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Monopar Therapeutics Inc.

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FY2017 Annual Report · Monopar Therapeutics Inc.
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UNITED STATES
SECURITIES AND EXCHANGE COMMISSION
Washington, D.C. 20549

FORM 10-K

(Mark One) 
☒ 

Annual Report Pursuant to Section 13 or 15(d) of the Securities Exchange Act of 1934

For the Fiscal Year Ended December 31, 2017

☐ 

Transition Report Pursuant to Section 13 or 15(d) of the Securities Exchange Act of 1934

For the transition period from                      to                      

Commission File Number:  000-55866

MONOPAR THERAPEUTICS INC.
(Exact name of registrant as specified in its charter)

DELAWARE
(State or other jurisdiction of incorporation or organization)

32-0463781
(I.R.S. employer  identification number)

1000 Skokie Blvd., Suite 350, Wilmette, IL
(Address of principal executive offices)

60091
(zip code)

(847) 388-0349
(Registrant’s telephone number, including area code)

Securities registered pursuant to Section 12(b) of the Act:

Title of each class
N/A

Name of each exchange on which registered
N/A

Securities registered pursuant to section 12(g) of the Act:
Common Stock, $0.001 par value

Indicate by check mark if the registrant is a well-known seasoned issuer, as defined in Rule 405 of the Securities Act. Yes  ☐    No  ☒

Indicate by check mark if the registrant is not required to file reports pursuant to Section 13 or Section 15(d) of the Act. Yes  ☐    No  ☒

Indicate by check mark whether the registrant (1) has filed all reports required to be filed by Section 13 or 15(d) of the Securities Exchange
Act of 1934 during the preceding 12 months (or for such shorter period that the registrant was required to file such reports), and (2) has
been subject to such filing requirements for the past 90 days. Yes  ☐    No  ☒

Indicate by check mark whether the registrant has submitted electronically and posted on its corporate Web site, if any, every Interactive
Data File required to be submitted and posted pursuant to Rule 405 of Regulation S-T (§ 232.405 of this chapter) during the preceding 12
months (or for such shorter period that the registrant was required to submit and post such files). Yes  ☒    No  ☐

Indicate  by  check  mark  if  disclosure  of  delinquent  filers  pursuant  to  Item  405  of  Regulation  S-K  (§  229.405  of  this  chapter)  is  not
contained  herein,  and  will  not  be  contained,  to  the  best  of  registrant’s  knowledge,  in  definitive  proxy  or  information  statements
incorporated by reference in Part III of this Form 10-K or any amendment to this Form 10-K. Yes  ☒    No  ☐

Indicate by check mark whether the registrant is a large accelerated filer, an accelerated filer, a non-accelerated filer, or a smaller reporting
company.  See  the  definitions  of  “large  accelerated  filer,”  “accelerated  filer”  and  “smaller  reporting  company”  in  Rule  12b-2  of  the
Exchange Act.
Large accelerated filer
Non-accelerated filer

☐  
☐    (Do not check if a smaller reporting company) Smaller reporting company
Emerging growth company

Accelerated filer

  ☐
☒
☒

If an emerging growth company, indicate by check mark if the registrant has elected not to use the extended transition period for complying
with any new or revised financial accounting standards provided pursuant to Section 13(a) of the Exchange Act. ☐

Indicate by check mark whether the registrant is a shell company (as defined in Rule 12b-2 of the Act).  Yes  ☐    No  ☒

Indicate by check mark whether the registrant has filed all documents and reports required to be filed by Section 12, 13 or 15(d) of the
Securities  Exchange Act  of  1934  (the  “Exchange Act”)  subsequent  to  the  distribution  of  securities  under  a  plan  confirmed  by  a  court.
Yes  ☐    No  ☐

The number of shares outstanding with respect to each of the classes of our common stock, as of March 26, 2018, is set forth below:
Class

Number of shares outstanding

Not Applicable.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Class A common stock, par value $0.001 per share
Documents incorporated by reference:

9,291,420.614

   
 
 
Part I

Part II

Part III

Part IV

MONOPAR THERAPEUTICS INC.
TABLE OF CONTENTS

  Item 1.
  Item 1A.
  Item 2.
  Item 3.

  Business
  Risk Factors
  Properties
  Legal Proceedings

  Item 5.

  Market for Registrant’s Common Equity, Related Stockholder Matters and Issuer Purchases of

Equity Securities

  Item 7.
  Item 8.
  Item 9.
  Item 9A.

  Management’s Discussion and Analysis of Financial Condition and Results of Operations
  Financial Statements and Supplementary Data
  Changes in and Disagreements with Accountants on Accounting and Financial Disclosures
  Controls and Procedures

  Item 10.
  Item 11.
  Item 12.

  Directors, Executive Officers and Corporate Governance
  Executive Compensation
  Security Ownership of Certain Beneficial Owners and Management and Related Stockholder

Matters

  Item 13.
  Item 14.

  Certain Relationships and Related Transactions and Director Independence
  Principal Accountant Fees and Services

  Item 15.

  Exhibits and Financial Statement Schedules
  Signatures

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Forward-Looking Statements

This Annual Report on Form 10-K contains “forward-looking statements” within the meaning of Section 27A of the Securities Act of 1933,
as  amended  (the  “Act”)  and  Section  21E  of  the  34 Act. All  statements  other  than  statements  of  historical  facts  included  in  this Annual
Report  on  Form  10-K  are  forward-looking  statements.  The  words  “hopes,”  “believes,”  “anticipates,”  “plans,”  “seeks,”  “estimates,”
“projects,”  “expects,”  “intends,”  “may,”  “could,”  “should,”  “would,”  “will,”  “continue,”  and  similar  expressions  are  intended  to  identify
forward-looking  statements.  Forward-looking  statements  contained  in  this  Annual  Report  on  Form  10-K  include  without  limitation
statements about the market for cancer products in general and statements about our:

●            projections and related assumptions;

●            business and corporate strategy;

●            plans, objectives, expectations, and intentions;

●            clinical and preclinical pipeline and the anticipated development of our technologies, products, and operations;

●            anticipated revenue and growth in revenue from various product offerings;

●            future operating results;

●            intellectual property portfolio;

●            projected liquidity and capital expenditures;

●            development and expansion of strategic relationships, collaborations, and alliances; and

●            market opportunity, including without limitation the potential market acceptance of our technologies and products and the size of

the market for cancer products.

Although we believe that the expectations reflected in such forward-looking statements are appropriate, we can give no assurance that such
expectations  will  be  realized.  Cautionary  statements  are  disclosed  in  this  Annual  Report  on  Form  10-K,  including  without  limitation
statements  in  the  section  entitled  “RISK  FACTORS,”  addressing  forward-looking  statements. All  subsequent  written  and  oral  forward-
looking statements attributable to us or persons acting on our behalf are expressly qualified in their entirety by the cautionary statements.
We undertake no obligation to update any statements made in this Annual Report on Form 10-K or elsewhere, including without limitation
any forward-looking statements, except as required by law.

2

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Item 1. Business

PART I

You  should  read  the  following  discussion  in  conjunction  with  our  financial  statements  as  of  December  31,  2017  and  the  notes  to

such financial statements included elsewhere in this Annual Report on Form 10-K.

Overview

We are a clinical-stage biotechnology company focused on developing innovative drugs and drug combinations to improve clinical
outcomes for cancer patients. We are building a drug development pipeline through the licensing or acquisition of oncology therapeutics at
the late preclinical through advanced clinical development stage, leveraging already existing scientific and clinical data as much as possible
to de-risk clinical development.

Our  lead  drug  product  candidate  is  Validive®  (clonidine  mucobuccal  tablet;  clonidine  MBT),  a  Phase  3-ready  molecule  for  the
prevention  and  treatment  of  severe  oral  mucositis  (“SOM”)  in  patients  undergoing  radiotherapy  for  oropharyngeal  cancer  (“OPC”).  In
September 2017, we exercised our exclusive option with Onxeo S.A. to license worldwide rights to Validive.

Increased  expression  of  pro-inflammatory  cytokines  by  macrophages  is  believed  to  be  the  mechanism  of  radiotherapy-induced
severe  oral  mucositis.  Oropharyngeal  cancer  arises  in  the  immune  tissue  at  the  back  of  the  throat,  which  is  characterized  by  a  high
localization  of  macrophages. As  a  mucoadhesive  tablet  that  works  locally  through  agonizing  a  receptor  on  macrophages  that  suppresses
cytokine  expression  at  the  sites  of  radiation,  we  believe  Validive ® has  significant  promise  in  addressing  this  large  unmet  medical  need.
Currently, there are no U.S. Food and Drug Administration (“FDA”)-approved preventive or therapeutic options for patients that develop
radiation-induced SOM.

A Phase 1 and Phase 2 trial with Validive have been completed, with encouraging results. We anticipate a pre-Phase 3 meeting with
the FDA in the second quarter of 2018, and are aiming to initiate our Phase 3 development program in the second half of 2018. Assuming
the FDA concurs with our clinical plan, an interim analysis of the Phase 3 clinical data is currently planned for the fourth quarter of 2019,
with  final  data  anticipated  to  be  released  in  the  first  half  of  2021.  In  anticipation  of  initiating  the  international  Phase  3  development
program for Validive, we created a wholly-owned French subsidiary, Monopar Therapeutics, SARL in January 2018, and a wholly-owned
Australian subsidiary, Monopar Therapeutics Australia Pty Ltd. in March 2018.

In August 2017, we acquired the clinical stage drug product candidate MNPR-201 (GPX-150) from TacticGem, LLC. MNPR-201 is
a  novel  doxorubicin  analog  engineered  to  eliminate  the  cardiotoxic  side  effects  typically  generated  by  anthracycline-based  cancer  drugs.
MNPR-201 has completed a small Phase 2 clinical trial in soft tissue sarcoma patients. We are aiming to initiate one or more Phase 2 trials
for MNPR-201 in the first half of 2019.

As part of the transaction to acquire MNPR-201, TacticGem, LLC became our majority shareholder. Surrounding this transaction,
we raised approximately $9.5 million (net of transaction costs) and filed a Form 10 with the SEC which became effective on January 8,
2018.

We  also  own  several  discovery  and  preclinical  stage  drug  product  candidates,  the  furthest  along  being  MNPR-101  (huATN-658).
MNPR-101  is  a  novel  first-in-class  humanized  monoclonal  antibody  to  the  urokinase  plasminogen  activator  receptor  (“uPAR”)  for  the
treatment of advanced cancers. It has nearly completed IND-enabling work and we anticipate a pre-IND meeting with the FDA in the third
quarter of 2018.

In  order  to  fund  our  planned  operations,  including  executing  our  clinical  development  plans  and  advancing  our  drug  product
candidates,  we  will  need  to  obtain  additional  significant  capital  through  the  sale  of  equity  securities  or  other  financial  arrangements;
however,  there  can  be  no  assurance  that  we  will  be  able  to  raise  needed  capital  under  acceptable  terms,  if  at  all.  The  sale  of  additional
equity will dilute our existing stockholders.

Corporate Information

We  were  formed  as  a  Delaware  limited  liability  company  in  December  2014,  with  the  name  Monopar  Therapeutics,  LLC.  In
December 2015, we converted into a Delaware C corporation. Our principal executive offices are located at 1000 Skokie Blvd, Suite 350,
Wilmette, IL 60091. Our telephone number is (847) 388-0349, and our email address is info@monopartx.com.

3

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Our corporate website is located at www.monopartx.com. Any information contained in, or that can be accessed through our website

is not incorporated by reference in this Annual Report on Form 10-K.

Our Strategy

Our goal is to leverage the experience and competencies of our management team to acquire, in-license and develop promising drug
product candidates and to commercialize cancer therapeutics that address unmet medical needs in the oncology market. The key elements
of our strategy include:

● Initiate our Phase 3 development program for Validive;

● Obtain FDA approval of Validive for reducing the risk of onset of SOM in patients undergoing radiotherapy for oropharyngeal

cancer;

● Commercialize Validive in the U.S. and EU;

● Maintain, expand and protect our intellectual property portfolio around Validive;

● Initiate clinical trial(s) for MNPR-201 in indications where we can leverage existing data of doxorubicin’s efficacy (breast cancer,

sarcoma, rare pediatric cancers);

● Request pre-IND meeting for MNPR-101; and

● Expand  our  product  portfolio  through  acquiring  or  in-licensing  additional  product  candidates,  especially  ones  where  we  can

leverage already existing scientific and clinical data to help de-risk further clinical development.

The Oncology Therapeutics Market

Cancer is a collection of diseases characterized by uncontrolled growth and spread of abnormal cells. In January 2018, the American
Cancer Society projected that there will be an estimated 1.7 million new cancer cases diagnosed and 609,640 cancer deaths in the U.S. in
2018.  Current  treatments  for  cancer  include  surgery,  radiation  therapy,  chemotherapy,  hormone  therapy,  targeted  therapy  and
immunotherapy.  The  IQVIA  Institute  for  Human  Data  Science  reported  in  2017  that  total  global  spending  on  oncology  medicines,
including therapeutic treatments and supportive care, reached $113 billion in 2016.

Many  currently  marketed  cancer  drugs  do  not  distinguish  between  rapidly  growing  healthy  cells  and  cancer  cells.  This  leads  to
serious  side  effects  and  a  very  narrow  therapeutic  index.  Often,  treatment  is  discontinued  because  of  adverse  effects  or  cumulative
toxicities,  rendering  chronic  treatment  impossible.  Since  tumors  are  generally  not  completely  eradicated  by  chemotherapy,  cessation  of
treatment often leads to a regrowth of the malignancy. Furthermore, many tumors mutate rapidly and develop resistance, thereby further
rendering  existing  treatments  ineffective.  While  newer  immunotherapies  have  shown  promising  results,  only  a  portion  of  patients  will
respond to such treatments. There is an urgent need for additional drugs to improve cancer treatment.

Advances in the understanding of how tumor cells differ from normal tissue have made possible the development of a new class of
targeted cancer therapies that interrupt processes important to tumor survival and progression. These include anti-angiogenic drugs, anti-
metastatic drugs, and cell-signaling inhibitors.

All of these approaches may be associated with various side effects experienced by cancer patients that result from the treatments
having  an  adverse  impact  on  normal  functioning  cells  and  organ  systems.  Supportive  care  products  are  frequently  prescribed  or
administered  to  cancer  patients  to  prevent  or  treat  these  side  effects  thereby  allowing  the  patients  to  continue  to  receive  potentially  life
prolonging cancer therapies and to minimize long term consequences from these treatments.

Our pipeline and strategy are aligned with the trends in cancer care. Validive is intended to reduce the incidence of SOM and keep
OPC patients on treatment longer. MNPR-201 is a novel analog of doxorubicin designed to eliminate formation of dose limiting cardiotoxic
metabolites  generated  by  doxorubicin  while  retaining  the  anti-cancer  activity.  MNPR-101  is  designed  to  bind  a  specific  cell  surface
receptor found cancer cells (uPAR), to thereby interrupt several pathways required for tumor growth and progression.

4

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Our Drug Product Candidates

MONOPAR PRODUCT PIPELINE

Validive® (clonidine mucobuccal tablet; clonidine MBT)

Validive  (clonidine  MBT)  is  a  mucobuccal  tablet  (“MBT”)  of  clonidine  based  on  the  Lauriad ®  mucoadhesive  technology.  The
Lauriad technology was developed for oral transmucosal drug delivery and significantly increases the mucous and salivary concentrations
of the active ingredient it contains, with decreased systemic absorption. The tablet is placed under the patient’s upper lip and remains there
for several hours a day, releasing the active ingredient into the saliva.

Mechanism of Action

Validive  is  designed  to  deliver  high  local  concentrations  of  the  active  pharmaceutical  ingredient  clonidine,  an  agonist  of  alpha-2
adrenergic receptors (“alpha-2AR”), to the oropharynx, the site of irradiation in the treatment of OPC. In the oropharynx, alpha-2AR are
expressed on macrophages, immune cells that produce cytokines, the molecules that are responsible for the development of SOM (Maria et
al., 2017). A recent clinical study demonstrated that radiation treatment substantially increased salivary cytokine levels and that these were
positively  associated  with  the  formation  of  SOM  in  patients  with  head  and  neck  cancer  (Bossi  et  al.,  2016).  OPC  patients  with  human
papilloma virus positive (“HPV+”) OPC demonstrate an increased accumulation of macrophages in the tumor microenvironment compared
to  patients  with  OPC  without  human  papilloma  virus  (“HPV–”),  thus  further  priming  HPV+  OPC  patients  for  the  development  of  SOM
(Oguejiofor  et  al.,  2017).  The  alpha-2AR  regulates  the  expression  of  cytokines  by  macrophages,  and  clonidine  reduces  this  cytokine
production  (Romero-Sandoval  et  al.,  2005;  Spengler  et  al.,  1990).  Macrophages  are  the  primary  immune  cells  that  express  alpha-2AR,
making clonidine’s mechanism of cytokine suppression macrophage selective and distinct from the mechanism of other anti-inflammatory
drugs  (Handy  et  al.,  1998;  Perälä  et  al.,  1992;  Laukova  et  al.,  2010).  Further,  Validive  delivers  clonidine  transmucosally,  to  the  sites  of
radiation  treatment  in  OPC.  This  results  in  high  salivary  concentrations  of  clonidine  and  minimizes  systemic  absorption,  allowing  for
maximal dosing of drug to the at-risk oral mucosa and the OPC microenvironment (Vasseur et al., 2017). Onxeo’s preclinical studies and
Phase  2  clinical  trial  have  provided  data  that  support  Validive’s  mechanism  of  action  and  therapeutic  potential  for  reducing  the
development  of  SOM  in  patients  with  OPC,  improving  oral  mucositis-related  symptoms,  and  decreasing  radiotherapy-related  adverse
events, while exhibiting a favorable safety profile and high compliance rate with patients.

5

 
 
 
 
 
 
 
 
 
 
 
Severe Oral Mucositis (“SOM”)

SOM is induced by radiation treatment and is the most frequent major radiation-induced side effect observed in patients with head
and neck cancer (“HNC”). SOM induces intense oral pain and dysphagia and limits a patient’s ability to eat and drink, which can lead to
severe weight loss and a requirement for enteral or parenteral nutritional support. Patients that develop SOM are often hospitalized, and
symptoms can force patients to stop cancer treatment for an undefined period of time or terminate early, thus reducing cancer treatment
efficacy  (Elting  et  al.,  2008;  Vera-Llonch  et  al.,  2006).  Thus,  SOM  impacts  both  quality  of  life  and  clinical  outcomes  in  HNC  patients.
Currently,  there  are  no  FDA-approved  preventive  or  therapeutic  options  for  patients  that  develop  radiation-induced  SOM.  Only
symptomatic treatments such as opioids and mouthwashes are currently considered as part of the standard of care for this indication.

The global incidence of HNC was approximately 690,000 cases in 2012 (Globocan 2012; Gupta, 2016). The incidence of HNC in the
U.S. was approximately 63,000 cases in 2017 (cancer.net) and is projected to increase to more than 93,000 new cases by 2030 (Gupta et al.,
2016). A similar increase is also predicted in the European Union (“EU”) Five (France, Germany, Italy, Spain and the United Kingdom).

These projections include all HNC patients, regardless of the anatomic location of their disease. However, the most rapidly growing
sub-population  of  HNC  are  patients  with  OPC  (Chaturvedi  et  al.,  2011;  Ramqvist  et  al.,  2010).  The  oropharynx  is  comprised  largely  of
immune tissue and includes the soft palate, the base (rear one third) of the tongue, and the tonsils. In the U.S., the incidence of OPC is
approaching 70% of all HNC, the majority of which (approximately 70%) is HPV+ (Chaturvedi et al., 2011; Jordan et al., 2012; Gooi et al.,
2016). The incidence of OPC is also increasing in the rest of the world (>30% of HNC) (Taberna et al., 2017), with >50% of all OPC being
HPV+ (Gupta et al., 2016; Fakhry et al., 2015).

Recent  data  (Vatca  et  al.,  2014)  have  demonstrated  that  HPV+  OPC  patients  have  a  6.9-fold  increased  risk  of  developing  SOM
during radiation treatment, and that onset of SOM occurs sooner than in HPV– OPC patients. These observations suggest that HPV+ OPC
patients may be more likely to benefit from Validive (clonidine MBT) treatment than other HNC patients. The incidence of HPV+ OPC has
outpaced the incidence of HPV– HNC by 4-5-fold over the past decade (Chaturvedi et al., 2011; Castellsagué et al., 2017). We project that
this trend will continue for at least the next 20-25 years (another generation) in the U.S. based on the predicted increase in high-risk oral
HPV  infections  due  to  the  lack  of  adequate  use  of  HPV  vaccinations  in  children  (Castellsagué  et  al.,  2017).  Thus,  the  HPV+  OPC
population  could  be  a  driver  of  market  growth  for  Validive  (clonidine  MBT),  and  also  represents  a  potentially  molecularly  defined
population for the clinical development of this drug (Taberna et al., 2017; Castellsagué et al., 2017).

Clinical Data

In November 2012, Onxeo submitted an Investigational New Drug application ("IND") for Validive with the FDA for the prevention
and  treatment  of  oral  mucositis  induced  by  radiotherapy  and/or  chemotherapy  in  cancer  patients.  On  March  12,  2018,  we  received  a
notification from the FDA confirming the IND transfer from Onxeo to us. We believe that Onxeo’s Phase 2 data support the development
of Validive for SOM in OPC patients, with an enhanced response anticipated in HPV+ patients. Patients with HPV+ OPC have a 6.9-fold
higher risk of developing SOM (Vatca et al., 2014) possibly due to the increased accumulation of immune cells in the tumor due to the
presence of the HPV infection (Lyford-Pike et al., 2013; Vatca et al., 2014; Oguejiofor et al., 2017). These immune cells may release oral
mucosa damaging cytokines in response to radiation and may therefore be more responsive to Validive, which suppresses the production of
these cytokines.

In  October  2015,  the  results  from  an  international  Phase  2  clinical  trial  of  Validive  were  announced  by  Onxeo,  demonstrating
encouraging signs of clinical activity and safety compared to placebo. The trial enrolled 183 patients and was conducted in more than thirty
centers in Europe and the U.S. This global, multi-center, double-blind, randomized, placebo-controlled, three-arm study (NCT01385748)
compared the efficacy and safety of Validive (50 microgram (µg) and 100 µg) to placebo in patients with HNC receiving chemoradiation
therapy.  Validive  and  placebo  were  applied  to  the  gum  of  the  mouth  once  daily  beginning  1  to  3  days  prior  to  chemoradiotherapy  and
continuing until the end of chemoradiation treatment.

6

 
 
 
 
 
 
 
 
 
 
 
The  safety  profile  of  Validive  was  similar  to  placebo.  Patients  treated  with  Validive  experienced  less  nausea  and  dysphagia

compared to placebo.

The mean overall patient compliance was approximately 90% across all treatment groups. Overall compliance according to patient

diaries was similar in all treatment groups and consistent with the compliance according to the investigator’s evaluation.

The analysis of OPC patients in this study showed:

● The  incidence  of  severe  oral  mucositis  (primary  endpoint)  was  reduced  by  26.3%  (40%  relative  to  placebo)  in  OPC  patients
treated with Validive (100 µg) (p=0.09† which is a meaningful trend but not statistically significant). 65.2% of OPC patients on
placebo experienced severe oral mucositis compared to only 38.9% of OPC patients on Validive 100 µg.

● Validive (100 µg) reduced the risk of onset of SOM by 52% compared to placebo
● Secondary endpoints of severe drinking, eating, and speaking limitations due to mouth and throat soreness (“MTS”) score were

reduced in the Validive (100µg) treated cohort.

● Decreases  in  other  indicators  of  clinical  benefit,  including  decreased  duration  of  severe  oral  mucositis  (by  15  days  versus
placebo),  weight  loss,  decreased  opiate  use  and  increased  cumulative  dose  of  radiation  received,  strongly  favored  the  Validive
(100 µg) treated cohort.

● A dose response was observed with the Validive (100 µg) dose, demonstrating a trend toward superiority over the Validive (50

µg) dose as well as placebo.

†p-value or probability value, is a statistical measurement of the likelihood a drug does not actually work based on the clinical data
compared to a control such as a placebo (with no active pharmaceutical ingredient). In general, the FDA requires a p-value of less than 5%
or p < 0.05, which is considered statistically significant, for marketing approval. A p-value of p<0.05 for a clinical trial comparing a drug
and placebo means that there is less than a 5% chance the drug is actually inactive.

Our review of Onxeo’s Phase 2 data indicated that the effect of Validive was much greater in OPC compared to non-OPC patients.
We  believe  the  data  along  with  the  mechanism  of  action  of  Validive  provide  a  rationale  for  developing  Validive  for  the  treatment  of
radiation induced SOM in OPC patients as a first indication. The most rapidly growing sub-population of HNC in the U.S. and Europe are
patients with HPV+ disease, which are primarily HNC patients with OPC. The oropharynx is the part of the throat at the back of the mouth,
which includes the soft palate, the base (rear one third) of the tongue, and the tonsils. HPV+ OPC is a molecularly defined population of
HNC characterized by the expression of a protein biomarker, p16 INK4a, and the presence of HPV DNA in the tumor. Evaluation of HPV
status is part of the routine clinical assessment of patients with OPC prior to initiating treatment. The incidence of HPV+ OPC has outpaced
the incidence of HPV– HNC in the U.S. and Europe by 4 to 5-fold over the past decade (Chaturvedi et al., 2011; Castellsagué et al., 2017).

Validive Development Strategy

Based  on  the  existing  Phase  2  data  in  patients  with  OPC  treated  with  Validive,  we  are  planning  an  adaptive  design  Phase  3
development program that will evaluate Validive compared to placebo in OPC patients stratified for HPV status. This design will allow us
to prospectively confirm the observation made from the Phase 2 trial, that Validive will be effective in preventing radiation-induced SOM
in  patients  with  OPC.  The  Phase  3  program  will  also  evaluate  if  Validive  performs  better  in  the  HPV+  OPC  cohort.  We  are  currently
working with the U.S. and EU regulatory agencies to design a development plan to move Validive toward registration in both a time- and
cost- efficient manner. An optimal timeline of development milestones related to Validive include: FDA meeting to discuss Phase 3 in the
second  quarter  of  2018,  with  Phase  3  trial  being  initiated  in  the  third  quarter  of  2018,  first  patient  dosed  in  the  fourth  quarter  of  2018,
interim analysis of Phase 3 trial in the fourth quarter of 2019, initiate stage 2 of the Phase 3 trial in the first half of 2020, data readout for
the Phase 3 trial in the first half of 2021, and NDA submission in the second half of 2021. However, there are many risk factors which
could delay or otherwise affect Validive’s development. See Item 1A – “Risk Factors.”

7

 
 
 
 
 
 
 
 
 
 
 
MNPR-201 (GPX-150; 5-imino-13-deoxydoxorubicin)

MNPR-201  (GPX-150;  5-imino-13-deoxydoxorubicin)  is  a  proprietary  doxorubicin  analog  that  is  selective  for  topoisomerase-
II-alpha.  Doxorubicin  is  used  to  treat  adult  and  pediatric  solid  and  blood  (hematologic)  cancers  including  breast,  gastric,  ovarian  and
bladder cancer, soft tissue sarcomas, leukemias and lymphomas. A number of clinical studies have demonstrated the anti-cancer benefit of
higher  doses  of  doxorubicin  administered  for  longer  periods  of  time.  The  optimal  clinical  efficacy  of  doxorubicin,  however,  has  been
limited  historically  by  the  risk  of  patients  developing  irreversible,  potentially  life-threatening  cardiotoxicity.  MNPR-201  has  been
engineered  specifically  to  retain  the  anticancer  activity  of  doxorubicin  while  minimizing  the  toxic  effects  on  the  heart.  We  believe  the
results of these studies, along with the potential to combine a less or non-cardiotoxic analog of doxorubicin with other anticancer agents,
emphasizes that there is a large market opportunity for MNPR-201 in a broad spectrum of cancer types.

The  antitumor  effects  of  MNPR-201  are  mediated  through  the  stabilization  of  the  topoisomerase  II  complex  after  a  DNA  strand
break and DNA intercalation leading to apoptosis (cell death) through a mechanism similar to doxorubicin and other anthracycline drugs.
Inhibiting the topoisomerase II-alpha isoform is desired for the anti-cancer effect, while inhibiting the topoisomerase II-beta isoform has
been  demonstrated  to  mediate,  at  least  in  part,  the  cardiotoxicity  associated  with  all  anthracycline  drugs  currently  used  in  the  clinic.
MNPR-201  is  substantially  more  selective  than  doxorubicin  for  inhibiting  topoisomerase  II-alpha  versus  topoisomerase  II-beta.  This
selectivity may at least partly explain the minimal cardiotoxicity that MNPR-201 has demonstrated in clinical studies to date.

Clinical Data

In February 2007, Gem Pharmaceuticals, LLC (a partner of TacticGem LLC) submitted an IND for MNPR-201 (GPX-150) for the
treatment of cancer. The IND remains open and was transferred to us in February 2018. Several clinical studies of MNPR-201 (GPX-150)
have been completed. A Phase I dose escalation study conducted at the University of Iowa enrolled 24 patients at 5 different dose levels of
MNPR-201  (GPX-150)  ranging  from  14-265  mg/m2.  No  evidence  of  irreversible  cardiotoxicity  was  observed  in  any  of  these  patients,
including 4 patients that had received prior anthracycline (doxorubicin or related molecules) treatment. In the four highest dose levels (>84
mg/m2), 9/17 patients showed a stabilization of disease including 3 out of 4 patients with leiomyosarcoma, which is a type of cancer that
originates in connective tissue and smooth muscle most commonly in the uterus, stomach and small intestine.

Based on the demonstration of stable disease in patients with leiomyosarcoma in the Phase I trial, a multi-center open label single
arm  Phase  2  trial  was  run  in  doxorubicin-naïve  patients  with  non-resectable  or  metastatic  soft  tissue  sarcoma  (“STS”).  Doxorubicin  has
historically been the standard of care for the treatment of leiomyosarcoma and other STS. This Phase 2 clinical trial enrolled 22 patients and
was completed in early 2017. MNPR-201 was administered intravenously at 265 mg/m2 every 3 weeks for up to 16 doses and there was
clear indication of anticancer activity and no evidence of irreversible cardiotoxicity. One patient went on compassionate use and received
20 cycles of MNPR-201, many more than the 6 to 8 cycles patients on doxorubicin are typically limited to. The progression free survival at
6 months was 38%, versus doxorubicin’s 6-month progression free survival of 25%, 33%, and 23% in three separate studies in this patient
population (Lorigan et al., 2007; Judson et al., 2014; Chawla et al., 2015).

MNPR-201 Development Strategy

We will need to raise additional funds to support the next stage of clinical development of MNPR-201, which is planned to include
Phase  2  trials  that  will  evaluate  MNPR-201  in  cancer  indications  where  doxorubicin  has  shown  efficacy  but  its  use  is  restricted  due  to
cardiotoxicity.  The  objective  of  these  trials  would  be  to  demonstrate  signals  of  efficacy  where  MNPR-201  dosing  does  not  have  to  be
restricted due to cardiotoxicity. For example, several clinical studies completed in the 1990s demonstrated that concurrent doxorubicin (60
mg/m2, 8 cycles) and paclitaxel gave a 94% overall response rate in patients with metastatic breast cancer but led to 18% of these patients
developing  congestive  heart  failure  (Gianni  et  al.,  1995).  Reduction  of  doxorubicin  to  4-6  cycles  of  treatment  decreased  occurrence  of
congestive heart failure, but also reduced response rate to 45-55% (Sparano et al., 1999; Valero et al., 2001). A potential Phase 2 screening
trial in patients with metastatic breast cancer would evaluate concurrent MNPR-201 plus paclitaxel to see if a higher response rate than 45-
55%  could  be  observed  in  the  absence  of  irreversible  cardiotoxicity.  Concomitant  administration  of  paclitaxel  and  MNPR-201  in  the
absence of cardiotoxicity would also provide rationale for this same combination in other clinical settings. Similar studies are also under
consideration  for  the  combination  of  MNPR-201  +  trastuzumab  in  metastatic  HER2+  breast  cancer  patients.  Additional  studies  will
evaluate cross-over to MNPR-201 in patients benefiting from doxorubicin that have reached their lifetime limit of doxorubicin exposure in
STS  and  other  cancer  indications  including  several  pediatric  cancer  indications.  The  results  of  these  Phase  2  studies  would  be  used  to
inform  an  initial  registration  strategy  for  MNPR-201,  as  well  as  to  support  collaborative  clinical  development  efforts  with  cooperative
groups  and  cancer-focused  foundations.  Ideally,  we  would  like  to  initiate  the  Phase  2  clinical  trial(s)  in  the  first  half  of  2019.  However,
there are many risk factors which could delay or otherwise affect MNPR-201’s development. See Item 1A – “Risk Factors.”

8

 
 
 
 
 
 
 
 
 
 
 
MNPR-101 (formerly huATN-658)

No IND is required for MNPR-101 at this time because it is not yet in human clinical trials.

uPA/uPAR Antibodies

A significant body of in vitro and in vivo data have established the urokinase plasminogen activator ("uPA") system as being central
to  the  processes  of  angiogenesis  and  metastasis,  and  therefore  as  a  potentially  promising  target  for  cancer  drug  development.  The  uPA
system is involved in the tissue remodeling and tumor signaling that leads to the progression of cancer. Recent evidence suggests that, in
addition to uPA, its cell surface receptor, uPAR, may also be a suitable target for cancer therapeutics and diagnostics because it:

● is selectively expressed on metastatic tumor, tumor-associated immune and angiogenic endothelial cells, but not on most normal
cells (several Phase 1 imaging studies in human advanced cancer patients show that uPAR can only be detected in the tumor and
not in normal tissues);

● is central to several extracellular and intracellular oncogenic pathways required for metastasis (inhibiting the uPA system in turn

inhibits many other downstream targets that are currently being targeted by other companies);
● is expressed on immune cells that allow the tumor to evade recognition by the immune system; and
● has the potential to interfere at several different signaling pathways that converge at uPAR.

Thus, uPAR-targeted therapies may have broad-spectrum activity against many different cancer types.

We  have  developed  a  set  of  monoclonal  antibodies  that  target  uPA  and  uPAR.  Our  lead  antibody,  MNPR-101,  demonstrated
significant anti-tumor activity in numerous preclinical models of tumor growth and is being advanced for clinical evaluation. Based on the
selective expression of uPAR in tumor, MNPR-101 is expected to be well-tolerated and amenable to a variety of combination treatment
approaches.

Efficacy and Safety

MNPR-101  is  designed  to  interrupt  several  pathways  required  for  tumor  growth  and  progression.  The  compound’s  mechanism  of
action is designed to block several particular cellular activities that are only turned “on” in a tumor rather than to destroy the tumor cell
directly.  For  this  reason,  we  believe  that  MNPR-101  may  have  fewer  side  effects  than  current  cytotoxic  agents  which  kill  cells
indiscriminately. In addition, by inhibiting multiple pathways required for tumor growth and progression, we believe MNPR-101 may lead
to more effective tumor control than therapies that target only a single such pathway. We believe that most tumors, regardless of the tissue
from which they originate, rely on the pathways that we are targeting; therefore, therapies directed at such pathways have the potential to
be used against many different types of cancers.

Drug Resistance

MNPR-101  may  also  avoid  some  of  the  drug  resistance  problems  caused  by  genetic  instability  that  plague  many  conventional
chemotherapies. Cancerous cells mutate and reproduce rapidly, meaning that there is great genetic heterogeneity among cells in a tumor. A
given  chemotherapy  may  be  effective  against  the  vast  majority  of  these  cells,  but  if  even  a  small  number  have  mutations  that  confer
resistance, these cells will likely survive the treatment. The tumor will grow back composed almost entirely of these mutated cells, making
the cancer resistant to further treatments with that particular chemotherapy. By targeting multiple tumor progression pathways, using drugs
in  combination  regimens,  and  targeting  more  genetically  stable  endothelial  and  immune  cells  in  addition  to  tumor  cells,  we  believe  that
MNPR-101 has the potential to avoid these drug resistance problems.

Combination Use

Published  preclinical  data  have  shown  the  ability  of  MNPR-101  to  enhance  the  anti-tumor  activity  of  chemotherapies  such  as
paclitaxel  and  gemcitabine  (Bauer  et  al.,  2005;  Kenny  et  al.,  2011).  The  expression  and  targeting  of  uPAR  in  general  also  suggests  that
MNPR-101 may combine with other targeted agents that affect signaling leading to tumor growth including the ability of tumors to evade
immune response. In particular, uPAR is selectively expressed on cells of the myeloid lineage such as myeloid derived suppressor cells,
neutrophils and macrophages, all of which drive tumor progression and may mediate resistance to immune checkpoint inhibitors.

9

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Reports  of  successful  cancer  therapy  increasingly  involve  the  use  of  drug  combinations  that  target  multiple  metabolic  pathways
simultaneously.  To  that  end,  oncologists  are  increasingly  exploring  the  combined  use  of  approved  drugs  when  treating  their  patients.
MNPR-101  is  not  expected  to  replace  existing  therapies,  but  rather  to  complement  them.  MNPR-101  is  intended  to  be  combined  with
existing therapies used to reduce tumor mass in order to make the overall treatment more effective in the acute setting. MNPR-101 could
make  chemotherapy  more  effective  by  making  tumors  more  susceptible  to  chemotherapy  by  interrupting  the  tumors’  protective
mechanisms. MNPR-101 could also potentially be used as a standard follow-up therapy after chemotherapy to prevent tumor regrowth and
metastasis  or  in  combination  with  immunotherapy  including  immune  checkpoint  inhibitors.  Many  cancers  are  not  fatal  unless  tumors
metastasize beyond their primary site and interfere with normal function in critical organs of the body. Current thinking suggests that by
containing or preventing tumor growth, it may be possible to transform cancer into a manageable, non-fatal condition treated with chronic
drug therapy. Given these potential uses, new treatments that target multiple pathways and are designed to be used in drug combinations,
like  MNPR-101,  have  the  potential  to  significantly  improve  treatment  outcomes,  rather  than  merely  competing  with  each  other  in  the
market.

MNPR-101 Development Strategy

We currently plan to request a pre-IND meeting with the FDA to discuss MNPR-101 in the third quarter of 2018. However, there are

many risk factors which could delay or otherwise affect MNPR-101’s development. See Item 1A – “Risk Factors.”

Material Agreements

Since our inception, we have entered into three material agreements, one with Onxeo S.A., one with Cancer Research UK, and one
with  XOMA  Ltd.  None  of  the  agreements  requires  any  issuance  of  equity  or  any  annual  maintenance  fee.  See  the  summary  of  each
material agreement below.

In  June  2016,  we  executed  an  option  agreement  with  Onxeo  S.A.,  a  French  public  company,  which  gave  us  the  option  to  license
Validive (clonidine mucobuccal tablet), a mucoadhesive tablet of clonidine based on the Lauriad mucoadhesive technology to potentially
treat severe oral mucositis in patients undergoing treatment for head and neck cancers. The pre-negotiated license terms included as part of
the option agreement included clinical, regulatory, developmental and sales milestones that could reach up to $108 million if we achieve all
milestones, and escalating royalties on net sales from 5 - 10%. On September 8, 2017, pursuant to the Onxeo license option agreement, we
exercised the option to license Validive for $1 million. The exercise of the option assigns all of Onxeo’s rights to the Validive intellectual
property to us, which allows us to commence the planning of our Phase 3 clinical trial in severe oral mucositis. Under the agreement, we
are required to pay royalties to Onxeo on a product-by-product and country-by-country basis until the later of (1) the date when a given
product is no longer within the scope of a patent claim in the country of sale or manufacture, (2) the expiry of any extended exclusivity
period in the relevant country (such as orphan drug exclusivity, pediatric exclusivity, new chemical entity exclusivity, or other exclusivity
granted beyond the expiry of the relevant patent), or (3) a specific time period after the first commercial sale of the product in such country.
In most countries, including the U.S., the patent term is generally 20 years from the earliest claimed filing date of a non-provisional patent
application in the applicable country, not taking into consideration any potential patent term adjustment that may be filed in the future or
any regulatory extensions that may be obtained. The royalty termination provision pursuant to (3) described above is shorter than 20 years
and is the least likely cause of termination of royalty payments.

The  Onxeo  license  agreement  does  not  have  a  pre-determined  term,  but  expires  on  a  product-by-product  and  country-by-country
basis;  that  is,  the  agreement  expires  with  respect  to  a  given  product  in  a  given  country  whenever  our  royalty  payment  obligations  with
respect to such product have expired. The agreement may also be terminated early for cause if either we or Onxeo materially breach the
agreement,  or  if  either  we  or  Onxeo  become  insolvent.  We  may  also  choose  to  terminate  the  agreement,  either  in  its  entirety  or  as  to  a
certain product and a certain country, by providing Onxeo with advance notice.

On May 15, 2015, we entered into a Clinical Trial and Option Agreement (“CTOA”) with Cancer Research UK. Being a new entity
at the time of the agreement negotiations, one of the requirements under the CTOA, which has already been fulfilled, was for us to deposit
$800,000  into  an  escrow  to  cover  indemnities  in  the  event  of  third  party  claims  resulting  from  actions  or  inactions  of  ours,  patent
infringement claims, or potential costs on termination of the CTOA by Cancer Research UK for cause. Pursuant to this agreement Cancer
Research  UK  conducted  preclinical  work,  improved  the  manufacturing,  and  planned  to  conduct  a  Phase  1a/1b  clinical  trial  in  cancer
patients. Under this agreement, Cancer Research UK was to cover all costs through Phase 1a/1b clinical studies, including manufacturing.
As part of a portfolio reprioritization review, on March 21, 2018, Cancer Research UK notified us it was terminating the agreement and
would  work  to  transfer  to  us  the  data  generated  under  the  agreement.    We  are  currently  reviewing  potential  alternative  collaboration
opportunities for MNPR-101 and continue to maintain the program’s intellectual property portfolio.

10

 
 
 
 
 
 
 
 
 
 
 
To humanize our MNPR-101 antibody, we have taken a non-exclusive license to XOMA Ltd.’s humanization technology and know-
how. Under the terms of the license, we are to pay only upon developmental and sales milestone achievements which could reach up to
$14.925 million if we achieve all milestones. The agreement does not require the payment of sales royalties. There can be no assurance that
we will reach any milestones. The first milestone payment is payable upon first dosing of a human patient in a Phase 2 clinical trial.

Oncology Market Competition

The pharmaceutical industry in general, and the oncology therapeutics sector in particular, are characterized by intense competition.
We face competition from pharmaceutical and biotechnology companies, many of which are larger and better financed than us. We also
face competition in our efforts to develop and commercialize new oncology therapeutics from academic and government laboratories. The
therapeutics that we are developing, if successfully commercialized, will have to compete with existing therapeutics already on the market
and  novel  therapeutics  currently  in  development,  as  well  as  new  therapeutics  that  may  be  discovered  and  developed  in  the  future.  Our
product  candidates  will  also  have  to  compete  with  alternate  treatment  modalities,  such  as  radiation,  which  is  also  subject  to  continual
innovation and improvement. Additional information can be found in the section entitled “Risk Factors – Risks Related to Our Business
Operations and Industry.”

Intellectual Property Portfolio and Exclusivity

An  important  part  of  our  strategy  is  obtaining  patent  protection  to  help  preserve  the  proprietary  nature  of  our  drug  product
candidates,  and  to  prevent  others  from  developing  competitive  agents  that  are  similar.  Our  patent  portfolio  includes  issued  patents  and
pending  patent  applications  in  the  U.S.  and  in  foreign  countries.  Our  general  practice  is  to  seek  patent  protection  in  major  markets
worldwide.

