recording its share of losses from RXi. 

F-16 

 
  
  
  
  
  
  
  
  
 
 
The following table presents summarized financial information for RXi for the years ended December 31, 2009 and 2008: 

Income Statement Data (in thousands)
Sales. . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   $
Gross profit . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Loss from continuing operations . . . . . . . . . . . . . .    
Net Loss . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    

Year Ended

December 31, 2009    

Year Ended 
December 31, 2008    
—  
—  
(14,553) 
(14,373) 

—    $
—     
(18,387)    
(18,387)    

Balance Sheet Data (in thousands)
Current assets . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   $
Noncurrent assets . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Current liabilities . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Stockholders’ equity . . . . . . . . . . . . . . . . . . . . . . . .    

  December 31, 2009     December 31, 2008    
9,929  
430  
1,387  
8,968  

5,805    $
448     
5,475     
743     

At December 31, 2009, the fair value of CytRx’s 5,768,881 shares of RXi common stock was $26.4 million based o the closing 
price of RXi common stock (NASDAQ: RXII) on that date. As CytRx accounts for its investment in RXi using the equity method, this 
value is not reflected 0n the CytRx balance sheet. 

15. Stock Options and Warrants 

CytRx Options 

The  Company  has  a  2000  Long-Term  Incentive  Plan  under  which  an  aggregate  of  10  million  shares  of  common  stock  were 
originally reserved for issuance. As of December 31, 2009, there were approximately 7.9 million shares subject to outstanding stock 
options and approximately 0.2 million shares available for future grant under this plan. 

On  July  1,  2009,  the  Company’s  stockholders  adopted  a  new  2008  Stock  Incentive  Plan  under  which  10  million  shares  of 
common  stock  were  reserved  for  issuance.  As  of  December  31,  2009,  there  were  1.1  million  shares  subject  to  outstanding  stock 
options under the plan and 8.9 million shares available for future grant under this plan. 

The Company has adopted the provisions of ASC 718 (previously SFAS No. 123(R), Share-Based Payment (“SFAS 123(R)”)), which 

requires the measurement and recognition of compensation expense for all stock-based awards made to employees and non-employees. 

For  stock  options  and  stock  warrants  paid  in  consideration  of  services  rendered  by  non-employees,  the  Company  recognizes 
compensation  expense  in  accordance  with  the  requirements  of  ASC  718  (previously  SFAS  No.  123(R)),  ASC  505-50  (previously 
Emerging  Issues  Task  Force  Issue  No.  96-18  (“EITF  96-18”)),  Accounting  for  Equity  Instruments  that  are  Issued  to  other  than 
Employees  for  Acquiring,  or  in  Conjunction  with  Selling  Goods  or  Services  and  ASC  505  (previously  EITF  00-18,  Accounting 
Recognition for Certain Transactions involving Equity Instruments Granted to Other Than Employees), as amended. 

Non-employee option grants that do not vest immediately upon grant are recorded as an expense over the vesting period. At the 
end of each financial reporting period prior to performance, the value of these options, as calculated using the Black-Scholes option-
pricing model, is determined, and compensation expense recognized or recovered during the period is adjusted accordingly. Since the 
fair  market  value  of  options  granted  to  non-employees  is  subject  to  change  in  the  future,  the  amount  of  the  future  compensation 
expense is subject to adjustment until the common stock options or warrants are fully vested. 

At  the  2009  Annual  Meeting  of  Stockholders  held  on  July  1,  2009,  the  Company’s  stockholders  approved  an  amendment  to  the 
Company’s 2000 Long-Term Incentive Plan to allow for a one-time stock option re-pricing program for employees and officers. Pursuant 
to  the  re-pricing  program,  3,265,500  eligible  stock  options  held  by  ten  eligible  employees  and  officers  were  amended  to  reduce  the 
exercise prices of the options to $1.15 per share, which was the closing sale price of CytRx’s common stock as reported on the Nasdaq 
Capital Market on the July 1, 2009 completion date of the re-pricing program, and to impose a new option vesting schedule. None of the 
amended options vested immediately. To the extent a participating employee’s or officer’s eligible options were vested on the amendment 
date, the amended options vested in full on December 31, 2009, so long as the employee or officer remained in the Company’s employ 
through  that  date.  To  the  extent  a  participating  employee’s  or  officer’s  eligible  options  were  unvested  as  of  July  1,  2009,  the  original 
scheduled vesting was suspended until December 31, 2009 and resumed after that date, so long as the employee or officer remained in the 
Company’s employ through such date. The incremental cost of the re-pricing program was approximately $0.4 million.