We  license  all  intellectual  property  related  to  Validive  from  Onxeo  S.A.,  a  French  public  company.  See  “Material Agreements”.
Validive  is  covered  by  32  issued  patents  and  allowed  patent  applications  and  corresponding  patents  and  applications  in  32  jurisdictions,
including the U.S., EU, Japan, and other Asian countries, and has orphan drug designation in the EU as well as Fast Track designation from
the FDA. These patents are methods of use patents that cover the use of Validive to prevent and/or treat inflammation and inflammatory
pain  of  the  mucosa  including  cancer  therapy-induced  mucositis,  and  have  been  assigned  to  us  pursuant  to  our  license  agreement  with
Onxeo. These patents expire in 2029.

MNPR-201  (GPX-150)  is  covered  by  both  composition  of  matter  as  well  as  manufacturing  process  patents.  We  have  a  patent  for
chemical synthesis technology that efficiently converts cardiotoxic "13-keto" anthracyclines such as doxorubicin, daunorubicin, epirubicin,
and idarubicin into novel, patentable, and most likely less-cardiotoxic "5-imino-13-deoxy" analogs. A novel chemical composition of an
intermediate for this synthesis is also patented. In addition, we have a patent covering the combination of MNPR-201 with paclitaxel for the
treatment of cancer, plus covering the method of use of these two drugs for this purpose. Our MNPR-201 patent portfolio, which is still in
the process of completing transfer of ownership subsequent to the purchase from TacticGem LLC, contains seven issued and allowed U.S.
patents and allowed patent applications and one U.S. pending patent application. We have certain corresponding patents and applications in
twenty-nine foreign jurisdictions, including the U.S., EU, Japan, and other Asian countries. The composition of matter patents will expire
in 2018, the process patents for the synthesis of MNPR-201 intermediates will expires in 2024 and the patents covering the combination
use of MNPR-201 and its analogs with taxanes will expire in 2026. We may pursue patent term extensions where appropriate. We do not
believe  that  expiration  of  the  MNPR-201  composition  of  matter  patents  will  significantly  affect  our  ability  to  develop  or  maintain  our
proprietary  position  around  MNPR-201,  given  that  we  have  obtained  patent  protection  around  the  intermediates  and  process  used  to
manufacture MNPR-201, will have Hatch-Waxman exclusivity (applicable to new chemical entities) for 5 years that will prevent generic
competition, and have obtained U.S. orphan drug status in soft tissue sarcoma with additional orphan cancer indications to follow. We also
have  a  pending  International  Nonproprietary  Name  (“INN”)  request  with  the  World  Health  Organization  for  a  non-proprietary  (generic)
name for MNPR-201.

Our patent portfolio for our MNPR-101 antibody (huATN-658), as well as its epitope, consists of two issued U.S. composition of
matter  and  their  methods  of  use  patents,  and  allowed  patent  applications  and  corresponding  (granted  and  pending)  patents  and  patent
applications in twenty-two foreign jurisdictions, including the European Union, Japan, and other Asian countries. These patents are owned
by us. The patents covering the composition of matter of MNPR-101 will expire in 2025 and the patents covering the MNPR-101 epitope
will expire in 2027. Being a novel biologic, it is eligible for 12 years of exclusivity in the U.S. under the Biologics Price Competition and
Innovation Act (“BPCI Act”), and in numerous other countries it will benefit from varying durations of similar exclusivity, as well.

11

 
 
 
 
 
 
 
 
 
 
 
Patent life determination depends on the date of filing of the application and other factors as promulgated under the patent laws. In
most countries, including the U.S., the patent term is generally 20 years from the earliest claimed filing date (the priority date) of a non-
provisional patent application in the applicable country, not taking into consideration any potential patent term adjustment that may be filed
in the future or any regulatory extensions that may be obtained. Some of our patents are currently near expiration and we may pursue patent
term extensions for these where appropriate. See “Risk Factors – Risks Related to Our Intellectual Property.”

Manufacturing

We do not currently own or operate manufacturing facilities for the production or testing of Validive, MNPR-201, MNPR-101 or any
other  product  candidates,  nor  do  we  have  plans  to  develop  our  own  manufacturing  operations  in  the  foreseeable  future.  We  presently
depend on third party contract manufacturers for all our required raw materials, Active Pharmaceutical Ingredients (“API”), and finished
drug  products  for  our  preclinical  and  clinical  studies.  We  have  not  yet  executed  manufacturing  agreements  for  our API  and  supplies  of
Validive, MNPR-201, or MNPR-101. See “Risk Factors – Risks Related to Our Reliance on Third Parties.”

Research and Development Costs

Research and development (“R&D”) costs including in-process R&D are expensed as incurred. Major components of R&D expenses
include R&D salaries and benefits, materials and supplies and fees paid to consultants and to the entities that conduct certain development
activities on our behalf. R&D expense, including upfront fees and milestones paid to collaborators, are expensed as goods are received or
services rendered. Costs to acquire technologies, including license fees, to be used in R&D that have not reached technological feasibility
and have no alternative future use are expensed as in-process R&D as incurred, except in the case of a business combination when such
costs are capitalized as part of the purchase price allocation. During the fiscal years ended December 31, 2017 and 2016, in aggregate we
spent  approximately  $15.7  million  (which  includes  $14.5  million  of  in-process  R&D)  on  research  and  development  costs  (not  including
approximately $1.5 million spent by Gem in development of MNPR-201). See “Risk Factors – Risks Related to Clinical Development and
Regulatory Approval.”

Government Regulation and Product Approval

Government authorities in the U.S., at the federal, state and local level, and other countries extensively regulate, among other things,
the  research,  development,  testing,  manufacture,  quality  control,  approval,  labeling,  packaging,  storage,  record-keeping,  promotion,
advertising,  distribution,  post-approval  monitoring  and  reporting,  marketing  and  export  and  import  of  products  such  as  those  we  are
developing.  The  pharmaceutical  drug  product  candidates  that  we  develop  must  be  approved  by  the  FDA  before  they  may  be  legally
marketed in the U.S. See “Risk Factors – Risks Related to Clinical Development and Regulatory Approval.”

U.S. Pharmaceutical Product Development Process

In  the  U.S.,  the  FDA  regulates  pharmaceutical  products  under  the  Federal  Food,  Drug  and  Cosmetic  Act  (“FDCA”)  and
implementing regulations. Pharmaceutical products are also subject to other federal, state and local statutes and regulations. The process of
obtaining  regulatory  approvals  and  the  subsequent  compliance  with  appropriate  federal,  state,  local  and  foreign  statutes  and  regulations
require  the  expenditure  of  substantial  time  and  financial  resources.  Failure  to  comply  with  the  applicable  U.S.  requirements  at  any  time
during  the  product  development  process,  approval  process  or  after  approval,  may  subject  an  applicant  to  administrative  or  judicial
enforcement. FDA enforcement could result in refusal to approve pending applications, withdrawal of an approval, a clinical hold, warning
letters, product recalls, product seizures, total or partial suspension of production or distribution injunctions, fines, refusals of government
contracts, restitution, disgorgement or civil or criminal penalties. Any agency or judicial enforcement action could have a material adverse
effect  on  us.  The  process  required  by  the  FDA  before  a  non-biological  pharmaceutical  product  may  be  marketed  in  the  U.S.  generally
involves the following:

● Completion  of  preclinical  laboratory  tests,  animal  studies  and  formulation  studies  according  to  Good  Laboratory  Practices

(“GLP”), or other applicable regulations;

● Submission to the FDA of an Investigational New Drug application (“IND”), which must become effective before human clinical

studies may begin;

● Performance  of  adequate  and  well-controlled  human  clinical  studies  according  to  the  FDA’s  current  Good  Clinical  Practices

(“GCP”), to establish the safety and efficacy of the proposed pharmaceutical product for its intended use;

12

 
 
 
 
 
 
 
 
 
 
 
 
 
● Submission to the FDA of a New Drug Application (“NDA”), for a new pharmaceutical product;
● Satisfactory  completion  of  an  FDA  inspection  of  the  manufacturing  facility  or  facilities  where  the  pharmaceutical  product  is
produced  to  assess  compliance  with  the  FDA’s  current  Good  Manufacturing  Practice  standards  (“cGMP:”),  to  assure  that  the
facilities, methods and controls are adequate to preserve the pharmaceutical product’s identity, strength, quality and purity;

● Potential FDA audit of the preclinical and clinical study sites that generated the data in support of the NDA; and
● FDA review and approval of the NDA.

The lengthy process of seeking required approvals and the continuing need for compliance with applicable statutes and regulations

require the expenditure of substantial resources and approvals are inherently uncertain.

Before  testing  any  compounds  with  potential  therapeutic  value  in  humans,  the  pharmaceutical  product  candidate  enters  the
preclinical testing stage. Preclinical tests include laboratory evaluations of product chemistry, toxicity and formulation, as well as animal
studies to assess the potential safety and activity of the pharmaceutical product candidate. These early proof-of-principle studies are done
using  sound  scientific  procedures  and  thorough  documentation.  The  conduct  of  the  single  and  repeat  dose  toxicology  and  toxicokinetic
studies  in  animals  must  comply  with  federal  regulations  and  requirements  including  GLP.  The  sponsor  must  submit  the  results  of  the
preclinical tests, together with manufacturing information, analytical data, any available clinical data or literature and a proposed clinical
protocol, to the FDA as part of the IND. The IND automatically becomes effective 30 days after receipt by the FDA, unless the FDA has
concerns and notifies the sponsor. In such a case, the IND sponsor and the FDA must resolve any outstanding concerns before the clinical
study can begin. If resolution cannot be reached within the 30-day review period, either the FDA places the IND on clinical hold or the
sponsor withdraws the application. The FDA may also impose clinical holds on a pharmaceutical product candidate at any time before or
during clinical studies due to safety concerns or non-compliance. Accordingly, it is not certain that submission of an IND will result in the
FDA allowing clinical studies to begin, or that, once begun, issues will not arise that suspend or terminate such clinical studies.

During the development of a new drug, sponsors are given opportunities to meet with the FDA at certain points. These points may be
prior to submission of an IND, at the end of Phase 2, and before an NDA is submitted. Meetings at other times may be requested. These
meetings can provide an opportunity for the sponsor to share information about the data gathered to date, for the sponsor to ask specific
questions to the FDA, for the FDA to provide advice, and for the sponsor and FDA to reach agreement on the next phase of development.
Sponsors typically use the end of Phase 2 meeting to discuss their Phase 2 clinical results and present their plans for the pivotal Phase 3
clinical (registration) trial(s) that they believe will support approval of the new drug. A sponsor may be able to request a Special Protocol
Assessment (“SPA”), the purpose of which is to reach agreement with the FDA on the design of the Phase 3 clinical trial protocol design
and analyses that will form the primary basis of an efficacy claim.

According to FDA guidance for industry on the SPA process, a sponsor which meets the prerequisites may make a specific request
for a SPA and provide information regarding the design and size of the proposed clinical trial. The FDA’s goal is to evaluate the protocol
within 45 days of the request to assess whether the proposed trial is adequate, and that evaluation may result in discussions and a request
for additional information. A SPA request must be made before the proposed trial begins, and all open issues must be resolved before the
trial begins. If a written agreement is reached, it will be documented and made part of the IND record. The agreement will be binding on
the FDA and may not be changed by the sponsor or the FDA after the trial begins except with the written agreement of the sponsor and the
FDA or if the FDA determines that a substantial scientific issue essential to determining the safety or efficacy of the drug was identified
after the testing began.

Clinical  studies  involve  the  administration  of  the  pharmaceutical  product  candidate  to  healthy  volunteers  or  patients  under  the
supervision of qualified investigators, generally physicians not employed by or under the clinical study sponsor’s control. Clinical studies
are conducted under protocols detailing, among other things, the objectives of the clinical study, dosing procedures, subject selection and
exclusion criteria, how the results will be analyzed and presented and the parameters to be used to monitor subject safety. Each protocol
must be submitted to the FDA as part of the IND. Clinical studies must be conducted in accordance with Good Clinical Practice (“GCP”)
guidelines.  Further,  each  clinical  study  must  be  reviewed  and  approved  by  an  independent  institutional  review  board  (“IRB”),  at,  or
servicing, each institution at which the clinical study will be conducted. An IRB is charged with protecting the welfare and rights of study
participants and is tasked with considering such items as whether the risks to individuals participating in the clinical studies are minimized
and  are  reasonable  in  relation  to  anticipated  benefits.  The  IRB  also  approves  the  informed  consent  form  that  must  be  provided  to  each
clinical study subject or his or her legal representative and must monitor the clinical study until completed.

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Human clinical studies are typically conducted in three sequential phases that may overlap or be combined:

● Phase I. The pharmaceutical product is initially introduced into healthy human subjects and tested for safety, dosage tolerance,

absorption, metabolism, distribution and excretion.

● Phase 2. The pharmaceutical product is evaluated in a limited patient population to identify possible adverse effects and safety
risks, to preliminarily evaluate the efficacy of the product for specific targeted diseases, to determine dosage tolerance, optimal
dosage and dosing schedule and to identify patient populations with specific characteristics where the pharmaceutical product may
be more effective.

● Phase 3. Clinical studies are undertaken to further evaluate dosage, clinical efficacy and safety in an expanded patient population
at geographically dispersed clinical study sites. These clinical studies are intended to establish the overall risk/benefit ratio of the
product and provide an adequate basis for product labeling. The studies must be well-controlled and usually include a control arm
for comparison. One or two Phase 3 studies are required by the FDA for an NDA approval, depending on the disease severity and
other available treatment options.

● Post-approval studies, or phase IV clinical studies, may be conducted after initial marketing approval. These studies are used to

gain additional experience from the treatment of patients in the intended therapeutic indication.

● Progress reports detailing the results of the clinical studies must be submitted at least annually to the FDA and written IND safety
reports must be submitted to the FDA and the investigators for serious and unexpected adverse events or any finding from tests in
laboratory animals that suggests a significant risk for human subjects. Phase I, Phase 2 and Phase 3 clinical studies may not be
completed  successfully  within  any  specified  period,  if  at  all.  The  FDA  or  the  sponsor  or  its  data  safety  monitoring  board  may
suspend  a  clinical  study  at  any  time  on  various  grounds,  including  a  finding  that  the  research  subjects  or  patients  are  being
exposed to an unacceptable health risk. Similarly, an IRB can suspend or terminate approval of a clinical study at its institution if
the  clinical  study  is  not  being  conducted  in  accordance  with  the  IRB’s  requirements  or  if  the  pharmaceutical  product  has  been
associated with unexpected serious harm to patients.

Concurrent with clinical studies, companies usually complete additional animal studies and must also develop additional information
about the chemistry and physical characteristics of the pharmaceutical product as well as finalize a process for manufacturing the product in
commercial  quantities  in  accordance  with  cGMP  requirements.  The  manufacturing  process  must  be  capable  of  consistently  producing
quality batches of the pharmaceutical product candidate and, among other things, must develop methods for testing the identity, strength,
quality and purity of the final pharmaceutical product. Additionally, appropriate packaging must be selected and tested and stability studies
must be conducted to demonstrate that the pharmaceutical product candidate does not undergo unacceptable deterioration over its shelf life.

U.S. Review and Approval Processes

The  results  of  product  development,  preclinical  studies  and  clinical  studies,  along  with  descriptions  of  the  manufacturing  process,
analytical tests conducted on the chemistry of the pharmaceutical product, proposed labeling and other relevant information are submitted
to  the  FDA  as  part  of  an  NDA  requesting  approval  to  market  the  product.  The  submission  of  an  NDA  is  subject  to  the  payment  of
substantial user fees; a waiver of such fees may be obtained under certain limited circumstances.

In addition, under the Pediatric Research Equity Act (“PREA”), an NDA or supplement to an NDA must contain data to assess the
safety and effectiveness of the pharmaceutical product for the claimed indications in all relevant pediatric subpopulations and to support
dosing and administration for each pediatric subpopulation for which the product is safe and effective. The FDA may grant deferrals for
submission of data or full or partial waivers. Unless otherwise required by regulation, PREA does not apply to any pharmaceutical product
for an indication for which orphan designation has been granted.

The FDA reviews all NDAs submitted before it accepts them for filing and may request additional information rather than accepting
an NDA for filing. Once the submission is accepted for filing, the FDA begins an in-depth review of the NDA. Under the goals and policies
agreed to by the FDA under the Prescription Drug User Fee Act (“PDUFA”), the FDA has 10 months in which to complete its initial review
of a standard NDA and respond to the applicant, and six months for a priority NDA. The FDA does not always meet its PDUFA goal dates
for standard and priority NDAs. The review process and the PDUFA goal date may be extended by three months if the FDA requests or if
the  NDA  sponsor  otherwise  provides  additional  information  or  clarification  regarding  information  already  provided  in  the  submission
within the last three months before the PDUFA goal date.

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After the NDA submission is accepted for filing, the FDA reviews the NDA application to determine, among other things, whether
the proposed product is safe and effective for its intended use, and whether the product is being manufactured in accordance with cGMP to
assure and preserve the product’s identity, strength, quality and purity. The FDA may refer applications for novel pharmaceutical products
or pharmaceutical products which present difficult questions of safety or efficacy to an advisory committee, typically a panel that includes
clinicians and other experts, for review, evaluation and a recommendation as to whether the application should be approved and under what
conditions.  The  FDA  is  not  bound  by  the  recommendations  of  an  advisory  committee,  but  it  considers  such  recommendations  carefully
when making decisions. During the pharmaceutical product approval process, the FDA also will determine whether a risk evaluation and
mitigation  strategy  (“REMS”),  is  necessary  to  assure  the  safe  use  of  the  pharmaceutical  product.  If  the  FDA  concludes  that  a  REMS  is
needed, the sponsor of the NDA must submit a proposed REMS; the FDA will not approve the NDA without a REMS, if required.

Before approving an NDA, the FDA will inspect the facilities at which the product is manufactured. The FDA will not approve the
product  unless  it  determines  that  the  manufacturing  processes  and  facilities  are  in  compliance  with  cGMP  requirements  and  adequate  to
assure consistent production of the product within required specifications. Additionally, before approving an NDA, the FDA will typically
inspect one or more clinical sites as well as the site where the pharmaceutical product is manufactured to assure compliance with GCP and
cGMP.  If  the  FDA  determines  the  application,  manufacturing  process  or  manufacturing  facilities  are  not  acceptable,  it  will  outline  the
deficiencies  in  the  submission  and  often  will  request  additional  testing  or  information.  In  addition,  the  FDA  will  require  the  review  and
approval of product labeling.

The  NDA  review  and  approval  process  is  lengthy  and  difficult  and  the  FDA  may  refuse  to  approve  an  NDA  if  the  applicable
regulatory criteria are not satisfied or may require additional clinical data or other data and information. Even if such data and information
are submitted, the FDA may ultimately decide that the NDA does not satisfy the criteria for approval. Data obtained from clinical studies
are  not  always  conclusive  and  the  FDA  may  interpret  data  differently  than  the  sponsor  interprets  the  same  data.  The  FDA  will  issue  a
complete response letter if the agency decides not to approve the NDA. The complete response letter usually describes all of the specific
deficiencies  in  the  NDA  identified  by  the  FDA.  The  deficiencies  identified  may  be  minor,  for  example,  requiring  labeling  changes,  or
major, for example, requiring additional clinical studies. Additionally, the complete response letter may include recommended actions that
the applicant might take to place the application in a condition for approval. If a complete response letter is issued, the applicant may either
resubmit the NDA, addressing all of the deficiencies identified in the letter, or withdraw the application.

If  a  product  receives  regulatory  approval,  the  approval  may  be  significantly  limited  to  specific  diseases  and  dosages  or  the
indications for use may otherwise be limited, which could restrict the commercial value of the product. Further, the FDA may require that
certain contraindications, warnings or precautions be included in the product labeling. In addition, the FDA may require Phase IV testing
which  involves  clinical  studies  designed  to  further  assess  pharmaceutical  product  safety  and  effectiveness  and  may  require  testing  and
surveillance programs to monitor the safety of approved products that have been commercialized.

Expedited Development and Review Programs

The FDA has a Fast Track program that is intended to expedite or facilitate the process for reviewing new pharmaceutical products
that meet certain criteria. Specifically, new pharmaceutical products are eligible for Fast Track designation if they are intended to treat a
serious  or  life-threatening  condition  and  demonstrate  the  potential  to  address  unmet  medical  needs  for  the  condition.  The  Fast  Track
designation must be requested by the sponsor. Fast Track designation applies to the combination of the product and the specific indication
for which it is being studied. With a Fast Track designated product, the FDA may consider for review sections of the NDA on a rolling
basis before the complete application is submitted, if the sponsor provides a schedule for the submission of the sections of the NDA, if the
FDA agrees to accept sections of the NDA and determines that the schedule is acceptable and if the sponsor pays any required user fees
upon submission of the first section of the NDA.

Any product submitted to the FDA for marketing approval, including a Fast Track program, may also be eligible for other types of
FDA programs intended to expedite development and review, such as priority review and accelerated approval. Any product is eligible for
priority review if it has the potential to provide safe and effective therapy where no satisfactory alternative therapy exists or a significant
improvement  in  the  treatment,  diagnosis  or  prevention  of  a  disease  compared  to  marketed  products.  The  FDA  will  attempt  to  direct
additional  resources  to  the  evaluation  of  an  application  for  a  new  pharmaceutical  product  designated  for  priority  review  in  an  effort  to
facilitate the review. Additionally, a product may be eligible for accelerated approval. Pharmaceutical products studied for their safety and
effectiveness in treating serious or life-threatening illnesses and that provide meaningful therapeutic benefit over existing treatments may
receive accelerated approval, which means that the products may be approved on the basis of adequate and well-controlled clinical studies
establishing that the product has an effect on a surrogate endpoint that is reasonably likely to predict a clinical benefit, or on the basis of an
effect on a clinical endpoint other than survival or irreversible morbidity. As a condition of approval, the FDA may require that a sponsor of
a pharmaceutical product receiving accelerated approval perform adequate and well-controlled post-marketing clinical studies. In addition,
the FDA currently requires as a condition for accelerated approval pre-approval of promotional materials, which could adversely impact the
timing  of  the  commercial  launch  of  the  product.  Fast  Track  designation,  priority  review  and  accelerated  approval  do  not  change  the
standards for approval but may expedite the development or approval process.

15

 
 
 
 
 
 
 
 
 
 
Breakthrough Therapy Designation

The FDA is also required to expedite the development and review of the application for approval of drugs that are intended to treat a
serious  or  life-threatening  disease  or  condition  where  preliminary  clinical  evidence  indicates  that  the  drug  may  demonstrate  substantial
improvement over existing therapies on one or more clinically significant endpoints. Under the breakthrough therapy program, the sponsor
of  a  new  drug  candidate  may  request  that  the  FDA  designate  the  drug  candidate  for  a  specific  indication  as  a  breakthrough  therapy
concurrent  with,  or  after,  the  filing  of  the  IND  for  the  drug  candidate.  The  FDA  must  determine  if  the  drug  candidate  qualifies  for
breakthrough  therapy  designation  within  60  days  of  receipt  of  the  sponsor’s  request.  Validive  and  MNPR-101  may  both  be  eligible  for
breakthrough therapy designation.

European Union Drug Review and Approval

In  the  European  Economic Area  (“EEA”)  (which  is  comprised  of  the  28  Member  States  of  the  European  Union  plus  Norway,
Iceland and Liechtenstein), medicinal products can only be commercialized after obtaining a Marketing Authorization (“MA”). There are
two types of MA:

The Community MA, which is issued by the European Commission through the Centralized Procedure, based on the opinion of the
CHMP, or Committee for Medicinal Products for Human Use, of the European Medicines Agency (“EMA”), is valid throughout the entire
territory  of  the  EEA.  The  Centralized  Procedure  is  mandatory  for  certain  types  of  products,  such  as  biotechnology  medicinal  products,
orphan  medicinal  products,  and  medicinal  products  containing  a  new  active  substance  indicated  for  the  treatment  of  AIDS,  cancer,
neurodegenerative disorders, diabetes and auto-immune and viral diseases. The Centralized Procedure is optional for products containing a
new  active  substance  not  yet  authorized  in  the  EEA,  or  for  products  that  constitute  a  significant  therapeutic,  scientific  or  technical
innovation or which are in the interest of public health in the EU.

National  MAs,  which  are  issued  by  the  competent  authorities  of  the  Member  States  of  the  EEA  and  only  cover  their  respective
territory, are available for products not falling within the mandatory scope of the Centralized Procedure. Where a product has already been
authorized for marketing in a Member State of the EEA, this National MA can be recognized in other Member States through the Mutual
Recognition Procedure. If the product has not received a National MA in any Member State at the time of application, it can be approved
simultaneously in various Member States through the Decentralized Procedure. Under the above described procedures, before granting the
MA, the EMA or the competent authorities of the Member States of the EEA make an assessment of the risk-benefit balance of the product
on the basis of scientific criteria concerning its quality, safety and efficacy.

PRIME Designation

The EMA launched its PRIME regulatory initiative to enhance support for the development of therapies that target an unmet medical
need.  The  initiative  focuses  on  drugs  that  may  offer  a  major  therapeutic  advantage  over  existing  treatments,  or  benefit  patients  with  no
treatment options. These therapies are considered priority medicines within the EU. Through PRIME, the EMA offers early, proactive and
enhanced  support  to  drug  developers  to  optimize  the  generation  of  robust  data  on  a  therapy’s  benefits  and  risks  and  enable  accelerated
assessment of drug applications. MNPR-101 may be eligible for PRIME designation.

Post-Approval Requirements

Any  pharmaceutical  products  for  which  a  sponsor  receives  FDA  approvals  are  subject  to  continuing  regulation  by  the  FDA,
including,  among  other  things,  record-keeping  requirements,  reporting  of  adverse  experiences  with  the  product,  providing  the  FDA  with
updated  safety  and  efficacy  information,  product  sampling  and  distribution  requirements,  complying  with  certain  electronic  records  and
signature requirements and complying with FDA and FTC promotion and advertising requirements, which include, among others, standards
for  direct-to-consumer  advertising,  prohibitions  on  promoting  pharmaceutical  products  for  uses  or  in  patient  populations  that  are  not
described  in  the  pharmaceutical  product’s  approved  labeling  (known  as  “off-label  use”),  industry-sponsored  scientific  and  educational
activities  and  promotional  activities  involving  the  internet.  Failure  to  comply  with  FDA  requirements  can  have  negative  consequences,
including adverse publicity, enforcement letters from the FDA, actions by the U.S. Department of Justice and/or U.S. Department of Health
and Human Services Office of Inspector General, mandated corrective advertising or communications with doctors, and civil or criminal
penalties. Although physicians may prescribe legally available pharmaceutical products for off-label uses, manufacturers may not directly
or indirectly market or promote such off-label uses.

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Manufacturers of FDA approved products are required to comply with applicable FDA manufacturing requirements contained in the
FDA’s  cGMP  regulations.  cGMP  regulations  require,  among  other  things,  quality  control  and  quality  assurance,  as  well  as  the
corresponding  maintenance  of  records  and  documentation.  Pharmaceutical  product  manufacturers  and  other  entities  involved  in  the
manufacture and distribution of approved pharmaceutical products are required to register their establishments with the FDA and certain
state agencies, and are subject to periodic unannounced inspections by the FDA and certain state agencies for compliance with cGMP and
other laws. Accordingly, manufacturers must continue to expend time, money and effort in the area of production and quality control to
maintain cGMP compliance. Discovery of problems with a product after approval may result in restrictions on a product, manufacturer or
holder  of  an  approved  NDA,  including  withdrawal  of  the  product  from  the  market.  In  addition,  changes  to  the  manufacturing  process
generally require prior FDA approval before being implemented and other types of changes to the approved product, such as adding new
indications and additional labeling claims, are also subject to further FDA review and approval. The FDA also may require post-marketing
testing, known as Phase IV testing, risk minimization action plans and surveillance to monitor the effects of an approved product or place
conditions on an approval that could restrict the distribution or use of the product.

U.S. Foreign Corrupt Practices Act

The U.S. Foreign Corrupt Practices Act (“FCPA”), prohibits certain individuals and entities from promising, paying, offering to pay,
or authorizing the payment of anything of value to any foreign government official, directly or indirectly, to obtain or retain business or an
improper  advantage.  The  U.S.  Department  of  Justice  and  the  SEC  have  increased  their  enforcement  efforts  with  respect  to  the  FCPA.
Violations of the FCPA may result in large civil and criminal penalties and could result in an adverse effect on a company’s reputation,
operations, and financial condition. A company may also face collateral consequences such as debarment and the loss of export privileges.

Federal and State Pharmaceutical Legislation

In  addition  to  FDA  restrictions  on  marketing  of  pharmaceutical  products,  several  other  types  of  state  and  federal  laws  have  been

applied to restrict certain business practices in the biopharmaceutical industry.

Anti-Kickback Statute of 1972

The federal Anti-Kickback Statute prohibits, among other things, knowingly and willfully offering, paying, soliciting, or receiving
remuneration to induce or in return for purchasing, leasing, ordering, or arranging for the purchase, lease, or order of any healthcare item or
service  reimbursable  under  Medicare,  Medicaid,  or  other  federally  financed  healthcare  programs.  The  term  “remuneration”  has  been
broadly  interpreted  to  include  anything  of  value,  including  for  example,  gifts,  discounts,  the  furnishing  of  supplies  or  equipment,  credit
arrangements,  payments  of  cash,  waivers  of  payment,  ownership  interests  and  providing  anything  at  less  than  its  fair  market  value.  The
Anti-Kickback Statute has been interpreted to apply to arrangements between pharmaceutical manufacturers on one hand and prescribers,
purchasers,  and  formulary  managers  on  the  other.  Although  there  are  a  number  of  statutory  exemptions  and  regulatory  safe  harbors
protecting  certain  common  activities  from  prosecution,  the  exemptions  and  safe  harbors  are  drawn  narrowly,  and  a  company’s  practices
may not in all cases meet all of the criteria for statutory exemptions or safe harbor protection. Practices that involve remuneration that may
be alleged to be intended to induce prescribing, purchases,  or  recommendations  may  be  subject  to  scrutiny  if  they  do  not  qualify  for  an
exemption or safe harbor. Several courts have interpreted the statute’s intent requirement to mean that if any one purpose of an arrangement
involving remuneration is to induce referrals of federal healthcare covered business, the statute has been violated. The reach of the Anti-
Kickback  Statute  was  also  broadened  by  the  PPACA,  which,  among  other  things,  amends  the  intent  requirement  of  the  federal Anti-
Kickback  Statute.  Pursuant  to  the  statutory  amendment,  a  person  or  entity  no  longer  needs  to  have  actual  knowledge  of  this  statute  or
specific intent to violate it in order to have committed a violation. In addition, the PPACA provides that the government may assert that a
claim including items or services resulting from a violation of the federal Anti-Kickback Statute constitutes a false or fraudulent claim for
purposes of the civil False Claims Act (discussed below) or the civil monetary penalties statute, which imposes penalties against any person
who is determined to have presented or caused to be presented a claim to a federal health program that the person knows or should know is
for an item or service that was not provided as claimed or is false or fraudulent.

False Claims Act of 1986

The federal False Claims Act prohibits any person from knowingly presenting, or causing to be presented, a false claim for payment
to  the  federal  government.  Recently,  several  pharmaceutical  and  other  healthcare  companies  have  been  prosecuted  under  these  laws  for
allegedly providing free product to customers with the expectation that the customers would bill federal programs for the product. Other
companies  have  been  prosecuted  for  causing  false  claims  to  be  submitted  because  of  the  companies’  marketing  of  the  product  for
unapproved, and thus non-reimbursable, uses. Many states also have statutes or regulations similar to the federal Anti-Kickback Statute and
False Claims Act, which state laws apply to items and services reimbursed under Medicaid and other state programs, or, in several states,
apply regardless of the payer.

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Health Insurance Portability and Accountability Act of 1996 (“HIPPA”)

The  federal  Health  Insurance  Portability  and Accountability Act  of  1996  (“HIPAA”),  created  new  federal  criminal  statutes  that
prohibit knowingly and willfully executing a scheme to defraud any healthcare benefit program, including private third-party payers and
knowingly  and  willfully  falsifying,  concealing  or  covering  up  a  material  fact  or  making  any  materially  false,  fictitious  or  fraudulent
statement in connection with the delivery of or payment for healthcare benefits, items or services. Because of the breadth of these laws and
the  narrowness  of  the  federal Anti-Kickback  Statute’s  safe  harbors,  it  is  possible  that  some  of  a  company’s  business  activities  could  be
subject  to  challenge  under  one  or  more  of  such  laws.  Such  a  challenge  could  have  a  material  adverse  effect  on  a  company’s  business,
financial condition and results of operations. See “Risk Factors - Risks Related to Commercialization of Our Product Candidates.”

Health Information Technology for Economic and Clinical Health Act of 2009 (“HITECH”)

HIPAA, as amended by the Health Information Technology and Clinical Health Act (“HITECH”), and its implementing regulations,
imposes certain requirements relating to the privacy, security and transmission of individually identifiable health information. Among other
things, HITECH makes HIPAA’s privacy and security standards directly applicable to “business associates”—independent contractors or
agents of covered entities that receive or obtain protected health information in connection with providing a service on behalf of a covered
entity.  HITECH  also  increased  the  civil  and  criminal  penalties  that  may  be  imposed  against  covered  entities,  business  associates  and
possibly other persons, and gave state attorneys general new authority to file civil actions for damages or injunctions in federal courts to
enforce the federal HIPAA laws and seek attorney’s fees and costs associated with pursuing federal civil actions. In addition, state laws
govern the privacy and security of health information in certain circumstances, many of which differ from each other in significant ways
and may not have the same effect, thus complicating compliance efforts. See “Risk Factors - Risks Related to Commercialization of Our
Product Candidates.”

The Medicare Prescription Drug, Improvement and Modernization Act of 2003 (“MMA”)

In  the  U.S.  and  foreign  jurisdictions,  there  have  been  a  number  of  legislative  and  regulatory  changes  to  the  healthcare  system,  in
particular, there have been and continue to be a number of initiatives at the U.S. federal and state levels that seek to reduce healthcare costs.
The Medicare Prescription Drug, Improvement, and Modernization Act of 2003 (“MMA”), imposed new requirements for the distribution
and pricing of prescription drugs for Medicare beneficiaries. Under Part D, Medicare beneficiaries may enroll in prescription drug plans
offered by private entities, which will provide coverage of outpatient prescription drugs. Part D plans include both stand-alone prescription
drug benefit plans and prescription drug coverage as a supplement to Medicare Advantage plans. Unlike Medicare Part A and B, Part D
coverage is not standardized. Part D prescription drug plan sponsors are not required to pay for all covered Part D drugs, and each drug plan
can develop its own drug formulary that identifies which drugs it will cover and at what tier or level. However, Part D prescription drug
formularies must include drugs within each therapeutic category and class of covered Part D drugs, though not necessarily all the drugs in
each  category  or  class. Any  formulary  used  by  a  Part  D  prescription  drug  plan  must  be  developed  and  reviewed  by  a  pharmacy  and
therapeutic  committee.  Moreover,  while  the  MMA  applies  only  to  drug  benefits  for  Medicare  beneficiaries,  private  payers  often  follow
Medicare coverage policy and payment limitations in setting their own payment rates. Any reduction in payment that results from Medicare
Part D may result in a similar reduction in payments from non-governmental payers.

The American Recovery and Reinvestment Act of 2009

The American Recovery and Reinvestment Act of 2009 provides funding for the federal government to compare the effectiveness of
different treatments for the same illness. A plan for the research will be developed by the Department of Health and Human Services, the
Agency for Healthcare Research and Quality and the National Institutes for Health, and periodic reports on the status of the research and
related expenditures will be made to Congress. Although the results of the comparative effectiveness studies are not intended to mandate
coverage policies for public or private payers, it is not clear what effect, if any, the research will have on the sales of any product, if any
such product or the condition that it is intended to treat is the subject of a study.

Physician Payments Sunshine Act of 2010

The federal Physician Payments Sunshine Act requires certain manufacturers of drugs, devices, biologics and medical supplies for
which  payment  is  available  under  Medicare,  Medicaid  or  the  Children’s  Health  Insurance  Program,  with  specific  exceptions,  to  report
annually to the Centers for Medicare & Medicaid Services (“CMS”) information related to payments or other transfers of value made to
physicians and teaching hospitals, and applicable manufacturers and applicable group purchasing organizations to report annually to CMS
ownership and investment interests held by the physicians and their immediate family members.

18

 
 
 
 
 
 
 
 
 
 
 
 
 
Patent Protection and Affordable Care Act of 2010

In March 2010, the PPACA was enacted, which includes measures to significantly change the way healthcare is financed by both
governmental and private insurers. Among the provisions of the PPACA of importance to the pharmaceutical and biotechnology industry
are the following:

● an annual, nondeductible fee on any entity that manufactures or imports certain branded prescription drugs and biologic agents,

apportioned among these entities according to their market share in certain government healthcare programs, that began in 2011;

● an increase in the rebates a manufacturer must pay under the Medicaid Drug Rebate Program to 23.1% and 13% of the average

manufacturer price for branded and generic drugs, respectively;

● a new Medicare Part D coverage gap discount program, in which manufacturers must agree to offer 50% point-of-sale discounts to
negotiated  prices  of  applicable  brand  drugs  to  eligible  beneficiaries  during  their  coverage  gap  period,  as  a  condition  for  the
manufacturer’s outpatient drugs to be covered under Medicare Part D;

● extension  of  manufacturers’  Medicaid  rebate  liability  to  covered  drugs  dispensed  to  individuals  who  are  enrolled  in  Medicaid

managed care organizations;

● expansion  of  eligibility  criteria  for  Medicaid  programs  by,  among  other  things,  allowing  states  to  offer  Medicaid  coverage  to
additional individuals and by adding new mandatory eligibility categories for certain individuals with income at or below 133% of
the Federal Poverty Level beginning in 2014, thereby potentially increasing manufacturers’ Medicaid rebate liability;

● expansion of the entities eligible for discounts under the Public Health Service pharmaceutical pricing program
● new  requirements  under  the  federal  Open  Payments  program,  created  under  Section  6002  of  the  PPACA  and  its  implementing
regulations, that manufacturers of drugs, devices, biologics and medical supplies for which payment is available under Medicare,
Medicaid or the Children’s Health Insurance Program (with certain exceptions) report annually to the U.S. Department of Health
and  Human  Services  (“HHS”),  information  related  to  “payments  or  other  transfers  of  value”  made  or  distributed  to  physicians
(defined  to  include  doctors,  dentists,  optometrists,  podiatrists  and  chiropractors)  and  teaching  hospitals,  and  that  applicable
manufacturers and applicable group purchasing organizations report annually to HHS ownership and investment interests held by
physicians (as defined above) and their immediate family members, with data collection required beginning August 1, 2013 and
reporting to the Centers for Medicare & Medicaid Services (“CMS”), required by March 31, 2014 and by the 90th day of each
subsequent calendar year;

● a requirement to annually report drug samples that manufacturers and distributors provide to physicians, effective April 1, 2012;
● expansion of health care fraud and abuse laws, including the False Claims Act and the Anti-Kickback Statute, new government

investigative powers, and enhanced penalties for noncompliance;

● a licensure framework for follow-on biologic products;
● a  new  Patient-Centered  Outcomes  Research  Institute  to  oversee,  identify  priorities  in,  and  conduct  comparative  clinical

effectiveness research, along with funding for such research;

● creation  of  the  Independent  Payment  Advisory  Board  which,  beginning  in  2014,  will  have  authority  to  recommend  certain
changes to the Medicare program that could result in reduced payments for prescription drugs and those recommendations could
have the effect of law even if Congress does not act on the recommendations; and

● establishment  of  a  Center  for  Medicare  Innovation  at  CMS  to  test  innovative  payment  and  service  delivery  models  to  lower

Medicare and Medicaid spending, potentially including prescription drug spending that began on January 1, 2011.

Budget Control Act of 2011

In August 2011, the President signed into law the Budget Control Act of 2011, which, among other things, created the Joint Select
Committee on Deficit Reduction, or joint committee, to recommend proposals in spending reductions to Congress. The joint committee did
not achieve its targeted deficit reduction of at least $1.2 trillion and for the years 2013 through 2021, triggering automatic reductions to
several  government  programs.  These  reductions  include  aggregate  reductions  to  Medicare  payments  to  providers  of  up  to  2%  per  fiscal
year, starting in 2013.

19

 
 
 
 
 
 
 
 
American Taxpayer Relief Act of 2012

In  January  2013,  the  President  signed  into  law  the American  Taxpayer  Relief Act  of  2012,  which,  among  other  things,  reduced
Medicare  payments  to  several  providers  and  increased  the  statute  of  limitations  period  for  the  government  to  recover  overpayments  to
providers from three to five years. These new laws may result in additional reductions in Medicare and other healthcare funding.

Proposals in Congress to repeal or replace parts of the PPACA

There have been a number of proposals in the U.S. Congress to repeal or replace parts of the PPACA. Some of the proposals include
the  repeal  of  the  tax  on  prescription  medications,  repeal  of  the  medical  device  excise  tax  for  sales,  and  repeal  of  the  elimination  of  a
deduction for expenses allocable to Medicare Part D subsidy. It is uncertain whether any repeal or replace legislation will be passed and
signed into law or what effect any such legislation may have on our commercialization strategy. See “Risk Factors - Future Legislation,
Executive  or  Private  Sector Action  May  Increase  the  Difficulty  and  Cost  for  us  to  Commercialize  our  Products  and Affect  the  Prices
Obtained for Such Products.”

Patent Term Restoration and Marketing Exclusivity

Depending upon the timing, duration and specifics of the FDA approval of the use of our pharmaceutical product candidates, some
of our products to be licensed under U.S. patents may be eligible for limited patent term extension under the Drug Price Competition and
Patent  Term  Restoration  Act  of  1984,  commonly  referred  to  as  the  Hatch-Waxman  Amendments.  The  Hatch-Waxman  Amendments
permits  a  patent  restoration  term  of  up  to  five  years  as  compensation  for  patent  term  lost  during  product  development  and  the  FDA
regulatory review process. However, patent term restoration cannot extend the remaining term of a patent beyond a total of 14 years from
the product’s approval date. The patent term restoration period is generally one-half the time between the effective date of an IND and the
submission date of an NDA plus the time between the submission date of an NDA and the approval of that application. Only one patent
applicable to an approved pharmaceutical product is eligible for the extension and the application for the extension must be submitted prior
to the expiration of the patent. The U.S. Patent and Trademark Office (“USPTO”), in consultation with the FDA, reviews and approves the
application for any patent term extension or restoration.

Market exclusivity provisions under the U.S. Food, Drug, and Cosmetic Act can also delay the submission or the approval of certain

applications of other companies seeking to reference another company’s NDA.

The Biologics Price Competition and Innovation Act (“BPCI Act”)

The  Biologics  Price  Competition  and  Innovation Act,  (“BPCI Act”),  authorizes  the  FDA  to  license  a  biological  product  that  is
biosimilar to an FDA-licensed biologic through an abbreviated pathway. The BPCI Act establishes criteria for determining that a product is
biosimilar to an already-licensed biologic, or reference product, and establishes a process by which an abbreviated BLA for a biosimilar
product  is  submitted,  reviewed  and  approved.  The  BPCI  Act  provides  periods  of  exclusivity  that  protect  a  reference  product  from
biosimilars competition. Under the BPCI Act, the FDA may not accept a biosimilar application for review until four years after the date of
first licensure of the reference product, and the biosimilar may not be licensed until at least 12 years after the reference product’s approval.
Additionally, the BPCI Act establishes procedures by which the biosimilar applicant provides information about its application and product
to the reference product sponsor, and by which information about potentially relevant patents may be shared and litigation over patents may
proceed in advance of approval. The BPCI Act also provides a period of exclusivity for the first biosimilar determined by the FDA to be
interchangeable with the reference product.

We anticipate that the contours of the BPCI Act will continue to be defined as the statute is implemented over a period of years. This
likely will be accomplished by a variety of means, including decisions related to the statute by the relevant federal courts, FDA issuance of
guidance documents, and FDA decisions in the course of considering specific applications. The FDA has to date issued various guidance
documents and other materials indicating the agency’s thinking regarding a number of issues implicated by the BPCI Act. Additionally, the
FDA’s approval of several biosimilar applications in recent years has helped define the agency’s approach to certain issues.