F-17 

  
 
 
 
  
  
  
  
  
  
  
  
ASC 718 (previously SFAS No. 123(R)) requires the re-pricing of equity awards to be treated as the repurchase of the old award 
for  a  new  award  of  equal  or  greater  value,  incurring  additional  compensation  cost  for  any  incremental  value.  This  incremental 
difference in value is measured as the excess of the fair value of the modified award determined in accordance with the provisions of 
ASC 718 over the fair value of the original award immediately before its terms are modified, measured based on the share price and 
other pertinent factors at that date. ASC 718 provides that this incremental fair value, plus the remaining unrecognized compensation 
cost from the original measurement of the fair value of the old option, must be recognized over the remaining vesting period. 

The fair value of the stock options at the date of grant was estimated using the Black-Scholes option-pricing model, based on the 

following assumptions: 

Risk-free interest rate . . . . . . . . .    
Expected volatility . . . . . . . . . . . .    
Expected lives (years) . . . . . . . . .    
Expected dividend yield . . . . . . .    

2009

2008

2007 

1.95%   
97%   
6      
0.00%   

2.68%   
102%   
6      
0.00%   

4.41%
108%
6  
0.00%

The  Company’s  computation  of  expected  volatility  is  based  on  the  historical  daily  volatility  of  its  publicly  traded  stock.  For 
option grants issued during years ended December 31, 2009, 2008 and 2007, the Company used a calculated volatility for each grant. 
The Company’s computation of expected lives was estimated using the simplified method provided for under ASC 718 (previously 
Staff Accounting Bulletin 107, Share-Based Payment (“SAB 107”)), which averages the contractual term of the Company’s options of 
ten years with the average vesting term of three years for an average of six years. The dividend yield assumption of zero is based upon 
the fact the Company has never paid cash dividends and presently has no intention of paying cash dividends. The risk-free interest rate 
used for each grant is equal to the U.S. Treasury rates in effect at the time of the grant for instruments with a similar expected life. 
Based on historical experience, for the year ended December 31, 2009, the Company has estimated an annualized forfeiture rate of 
14% for options granted to its employees, 2% for options granted to senior management and 0% for options granted to directors. For 
the years ended December 31, 2008 and 2007, the Company has estimated an annualized forfeiture rate for each period of 10% for 
options granted to its employees, 3% for options granted to senior management and 0% for options granted to directors. Compensation 
costs will be adjusted for future changes in estimated forfeitures. The Company will record additional expense if the actual forfeitures 
are  lower  than  estimated  and  will  record  a  recovery  of  prior  expense  if  the  actual  forfeiture  rates  are  higher  than  estimated.  No 
amounts relating to employee stock-based compensation have been capitalized. 

At  December  31,  2009,  there  remained  approximately  $2.5  million  of  unrecognized  compensation  expense  related  to  unvested 
stock options granted to current and former employees and directors, to be recognized as expense over a weighted-average period of 
1.12 years. Presented below is the Company’s stock option activity for employees and directors: 

2009 

Outstanding — beginning of year . . .        6,409,940     
Granted . . . . . . . . . . . . . . . . . . . . . . . . . . .        2,351,000     
Exercised . . . . . . . . . . . . . . . . . . . . . . . . .       
(8,333)    
Forfeited . . . . . . . . . . . . . . . . . . . . . . . . . .       
(713,018)    
Expired . . . . . . . . . . . . . . . . . . . . . . . . . . .       
(27,499)    
Outstanding — end of year . . . . . . . . .        8,012,090     
Exercisable at end of year . . . . . . . . . .        2,261,309     
Weighted average fair value of stock 

Stock Options
2008
4,932,273     
2,021,500     
(54,737)    
(473,096)    
(16,000)    
6,409,940     
4,109,839     

2007
4,500,208    $
1,685,500     
(1,030,932)    
(222,503)    
—     
4,932,273     
3,210,320    $

Weighted Average Exercise Price
2008 

2009

2007

1.99    $ 
1.00      
0.37      
2.57      
1.07      
1.02      
1.16    $ 

2.46    $
0.79     
0.92     
2.08     
1.00     
1.99     
2.07    $

1.66 
4.02 
1.76 
1.24 
— 
2.46 
1.93 

options granted during the year: . . .     $ 

0.77    $

0.63    $

3.34     

A summary of the activity for unvested employee stock options (excluding re-priced options) as of December 31, and changes 

during the year is presented below: 

2009 

Nonvested at January 1, . . . . . . . . . . . .        2,300,100     
Granted . . . . . . . . . . . . . . . . . . . . . . . . . . .        2,351,000     
Vested . . . . . . . . . . . . . . . . . . . . . . . . . . . .       
(924,392)    
Pre-vested forfeitures . . . . . . . . . . . . . .       
(713,018)    
Nonvested at December 31, . . . . . . . .        3,013,690     

Stock Options
2008
1,721,952     
2,021,500     
(970,256)    
(473,096)    
2,300,100     

F-18 

2007
1,183,214    $
1,685,500     
(924,259)    
(222,503)    
1,721,952    $

Weighted Average Grant Date Fair Value per Share
2008 

2007

2009

1.52    $ 
0.77      
2.10      
2.11      
0.70    $ 

2.92    $
0.63     
2.10     
1.74     
1.52    $

0.99 
3.34 
1.67 
1.06 
2.92 

  
  
  
 
    
    
  
 
  
  
  
  
  
  
     
      
     
 
 
  
  
  
  
     
 
 
For stock options paid in consideration of services rendered by non-employees, the Company recognizes compensation expense in 
accordance with the requirements of ASC 718, ASC 503-50 (formerly Emerging Issues Task Force Issue No. 96-18 (“EITF 96-18”), 
Accounting for Equity Instruments that are Issued to other than Employees for Acquiring, or in Conjunction with Selling Goods or 
Services and formerly EITF 00-18, Accounting Recognition for Certain Transactions involving Equity Instruments Granted to Other 
Than Employees, as amended). 

Non-employee option grants that do not vest immediately upon grant are recorded as an expense over the vesting period. At the 
end of each financial reporting period prior to performance, the value of these options, as calculated using the Black-Scholes option-
pricing model, is determined, and compensation expense recognized or recovered during the period is adjusted accordingly. Since the 
fair  market  value  of  options  granted  to  non-employees  is  subject  to  change  in  the  future,  the  amount  of  the  future  compensation 
expense is subject to adjustment until the common stock options are fully vested. 

The Company recorded approximately $0, ($0.4) million and $0.4 million of non-cash charges related to the issuance of stock 

options to certain consultants in exchange for services during 2009, 2008 and 2007, respectively. 

At  December  31,  2009,  there  remained  approximately  $0.1  million  (subject  to  change  in  the  future  based  on  vesting  date  fair 
value)  of  unrecognized  compensation  expense  related  to  unvested  non-employee  stock  options  to  be  recognized  as  expense  over  a 
weighted-average period of 2.0 years. Presented below is the Company’s non-employee stock option activity: 

Outstanding — beginning of year . . .       
Granted . . . . . . . . . . . . . . . . . . . . . . . . . . .       
Exercised . . . . . . . . . . . . . . . . . . . . . . . . .       
Forfeited . . . . . . . . . . . . . . . . . . . . . . . . . .       
Expired . . . . . . . . . . . . . . . . . . . . . . . . . . .       
Outstanding — end of year . . . . . . . . .       
Exercisable at end of year . . . . . . . . . .       
Weighted average fair value of stock 

options granted during the year: . . .     $ 

Stock Options

2009 
995,000     
—     
—     
—     
—     
995,000     
545,080     

2008
1,067,000     
350,000     
—     
(402,000)    
(20,000)    
995,000     
445,000     

2007
2,358,000    $
—     
(728,500)    
(562,500)    
—     
1,067,000     
817,000    $

0    $

0.33    $

0     

Weighted Average
Exercise Price
2008 

2009

2007

0.91    $ 
—      
—      
—      
—      
0.91      
1.00    $ 

1.44    $
0.35     
—     
1.85     
0.30     
0.91     
1.18    $

1.66 
— 
1.86 
1.85 
— 
1.44 
1.54 

The fair value of the stock options at the date of grant was estimated using the Black-Scholes option-pricing model, based on the 

following assumptions: 

Risk-free interest rate . . . . . . . . .    
Expected volatility . . . . . . . . . . . .    
Expected lives (years) . . . . . . . . .    
Expected dividend yield . . . . . . .    

2009

2008

2007 

—     
—     
—     
—     

2.68%   
123%   
10      
0%   

—  
—  
—  
—  

A  summary  of  the  activity  for  nonvested,  non-employee  stock  options  as  of  December  31,  and  changes  during  the  years  are 

presented below: 

Nonvested at January 1, . . . . . . . . . . . .       
Granted . . . . . . . . . . . . . . . . . . . . . . . . . . .       
Vested . . . . . . . . . . . . . . . . . . . . . . . . . . . .       
Pre-vested forfeitures . . . . . . . . . . . . . .       
Nonvested at December 31, . . . . . . . .       