20

 
 
 
 
 
 
 
 
 
 
 
 
 
Pharmaceutical Coverage, Pricing and Reimbursement

Significant uncertainty exists as to the coverage and reimbursement status of any pharmaceutical product candidates for which we
obtain regulatory approval. In the U.S. and markets in other countries, sales of any products for which we receive regulatory approval for
commercial sale will depend in part upon the availability of reimbursement from third-party payers. Third-party payers include government
payers  such  as  Medicare  and  Medicaid,  managed  care  providers,  private  health  insurers  and  other  organizations.  The  process  for
determining whether a payer will provide coverage for a pharmaceutical product may be separate from the process for setting the price or
reimbursement  rate  that  the  payer  will  pay  for  the  pharmaceutical  product.  Third-party  payers  may  limit  coverage  to  specific
pharmaceutical products on an approved list, or formulary, which might not include all of the FDA-approved pharmaceutical products for a
particular indication. Third-party payers are increasingly challenging the price and examining the medical necessity and cost-effectiveness
of medical products and services, in addition to their safety and efficacy. We may need to conduct expensive pharmaco-economic studies in
order  to  demonstrate  the  medical  necessity  and  cost-effectiveness  of  its  products,  in  addition  to  the  costs  required  to  obtain  the  FDA
approvals. A payer’s decision to provide coverage for a pharmaceutical product does not imply that an adequate reimbursement rate will be
approved.

In  2003,  the  federal  government  enacted  legislation  providing  a  partial  prescription  drug  benefit  for  Medicare  recipients,  which
became effective at the beginning of 2006. However, to obtain payments under this program, a company would be required to sell products
to Medicare recipients through prescription drug plans operating pursuant to this legislation. As part of their participation in the Medicare
prescription drug program, these plans negotiate discounted prices for prescription drugs. Federal, state and local governments in the U.S.
continue  to  consider  legislation  to  limit  the  growth  of  health  care  costs,  including  the  cost  of  prescription  drugs.  Future  legislation  and
regulations could limit payments for pharmaceuticals such as the drug product candidates that we are developing.

Different pricing and reimbursement schemes exist in other countries. In the European Community, governments influence the price
of pharmaceutical products through their pricing and reimbursement rules and control of national health care systems that fund a large part
of the cost of those products to consumers. Some jurisdictions operate positive and negative list systems under which products may only be
marketed once a reimbursement price has been agreed upon. To obtain reimbursement or pricing approval, some of these countries may
require the completion of clinical studies that compare the cost-effectiveness of a particular pharmaceutical product candidate to currently
available therapies. Other member states allow companies to fix their own prices for medicines, but monitor and control company profits.
The downward pressure on health care costs in general, particularly prescription drugs, has become very intense. As a result, increasingly
high barriers are being erected to the entry of new products. In addition, in some countries, cross-border imports from low-priced markets
exert a commercial pressure on pricing within a country.

International Regulation

In addition to regulations in the U.S., there are a variety of foreign regulations governing clinical studies and commercial sales and
distribution  of  our  future  product  candidates.  Whether  or  not  FDA  approval  is  obtained  for  a  product,  approval  of  a  product  must  be
obtained by the comparable regulatory authorities of foreign countries before clinical studies or marketing of the product can commence in
those countries. The approval process varies from country to country, and the time may be longer or shorter than that required for FDA
approval.  The  requirements  governing  the  conduct  of  clinical  studies,  product  licensing,  pricing  and  reimbursement  vary  greatly  from
country to country. In addition, certain regulatory authorities in select countries may require us to repeat previously conducted preclinical
and/or clinical studies under specific criteria for approval in their respective country which may delay and/or greatly increase the cost of
approval in certain markets targeted for approval by us.

Under E.U. regulatory systems, marketing applications for pharmaceutical products must be submitted under a centralized procedure
to the EMA. The centralized procedure provides for the grant of a single marketing authorization that is valid for all E.U. member states.
The EMA also has designations for Orphan Drugs, which, if applicable, can provide for faster review, lower fees and more access to advice
during  drug  development.  While  the  marketing  authorization  in  the  European  Union  is  centralized,  the  system  for  clinical  studies
(application,  review  and  requirements)  is  handled  by  each  individual  country. Approval  to  run  a  clinical  study  in  one  country  does  not
guarantee approval in any other country. The pharmaceutical industry in Canada is regulated by Health Canada. A New Drug Submission
(“NDS”) is the equivalent of a U.S. NDA and must be filed to obtain approval to market a pharmaceutical product in Canada. Marketing
regulations and reimbursement are subject to national and provincial laws. In Japan, applications for approval to manufacture and market
new drugs must be approved by the Ministry of Health, Labor and Welfare. Nonclinical and clinical studies must meet the requirements of
Japanese  laws.  Results  from  clinical  studies  conducted  outside  of  Japan  must  be  supplemented  with  at  least  a  bridging  clinical  study
conducted in Japanese patients.

21

 
 
 
 
 
 
 
 
 
 
In addition to regulations in Europe, Canada, Japan and the U.S., there are a variety of foreign regulations governing clinical studies,
commercial distribution and reimbursement of future product candidates which we may be subject to as we pursue regulatory approval and
commercialization of Validive, MNPR-201, MNPR-101, or any future product candidates internationally.

Compliance with Environmental Laws

Since we do not have our own laboratory facilities, we do not estimate any annual costs of compliance with environmental laws.

Employees

Our operations are currently overseen by five individuals, of which three have a PhD, two have an MD, one has an MBA, one has an
MSc in health economics and policy, and one has an inactive CPA. They have worked at industry leading companies such as BioMarin
Pharmaceutical  Inc.,  Raptor  Pharmaceuticals,  Abbott  Laboratories,  and  Onyx  Pharmaceuticals.  As  of  March  1,  2018,  we  have  five
employees;  four  of  them  are  full-time  employees.  For  information  regarding  our  executive  officers,  see  the  section  entitled  “Executive
Officers and Board Members.”

Available Information

Our Annual  Reports  on  Form  10-K,  Quarterly  Reports  on  Form  10-Q,  Current  Reports  on  Form  8-K  and  amendments  to  those
reports  filed  or  furnished  pursuant  to  Section  13(a)  or  15(d)  of  the  Exchange  Act  may  be  accessed  through  the  SEC’s  website  at
www.sec.gov  and  on  our  website  at www.monopartx.com  free  of  charge.  Such  filings  are  placed  on  our  website  as  soon  as  reasonably
practicable after they are filed with the SEC. Our Code of Business Conduct and Ethics and our Audit Committee Charter are also posted
on the Investor Highlight page on our website.

Item 1A. Risk Factors

RISK FACTORS

An investment in our common stock involves a high degree of risk. A prospective investor should carefully consider the following
information about these risks, together with other information appearing elsewhere in this Annual Report on Form 10-K, before deciding to
invest in our common stock. The occurrence of any of the following risks could have a material adverse effect on our business, financial
condition, results of operations and future prospects and prospective investors could lose all or part of their investment. The risk factors
discussed  below  and  elsewhere  in  this Annual  Report  on  Form  10-K  are  not  exhaustive;  other  significant  risks  may  exist  that  are  not
identified  in  this Annual  Report  on  Form  10-K,  but  that  might  still  materially  and  adversely  affect  our  business,  prospects,  financial
condition, and results of operations were any of such risks to occur.

Risks Related to Our Financial Condition and Capital Requirements

We have a limited operating history, expect to incur significant operating losses, and have a high risk of never being profitable.

We commenced operations in December 2014 and have a limited operating history of almost three years. Therefore, there is limited
historical financial or operational information upon which to evaluate our performance. Our prospects must be considered in light of the
uncertainties, risks, expenses, and difficulties frequently encountered by companies in their early stages of operations. Most companies in
our industry at our stage of development never become profitable, and are acquired or go out of business without successfully developing
any product that generates revenue from commercial sales.

From inception in December 2014 through December 31, 2017, we have incurred losses of approximately $18.4 million. We expect
to continue to incur substantial operating losses over the next several years for the clinical development of our current and future licensed or
purchased drug product candidates.

The  amount  of  future  losses  and  when,  if  ever,  we  will  become  profitable  are  uncertain.  We  do  not  have  any  products  that  have
generated any revenues from commercial sales, and do not expect to generate revenues from the commercial sale of products in the near
future, if ever. Our ability to generate revenue and achieve profitability will depend on, among other things, successful completion of the
development  of  our  product  candidates;  obtaining  necessary  regulatory  approvals  from  the  FDA  and  international  regulatory  agencies;
establishing manufacturing, sales, and marketing arrangements with third parties; obtaining adequate reimbursement by third party payers;
and  raising  sufficient  funds  to  finance  our  activities.  If  we  are  unsuccessful  at  some  or  all  of  these  undertakings,  our  business,  financial
condition, and results of operations are expected to be materially and adversely affected.

22

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
As a new public reporting company, we are subject to SEC reporting and other requirements, which will lead to increased operating

costs in order to meet these requirements.

If we continue to incur operating losses and fail to obtain the capital necessary to fund our operations, we will be unable to advance our
development  programs,  complete  our  clinical  trials,  or  bring  products  to  market,  or  may  be  forced  to  cease  operations  entirely.  In
addition, any capital obtained by us may be obtained on terms that are unfavorable to us, our investors, or both.

Developing  a  new  drug  and  conducting  clinical  trials  for  one  or  more  disease  indications  involves  substantial  costs.  We  have
projected  cash  requirements  for  the  near  term  based  on  a  variety  of  assumptions,  but  some  or  all  of  such  assumptions  are  likely  to  be
incorrect  and/or  incomplete,  possibly  materially  in  an  adverse  direction.  Our  actual  cash  needs  may  deviate  materially  from  those
projections, changes in market conditions or other factors may increase our cash requirements, or we may not be successful even in raising
the  amount  of  cash  we  currently  project  will  be  required  for  the  near  term.  See  discussion  of  our  material  development  agreements  in
“Material Agreements”. We will need to raise additional capital in the future; the amount of additional capital needed will vary as a result
of a number of factors, including without limitation the following:

● receiving less funding than we require;
● higher than expected costs to manufacture our active pharmaceutical ingredient and our drug product candidates;
● higher than expected costs for preclinical testing;
● an increase in the number, size, duration, or complexity of our clinical trials;
● slower  than  expected  progress  in  developing  Validive,  MNPR-201,  MNPR-101,  or  other  drug  product  candidates,  including

without limitation, additional costs caused by program delays;

● higher than expected costs associated with attempting to obtain regulatory approvals, including without limitation additional costs

caused by additional regulatory requirements or larger clinical trial requirements;

● higher than expected personnel or other costs, such as adding personnel or pursuing the licensing/acquisition of additional assets;

and

● higher than expected costs to protect our intellectual property portfolio or otherwise pursue our intellectual property strategy.

If  we  attempt  to  raise  additional  financing,  there  can  be  no  assurance  that  we  will  be  able  to  secure  such  additional  financing  in
sufficient  quantities  or  at  all.  We  may  be  unable  to  raise  additional  capital  for  reasons  including  without  limitation  our  financial
performance, investor confidence in us and the biopharmaceutical industry, credit availability from banks and other financial institutions,
the status of current projects, and our prospects for obtaining any necessary regulatory approvals. Potential investors’ capital investments
may be shifted to other opportunities with perceived greater returns and/or lower risk thereby reducing capital available to us, if at all.

In addition, any additional financing might not be available and even if available, may not be available on terms favorable to us or
our then-existing investors. We may seek to raise funds through public or private equity offerings, debt financings, corporate collaboration
or licensing arrangements, mergers, acquisitions, sales of intellectual property, or other financing vehicles or arrangements. To the extent
that  we  raise  additional  capital  by  issuing  equity  securities  or  other  securities,  our  then-existing  investors  may  experience  significant
dilution.  If  we  raise  funds  through  debt  financings  or  bank  loans,  we  may  become  subject  to  restrictive  covenants,  our  assets  may  be
pledged as collateral for the debt, and the interests of our then-existing investors would be subordinated to the debt holders or banks. In
addition, our use of and ability to exploit assets pledged as collateral for debt or loans may be restricted or forfeited. To the extent that we
raise  additional  funds  through  collaboration  or  licensing  arrangements,  we  may  be  required  to  relinquish  significant  rights  (including
without limitation intellectual property rights) to our technologies or product candidates, or grant licenses on terms that are not favorable to
us. If we are not able to raise needed funding under acceptable terms or at all, then we will have to reduce expenses, including the possible
options of curtailing operations, abandoning opportunities, selling off assets, reducing costs, or ceasing operations entirely.

23

 
 
 
 
 
 
 
 
 
Risks Related to Clinical Development and Regulatory Approval

We do not have and may never have any approved products on the market. Our business is highly dependent upon receiving approvals
from various U.S. and international governmental agencies and will be severely harmed if we are not granted approval to manufacture
and sell our drug product candidates.

In order for us to commercialize any treatment for a cancer indication or for any other clinical indication, we must obtain regulatory
approvals of such treatment for that indication. Satisfying regulatory requirements is an expensive process that typically takes many years
and  involves  compliance  with  requirements  covering  research  and  development,  testing,  manufacturing,  quality  control,  labeling,  and
promotion of drugs for human use. To obtain necessary regulatory approvals, we must, among other requirements, complete clinical trials
demonstrating that our products are safe and effective for a particular indication. There can be no assurance that our products are safe and
effective,  that  our  clinical  trials  will  demonstrate  the  necessary  safety  and  effectiveness  of  our  drug  product  candidates,  or  that  we  will
succeed in obtaining regulatory approval for any treatment we develop even if such safety and effectiveness are demonstrated.

Any  delays  or  difficulties  we  encounter  in  our  clinical  trials  may  delay  or  preclude  regulatory  approval  from  the  FDA  or  from
international  regulatory  organizations.  Any  delay  or  preclusion  of  regulatory  approval  would  be  expected  to  delay  or  preclude  the
commercialization of our products. Examples of delays or difficulties that we may encounter in our clinical trials include without limitation
the following:

● Clinical trials may not yield sufficiently conclusive results for regulatory agencies to approve the use of our products.
● Our products may fail to be more effective than current therapies, or to be effective at all.
● We may discover that our products have adverse side effects, which could cause our products to be delayed or precluded from

receiving regulatory approval or otherwise expose us to significant commercial and legal risks.

● It may take longer than expected to determine whether or not a treatment is effective.
● Patients involved in our clinical trials may suffer severe adverse side effects even up to death, whether as a result of treatment

with our products, the withholding of such treatment, or other reasons (whether within or outside of our control).

● We may fail to enroll a sufficient number of patients in our clinical trials.
● Patients  enrolled  in  our  clinical  trials  may  not  have  the  characteristics  necessary  to  obtain  regulatory  approval  for  a  particular

indication.

● We may be unable to produce sufficient quantities of product to complete the clinical trials.
● Even if we are successful in our clinical trials, any required governmental approvals may still not be obtained or, if obtained, may

not be maintained.

● If  approval  for  commercialization  is  granted,  it  is  possible  the  authorized  use  will  be  more  limited  than  is  necessary  for
commercial  success,  or  that  approval  may  be  conditioned  on  completion  of  further  clinical  trials  or  other  activities,  which  will
cause a substantial increase in costs and which we might not succeed in performing or completing.

● If granted, approval may be withdrawn or limited if problems with our products emerge or are suggested by the data arising from

their use or if there is a change in law or regulation.

Any success we may achieve at a given stage of our clinical trials does not guarantee that we will achieve success at any subsequent

stage, including without limitation final FDA approval.

We  may  encounter  delays  or  rejections  in  the  regulatory  approval  process  because  of  additional  government  regulation  resulting
from future legislation or administrative action, or from changes in the policies of the FDA or other regulatory bodies during the period of
product development, clinical trials, or regulatory review. Failure to comply with applicable regulatory requirements may result in criminal
prosecution,  civil  penalties,  recall  or  seizure  of  products,  total  or  partial  suspension  of  production,  or  an  injunction  preventing  certain
activity,  as  well  as  other  regulatory  action  against  our  product  candidates  or  us. As  a  company,  we  have  no  experience  in  successfully
obtaining  regulatory  approval  for  a  drug  and  thus  may  be  poorly  equipped  to  gauge,  and  may  prove  unable  to  manage  risks  relating  to
obtaining such approval.

Outside  the  U.S.,  our  ability  to  market  a  product  is  contingent  upon  receiving  clearances  from  appropriate  non-U.S.  regulatory
authorities. Non-U.S. regulatory approval typically includes all of the risks associated with FDA clearance discussed above as well as the
additional uncertainties and potential prejudices faced by U.S. companies conducting business abroad. In certain cases, pricing restrictions
and practices can make achieving even limited profitability very difficult.

24

 
 
 
 
 
 
 
 
 
 
 
If  we  or  our  licensees,  development  collaborators,  or  suppliers  are  unable  to  manufacture  our  products  in  sufficient  quantities  or  at
defined quality specifications, or are unable to obtain regulatory approvals for the manufacturing facility, we may be unable to develop
and/or meet demand for our products and lose time to market and potential revenues.

Completion of our clinical trials and commercialization of our product candidates require access to, or development of, facilities to
manufacture a sufficient supply of our product candidates. We currently contract with outside sources to manufacture MNPR-101. In order
to  be  able  to  manufacture  sufficient  quantities  of  MNPR-101  to  be  able  to  proceed  with  human  clinical  trials,  Cancer  Research  UK
developed a new cell line under our CTOA. We received notification of termination of CRUK’s work on MNPR-101 under the CTOA on
March 21, 2018. There can be no assurance that this new cell line will be successful or that sufficient quantities of MNPR-101 will be able
to  be  manufactured.  Since  Cancer  Research  UK  has  decided  to  terminate  its  involvement  with  MNPR-101,  we  will  need  to  make  other
arrangements  for  the  clinical  testing,  development  and  manufacture  of  our  drug  product  candidate.  There  can  be  no  assurance  that  such
alternative arrangements can be made or on terms favorable to us. We in the future may become unable, for various reasons, to rely on our
sources for the manufacture of our product candidates, either for clinical trials or, at some future date, for commercial distribution. We may
not  be  successful  in  identifying  additional  or  replacement  third-party  manufacturers,  or  in  negotiating  acceptable  terms  with  any  we  do
identify.  We  may  face  competition  for  access  to  these  manufacturers’  facilities  and  may  be  subject  to  manufacturing  delays  if  the
manufacturers give other clients higher priority than they give to us. Even if we are able to identify an additional or replacement third-party
manufacturer, the delays and costs associated with establishing and maintaining a relationship with such manufacturer may have a material
adverse effect on us.

Before  we  can  begin  to  commercially  manufacture  Validive,  MNPR-201,  MNPR-101,  or  any  other  product  candidate,  we  must
obtain regulatory approval of the manufacturing facility and process. Manufacturing of drugs for clinical and commercial purposes must
comply  with  the  FDA's  current  Good  Manufacturing  Practices  requirements,  commonly  known  as  “cGMP”,  and  applicable  non-U.S.
regulatory  requirements.  The  cGMP  requirements  govern  quality  control  and  documentation  policies  and  procedures.  Complying  with
cGMP and non-U.S. regulatory requirements will require that we expend time, money, and effort in production, recordkeeping, and quality
control  to  ensure  that  the  product  meets  applicable  specifications  and  other  requirements.  We,  or  our  contracted  manufacturing  facility,
must also pass a pre-approval inspection prior to FDA approval. Failure to pass a pre-approval inspection may significantly delay or prevent
FDA approval of our products. If we fail to comply with these requirements, we would be subject to possible regulatory action and may be
limited in the jurisdictions in which we are permitted to sell our products and will lose time to market and potential revenues.

It  is  uncertain  whether  insurance  will  be  adequate  to  address  product  liability  claims,  or  that  insurance  against  such  claims  will  be
affordable or available on acceptable terms in the future.

Clinical research involves the testing of new drugs on human volunteers pursuant to a clinical trial protocol. Such testing involves a
risk of liability for personal injury to or death of patients due to, among other causes, adverse side effects, improper administration of the
new  drug,  or  improper  volunteer  behavior.  Claims  may  arise  from  patients,  clinical  trial  volunteers,  consumers,  physicians,  hospitals,
companies,  institutions,  researchers,  or  others  using,  selling,  or  buying  our  products,  as  well  as  from  governmental  bodies.  In  addition,
product liability and related risks are likely to increase over time, in particular upon the commercialization or marketing of any products by
us  or  parties  with  which  we  enter  into  development,  marketing,  or  distribution  collaborations. Although  we  are  contracting  for  general
liability  insurance  in  connection  with  our  ongoing  business,  there  can  be  no  assurance  that  the  amount  and  scope  of  such  insurance
coverage  will  be  appropriate  and  sufficient  in  the  event  any  claims  arise,  that  we  will  be  able  to  secure  additional  coverage  should  we
attempt to do so, or that our insurers would not contest or refuse any attempt by us to collect on such insurance policies. Furthermore, there
can  be  no  assurance  that  suitable  insurance  will  continue  to  be  available  on  terms  acceptable  to  us  or  at  all,  or  that,  if  obtained,  the
insurance coverage will be appropriate and sufficient to cover any potential claims or liabilities.

Risks Related to Our Reliance on Third Parties

Corporate, non-profit, and academic collaborators may take actions (including lack of effective actions) to delay, prevent, or undermine
the success of our products.

Our  operating  and  financial  strategy  for  the  development,  clinical  testing,  manufacture,  and  commercialization  of  drug  product
candidates  is  heavily  dependent  on  us  entering  into  collaborations  with  corporations,  non-profit  organizations,  academic  institutions,
licensors, licensees, and other parties. There can be no assurance that we will be successful in establishing such collaborations. Some of our
existing  collaborations  are,  and  future  collaborations  may  be  terminable  at  the  sole  discretion  of  the  collaborator.  For  example,  our
collaboration with Cancer Research UK on MNPR-101, we recently received notification of termination by CRUK of its involvement with
MNPR-101 and we will need to seek alternate arrangements. Replacement collaborations might not be available on attractive terms, or at
all. The activities of any collaborator will not be within our control and may not be in our power to influence. There can be no assurance
that any collaborator will perform its obligations to our satisfaction or at all; that we will derive any revenue, profits, or benefit from such
collaborations; or that any collaborator will not compete with us. If any collaboration is not pursued, we may require substantially greater
capital to undertake development and commercialization of our proposed products, and may not be able to develop and commercialize such
products  effectively,  if  at  all.  In  addition,  a  lack  of  development  and  commercialization  collaborations  may  lead  to  significant  delays  in
introducing  proposed  products  into  certain  markets  and/or  reduced  sales  of  proposed  products  in  such  markets.  Furthermore,  current  or
future collaborators may act deliberately or inadvertently in ways detrimental to our interests.

25

 
 
 
 
 
 
 
 
 
 
 
The termination of third-party licenses could adversely affect our rights to important compounds.

We rely on certain rights to MNPR-101 that we have secured through a non-exclusive license agreement with XOMA. XOMA, as
licensor, has the ability to terminate the license if we breach our obligations under the license agreement and do not remedy any such breach
in  time  after  receiving  written  notice  of  such  breach  from  XOMA.  A  termination  of  the  license  agreement  might  force  us  to  cease
developing and/or selling MNPR-101, if it gets to market. We have exercised our option to license Validive; as such, Onxeo has the ability
to  terminate  the  license  if  we  breach  our  obligations  under  the  option  and  license  agreement. A  termination  of  the  option  and  license
agreement might force us to cease developing and/or selling Validive.

Data provided by collaborators and other parties upon which we rely have not been independently verified and could turn out to be false,
misleading, or incomplete.

We rely on third-party vendors, scientists, and collaborators to provide us with significant data and other information related to our
projects, clinical trials, and business. We do not independently verify or audit all of such data (including possibly material portions thereof).
As a result, such data may be inaccurate, misleading, or incomplete.

In certain cases, we rely on a single supplier for a particular manufacturing material, and any interruption in or termination of service
by such supplier could delay or disrupt the commercialization of our products.

We  rely  on  third-party  suppliers  for  the  materials  used  to  manufacture  our  compounds.  Some  of  these  materials  may  only  be
available  from  one  supplier.  Any  interruption  in  or  termination  of  service  by  such  single  source  suppliers  could  result  in  a  delay  or
disruption  in  manufacturing  until  we  locate  an  alternative  source  of  supply.  There  can  be  no  assurance  that  we  would  be  successful  in
locating such alternative source of supply or in negotiating acceptable terms with such prospective supplier.

Risks Related to Commercialization of Our Product Candidates

Our  product  development  efforts  are  at  an  early  stage.  We  have  not  yet  undertaken  any  marketing  efforts,  and  there  can  be  no
assurances  that  future  anticipated  market  testing  and  analyses  will  validate  our  marketing  strategy  and  therefore  we  may  need  to
modify the products, or will not be successful in either developing or marketing those products.

We have not completed the development or clinical trials of any product candidates and, accordingly, have not yet begun to market
or  generate  revenue  from  the  commercialization  of  any  products.  Commercializing  these  product  candidates  will  require  substantial
additional  research  and  development  as  well  as  costly  clinical  trials.  There  can  be  no  assurance  that  we  will  successfully  complete
development  of  our  product  candidates  or  successfully  market  them.  We  may  encounter  problems  and  delays  relating  to  research  and
development, regulatory approval, intellectual property rights of product candidates, or other factors. There can be no assurance that our
development programs will be successful, that our products, if successfully developed, will prove to be safe and effective in or after clinical
trials, that the necessary regulatory approvals for any product candidates will be obtained, or, even if obtained, will be as broad as sought or
will be maintained for any period thereafter, that patents will issue on our patent applications, that any intellectual property protections we
secure will be adequate, or that our collaboration arrangements will not diminish the value of our intellectual property through licensing or
other  arrangements.  Furthermore,  there  can  be  no  assurance  that  any  product  we  might  market  will  be  received  favorably  by  customers
(whether physicians, patients, or both), adequately reimbursed by third party payers, or that competitive products will not perform better
and/or be marketed more successfully. Additionally, there can be no assurances that any future market testing and analyses will validate
our marketing strategies. We may need to seek to modify the product labels through additional studies in order to be able to market them
successfully.

If we are unable to establish relationships with licensees or collaborators to carry out sales, marketing, and distribution functions or to
create effective marketing, sales, and distribution capabilities, we will be unable to market our products successfully.

Our  business  strategy  may  include  out-licensing  product  candidates  to  or  collaborating  with  larger  firms  with  experience  in
marketing and selling pharmaceutical products. There can be no assurance that we will successfully be able to establish marketing, sales, or
distribution  relationships  with  any  third  party,  that  such  relationships,  if  established,  will  be  successful,  or  that  we  will  be  successful  in
gaining  market  acceptance  for  any  products  we  might  develop.  To  the  extent  that  we  enter  into  any  marketing,  sales,  or  distribution
arrangements with third parties, our product revenues per unit sold are expected to be lower than if we marketed, sold, and distributed our
products directly, and any revenues we receive will depend upon the efforts of such third parties.

If we are unable to establish such third-party marketing and sales relationships, or choose not to do so, we would have to establish in-
house  marketing  and  sales  capabilities.  We  have  no  experience  in  marketing  or  selling  oncology  pharmaceutical  products,  and  currently
have  no  marketing,  sales,  or  distribution  infrastructure  and  no  experience  developing  or  managing  such  infrastructure  for  an  oncology
product. To market any products directly, we would have to establish a marketing, sales, and distribution force that had technical expertise
and could support a distribution capability. Competition in the biopharmaceutical industry for technically proficient marketing, sales, and
distribution personnel is intense and attracting and retaining such personnel may significantly increase our costs. There can be no assurance
that we will be able to establish internal marketing, sales, or distribution capabilities or that these capabilities will be sufficient to meet our
needs.

26

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Commercial success of our product candidates will depend on the acceptance of these products by physicians and patients.

Any product candidate that we may develop may not gain market acceptance among physicians and patients. Market acceptance of

and demand for any product that we may develop will depend on many factors, including without limitation:

● prevalence and severity of adverse side effects;
● potential advantages over alternative treatments;
● cost effectiveness;
● convenience and ease of administration;
● sufficient third-party coverage or reimbursement;
● strength of marketing and distribution support; and
● our ability to provide acceptable evidence of safety and efficacy.

If any product candidate developed by us receives regulatory approval but does not achieve an adequate level of market acceptance

by physicians and patients, we may generate little or no product revenue and may not become profitable.

Our products may not be accepted for reimbursement or properly reimbursed by third-party payers.

The successful commercialization of any products we might develop will depend substantially on whether the costs of our products
and  related  treatments  are  reimbursed  at  acceptable  levels  by  government  authorities,  private  healthcare  insurers,  and  other  third-party
payers,  such  as  health  maintenance  organizations.  Reimbursement  rates  may  vary,  depending  upon  the  third-party  payer,  the  type  of
insurance  plan,  and  other  similar  or  dissimilar  factors.  If  our  products  are  not  subject  to  adequate  reimbursement,  physicians  may  not
prescribe for our products in sufficient amounts to make our products profitable.

Comparative  effectiveness  research  demonstrating  benefits  in  a  competitor’s  product  could  adversely  affect  the  sales  of  our  drug
product candidates. If third-party payers do not consider our products to be cost-effective compared to other available therapies, they may
not cover our products as a benefit under their plans or, if they do, the level of payment may not be sufficient to allow us to sell our products
on a profitable basis.

Adequate third-party reimbursement may not be available to enable us to maintain price levels sufficient to realize an appropriate
return  on  our  investment  in  product  development.  In  addition,  in  the  U.S.  there  is  a  growing  emphasis  on  comparative  effectiveness
research, both by private payers and by government agencies. To the extent other drugs or therapies are found to be more effective than our
products, payers may elect to cover such therapies in lieu of our products and/or reimburse our products at a lower rate.

In  addition,  emphasis  on  managed  care  in  the  U.S.  has  increased  and  we  expect  this  will  continue  to  increase  the  pressure  on
pharmaceutical  pricing.  Coverage  policies  and  third-party  reimbursement  rates  may  change  at  any  time.  Even  if  favorable  coverage  and
reimbursement status is attained for one or more products for which we receive regulatory approval, less favorable coverage policies and
reimbursement rates may be implemented in the future.

Any development along these lines could materially and adversely affect our prospects. We are unable to predict what legislative or
regulatory changes relating to the healthcare industry, including without limitation any changes affecting governmental and/or private or
third party coverage and reimbursement, may be enacted in the future, or what effect such legislative or regulatory changes would have on
our business.

If  we  obtain  FDA  approval  for  any  of  our  product  candidates,  we  will  be  subject  to  various  federal  and  state  fraud  and  abuse  laws;
these  laws  may  impact,  among  other  things,  our  proposed  sales,  marketing  and  education  programs.  Fraud  and  abuse  laws  are
expected to increase in breadth and in detail, which will likely increase our operating costs and the complexity of our programs to insure
compliance with such enhanced laws.

If we obtain FDA approval for any of our product candidates and begin commercializing those products in the U.S., our operations
may be directly, or indirectly through our customers, distributors, or other business partners, subject to various federal and state fraud and
abuse laws, including, without limitation, anti-kickback statutes and false claims statutes which may  increase  our  operating  costs.  These
laws  may  impact,  among  other  things,  our  proposed  sales,  marketing  and  education  programs.  In  addition,  we  may  be  subject  to  data
privacy and security regulation by both the federal government and the states in which we conduct business.

27

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
If our operations are found to be in violation of any of the federal and state laws or any other governmental regulations that apply to us,
we may be subject to criminal actions and significant civil monetary penalties, which would adversely affect our ability to operate our
business and our results of operations.

If  our  operations  are  found  to  be  in  violation  of  any  of  the  federal  and  state  laws  described  above  or  any  other  governmental
regulations  that  apply  to  us,  we  may  be  subject  to  penalties,  including  criminal  and  significant  civil  monetary  penalties,  damages,  fines,
imprisonment, exclusion from participation in government healthcare programs, and the curtailment or restructuring of our operations, any
of  which  could  adversely  affect  our  ability  to  operate  our  business  and  our  results  of  operations.  To  the  extent  that  any  of  our  product
candidates  are  ultimately  sold  in  a  foreign  country,  we  may  be  subject  to  similar  foreign  laws  and  regulations,  which  may  include,  for
instance, applicable post-marketing requirements, including safety surveillance, anti-fraud and abuse laws, and implementation of corporate
compliance programs and reporting of payments or transfers of value to healthcare professionals.

Negotiated prices for our products covered by a Part D prescription drug plan will likely be lower than the prices we might otherwise
obtain.

Government  payment  for  some  of  the  costs  of  prescription  drugs  may  increase  demand  for  our  products  for  which  we  receive
marketing approval, however, any negotiated prices for our products covered by a Part D prescription drug plan will likely be lower than
the prices we might otherwise obtain.

Risks Related to Our Intellectual Property

If we and our third-party licensors do not obtain and preserve protection for our respective intellectual property rights, our competitors
may be able to take advantage of our (and our licensors’) development efforts to develop competing drugs.

Our  commercial  success  will  depend  in  part  on  obtaining  patent  protection  for  any  products  and  other  technologies  we  might
develop,  and  successfully  defending  any  patents  we  obtain  against  third-party  challenges.  We  license  all  intellectual  property  related  to
Validive from Onxeo S.A., a French public company. See “Material Agreements”. The assignment and transfer of the MNPR-201 (GPX-
150) patent portfolio from TacticGem, LLC to us has been completed. We filed and have been granted in the U.S. and various countries
around the world patents for antibodies that target uPAR. We have also been granted in the U.S. and various countries around the world
patents to a specific sequence of amino acids on uPAR, to which our MNPR-101 antibody binds. We are currently prosecuting this patent in
other countries around the world to further protect MNPR-101. The patent process is subject to numerous risks and uncertainties, and there
can be no assurance that we will be successful in obtaining and defending patents. See “Intellectual Property Portfolio”. These risks and
uncertainties include without limitation the following:

● Patents  that  may  be  issued  or  licensed  may  be  challenged,  invalidated,  or  circumvented;  or  may  not  provide  any  competitive

advantage for other reasons.

● Our competitors, many of which have substantially greater resources than us and have made significant investments in competing
technologies, may seek, or may already have obtained, patents that will limit, interfere with, or eliminate our ability to make, use,
and sell our potential products either in the U.S. or in international markets.

● As a matter of public policy regarding worldwide health concerns, there may be significant pressure on the U.S. government and
other international governmental bodies to limit the scope of domestic and international patent protection for cancer treatments
that prove successful.

● Countries  other  than  the  U.S.  may  have  less  restrictive  patent  laws  than  those  upheld  by  the  U.S.  courts;  therefore,  non-U.S.

competitors could exploit these laws to create, develop, and market competing products.

In  addition,  the  USPTO  and  patent  offices  in  other  jurisdictions  have  often  required  that  patent  applications  concerning
pharmaceutical  and/or  biotechnology-related  inventions  be  limited  or  narrowed  substantially  to  cover  only  the  specific  innovations
exemplified  in  the  patent  application,  thereby  limiting  their  scope  of  protection  against  competitive  challenges.  Thus,  even  if  we  or  our
licensors are able to obtain patents, the patents may be substantially narrower than anticipated.

If we permit our patents to lapse or expire, we will not be protected and will have less of a competitive advantage. The value of our
products may be greatly reduced if this occurs. Our patents expire at different times and are subject to the laws of multiple countries. Some
of  our  patents  are  currently  near  expiration  and  we  may  pursue  patent  term  extensions  for  these  where  appropriate.  See  “Intellectual
Property Portfolio”.

In addition to patents, we also rely on trade secrets and proprietary know-how. While we take measures to protect this information by
entering into confidentiality and invention agreements with our consultants and collaborators, we cannot provide any assurances that these
agreements  will  be  fully  enforceable  and  will  not  be  breached,  that  we  will  be  able  to  protect  ourselves  from  the  harmful  effects  of
disclosure  if  they  are  not  fully  enforceable  or  are  breached,  that  any  remedy  for  a  breach  will  adequately  compensate  us,  that  these
agreements will achieve their intended aims, or that our trade secrets will not otherwise become known or be independently discovered by
competitors. If any of these events for which we cannot provide assurances occurs, or we otherwise lose protection for our trade secrets or
proprietary know-how, the value of this information may be greatly reduced.

28

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Intellectual  property  disputes  could  require  us  to  spend  time  and  money  to  address  such  disputes  and  could  limit  our  intellectual
property rights.

The  biopharmaceutical  industry  has  been  characterized  by  extensive  litigation  regarding  patents  and  other  intellectual  property
rights,  and  companies  have  employed  intellectual  property  litigation  to  gain  a  competitive  advantage.  We  may  become  subject  to
infringement claims or litigation arising out of patents and pending applications of our competitors, or additional interference proceedings
declared  by  the  USPTO  to  determine  the  priority  of  inventions.  The  defense  and  prosecution  of  intellectual  property  suits,  USPTO
proceedings,  and  related  legal  and  administrative  proceedings  are  costly  and  time-consuming  to  pursue,  and  their  outcome  is  uncertain.
Litigation may be necessary to enforce our issued patents, to protect our trade secrets and know-how, or to determine the enforceability,
scope, and validity of the proprietary rights of others. An adverse determination in litigation or interference proceedings to which we may
become  a  party  could  subject  us  to  significant  liabilities,  require  us  to  obtain  licenses  from  third  parties,  or  restrict  or  prevent  us  from
selling  our  products  in  certain  markets.  Even  if  a  given  patent  or  intellectual  property  dispute  were  settled  through  licensing  or  similar
arrangements, our costs associated with such arrangements may be substantial and could include the payment by us of large fixed payments
and ongoing royalties. Furthermore, the necessary licenses may not be available on satisfactory terms or at all. In addition, even where we
have  meritorious  claims  or  defenses,  the  costs  of  litigation  may  prevent  us  from  pursuing  these  claims  or  defenses  and/or  may  require
extensive financial and personnel resources to pursue these claims or defenses.

Risks Related to Our Business Operations and Industry

We have a limited operating history as we are a new entity.

As  of  March  1,  2018,  we  have  engaged  exclusively  in  acquiring  pharmaceutical  drug  product  candidates,  licensing  rights  to  drug
product  candidates  and  entering  into  collaboration  agreements,  and  have  not  completed  any  clinical  trials,  received  any  governmental
approvals,  brought  any  product  to  market,  manufactured  or  produced  products  in  commercial  quantities  or  sold  any  pharmaceutical
products.  We  have  limited  experience  in  negotiating,  establishing,  and  maintaining  strategic  relationships,  conducting  clinical  trials,  and
managing the regulatory approval process, all of which will be necessary if we are to be successful. Our lack of experience in these critical
areas makes it difficult for a prospective investor to evaluate our abilities, and increases the risk that we will fail to successfully execute our
strategies.

Furthermore,  if  our  business  grows  rapidly,  our  operational,  managerial,  legal,  and  financial  resources  will  be  strained.  Our
development  will  require  continued  improvement  and  expansion  of  our  management  team  and  our  operational,  managerial,  legal,  and
financial systems and controls.

In  the  normal  course  of  business,  we  have  evaluated  and  expect  to  evaluate  potential  acquisitions  and/or  licenses  of  patents,
compounds,  and  technologies  that  our  management  believes  could  complement  or  expand  our  business.  We  have  limited  history  of
conducting acquisitions, and negotiating and acquiring licenses. In the event that we identify an acquisition or license candidate we find
attractive, there is no assurance that we will be successful in negotiating an agreement to acquire or license, or in financing or profitably
exploiting,  such  patents,  compounds,  or  technologies.  Furthermore,  such  an  acquisition  or  license  could  divert  management  time  and
resources away from other activities that would further our business development.

If we lose key management leadership, and/or scientific personnel, and if we cannot recruit qualified employees, managers, directors,
officers,  or  other  significant  personnel,  we  may  experience  delays  and  increases  in  compensation  costs,  and  our  business  materially
disrupted.

Our future success is highly dependent on the continued service of principal members of our management, leadership, and scientific
personnel, who are able to terminate their employment with us at any time, and may be able to compete with us. The loss of any of our key
management,  leadership,  or  scientific  personnel  including  in  particular,  Chandler  D.  Robinson,  our  President  and  CEO,  and Andrew  P.
Mazar, our Executive Vice President of Research and Development, and Chief Scientific Officer, could materially disrupt our business and
materially  delay  or  prevent  the  successful  commercialization  of  our  product  candidates.  We  have  employment  agreements  with  Dr.
Robinson  and  Dr.  Mazar  which  have  no  term  but  are  for  at-will  employment,  meaning  the  executives  have  the  ability  to  terminate  their
employment at any time.

Our future success will also depend on our continuing ability to identify, hire, and retain highly skilled personnel for all areas of the
organization. Competition in the biopharmaceutical industry for scientifically and technically qualified personnel is intense, and we may be
unsuccessful  in  identifying,  hiring,  and  retaining  qualified  personnel.  Our  continued  ability  to  identify,  hire,  and  retain  highly  skilled
personnel may cause our compensation costs to increase materially.

We are an emerging growth company and we cannot be certain if the reduced disclosure requirements applicable to emerging growth
companies will make our common stock less attractive to investors.

We are an emerging growth company. Under the Jumpstart Our Business Startups Act of 2012 (the “JOBS Act”), emerging growth
companies  can  delay  adopting  new  or  revised  accounting  standards  until  such  time  as  those  standards  apply  to  private  companies.
Therefore, we may not be subject to the same new or revised accounting standards as other public companies that are not “emerging growth
companies.”

29

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
For as long as we continue to be an emerging growth company, we also intend to take advantage of certain other exemptions from
various reporting requirements that are applicable to other public companies including, but not limited to, reduced disclosure obligations
regarding executive compensation in our periodic reports and proxy statements, exemptions from the requirements of holding a nonbinding
advisory  stockholder  vote  on  executive  compensation  and  any  golden  parachute  payments  not  previously  approved,  exemption  from  the
requirement of auditor attestation in the assessment of our internal control over financial reporting and exemption from any requirement
that may be adopted by the Public Company Accounting Oversight Board regarding mandatory audit firm rotation or a supplement to the
auditor’s report providing additional information about the audit and the financial statements (auditor discussion and analysis). If we do
take advantage of these exemptions, the information that we provide stockholders will be different than what is available with respect to
other  public  companies.  We  cannot  predict  if  investors  will  find  our  Common  Stock  less  attractive  because  we  will  rely  on  these
exemptions. If investors find our Common Stock less attractive as a result of our status as an emerging growth company, there may be less
liquidity for our Common Stock and our stock price may be more volatile.

We  will  remain  an  emerging  growth  company  until  the  earliest  of  (i)  the  end  of  the  fiscal  year  in  which  the  market  value  of  our
common stock that is held by non-affiliates exceeds $700 million as of the end of the second fiscal quarter, (ii) the end of the fiscal year in
which  we  have  total  annual  gross  revenues  of  $1  billion  or  more  during  such  fiscal  year,  (iii)  the  date  on  which  we  issue  more  than  $1
billion in non-convertible debt in a three-year period or (iv) the end of the fiscal year following the fifth anniversary of the date of the first
sale of our Common Stock pursuant to an effective registration statement filed under the Act.

Competition and technological change may make our product candidates obsolete or non-competitive.

The biopharmaceutical industry is subject to rapid technological change. We have many potential competitors, including major drug
and chemical companies, specialized biopharmaceutical firms, and universities and other research institutions. These companies, firms, and
other  institutions  may  develop  products  that  are  more  effective  than  our  product  candidates  or  that  would  make  our  product  candidates
obsolete or non-competitive. Many of these companies, firms, and other institutions have greater financial resources than us and may be
better able to withstand and respond to adverse market conditions within the biopharmaceutical industry, including without limitation the
lengthy regulatory approval process for product candidates.

If product liability lawsuits are brought against us, we may incur substantial costs to defend them and address any damages awarded,
and demand for our products could be reduced as a result of such lawsuits.

The testing and marketing of medical products is subject to an inherent risk of product liability claims. Since we currently are not
sponsoring  a  clinical  trial,  we  do  not  have  product  liability  insurance  coverage,  but  plan  to  obtain  appropriate  coverage  when  we  enroll
patients in a Validive or other clinical trial. Regardless of their merit or eventual outcome, product liability claims may result in:

● decreased demand for our products;
● injury to our reputation and significant, adverse media attention;
● withdrawal of clinical trial volunteers; and
● potentially  significant  litigation  costs,  including  without  limitation  any  damages  awarded  to  the  plaintiffs  if  we  lose  or  settle

claims.

We use hazardous materials, including radioactive materials, in our business, and any claims relating to improper handling, storage, or
disposal of these materials could materially harm our business.

Our business involves the use of a broad range of hazardous chemicals and materials, including radioactive materials. Environmental
laws impose stringent civil and criminal penalties for improper handling, disposal, and storage of these materials. In addition, in the event
of an improper or unauthorized release of, or exposure of individuals to, hazardous materials, we could be subject to civil damages due to
personal injury or property damage caused by the release or exposure. A failure to comply with environmental laws could result in fines
and the revocation of environmental permits, which could prevent us from conducting our business.

We have limited the liability of and indemnified our directors and officers.

Although our directors and officers are accountable to us and must exercise good faith, good business judgement, and integrity in
handling our affairs, our Second Amended and Restated Certificate of Incorporation (the “Certificate of Incorporation”), provides that our
directors will be indemnified to the fullest extent permitted under Delaware law. As a result, our stockholders may have fewer rights against
our  directors  than  they  would  have  absent  such  provisions  in  our  Certificate  of  Incorporation,  and  a  stockholder’s  ability  to  seek  and
recover damages for a breach of fiduciary duties may be reduced or restricted. Delaware law allows indemnification if our Board Member
(a) has acted in good faith, in a manner the Board Member reasonably believes to be in or not opposed to our best interests, and (b) with
respect to any criminal action or proceeding, if the Board Member had no reasonable cause to believe the conduct was unlawful.

30

 
 
 
 
 
 
 
 
 
 
 
 
 
 
Pursuant to the Certificate of Incorporation, each director and (to the extent approved by our Board) each of our officers who is made
a party to a legal proceeding because he or she is or was a Board Member or officer, is indemnified by us from and against any and all
liability, except that we may not indemnify a Board Member or officer: (a) for any liability incurred in a proceeding in which such person is
adjudged  liable  to  Monopar  or  is  subjected  to  injunctive  relief  in  favor  of  Monopar;  (b)  for  acts  or  omissions  that  involve  intentional
misconduct or a knowing violation of law, fraud or gross negligence; (c) for unlawful distributions; (d) for any transaction for which such
Board Member or officer received a personal benefit or as otherwise prohibited by or as may be disallowed under Delaware law; or (e) with
respect to any dispute or proceeding between us and such Board Member or officer unless such indemnification has been approved by a
disinterested  majority  of  Board  Members  or  by  a  majority  in  interest  of  disinterested  stockholders.  We  are  required  to  pay  or  reimburse
attorney’s fees and expenses of a Board Member seeking indemnification as they are incurred, provided the director executes an agreement
to repay the amount to be paid or reimbursed if there is a final determination by a court of competent jurisdiction that such person is not
entitled to indemnification.

Future legislation or executive or private sector actions may increase the difficulty and cost for us to commercialize our products and
affect the prices obtained for such products.

There have been several attempts made to repeal the Patient Protection and Affordable Care Act (the “PPACA”), and modification
and  partial  or  complete  repeal  of  the Affordable  Care Act  in  the  future  is  possible.  On  December  22,  2017,  the  Tax  Cuts  and  Jobs Act
became  law  –  one  of  its  provisions  repealed  what  is  known  as  the  individual  mandate  under  PPACA  which  could  have  the  effect  of
negating such law. Healthcare reform measures that may be adopted in the future may result in more rigorous coverage criteria and lower
reimbursement, and in additional downward pressure on the price that may be charged for any of our product candidates, if approved.

The  increasing  cost  of  healthcare  as  a  percentage  of  GDP  and  the  increasing  deferred  liabilities  behind  most  governmental  health
care programs (such as Medicare and Medicaid) continue to be an economic challenge which affects the overall economic health of the U.S.
High cost products and therapies that are early in their life cycle, are attractive targets for parties that believe that the cost of healthcare
must  be  better  controlled  and  reduced.  Pharmaceutical  prices  and  healthcare  reform  has  been  debated  and  acted  upon  by  legislators  for
many years. Future legislation or executive or private sector actions related to healthcare reform could materially and adversely affect our
business by reducing our ability to generate revenue at prices sufficient to reward for the risks and costs of development, to raise capital,
and to market our products.

Additionally, Executive Orders and policy statements issued by President Trump have increased the uncertainty regarding the timing
for  the  FDA’s  interpretation  and  implementation  of  requirements  under  the  Federal  Food,  Drug  and  Cosmetic Act  (“FDCA”).  Some  of
these  executive  actions  may  also  negatively  affect  the  FDA’s  exercise  of  regulatory  oversight  and  ability  to  timely  review  industry
submissions and applications in connection with the drug development and approval process. Notably, on April 12, 2017, the Director for
the Office of Management and Budget (“OMB”) implemented a long-term plan to reduce the size of the federal workforce. Although the
FDA is funded in the near-term, in the future, an under-staffed FDA could result in increasing delays in the FDA’s responsiveness or in its
ability to review applications, issue regulations or guidance, or implement or enforce regulatory requirements in a timely fashion or at all. A
January 30, 2017 Executive Order also included a budget neutrality provision that requires the total incremental cost of all new regulations
in the 2017 fiscal year, including repealed regulations, to be no greater than zero, except in limited circumstances. It is difficult to predict
how  these  requirements  will  be  interpreted  and  implemented,  and  the  extent  to  which  they  will  impact  the  FDA’s  ability  to  continue
engaging in its regulatory authorities under the FDCA. If executive or legislative actions impose restrictions on the FDA’s ability to engage
in oversight and implementation activities in the normal course, our business may be negatively impacted. On August 18, 2017, the FDA
Reauthorization Act  of  2017  was  signed  which,  among  other  things,  established  user  fees  for  human  drug  applications  which  are  to  be
directed toward expediting the drug development process. On December 12, 2017, an amendment to the FDCA was passed to authorize
additional emergency uses for medical products during a military emergency. Both of these actions restore increased funding for the FDA.
The user fees for human drug applications can result in funding which is variable depending on the work load created by applications that
is supported by the user fees. There is no assurance that federal or state health care reform will not adversely affect our future business and
financial  results,  and  we  cannot  predict  how  future  federal  or  state  legislative,  judicial  or  administrative  changes  relating  to  healthcare
reform and third party payers will affect the pharmaceutical industry in general and our business in particular.

Future tax reform measures may negatively impact our financial position.

Our business may be negatively impacted by tax reform measures. If tax reform measures are passed, there can be no assurance that
we will continue to receive favorable tax treatment related to our patents. For example, on December 22, 2017, the Tax Cuts and Jobs Act
of 2017 was signed into law that significantly revises the Internal Revenue Code of 1986, as amended. The newly enacted federal income
tax  law,  among  other  things,  contains  significant  changes  to  corporate  taxation,  including  reduction  of  the  corporate  tax  rate  from  a  top
marginal  rate  of  35%  to  a  flat  rate  of  21%,  limitation  of  the  tax  deduction  for  interest  expense  to  30%  of  adjusted  earnings  (except  for
certain small businesses), limitation of the deduction for net operating losses to 80% of current year taxable income and elimination of net
operating  loss  carrybacks,  treatment  of  proceeds  from  the  sale  of  “self-created”  patents  as  ordinary  income,  and  modifying  or  repealing
many business deductions and credits (including reducing the business tax credit for certain clinical testing expenses incurred in the testing
of orphan drugs from 50% to 25%). Notwithstanding the reduction in the corporate income tax rate, the overall impact of the new federal
tax law is uncertain and our business and financial condition could be adversely affected. In addition, it is uncertain if and to what extent
various states will conform to the newly enacted federal tax law. The impact of this tax reform on holders of our common stock is also
uncertain.  We  urge  our  stockholders  to  consult  with  their  legal  and  tax  advisors  with  respect  to  this  legislation  and  the  potential  tax
consequences  of  investing  in  or  holding  our  common  stock.  It  is  difficult  to  predict  what  future  tax  reform  measures,  if  any,  could  be
implemented and the extent to which they will impact our accounting practices and our business.

31

 
 
 
 
 
 
 
 
 
 
Our  anticipated  operating  expenses  over  the  next  year  are  based  upon  our  management’s  estimates  of  possible  future  events.  Actual
amounts could differ materially from those estimated by our management.

Development of pharmaceuticals and cancer drugs is extremely risky and unpredictable. We have estimated operating expenses and
capital expenditures over the next year based on certain assumptions. Any change in the assumptions could and will cause the actual results
to  vary  substantially  from  the  anticipated  expenditures,  and  could  result  in  material  differences  in  actual  versus  forecasted  expenses  or
expenditures. Furthermore, all of the factors are subject to the effect of unforeseeable future events. The estimates of capital expenditures
and operating expenses represent forward-looking statements within the meaning of the federal securities laws. Prospective investors are
cautioned that any such forward-looking statements are not guarantees of future performance and involve risks and uncertainties. Actual
events or results may differ materially from those discussed in the forward-looking statements as a result of various factors, including the
risk  factors  set  forth  under  "Risk  Factors"  in  this  Form  10-K.  In  view  of  the  foregoing,  investors  should  not  rely  on  these  estimates  in
making a decision to invest in us.

Risks Associated with Our Capital Stock

We may never provide liquidity to our investors.

No public market exists with respect to any of our securities. There is no assurance that any public offering, merger, combination,
sale, or other liquidity event relating to us will ever take place, or that any public offering, merger, combination, sale, or other event that
might take place would provide liquidity for our investors or that we will be able to provide liquidity to our investors in any fashion. In the
event that we are unable to affect a public offering, merger, combination, sale, or other liquidity event, our investors would likely be unable
to sell their interests in us.

Existing  and  new  investors  will  experience  dilution  as  a  result  of  future  sales  or  issuances  of  our  common  stock  and  future  option
exercises under our stock option plan.

Our Board Members, employees, and certain of our consultants have been and will be issued equity and/or granted options that vest
with the passage of time. Up to a total of 1,600,000 shares of our Common Stock may be issued as stock options or restricted stock under
the Amended  and  Restated  Monopar  Therapeutics  Inc.  2016  Stock  Incentive  Plan,  and  stock  options  for  the  purchase  of  up  to  690,596
shares of our common stock have already been granted. See Item 11 - “Stock Option Plan.” The issuance of such equity and/or the exercise
of such options will dilute both our existing and our new investors. As of March 1, 2018, no stock options have been exercised.

Our  existing  and  our  new  investors  will  likely  also  experience  substantial  dilution  resulting  from  the  issuance  by  us  of  equity
securities  in  connection  with  certain  transactions,  including  without  limitation,  future  offering  of  shares,  intellectual  property  licensing,
acquisition, or commercialization arrangements.

Holders of the shares of our Common Stock will have no control of our operations or of decisions on major transactions.

Our business and affairs are managed by or under the direction of our Board. Our Stockholders are entitled to vote only on actions
that require a Stockholder vote under federal or state law. Stockholder approval requires the consent and approval of holders of a majority
or more of our outstanding stock. Shares of stock do not have cumulative voting rights and therefore, holders of a majority of the shares of
our outstanding stock will be able to elect all Board Members. TacticGem, LLC owns 7,166,667 shares of common stock (77.1%). The
limited liability company agreement of TacticGem, LLC provides that the manager will vote its shares of Monopar to elect to the Board of
Directors those persons nominated by TacticPharma LLC plus one person nominated by Gem Pharmaceuticals, LLC. Additionally, other
than  in  the  elections  of  directors  the  limited  liability  company  agreement  requires  TacticGem  to  pass  through  votes  to  its  members  in
proportion  to  their  membership  percentages  in  TacticGem. As  a  result,  Tactic  Pharma,  our  initial  investor,  holds  an  approximately  46%
beneficial  interest  in  us  and  together  with  Gem’s  beneficial  ownership  of  approximately  33%,  the  two  entities  control  a  majority  of  our
stock and will be able to elect all Board Members and control our affairs. Some of our Board Members and executive officers own and
control  Tactic  Pharma. Although  no  single  person  has  a  controlling  interest  in  Tactic  Pharma,  acting  together,  they  are  able  to  control
Tactic Pharma and a large voting block of Monopar and elect over a majority of our Board of Directors. See Item 12 - “Security Ownership
of Certain Beneficial Owners and Management.”

Our  ability  to  list  on  Nasdaq  in  the  future  will  require  raising  significant  additional  capital  and  likely  require  a  public  stock
transaction; failure to qualify to trade on Nasdaq will make it more difficult to raise capital.

We will need to raise significant funds in the next 24 months to execute our clinical development plans and we believe that if our
stock  is  trading  on  Nasdaq’s  Capital  Market  it  will  enable  better  access  to  capital.  Nasdaq  has  listing  requirements  for  inclusion  of
securities  for  trading  on  the  Nasdaq  Capital  Market,  including  stockholders  equity  of  $4  million  (market  value  standard)  or  $5  million
(equity standard), market value of publicly held shares of $15 million, an operating history of 2 years under the equity standard or a market
value  of  listed  securities  of  $50  million  under  the  market  value  standard,  1  million  publicly  held  shares,  300  shareholders,  three  market
makers and a $4 bid price or a closing price of $3 (equity standard) or $2 (market value standard). If we are unable to list on Nasdaq, it
could make it harder for us to raise capital in both the immediate time frame and in the long-term. If we are unable to raise capital when
needed in the future, we may have to cease or reduce operations.

32

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Item 2. Properties

We lease approximately 1,202 square feet of space in the Village of Wilmette, Illinois for our corporate offices, under a lease which
runs through the end of 2019. We lease approximately 160 square feet for our Seattle, Washington office. We believe that we will require
additional office space within the next 12 months as we begin to hire additional personnel.

Item 3. Legal

We are not party to any material legal proceedings.

PART II

Item 5. Market for Registrant’s Common Equity, Related Stockholder Matters and Issuer Purchases of Equity Securities

Market Information

There is no established public trading market in our common stock. Our securities are not listed for trading on any national securities

exchange nor are bid or asked quotations reported in any over-the-counter quotation service.

Rule 144 Eligibility

As of March 1, 2018, 1,335,079.3 shares of our common stock are eligible for sale under Rule 144.

We cannot estimate the number of shares of our common stock that our existing stockholders will elect to sell under Rule 144.

Holders

As of March 1, 2018, there were 9,291,420.614 shares of our common stock outstanding held by 43 holders. In addition, there were

nine holders of stock options to purchase up to 690,596 shares of our common stock.

Dividends

We have never paid cash dividends on any of our capital stock and we currently intend to retain our future earnings, if any, to fund
the development and growth of our business. We do not intend to pay cash dividends to holders of our common stock in the foreseeable
future.

Securities Authorized for Issuance Under Equity Compensation Plans

The following table provides information as of December 31, 2017, with respect to shares of our common stock that may be issued

under existing equity compensation plans. There are no equity compensation plans that have not been approved by our security holders.

33

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Number of
Securities to
be Issued
Upon Exercise
of
Outstanding
Options,
Warrants and
Rights

Weighted
Average
Exercise Price
of
Outstanding
Options,
Warrants and
Rights

658,592 

  $

0.94 

Number of
Securities
Remaining
Available For
Future
Issuance
under Equity
Compensation
Plans
941,408 

Plan Category
Equity compensation plans approved by security holders (1)

(1) The Monopar Therapeutics Inc. 2016 Stock Incentive Plan.

Registration Rights

We  are  subject  to  an  agreement  with  TacticGem  (pursuant  to  the  Gem  Transaction  as  discussed  later  in  this  document),  which
obligates  us  to  file  Form  S-3  or  other  appropriate  form  of  registration  statement  covering  the  resale  of  any  of  our  Common  Stock  by
TacticGem, Gem, or Tactic, upon direction by TacticGem at any time after we have been subject to the reporting requirements of the 1934
Act for at least twelve months (the “Initial Holding Period’). We are required to use our best efforts to have such registration statement
declared effective as soon as practical after it is filed. In the event that such registration statement for resale is not approved by the SEC,
and  TacticGem  submits  a  written  request,  we  are  required  to  prepare  and  file  a  registration  statement  on  Form  S-1  registering  such
Common Stock for resale and to use our best efforts to have such registration statement declared effective as soon as practical thereafter.
After registration, pursuant to these rights, these shares will become freely tradable without restriction under the Securities Act other than
pursuant to restrictions on affiliates under Rule 144.

Recent Sales of Unregistered Securities.

Set forth below is information regarding shares of common stock issued and options granted by us in the year ended December 31,
2017,  that  were  not  registered  under  the  Securities Act. Also  included  is  the  consideration,  if  any,  received  by  us,  for  such  shares  and
options  and  information  relating  to  the  Securities Act,  or  rule  of  the  SEC,  under  which  exemption  from  registration  was  claimed.  No
underwriters  were  involved  in  the  foregoing  issuances  of  securities.  Below  this  description  of  recent  sales  of  unregistered  securities  is  a
description of the exemptions from registration which were applicable to each sale or grant.

(a)  On  February  20,  2017,  we  granted  stock  options  for  1,200  shares  of  our  Common  Stock  to  each  of  Dr.  Christopher  M.  Starr,  Dr.
Chandler  D.  Robinson,  and  Dr. Andrew  P.  Mazar  in  exchange  for  services.  Pursuant  to  the  “Conversion”  in  March  2017,  these  stock
options were each adjusted to be for 84,000 shares. On the same date, we granted a stock option for 336 shares of our Common Stock to
Kim R. Tsuchimoto in exchange for services, which was adjusted to be for 23,520 shares pursuant to the Conversion. The exercise price of
each of these options was $0.001 per share and the options expire on February 19, 2027.

(b) During March 2017 through June 2017, 340,840.33 shares of Common Stock were sold to accredited investors at a price of $6.00 per
share.

(c) During August 2017 through September 2017, 448,834 shares of Common Stock were sold to accredited investors at a price of $6.00 per
share.

(d) On September 1, 2017, we granted options for 21,024 shares of Common Stock to Arthur Klausner, and on September 18, 2017, we
granted options for 21,024 shares of Common Stock to each of Michael J. Brown and Raymond W. Anderson, in exchange for services as
Directors.  The  exercise  price  of  the  options  was  $6.00  per  share  and  the  options  expire  on August  31,  2027  and  September  17,  2027,
respectively.

(e) On August 25, 2017, 3,055,394.12 shares of our Common Stock were issued to TacticGem in exchange for the Gem Contributed Assets
(including assets and $5 million in cash) as part of the Gem Transaction.

(f)  On  November  1,  2017,  we  granted  options  for  40,000  shares  of  Common  Stock  to  Kirsten Anderson  in  exchange  for  services.  The
exercise price of the options was $6.00 per share and the options expire on October 31, 2027.

(g) On January 1, 2018, we granted options for 32,004 shares of Common Stock to Patrice Rioux in exchange for services. The exercise
price of the option was $6.00 per share and the options expire on December 31, 2027.

34

 
 
 
 
 
 
 
 
   
   
 
 
 
 
 
 
 
 
 
 
 
 
 
 
The  offers,  sales  and  issuances  of  the  securities  described  in  paragraphs  (a),  (d),  (f),  and  (g)  were  deemed  to  be  exempt  from
registration  under  the  Securities Act  in  reliance  on  both  Section  4(a)(2)  of  the Act  and  Rule  701  in  that  the  transactions  were  under
compensatory benefit plans and contracts relating to compensation as provided under Rule 701. The recipients of such securities were our
employees, officers, bona fide consultants and advisors and received the securities under our Plan. Appropriate legends were affixed to the
securities issued in these transactions. Each of the recipients of securities in these transactions had adequate access, through employment,
business or other relationships, to information about us and had knowledge and experience to make the decision to accept the stock options.

The offers, sales and issuances of the securities described in paragraph (b), (c), and (e) were deemed to be exempt from registration
under the Securities Act in reliance on Rule 506(b) of Regulation D in that the issuance of securities to the accredited  investors  did  not
involve a public offering. The recipients of securities in each of these transactions acquired the securities for investment only and not with a
view to or for sale in connection with any distribution thereof. Each of the recipients of securities in these transactions was an accredited
investor under Rule 501 of Regulation D. Form D was filed related to the offer described in paragraph (b) on March 28, 2017; and Form D
was filed related to the offer described in paragraph (c) on August 23, 2017.

Item 7. Management's Discussion and Analysis of Financial Condition and Results of Operations.

You should read the following discussion and analysis of our financial condition and results of operations together with our financial
statements  and  related  notes  appearing  at  the  end  of  this  Annual  Report  on  Form  10-K.  Some  of  the  information  contained  in  this
discussion and analysis or set forth elsewhere in this Annual Report on Form 10-K, including information with respect to our plans and
strategy for our business and related financing, includes forward-looking statements that involve risks and uncertainties. You should read
the  "Risk  Factors"  section  of  this Annual  Report  on  Form  10-K,  Item  1A,  for  a  discussion  of  important  factors  that  could  cause  actual
results to differ materially from the results described in or implied by the forward-looking statements contained in the following discussion
and analysis.

Overview

Our mission is to develop innovative drugs and drug combinations to improve clinical outcomes for cancer patients. We are building
a drug development pipeline through the licensing or acquisition of oncology therapeutics at the late preclinical through advanced clinical
development stage.

Validive is being developed for the treatment of radiation-induced SOM. SOM is a frequent major adverse side effect for patients
with head and neck cancer who are treated by radiation treatment. SOM causes intense oral pain and limits a patient’s ability to eat and
drink, which causes additional treatment complications. Many affected patients require hospitalization and the SOM symptoms can force
patients  to  stop  cancer  treatments  early,  which  reduces  the  success  of  treatments.  Validive  is  designed  to  deliver  the  active  ingredient,
clonidine,  to  the  at-risk  oropharyngeal  mucosa.  Clonidine  reduces  the  production  of  cytokines,  the  molecules  that  cause  ulcerations  and
pain  in  patients  that  develop  SOM.  Preclinical  studies  and  a  Phase  2  clinical  trial  have  demonstrated  that  Validive  has  the  potential  for
reducing the frequency of developing SOM in addition to improving its symptoms, as compared to a placebo. On September 8, 2017, we
exercised our exclusive option to license in order to advance the development of Validive with the near-term goal of commencing a Phase 3
development program. If successful, this Phase 3 program may allow us to apply for marketing approval. See “Material Agreements” and
“Strategy.”

In August  2017,  we  acquired  MNPR-201  (GPX-150;  5-imino-13-deoxydoxorubicin),  a  proprietary  analog  of  doxorubicin  that  is
selective for  topoisomerase-II-alpha  from  TacticGem.  MNPR-201  has  been  engineered  specifically  to  retain  the  anticancer  activity  of
doxorubicin while minimizing toxic effects on the heart.

MNPR-101 is a drug product candidate designed to reduce tumor growth by targeting a specific receptor, uPAR, which is present in
a  range  of  tumor  types,  including  pancreatic  and  ovarian  tumors.  uPAR  is  part  of  the  normal  cell  repair  process  in  non-cancerous  cells;
however, in cancerous cells the tumor hijacks uPAR to help the tumor grow and spread. Preclinical models have shown that MNPR-101 is
effective at reducing tumor growth, both used alone and in combination with existing therapies. In May 2015, we entered into a Clinical
Trial  and  Option Agreement  with  Cancer  Research  UK  with  respect  to  our  drug  product  candidate  MNPR-101  (formerly  huATN-658).
Pursuant to this agreement Cancer Research UK conducted preclinical work, improved the manufacturing, and planned to conduct a Phase
1a/1b clinical trial in cancer patients. As part of a portfolio reprioritization review, on March 21, 2018 Cancer Research UK notified us it
was closing its project related to MNPR-101 and would work to make arrangements to formally terminate the agreement.  We are currently
reviewing  potential  alternative  collaboration  opportunities  for  MNPR-101  and  continue  to  maintain  the  program’s  intellectual  property
portfolio.

35

 
 
 
 
 
 
 
 
 
 
 
 
Over  the  next  three  years,  we  plan  to  execute  a  Phase  3  clinical  trial  for  Validive,  continue  clinical  development  of  MNPR-201,
pursue  collaboration  opportunities  for  MNPR-101  for  initial  clinical  development,  raise  additional  capital  to  fund  our  drug  development
programs, acquire or in-license additional drug product candidates and promote public and biotech investor awareness of us.

Developing a new drug and conducting clinical trials for one or more disease indications involves substantial costs and resources.
Our operating and financial strategy for the development, clinical testing, manufacture and commercialization of drug product candidates is
heavily dependent on our entering into collaborations with corporations, non-profits, scientific institutions, licensors, licensees and other
parties,  which  enables  us  to  utilize  their  financial  and  other  resources  to  assist  in  drug  development. Additionally,  we  will  need  to  raise
significant funds in the next 12–24 months to execute our clinical development of Validive and potential approval and commercialization
plans. We believe that we will have better access to capital as a public reporting company and if a trading market develops for our stock.
This  would  increase  corporate  visibility,  provide  increased  liquidity  for  our  stockholders,  and  create  a  market  value  for  our  pipeline  of
oncology drug product candidates. Therefore, we became a public reporting company under the Securities Exchange Act of 1934 (the “34
Act”) through the filing of a Form 10 registration statement with the SEC. We are working with investment bankers and market makers,
with the intention of listing on Nasdaq as soon as we are able to meet the shareholder number, capitalization and other requirements for
such a listing, which will likely require a public offering of our stock or other public stock transaction. See “Risk Factors – Our ability to
list on Nasdaq in the future will require raising significant additional capital and likely require a public stock transaction; failure to qualify
to trade on Nasdaq will make it more difficult to raise capital.” There can be no assurance that we will be successful in including our stock
for trading on Nasdaq or that a market will develop for our stock. See Item 1A - “Risk Factors – Risks Related to Our Financial Condition
and Capital Requirements”, and “Risks Related to Our Business Operations and Industry.”

Revenues

We are an emerging growth company, have no approved drugs and have not generated any revenues.

Conversion of Preferred Stock to Common Stock

In March 2017, holders of a majority in interest of our Series A Preferred Stock and holders of a majority in interest of our Series Z
Preferred  Stock  voted  to  adopt  the  Second  Amended  and  Restated  Certificate  of  Incorporation  of  the  Company  (the  “Certificate  of
Incorporation”). When the Certificate of Incorporation took effect, each share of Series A Preferred Stock was automatically converted into
84 shares of common stock of the Company (a 1.2 for 1 conversion to Common Stock concurrent with a 70 for 1 stock split) and each share
of Series Z Preferred Stock was automatically converted into 70 shares of common stock of the Company (a 1 for 1 conversion to common
stock concurrent with a 70 for 1 stock split) and Series A Preferred Stock and Series Z Preferred Stock were eliminated (the “Conversion”).
100,000 shares of Series Z Preferred Stock were converted into 7,000,000 shares of common stock and 15,894 shares of Series A Preferred
Stock  were  converted  into  1,335,079.284  shares  of  common  stock. All  references  in  this  “Management’s  Discussion  and Analysis  of
Financial Conditions and Results of Operations” to common stock authorized, issued and outstanding and common stock options take into
account the stock split that occurred as part of the Conversion.

Critical Accounting Policies and Use of Estimates

While our significant accounting policies are described in more detail in Note 2 of our financial statements included elsewhere in this
Annual  Report  on  Form  10-K,  we  believe  the  following  accounting  policies  to  be  critical  to  the  judgments  and  estimates  used  in  the
preparation of our financial statements.

Use of Estimates

The preparation of financial statements in conformity with GAAP requires our management to make estimates and assumptions that
affect the reported amounts of assets and liabilities, disclosure of contingent assets and liabilities, and reported amounts of revenues and
expenses in the financial statements and accompanying notes. Actual results could differ from those estimates.

Going Concern Assessment

We adopted Accounting Standards Updates (“ASU”) 2014-15, Disclosure of Uncertainties about an Entity’s Ability to Continue as a
Going  Concern,  which  the  Financial Accounting  Standards  Board  (“FASB”)  issued  to  provide  guidance  on  determining  when  and  how
reporting  companies  must  disclose  going-concern  uncertainties  in  their  financial  statements.  The ASU  requires  management  to  perform
interim and annual assessments of an entity’s ability to continue as a going concern within one year of the date of issuance of the entity’s
financial  statements  (or  within  one  year  after  the  date  on  which  the  financial  statements  are  available  to  be  issued,  when  applicable).
Further, a company must provide certain disclosures if there is “substantial doubt about the entity’s ability to continue as a going concern.”
In  February  2018,  we  analyzed  our  minimum  cash  requirements  through  March  2019  and  have  determined  that,  based  upon  our  current
available  cash,  we  have  no  substantial  doubt  about  our  ability  to  continue  as  a  going  concern.  See  Item  1A  -  “Risk  Factors”  –  our
anticipated operating expenses over the next year are based upon our management’s estimates of possible future events. Actual operating
expenses could differ materially from those projected by our management.

36

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Revenue

We are an emerging growth company, have no approved drugs and have not generated any revenues. See “Overview – Revenues”.
To date, we have engaged in acquiring pharmaceutical drug product candidates, licensing rights to drug product candidates, entering into
collaboration agreements for testing and clinical development of our drug product candidates and providing the infrastructure to support the
clinical development of drug product candidates. We do not anticipate revenues from operations until we complete testing and development
of one of our drug product candidates and obtain marketing approval or we sell or out-license one of our drug product candidates to another
party. See “Liquidity and Capital Resources”.

Research and Development Expenses

Research  and  development  (“R&D”)  costs  are  expensed  as  incurred.  Major  components  of  research  and  development  expenses
include salaries and benefits of R&D staff, fees paid to consultants and to the entities that conduct certain development activities on our
behalf and materials and supplies.

We  accrue  and  expense  the  costs  for  clinical  trial  activities  performed  by  third  parties  based  upon  estimates  of  the  percentage  of
work completed over the life of the individual study in accordance with agreements established with contract research organizations and
clinical  trial  sites.  We  determine  the  estimates  through  discussions  with  internal  clinical  personnel  and  external  service  providers  as  to
progress or stage of completion of trials or services and the agreed upon fee to be paid for such services. Costs of setting up clinical trial
sites for participation in the trials are expensed immediately as research and development expenses. Clinical trial site costs related to patient
enrollment are accrued as patients are entered into the trial. During the previous two fiscal years, we had no clinical trials in progress.

The successful development of our product pipeline is highly uncertain. We cannot reasonably estimate the nature, timing or costs of
the efforts that will be necessary to complete the remainder of the development of any of our drug product candidates or the period, if any,
in which material net cash inflows from our drug product candidates may commence. This is due to the numerous risks and uncertainties
associated with developing drug product candidates, including:

● receiving less funding than we require;
● slower than expected progress in developing Validive, MNPR-201, MNPR-101 or other drug product candidates;
● higher than expected costs to produce our current and future drug product candidates;
● higher than expected costs for preclinical testing of our future and current acquired and/or in-licensed programs;
● future clinical trial costs, including an increase in the number, size, duration, or complexity of future clinical trials;
● future clinical trial results;
● higher than expected costs associated with attempting to obtain regulatory approvals, including without limitation additional costs

caused by delays;

● higher  than  expected  personnel  or  other  costs,  such  as  adding  personnel  or  pursuing  the  acquisition  or  licensing  of  additional

assets;

● higher than expected costs to protect our intellectual property portfolio or otherwise pursue our intellectual property strategy;
● the potential benefits of our product candidates over other therapies; and
● our ability to market, commercialize and achieve market acceptance for any of our product candidates that we are developing or

may develop in the future.

There are other risks described in Item 1A - “Risk Factors”. A change in the outcome of any of these variables with respect to the
development of a drug product candidate could mean a significant change in the costs and timing associated with the development of that
drug  product  candidate.  We  expect  that  research  and  development  expenses  will  increase  in  future  periods  as  a  result  of  increased
personnel, increased consulting, future preclinical and clinical trial costs, including clinical drug product manufacturing and related costs.

37

 
 
 
 
 
 
 
 
 
 
 
In-process Research and Development

In-process  research  and  development  (“IPR&D”)  expense  represents  the  costs  to  acquire  technologies  to  be  used  in  research  and
development  that  have  not  reached  technological  feasibility,  have  no  alternative  future  uses,  and  are  thus  expensed  as  incurred.  IPR&D
expense also includes upfront license fees and milestones paid to collaborators, with no alternative use, which are expensed as goods are
received or services rendered.

General and Administrative Expenses

General  and  administrative  expenses  consist  primarily  of  compensation  and  expenses  for  our  executive  personnel,  stock-based
compensation  expense  related  to  stock  options  issued  to  our  executive  team,  legal  and  audit  expenses,  general  and  administrative
consulting, board fees and expenses, patent legal and application fees, and facilities and related expenses. Future general and administrative
expenses may also include: compensation and expenses related to the employment of finance, human resources and business development
personnel,  depreciation  and  amortization  of  general  and  administrative  fixed  assets,  investor  relations  and  annual  meeting  expense,  and
stock-based compensation expense related to general and administrative personnel. We expect that our general and administrative expenses
will  increase  in  future  periods  as  a  result  of  increased  personnel,  expanded  infrastructure,  increased  consulting,  legal,  accounting  and
investor relations expenses associated with being a public company and costs incurred to seek and establish collaborations with respect to
any of our drug product candidates.

Collaborative Arrangements

We  and  our  collaborative  partners  are  active  participants  in  a  collaborative  arrangement  and  all  parties  are  exposed  to  significant
risks and rewards depending on the development and commercial success of the activities. Contractual payments to the other parties in the
collaboration agreement and costs incurred by us when we are deemed to be the principal participant for a given transaction are recognized
on a gross basis in research and development expenses. Royalties and license payments are recorded as earned.

In May 2015, we entered into a Clinical Trial and Option Agreement with Cancer Research UK with respect to our drug product
candidate MNPR-101 (formerly huATN-658). Pursuant to this agreement Cancer Research UK conducted preclinical work, improved the
manufacturing, and planned to conduct a Phase 1a/1b clinical trial in cancer patients. Under this agreement, Cancer Research UK was to
cover all costs through Phase 1a/1b clinical studies, including manufacturing. As part of a portfolio reprioritization review, on March 21,
2018 Cancer Research UK notified us it was closing its project related to MNPR-101 and would work to make arrangements to formally
terminate  the  agreement.    We  are  currently  reviewing  potential  alternative  collaboration  opportunities  for  MNPR-101  and  continue  to
maintain the program’s intellectual property portfolio.

In  addition,  we  have  a  non-exclusive  license  with  XOMA  Ltd.  for  its  humanization  technology  and  know-how  utilized  in  the
development of MNPR-101. Under the terms of the license, we are required to pay developmental and sales milestones which could reach
up  to  $14.925  million  if  we  achieve  all  milestones.  The  agreement  does  not  require  the  payment  of  sales  royalties.  There  can  be  no
assurance that we will reach any milestones.

From inception in December 2014 through March 1, 2018, no milestones were met and no royalties were earned, therefore, we did

not pay or accrue/expense any milestone or royalty payments under the CTOA and XOMA Ltd. license agreement.

License Option Agreement

In June 2016, we executed an agreement with Onxeo S.A., a French public company, which gave us the option to license Validive
(clonidine  mucobuccal  tablet),  a  mucoadhesive  tablet  of  clonidine  based  on  the  Lauriad  mucoadhesive  technology  to  potentially  treat
severe oral mucositis in patients undergoing treatment for head and neck cancers. The pre-negotiated license terms included as part of the
option agreement included clinical, regulatory, developmental and sales milestones that could reach up to $108 million if we achieve all
milestones, and escalating royalties on net sales from 5 - 10%. On September 8, 2017, we exercised the option to license Validive in order
to commence the clinical development of the drug product candidate in exchange for a one-time option fee payment of $1 million.

Under the agreement, we are required to pay royalties to Onxeo on a product-by-product and country-by-country basis until the later
of (1) the date when a given product is no longer within the scope of a patent claim in the country of sale or manufacture, (2) the expiry of
any  extended  exclusivity  period  in  the  relevant  country  (such  as  orphan  drug  exclusivity,  pediatric  exclusivity,  new  chemical  entity
exclusivity, or other exclusivity granted beyond the expiry of the relevant patent), or (3) a specific time period after the first commercial
sale of the product in such country. In most countries, including the U.S., the patent term is generally 20 years from the earliest claimed
filing  date  of  a  non-provisional  patent  application  in  the  applicable  country,  not  taking  into  consideration  any  potential  patent  term
adjustment that may be filed in the future or any regulatory extensions that may be obtained. The royalty termination provision pursuant to
(3) described above is shorter than 20 years and is the least likely cause of termination of royalty payments.

38

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
The  Onxeo  license  agreement  does  not  have  a  pre-determined  term,  but  expires  on  a  product-by-product  and  country-by-country
basis;  that  is,  the  agreement  expires  with  respect  to  a  given  product  in  a  given  country  whenever  our  royalty  payment  obligations  with
respect to such product have expired. The agreement may also be terminated early for cause if either we or Onxeo materially breach the
agreement,  or  if  either  we  or  Onxeo  become  insolvent.  We  may  also  choose  to  terminate  the  agreement,  either  in  its  entirety  or  as  to  a
certain product and a certain country, by providing Onxeo with advance notice.

From the execution of the agreement through March 1, 2018, no milestones were met and no royalties were earned, therefore, we did

not pay or accrue/expense any milestone or royalty payments under the Onxeo option agreement.

Income Taxes

We use an asset and liability approach for accounting for deferred income taxes, which requires recognition of deferred income tax
assets and liabilities for the expected future tax consequences of events that have been recognized in our financial statements, but have not
been reflected in our taxable income. Estimates and judgments occur in the calculation of certain tax liabilities and in the determination of
the recoverability of certain deferred income tax assets, which arise from temporary differences and carry forwards. Deferred income tax
assets and liabilities are measured using the currently enacted tax rates that apply to taxable income in effect for the years in which those
tax assets and liabilities are expected to be realized or settled.

We regularly assess the likelihood that our deferred income tax assets will be realized from recoverable income taxes or recovered
from future taxable income. To the extent that we believe any amounts are more likely not to be realized, we record a valuation allowance
to reduce the deferred income tax assets. In the event we determine that all or part of the net deferred tax assets are not realizable in the
future, an adjustment to the valuation allowance would be charged to earnings in the period such determination is made. Similarly, if we
subsequently  realize  deferred  income  tax  assets  that  were  previously  determined  to  be  unrealizable,  the  respective  valuation  allowance
would be reversed, resulting in an adjustment to earnings in the period such determination is made.

Internal Revenue Code Section 382 provides that, after an ownership change, the amount of a loss corporation’s net operating loss
(“NOL”) for any post-change year that may be offset by pre-change losses shall not exceed the section 382 limitation for that year. Because
we will continue to raise equity in the coming years, section 382 may limit our usage of NOLs in the future.

Based on the available evidence, we believe that the Company was not likely to be able to utilize our minimal deferred tax assets in
the future and, as a result, we recorded a full valuation allowance for the years ended December 31, 2017 and 2016. We intend to maintain
the valuation allowance until sufficient evidence exists to support their reversal. We regularly review our tax positions and for a tax benefit
to  be  recognized,  the  related  tax  position  must  be  more  likely  than  not  to  be  sustained  upon  examination. Any  amount  recognized  is
generally the largest benefit that is more likely than not to be realized upon settlement. Our policy is to recognize interest and penalties
related to income tax matters as an income tax expense. For the years ended December 31, 2017 and 2016, the Company did not have any
interest or penalties associated with unrecognized tax benefits.

We  are  subject  to  U.S.  federal,  Illinois  and  California  income  taxes.  Tax  regulations  within  each  jurisdiction  are  subject  to  the
interpretation of the related tax laws and regulations and require significant judgment to apply. We are subject to U.S. federal, state and
local tax examinations by tax authorities for the years ended December 31, 2017 and 2016. We plan on filing our tax returns for the year
ending December 31, 2017 prior to the respective filing deadlines in all applicable jurisdictions.

On December 22, 2017, the Tax Cuts and Jobs Act of 2017 was enacted by the U.S. President. The Tax Reform Bill is effective as
of January 1, 2018. In accordance with ASC guidance, deferred tax assets/liabilities in our financial statements are to be reflected at the tax
rate in which the deferred tax assets/liabilities are anticipated to be realized. As a result, we changed the tax rate for tax provision purposes
at December 31, 2017 from 34% to 21%.

Stock-Based Compensation

We account for stock-based compensation arrangements with employees, nonemployee directors and consultants using a fair value
method, which requires the recognition of compensation expense for costs related to all stock-based payments, including stock options. The
fair value method requires us to estimate the fair value of stock-based payment awards on the date of grant using an option pricing model.

39

 
 
 
 
 
 
 
 
 
 
 
 
 
 
Stock-based compensation costs for options granted to our employees and nonemployee directors are based on the fair value of the
underlying  option  calculated  using  the  Black-Scholes  option-pricing  model  on  the  date  of  grant  for  stock  options  and  recognized  as
expense on a straight-line basis over the requisite service period, which is the vesting period. Determining the appropriate fair value model
and  related  assumptions  requires  judgment,  including  estimating  stock  price  volatility,  forfeiture  rates  and  expected  term.  The  expected
volatility  rates  are  estimated  based  on  the  actual  volatility  of  comparable  public  companies  over  the  expected  term.  We  selected  these
companies  based  on  comparable  characteristics,  including  market  capitalization,  risk  profiles,  stage  of  development  and  with  historical
share price information sufficient to meet the expected life of the stock-based awards. The expected term for options granted during the
years  ended  December  31,  2017  and  2016  is  estimated  using  the  simplified  method.  Forfeitures  are  estimated  at  the  time  of  grant  and
revised,  if  necessary,  in  subsequent  periods  if  actual  forfeitures  differ  from  those  estimates.  We  have  not  paid  dividends  and  do  not
anticipate  paying  a  cash  dividend  in  the  future  vesting  period  and,  accordingly,  use  an  expected  dividend  yield  of  zero.  The  risk-free
interest rate is based on the rate of U.S. Treasury securities with maturities consistent with the estimated expected term of the awards. The
measurement of consultant share-based compensation is subject to periodic adjustments as the underlying  equity  instruments  vest  and  is
recognized as an expense over the period over which services are rendered.

Stock Option Plan

In April  2016,  our  Board  and  the  preferred  stockholders  representing  a  majority  in  interest  of  our  outstanding  stock  approved  the
Amended and Restated Monopar Therapeutics Inc. 2016 Stock Incentive Plan (the “Plan”), allowing us to grant up to an aggregate 700,000
shares (as adjusted subsequent to the Conversion) of stock awards, stock options, stock appreciation rights and other stock-based awards to
our employees, non-employee directors and consultants. In October 2017, our Board increased the stock option pool up to 1,600,000 shares.
Through December 31, 2017, our Board granted to Board Members, our Chief Financial Officer, our Acting Chief Medical Officer, and our
Senior Vice President of Clinical Development stock options to purchase up to an aggregate 555,520 shares of our common stock at an
exercise price of $0.001 par value and stock options to purchase up to an aggregate 103,072 shares of our common stock at an exercise price
of $6.00 based upon third party valuations of our common stock and based on the price per share at which common stock was sold in our
most recent private offering.

Under  the  Plan,  the  per  share  exercise  price  for  the  shares  to  be  issued  upon  exercise  of  an  option  is  determined  by  our  Plan
administrator,  except  that  the  per  share  exercise  price  cannot  be  less  than  100%  of  the  fair  market  value  per  share  on  the  grant  date.  In
connection with our stock options issued in April 2016, December 2016, and February 2017, fair market value was established by our Plan
Administrator  using  recently  obtained  third  party  valuation  reports.  In  connection  with  our  stock  options  issued  in  September  2017,
November  2017,  and  January  2018,  fair  market  value  was  established  by  our  Plan Administrator  based  on  the  price  per  share  at  which
common stock was sold in our most recent private offering. Options generally expire after ten years.