Stock Options

2009 
550,000     
—     
(100,080)    
—     
449,920     

2008
250,000     
350,000     
(50,000)    
—     
550,000     

2007
916,663    $
—     
(104,163)    
(562,500)    
250,000    $

Weighted Average
Grant Date Fair 
Value per Share
2008 

2009

0.58    $ 
—      
0.33      
—      
1.38    $ 

1.00    $
0.33     
2.33     
—     
0.58    $

2007

1.44 
— 
1.63 
1.63 
1.00 

F-19 

 
  
  
  
  
  
   
 
  
  
   
   
   
     
   
 
      
     
 
 
  
 
   
    
  
 
  
  
  
  
   
 
  
  
   
   
   
     
   
 
 
 
 
The following table summarizes significant ranges of outstanding stock options under the three plans at December 31, 2009: 

Range of 

Exercise Prices       
$  0.30 — 1.00      
$  1.01 — 1.50      
$  2.35 — 3.33      

Number of 
Options 

Weighted Average
RemainingContractual 
Life 
(years) 

Weighted Average
Exercise Price

Number of 
Options 
Exercisable

Weighted Average
Contractual Life   

Weighted Average
Exercise Price

2,302,607      
6,176,483      
528,000      
9,007,090      

7.89    $
7.20     
4.55     
7.22    $

0.57     
1.13     
2.27     
1.05     

1,290,762      
3,723,317      
528,000      
5,542,079      

7.89    $
7.20     
4.55     
7.22    $

0.62 
1.16 
2.27 
1.16 

The aggregate intrinsic value of outstanding options as of December 31, 2009 was $1.3 million, which represents options whose 

exercise price was less than the closing fair market value of the Company’s common stock on December 31, 2009 of $1.12. 

RXi Pharmaceuticals 

RXi has its own stock option plan. RXi accounted for stock option expense in the same manner as CytRx as described above. 

As discussed in Note 2, the Company has accounted for its investment in RXi under the equity method since March 2008, and 
accordingly, the following table sets forth the total stock-based compensation expense for January and February 2008 resulting from 
RXi stock options that is included in the Company’s consolidated statements of operations: 

Research and development — 

employee . . . . . . . . . . . . . . . . . .   $

General and administrative — 

employee . . . . . . . . . . . . . . . . . .    

Total employee stock-based 

compensation . . . . . . . . . . . . . .   $

Research and development — 

non-employee . . . . . . . . . . . . . .   $

General and administrative — 

non-employee . . . . . . . . . . . . . .    

Total non-employee stock-

based compensation . . . . . . . .   $

2009

2008

2007 

—    $

28,000    $

120,000  

—     

369,000     

931,000  

—    $

397,000    $

1,051000  

—    $

121,000    $ 1,043,000  

—     

—     

—  

—    $

121,000    $ 1,043,000  

CytRx Warrants 

A summary of the Company’s warrant activity and related information for the years ended December 31 are shown below. 

2009 

Warrants

2008

2007

2009

Outstanding — beginning of year . . .        10,634,848      13,031,515      23,360,165    $
Granted . . . . . . . . . . . . . . . . . . . . . . . . . . .        6,328,330     
Exercised . . . . . . . . . . . . . . . . . . . . . . . . .       
(250,000)    
(951,665)     (10,233,650)    
Forfeited . . . . . . . . . . . . . . . . . . . . . . . . . .       
—     
—     
Expired . . . . . . . . . . . . . . . . . . . . . . . . . . .        (1,295,000)    
(95,000)    
Outstanding — end of year . . . . . . . . .        15,418,178      10,634,848      13,031,515     
Exercisable at end of year . . . . . . . . . .        15,418,178      10,634,848      13,031,515    $
Weighted average fair value of 

—     
(1,445,002)    

—     

— 

warrants granted during the year: .     $ 

1.61    $

—    $

—     

F-20 

Weighted Average
Exercise Price
2008 

2007

1.40    $ 
1.61      
1.16      
—      
1.28      
1.50      
1.50    $ 

1.87    $
—     
0.97     
—     
2.60     
1.40     
1.40    $

1.83 
— 
1.77 
— 
2.25 
1.87 
1.87 

  
    
   
  
   
 
 
 
 
  
      
 
  
  
  
  
  
 
   
   
  
   
     
     
  
 
  
  
  
  
   
 
  
  
   
   
   
     
   
 
 
      
     
 
 
 
 
The following table summarizes additional information concerning warrants outstanding and exercisable at December 31, 2009: 

Range of Exercise 
Prices 
0.26 — 1.26        
1.51 — 1.62        
1.70 — 1.84        
2.25 — 4.00        

$ 
$ 
$ 
$ 

Number of 
Shares 

3,322,767        
6,861,790        
4,735,973        
497,648        
15,418,178        

16. ALSCRT Amendment 

Weighted
Average 
Remaining 
Contractual Life 
(years)