The fair market value of the 273,000 options granted in April 2016, the 7,000 options granted in December 2016 and the 275,520
options granted in February 2017 was nominal at the time of grant because of both the low number of options granted prior to Conversion
in March 2017 and the low exercise price (equal to par value $0.001). For employees that were previously consultants at the time of grant,
the  fair  market  value  during  the  year  ended  December  31,  2017  totaled  $32,401  of  which  $26,498  was  recorded  as  research  and
development  expenses  and  $5,903  was  recorded  as  general  and  administrative  expenses.  In  September  2017,  we  granted  three  Board
members  options  to  purchase  up  to  21,024  shares  of  our  common  stock  each.  The  options  for  these  board  members  have  a  six-month
vesting cliff and vest between 24 and 48 months, depending on the Board member's prior months of service. The fair market value of the
aggregate 63,072 options granted to Board members totaled $20,962 during the year ended December 31, 2017 and was recorded as general
and administrative expenses. In November 2017, we granted options to purchase up to 40,000 shares of our common stock to an employee.
The options for the employee have a six-month vesting cliff and vest over 48 months. The fair market value of the 40,000 options granted
to an employee during the year ended December 31, 2017 totaled $5,502 and was recorded as general and administrative expenses.

We recognize as an expense the fair value of options granted to persons who are neither employees nor directors. The fair value of
expensed options was based on the Black-Scholes option-pricing model assuming the following factors: 6.1 to 5.3 year expected term, 57%
volatility, 2.2% to 1.2% risk free interest rate and zero dividends. Stock-based compensation expense for non-employees for the year ended
December 31, 2017 and 2016 was $251,842 and $0, respectively, of which $199,769 and $0, respectively, was recorded as research and
development expenses and $52,073 and $0, respectively, as general and administrative expenses.

40

 
 
 
 
 
 
 
 
 
Stock option activity under the Plan from January 1, 2017 through December 31, 2017 is as follows:

Balances, January 1, 2017
Increase in option pool(1)
Granted(2)
Forfeited
Exercised
Balances, December 31, 2017

Options Outstanding

Options
Available

Number of
Options

420,000 
900,000 
(378,592)    

- 
- 
941,408 

280,000 
- 
378,592 
- 
- 
658,592 

  $

Weighted-
Average
Exercise Price  
0.001 
- 
1.63 
- 
- 
0.94 

(1) The option pool was increased to 1,600,000 effective October 26, 2017.
(2) 336,544  options  vest  6/48ths  at  the  six-month  anniversary  of  grant  date  and  1/48th  per  month  thereafter,  21,024  options  vest
6/24ths on the six-month anniversary of grant date and 1/24th per month thereafter, and 21,024 options vest 6/42nds on the six-
month anniversary of grant date and 1/42nd per month thereafter.

A summary of options outstanding as of December 31, 2017 is shown below:

Exercise Prices

  $
  $

0.001 
6.00 

Number of Shares
Subject to Options
Outstanding

555,520 
103,072 
658,592 

Weighted Average Remaining
Contractual Term
8.7 years
9.6 years

Number of Shares
Subject to Options Fully
Vested and Exercisable  
337,400 
- 
337,400 

Weighted Average
Remaining Contractual
Term
8.4 years
N/A     

No income tax benefits have been recognized in the statements of operations for stock-based compensation arrangements.

We recognize as an expense the fair value of options granted to persons who are neither our employees nor directors. The fair value

of expensed options is based on the Black-Scholes option-pricing.

Results of Operations

Comparison of the Years Ended December 31, 2017 and December 31, 2016

The following table summarizes the results of our operations for the years ended December 31, 2017 and 2016:

(in thousands)
Revenue

Research and development expenses
In-process research and development expenses
General and administrative expenses

Total operating expenses

Operating loss
Interest and other income
Net loss

41

Year Ended December 31,

2017

2016

Increase
(Decrease)

  $

- 

  $

- 

  $

- 

935 
14,502 
1,166 

280 
- 
913 

655 
14,502 
253 

16,603 

1,193 

15,410 

(16,603)    
48 
(16,555)   $

(1,193)    
7 
(1,186)   $

(15,410)
41 
(15,369)

  $

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
  
 
 
 
 
 
 
 
  
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
  
   
  
   
  
   
   
   
   
   
   
   
   
   
 
   
  
   
  
   
  
   
   
   
 
   
  
   
  
   
  
   
   
   
   
 
 
R&D Expenses

R&D expenses for the year ended December 31, 2017 were approximately $0.94 million, compared to approximately $0.28 million

for the year ended December 31, 2016, an increase of approximately $0.66 million. This increase was primarily attributed to:

Research and Development Expense (in thousands)
Increased consulting in clinical development for Validive
Stock-based compensation (non-cash) for consultants
Salaries and benefits for R&D staff hired in Q4 2017
Stock-based compensation (non-cash) for employees in Q4 2017
Other, net
Net increase in R&D expenses

In-process Research and Development ("IPR&D") Expenses

Year ended
December 31,
2017 versus
year ended
December 31,
2016

  $

  $

254 
200 
152 
26 
23 
655 

IPR&D expenses for the year ended December 31, 2017 of $14.5 million represents the $1 million license fee for Validive and $13.5
million  representing  the  value  of  MNPR-201,  including  transaction  costs,  acquired  from  TacticGem  LLC  in  August  2017.  IPR&D
represents the costs of acquiring or licensing technologies that have not reached technological feasibility and have no alternative future use.

General and Administrative (“G&A”) Expenses

G&A expenses for the year ended December 31, 2017 were approximately $1.18 million, compared to approximately $0.91 million

for the year ended December 31, 2016, an increase of approximately $0.27 million. This increase was primarily attributed to:

Year ended
December 31,
2017 versus
year ended
December 31,
2016

General and Administration Exp. (in thousands)

Intellectual property legal costs for MNPR-201 (GPX-150) and international filings for MNPR-101
Increase in CEO’s salary plus new hires in Q4 2017
Fees and expenses for new Board members
Stock-based compensation (non-cash) for consultant
Audit services related to quarterly reviews
Stock-based compensation (non-cash) for new Board members
Website revisions
Consulting in 2016 for potential transaction not repeated in 2017
Legal expenses in 2016 were recorded as G&A expenses, in 2017 were recorded as IPR&D expense and deferred offering
costs (a current asset)

  $

197 
95 
76 
52 
46 
21 
17 
(36)

(215)

Net increase in G&A expenses

Interest Income

  $

253 

Interest income for the year ended December 31, 2017 increased by approximately $0.04 million versus the year ended December
31,  2016  due  to  higher  bank  balances  resulting  from  funds  raised  in  2017.  Interest  income  was  related  to  interest  earned  on  our  cash
equivalent investments in two business savings accounts and on our escrow account.

42

 
 
 
 
 
 
 
 
 
 
   
   
   
   
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
   
   
   
   
   
   
   
 
   
  
 
 
 
 
Liquidity and Capital Resources

Sources of Liquidity

We  have  incurred  losses  and  cumulative  negative  cash  flows  from  operations  since  our  inception  in  December  2014  and,  as  of
December 31, 2017 we had an accumulated deficit of approximately $18.4 million. We anticipate that we will continue to incur losses for
the foreseeable future. We expect that our research and development and general and administrative expenses will increase, and, as a result,
we anticipate that we will need to raise additional capital to fund our operations, which we may seek to obtain through a combination of
equity offerings, debt financings, strategic collaborations and grant funding. From our inception, through March 1, 2018, we have financed
our operations primarily through private placements of our preferred stock and common stock, the $4.8 million received (net of transaction
costs)  received  in  the  Gem  Transaction  (as  defined  below),  and  our  Cancer  Research  UK  collaboration. As  of  March  1,  2018,  we  have
received  net  proceeds  of  approximately  $4.70  million  (net  of  issuance  costs)  from  the  sale  of  our  preferred  stock  which  have  been
converted into common stock and we sold 789,674.33 shares of our common stock for net proceeds of approximately $4.71 million. We
anticipate that the funds raised to-date will fund our minimal operations through March 2019.

We invest our cash equivalents in a money market account.

Contribution to Capital

In August  2017,  our  largest  stockholder,  Tactic  Pharma,  LLC,  surrendered  2,888,727.12  shares  of  common  stock  back  to  us  as  a

contribution to the capital of the Company. This resulted in reducing Tactic Pharma’s ownership in us from 79.5% to 69.9%.

The Gem Transaction

On August  25,  2017,  Tactic  Pharma  and  Gem  Pharmaceuticals  formed  a  limited  liability  company,  TacticGem,  LLC,  with  Tactic
Pharma contributing 4,111,272.88 shares of our common stock and Gem contributing assets and $5 million in cash before transaction costs.
TacticGem then contributed the Gem assets and cash to us in exchange for 3,055,394.12 shares of our common stock. This has resulted in
TacticGem owning 77.1% of our outstanding common stock as of March 1, 2018. The contribution by TacticGem, made in conjunction
with contributions from outside investors in a private offering, was intended to qualify for tax-free treatment.

It  is  anticipated  that  this  transaction  will  increase  the  Company’s  annual  cash  burn  by  at  least  $750,000  and  will  be  significantly

higher if the Company chooses to conduct clinical trials with the Gem drug candidate programs.

The Gem Transaction was recorded on our financial statements for the year ended December 31, 2017 as follows:

Cash to be recorded on our Balance Sheet
Assembled Workforce to be recorded as In-process Research and Development Expense on our Statement of Operations
MNPR-201 (GPX-150) recorded as In-process Research and Development Expense on our Statement of Operations
Total Gem Transaction

  $ 5,000,000 
9,886 
    13,491,736 
  $ 18,501,622 

Cash Flows

The following table provides information regarding our cash flows for the years ended December 31, 2017 and 2016.

(in thousands)

Year ended December 31,

2017

2016

Increase
(decrease)
year ended
December 31,
2017 over
December 31,
2016

Cash used in operating activities
Cash provided by financing activities
Net change in cash, cash equivalents and restricted cash

  $

  $

(2,627)   $
9,536 
6,909 

  $

(1,195)   $
1,263 
68 

  $

(1,432)
8,273 
6,841 

43

 
 
 
 
 
 
 
 
 
 
 
 
   
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
   
   
 
 
During the years ended December 31, 2017 and 2016, we had net cash inflows of $6.91 million and $0.07 million, respectively.

Cash Flow Used in Operating Activities

The increase to cash used in operating activities during the year ended December 31, 2017 compared to the year ended December 31,
2016 of approximately $1.43 million was primarily due to the $1.0 million license fee for Validive paid in 2017 plus the increase in clinical
development consulting for planning our Phase 3 clinical trial for Validive. Cash used in operating activities of approximately $2.63 million
for the year ended December 31, 2017 was primarily a result of our approximately $16.55 million net loss offset by non-cash in-process
research  and  development  of  $13.50  million,  non-cash  stock-based  compensation  of  $0.31  million  and  changes  in  operating  assets  and
liabilities of approximately $0.12 million. Cash used in operating activities of approximately $1.19 million for the year ended December
31, 2016 was primarily a result of our approximately $1.19 million net loss.

Cash Flow Used in Investing Activities

There was no cash provided by or used in investing activities for the years ended December 31, 2017 and 2016.

Cash Flow Provided by Financing Activities

The  increase  of  cash  provided  by  financing  activities  during  the  year  ended  December  31,  2017  compared  to  the  year  ended
December  31,  2016  of  approximately  $8.27  million  was  due  to  the  sale  of  common  stock  during  the  year  ended  December  31,  2017  at
$6.00  per  share  for  aggregate  net  proceeds  of  $4.70  million  plus  $4.83  million  of  net  proceeds  from  the  Gem  Transaction  compared  to
$1.26 million raised during the year ended December 31, 2016 from the sale of Series A Preferred Stock.

Future Funding Requirements

We have not generated any revenue from product sales. We do not know when, or if, we will generate any revenue from product
sales. We do not expect to generate any revenue from product sales unless and until we obtain regulatory approval of and commercialize
any of our current or future drug product candidates or we out-license or sell a drug product candidate to another party. At the same time,
we  expect  our  expenses  to  increase  in  connection  with  our  ongoing  development  activities,  particularly  as  we  continue  the  research,
development, future preclinical and clinical trials of, and seek regulatory approval for, our current and future drug product candidates. If we
are able to list on Nasdaq or another national stock exchange, we expect to incur additional costs associated with operating as a listed public
company. In addition, if we obtain regulatory approval of any of our current and future drug product candidates, we will need substantial
additional funding in connection with our future continuing operations.

As a company, we have not completed development of any therapeutic products. We expect to continue to incur significant expenses

and increasing operating losses for the foreseeable future. We anticipate that our expenses will increase substantially as we:

● advance the clinical development and execute the regulatory strategy of Validive;

● continue the clinical development of MNPR-201;

● continue the preclinical and clinical development of MNPR-101;

● acquire and/or license additional pipeline drug product candidates and pursue the future preclinical and/or clinical development of

such drug product candidates;

● seek regulatory approvals for any of our current and future drug product candidates that successfully complete registration trials;

● establish  a  sales,  marketing  and  distribution  infrastructure  and  increase  or  develop  our  manufacturing  capabilities  to

commercialize any products for which we may obtain regulatory approval; and

● add operational, financial and management information systems and personnel, including personnel to support our drug product

candidate development and planned commercialization efforts.

44

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
We anticipate that the funds raised to-date will fund our minimal operations through at least the next 12 months. We have based this
estimate on assumptions that may prove to be wrong, and we could use our available capital resources sooner than we currently expect.
Because of the numerous risks and uncertainties associated with the development and commercialization of our drug product candidates,
and the extent to which we enter into collaborations with third parties to participate in the development and commercialization of our drug
product  candidates,  we  are  unable  to  estimate  the  amounts  of  increased  capital  outlays  and  operating  expenditures  associated  with  our
current  and  anticipated  drug  product  candidate  development  programs.  Our  future  capital  requirements  will  depend  on  many  factors,
including:

● the progress of regulatory interactions and clinical development of Validive;

● the progress of clinical development of MNPR-201;

● the progress of preclinical and clinical development of MNPR-101;

● the number and characteristics of other drug product candidates that we may pursue;

● the scope, progress, timing, cost and results of research, preclinical development and clinical trials;

● the costs, timing and outcome of seeking and obtaining FDA and international regulatory approvals;

● the costs associated with manufacturing and establishing sales, marketing and distribution capabilities;

● our ability to maintain, expand and defend the scope of our intellectual property portfolio, including the amount and timing of any
payments we may be required to make in connection with the licensing, filing, defense and enforcement of any patents or other
intellectual property rights;

● our need and ability to hire additional management, scientific and medical personnel;

● the effect of competing products that may limit market penetration of our drug product candidates;

● our need to implement additional internal systems and infrastructure; and

● the economic and other terms, timing and success of our existing collaboration and licensing arrangements and any collaboration,
licensing or other arrangements into which we may enter in the future, including the timing of receipt of or payment to or from
others of any milestone or royalty payments under these arrangements

See  Item  1A  -  “Risk  Factors”.  In  the  first  quarter  of  2018,  expenditures  are  expected  to  increase  in  employee  compensation  as  a
result of hiring various employees and consultants to support the planning of our Phase 3 clinical trial of Validive, in preparation for public
market listing via the Form 10 process, and in adjusting employee compensation to align with comparable public companies. There can be
no  assurance  that  any  such  events  will  occur.  We  intend  to  continue  evaluating  drug  product  candidates  for  the  purpose  of  growing  our
pipeline. Identifying and securing high quality compounds usually takes time; however, our spending could be significantly accelerated in
2018  if  additional  product  candidates  are  acquired  and  enter  clinical  development.  In  this  event,  we  may  be  required  to  expand  our
management team, and pay much higher insurance rates, contract manufacturing costs, contract research organization fees or other clinical
development costs that are not currently anticipated. We, under this scenario, would plan to pursue raising additional capital in the next 12
months. The anticipated operating cost increases from 2018 through 2019 are expected to be primarily driven by the funding of our planned
Validive Phase 3 clinical program. Office space rent in 2018 and 2019 will also likely increase as a result of requiring additional space as
we hire additional employees.

Until we can generate a sufficient amount of product revenue to finance our cash requirements, we expect to finance our future cash
needs primarily through a combination of equity offerings, debt financings, strategic collaborations and grant funding. To the extent that we
raise additional capital through the sale of equity or convertible debt securities, the ownership interest of our stockholders will be diluted,
and the terms of these securities may include liquidation or other preferences that adversely affect our stockholders’ rights. See Item 1A -
“Risk Factors – Existing and new investors will experience dilution as a result of our option plan and potential future stock sales.” Debt
financing, if available, may involve agreements that include covenants limiting or restricting our ability to take specific actions, such as
incurring  additional  debt,  making  capital  expenditures  or  declaring  dividends.  If  we  raise  additional  funds  through  marketing  and
distribution  arrangements  or  other  collaborations,  strategic  alliances  or  licensing  arrangements  with  other  parties,  we  may  have  to
relinquish valuable rights to our technologies, future revenue streams, research programs or product candidates or grant licenses on terms
that  may  not  be  favorable  to  us.  If  we  are  unable  to  raise  additional  funds  through  equity  or  debt  financings  when  needed,  we  may  be
required  to  delay,  limit,  reduce  or  terminate  our  pipeline  product  development  or  commercialization  efforts  or  grant  rights  to  others  to
develop and market product candidates that we would otherwise prefer to develop and market ourselves.

45

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Contractual Obligations and Commitments

Development and Collaboration Agreements

Onxeo SA

In June 2016, we executed an agreement with Onxeo S.A., a French public company, which gave us the exclusive option to license
(on a world-wide exclusive basis) Validive (clonidine mucobuccal tablet; clonidine MBT a mucoadhesive tablet of clonidine based on the
Lauriad mucoadhesive technology) to pursue treating severe oral mucositis in patients undergoing chemoradiation treatment for head and
neck cancers. The agreement includes clinical, regulatory, developmental and sales milestones that could reach up to $108 million if we
achieve all milestones, and escalating royalties on net sales from 5 - 10%. In September 2017, we exercised the option to license Validive
from Onxeo for $1 million, but as of March 1, 2018, we have not been required to pay Onxeo any other funds under the agreement.

Under the agreement, we are required to pay royalties to Onxeo on a product-by-product and country-by-country basis until the later
of (1) the date when a given product is no longer within the scope of a patent claim in the country of sale or manufacture, (2) the expiry of
any  extended  exclusivity  period  in  the  relevant  country  (such  as  orphan  drug  exclusivity,  pediatric  exclusivity,  new  chemical  entity
exclusivity, or other exclusivity granted beyond the expiry of the relevant patent), or (3) a specific time period after the first commercial
sale of the product in such country. In most countries, including the U.S., the patent term is generally 20 years from the earliest claimed
filing  date  of  a  non-provisional  patent  application  in  the  applicable  country,  not  taking  into  consideration  any  potential  patent  term
adjustment that may be filed in the future or any regulatory extensions that may be obtained. The royalty termination provision pursuant to
(3) described above is shorter than 20 years and is the least likely cause of termination of royalty payments.

The  Onxeo  license  agreement  does  not  have  a  pre-determined  term,  but  expires  on  a  product-by-product  and  country-by-country
basis;  that  is,  the  agreement  expires  with  respect  to  a  given  product  in  a  given  country  whenever  our  royalty  payment  obligations  with
respect to such product have expired. The agreement may also be terminated early for cause if either we or Onxeo materially breach the
agreement,  or  if  either  we  or  Onxeo  become  insolvent.  We  may  also  choose  to  terminate  the  agreement,  either  in  its  entirety  or  as  to  a
certain product and a certain country, by providing Onxeo with advance notice.

Given the strength of the Phase 2 data, we paid the $1 million fee to Onxeo and exercised the license option in order to advance the
clinical development of Validive. We fully anticipate the need to raise significant funds to support the completion of clinical development
of Validive.

Cancer Research UK

In  July  2015,  we  entered  into  a  Clinical  Trial  and  Option Agreement  (“CTOA”)  with  Cancer  Research  UK  and  Cancer  Research
Technology Limited, a wholly-owned subsidiary of Cancer Research UK. As part of the CTOA, we were obligated to deposit $0.8 million
in escrow to cover certain potential future claims, intellectual property infringement costs or termination costs incurred by Cancer Research
UK. Pursuant to this agreement Cancer Research UK conducted preclinical work, improved the manufacturing, and planned to conduct a
Phase 1a/1b clinical trial in cancer patients. Under this agreement, Cancer Research UK was to cover all costs through Phase 1a/1b clinical
studies, including manufacturing. As part of a portfolio reprioritization review, on March 21, 2018 Cancer Research UK notified us it was
closing  its  project  related  to  MNPR-101  and  would  work  to  make  arrangements  to  formally  terminate  the  agreement.    We  are  currently
reviewing  potential  alternative  collaboration  opportunities  for  MNPR-101  and  continue  to  maintain  the  program’s  intellectual  property
portfolio.

XOMA Ltd.

The intellectual property rights contributed by Tactic Pharma, LLC to us included the non-exclusive license agreement with XOMA
Ltd. for the humanization technology used in the development of MNPR-101. Pursuant to such license agreement, we are obligated to pay
XOMA Ltd. clinical, regulatory and sales milestones which could reach up to $14.925 million if we achieve all milestones for MNPR-101
The agreement does not require the payment of sales royalties. There can be no assurance that we will achieve any milestones. As of March
1, 2018, we had not reached any milestones and had not been required to pay XOMA Ltd. any funds under this license agreement.

46

 
 
 
 
 
 
 
 
 
 
 
 
 
 
Service Providers

In  the  normal  course  of  business,  we  contract  with  service  providers  to  assist  in  the  performance  of  research  and  development,
financial strategy, audit, tax and legal support. We can elect to discontinue the work under these agreements at any time. We could also
enter  into  collaborative  research,  contract  research,  manufacturing  and  supplier  agreements  in  the  future,  which  may  require  upfront
payments and/or long-term commitments of cash.

Office Lease

In May 2016, we executed a six-month office lease in Northbrook, Illinois for $1,340 per month, which was extended to December
31, 2017. Effective January 1, 2018, we leased office space in the Village of Wilmette for $2,379 per month for 24 months. This office
space  houses  our  current  headquarters.  On  November  1,  2017,  we  executed  a  month-to-month  office  lease  in  Seattle,  Washington  for
$1,249 per month for the first three months, but which tiers up to $2,495 on the last month.

Legal Contingencies

We are currently not, and to date have never been, a party to any material legal proceedings.

Indemnification

In the normal course of business, we enter into contracts and agreements that contain a variety of representations and warranties and
provide for general indemnification. Our exposure under these agreements is unknown because it involves claims that may be made against
us in the future, but that have not yet been made. To date, we have not paid any claims or been required to defend any action related to our
indemnification obligations. However, we may record charges in the future as a result of these indemnification obligations.

In  accordance  with  our  Second Amended  and  Restated  Certificate  of  Incorporation  and Amended  and  Restated  Bylaws  we  have
indemnification obligations to our officers and Board Members for certain events or occurrences, subject to certain limits, while they are
serving at our request in such capacity. There have been no claims to date. See Item 1A - “Risk Factors -  We have limited the liability of
and indemnified our directors and officers.”

Off-Balance Sheet Arrangements

To date, we have not had any off-balance sheet arrangements, as defined under SEC rules.

Recent Accounting Pronouncements

In August 2014, FASB issued ASU 2014-15, Disclosure of Uncertainties about an Entity’s Ability to Continue as a Going Concern,
which provides guidance on determining when and how reporting companies must disclose going-concern uncertainties in their financial
statements. The ASU requires management to perform interim and annual assessments of an entity’s ability to continue as a going concern
within  one  year  of  the  date  of  issuance  of  the  entity’s  financial  statements  (or  within  one  year  after  the  date  on  which  the  financial
statements are available to be issued, when applicable). Further, a company must provide certain disclosures if there is “substantial doubt
about the entity’s ability to continue as a going concern.” This ASU is effective for annual periods ending after December 15, 2016 and
interim  periods  within  annual  periods  beginning  after  December  15,  2016.  Early  adoption  is  permitted.  We  have  adopted  this  new
accounting standard in our financial statements and footnote disclosures.

In  November  2015,  the  FASB  issued  ASU  2015-17,  Balance  Sheet  Classification  of  Deferred  Taxes.  This  is  part  of  FASB’s
simplification  initiative.  The  amendments  in  this  ASU  require  that  deferred  tax  liabilities  and  assets  be  classified  as  noncurrent  in  a
classified statement of financial position. This ASU is effective for us in the first quarter of 2017. Early adoption is permitted. We have
adopted this ASU and determined that it does not have a material effect on our financial condition and results of operations for the year
ended December 31, 2017.

In January 2016, the FASB issued ASU 2016-01, Recognition and Measurement of Financial Assets and Financial Liabilities. The
purpose  is  to  enhance  the  reporting  model  for  financial  instruments  to  provide  users  of  financial  statements  with  more  decision-useful
information. This ASU is effective for us in the first quarter of 2018. Early adoption is not permitted except for limited provisions. We do
not expect the adoption of this amendment to have a material effect on our financial condition and results of operations.

47

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
In February 2016, the FASB issued ASU 2016-02, Leases, which for operating leases, requires a lessee to recognize a right-of-use
asset and a lease liability, initially measured at the present value of the lease payments, in its balance sheet. The standard also requires a
lessee to recognize a single lease cost, calculated so that the cost of the lease is allocated over the lease term, on a generally straight-line
basis. ASU  2016-02  will  be  effective  for  us  in  the  first  quarter  of  2019,  and  early  adoption  is  permitted.  We  are  currently  assessing  the
impact that adopting this new accounting standard will have on our financial statements and footnote disclosures.

In  March  2016,  the  FASB  issued ASU  2016-09,  Improvements  to  Employee  Share-Based  Payment Accounting,  which  simplifies
several aspects of the accounting for employee share-based payment transactions for both public and nonpublic companies, including the
accounting  for  income  taxes,  forfeitures,  and  statutory  tax  withholding  requirements,  as  well  as  classification  in  the  statement  of  cash
flows.  The ASU  will  be  effective  for  us  in  the  first  quarter  of  2017,  and  early  adoption  is  permitted.  We  have  adopted  this ASU  and
determined that it does not have a material effect on our financial condition and results of operations for the year ended December 31, 2017.

In November 2016, the FASB issued ASU 2016-18, Statement of Cash Flows (Topic 230): Restricted Cash. The amendments apply
to all entities that have restricted cash or restricted cash equivalents and are required to present a statement of cash flows. The amendments
address diversity in practice that exists in the classification and presentation of changes in restricted cash on the statement of cash flows.
The  amendments  require  that  a  statement  of  cash  flows  explain  the  change  during  the  period  in  the  total  of  cash,  cash  equivalents,  and
amounts generally described as restricted cash or restricted cash equivalents. As a result, amounts generally described as restricted cash and
restricted cash equivalents should be included with cash and cash equivalents when reconciling the beginning-of-period and end-of-period
total  amounts  shown  on  the  statement  of  cash  flows.  The  amendments  do  not  provide  a  definition  of  restricted  cash  or  restricted  cash
equivalents.  The  amendments  are  effective  for  public  business  entities  for  fiscal  years  beginning  after  December  15,  2017,  and  interim
periods within those fiscal years. For all other entities, the amendments are effective for fiscal years beginning after December 15, 2018,
and  interim  periods  within  fiscal  years  beginning  after  December  15,  2019.  Early  adoption  is  permitted.  We  have  early  adopted  the
amendments and have applied them using a retrospective transition method to each period presented. Therefore, we have included restricted
cash in cash equivalents and restricted cash on our statements of cash flows for the years ended December 31, 2017 and 2016.

In January 2017, the FASB issued ASU No. 2017-01, Business Combinations (Topic 805): Clarifying the Definition of a Business
(“ASU No. 2017-01”). The amendments in ASU No. 2017-01 clarify the definition of a business with the objective of adding guidance to
assist  entities  with  evaluating  whether  transactions  should  be  accounted  for  as  acquisitions  (or  disposals)  of  assets  or  businesses.  The
definition  of  a  business  affects  many  areas  of  accounting  including  acquisitions,  disposals,  goodwill  and  consolidation.  For  public
companies,  the  amendments  are  effective  for  annual  periods  beginning  after  December  15,  2017,  including  interim  periods  within  those
periods. For all other companies and organizations, the amendments are effective for annual periods beginning after December 15, 2018,
and interim periods within annual periods beginning after December 15, 2019. We are currently assessing the impact that adopting this new
accounting standard will have on our financial statements and footnote disclosures.

In  May  2017,  the  FASB  issued  ASU  No.  2017-09,  Compensation-Stock  Compensation  (Topic  718):  Scope  of  Modification
Accounting. The amendment amends the scope of modification accounting for share-based payment arrangements, provides guidance on
the types of changes to the terms or conditions of share-based payment awards to which an entity would be required to apply modification
accounting  under ASC  718.  This ASU  is  effective  for  all  entities  for  annual  periods,  and  interim  periods  within  those  annual  periods,
beginning after December 15, 2017. Early adoption is permitted, including adoption in any interim period for: (a) public business entities
for  reporting  periods  for  which  financial  statements  have  not  yet  been  issued,  and  (b)  all  other  entities  for  reporting  periods  for  which
financial  statements  have  not  yet  been  made  available  for  issuance.  We  are  currently  assessing  the  impact  that  adopting  this  new
accounting standard will have on our financial statements and footnote disclosures.

In  July  2017,  the  FASB  issued ASU  No.  2017-11,  Earnings  Per  Share  (Topic  260)  Distinguishing  Liabilities  from  Equity  (Topic
480)  Derivatives  and  Hedging  (Topic  815)  (Part  I) Accounting  for  Certain  Financial  Instruments  with  Down  Round  Features,  (Part  II)
Replacement  of  the  Indefinite  Deferral  for  Mandatorily  Redeemable  Financial  Instruments  of  Certain  Nonpublic  Entities  and  Certain
Mandatorily  Redeemable  Noncontrolling  Interests  with  a  Scope  Exception.  This  ASU  simplifies  the  accounting  for  certain  financial
instruments with down round features, a provision in an equity-linked financial instrument (or embedded feature) that provides a downward
adjustment  of  the  current  exercise  price  based  on  the  price  of  future  equity  offerings.  Down  round  features  are  common  in  warrants,
preferred shares, and convertible debt instruments issued by private companies and development-stage public companies. This new ASU
requires companies to disregard the down round feature when assessing whether the instrument is indexed to its own stock, for purposes of
determining  liability  or  equity  classification.  The  provisions  of  this  new ASU  related  to  down  rounds  are  effective  for  public  business
entities  for  fiscal  years,  and  interim  periods  within  those  fiscal  years,  beginning  after  December  15,  2018.  For  all  other  entities,  the
amendments  are  effective  for  fiscal  years  beginning  after  December  15,  2019,  and  interim  periods  within  fiscal  years  beginning  after
December 15, 2020. Early adoption is permitted for all entities. We are currently assessing the impact that adopting this new accounting
standard will have on our financial statements and footnote disclosures.

48

 
 
 
 
 
 
 
 
 
Item 8. Financial Statements and Supplementary Data

The information required to be filed in this item appears on pages F-1 to F-24 of this Annual Report on Form 10-K.

Documents filed as part of this Annual Report on Form 10-K:

Report of Independent Registered Public Accounting Firm

Balance Sheets as of December 31, 2017 and 2016

Statements of Operations for the Years Ended December 31, 2017 and 2016

Statements of Stockholders’ Equity for the Years Ended December 31, 2017 and 2016

Statements of Cash Flows for the Years Ended December 31, 2017 and 2016

Notes to Financial Statements

Page
F-2

F-3

F-4

F-5

F-6

F-7 to F-24

49

 
 
 
 
  
 
 
 
 
   
 
 
   
 
 
   
 
 
   
 
 
   
 
 
 
 
 
 
 
Item 9: Changes in and Disagreements with Accountants on Accounting and Financial Disclosure

PART II – FINANCIAL INFORMATION

None.

 Item 9a: Controls and Procedures

Our  Chief  Executive  Officer  and  Chief  Financial  Officer  have  provided  certifications  filed  as  Exhibits  31.1  and  32.1,  and  31.2,
respectively.  Such  certifications  should  be  read  in  conjunction  with  the  information  contained  in  this  Item  9A  for  a  more  complete
understanding of the matters covered by those certifications.

(a) Management’s Annual Report on Internal Control over Financial Reporting

Our  management  is  responsible  for  establishing  and  maintaining  adequate  internal  control  over  financial  reporting,  as  defined  in
Rule  13a15(f)  of  the  Securities  Exchange Act  of  1934  (the  “Exchange Act”).  Our  internal  control  over  financial  reporting  is  a  process
designed to provide reasonable assurance regarding the reliability of the financial reporting and the preparation of financial statements for
external purposes in accordance with U.S. generally accepted accounting principles. This process includes those policies and procedures (i)
that  pertain  to  the  maintenance  of  records  that,  in  reasonable  detail,  accurately  and  fairly  reflect  the  transactions  and  dispositions  of  our
assets. (ii) that receipts and expenditures are being made only in accordance with authorizations of our management and directors. (iii) that
provide  reasonable  assurance  regarding  prevention  or  timely  detection  of  unauthorized  acquisition,  use,  or  disposition  of  our  assets  that
could  have  a  material  effect  on  our  financial  statements.  and  (iv)  that  provide  reasonable  assurance  that  transactions  are  recorded  as
necessary to permit preparation of financial statements in accordance with GAAP. Because of its inherent limitations, internal control over
financial  reporting  may  not  prevent  or  detect  misstatements. Also,  projections  of  any  evaluation  of  the  internal  control  over  financial
reporting to future periods are subject to risk that the internal control may become inadequate because of changes in conditions, or that the
degree of compliance with policies or procedures may deteriorate.

This annual report does not include a report of management's assessment regarding internal controls over financial reporting or an
attestation report of the Company's registered public accounting firm due to a transition period established by SEC rules for newly public
companies.

(b) Disclosure Controls and Procedures

We carried out an evaluation, under the supervision and with the participation of our management, including our Chief Executive
Officer and Chief Financial Officer, of the effectiveness of our disclosure controls and procedures as of December 31, 2017, pursuant to
Rules 13a15(e) and 15d15(e) under the Exchange Act. Based on that evaluation, our Chief Executive Officer and Chief Financial Officer
have concluded that our disclosure controls and procedures, as of such date, were effective.

(c) Changes in Internal Control over Financial Reporting

We have concluded that the financial statements and other financial information included in this Annual Report on Form 10-K fairly

present in all material respects our financial condition, results of operations and cash flows as of, and for, the periods presented.

There have been no changes in our internal control over financial reporting during the fourth quarter and the year ended December

31, 2017 that have materially affected, or are reasonably likely to materially affect, our internal control over financial reporting.

50

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Item 10. Directors and Executive Officers and Corporate Governance.

PART III

The  Members  of  our  Board  of  Directors,  each  of  whom  serves  until  the  next  annual  meeting  of  stockholders,  and  the  executive

officers of the Company, each of whom serves at the discretion of the Board of Directors are as follows:

Name
Christopher M. Starr, Ph.D.

Age
65

Chandler D. Robinson, MD
MBA MSc

Andrew P. Mazar, Ph.D.

Kim R. Tsuchimoto

Patrice Rioux, MD Ph.D.

Michael J. Brown, MSc

Raymond “Bill” Anderson,
MBA

Arthur Klausner, MBA

34

56

55

66

60

76

57

  Positions

Executive Chairman, Director, Member of the Audit
Committee, the Compensation Committee, and the
Corporate Governance & Nominating Committee

Director Since
December 2014

Chief Executive Officer, Director

December 2014

Executive Vice President of Research and
Development, Chief Scientific Officer, Director

December 2014

  Chief Financial Officer

  Acting Chief Medical Officer

Director, Member of the Audit Committee, the
Compensation Committee, and the Corporate
Governance & Nominating Committee

Director, Chair of the Audit Committee, Member of
the Compensation Committee and the Corporate
Governance & Nominating Committee

Director, Member of the Audit Committee, the
Compensation Committee, and the Corporate
Governance & Nominating Committee

-

-

December 2014

April 2017

August 2017

Kirsten Anderson

50

  Senior Vice President, Clinical Development

-

Backgrounds of our executive officers and board members are discussed below.

Executive Officers and Board Members

Christopher M. Starr, PhD - Executive Chairman

Dr.  Starr  is  a  co-founder  and  has  been  our  Executive  Chairman  and  a  Board  Member  of  ours  and  our  predecessor  Monopar
Therapeutics, LLC since its inception in December 2014. Dr. Starr’s primary responsibility as our Executive Chairman is to work with our
Chief  Executive  Officer  and  the  rest  of  our  Board  to  set  our  strategic  direction  and  provide  guidance  to,  and  oversight  of  our  Chief
Executive Officer. Our Chairman also sets the agenda for Board meetings and presides over them. Dr. Starr was the co-Founder and served
as the initial chief executive officer (“CEO”) at Raptor Pharmaceuticals (“Raptor”), a public company (Nasdaq: RPTP), since its inception
in  2006  through  December  2014  and  continued  to  serve  Raptor  as  a  member  of  its  board  of  directors  until  Raptor  was  sold  to  Horizon
Pharma plc in October 2016. The principal business of Raptor is the development and commercialization of treatments for rare diseases.
Dr. Starr’s primary responsibilities as CEO included the day to day leadership and performance of Raptor which had one approved drug
marketed  in  the  U.S.  and  Europe.  Dr.  Starr  co-founded  BioMarin  in  1997,  a  public  company  (Nasdaq:  BMRN)  where  he  last  served  as
Senior  Vice  President  and  Chief  Scientific  Officer  overseeing  the  approval  of  three  drugs  until  starting  Raptor  in  2006. As  Senior  Vice
President  at  BioMarin,  Dr.  Starr  was  responsible  for  managing  a  Scientific  Operations  team  of  181  research,  process  development,
manufacturing and quality personnel through the successful development of commercial manufacturing processes for its biologic enzyme
replacement therapy and small molecule products, and supervised the cGMP design, construction and licensing of BioMarin’s proprietary
biological manufacturing facility. From 1991 to 1997, Dr. Starr supervised research and commercial programs at BioMarin’s predecessor
company, Glyko, Inc., where he served as Vice President of Research and Development. Prior to his tenure at Glyko, Inc., Dr. Starr was a
National Research Council Associate at the National Institutes of Health. Dr. Starr earned a B.S. from Syracuse University and a Ph.D. in
Biochemistry and Molecular Biology from the State University of New York Health Science Center, in Syracuse, New York.

51

 
 
 
 
 
 
 
 
 
 
 
   
   
   
 
 
 
 
   
   
   
 
 
 
 
   
   
   
 
 
 
   
   
   
 
 
 
   
   
   
 
 
 
 
   
   
   
 
 
 
 
   
   
   
 
 
 
 
   
   
   
 
 
 
 
 
 
 
 
Chandler D. Robinson, MD MBA MSc - Chief Executive Officer

Dr. Robinson is a co-founder and has been our CEO and a Board Member of ours and our predecessor Monopar Therapeutics, LLC
since its inception in December 2014. Dr. Robinson’s primary responsibilities as CEO are for our day to day leadership and performance.
Since 2010, Dr. Robinson has been, and continues to be, a manager of Tactic Pharma LLC (“Tactic”), which he co-founded and led as CEO
until it became a holding company in April 2014. Tactic acquired and developed preclinical and clinical stage compounds. In 2010, Tactic
acquired a drug on which Dr. Robinson conducted research at Northwestern University. Tactic licensed the drug to a company in Europe
and manufactured it for sale on a Named Patient basis throughout Europe. In April 2014, Tactic sold its remaining rights to the compound
to three large European investment firms and this compound is currently in a Phase 3 clinical trial for Wilson disease. Among his previous
experiences,  Dr.  Robinson  in  2008  worked  at  Onyx  Pharmaceuticals  in  their  Nexavar  marketing  division,  from  2008  to  2009  as  a  co-
manager of a healthcare clinic in San Jose CA, from 2004 to present as Founder and President of an undergraduate research focused non-
profit now in its 14th year, and from 2006 to 2007 as part of a quantitative internal hedge-fund style team at Bear Stearns investment bank.
He  was  previously  on  the  board  of  Wilson  Therapeutics  (Nasdaq:  WTX)  and  is  currently  on  the  board  of  Northwestern  University’s
Chemistry of Life Processes Institute. Dr. Robinson graduated summa cum laude from Northwestern University, earned a master's degree
in  International  Health  Policy  and  Health  Economics  from  the  London  School  of  Economics  on  a  Fulbright  Scholarship,  an  MBA  from
Cambridge University on a Gates Scholarship through Bill Gates’ Trust, and an MD from Stanford University.

Andrew P. Mazar, PhD – Executive Vice President of Research and Development, and Chief Scientific Officer

Dr.  Mazar  is  a  co-founder  and  has  been  our  Chief  Scientific  Officer  and  a  Board  Member  of  ours  and  our  predecessor  Monopar
Therapeutics,  LLC,  since  inception  in  December  2014.  Dr.  Mazar  became  our  Executive  Vice  President  of  Research  and  Development
effective as of November 1, 2017. Dr. Mazar’s primary responsibilities for us are the day to day leadership and performance of our research
and  development  activities.  Dr.  Mazar  has  spent  28  years  working  on  drug  discovery  and  development  at  the  interface  of  academia  and
industry  and  has  founded  or  co-founded  8  start-up  companies  to  commercialize  new  drug  discoveries,  including  Tactic  Pharma  LLC
(“Tactic”),  which  acquired  and  developed  preclinical  and  clinical  stage  compounds.  He  is  also  internationally  recognized  for  his  basic
research  work  on  the  role  of  the  urokinase  plasminogen  activator  (uPA)  system  in  tumor  progression  as  well  as  mechanisms  of  cancer
invasion and metastasis. Prior to joining Tactic in 2010 and the Chemistry of Life Processes Institute at Northwestern University in 2009,
Dr. Mazar was the Chief Scientific Officer at Attenuon, LLC in San Diego from 2000 to 2009 and led discovery and development efforts
resulting in three drugs entering oncology clinical trials. Dr. Mazar has now overseen 18 IND-enabling efforts, many of these focused on
drugs discovered in academia.

Dr.  Mazar  is  the  previous  Chair  of  the  NCI  Nanotechnology Alliance Animal  Model  working  group  (2011-2015)  and  has  been  a
member of the NHLBI Scientific Review Board (SRB) for the SMARTT program since 2011. Dr. Mazar served as Associate Editor for
Recent Patent Reviews on Anti - Cancer Drug Discovery (2010-2013) and is currently a member of the editorial board of Clinical Cancer
Research. He most recently served as a charter member of the NIH Developmental Therapeutics Study Section (2012-2016), and has also
served on study sections for the NCI, NIDDK, NHLBI, NIH Special Emphasis Panels, VA Oncology Merit Review, AHA and the Phillip
Morris  External  Research  Program.  He  is  also  the  co-author  of  110  peer  reviewed  publications  and  18  reviews  and  book  chapters,  most
recently contributing chapters on Cancer Invasion and Metastasis to the Oxford Textbook of Clinical Oncology and The Oxford Textbook
of  Cancer  Biology.  Dr.  Mazar  has  founded  or  advised  several  start-up  companies  over  the  past  5  years  including  Tactic  Pharma  LLC,
Valence Therapeutics, Wilson Therapeutics, Panther Biotechnology, Lung Therapeutics Inc., Actuate Therapeutics, AvidTox and Tempus.

Kim R. Tsuchimoto –Chief Financial Officer

Ms.  Tsuchimoto  was  our Acting  Chief  Financial  Officer  since  June  2015,  and  became  employed  as  our  Chief  Financial  Officer
effective November 1, 2017. Ms. Tsuchimoto spent over nine years at Raptor, as its Chief Financial Officer from Raptor’s inception in May
2006 until September 2012, as Raptor’s Vice President of International Finance, Tax & Treasury from September 2012 to February 2015,
and  lastly  served  as  Raptor’s  Vice  President,  Financial  Planning  & Analysis  and  Internal  Controls  from  February  to  May  2015.  Prior  to
Raptor,  Ms.  Tsuchimoto  spent  eight  years  at  BioMarin  and  its  predecessor,  Glyko,  Inc.,  where  she  held  the  positions  of  Vice  President-
Treasurer, Vice President-Controller and Controller. Ms. Tsuchimoto received a B.S. in Business Administration from San Francisco State
University. She holds an inactive California Certified Public Accountant license.