Weighted 
Average 
Exercise Price

Warrants 
Number of 
Shares 
Exercisable 

Exercisable 
Weighted Average 
Exercise Price

2.22      $
0.07        
4.57        
0.90        
1.94      $

0.94        
1.51        
1.70        
3.07        
1.48        

3,322,767      $
6,861,790        
4,735,973        
497,648        
15,418,178      $

0.94  
1.51  
1.70  
3.07  
1.50  

Pursuant to an amendment signed between the Company and the beneficiary of the ALSCRT on August 6, 2009, the Company 
was released from all restrictions on the use of any proceeds previously paid to the Company in connection with the arrangement. As a 
result, the Company recognized $6.7 million as service revenue in the third quarter of 2009, which represented the remaining deferred 
revenue and previously un-recognized portion of the value received. 

17. Stockholder Protection Rights Plan 

Effective April 16, 1997, the Company’s board of directors declared a distribution of one right (“Rights”) for each outstanding 
share  of  the  Company’s  common  stock  to  stockholders  of  record  at  the  close  of  business  on  May  15,  1997  and  for  each  share  of 
common  stock  issued  by  the  Company  thereafter  and  prior  to  a  Flip-in  Date  (as  defined  below).  Each  Right  entitles  the  registered 
holder to purchase from the Company one-ten thousandth (1/10,000th) of a share of Series A Junior Participating Preferred Stock, at 
an exercise price of $30. The Rights are generally not exercisable until 10 business days after an announcement by the Company that a 
person or group of affiliated persons (an “Acquiring Person”) has acquired beneficial ownership of 15% or more of the Company’s 
then outstanding shares of common stock (a “Flip-in Date”). 

In the event the Rights become exercisable as a result of the acquisition of shares, each Right will enable the owner, other than the 
Acquiring  Person,  to  purchase  at  the  Right’s  then-current  exercise  price  a  number  of  shares  of  common  stock  with  a  market  value 
equal to twice the exercise price. In addition, unless the Acquiring Person owns more than 50% of the outstanding shares of common 
stock, the Board of Directors may elect to exchange all outstanding Rights (other than those owned by such Acquiring Person) at an 
exchange ratio of one share of common stock per Right. All Rights that are owned by any person on or after the date such person 
becomes an Acquiring Person will be null and void. 

The Rights have been distributed to protect the Company’s stockholders from coercive or abusive takeover tactics and to give the 
Board  of  Directors  more  negotiating  leverage  in  dealing  with  prospective  acquirors.  In  April  2007,  the  Company  extended  the 
stockholder rights plan through April 2017. 

18. Income Taxes 

At December 31, 2009, the Company had federal and state net operating loss carryforwards of $91.6 million and $81.9 million, 
respectively, available to offset against future taxable income, which expire in 2011 through 2029. As a result of a change in-control 
that  occurred  in  the  CytRx  shareholder  base  in  July  2002,  approximately  $34.7  million  in  federal  net  operating  loss  carryforwards 
became  limited  in  their  availability  to  $0.3  million  annually.  Management  currently  believes  that  the  remaining  $56.9  million  in 
federal net operating loss carryforwards, and the $57.6 million in state net operating loss carryforwards, are unrestricted. However, 
management  is  reviewing  its  recent  equity  transactions  to  determine  if  they  may  have  resulted  in  any  further  restrictions  on  the 
Company’s  net  operating  loss  carryforwards.  As  of  December  31,  2009,  CytRx  also  had  research  and  development  and  alternative 
minimum  tax  credits  for  federal  and  state  purposes  of  approximately  $8.9  million  and  $0,  respectively,  available  for  offset  against 
future income taxes, which expire in 2022 through 2029. Based on an assessment of all available evidence including, but not limited 
to, the Company’s limited operating history in its core business and lack of profitability, uncertainties of the commercial viability of 
its  technology,  the  impact  of  government  regulation  and  healthcare  reform  initiatives,  and  other  risks  normally  associated  with 
biotechnology companies, the Company has concluded that it is more likely than not that these net operating loss carryforwards and 
credits will not be realized and, as a result, a 100% deferred tax valuation allowance has been recorded against these assets.