52

 
 
 
 
 
 
 
 
 
 
Patrice Rioux, MD Ph.D. – Acting Chief Medical Officer

Dr.  Rioux  has  been  our Acting  Chief  Medical  Officer  since  December  2016.  Dr.  Rioux’s  primary  responsibilities  include  clinical
development  and  regulatory  (FDA  &  EMA)  planning,  coordination  of  clinical  operations  and  statistical  strategy,  support  of  investor
relationship. Dr. Rioux has been deeply involved in development of drugs for rare diseases for the last 20 years. His background includes
development  of  drugs  and  biologic  products  for  various  indications  across  neurodegenerative  diseases,  immunology,  pain  management,
oncology and metabolic diseases. Dr. Rioux has been performing development, medical/regulatory, and clinical consulting services through
his  consulting  company,  pRx  Consulting,  LLC  from  June  2004  to  the  present.  From  2009  to  October  2014,  Dr.  Rioux  was  the  Chief
Medical Officer at Raptor where he was responsible for securing regulatory approval of PROCYSBI, a delayed-release cysteamine for the
treatment of a lysosomal storage disease, nephropathic cystinosis, in both the U.S. and Europe. From 2005 to 2008 he served as the Chief
Medical Officer at Edison Pharmaceuticals, and as from 2000 to 2003, he served as Vice President Clinical at Repligen, where he gained
significant orphan disease experience in mitochondrial diseases as well as in autism, and auto-immune diseases. After several years as a
clinical  researcher  at  INSERM  (France),  he  started  his  career  in  the  pharmaceutical  industry  at  Biogen  in  October  1995,  working  on
multiple sclerosis, before joining Variagenics, Inc. in 1998, one of the first pharmacogenomic companies. Dr. Rioux received his Medical
Education  at  Faculté  de  Médecine  Pitié-Salpetriere,  his  Ph.D.  in  Mathematical  Statistics  at  Faculté  des  Sciences,  and  his  Degree  of
Pharmacology (pharmacokinetics and clinical pharmacology) at Faculté de Médecine Pitié-Salpetriere.

Kirsten Anderson - Senior Vice President, Clinical Development

Ms. Anderson  has  more  than  25  years  of  experience  in  the  biotech  and  pharmaceutical  industry,  with  expertise  in  oncology  drug
development,  most  recently  as  an  independent  clinical  development  consultant  for  us  from  February  2017  through  October  2017.  She
became  our  Senior  Vice  President  of  Clinical  Development  effective  November  1,  2017.  From  2008  to  2016,  she  was  at  OncoGenex
Pharmaceuticals,  where  she  served  as  Vice  President  of  Clinical  Operations  (March  2015  to  November  2016).  Since  2008,  she  has  also
held the following positions with OncoGenex: Director, Clinical Research (2008 to December 2010) and Senior Director, Clinical Research
(January  2012  to  February  2015).  Prior  to  joining  OncoGenex,  Ms  Anderson  held  clinical  trial  management  positions  at  Sonus
Pharmaceuticals, Xcyte Therapies, and Immunex, including the oversight of global clinical operations, drug safety and data management.
She has a laboratory research background and began her career at the University of Pennsylvania. Ms. Anderson earned a degree in Biology
from the University of Vermont and is completing her Masters in Biotech Enterprise (expected 2018) from Johns Hopkins University.

Michael J. Brown, MSc – Board Member

Mr.  Brown  has  been  a  Board  Member  of  ours  and  our  predecessor,  Monopar  Therapeutics,  LLC  since  its  inception  in  December
2014. Mr. Brown is also the Administrator of the Monopar 2016 Stock Incentive Plan. Mr. Brown is the Co-Founder, and since 1994 has
served  as  Chairman,  and  since  1996  as  CEO,  of  Euronet  Worldwide  Inc.  (“Euronet”),  a  public  company  (Nasdaq:  EEFT)  which  offers
payment and transaction processing and distribution solutions to financial institutions, retailers, service providers and individual consumer.
Mr. Brown has been President of Euronet since December 2014 and also served as President of Euronet from December 2006 to June 2007.
Mr.  Brown  has  been  a  member  of  the  Euronet  board  of  directors  since  December  1996  and  also  served  on  the  boards  of  Euronet’s
predecessor companies. He has a Master of Science in molecular and cellular biology.

Raymond W. Anderson, MBA MS – Board Member

Mr. Anderson  has  been  a  Board  Member  of  Monopar  since April  2017.  He  has  been  chair  of  the  audit  committee  since  October
2017.  Mr. Anderson  has  more  than  35  years  of  biopharmaceutical/medical  technology  sector  experience,  primarily  focused  in  financial
management.  Mr. Anderson  worked  at  Dow  Pharmaceutical  Sciences,  Inc.  from  July  2003  until  June  2010.  He  most  recently  served  as
Dow’s Managing Director from January 2009 to June 2010, and previously served as Dow’s Chief Financial Officer and Vice President,
Finance  and Administration.  Prior  to  joining  Dow  in  2003,  Mr. Anderson  was  Chief  Financial  Officer  for  Transurgical,  Inc.,  a  private
medical  technology  company.  Prior  to  that,  Mr. Anderson  served  as  Chief  Operating  Officer  and  Chief  Financial  Officer  at  BioMarin
Pharmaceutical Inc. from June 1998 to January 2002. Prior to June 1998, Mr. Anderson held similar executive-level positions with other
biopharmaceutical  companies,  including  Syntex  Laboratories,  Chiron  Corporation,  Glycomed  Incorporated  and  Fusion  Medical
Technologies. Mr. Anderson served as a board member and chair of the audit committee at Raptor Pharmaceutical Inc. from its founding in
2006 to its acquisition in 2016. Mr. Anderson also served as an officer in the U.S. Army Corps of Engineers, as a strategic planner and
operational profit and loss manager at General Electric and as a finance manager at Memorex. Mr. Anderson holds an M.B.A. from Harvard
University, an M.S. in Administration from George Washington University and a B.S. in Engineering from the U.S. Military Academy.

53

 
 
 
 
 
 
 
 
 
 
 
Arthur Klausner, MBA – Board Member

Mr.  Klausner  has  been  a  consultant  to  the  biopharmaceutical  industry  since  2009.  He  served  as  Chief  Executive  Officer  of  Gem
Pharmaceuticals,  LLC  (“Gem”)  from  September  2012  until  Gem’s  drug  development  assets  were  acquired  by  us  in  2017.  Gem’s  lead,
Phase 2 drug product candidate was GPX-150 (renamed MNPR-201) (5-imino-13-deoxydoxorubicin), a proprietary analog of doxorubicin
engineered specifically to retain the anticancer activity of doxorubicin while minimizing toxic effects on the heart. In addition to his role at
Gem, Mr. Klausner served as CEO of Jade Therapeutics Inc. (“Jade”) from September 2012 until December 2015. Jade’s focus was on the
development  of  proprietary,  cross-linked  hyaluronic  acid  formulations  for  ophthalmic  applications  until  its  March  2016  acquisition  by
EyeGate Pharmaceuticals, Inc. (Nasdaq: EYEG). Previously, Mr. Klausner spent a total of 18 years at the life science venture capital firms
Domain  Associates  and  Pappas  Ventures,  where  he  was  involved  in  the  investment  in  and  subsequent  nurturing  of  a  variety  of
biotechnology, specialty pharmaceutical, and medical device companies. During that time, he was a member of the board of directors at
Santarus (acquired by Salix Pharmaceuticals), X-Ceptor Therapeutics (acquired by Exelixis), Orexigen Therapeutics, Inc. (Nasdaq: OREX),
and Syndax Pharmaceuticals (Nasdaq: SNDX), and a board observer at Peninsula Pharmaceuticals (acquired by Johnson & Johnson) and
Cerexa  (acquired  by  Forest  Laboratories).  Mr.  Klausner  currently  serves  on  the  board  of  directors  of  Cennerv  Pharma  (S)  Pte.  Ltd.
(Singapore), and on advisory boards for Neurotez, Inc., and the New York University Innovation Venture Fund. He received his M.B.A.
from the Stanford University Graduate School of Business and his undergraduate degree in Biology from Princeton University.

Agreement Regarding Election of Directors

The  limited  liability  company  agreement  of  TacticGem  provides  that  the  Manager  of  TacticGem  is  required  to  vote  TacticGem’s
shares  of  our  common  stock  to  elect  Tactic  Pharma’s  nominees  to  our  Board  plus  one  person  designated  by  Gem.  The  Gem  board
nomination right terminates at such time as we achieve a listing on a national stock exchange (e.g. Nasdaq, the NYSE or similar national
stock exchange). Gem’s initial designee for election to our Board was Arthur Klausner.

Board Composition and Election of Directors

Independence of the Board of Directors

We  believe  it  is  important  to  have  independent  directors  on  our  Board  who  can  make  decisions  without  being  influenced  by
personal  interests. Additionally,  because  one  of  our  goals  is  to  qualify  for  listing  with  NADSDAQ  we  are  following  the  Nasdaq  Stock
Market  (“Nasdaq”)  listing  standards,  which  requires  that  a  majority  of  the  members  of  our  Board  of  Directors  must  qualify  as
“independent,” as affirmatively determined by our Board. Our Board consults with our counsel to ensure that our Board’s determinations
are consistent with relevant securities and other laws and regulations regarding the definition of “independent,” including those set forth in
pertinent listing standards of Nasdaq, as in effect from time to time.

Consistent with these considerations, after review of all relevant identified transactions or relationships between each director, or any
of his family members, and us, our senior management and our independent registered public accounting firm, our Board has affirmatively
determined that the following directors are independent directors within the meaning of the applicable Nasdaq listing standards: Dr. Starr,
Mr. Brown, Mr. Anderson and Mr. Klausner. In making this determination, our Board found that none of the directors had a material or
other disqualifying relationship with us. Dr. Robinson, our President and Chief Executive Officer, is not an independent director by virtue
of his employment relationship with us, and similarly Dr. Mazar by virtue of his employment relationship with us is not an independent
director.

There are no family relationships among any of our directors or executive officers.

Board Leadership Structure

We have structured our Board in a way that we believe effectively serves our objectives of corporate governance and management
oversight. We separate the roles of Chief Executive Officer and Chairman of the Board in recognition of the differences between the two
roles. We believe that the Chief Executive Officer should be responsible for Monopar’s day to day leadership and performance, while our
Executive Chairman of the Board should work with our Chief Executive Officer and the rest of our Board to set our strategic direction and
provide guidance to, and oversight of our Chief Executive Officer. Our Executive Chairman also sets the agenda for Board meetings and
presides over them.

54

 
 
 
 
 
 
 
 
 
 
 
 
 
 
Audit Committee

Our  Board  has  formed  an  audit  committee.  Mr. Anderson  has  been  appointed  as  chair  of  the  audit  committee.  Mr. Anderson  is  a
financial expert as defined by Nasdaq and is an independent board member as contemplated by Rule 10A-3 under the Exchange Act. In
addition, Dr. Starr, Mr. Klausner and Mr. Brown have been appointed as independent members of the audit committee.

The functions of our Audit Committee include, among other duties and responsibilities:

● to assist the Board of Directors in its oversight responsibilities for the integrity of the Company’s financial statements;
● to assure the quality of the accounting and financial reporting processes of the Company;
● to assure the effectiveness of the Company’s internal controls over financial reporting;
● to assist with the Company’s compliance with legal and regulatory requirements;
● to  review  and  discuss  with  management  and  the  independent  registered  public  accounting  firm  the  Company’s  annual  and
quarterly SEC reports including the audit of the annual financial statements and the reviews of the quarterly financial statements
and related disclosures;

● to be directly responsible for the appointment, compensation, retention, and oversight of the work of the independent registered
public  accounting  firm  and  any  other  independent  registered  public  accounting  firm  performing  other  audit,  review,  or  attest
services for the Company;

● to review and discuss with the Company’s management the risk assessment and risk management policies of the Company;
● to  oversee  systems  and  procedures  for  the  receipt,  retention  and  resolution  of  complaints  received  by  the  Company  regarding
accounting,  internal  financial  controls  or  auditing  matters  and  for  the  confidential  and  anonymous  submission  by  Company
employees  of  concerns  regarding  potential  fraud  or  questionable  financial,  accounting,  internal  financial  controls  or  auditing
matters;

● to  periodically  review  and  update  the  Company’s  Code  of  Business  Conduct  and  Ethics  and  review  programs  established  to

monitor compliance with and to improve employees’ knowledge of the Code;

● to review and approve or disapprove any transaction required to be disclosed according to SEC regulations between the Company
and any related party and to oversee the Company’s policies and procedures for judgments as to related party transactions; and

● to prepare the Audit Committee’s report required by SEC rules, when such requirement becomes applicable to the Company.

Code of Conduct and Business Ethics

We  have  adopted  a  Code  of  Conduct  and  Business  Ethics  that  is  applicable  to  our  principal  executive  officer,  principal  financial
officer, principal accounting officer or controller, or persons performing similar functions. It also applies to all of our employees and our
non-employee  directors.  Our  Code  of  Conduct  and  Business  Ethics  is  available  on  our  website,  will  be  provided  to  any  person  without
charge upon request, and is filed as an exhibit to this Annual Report on Form 10-K.

55

 
 
 
 
 
 
 
 
 
Corporate Governance and Nominating Committee

The Board has formed a Corporate Governance and Nominating Committee and has appointed Dr. Starr, Mr. Brown, Mr. Anderson

and Mr. Klausner as members of the committee.

It is anticipated that the functions of our corporate governance and nominating committee will include, among other things:

● identifying individuals qualified to become board members;
● recommending to our board the persons to be nominated for election as directors and to each of the board's committees;
● reviewing and making recommendations to the board with respect to management succession planning;
● developing and recommending to the board corporate governance guidelines; and
● overseeing an annual evaluation of the board.

Compensation Committee

Our  Board  has  also  formed  a  Compensation  Committee  consisting  of  Mr.  Brown  Dr.  Starr,  Mr. Anderson  and  Mr.  Klausner  as
independent  members.  It  is  anticipated  that  the  compensation  committee  will  engage  independent  third-party  compensation  experts  as
needed.

The functions of our Compensation Committee is anticipated to include, among other things:

● annually reviewing and approving corporate goals and objectives relevant to our chief executive officer's compensation;
● determining our chief executive officer's compensation;
● reviewing  and  approving,  or  making  recommendations  to  our  board  with  respect  to,  the  compensation  of  our  other  executive

officers;

● overseeing an evaluation of our senior executives;
● overseeing and administering our equity incentive plans;
● reviewing and making recommendations to our board with respect to director compensation; and
● preparing  the  annual  compensation  committee  report  to  the  extent  required  by  SEC  rules,  when  such  requirement  becomes

applicable to us.

56

 
 
 
 
 
 
 
 
 
  
 
Item 11. Executive Compensation.

Summary Compensation Table

The following table sets forth for the fiscal years  ended  December  31, 2017 and 2016, the compensation of the Company’s Chief
Executive Officer and the Company's two highest compensated executive officers whose compensation exceeded $100,000  during our last
fiscal year.

Name and
Positions

Chandler D. Robinson, M.D.,
Chief Executive Officer and Director

Andrew P. Mazar, Ph.D.,
Chief Scientific Officer and Director

Kirsten Anderson,
Senior Vice President, Clinical Development(4)

Fiscal
Year
2017
2016

2017
2016

2017
2016

Salary
($)
    318,750 
    300,000 

Bonus
($)

- 

Option
Awards
($)

All Other
Compensation 
($)
70,000(2)    388,773 
75,000(2)    375,041 

Total
($)

23(1)   
41(1)   

87,500 
- 

43,333 
- 

- 
- 

    220,466(1)    238,750(3)    546,716 
41(1)    197,500(3)    197,541 

25,000 
- 

5,502 
- 

78,550 
- 

    152,385 
- 

(1) In 2016, each of Dr. Robinson and Dr. Mazar was granted options to purchase up to 84,000 shares of our common stock as discussed
below in the section Outstanding Equity Awards at Fiscal Year End . Based upon the Black-Scholes valuation model for stock option
compensation expense, the value of Dr. Robinson’s stock options was $ 41 and the value of Dr. Mazar’s stock options was $ 41 for the year
ended December 31, 2016. The options vested 50% on the grant date (April 4, 2016), 25% on the six-month anniversary of the grant date
(October 4, 2016) and 25% on the one year anniversary of the grant date (April 3, 2017).

In 2017, each of Dr. Robinson and Dr. Mazar was granted options to purchase up to 84,000 shares of our common stock as discussed below
in  the  section  Outstanding  Equity  Awards  at  Fiscal  Year  End .  Based  upon  the  Black-Scholes  valuation  model  for  stock  option
compensation  expense,  the  value  of  Dr.  Robinson’s  stock  options  outstanding  as  of  December  31,  2017  was  $23  and  the  value  of  Dr.
Mazar’s stock options outstanding as of December 31, 2017 was $220,466 for the year ended December 31, 2017. The options granted in
2017 vested 6/48ths on the six month anniversary of grant date (August 20, 2017) and 1/48th per month thereafter.

(2)  Consisting  of  an  employer  funded  401(k)  in  the  amount  of $54,000 and  $53,000 for  2017  and  2016,  respectively,  plus $16,000  and
$22,000 in lieu of benefits for 2017 and 2016, respectively.

(3) Until November 1, 2017, Dr. Mazar was a consultant acting as chief scientific officer for  $225,000 and $197,500 in consulting fees in
2017 and 2016, respectively,  with  no  additional  compensation  for  board  member  services. As  of  November  1,  2017,  Dr.  Mazar  became
employed as our Executive Vice President of Research and Development, and Chief Scientific Officer  at an annual base salary of $350,000
and an amount in lieu of benefits of $55,000. A pro rata amount of in lieu of benefits of $13,750 is included in All Other Compensation.

(4) Until November 1, 2017, Ms. Anderson was a consultant during 2017 providing clinical development strategy for $78,550 in consulting
fees. As  of  November  1,  2017,  Ms. Anderson  became  employed  as  our  Senior  Vice  President,  Clinical  Development  at  an  annual  base
salary of $260,000 and a sign-on bonus of $25,000. On November 1, 2017, Ms. Anderson was granted options to purchase up to 40,000
shares of our common stock as discussed below in the section Outstanding Equity Awards at Fiscal Year End . Based upon the Black-
Scholes valuation model for stock option compensation expense, the value of Ms. Anderson’s stock options outstanding as of December 31,
2017 was $5,502. The options vest 6/48ths on the six month anniversary of grant date (May 1, 2018) and 1/48th per month thereafter.

57

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
   
   
  
   
 
 
   
  
   
  
   
  
   
  
   
  
   
   
   
   
   
 
 
   
  
   
  
   
  
   
  
   
  
   
   
   
   
   
   
   
   
   
 
 
 
 
 
 
 
Employment Agreements

In  December  2016,  we  entered  into  an  employment  agreement  with  Dr.  Robinson  for  his  role  as  our  chief  executive  officer.
Although we have been paying Dr. Robinson as our employee since January 1, 2016, we did not enter into a formal employment agreement
until  December  2016.  Dr.  Robinson’s  employment  agreement  is  for  an  indefinite  term  (for  at-will  employment).  The  agreement  was
amended and restated on November 1, 2017.

Under  his  employment  agreement,  Dr.  Robinson  currently  receives  a  $375,000  per  year  base  salary,  which  may  be  adjusted  from
time to time in accordance with normal business practice and in our sole discretion. In addition, Dr. Robinson will be eligible for an annual
performance  bonus,  of  up  to  50%  of  his  base  salary,  based  on  achieving  goals  as  determined  by  our  Board  and  our  Compensation
Committee. Until we obtain retirement and healthcare benefits for our eligible employees and Dr. Robinson elects to opt in to such benefits,
Dr. Robinson is entitled to an additional salary of at least $4,583.33 per month (or such greater amount as determined by our Board) in lieu
of such benefits.

On November 1, 2017, we entered into an employment agreement with Dr. Mazar for his role as our Executive Vice President of
Research  and  Development  and  Chief  Scientific  Officer.  Dr.  Mazar’s  employment  agreement  is  for  an  indefinite  term  (for  at-will
employment). Under his employment agreement, Dr. Mazar receives a $350,000 per year base salary, which may be adjusted from time to
time  in  accordance  with  normal  business  practice  and  in  our  sole  discretion.  In  addition,  Dr.  Mazar  will  be  eligible  for  an  annual
performance  bonus,  of  up  to  40%  of  his  base  salary,  based  on  achieving  goals  as  determined  by  our  Board  and  our  Compensation
Committee. Until we obtain retirement and healthcare benefits for our eligible employees and Dr. Mazar elects to opt in to such benefits,
Dr. Mazar is entitled to an additional salary of at least $4,583.33 per month (or such greater amount as determined by our Board) in lieu of
such benefits.

On November 1, 2017, we entered into an employment agreement with Ms. Tsuchimoto for her role as our Chief Financial Officer.
Ms.  Tsuchimoto’s  employment  agreement  is  for  an  indefinite  term  (for  at-will  employment).  The  agreement  was  amended  on  March  1,
2018.  Under  her  employment  agreement,  Ms.  Tsuchimoto  receives  a  $137,500  per  year  base  salary  to  reflect  50%  time,  which  may  be
adjusted  from  time  to  time  in  accordance  with  normal  business  practice  and  in  our  sole  discretion.  Ms.  Tsuchimoto  is  entitled  to  an
additional salary of up to $1,800 per month in lieu of medical, dental and vision benefits until such time the Company has such benefit
plans  in  place.  In  addition,  Ms.  Tsuchimoto  will  be  eligible  for  an  annual  performance  bonus  determined  by  our  Board  and  our
Compensation Committee.

On November 1, 2017, we entered into an employment agreement with Ms. Anderson for her role as our Senior Vice President of
Clinical Development. Ms. Anderson’s employment agreement is for an indefinite term (for at-will employment). Under her employment
agreement, Ms. Anderson receives a $260,000 per year base salary, which may be adjusted from time to time in accordance with normal
business  practice  and  in  our  sole  discretion. Ms.  Anderson's  employment  agreement  included  a  $25,000  sign-on  bonus.  In  addition,
beginning  in  2018,  Ms. Anderson  will  be  eligible  for  an  annual  performance  bonus  determined  by  our  Board  and  our  Compensation
Committee.

Outstanding Equity Awards at Fiscal Year End

The following table sets forth outstanding stock option awards held by named executive officers as of December 31, 2017.  There

were no outstanding stock awards as of December 31, 2017.

Name

Chandler D. Robinson, M.D.

Andrew P. Mazar, Ph.D

Number of
securities
underlying
unexercised
options (#)
exercisable

Number of
securities
underlying
unexercised
options (#)
unexercisable

    17,500(1)
84,000(2)  

    66,500(1)
-

    17,500(1)
84,000(2)  

    66,500(1)
-

Option exercise
price ($)

  $0.001
$0.001

  $0.001
$0.001

Option expiration date
02/19/2027
04/03/2026

02/19/2027
04/03/2026

Kirsten Anderson

    - (3)  

    40,000(3)  

  $6.00  

10/31/2027

58

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
         
         
         
 
 
 
 
 
 
         
         
         
 
 
 
 
(1) Both  Dr.  Robinson  and  Dr.  Mazar  were  granted  stock  option  awards  on  February  20,  2017  which  vested  6/48ths  on  the  six  month

anniversary of grant date (August 20, 2017) and 1/48th per month thereafter.

(2) Both  Dr.  Robinson  and  Dr.  Mazar  were  granted  stock  option  awards  on April  4,  2016  which  vested  50%  on  the  grant  date  (April  4,
2016), 25% on the six-month anniversary of the grant date (October 4, 2016) and 25% on the one year anniversary of  the  grant  date
(April 3, 2017).

(3) Ms. Anderson was granted a stock option award on November 1, 2017 which vests 6/48ths on the six month anniversary of grant date

(May 1, 2018) and 1/48th per month thereafter.

Potential Payments upon Termination or Change in Control

Each  of  Dr.  Mazar’s  and  Dr.  Robinson’s  employment  agreements  provides  that  upon  execution  and  effectiveness  of  a  release  of
claims, Dr. Mazar and Dr. Robinson will be entitled to severance payments if we terminate their employment without cause, as defined in
the  employment  agreement,  or  if  Dr.  Mazar  or  Dr.  Robinson  terminates  his  employment  with  us  for  good  reason,  as  defined  in  the
employment  agreement.  If  employment  terminates  under  these  circumstances,  in  each  case  absent  a  change  in  control,  as  defined  in  the
employment agreements, we will be obligated for a period of twelve months, (1) to pay base salary, (2) to provide that any equity awards
will continue vesting, (3) to pay the monthly premiums for COBRA coverage equal to the amount paid for similarly situated employees and
(4) to the extent allowed by applicable law and the applicable plan documents, continue to provide all of our employee benefit plans and
arrangements that the employee was receiving at the time of termination. In addition, equity awards held by the terminated employee, that
vest  solely  on  the  passage  of  time,  will  be  accelerated  by  12  months.  If  employment  terminates  under  these  circumstances,  within  12
months following a change in control, in addition to the severance described above, we will be obligated to accelerate in full the vesting of
all of the employee’s outstanding equity awards. In the case of a change in control, instead of the 12 months of base salary described above,
we will be obligated to provide an amount equal to one-and-a-half times the sum of the base salary and target bonus for the fiscal year in
which termination occurred. If either of Dr. Mazar’s or Dr. Robinson’s employment is terminated because of death or permanent disability,
we will be obligated to provide the severance described above, but for a period of three months instead of twelve months.

Ms. Anderson’s employment agreement provides that upon execution and effectiveness of a release of claims, Ms. Anderson will be
entitled to severance payments if we terminate her employment without cause, as defined in the employment agreement, or if Ms. Anderson
terminates  her  employment  with  us  for  good  reason,  as  defined  in  the  employment  agreement.  If  employment  terminates  under  these
circumstances, absent a change in control, as defined in the employment agreement, we will be obligated for a period of three months to
pay base salary, and for a period of six months (1) to provide that any vested and unexercised equity awards continue to be exercisable and
(2) to pay the monthly premiums for COBRA coverage. If employment terminates within six months following a change in control, we will
be obligated to pay six months base salary and monthly premiums for COBRA coverage for six months and accelerate in full the vesting of
all of the employee’s outstanding equity awards which would be exercisable for two years from termination. If Ms. Anderson's employment
is terminated because of death or permanent disability, we will be obligated to provide base salary for two months and monthly premiums
for COBRA coverage for two months.

Stock Option Plan

In April 2016, our Board and stockholders holding more than a majority of our outstanding convertible preferred stock approved the
Monopar  Therapeutics  Inc.  2016  Stock  Incentive  Plan  (as  subsequently  amended,  the  “Plan”),  allowing  us  to  grant  up  to  an  aggregate
700,000 shares of stock awards, stock options, stock appreciation rights and other stock-based awards to employees, non-employee directors
and consultants. Concurrently, our Board granted to non-employee board members and our acting chief financial officer stock options to
purchase up to an aggregate 273,000 shares of our common stock at an exercise price of $0.001 per share (the par value) based upon a third
party valuation of our common stock. Such stock options vest 50% on grant date, 25% on the six month anniversary of the grant date and
25%  on  the  one  year  anniversary  of  the  grant  date.  In  December  2016,  our  Board  granted  to  our  acting  chief  medical  officer  options  to
purchase up to 7,000 shares of our common stock. Such options vest monthly over six months from the grant date. In February 2017, our
Board granted to board members and our acting chief financial officer stock options to purchase up to an aggregate 275,520 shares of our
common  stock  at  an  exercise  price  of  $0.001  per  share  (the  par  value)  based  upon  a  third  party  valuation  of  our  common  stock.  Such
options vest 6/48ths upon the six month anniversary of the grant date and 1/48th per month thereafter. In September 2017 and November
2017, stock options to purchase up to an aggregate 103,072 shares of our common stock were granted at an exercise price of $6.00, based
on the price per share at which common stock was sold in our most recent private offering. 61,024 of such options vest 6/48ths upon the six
month anniversary of the grant date and 1/48th per month thereafter, 21,024 of such options vest 6/42nd upon the six month anniversary of
the grant date and 1/42nd per month thereafter and 21,024 of such options vest 6/24ths upon the six month anniversary of the grant date and
1/24th per month thereafter. On January 1, 2018, our Board granted to our acting chief medical officer options to purchase up to 32,004
shares of our common stock at an exercise price of $6 per share based upon the price per share at which common stock was sold in our most
recent  private  offering,  and  such  options  vest  12,000  on  the  date  of  grant  and  1,667  options  on  the  1st  of  each  month  thereafter.  All
outstanding stock options have a ten year term. 690,596 stock options were outstanding as of March 1, 2018.

59

 
 
 
 
 
 
 
 
 
 
 
Under the Plan, the per share exercise price for the shares to be issued upon exercise of an option is to be determined by the Plan
administrator, except that the per share exercise price may be no less than 100% of the fair market value per share on the grant date. Fair
market value is established by our Board, using third party valuation reports and recent financings. Stock options generally expire after ten
years.

The Plan provides that the Plan administrator will be our Board, a committee designated by our Board, or an individual designee. On
February 28, 2018, our independent Directors approved the appointment of a committee (the “Plan Administrator Committee”) consisting
of three independent, non-employee Directors (Dr. Starr, Mr. Brown, and Mr. Anderson) to serve as the Administrator of our 2016 Stock
Incentive  Plan.  The  Plan Administrator  Committee  will  require  a  quorum  of  at  least  two  of  the  three  Directors  on  all  decisions.  The
Administrator  has  exclusive  authority,  consistent  with  laws  and  the  terms  of  the  Plan,  to  designate  recipients  of  options  to  be  granted
thereunder  and  to  determine  the  number  and  type  of  options  and  the  number  of  shares  subject  thereto.  Prior  to  February  28,  2018,  Mr.
Brown was the Board-representative Administrator of our 2016 Stock Incentive Plan. In March 2017, at the time of the Conversion, which
resulted in a 70 for 1 split of our common stock, the Administrator effected the 70 for 1 stock split for the Plan which increased the stock
option pool from 10,000 to 700,000 and changed the stock options granted in 2016 and in February 2017 by a 70 for 1 factor. No other
features were changed on the outstanding stock options granted.

The  Plan  was  subsequently  amended  and  restated  in  October  2017,  which  was  approved  by  stockholders  holding  more  than  a
majority of our outstanding common stock, as the Amended and Restated Monopar Therapeutics Inc. 2016 Stock Incentive Plan, in order to
increase the maximum aggregate grants under the Plan from 700,000 to 1,600,000 shares of stock awards, stock options, stock appreciation
rights and other stock-based awards.

Director Compensation for Fiscal Year Ended December 31, 2017

The following table sets forth the compensation of our non-employee Board of Directors during the year ended December 31, 201 7.

Name

Christopher M. Starr, Ph.D.
Michael J. Brown
Raymond "Bill" Anderson
Arthur Klausner

Fees earned or
paid in cash
($)
100,897 
20,000 
37,500 
14,022 

Option Awards
($)

All Other
Compensation
($)

23(1)   
9,652(2)   
5,672(3)   
5,615(4)   

- 
- 
- 
- 

Total
($)
100,920 
29,652 
43,172 
19,637 

(1)  Based  upon  the  Black-Scholes  valuation  model  for  stock  option  compensation  expense,  the  value  of  Dr.  Starr’s  stock  option s
outstanding  as  of  December  31,  2017  was  $23  for  the  year  ended  December  31,  2017.  Dr.  Starr was granted  a  stock  option  award  on
February 20, 2017 which vested 6/48ths on the six month anniversary of grant date (August 20, 2017) and 1/48th per month thereafter. In
2016, Dr. Starr was granted a stock option award on April 4, 2016 which vested 50% on the grant date (April 4, 2016), 25% on the six-
month anniversary of the grant date (October 4, 2016) and 25% on the one year anniversary of the grant date (April 3, 2017).

(2)  Based  upon  the  Black-Scholes  valuation  model  for  stock  option  compensation  expense,  the  value  of  Mr.  Brown’s  stock  options
outstanding as of December 31, 2017 was $9,652 for the year ended December 31, 2017. Mr. Brown was granted a stock option award on
September 18, 2017 which vests 6/24ths on the six month anniversary of grant date (March 18, 2018) and 1/24th per month thereafter.

(3)  Based  upon  the  Black-Scholes  valuation  model  for  stock  option  compensation  expense,  the  value  of  Mr. Anderson’s  stock  options
outstanding as of December 31, 2017 was $5,672 for the year ended December 31, 2017. Mr. Anderson was granted a stock option award
on September 18, 2017 which vests 6/42nds on the six month anniversary of grant date (March 18, 2018) and 1/42nd per month thereafter.

(4)  Based  upon  the  Black-Scholes  valuation  model  for  stock  option  compensation  expense,  the  value  of  Mr.  Klausner’s  stock  options
outstanding as of December 31, 2017 was $5,615 for the year ended December 31, 2017. Mr. Klausner was granted a stock option award
on September 1, 2017 which vests 6/48ths on the six month anniversary of grant date (March 1, 2018) and 1/48th per month thereafter.

60

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
   
   
   
   
   
   
   
   
   
   
   
 
 
 
 
 
 
Options Exercised and Stock Vested

None  of  our  executive  officers  or  non-employee  directors  exercised  any  options  during  the  years  ended  December  31,  2017  and

2016.

Item 12. Security Ownership of Certain Beneficial Owners and Management and Related Stockholder Matters.

Securities Authorized for Issuance Under Equity Compensation Plans

The following table provides information as of December 31, 2017, with respect to shares of our common stock that may be issued

under existing equity compensation plans. There are no equity compensation plans that have not been approved by our security holders.

Number of
Securities to
be Issued
Upon Exercise
of
Outstanding
Options,
Warrants and
Rights

Weighted
Average
Exercise Price
of
Outstanding
Options,
Warrants and
Rights

658,592 

  $

0.94 

Number of
Securities
Remaining
Available For
Future
Issuance
under Equity
Compensation
Plans
941,408 

Plan Category
Equity compensation plans approved by security holders (1)

(1) The Monopar Therapeutics Inc. 2016 Stock Incentive Plan.

61

 
 
 
 
 
 
 
 
 
 
 
 
 
   
   
 
 
 
The following table and the related notes present information on the beneficial ownership of shares of our common stock, our only

outstanding class of stock, as of March 1, 2018 (subsequent to the Conversion) by:

● each of our directors;

● each of our named executive officers;

● all of our current directors and executive officers as a group; and

● each person known by us to beneficially own more than five percent of our common stock

Beneficial ownership is determined in accordance with the rules of the SEC and includes voting or investment power with respect to
the securities. Shares of our common stock that may be acquired by an individual or group within 60 days of March 1, 2018, pursuant to the
exercise of options or warrants, are deemed to be outstanding for the purpose of computing the percentage ownership of such individual or
group, but are not deemed to be outstanding for the purpose of computing the percentage ownership of any other person shown in the table.

Except as indicated in footnotes to this table, we believe that the stockholders named in this table have sole voting and investment
power with respect to all shares of common stock shown to be beneficially owned by them, based on information provided to us by such
stockholders.

Name and Address of Beneficial Owner
*Unless otherwise noted, addresses are: 1000 Skokie Blvd., Suite 350, Wilmette, IL 60091
TacticGem, LLC
Tactic Pharma LLC
Gem Pharmaceutical LLC
941 Lake Forest Cir.
Birmingham, AL 35244
Chandler D. Robinson, Chief Executive Officer and Director
Christopher M. Starr, Executive Chairman
Andrew P. Mazar, Executive Vice President of Research and Development, Chief
Scientific Officer and Director
Michael J. Brown, Director
Raymond “Bill” Anderson, Director

Arthur Klausner, Director
Kim R. Tsuchimoto, Chief Financial Officer
Patrice P. Rioux, Acting Chief Medical Officer
Named executive officers and directors as a group(C)

Shares of Common Stock
Beneficially Owned (A)

7,166,667(B)
4,277,939.88(B)

3,055,394.12(B)
122,502.8
157,900

122,502.8
216,132
4,504
8,066

27,860
24,001
7,850,135.6

Percent of Class Held (A)

77.1%
46.0%

32.9%
1.3%
1.7%

1.3%
2.3%
*
*

*
*
81.1%

(A) Beneficial ownership is based upon 9,291,420.614 shares of our Common Stock outstanding; and includes common stock options that
vest  within  60  days  after  March  1,  2018  as  follows  –  Chandler  D.  Robinson,  Christopher  M.  Starr  and Andrew  P.  Mazar  options  to
purchase  up  to  108,500  shares  of  common  stock,  Kim  R.  Tsuchimoto  options  to  purchase  up  to  27,860  shares  of  common  stock  and
Patrice  P.  Rioux  options  to  purchase  up  to  24,001  shares.  These  vested  option  shares  are  deemed  to  be  outstanding  and  beneficially
owned by the person holding the applicable options for the purpose of computing the percentage ownership of that person, but they are
not treated as outstanding for the purpose of computing the percentage ownership of any other person.

(B) Tactic Pharma LLC (“Tactic Pharma”) shares voting and investment power over 4,111,272.88 shares of our common stock owned by
TacticGem, and Gem Pharmaceutical LLC (“Gem”) shares voting and investment power over 3,055,394.12 shares of our common stock
owned by TacticGem, because pursuant to the TacticGem limited liability company agreement all votes of our common stock (other than
votes  for  the  election  of  directors)  are  passed  through  to  Tactic  Pharma  and  Gem  in  proportion  to  their  percentage  interests  in
TacticGem, and after an initial holding period, which ends after we have been subject to the reporting requirements of the Exchange Act
and  have  filed  all  required  reports  for  a  period  of  at  least  12  months,  either  member  of  TacticGem  can  cause  up  to  its  proportionate
shares of our common stock to be distributed to it. Tactic Pharma holds 166,667 shares of stock in its own name. Mr. Brown, Dr. Mazar
and Dr. Robinson are managers of Tactic Pharma; because of this, they control voting and dispositive power over 4,111,272.88 shares of
our  common  stock  owned  by  TacticGem,  and  over  our  Common  Stock  owned  by  Tactic  Pharma.  Gem  is  controlled  by  Pharma
Investments, LLC, which is in turn controlled by Diane M. Hendricks.

62

 
 
 
 
 
 
 
 
 
 
 
 
 
(C) Shares held by TacticGem are only included in the total beneficial ownership of our named executive officers and directors because the
limited liability agreement of TacticGem provides that the Manager of TacticGem will vote our common stock held by TacticGem to
elect Tactic Pharma’s nominees plus one person designated by Gem (until we achieve listing on a national stock exchange) to our Board,
and acting together the directors are able to control Tactic Pharma, LLC, and how it selects its nominees for our Board of Directors.

* Less than 1%

Item 13. Certain Relationships and Related Transactions, and Director Independence.

Since January 2015, we (including as Monopar Therapeutics, LLC) have engaged in the following transactions with our directors,
executive officers, holders of more than 5% of our voting securities, and affiliates or immediate family members of our directors, executive
officers and holders of more than 5% of our voting securities, and our co-founders. We believe that all of these transactions were on terms
as favorable as could have been obtained from unrelated third parties.

During the years ended December 31, 2017 and 2016, we paid or accrued legal fees to Baker & Hostetler, LLP, a large national law
firm in which our Chief Executive Officer’s family member is a law partner, approximately $300,140 and $54,000, respectively. The family
member billed a de minimis amount of time on our legal engagement with Baker & Hostetler, LLP.

Contributions by Tactic Pharma, LLC

We were initially formed as a Delaware limited liability company in December 2014, with the name Monopar Therapeutics, LLC, at
which time Tactic Pharma contributed technology and related assets to us, in exchange for 1,000,000 shares of Series Z Preferred Units,
which were exchanged for 100,000 shares of Series Z Preferred Stock at the time of our conversion to a corporation. The issued Series Z
Preferred Stock was recorded at par value $0.001 per share on our balance sheet reflecting the historical capitalized cost basis, due to the
fact that MNPR-101’s development costs were previously expensed (not capitalized) by Tactic Pharma. In March 2017, the 100,000 shares
of  Series  Z  Preferred  Stock  were  converted  into  7,000,000  shares  of  our  common  stock,  $.0001  par  value  in  connection  with  the
Conversion. See “Conversion of Preferred Stock to Common Stock”.

In August 2017, Tactic Pharma surrendered 2,888,727.12 shares of our common stock back to us as a contribution to the capital of

the Company. This reduced its ownership percentage of our common stock from 79.5% to 69.9%.

We reimbursed Tactic Pharma, a de minimis amount in monthly storage fees during the years ended December 31, 2017 and 2016. In
March 2017, Tactic Pharma wired $1 million to us in advance of the sale of our common stock at $6 per share under a private placement
memorandum. In April, we issued to Tactic Pharma 166,667 shares in exchange for the $1 million at $6 per share once we began selling
stock to unaffiliated parties under the private placement memorandum. In August 2017, Tactic Pharma surrendered 2,888,727.12 shares of
our common stock back to us as a contribution to the capital of the Company. This resulted in reducing Tactic Pharma’s ownership in us
from 79.5% to 69.9%. Following the surrender of the common stock, Tactic Pharma contributed 4,111,272.88 shares of its holdings in our
common stock to TacticGem pursuant to the Gem Transaction discussed in detail in Note 6 of our audited financial statements below. As of
December 31, 2017, Tactic Pharma beneficially owned 46% of our common stock, and TacticGem owned 77% of our common stock.

Gem Transaction

On June 27, 2017, we signed a term sheet with Gem Pharmaceuticals, LLC (“Gem”) pursuant to which Gem was to transfer assets
related to certain of its drug product candidate programs to us in exchange for 32% of our outstanding common stock on a fully-diluted
basis. The Gem transaction was structured through a limited liability company, TacticGem, which Gem formed with Tactic Pharma, LLC
(“Tactic Pharma”), our largest shareholder at that time. Gem contributed certain of Gem’s drug product candidates’ intellectual property
and agreements associated primarily with Gem’s GPX-150 (renamed MNPR-201) drug product candidate program, along with $5,000,000
in cash (the “Gem Contributed Assets”) to TacticGem for a 42.633% interest, and Tactic Pharma contributed 4,111,272.88 shares of our
common  stock  to  TacticGem  for  a  57.367%  interest.  Then,  TacticGem  contributed  the  Gem  Contributed Assets  to  us  in  exchange  for
3,055,394.12  newly  issued  shares  of  our  common  stock  (31.4%  on  a  fully-diluted  basis)  (the  two  contributions  collectively,  the  “Gem
Transaction”).  The  contribution  by  TacticGem,  made  in  conjunction  with  contributions  from  outside  investors  in  a  private  offering,  was
intended to qualify for tax-free treatment. The Gem Transaction closed on August 25, 2017. Following the Gem Transaction, TacticGem
owns  7,166,667  shares  of  our  stock.  Pursuant  to  the  TacticGem  limited  liability  company  agreement,  all  votes  of  our  common  stock  by
TacticGem (aside from the election of our Board of Directors) is required to be passed through to Tactic Pharma and Gem based on their
percentage interest (currently pursuant to this voting agreement, Tactic has voting and investment power over 4,111,272.88 shares of our
common stock and Gem has voting and investment power over 3,055,394.12 shares of our common stock). Neither Gem nor TacticGem
was a related person prior to the Gem Transaction. The TacticGem limited liability company agreement provides that its manager will vote
all shares of our common stock held by it to elect Tactic Pharma’s nominees to our Board of Directors plus one person nominated by Gem,
initially Arthur Klausner.