F-21 

  
     
     
     
  
     
     
  
  
  
        
 
  
  
  
  
  
  
  
Deferred income taxes reflect the net effect of temporary differences between the financial reporting carrying amounts of assets 
and liabilities and income tax carrying amounts of assets and liabilities. The components of the Company’s deferred tax assets and 
liabilities, all of which are long-term, are as follows (in thousands): 

Net operating loss carryforwards. . . . . . . . . . . .   $
Tax credit carryforwards . . . . . . . . . . . . . . . . . . .    
Equipment, furnishings and other . . . . . . . . . . .    
Deferred revenue . . . . . . . . . . . . . . . . . . . . . . . . . .    
Total deferred tax assets . . . . . . . . . . . . . . . . . . . . . .    
Deferred tax liabilities . . . . . . . . . . . . . . . . . . . . . . .    
Net deferred tax assets . . . . . . . . . . . . . . . . . . . . . . .    
Valuation allowance . . . . . . . . . . . . . . . . . . . . . . . . .    
  $

December 31,

2009

2008 

35,285    $
8,957     
8,142     
—     
52,384     
(560)    
51,824     
(51,824)    
—    $

34,407  
6,071  
4,358  
3,744  
48,580  
(407) 
48,173  
(48,173) 
—  

For  all  years  presented,  the  Company  did  not  recognize  any  deferred  tax  assets  or  liabilities.  The  net  change  in  valuation 

allowance for the years ended December 31, 2009 and 2008 was $3,651,000 and ($5,073,000), respectively. 

The  provision  for  income  taxes  differs  from  the  provision  computed  by  applying  the  Federal  statutory  rate  to  net  loss  before 

income taxes as follows (in thousands): 

Federal benefit at statutory rate   $
State income taxes, net of 

Federal taxes . . . . . . . . . . . . . . .    
Permanent differences . . . . . . . .    
Provision related to change in 

valuation allowance. . . . . . . . .    

Net change in research and 

development tax credits . . . . .    
Other, net . . . . . . . . . . . . . . . . . . . .    
  $

Years ended December 31,

2009

2008

2007 

(1,809)   $

(8,899)   $

(7,781) 

(310)    
(136)    

(1,525)    
16,272     

(908) 
65  

3,651     

(5,073)    

9,416  

(2,826)    
911     
(519)   $

(2,207)    
(2,304)    
872    $

(1,125) 
373  
40  

As of January 1, 2007, the Company had no unrecognized tax benefits and there was no effect on its financial condition or results 
of  operations  as  a  result  of  implementing  ASC  740.  There  have  been  no  changes  to  the  Company’s  liability  for  unrecognized  tax 
benefits during the year ended December 31, 2009. 

The Company and its Subsidiaries file income tax returns in the U.S. Federal jurisdiction and various state jurisdictions. As of the 
date  of  adoption  of  ASC  740  and  the  year  ended  December  31,  2009,  the  tax  returns  for  2006  through  2008  remain  open  to 
examination by the Internal Revenue Service and various state tax authorities. 

The Company’s policy is to recognize any interest and penalties related to unrecognized tax benefits as a component of income 
tax expense. As of the date of adoption of ASC 740 and the years ended December 31, 2009 and 2008, the Company had accrued no 
interest or penalties related to uncertain tax positions. 

F-22 

 
  
 
  
  
 
   
  
 
  
  
  
 
  
  
 
   
   
  
 
  
  
 
 
19. Quarterly Financial Data (unaudited) 

Summarized quarterly financial data for 2009 and 2008 is as follows (in thousands, except per share data): 

Quarters Ended 

  March 31

June 30

      September 30     December 31  

(In thousands, except per share data)

2009 
Total revenues . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   $
Net income (loss) . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Net income (loss) applicable to common stockholders . . . . . . . . . . . . . .   $
Basic and diluted loss per share applicable to common stock . . . . . .   $

1,483    $
(3,973)    
(3,973)   $
(0.04)   $

1,000    $ 
(2,226)     
(2,226)   $ 
(0.02)   $ 

6,954    $
3,863     
3,863    $
0.04    $

2008 
Total revenues . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   $
Net loss . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Deemed dividend for anti-dilution adjustments made to outstanding 

common stock warrants . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .    
Net loss applicable to common stockholders . . . . . . . . . . . . . . . . . . . . . . .   $

Basic and diluted income (loss) per share applicable to common 

stock . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . .   $

2,181    $
(5,374)    

1,740    $ 
(5,826)     

917    $
(12,316)    

(757)    
(6,131)   $

—      
(5,826)   $ 

—     
(12,316)   $

(0.07)   $

(0.06)   $ 

(0.14)   $

(0.03)

100 
(2,464)
(2,464)
(0.03)

1,428 
(3,530)

— 
(3,530)

Quarterly and year-to-date loss per share amounts are computed independently of each other. Therefore, the sum of the per share 

amounts for the quarters may not agree to the per share amounts for the year. 