63

 
 
 
 
 
 
 
 
 
 
 
 
 
 
Pursuant to the Conversion and the Gem Transaction and sales of our common stock in September 2017, Tactic Pharma now holds
voting and investment power over 4,277,939.88 shares of our Common Stock, which is 46.0% of our outstanding common stock. In the
ordinary  course  of  business,  we  have  reimbursed  and  continue  to  reimburse  Tactic  Pharma  for  expenses  Tactic  Pharma  has  paid  on  our
behalf, which historically included legal patent fees and storage rental fees. Certain of our Board Members and executive officers own and
control Tactic Pharma. Although no single person has a controlling interest in Tactic Pharma, acting together they are able to control Tactic
Pharma and a large voting block of our common stock.

Stock Purchases by Directors and Executive Officers

The following table sets forth the number of shares of our common stock owned by our co-founders; each co-founder purchased such

shares at $3.57 per share (taking into account the Conversion) in 2016.

Name

Christopher M. Starr, Ph.D.
Chandler D. Robinson, M.D.
Andrew P. Mazar, Ph.D.

Related Person Status
Executive Chairman
Director, Chief Executive Officer
Director, Chief Scientific Officer

# Shares of Common
Stock
29,400
14,002.3
14,002.3

Transaction Value (and Related Person’s Interest)
($)
105,000
50,010
50,010

Also, in 2016, Michael Brown (Director), purchased 210,000 shares of our common stock (taking into account the Conversion), at

$3.57 per share, for a total transaction value of $750,000.

In 2017, Board members purchased shares of our common stock at $6 per share, as follows: Dr. Starr purchased 20,000 shares for a
transaction value of $120,000; Mr. Anderson purchased 1,000 shares for a transaction value of $6,000; and Mr. Klausner purchased 5,000
shares for a transaction value of $30,000.

Promoters and Certain Control Persons

We have not had any promoters since our formation in December 2014.

Parent Companies

Prior  to  the  Gem  Transaction,  Tactic  Pharma  was  our  parent  company,  having  a  controlling  interest  in  us.  After  the  Gem
Transaction, TacticGem became our parent company, currently having a 77.1% controlling interest in us. See “ Contributions by Tactic
Pharma, LLC” and “Gem Transaction”.

Director Independence

We have decided to follow the Nasdaq Stock Market, or Nasdaq, listing standards, which require that a majority of the members of
our Board of Directors, or our Board, must qualify as “independent,” as affirmatively determined by our Board. Our Board consults with
our counsel to ensure that our Board’s determinations are consistent with relevant securities and other laws and regulations regarding the
definition of “independent,” including those set forth in pertinent listing standards of Nasdaq, as in effect from time to time.

Consistent with these considerations, after review of all relevant identified transactions or relationships between each director, or any
of his family members, and us, our senior management and our independent registered public accounting firm, our Board has affirmatively
determined that the following four directors are independent directors within the meaning of the applicable Nasdaq listing standards: Dr.
Starr, Mr. Brown, Mr. Anderson and Mr. Klausner. In making this determination, our Board found that none of the directors had a material
or  other  disqualifying  relationship  with  us.  Dr.  Robinson,  our  President  and  Chief  Executive  Officer  is  not  an  independent  director  by
virtue  of  his  employment  relationship  with  us,  and  similarly,  Dr.  Mazar  by  virtue  of  his  employment  relationship  with  us  is  not  an
independent director.

There are no family relationships among any of our directors or executive officers.

Relationships Considered in Determining Director Independence

In  addition  to  the  stock  transactions  described  above,  in  considering  director  independence,  we  considered  the  following

transactions:

64

 
 
 
 
 
 
 
 
  
 
 
 
 
 
 
 
 
 
 
 
During  the  years  ended  December  31,  2017  and  2016,  we  were  advised  by  four  members  of  our  Board  of  Directors,  who  were
Managers  of  our  predecessor  LLC  prior  to  our  conversion  to  a  C  Corporation.  The  four  former  Managers  are  also  our  current  common
stockholders (owning approximately an aggregate 3% of our common stock outstanding as of December 31, 2017). Three of the former
Managers  are  also  Managing  Members  of  Tactic  Pharma,  LLC,  which  was,  prior  to  the  Gem  Transaction,  our  largest  and  controlling
stockholder (owning a 46% beneficial interest in us at December 31, 2017 and in partnership with Gem through TacticGem owning 77.1%).
We paid the Managing Members of Tactic Pharma, LLC the following during the years ended December 31, 2017 and 2016: Chandler D.
Robinson,  our  Co-Founder,  Chief  Executive  Officer,  common  stockholder,  Managing  Member  of  Tactic  Pharma,  LLC  and  former
Manager of our predecessor LLC, $346,545 and $322,000, respectively; and Andrew P. Mazar, our Co-Founder, Chief Scientific Officer,
common stockholder, Managing Member of Tactic Pharma, LLC and former Manager of our predecessor LLC, $300,731 and $197,500,
respectively. We also paid Christopher M. Starr, our Co-Founder, Executive Chairman of the Board of Directors, common stockholder and
former Manager of our predecessor LLC, $100,897 and $96,339 during the years ended December 31, 2017 and 2016, respectively.

In the normal course of business, our Chief Executive Officer, Board Members and consultants incur expenses on behalf of us and

are reimbursed within 30 days of submission of relevant expense reports.

Item 14. Principal Accounting Fees and Services

The  following  is  a  summary  of  the  fees  billed  and  services  provided  by  our  independent  registered  public  accounting  firm,  BPM

LLP during the years ended December 31, 2017 and 2016, respectively.

Description of Services Provided by BPM LLP
Audit Fees
Audit-Related Fees: These services relate to assurance and services reasonably related to the

performance of the audit or review of financial statements not included above.

Tax Compliance Fees: These services relate to the preparation of federal, state and foreign tax returns

and other filings.

Tax Consulting and Advisory Services: These services primarily relate to the area of tax strategy and

minimizing Federal, state, local and foreign taxes.

All Other Fees

For the year
ended
December 31,
2017 

For the year
ended
December 31,
2016

  $

83,815 

  $

32,036 

28,325 

3,150 

1,250 
0 

0 

4,910 

35,680 

65

 
 
 
 
 
 
 
 
 
 
   
   
   
   
   
   
  
   
   
 
 
Item 15. Exhibits, Financial Statement Schedule

(a)

PART IV

INDEX TO FINANCIAL STATEMENTS

Report of Independent Registered Public Accounting Firm

Balance Sheets as of December 31, 2017 and 2016

Statements of Operations for the Years Ended December 31, 2017 and 2016

Statements of Stockholders’ Equity for the Years Ended December 31, 2017 and 2016

Statements of Cash Flows for the Years Ended December 31, 2017 and 2016

Notes to Financial Statements

Page
F-2

F-3

F-4

F-5

F-6

F-7 to F-24

66

 
 
 
 
 
 
 
 
 
 
   
 
 
   
 
 
   
 
 
   
 
 
   
 
 
 
 
 
 
 
 
(b) Exhibits

The following exhibits are filed as part of this Annual Report on Form 10-K.

Document

Amended and Restated Bylaws

  Second Amended and Restated Certificate of Incorporation

Exhibit
3.1
3.2
  Clinical Trial and Option Agreement with Cancer Research UK
10.1*
  License Agreement with XOMA Ltd.
10.2*
  Option and License Agreement with Onxeo S.A.
10.3*
  Contribution Agreement (351) – Containing Registration Rights Agreement with TacticGem
10.4*
  Amended and Restated 2016 Stock Incentive Plan
10.5
  Employment Agreement of Chandler D. Robinson – terminated October 31, 2017
10.6
  Employment Agreement of Chandler D. Robinson – effective November 1, 2017
10.7
  Consulting Agreement of Kim Tsuchimoto – terminated October 31, 2017
10.8
Employment Agreement of Kim Tsuchimoto – effective November 1, 2017
10.9
  Consulting Agreement of Andrew P. Mazar – terminated October 31, 2017
10.10
  Employment Agreement of Andrew P. Mazar – effective November 1, 2017
10.11
  Consulting Agreement of pRx Consulting (Patrice Rioux) – terminated December 31, 2017
10.12
  Employment Agreement of Kirsten Anderson
10.13
  Consulting Agreement of pRx Consulting (Patrice Rioux) - effective January 1, 2018
10.14
  Amendment One to Employment Agreement of Kim Tsuchimoto – effective March 1, 2018
10.15
  Cancer Research UK Letter Dated March 21, 2018
10.16
  Statement Regarding Computation of Per Share Earnings
11
  Code of Conduct and Business Ethics
14
  Power of Attorney (included in the signature page hereto)
24.1
  Certification of Chandler Robinson, Chief Executive Officer
31.1
  Certification of Kim Tsuchimoto, Chief Financial Officer
31.2
  Certification of Chandler Robinson, Chief Executive Officer and Kim Tsuchimoto, Chief Financial Officer
32.1
101.INS
  XBRL Instance Document
101.SCH   XBRL Taxonomy Extension Schema
101.CAL   XBRL Taxonomy Extension Calculation Linkbase
101.DEF   XBRL Taxonomy Extension Definition Linkbase
101.LAB   XBRL Taxonomy Extension Label Linkbase
101.PRE   XBRL Taxonomy Extension Presentation Linkbase

Confidential Information has been omitted and filed separately with the Securities and Exchange Commission on exhibits marked with (*).
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

67

 
 
 
 
 
 
 
 
Pursuant to the requirements of Section 13 or 15(d) of the Securities Exchange Act of 1934, the registrant has duly caused this report

to be signed on its behalf by the undersigned, thereunto duly authorized.

SIGNATURES

Dated: March 26, 2018

Company MONOPAR THERAPEUTICS INC.

By:  /s/ Kim Tsuchimoto
Kim Tsuchimoto 
Chief Financial Officer (Principal Financial
Officer) 

KNOW  ALL  PERSONS  BY  THESE  PRESENTS,  that  each  person  whose  signature  appears  below  constitutes  and  appoints
Chandler Robinson and Kim Tsuchimoto, his attorneyinfact, with the power of substitution, for him in any and all capacities, to sign any
amendments to this Annual Report on Form 10K and to file the same, with exhibits thereto and other documents in connection therewith,
with  the  Securities  and  Exchange  Commission,  hereby  ratifying  and  confirming  all  that  each  of  said  attorneysinfact,  or  his  substitute  or
substitutes, may do or cause to be done by virtue hereof.

Pursuant to the requirements of the Securities Exchange Act of 1934, this report has been signed below by the following persons on

behalf of the registrant and in the capacities and on the dates indicated:

Signatures

Title

/s/ Chandler Robinson
Chandler Robinson

/s/ Kim Tsuchimoto
Kim Tsuchimoto

/s/ Andrew Mazar
Andrew Mazar

/s/ Christopher Starr
Christopher Starr

/s/ Raymond W. Anderson
Raymond W. Anderson

/s/ Michael Brown
Michael Brown

/s/ Arthur Klausner
Arthur Klausner

  Chief Executive Officer and Director

(Principal Executive Officer)

  Chief Financial Officer (Principal Financial
Officer and Principal Accounting Officer)

  Chief Scientific Officer and Director

  Executive Chairman of the Board and Director

  Director

  Director

  Director

68

Date

  March 26, 2018

  March 26, 2018

  March 26, 2018

  March 26, 2018

  March 26, 2018

  March 26, 2018

  March 26, 2018

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
  
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
    
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
INDEX TO FINANCIAL STATEMENTS

Report of Independent Registered Public Accounting Firm

Balance Sheets as of December 31, 2017 and 2016

Statements of Operations for the Years Ended December 31, 2017 and 2016

Statements of Stockholders’ Equity for the Years Ended December 31, 2017 and 2016

Statements of Cash Flows for the Years Ended December 31, 2017 and 2016

Notes to Financial Statements

F-1

Page
F-2

F-3

F-4

F-5

F-6

F-7 to F-24

 
 
 
 
 
 
 
   
 
 
   
 
 
   
 
 
   
 
 
   
 
 
 
REPORT OF INDEPENDENT REGISTERED PUBLIC ACCOUNTING FIRM

To the Stockholders and Board of Directors of
Monopar Therapeutics Inc.

Opinion on the Financial Statements

We have audited the accompanying balance sheets of Monopar Therapeutics Inc. (the "Company") as of December 31, 2017 and 2016, the
related statements of operations, stockholders’ equity and cash flows, for each of the two years in the period ended December 31, 2017, and
the related notes (collectively referred to as the "financial statements"). In our opinion, the financial statements present fairly, in all material
respects, the financial position of the Company as of December 31, 2017 and 2016, and the results of its operations and its cash flows for
each of the two years in the period ended December 31, 2017, in conformity with accounting principles generally accepted in the United
States of America.

Basis for Opinion

These  financial  statements  are  the  responsibility  of  the  Company's  management.  Our  responsibility  is  to  express  an  opinion  on  the
Company's  financial  statements  based  on  our  audits.  We  are  a  public  accounting  firm  registered  with  the  Public  Company Accounting
Oversight Board (United States) ("PCAOB") and are required to be independent with respect to the Company in accordance with the U.S.
federal securities laws and the applicable rules and regulations of the Securities and Exchange Commission and the PCAOB.

We conducted our audits in accordance with the standards of the PCAOB. Those standards require that we plan and perform the audit to
obtain reasonable assurance about whether the financial statements are free of material misstatement, whether due to error or fraud. The
Company is not required to have, nor were we engaged to perform, an audit of its internal control over financial reporting. As part of our
audits,  we  are  required  to  obtain  an  understanding  of  internal  control  over  financial  reporting  but  not  for  the  purpose  of  expressing  an
opinion on the effectiveness of the Company's internal control over financial reporting. Accordingly, we express no such opinion.

Our audits included performing procedures to assess the risks of material misstatement of the financial statements, whether due to error or
fraud, and performing procedures that respond to those risks. Such procedures included examining, on a test basis, evidence regarding the
amounts  and  disclosures  in  the  financial  statements.  Our  audits  also  included  evaluating  the  accounting  principles  used  and  significant
estimates  made  by  management,  as  well  as  evaluating  the  overall  presentation  of  the  financial  statements.  We  believe  that  our  audits
provide a reasonable basis for our opinion.

/s/ BPM LLP

We have served as the Company's auditor since 2015.

San Francisco, California

March 26, 2018

F-2

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Monopar Therapeutics Inc.
Balance Sheet

Current assets:

Cash and cash equivalents
Prepaid expenses and other current assets

Total current assets

Assets

Restricted cash

Total assets

Liabilities and Equity

Current liabilities:

Accounts payable and accrued expenses

Total current liabilities

Long term liabilities

Total liabilities

Commitments and contingencies (Note 9)

Stockholders’ equity:
Preferred stock, par value of $0.001 per share, zero shares authorized at December 31, 2017, and

200,000 shares authorized at December 31, 2016; 115,894 shares issued and outstanding, aggregate
liquidation preference of $34,768,140 at December 31, 2016

Common stock, par value of $0.001 per share, 40,000,000 authorized, 9,291,421 shares issued and

outstanding at December 31, 2017; zero shares issued and outstanding at December 31, 2016

Additional paid-in capital

Accumulated deficit

Total stockholders’ equity

Total liabilities and stockholders’ equity

The accompanying notes are an integral
part of these financial statements.

F-3

December 31

2017

2016

  $ 8,981,894 
149,342 
9,131,236 

  $ 2,072,611 
22,562 
    2,095,173 

800,031 

800,393 

  $ 9,931,267 

  $ 2,895,566 

  $

  $

311,867 
311,867 
— 

64,510 
64,510 
— 

311,867 

64,510 

— 

116 

— 
9,291 
    28,037,889 
    4,703,848 
    (18,427,780)     (1,872,908)

9,619,400     2,831,056 
  $ 2,895,566 

  $ 9,931,267 

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
   
   
 
   
  
   
  
   
   
 
   
  
   
  
   
  
   
  
   
  
   
  
   
   
   
   
 
   
  
   
  
   
   
   
  
   
  
 
   
  
   
  
   
  
   
  
   
   
   
   
   
 
 
 
Revenues

Operating expenses:

Research and development
In-process research and development
General and administrative
Total operating expenses

Loss from operations
Other income:

Interest and other income

Net loss
Net loss per share:
     Basic and diluted
Weighted average shares outstanding:
     Basic and diluted

Monopar Therapeutics Inc.
Statements of Operations

F-4

December 31,

2017

2016

  $

  $

— 
— 

— 
— 

280,355 
935,319 
— 
    14,501,622 
912,474 
1,166,186 
    1,192,829 
    16,603,127 
    (16,603,127)     (1,192,829)

48,255 

7,232 
  $(16,554,872)   $ (1,185,597)

  $

(1.89)    

8,782,037 

N/A 

N/A 

 
 
 
 
 
 
 
 
 
 
 
 
   
   
   
  
   
  
   
   
   
   
   
   
  
   
  
   
   
   
  
   
  
   
  
   
  
   
   
 
 
Monopar Therapeutics Inc.
Statement of Stockholders’ Equity

Balance at January 1, 2016
Issuance of Series A Preferred Stock at $300 per
share for cash, net of $12,500 issuance costs
Net loss
Balance at December 31, 2016
Conversion of preferred stock to common stock
Issuance of common stock at $6 per share for
cash, net of $32,400 issuance costs
Tactic Pharma shares surrendered
Shares issued in Gem transaction, net of issuance
costs of $169,257
Non-cash stock compensation
Net loss
Balance at December 31, 2017

Series A and Z
Preferred Stock

Common Stock

Additional
Paid-

  Accumulated 

  Shares

111,644 

  Amount  
112 

  Shares

  Amount  
— 

  in Capital 
    3,441,352 

0 

  Deficit  

Total
Equity  
(687,311)     2,754,153 

4,250 
— 
115,894 
(115,894)    

— 
4 
— 
— 
116 
0 
(116)     8,335,080 

— 
— 
— 
8,335 

    1,262,496 
— 
    4,703,848 

(8,219)    

    1,262,500 
(1,185,597)     (1,185,597)
(1,872,908)     2,831,056 
— 

— 

— 
— 

— 
— 
— 
— 

  $

— 
— 

789,674 
    (2,888,727)    

790 
(2,889)    

    4,704,856 
2,889 

— 
— 

    4,705,646 
— 

— 
— 
— 
— 

    3,055,394 
— 
— 
    9,291,421 

  $

3,055 
— 
— 
9,291 

    18,329,310 
305,205 
— 
  $ 28,037,889 

— 
— 

    18,332,365 
305,205 
    (16,554,872)     (16,554,872)
  $(18,427,780)   $ 9,619,400 

The accompanying notes are an integral
part of these financial statements.

F-5

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
   
   
   
   
   
   
   
   
   
  
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
 
 
 
Monopar Therapeutics Inc.
Statement of Cash Flows

Cash flows from operating activities:
Net loss
Adjustments to reconcile net loss to net cash used in operating activities:

Stock compensation expense (non-cash)
In process research and development (non-cash)

Changes in operating assets and liabilities, net
Prepaid expenses and other current assets
Accounts payable and accrued expenses
Net cash used in operating activities

Cash flows from financing activities:

Proceeds from sale of Series A Preferred Stock, net of $12,500 of issuance costs
Cash received from Gem, net of $169,257 of transaction costs
Proceeds from the sale of common stock, net of $32,400 of issuance costs
Net cash provided by financing activities
Net increase in cash, cash equivalents and restricted cash
Cash, cash equivalents and restricted cash at beginning of period
Cash, cash equivalents and restricted cash at end of period
Supplemental disclosure of non-cash items for cash flow information:
    Value of shares issued in Gem transaction

The accompanying notes are an integral
part of these financial statements.

F-6

December 31,

2017

2016

  $(16,554,872)   $ (1,185,597)

305,205 
    13,501,622 

— 
— 

(126,780)    
247,357 

298 
(9,333)
(2,627,468)     (1,194,632)

— 
4,830,743 
4,705,646 
9,536,389 
6,908,921 
2,873,004 
  $ 9,781,925 

    1,262,500 
— 
— 
    1,262,500 
67,868 
    2,805,136 
  $ 2,873,004 

    18,332,365 

- 

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
  
   
  
   
   
   
   
  
   
  
   
   
   
   
   
  
   
  
   
   
   
   
   
   
   
   
   
   
  
   
  
   
 
 
 
MONOPAR THERAPEUTICS INC.
NOTES TO FINANCIAL STATEMENTS
December 31, 2017

Note 1 -    Nature of Business and Liquidity

Nature of Business

Monopar  Therapeutics  Inc.  (the  ”Company”)  is  an  emerging  biopharmaceutical  company  focused  on  developing  innovative  drug
candidates  to  improve  clinical  outcomes  in  cancer  patients.  Monopar  currently  has  three  compounds  in  development:  Validive®
(clonidine mucobuccal tablet; clonidine MBT), a Phase 3-ready, first-in-class mucoadhesive local anti-inflammatory tablet for the
prevention and treatment of radiation induced severe oral mucositis (“SOM”) in oropharyngeal cancer patients; MNPR-201 (GPX-
150; 5-imino-13-deoxydoxorubicin), a proprietary topoisomerase-II-alpha targeted analog of doxorubicin engineered specifically to
retain  the  anticancer  activity  while  minimizing  toxic  effects  on  the  heart;  and  MNPR-101  (formerly  huATN-658),  a  near-to-the-
clinic humanized monoclonal antibody, which targets the urokinase plasminogen activator receptor (“uPAR”), for the treatment of
advanced solid cancers.

The Company was originally formed in the State of Delaware on December 5, 2014 as a limited liability company (“LLC”) and on
December 16, 2015 converted to a C Corporation in a tax-free exchange. In March 2017, the Company’s Series A Preferred Stock
and Series Z Preferred Stock converted into common stock at a conversion rate of 1.2 for 1 and 1 for 1, respectively, along with a
concurrent common stock split of 70 for 1 which eliminated all shares of Series A Preferred Stock and Series Z Preferred Stock. All
references to common stock authorized, issued and outstanding and common stock options take into account the 70 for 1 stock split.

Liquidity

The Company has incurred an accumulated loss of approximately $18.4 million as of December 31, 2017. To date, the Company
has primarily funded its operations with the net proceeds from private placements of convertible preferred stock and common stock
and  from  the  cash  provided  in  the  Gem  transaction  discussed  in  detail  in  Note  6  below.  Management  believes  that  currently
available resources will provide sufficient funds to enable the Company to meet its minimum obligations through March 2019. The
Company’s  ability  to  fund  its  future  operations,  including  the  clinical  development  of  Validive,  is  dependent  primarily  upon  its
ability to execute on its business strategy and obtain additional funding or execute collaboration research transactions. There can be
no certainty that future financing or collaborative research transactions will occur.

Note 2 - Significant Accounting Policies

Basis of Presentation

These  financial  statements  include  the  books  of  Monopar  Therapeutics  Inc.,  its  French  branch  and  its  wholly-owned  French
subsidiary, Monopar Therapeutics, SARL and have been prepared in accordance with accounting principles generally accepted in
the United States (“GAAP”) and include all disclosures required by GAAP for financial reporting. The principal accounting policies
applied in the preparation of these financial statements are set out below and have been consistently applied in all periods presented.
The Company has been primarily involved in performing research activities, developing product technologies, and raising capital to
support and expand these activities.

Comprehensive Loss

Comprehensive  loss  represents  net  loss  plus  any  gains  or  losses  not  reported  in  the  statements  of  operations,  such  as  foreign
currency translations gains and losses that are typically reflected on a company’s statements of stockholders’ equity. There were no
differences between net loss for the years ended December 31, 2017 and 2016, and comprehensive loss for those periods.

F-7

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
MONOPAR THERAPEUTICS INC.
NOTES TO FINANCIAL STATEMENTS
December 31, 2017

Use of Estimates

The  preparation  of  financial  statements  in  conformity  with  GAAP  requires  management  to  make  estimates  and  assumptions  that
affect the reported amounts of assets and liabilities, disclosure of contingent assets and liabilities, and reported amounts of revenues
and expenses in the financial statements and accompanying notes. Actual results could differ from those estimates.

Going Concern Assessment

The Company adopted Accounting Standards Updates (“ASU”) 2014-15,  Disclosure of Uncertainties about an Entity’s Ability to
Continue  as  a  Going  Concern,  which  the  Financial  Accounting  Standards  Board  (“FASB”)  issued  to  provide  guidance  on
determining when and how reporting companies must disclose going-concern uncertainties in their financial statements. The ASU
requires  management  to  perform  interim  and  annual  assessments  of  an  entity’s  ability  to  continue  as  a  going  concern  within  one
year of the date of issuance of the entity’s financial statements (or within one year after the date on which the financial statements
are available to be issued, when applicable). Further, a company must provide certain disclosures if there is “substantial doubt about
the  entity’s  ability  to  continue  as  a  going  concern.”  In  February  2018,  the  Company  analyzed  its  minimum  cash  requirements
through March 2019 and has determined that, based upon the Company’s current available cash, the Company has no substantial
doubt about its ability to continue as a going concern.

Cash Equivalents

The Company considers all highly liquid investments purchased with an original maturity of 90 days or less to be cash equivalents.
Cash equivalents as of December 31, 2017 and December 31, 2016 consist entirely of money market accounts.

Restricted Cash

On July 9, 2015, the Company entered into a Clinical Trial and Option Agreement (“CTOA”) with Cancer Research UK. Pursuant
to the CTOA, the Company deposited $0.8 million into an escrow account to cover certain future indemnities, claims or potential
termination costs incurred by Cancer Research UK. Restricted cash was $0.8 million as of December 31, 2017 and December 31,
2016.

Prepaid Expenses

Prepayments  are  expenditures  for  goods  or  services  before  the  goods  are  used  or  the  services  are  received  and  are  charged  to
operations as the benefits are realized. Prepaid expenses include insurance premiums and software costs that are expensed monthly
over the life of the contract and prepaid legal patent fees that will be expensed as incurred.

Concentration of Credit Risk

Financial instruments that potentially subject the Company to concentration of credit risk consist of cash and cash equivalents and
restricted  cash.  The  Company  maintains  cash  and  cash  equivalents  at  one  financial  institution  and  restricted  cash  at  another
financial institution. As of December 31, 2017, and December 31, 2016, cash and cash equivalents and restricted cash balances at
these two financial institutions were in excess of the $250,000 Federal Deposit Insurance Corporation (“FDIC”) insurable limit.

Fair Value of Financial Instruments

For financial instruments consisting of cash and cash equivalents, prepaid expenses, deferred offering costs, accounts payable and
accrued expenses, the carrying amounts are reasonable estimates of fair value due to their relatively short maturities.

F-8

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
MONOPAR THERAPEUTICS INC.
NOTES TO FINANCIAL STATEMENTS
December 31, 2017

The Company adopted Accounting Standard Codification  (“ASC”) 820, Fair Value Measurements and Disclosures,  as  amended,
addressing the measurement of the fair value of financial assets and financial liabilities. Under this standard, fair value is defined as
the price that would be received to sell an asset or paid to transfer a liability (i.e., the “exit price”) in an orderly transaction between
market participants at the measurement date.

In determining fair values of all reported assets and liabilities that represent financial instruments, the Company uses the carrying
market values of such amounts. The standard establishes a hierarchy for inputs used in measuring fair value that maximizes the use
of  observable  inputs  and  minimizes  the  use  of  unobservable  inputs  by  requiring  that  the  most  observable  inputs  be  used  when
available. Observable inputs reflect assumptions market participants would use in pricing an asset or liability based on market data
obtained from independent sources. Unobservable inputs reflect a reporting entity’s pricing an asset or liability developed based on
the best information available in the circumstances. The fair value hierarchy consists of the following three levels:

Level 1 - instrument valuations are obtained from real-time quotes for transactions in active exchange markets involving identical
assets.

Level 2 - instrument valuations are obtained from readily-available pricing sources for comparable instruments.

Level 3 - instrument valuations are obtained without observable market values and require a high-level of judgment to determine
the fair value.

Determining which category an asset or liability falls within the hierarchy requires significant judgment. The Company evaluates its
hierarchy disclosures each reporting period. There were no transfers between Level 1, 2 or 3 of the fair value hierarchy during the
years ended December 31, 2017 and 2016. The following table presents the assets and liabilities recorded that are reported at fair
value on our balance sheets on a recurring basis.

Assets and Liabilities Measured at Fair Value on a Recurring Basis

December 31, 2017

Level 1

Level 2

Total

Assets
Cash equivalents(1)
Restricted cash(2)
Total

  $ 8,872,982 
31 
  $ 8,873,013 

  $

  $

- 
800,000 
800,000 

  $ 8,872,982 
800,031 
  $ 9,673,013 

(1) Cash equivalents represent the fair value of the Company’s investments in two money market accounts at December 31, 2017.
(2) Restricted cash represents the fair value of the Company’s investments in an $800,000 certificate of deposit and $31 in a money

market account at December 31, 2017.

December 31, 2016

Level 1

Level 2

Total

Assets
Cash equivalents(1)
Restricted cash(2)
Total

  $ 2,009,018 
393 
  $ 2,009,411 

  $

  $

- 
800,000 
800,000 

  $ 2,009,018 
800,393 
  $ 2,809,411 

(1)         Cash equivalents represent the fair value of the Company’s investments in a money market account at December 31, 2016.
Restricted cash represents the fair value of the Company’s investments in an $800,000 certificate of deposit and $393 in a
(2) 
money market account at December 31, 2016.

Net Loss per Share

Net  loss  per  share  for  the  year  ended  December  31,  2017  is  calculated  by  dividing  net  loss  by  the  weighted-average  shares  of
common  stock  outstanding  during  the  period.  Diluted  net  loss  per  share  for  the  year  ended  December  31,  2017  is  calculated  by
dividing net loss by the weighted-average shares of common stock outstanding and potential

F-9

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
   
   
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
   
   
 
 
 
 
 
MONOPAR THERAPEUTICS INC.
NOTES TO FINANCIAL STATEMENTS
December 31, 2017

shares  of  common  stock  during  the  period. As  of  December  31,  2017,  potentially  dilutive  securities  included  658,592  options  to
purchase common stock.

During the year ended December 31, 2016 there were no shares of common stock outstanding.

Research and Development Expenses

Research  and  development  (“R&D”)  costs  are  expensed  as  incurred.  Major  components  of  research  and  development  expenses
include  salaries  and  benefits  paid  to  the  Company’s  R&D  staff,  fees  paid  to  consultants  and  to  the  entities  that  conduct  certain
development activities on the Company’s behalf and materials and supplies.

The  Company  accrues  and  expenses  the  costs  for  clinical  trial  activities  performed  by  third  parties  based  upon  estimates  of  the
percentage of work completed over the life of the individual study in accordance with agreements established with contract research
organizations and clinical trial sites. The Company determines the estimates through discussions with internal clinical personnel and
external  service  providers  as  to  progress  or  stage  of  completion  of  trials  or  services  and  the  agreed  upon  fee  to  be  paid  for  such
services. Costs of setting up clinical trial sites for participation in the trials are expensed immediately as research and development
expenses.  Clinical  trial  site  costs  related  to  patient  enrollment  are  accrued  as  patients  are  entered  into  the  trial.  During  the  year
ended December 31, 2017 and 2016, the Company had no clinical trials in progress.

In-process Research and Development

In-process research and development expense represents the costs to acquire technologies to be used in research and development
that have not reached technological feasibility, have no alternative future uses and thus are expensed as incurred. IPR&D expense
also  includes  upfront  license  fees  and  milestones  paid  to  collaborators,  with  no  alternative  use,  which  are  expensed  as  goods  are
received or services rendered.

Collaborative Arrangements

The  Company  and  its  collaborative  partner  are  active  participants  in  a  collaborative  arrangement  and  all  parties  are  exposed  to
significant risks and rewards depending on the technical and commercial success of the activities. Contractual payments to the other
party  in  the  collaboration  agreement  and  costs  incurred  by  the  Company  when  the  Company  is  deemed  to  be  the  principal
participant  for  a  given  transaction  are  recognized  on  a  gross  basis  in  research  and  development  expenses.  Royalties  and  license
payments are recorded as earned.

During the years ended December 31, 2017 and 2016, no milestones were met and no royalties were earned, therefore, the Company
did not pay or accrue/expense any milestone or royalty payments.

Licensing Agreements

The  Company  has  various  agreements  to  license  technology  utilized  in  the  development  of  its  programs.  The  licenses  contain
success milestone obligations and royalties on future sales. During the year ended December 31, 2017 and 2016, no milestones were
met and no royalties were earned, therefore, the Company did not pay or accrue/expense any milestone or royalty payments under
any of its license agreements.

Patent Costs

The  Company  expenses  costs  relating  to  issued  patents  and  patent  applications,  including  costs  relating  to  legal,  renewal  and
application fees, as a component of general and administrative expenses in its statements of operations.

F-10

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
MONOPAR THERAPEUTICS INC.
NOTES TO FINANCIAL STATEMENTS
December 31, 2017

Income Taxes

From December 2014 to December 16, 2015, the Company was an LLC taxed as a partnership under the Internal Revenue Code,
during  which  period  the  members  separately  accounted  for  their  pro-rata  share  of  income,  deductions,  losses,  and  credits  of  the
Company. On December 16, 2015, the Company converted from an LLC to a C Corporation. Beginning on December 16, 2015, the
Company  uses  an  asset  and  liability  approach  for  accounting  for  deferred  income  taxes,  which  requires  recognition  of  deferred
income  tax  assets  and  liabilities  for  the  expected  future  tax  consequences  of  events  that  have  been  recognized  in  its  financial
statements,  but  have  not  been  reflected  in  its  taxable  income.  Estimates  and  judgments  occur  in  the  calculation  of  certain  tax
liabilities  and  in  the  determination  of  the  recoverability  of  certain  deferred  income  tax  assets,  which  arise  from  temporary
differences  and  carry  forwards.  Deferred  income  tax  assets  and  liabilities  are  measured  using  the  currently  enacted  tax  rates  that
apply to taxable income in effect for the years in which those tax assets and liabilities are expected to be realized or settled.

The Company regularly assesses the likelihood that its deferred income tax assets will be realized from recoverable income taxes or
recovered from future taxable income. To the extent that the Company believes any amounts are more likely not to be realized, the
Company records a valuation allowance to reduce the deferred income tax assets. In the event the Company determines that all or
part  of  the  net  deferred  tax  assets  are  not  realizable  in  the  future,  an  adjustment  to  the  valuation  allowance  would  be  charged  to
earnings in the period such determination is made. Similarly, if the Company subsequently realizes deferred income tax assets that
were previously determined to be unrealizable, the respective valuation allowance would be reversed, resulting in an adjustment to
earnings in the period such determination is made.

Internal Revenue Code Section 382 provides that, after an ownership change, the amount of a loss corporation’s net operating loss
(“NOL”) for any post-change year that may be offset by pre-change losses shall not exceed the section 382 limitation for that year.
Because the Company will continue to raise equity in the coming years, section 382 may limit the Company’s usage of NOLs in the
future.

Based on the available evidence, the Company believed it was not likely to utilize its minimal deferred tax assets in the future and
as a result, the Company recorded a full valuation allowance as of December 31, 2017 and 2016. The Company intends to maintain
the valuation allowance until sufficient evidence exists to support their reversal. The Company regularly reviews its tax positions
and for a tax benefit to be recognized, the related tax position must be more likely than not to be sustained upon examination. Any
amount recognized is generally the largest benefit that is more likely than not to be realized upon settlement. The Company’s policy
is  to  recognize  interest  and  penalties  related  to  income  tax  matters  as  an  income  tax  expense.  For  the  years  ended  December  31,
2017 and 2016, the Company did not have any interest or penalties associated with unrecognized tax benefits.

The Company is subject to U.S. Federal, Illinois and California income taxes. Tax regulations within each jurisdiction are subject to
the interpretation of the related tax laws and regulations and require significant judgment to apply. The Company was incorporated
on  December  16,  2015  and  is  subject  to  U.S.  Federal,  state  and  local  tax  examinations  by  tax  authorities  for  the  years  ended
December  31,  2017  and  2016  and  for  the  short  tax  period  December  16,  2015  to  December  31,  2015.  The  Company  does  not
anticipate significant changes to its current uncertain tax positions through December 31, 2017. The Company plans on filing its tax
returns for the year ending December 31, 2017 prior to the filing deadlines in all jurisdictions.

F-11

 
 
 
 
 
 
 
 
 
 
MONOPAR THERAPEUTICS INC.
NOTES TO FINANCIAL STATEMENTS
December 31, 2017

Stock-Based Compensation

The Company accounts for stock-based compensation arrangements with employees, nonemployee directors and consultants using a
fair value method, which requires the recognition of compensation expense for costs related to all stock-based payments, including
stock options. The fair value method requires the Company to estimate the fair value of stock-based payment awards on the date of
grant using an option pricing model.

Stock-based  compensation  costs  for  options  granted  to  employees  and  nonemployee  directors  are  based  on  the  fair  value  of  the
underlying option calculated using the Black-Scholes option-pricing model on the date of grant for stock options and recognized as
expense on a straight-line basis over the requisite service period, which is the vesting period. Determining the appropriate fair value
model and related assumptions requires judgment, including estimating stock price volatility, forfeiture rates and expected term. The
expected volatility rates are estimated based on the actual volatility of comparable public companies over the expected term. The
Company  selected  these  companies  based  on  comparable  characteristics,  including  enterprise  value,  risk  profiles,  stage  of
development and with historical share price information sufficient to meet the expected life of the stock-based awards. The expected
term for options granted to date is estimated using the simplified method. Forfeitures are estimated at the time of grant and revised,
if necessary, in subsequent periods if actual forfeitures differ from those estimates. The Company has not paid dividends and does
not anticipate paying a cash dividend in the future vesting period and, accordingly, uses an expected dividend yield of zero. The
risk-free interest rate is based on the rate of U.S. Treasury securities with maturities consistent with the estimated expected term of
the awards. The measurement of consultant share-based compensation is subject to periodic adjustments as the underlying equity
instruments vest and is recognized as an expense over the period over which services are rendered.

Recent Accounting Pronouncements

In August 2014, FASB issued ASU 2014-15, Disclosure of Uncertainties about an Entity’s Ability to Continue as a Going Concern,
which  provides  guidance  on  determining  when  and  how  reporting  companies  must  disclose  going-concern  uncertainties  in  their
financial statements. The ASU requires management to perform interim and annual assessments of an entity’s ability to continue as
a  going  concern  within  one  year  of  the  date  of  issuance  of  the  entity’s  financial  statements  (or  within  one  year  after  the  date  on
which the financial statements are available to be issued, when applicable). Further, a company must provide certain disclosures if
there is “substantial doubt about the entity’s ability to continue as a going concern.” This ASU became effective for annual periods
ending after December 15, 2016 and interim periods within annual periods beginning after December 15, 2016. The Company has
adopted this new accounting standard in its financial statements and footnote disclosures.

In  November  2015,  the  FASB  issued  ASU  2015-17,  Balance  Sheet  Classification  of  Deferred  Taxes.  This  is  part  of  FASB’s
simplification initiative. The amendments in this ASU require that deferred tax liabilities and assets be classified as noncurrent in a
classified statement of financial position. This ASU became effective for the Company in the first quarter of 2017. The Company
has adopted this ASU and determined that it does not have a material effect on its financial condition and results of operations for
the year ended December 31, 2017.

In January 2016, the FASB issued ASU 2016-01,  Recognition and Measurement of Financial Assets and Financial Liabilities. The
purpose  is  to  enhance  the  reporting  model  for  financial  instruments  to  provide  users  of  financial  statements  with  more  decision-
useful information. This ASU is effective for the Company in the first quarter of 2018. Early adoption is not permitted except for
limited provisions. The Company does not expect the adoption of this amendment to have a material effect on its financial condition
and results of operations.

F-12

 
 
 
 
 
 
 
 
 
 
 
MONOPAR THERAPEUTICS INC.
NOTES TO FINANCIAL STATEMENTS
December 31, 2017

In February 2016, the FASB issued ASU 2016-02,  Leases, which for operating leases, requires a lessee to recognize a right-of-use
asset  and  a  lease  liability,  initially  measured  at  the  present  value  of  the  lease  payments,  in  its  balance  sheet.  The  standard  also
requires a lessee to recognize a single lease cost, calculated so that the cost of the lease is allocated over the lease term, generally on
a straight-line basis. ASU 2016-02 will be effective for the Company in the first quarter of 2019, and early adoption is permitted.
The Company is currently assessing the impact that adopting this new accounting standard will have on its financial statements and
footnote disclosures.

In  March  2016,  the  FASB  issued ASU  2016-09,  Improvements  to  Employee  Share-Based  Payment  Accounting,  which  simplifies
several  aspects  of  the  accounting  for  employee  share-based  payment  transactions  for  both  public  and  nonpublic  companies,
including the accounting for income taxes, forfeitures, and statutory tax withholding requirements, as well as classification in the
statement of cash flows. The ASU became effective for the Company in the first quarter of 2017. The Company has adopted this
ASU and determined that it does not have a material effect on its financial condition and results of operations for the year ended
December 31, 2017.

In November 2016, the FASB issued ASU 2016-18,  Statement of Cash Flows (Topic 230):Restricted Cash. The amendments apply
to  all  entities  that  have  restricted  cash  or  restricted  cash  equivalents  and  are  required  to  present  a  statement  of  cash  flows.  The
amendments  address  diversity  in  practice  that  exists  in  the  classification  and  presentation  of  changes  in  restricted  cash  on  the
statement of cash flows. The amendments require that a statement of cash flows explain the change during the period in the total of
cash,  cash  equivalents,  and  amounts  generally  described  as  restricted  cash  or  restricted  cash  equivalents. As  a  result,  amounts
generally  described  as  restricted  cash  and  restricted  cash  equivalents  should  be  included  with  cash  and  cash  equivalents  when
reconciling the beginning-of-period and end-of-period total amounts shown on the statement of cash flows. The amendments do not
provide a definition of restricted cash or restricted cash equivalents. The amendments are effective for public business entities for
fiscal years beginning after December 15, 2017, and interim periods within those fiscal years. For all other entities, the amendments
are effective for fiscal years beginning after December 15, 2018, and interim periods within fiscal years beginning after December
15, 2019. Early adoption is permitted. The Company has early adopted the amendments and has applied them using a retrospective
transition method to each period presented. Therefore, the Company has included restricted cash in cash equivalents and restricted
cash on its statements of cash flows for the years ended December 31, 2017 and 2016.

In January 2017, the FASB issued ASU No. 2017-01,  Business Combinations (Topic 805): Clarifying the Definition of a Business
(“ASU  No.  2017-01”).  The  amendments  in ASU  No.  2017-01  clarify  the  definition  of  a  business  with  the  objective  of  adding
guidance to assist entities with evaluating whether transactions should be accounted for as acquisitions (or disposals) of assets or
businesses.  The  definition  of  a  business  affects  many  areas  of  accounting  including  acquisitions,  disposals,  goodwill  and
consolidation.  For  public  companies,  the  amendments  are  effective  for  annual  periods  beginning  after  December  15,  2017,
including interim periods within those periods. For all other companies and organizations, the amendments are effective for annual
periods  beginning  after  December  15,  2018,  and  interim  periods  within  annual  periods  beginning  after  December  15,  2019.  The
Company  is  currently  assessing  the  impact  that  adopting  this  new  accounting  standard  will  have  on  its  financial  statements  and
footnote disclosures.

In  May  2017,  the  FASB  issued  ASU  No.  2017-09,  Compensation-Stock  Compensation  (Topic  718):  Scope  of  Modification
Accounting.  The  amendment  amends  the  scope  of  modification  accounting  for  share-based  payment  arrangements,  provides
guidance on the types of changes to the terms or conditions of share-based payment awards to which an entity would be required to
apply modification accounting under ASC 718. This ASU is effective for all entities for annual periods, and interim periods within
those annual periods, beginning after December 15, 2017. Early adoption is permitted, including adoption in any interim period for:
(a) public business entities for reporting periods for which financial statements have not yet been issued, and (b) all other entities
for  reporting  periods  for  which  financial  statements  have  not  yet  been  made  available  for  issuance.  The  Company  is  currently
assessing the impact that adopting this new accounting standard will have on its financial statements and footnote disclosures.