In connection with the Company’s adjustment to the exercise terms of certain outstanding warrants to purchase common stock on 
March 11, 2008, the Company recorded a deemed dividend of $757,000. That deemed dividend is reflected as an adjustment to net 
loss for the first quarter of 2008 to arrive at net loss applicable to common stockholders on the consolidated statements of operations 
and for purposes of calculating basic and diluted earnings per shares. 

20. Acquisition of Innovive Pharmaceuticals 

On September  19,  2008,  the Company  completed  the  merger of Innovive  with  CytRx Merger  Subsidiary,  Inc.,  the Company’s 
wholly  owned  subsidiary,  with  Innovive  continuing  as  the  surviving  corporation.  As  a  result,  Innovive  became  a  wholly  owned 
subsidiary  of  CytRx  and  changed  its  name  to  CytRx  Oncology  Corporation.  Because  Innovive  was  a  development  stage  company, 
under  accounting  principles  generally  accepted  in  the  United  States  and  the  SEC  regulations,  it  was  not  considered  a  business. 
Accordingly, CytRx accounted for the merger in accordance with ASC 350 (previously Statement of Financial Accounting Standards 
No. 142, Goodwill and Other Intangible Assets), for transactions other than a business combination. The initial merger consideration, 
together  with  direct  costs  incurred  to  effect  the  merger,  were  allocated  to  the  individual  assets  acquired,  including  identifiable 
intangible  assets  and  liabilities  assumed  based  on  the  relative  fair  value.  No  goodwill  was  recorded.  The  Company’s  consolidated 
financial statements reflect these fair values and were not restated retroactively to reflect the historical financial position or results of 
operations of Innovive. In connection with the merger, the Company recorded a one-time expense for acquired in-process research and 
development.  Under  the  merger  agreement  by  which  the  Company  acquired  Innovive,  it  agreed  to  pay  the  former  Innovive 
stockholders  a  total  of  up  to  approximately  $18.3  million  of  future  earnout  merger  consideration,  subject  to  the  Company’s 
achievement of specified net sales under the Innovive license agreements. The earnout merger consideration, if any, will be payable in 
shares of CytRx common stock, subject to specified conditions, or, at the Company’s election, in cash or by a combination of shares of 
CytRx common stock and cash. The Company’s common stock will be valued for purposes of any future earnout merger consideration 
based upon the trading price of its common stock at the time the earnout merger consideration is paid. 

F-23 

  
  
  
 
 
  
   
 
 
    
      
        
      
 
   
     
      
     
 
   
     
      
     
 
 
  
  
  
 
 
REPORT OF INDEPENDENT REGISTERED PUBLIC ACCOUNTING FIRM 

Board of Directors and Stockholders 
CytRx Corporation 
Los Angeles, California 

We have audited the accompanying consolidated balance sheets of CytRx Corporation (“the Company”) as of December 31, 2009 
and 2008 and the related consolidated statements of operations, stockholders’ equity, and cash flows for each of the three years in the 
period  ended  December  31,  2009.  We  have  also  audited  the  schedule  listed  in  the  accompanying  index  under  Item  15a  (2).  These 
financial statements and schedule are the responsibility of the Company’s management. Our responsibility is to express an opinion on 
these financial statements and schedule based on our audits. 

We conducted our audits in accordance with the standards of the Public Company Accounting Oversight Board (United States). 
Those standards require that we plan and perform the audit to obtain reasonable assurance about whether the financial statements are 
free of material misstatement. An audit also includes examining, on a test basis, evidence supporting the amounts and disclosures in 
the  financial  statements,  assessing  the  accounting  principles  used  and  significant  estimates  made  by  management,  as  well  as 
evaluating the overall financial statement presentation. We believe that our audits provide a reasonable basis for our opinion. 

In our opinion, the consolidated financial statements referred to above present fairly, in all material respects, the financial position 
of CytRx Corporation at December 31, 2009 and 2008, and the results of its operations and its cash flows for each of the three years in 
the period ended December 31, 2009, in conformity with accounting principles generally accepted in the United States of America. 

As more fully described in Note 3 to the consolidated financial statements, effective January 1, 2009, the Company adopted the 
Amendments to the provisions of Accounting Standards Codification 810-10, Consolidation. 

Also, in our opinion, the financial statement schedule, when considered in relation to the basic consolidated financial statements 

taken as a whole, present fairly, in all material respects, the information set forth therein. 

We  also  have  audited,  in  accordance  with  the  standards  of  the  Public  Company  Accounting  Oversight  Board  (United  States), 
CytRx  Corporation's  internal  control  over  financial  reporting  as  of  December  31,  2009,  based  on  criteria  established  in  Internal 
Control – Integrated Framework issued by the Committee of Sponsoring Organizations of the Treadway Commission (COSO) and 
our report dated March 12, 2010 expressed an unqualified opinion thereon. 

/s/ BDO SEIDMAN, LLP 

Los Angeles, California 
March 12, 2010 

F-24 

 
  
  
  
  
 
  
  
  
 
 
 
 
REPORT OF INDEPENDENT REGISTERED PUBLIC ACCOUNTING FIRM 

Board of Directors and Shareholders 
CytRx Corporation 
Los Angeles, California 

We have audited CytRx Corporation’s (“the Company”) internal control over financial reporting as of December 31, 2009, based 
on  criteria  established  in  Internal  Control  –  Integrated  Framework  issued  by  the  Committee  of  Sponsoring  Organizations  of  the 
Treadway  Commission  (the  COSO  criteria).  CytRx  Corporation’s  management  is  responsible  for  maintaining  effective  internal 
control over financial reporting and for its assessment of the effectiveness of internal control over financial reporting, included in the 
accompanying  “Item  9A,  Controls  and  Procedures.”  Our  responsibility  is  to  express  an  opinion  on  the  Company’s  internal  control 
over financial reporting based on our audit. 

We conducted our audit in accordance with the standards of the Public Company Accounting Oversight Board (United States). 
Those  standards  require  that  we  plan  and perform  the  audit  to  obtain  reasonable  assurance  about  whether  effective  internal  control 
over financial reporting was maintained in all material respects. Our audit included obtaining an understanding of internal control over 
financial reporting, assessing the risk that a material weakness exists, and testing and evaluating the design and operating effectiveness 
of internal control based on the assessed risk. Our audit also included performing such other procedures as we considered necessary in 
the circumstances. We believe that our audit provides a reasonable basis for our opinion. 

A  company’s  internal  control  over  financial  reporting  is  a  process  designed  to  provide  reasonable  assurance  regarding  the 
reliability  of  financial  reporting  and  the  preparation  of  financial  statements  for  external  purposes  in  accordance  with  generally 
accepted accounting principles. A company’s internal control over financial reporting includes those policies and procedures that (1) 
pertain to the maintenance of records that, in reasonable detail, accurately and fairly reflect the transactions and dispositions of the 
assets of the company; (2) provide reasonable assurance that transactions are recorded as necessary to permit preparation of financial 
statements in accordance with generally accepted accounting principles, and that receipts and expenditures of the company are being 
made  only  in  accordance  with  authorizations  of  management  and  directors  of  the  company;  and  (3)  provide  reasonable  assurance 
regarding  prevention  or  timely  detection  of  unauthorized  acquisition,  use,  or  disposition  of  the  company’s  assets  that  could  have  a 
material effect on the financial statements. 

Because  of  its  inherent  limitations,  internal  control  over  financial  reporting  may  not  prevent  or  detect  misstatements.  Also, 
projections of any evaluation of effectiveness to future periods are subject to the risk that controls may become inadequate because of 
changes in conditions, or that the degree of compliance with the policies or procedures may deteriorate. 

In  our  opinion,  CytRx  Corporation  maintained,  in  all  material  respects,  effective  internal  control  over  financial  reporting  as  of 

December 31, 2009, based on the COSO criteria. 

We also have audited, in accordance with the standards of the Public Company Accounting Oversight Board (United States), the 
balance sheets of the Company as of December 31, 2009 and 2008, and the related statements of operations, stockholders’ equity, and 
cash  flows  for  each  of  the  three  years  in  the  period  ended  December  31,  2009  and  our  report  dated  March  12,  2010  expressed  an 
unqualified opinion thereon. 

/s/ BDO SEIDMAN, LLP 

Los Angeles, California 
March 12, 2010 

F-25 

  
  
  
  
  
  
  
 
  
 
 
CYTRX CORPORATION 
SCHEDULE II — VALUATION AND QUALIFYING ACCOUNTS 
For the Years Ended December 31, 2009, 2008 and 2007 

Description 
Reserve Deducted in the Balance Sheet from the 

Additions

Balance at
Beginning of 
Year

Charged to 
Costs  
and Expenses    

Charged to  
Other Accounts     

Deductions

Balance at 
End of Year  

Asset to Which it Applies: 
Allowance for Deferred Tax Assets 
Year ended December 31, 2009 . . . . . . . . . . . . . . . . . .   $ 48,998,000    $
Year ended December 31, 2008 . . . . . . . . . . . . . . . . . .   $ 53,246,000    $
Year ended December 31, 2007 . . . . . . . . . . . . . . . . . .   $ 43,830,000    $

—    $ 2,826,000    $ 
—    $
—    $ 9,416,000    $ 

—    $ 51,824,000 
—    $  4,248,000    $ 48,998,000 
—    $ 53,246,000 

F-26