F-13

 
 
 
 
 
 
 
 
 
MONOPAR THERAPEUTICS INC.
NOTES TO FINANCIAL STATEMENTS
December 31, 2017

In July 2017, the FASB issued ASU No. 2017-11,  Earnings Per Share (Topic 260) Distinguishing Liabilities from Equity (Topic
480) Derivatives and Hedging (Topic 815) (Part I) Accounting for Certain Financial Instruments with Down Round Features, (Part
II)  Replacement  of  the  Indefinite  Deferral  for  Mandatorily  Redeemable  Financial  Instruments  of  Certain  Nonpublic  Entities  and
Certain Mandatorily Redeemable Noncontrolling Interests with a Scope Exception. This ASU simplifies the accounting for certain
financial  instruments  with  down  round  features,  a  provision  in  an  equity-linked  financial  instrument  (or  embedded  feature)  that
provides a downward adjustment of the current exercise price based on the price of future equity offerings. Down round features are
common in warrants, convertible preferred shares, and convertible debt instruments issued by private companies and development-
stage  public  companies.  This  new  ASU  requires  companies  to  disregard  the  down  round  feature  when  assessing  whether  the
instrument is indexed to its own stock, for purposes of determining liability or equity classification. The provisions of this new ASU
related  to  down  rounds  are  effective  for  public  business  entities  for  fiscal  years,  and  interim  periods  within  those  fiscal  years,
beginning after December 15, 2018. For all other entities, the amendments are effective for fiscal years beginning after December
15, 2019, and interim periods within fiscal years beginning after December 15, 2020. Early adoption is permitted for all entities.
The Company is currently assessing the impact that adopting this new accounting standard will have on its financial statements and
footnote disclosures.

Note 3 - Capital Stock

On December 16, 2015, the Company converted from an LLC to a C Corporation at which time the Company effected a 1 for 10
reverse  stock  split. All  references  to  preferred  stock  authorized,  issued  and  outstanding  and  common  stock  authorized  take  into
account  the  1  for  10  reverse  stock  split.  In  March  2017,  the  Company’s  Series A  Preferred  Stock  and  Series  Z  Preferred  Stock
converted to common stock at a conversion rate of 1.2 for 1 and 1 for 1, respectively, along with a simultaneous common stock split
of 70 for 1 and the elimination all shares of Series A Preferred Stock and Series Z Preferred Stock (collectively, the “Conversion”).
100,000 shares of Series Z Preferred Stock were converted into 7,000,000 shares of common stock and 15,894 shares of Series A
Preferred  Stock  were  converted  into  1,335,079  shares  of  common  stock. All  references  to  common  stock  authorized,  issued  and
outstanding and common stock options take into account the 70 for 1 stock split.

Holders  of  the  common  stock  are  entitled  to  receive  such  dividends  as  may  be  declared  by  the  Board  of  Directors  out  of  funds
legally available therefor. Upon dissolution and liquidation of the Company, holders of the common stock are entitled to a ratable
share of the net assets of the Company remaining after payments to creditors of the Company. The holders of shares of common
stock are entitled to one vote per share for the election of directors and on all other matters submitted to a vote of stockholders.

The Company’s amended and restated certificate of incorporation authorizes the Company to issue 40,000,000 shares of common
stock with a par value of $0.001 per share.

Contribution to Capital

In August  2017,  the  Company’s  largest  stockholder,  Tactic  Pharma,  LLC  (“Tactic  Pharma”),  surrendered  2,888,727.12  shares  of
common  stock  back  to  the  Company  as  a  contribution  to  the  capital  of  the  Company.  This  resulted  in  reducing  Tactic  Pharma’s
ownership in Monopar from 79.5% to 69.9%.

Sales of Common Stock

Pursuant to an active private placement memorandum, during the period from July 1, 2017 through September 30, 2017, Monopar
sold  448,834  shares  of  common  stock  at  $6  per  share  for  proceeds  of  approximately  $2.7  million.  This  financing  closed  on
September 30, 2017.

F-14

 
 
 
 
 
 
 
 
 
 
 
 
 
MONOPAR THERAPEUTICS INC.
NOTES TO FINANCIAL STATEMENTS
December 31, 2017

Issuance of Common Stock in the Gem Transaction

Pursuant to the Gem Transaction, discussed in detail in Note 6 below, the Company issued 3,055,394.12 shares of its common stock
in exchange for cash and intellectual property related to GPX-150 (renamed MNPR-201).

As  of  December  31,  2017,  the  Company  had  9,291,420.614  shares  of  common  stock  issued  and  outstanding.  The  Company  no
longer has any shares of preferred stock authorized or outstanding.

In April 2016, the Company adopted the 2016 Stock Incentive Plan and the Company’s Board of Directors reserved 700,000 shares
of common stock for issuances under the plan (as adjusted subsequent to the Conversion). In October 2017, the Company’s Board
of Directors increased the stock option pool to 1,600,000 shares of common stock.

Note 4 - Stock Option Plan

In  April  2016,  the  Company’s  Board  of  Directors  and  the  convertible  preferred  stockholders  representing  a  majority  of  the
Company’s  outstanding  stock  approved,  the  Monopar  Therapeutics  Inc.  2016  Stock  Incentive  Plan  (the  “Plan”)  allowing  the
Company to grant up to an aggregate 700,000 shares of stock awards, stock options, stock appreciation rights and other stock-based
awards  to  employees,  directors  and  consultants.  Concurrently,  the  Board  of  Directors  granted  to  certain  Board  members  and  the
Company’s acting chief financial officer stock options to purchase up to an aggregate 273,000 shares of the Company’s common
stock at an exercise price of $0.001 par value based upon a third-party valuation of the Company’s common stock.

In December 2016, the Board of Directors granted stock options to purchase up to 7,000 shares of the Company’s common stock at
an exercise price of $0.001 par value to the Company’s acting chief medical officer.

In February 2017, the Board of Directors granted to certain Board members and the Company’s acting chief financial officer stock
options to purchase up to an aggregate 275,520 shares of the Company’s common stock at an exercise price of $0.001 par value
based upon a third-party valuation of the Company’s common stock. In September 2017, the Board of Directors represented by the
designated Plan Administrator, granted options to purchase up to 21,024 shares of common stock to each of the three new Board
members at an exercise price of $6 per share based on the price per share at which common stock was sold in the Company’s most
recent private offering.

Under the Plan, the per share exercise price for the shares to be issued upon exercise of an option shall be determined by the Plan
administrator, except that the per share exercise price shall be no less than 100% of the fair market value per share on the grant date.
Fair  market  value  is  established  by  the  Company’s  Board  of  Directors,  using  third  party  valuation  reports  and  recent  financings.
Options generally expire after ten years.

F-15

 
 
 
 
 
 
 
 
 
 
 
 
 
MONOPAR THERAPEUTICS INC.
NOTES TO FINANCIAL STATEMENTS
December 31, 2017

Stock option activity under the Plan was as follows:

Balances at January 1, 2016
Initial option pool
Granted (1)
Forfeited
Exercised
Balances at December 31, 2016
Option pool increase (2)
Granted (3)
Forfeited
Exercised
Balances at December 31, 2017

Options Outstanding

Options
Available

Number
ofOptions

Weighted-
Average
Exercise
Price

— 
700,000 
(280,000)    

— 
— 
420,000 
900,000 
(378,592)    

— 
— 
941,408 

— 

  $

— 

280,000 
— 
— 
280,000 
— 
378,592 
— 
— 
658,592 

0.001 
— 
— 
0.001 
— 
1.63 
— 
— 
0.94 

(1) 273,000  options  vested  50%  upon  grant  date,  25%  upon  the  6-month  anniversary  of  grant  date  and  25%  upon  the  1-year

anniversary of grant date; 7,000 options vested monthly over 6 months.

(2) In October 2017, the Company’s Board of Directors increased the option pool to 1,600,000 shares.

(3) 336,544  options  vest  6/48ths  at  the  six-month  anniversary  of  grant  date  and  1/48th  per  month  thereafter  21,024  options  vest
6/24ths on the six-month anniversary of grant date and 1/24th per month thereafter; and 21,024 options vest 6/42nds on the six-
month anniversary of grant date and 1/42nd per month thereafter.

A summary of options outstanding as of December 31, 2017 is shown below:

Exercise Prices

  $
  $

0.001 
6.00 

Numberof Shares
Outstanding

Weighted Average
Remaining Contractual
Term

Number of Shares
Fully Vested and
Exercisable

555,520 
103,072 
658,592 

 8.7 years  
 9.6 years  

337,400 
— 
337,400 

Weighted Average
Remaining

Contractual Term  

 8.4 years

N/A 

During  the  years  ended  December  31,  2017  and  2016,  the  Company  recognized  $26,864  and  $0  of  employee  and  non-employee
director  stock-based  compensation  expense  as  general  and  administrative  expenses,  respectively,  and  $26,499  and  $0  as  research
and development expenses, respectively. The compensation expense is allocated on a departmental basis, based on the classification
of the option holder. No income tax benefits have been recognized in the statements of operations for stock-based compensation
arrangements.

F-16

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
   
   
   
  
   
  
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
   
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
  
 
 
 
MONOPAR THERAPEUTICS INC.
NOTES TO FINANCIAL STATEMENTS
December 31, 2017

The Company recognizes as an expense the fair value of options granted to persons who are neither employees nor directors. The
fair  value  of  expensed  options  was  based  on  the  Black-Scholes  option-pricing  model  assuming  the  following  factors:  6.1  to  5.3
years expected term, 57% volatility, 2.2% to 1.2% risk free interest rate and zero dividends.  The expected term for options granted
to  date  is  estimated  using  the  simplified  method.  Stock-based  compensation  expense  for  non-employees  for  the  years  ended
December 31, 2017 and 2016 was $251,842 and $0, respectively, of which $199,769 and $0, respectively was recorded as research
and development expenses and $52,073 and $0, respectively, as general and administrative expenses. For the years ended December
31, 2017 and 2016: the weighted average grant date fair value was $0.88 and $0.00 per share, respectively; and the fair value of
shares vested were approximately $0.3 million and nominal, respectively.  At December 31, 2017, the aggregate intrinsic value was
approximately $3.3 million of which approximately $2.0 million was vested and approximately $1.3 million is expected to vest and
the weighted average exercise price in aggregate was $0.94 which includes $0.001 for fully vested stock options and $1.93 for stock
options  expected  to  vest. At  December  31,  2017  unamortized  unvested  balance  of  stock  base  compensation  was  $925,126,  to  be
amortized over 3.3 years.

Note 5 - Development and Collaboration Agreements

Onxeo SA

The  pre-negotiated  Onxeo  license  agreement  for  Validive  included  as  part  of  the  option  agreement  includes  clinical,  regulatory,
developmental  and  sales  milestones  that  could  reach  up  to  $108  million  if  the  Company  achieves  all  milestones,  and  escalating
royalties on net sales from 5 - 10%. On September 8, 2017, the Company exercised the option, and therefore was required to pay
Onxeo the $1 million fee under the option and license agreement.

Under  the  agreement,  the  Company  is  required  to  pay  royalties  to  Onxeo  on  a  product-by-product  and  country-by-country  basis
until  the  later  of  (1)  the  date  when  a  given  product  is  no  longer  within  the  scope  of  a  patent  claim  in  the  country  of  sale  or
manufacture, (2) the expiry of any extended exclusivity period in the relevant country (such as orphan drug exclusivity, pediatric
exclusivity, new chemical entity exclusivity, or other exclusivity granted beyond the expiry of the relevant patent), or (3) a specific
time period after the first commercial sale of the product in such country. In most countries, including the U.S., the patent term is
generally 20 years from the earliest claimed filing date of a non-provisional patent application in the applicable country, not taking
into  consideration  any  potential  patent  term  adjustment  that  may  be  filed  in  the  future  or  any  regulatory  extensions  that  may  be
obtained. The royalty termination provision pursuant to (3) described above is shorter than 20 years and is the least likely cause of
termination of royalty payments.

The  Onxeo  license  agreement  does  not  have  a  pre-determined  term,  but  expires  on  a  product-by-product  and  country-by-country
basis; that is, the agreement expires with respect to a given product in a given country whenever the Company’s royalty payment
obligations with respect to such product have expired. The agreement may also be terminated early for cause if either the Company
or Onxeo materially breach the agreement, or if either the Company or Onxeo become insolvent. The Company may also choose to
terminate  the  agreement,  either  in  its  entirety  or  as  to  a  certain  product  and  a  certain  country,  by  providing  Onxeo  with  advance
notice.

The  Company  plans  to  internally  develop  Validive  with  the  near-term  goal  of  commencing  a  Phase  3  clinical  trial,  which,  if
successful,  may  allow  the  Company  to  apply  for  marketing  approval  within  the  next  few  years.  The  Company  will  need  to  raise
significant funds to support the further development of Validive.

Cancer Research UK

In May 2015, the Company entered into a CTOA with Cancer Research UK and Cancer Research Technology Limited, a wholly-
owned subsidiary of Cancer Research UK. As part of the CTOA, the Company was obligated to submit $0.8 million in escrow to
cover certain potential future claims, intellectual property infringement costs or termination costs incurred by Cancer Research UK.
Pursuant to this agreement Cancer Research UK conducted preclinical work, improved the manufacturing, and planned to conduct a
Phase 1a/1b clinical trial in cancer patients. As part of a portfolio reprioritization review, on March 21, 2018 Cancer Research UK
notified the Company that it was terminating the CTOA and would work to transfer to the Company the data generated under the
CTOA.    The  Company  is  currently  reviewing  potential  alternative  collaboration  opportunities  for  MNPR-101  and  continues  to
maintain the program’s intellectual property portfolio.

F-17

 
 
 
 
 
 
 
 
 
 
 
 
 
MONOPAR THERAPEUTICS INC.
NOTES TO FINANCIAL STATEMENTS
December 31, 2017

XOMA Ltd.

The intellectual property rights contributed by Tactic Pharma to the Company included the non-exclusive license agreement with
XOMA  Ltd.  for  the  humanization  technology  used  in  the  development  of  MNPR-101.  Pursuant  to  such  license  agreement,  the
Company is obligated to pay XOMA Ltd. clinical, regulatory and sales milestones for MNPR-101 that could reach up to $14.925
million  if  the  Company  achieves  all  milestones.  The  agreement  does  not  require  the  payment  of  sales  royalties.  There  can  be  no
assurance that the Company will reach any milestones. As of December 31, 2017, the Company has not reached any milestones and
has not been required to pay XOMA Ltd. any funds under this license agreement.

Note 6 - The Gem Transaction

On August  25,  2017,  the  Company  executed  definitive  agreements  with  Gem  Pharmaceuticals,  LLC  (“Gem”),  pursuant  to  which
Gem formed a limited liability company, TacticGem LLC (“TacticGem”) with Tactic Pharma, the Company’s largest shareholder at
that time. Gem contributed certain of Gem’s drug candidates’ intellectual property and agreements associated primarily with Gem’s
GPX-150  (renamed  MNPR-201)  drug  candidate  program,  along  with  $5,000,000  in  cash  (the  “Gem  Contributed  Assets”)  to
TacticGem for a 42.633% interest, and Tactic Pharma contributed 4,111,272.88 shares of common stock of Monopar to TacticGem
for a 57.367% interest. Then, TacticGem contributed the Gem Contributed Assets to the  Company  in  exchange  for  3,055,394.12
newly  issued  shares  of  common  stock  of  the  Company  (31.4%  on  a  fully-diluted  basis)  (the  two  contributions  collectively,  the
“Gem  Transaction”).  The  Gem  Transaction  closed  on  August  25,  2017.  Following  the  Gem  Transaction,  TacticGem  owns
7,166,667 (77.1%) shares of Monopar’s common stock as of December 31, 2017.

The transaction was recorded as an asset acquisition on August 25, 2017 as follows:

Cash recorded on the Company’s Balance Sheet
Assembled Workforce recorded as In-process Research and Development Expense on
the Company’s Statement of Operations
MNPR-201 (GPX-150) recorded as In-process Research and Development Expense on
the Company’s Statement of Operations
Total Gem Transaction

  $ 5,000,000 

9,886 

    13,491,736 
  $18,501,622 

Within 90 days of the effective date of the transaction, the Company was required to use its best efforts to file a Form 10 to register
its common stock under the Securities Exchange Act of 1934. The Company filed its Form 10 on November 9, 2017. Additionally,
Arthur  Klausner,  current  CEO  of  Gem,  has  been  added  to  the  Company’s  Board  of  Directors  and  will  remain  on  the  Board  of
Directors at least until the Company achieves a listing on a major stock exchange (such as Nasdaq or NYSE). Richard Olson and
Gerald  Walsh,  CSO  and  President  of  Gem,  respectively,  have  been  retained  with  one-year  consulting  agreements  to  aid  in  an
efficient transfer of Gem’s GPX-150 (renamed MNPR-201) and associated programs.

It is anticipated that this transaction will increase the Company’s annual cash burn by at least $750,000, and will be significantly
higher if the Company chooses to conduct clinical trials with the Gem drug candidate programs.

F-18

 
 
 
 
 
 
 
  
 
   
 
 
 
 
MONOPAR THERAPEUTICS INC.
NOTES TO FINANCIAL STATEMENTS
December 31, 2017

Note 7 - Related Party Transactions

During the years ended December 31, 2017 and 2016, the Company was advised by four members of its Board of Directors, who
were  Managers  of  the  LLC  prior  to  the  Company’s  conversion  to  a  C  Corporation.  The  four  former  Managers  are  also  current
common stockholders (owning approximately an aggregate 3% of the common stock outstanding as of December 31, 2017). Three
of  the  former  Managers  are  also  Managing  Members  of  Tactic  Pharma  the  Company’s  largest  and  controlling  stockholder
(beneficially owning 46% of the Company at December 31, 2017 and in partnership with Gem through TacticGem owning 77%).
Monopar paid Managing Members of Tactic Pharma the following during the years ended December 31, 2017 and 2016: Chandler
D. Robinson, the Company’s Co-Founder, Chief Executive Officer, common stockholder, Managing Member of Tactic Pharma and
former Manager of the predecessor LLC $346,545 and $322,000, respectively; and Andrew P. Mazar, the Company’s Co-Founder,
Chief Scientific Officer, common stockholder, Managing Member of Tactic Pharma and former Manager of the predecessor LLC,
$300,731  and  $197,500,  respectively.  The  Company  also  paid  Christopher  M.  Starr,  the  Company’s  Co-Founder,  Executive
Chairman  of  the  Board  of  Directors,  common  stockholder  and  former  Manager  of  the  predecessor  LLC  $100,897  and  $96,339
during the years ended December 31, 2017 and 2016, respectively.

In the normal course of business, the Company’s Chief Executive Officer, Board Members and consultants incur expenses on behalf
of the Company and are reimbursed within 30 days of submission of relevant expense reports.

The Company reimbursed Tactic Pharma, a  de minimis amount in monthly storage fees during the years ended December 31, 2017
and 2016. In March 2017, Tactic Pharma wired $1 million to the Company in advance of the sale of the Company’s common stock
at $6 per share under a private placement memorandum. In April, the Company issued to Tactic Pharma 166,667 shares in exchange
for  the  $1  million  at  $6  per  share  once  the  Company  began  selling  stock  to  unaffiliated  parties  under  the  private  placement
memorandum.  In  August  2017,  Tactic  Pharma  surrendered  2,888,727  shares  of  common  stock  back  to  the  Company  as  a
contribution to the capital of the Company. This resulted in reducing Tactic Pharma’s ownership in Monopar from 79.5% to 69.9%.
Following the surrender of the common stock, Tactic Pharma contributed 4,111,272.88 shares of its holdings in Monopar’s common
stock to TacticGem pursuant to the Gem Transaction discussed in detail in Note 6 above. As of December 31, 2017, Tactic Pharma
beneficially owned 46% of Monopar’s common stock, and TacticGem owned 77% of Monopar’s common stock.

During the years ended December 31, 2017 and 2016, the Company paid or accrued legal fees to a large national law firm, in which
a family member of the Company’s Chief Executive Officer is a law partner, approximately $300,140 and $54,000, respectively.
The family member personally billed a de minimis amount of time on the Company’s legal engagement with the law firm in these
periods.

Note 8 – Income Taxes

ASC 740 requires that the tax benefit of net operating losses, temporary differences, and credit carryforwards be recorded as an asset
to the extent that management assesses that realization is "more likely than not." Realization of the future tax benefits is dependent
on  the  Company's  ability  to  generate  sufficient  taxable  income  within  the  carryforward  period.  The  Company  has  reviewed  the
positive and negative evidence relating to the realizability of the deferred tax assets and has concluded that the deferred tax assets
are not more likely than not to be realized with the exception of $4,358 of U.S. Federal R&D tax credits. These tax credits will be
utilized to reduce payroll taxes in 2018. Accordingly, the valuation allowance has not been released related to these assets with the
exception of $4,000 in U.S. Federal R&D tax credits. The valuation allowance increased by approximately $470,000 and $460,000
during the years ended December 31, 2017 and 2016, respectively.

F-19

 
 
 
 
 
 
 
 
 
 
 
MONOPAR THERAPEUTICS INC.
NOTES TO FINANCIAL STATEMENTS
December 31, 2017

The provision for income taxes for December 31, 2017 and 2016 consists of the following:

Current:
Federal
State

Total current

Deferred:

Federal
State

Total deferred
Full valuation allowance
Total provision(1)

(1) Total provision consists of U.S. Federal R&D credits, net of California minimum tax.

The difference between the effective tax rate and the U.S. federal tax rate is as follows:

Federal income tax
State income taxes, less federal benefit
Tax credits
Permanent differences
Tax basis intangibles
Change in valuation allowance
Other (Release of VA)
Effective tax rate benefit (expense)

F-20

As of December 31,
2017

2016

  $

  $

- 
800 
800 

- 
800 
800 

980,176 
25,169 
    1,005,345 
    (1,000,987)    
(3,558)   $
  $

463,520 
71,734 
535,254 
(535,254)
800 

 %

34.00%
0.07%
0.09%
-27.38%
-4.90%
-1.88%
0.03%
0.03%

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
   
   
   
   
  
   
  
   
   
   
   
   
 
 
 
 
 
 
   
   
   
   
   
   
   
   
 
 
MONOPAR THERAPEUTICS INC.
NOTES TO FINANCIAL STATEMENTS
December 31, 2017

Deferred tax assets and liabilities consist of the following:

Deferred tax assets:

Net operating loss carryforwards
Tax credit carryforwards
Stock compensation
Intangible asset basis differences
Gross deferred tax assets
Valuation allowance
Total deferred tax assets, net of valuation allowance

Deferred tax liabilities:

Net deferred tax liability
Net deferred taxes

As of December 31,

2017

2016

  $

  $

186,019 
30,143 
58,536 
730,647 
    1,005,345 
    (1,000,987)    

4,358 

111,245 
4,470 
— 
419,539 
535,254 
(535,254)
0 

— 
4,358 

  $

  $

— 
0 

As of December 31, 2017, Company had federal net operating loss carryforwards of approximately $820,000 which will begin to
expire  in  2035  for  federal  tax  purposes.  At  December  31,  2017,  the  Company  had  state  net  operating  loss  carryforwards  of
approximately $260,000 which will begin to expire in 2027. The net operating loss related deferred tax assets do not include excess
tax benefits from employee stock option exercises.

As  of  December  31,  2017,  Company  had  R&D  credit  carryforwards  of  approximately  $19,000  and  $14,000  available  to  reduce
future  taxable  income,  if  any,  for  both  federal  and  state  income  tax  purposes,  respectively.  In  addition,  Company  had  $4,358
available to reduce future payroll taxes, if any, for Federal tax purposes. The federal R&D credit carryforwards expire beginning
2035 and Illinois R&D credit carryforwards expire beginning 2020.

The Tax Reform Act of 1986 limits the use of net operating carryforwards in certain situations where changes occur in the stock
ownership  of  a  company.  In  the  event  the  Company  has  had  a  change  in  ownership,  utilization  of  the  carryforwards  could  be
limited. The Company has not performed such a study.

On January 1, 2015, the Company adopted the provisions of FASB Accounting Standards Codification (ASC 740-10), " Accounting
for Uncertainty in Income Taxes ." ASC 740-10 prescribes a comprehensive model for the recognition, measurement, presentation
and disclosure in financial statements of any uncertain tax positions that have been taken or expected to be taken on a tax return.
The  cumulative  effect  of  adopting ASC  740-10  resulted  in  no  adjustment  to  retained  earnings  as  of  December  31,  2017.  It  is
Company's policy to include penalties and interest expense related to income taxes as a component of other expense and interest
expense, respectively, as necessary.

No liability related to uncertain tax positions is recorded on the financial statements related to uncertain tax positions. There are no
unrecognized  tax  benefits  as  of  December  31,  2017.  The  Company  does  not  expect  that  uncertain  tax  benefits  will  materially
change in the next 12 months.

F-21

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
   
   
   
   
   
   
   
   
   
  
   
  
   
   
 
 
 
 
 
 
 
MONOPAR THERAPEUTICS INC.
NOTES TO FINANCIAL STATEMENTS
December 31, 2017

Company  files  U.S.  federal,  California  and  Illinois  State  tax  returns.  Company  is  subject  to  California  State  minimum  franchise
taxes.  All  tax  returns  will  remain  open  for  examination  by  the  federal  and  state  taxing  authorities  for  three  and  four  years,
respectively, from the date of utilization of any net operating loss carryforwards or R&D credits.

On December 22, 2017, the Tax  Cuts and Jobs Act of 2017 was enacted by the U.S. President. The Tax  Cuts and Jobs Act of 2017
is  effective  as  of  January  1,  2018.  In  accordance  with ASC  guidance,  deferred  tax  assets/liabilities  in  the  Company’s  financial
statements are to be reflected at the tax rate in which the deferred tax assets/liabilities are anticipated to be realized. As a result, the
Company changed the tax rate for tax provision purposes at December 31, 2017 from 34% to 21%. This resulted in a reduction of
the value of the Company’s deferred tax asset balances in the amount of approximately $176,000.

Note 9 – Commitments and Contingencies

Development and Collaboration Agreements

The intellectual property rights contributed by Tactic Pharma, LLC to the Company included the non-exclusive license agreement
with XOMA Ltd. for the humanization technology used in the development of MNPR-101. Pursuant to such license agreement, the
Company  is  obligated  to  pay  XOMA  Ltd.  clinical,  regulatory  and  sales  milestones  for  MNPR-101  and  zero  royalties.  As  of
December 31, 2017, the Company has not reached any milestones and has not been required to pay XOMA Ltd. any funds under
this license agreement.

Leases

The Company leases office space at 500 Mercer St., Seattle, WA. The lease commenced on November 1, 2017 and is extendable on
a  month-to-month  basis.  Commencing  January  1,  2018,  the  Company  entered  into  a  lease  for  its  executive  headquarters  at  1000
Skokie  Blvd.,  Suite  350,  Wilmette,  IL.  The  lease  term  is  January  1,  2018  through  December  31,  2019.  The  future  lease
commitments as presented below include amounts for these two leases.

2018
2019
2020

Total future lease payments

Legal Contingencies

  $

  $

30,234 
30,234 
- 
60,468 

The  Company  is  subject  to  claims  and  assessments  from  time  to  time  in  the  ordinary  course  of  business.  The  Company’s
management  does  not  believe  that  any  such  matters,  individually  or  in  the  aggregate,  will  have  a  material  adverse  effect  on  the
Company’s business, financial condition, results of operations or cash flows.

F-22

 
 
 
 
 
 
 
 
 
 
 
   
   
 
 
 
 
MONOPAR THERAPEUTICS INC.
NOTES TO FINANCIAL STATEMENTS
December 31, 2017

Indemnification

In the normal course of business, the Company enters into contracts and agreements that contain a variety of representations and
warranties  and  provide  for  general  indemnification.  The  Company’s  exposure  under  these  agreements  is  unknown  because  it
involves claims that may be made against the Company in the future, but that have not yet been made. To date, the Company has
not paid any claims or been required to defend any action related to its indemnification obligations. However, the Company may
record charges in the future as a result of these indemnification obligations.

In accordance with its amended and restated certificate of incorporation and bylaws, the Company has indemnification obligations
to  its  officers  and  directors  for  certain  events  or  occurrences,  subject  to  certain  limits,  while  they  are  serving  at  the  Company’s
request in such capacity. There have been no claims to date.

Note 10 - Subsequent Events

Cancer Research UK Termination of CTOA

On March 21, 2018 Cancer Research UK notified the Company that it was terminating the CTOA and would work to transfer to the
Company  the  data  and  know-how  generated  under  the  CTOA.  The  Company  is  currently  reviewing  potential  alternative
collaboration opportunities for MNPR-101 and continues to maintain the program’s intellectual property portfolio.

The Company has evaluated all events occurring from December 31, 2017 through March 26, 2018, the date which these financial
statements were available to be issued, and did not identify any additional material disclosable subsequent events.

F-23

 
 
 
 
 
 
 
 
 
 
 
 
Schedule II: Valuation and Qualifying Accounts
Valuation Allowance for Deferred Tax Assets

(In thousands) 
Balance at beginning of year
Additions to charged to expenses/other accounts

Balance at end of year

    Year Ended December 31, 

  $

2017
535,254 
465,733 
  $ 1,000,987 

  $

  $

2016

75,251 
460,003 
535,254 

F-24

 
 
 
 
 
 
 
 
 
 
   
   
 
 
 
 
 
 
 
SECOND AMENDED AND RESTATED CERTIFICATE OF INCORPORATION OF MONOPAR
THERAPEUTICS INC.

This  Second  Amended  and  Restated  Certificate  of  Incorporation  (the  “Certificate”)  amends  and  restates  the  Certificate  of
Incorporation  of  Monopar  Therapeutics  Inc.,  originally  filed  with  the  Delaware  Secretary  of  State  on  December  16,  2015,  which  was
amended and restated on March 15, 2016, under the provisions of and subject to the requirements of the General Corporation Law of the
State of Delaware (the "DGCL"). This Certificate has been duly adopted in accordance with Section 245 of the DGCL, and by written
consent of a majority of stockholders under Section 228 of the DGCL.

FIRST: The name of the corporation is Monopar Therapeutics Inc. (the "Corporation").

SECOND:  The  address  of  the  registered  office  of  the  Corporation  in  the  State  of  Delaware  is  Corporation  Trust  Center,  1209  Orange
Street,  Wilmington,  DE  19801,  in  New  Castle  County.  The  name  of  the  registered  agent  of  the  Corporation  at  such  address  is  The
Corporation Trust Company.

THIRD: The nature of the business or purposes to be conducted or promoted by the Corporation is to engage in any lawful act or activity
for which corporations may be organized under the DGCL.

FOURTH: The total number of shares of stock which the Corporation is authorized to issue is 40,000,000; all of which shall be common
stock having $0.001 par value per share (“Common Stock”). The Common Stock, and any other stock issued by the board of directors of
the Corporation (the “Board”) (together, the “Stock”)  of  the  Corporation  shall  be  governed  by  the  Bylaws  of  the  Corporation  and  this
Certificate.  Upon  the  effectiveness  of  this  Certificate,  (a)  each  share  of  Series A  Preferred  Stock,  $0.001  par  value  per  share  of  the
Corporation authorized and outstanding immediately prior to the effectiveness of this Certificate shall be automatically converted into 84
shares of Common Stock, $0.001 par value per share, and (b) each share of Series Z Preferred Stock, $0.001 par value per share, of the
Corporation authorized and outstanding immediately prior to the effectiveness of this Certificate shall be automatically converted into 70
shares of Common Stock, $0.001 par value per share.

Section 1. General. The terms of each of the shares of Stock of the Corporation shall be equal to and identical in all respects with every
other share of Stock, irrespective of class.

Section 2. Additional Stockholders. Additional persons may be admitted to the Corporation as Stockholders, and shares (of any existing or
new classes) may be created for issuance to such persons, on such terms and conditions as the Board may determine.

Section  3. Conversion. The certificates representing shares of Series A Preferred Stock or Series Z Preferred Stock, as applicable, shall
continue  to  represent  the  holders’  ownership  in  the  Corporation  until  returned  to  the  Corporation  for  replacement,  at  which  time  the
Corporation shall issue and deliver to such holder of Series A Preferred Stock or Series Z Preferred Stock, or

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
to his or its nominees, a certificate or certificates for the number of shares of Common Stock to which the holder is entitled.

FIFTH: To the extent permitted by law, the Corporation may purchase or otherwise acquire shares of stock of any class issued by it for
such consideration and upon such terms and conditions as may be authorized by the Board from time to time.

SIXTH: In furtherance of and not in limitation of powers conferred by statute, this Article is inserted for the management of the business
and for the conduct of the affairs of the Corporation.

1. General Powers. The business and affairs of the Corporation shall be managed by or under the direction of the Board

pursuant to the provisions of this Certificate of Incorporation and the Bylaws of the Corporation, as amended, restated and/or modified
from time to time.

2. Election of Directors. Election of directors need not be by written ballot. Voting rights with respect to election or removal of

members of the Board are set forth in the Bylaws of the Corporation.

3. Authority to Amend Bylaws. In furtherance and not in limitation of the rights, powers, privileges and discretionary authority

granted or conferred by the General Corporation Law of the State of Delaware or other statutes or laws of the State of Delaware, but
subject to the express provisions of this Certificate, the Board is expressly authorized to adopt, make, alter, amend or repeal the Bylaws of
the Corporation, without any action on the part of the stockholders (except to the extent specifically set forth in such Bylaws), but the
Stockholders may adopt or make additional Bylaws and may alter, amend or repeal any Bylaw whether adopted by the Stockholders or
otherwise.

The Corporation may in its Bylaws confer powers upon its Board in addition to the foregoing and in addition to the powers and authorities
expressly conferred upon the Board by applicable law.

SEVENTH: To the fullest extent permitted by Delaware law, no director of the Corporation shall be personally liable to the Corporation
or  its  stockholders  (the  “Stockholders”)  for  monetary  damages  for  any  breach  of  fiduciary  duty  as  a  director,  notwithstanding  any
provision of law (other than any provision of the DGCL) imposing such liability. No amendment to or repeal of this provision shall apply
to or have any effect on the liability or alleged liability of any director of the Corporation for or with respect to any acts or omissions of
such director occurring prior to such amendment or repeal.

EIGHTH: The Corporation shall, to the fullest extent permitted by the DGCL, as amended from time to time, indemnify each person who
was or is a party or is threatened to be made a party to any threatened, pending, or completed action, suit, or proceeding, whether civil,
criminal, administrative, or investigative, by reason of the fact that he or she is or was, or has agreed to become, a director or officer of the
Corporation,  or  is  or  was  serving,  or  has  agreed  to  serve,  at  the  request  of  the  Corporation,  as  a  director,  officer,  manager,  partner,
employee, or trustee of, or in a similar capacity with, another corporation, limited liability company, partnership, joint venture, trust, or
other enterprise (including any employee benefit plan) (all such persons being

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
referred to hereafter as an “Indemnitee”), or by reason of any action alleged to have been taken or omitted in such capacity, against all
expenses (including attorneys’ fees), judgments, fines, and amounts paid in settlement actually and reasonably incurred by or on behalf of
an Indemnitee in connection with such action, suit, or proceeding and any appeal therefrom.

As a condition precedent to an Indemnitee’s right to be indemnified, the Indemnitee must notify the Corporation in writing as
soon  as  practicable  of  any  action,  suit,  proceeding,  or  investigation  involving  such  Indemnitee  for  which  indemnity  will  or  could  be
sought.  With  respect  to  any  action,  suit,  proceeding,  or  investigation  of  which  the  Corporation  is  so  notified,  the  Corporation  will  be
entitled to participate therein at its own expense and/or to assume the defense thereof at its own expense, with legal counsel reasonably
acceptable to the Indemnitee.

In  the  event  that  the  Corporation  does  not  assume  the  defense  of  any  action,  suit,  proceeding,  or  investigation  of  which  the
Corporation receives notice under this Article, the Corporation shall pay in advance of the final disposition of such matter any expenses
(including  attorneys’  fees)  incurred  by  an  Indemnitee  in  defending  a  civil  or  criminal  action,  suit,  proceeding,  or  investigation  or  any
appeal therefrom; provided, however, that the payment of such expenses incurred by an Indemnitee in advance of the final disposition of
such matter shall be made only upon receipt of an undertaking by or on behalf of the Indemnitee to repay all amounts so advanced in the
event that it shall ultimately be determined that the Indemnitee is not entitled to be indemnified by the Corporation as authorized in this
Article,  which  undertaking  shall  be  accepted  without  reference  to  the  financial  ability  of  the  Indemnitee  to  make  such  repayment;  and
further  provided  that  no  such  advancement  of  expenses  shall  be  made  under  this  Article  if  it  is  reasonably  determined  that  (i)  the
Indemnitee did not act in good faith and in a manner he or she reasonably believed to be in, or not opposed to, the best interests of the
Corporation, or (ii) with respect to any criminal action or proceeding, the Indemnitee had reasonable cause to believe his or her conduct
was unlawful.

The  Corporation  shall  not  indemnify  an  Indemnitee  pursuant  to  this Article  in  connection  with  a  proceeding  (or  part  thereof)
initiated by such Indemnitee unless the initiation thereof was approved by the Board of the Corporation. In addition, the Corporation shall
not indemnify an Indemnitee to the extent such Indemnitee is reimbursed from the proceeds of insurance, and in the event the Corporation
makes any indemnification payments to an Indemnitee and such Indemnitee is subsequently reimbursed from the proceeds of insurance,
such Indemnitee shall promptly refund such indemnification payments to the Corporation to the extent of such insurance reimbursement.

The Corporation may not indemnify an Indemnitee (i) for any liability incurred in a proceeding in which such person is adjudged
liable to the Corporation or is subjected to injunctive relief in favor of the Corporation (ii) for acts or omissions that involve intentional
misconduct or a knowing violation of law, fraud or gross negligence, (iii) for unlawful distributions (iv) for any transaction for which such
Indemnitee received a personal benefit in violation or breach of any provision of this Certificate or the Bylaws of the Corporation, or as
otherwise  prohibited  by  or  as  may  be  disallowed  under  Delaware  law  or  (v)  with  respect  to  any  dispute  or  proceeding  between  the
Corporation and such Indemnitee unless such

 
 
 
 
 
 
 
 
 
 
 
 
 
indemnification has been approved by a disinterested majority of the Board or by a majority in interest of disinterested Stockholders who
are entitled to vote.

All determinations hereunder as to the entitlement of an Indemnitee to indemnification or advancement of expenses shall be made
in  each  instance  (a)  by  a  majority  vote  of  the  directors  of  the  Corporation  consisting  of  persons  who  are  not  at  that  time  parties  to  the
action, suit, or proceeding in question (“disinterested directors”), whether or not a quorum, (b) by a committee of disinterested directors
designated  by  majority  vote  of  disinterested  directors,  whether  or  not  a  quorum,  (c)  if  there  are  no  disinterested  directors,  or  if  the
disinterested directors so direct, by independent legal counsel (who may, to the extent permitted by law, be regular legal counsel to the
Corporation) in a written opinion, or (d) by the Stockholders of the Corporation.

The rights provided in this Article (i) shall not be deemed exclusive of any other rights to which an Indemnitee may be entitled
under any law, agreement, or vote of Stockholders or disinterested directors or otherwise, and (ii) shall inure to the benefit of the heirs,
executors  and  administrators  of  the  Indemnitees.  The  Corporation  may,  to  the  extent  authorized  from  time  to  time  by  its  Board,  grant
indemnification rights to other employees or agents of the Corporation or other persons serving the Corporation and such rights may be
equivalent to, or greater or less than, those set forth in this Article.

The Corporation shall have power to purchase and maintain insurance on behalf of any person who is or was a director, officer,
employee or agent of the Corporation, or is or was serving at the request of the Corporation as a director, officer, employee or agent of
another corporation, partnership, joint venture, trust or other enterprise against any expense, liability or loss incurred by such person in any
such capacity or arising out of his status as such, whether or not the Corporation would have the power to indemnify him against such
liability under the DGCL.

No amendment, termination, or repeal of this Article or of the relevant provisions of the DGCL or any other applicable laws shall
affect or diminish in any way the rights of any Indemnitee to indemnification under the provisions hereof with respect to any action, suit,
proceeding,  or  investigation  arising  out  of  or  relating  to  any  actions,  transactions,  or  facts  occurring  prior  to  the  final  adoption  of  such
amendment, termination or repeal.

NINTH: Meetings of Stockholders may be held within or without the State of Delaware, as the By-laws of the Corporation may provide.
The books of the Corporation may be kept outside the State of Delaware at such place as may be designated from time to time by the
Board or in the By-laws of the Corporation.

TENTH: The Corporation shall have the right from time to time, to amend this Certificate or any provision thereof in any manner now or
hereafter provided by law. Except as expressly set forth herein, all rights and powers of any kind conferred upon a director or stockholder
of the Corporation by this Certificate or any amendment thereof are conferred subject to such right.

[SIGNATURE PAGE FOLLOWS]

 
 
 
 
 
 
 
 
 
 
 
 
 
 
In witness whereof, the Corporation has caused this Second Amended and Restated Certificate of Incorporation to be signed this
17th day of March, 2017.

By: /s/ Chandler D. Robinson

Chandler D. Robinson. President

 
 
 
 
 
 
AMENDED AND RESTATED
BY-LAWS OF MONOPAR THERAPEUTICS INC.

ARTICLE I OFFICES

Section 1.01 Registered Office.  The  address,  principal  office,  and  principal  place  of  business  of  Monopar  Therapeutics  Inc.
(hereinafter  called  the  "Corporation")  in  the  State  of  Delaware  shall  be  at  5  Revere  Dr.,  Suite  200,  Northbrook,  Illinois  60062.  The
address of the Corporation’s registered office in Delaware shall be Corporation Trust Center, 1209 Orange Street, Wilmington, DE 19801.

Section 1.02 Other Offices. The Corporation may also have offices at such other places, both within  and  outside  the  State  of
Delaware, as the acting board of directors of the Corporation (the "Board of Directors") from time to time shall determine or the business
of the Corporation may require.

Section 1.03 Books and Records. Any records maintained by the Corporation in the regular course of its business, including its
stock  ledger,  books  of  account  and  minute  books,  may  be  maintained  on  any  information  storage  device  or  method; provided that  the
records so kept can be converted into clearly legible paper form within a reasonable time. The Corporation shall so convert any records so
kept upon the request of any person entitled to inspect such records pursuant to applicable law.

ARTICLE II
MEETINGS OF THE STOCKHOLDERS

Section 2.01 Place of Meetings. All meetings of the stockholders shall be held at such place, if any, either within or without the
State of Delaware, as shall be designated from time to time by resolution of the Board of Directors and stated in the notice of meeting. If
authorized by the Board of Directors in its sole discretion, and subject to such guidelines and procedures as the Board of Directors may
adopt,  stockholders  and  proxyholders  not  physically  present  at  a  meeting  of  stockholders  may,  by  means  of  remote  communication
participate in a meeting of stockholders; and be deemed present in person and vote at a meeting of stockholders, whether such meeting is
to  be  held  at  a  designated  place  or  solely  by  means  of  remote  communication,  provided  that  (i)  the  Corporation  shall  implement
reasonable measures to verify that each person deemed present and permitted to vote at the meeting by means of remote communication is
a stockholder or proxyholder, (ii) the Corporation shall implement reasonable measures to provide such stockholders and proxyholders a
reasonable opportunity to participate in the meeting and to vote on matters submitted to the stockholders, including an opportunity to read
or hear the proceedings of the meeting substantially concurrently with such proceedings, and (iii) if any stockholder or proxyholder votes
or takes other action at the meeting by means of remote communication, a record of such vote or other action shall be maintained by the
Corporation.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Section 2.02 Annual Meeting. Unless directors are elected by written consent in lieu of an annual meeting as permitted by

Section 2.11, the annual meeting of the stockholders for the election of directors and for the transaction of such other business as may
properly come before the meeting shall be held at such date, time and place, if any, as shall be determined by the Board of Directors and
stated in the notice of the meeting.

Section 2.03  Special  Meetings.  Special  meetings  of  stockholders  for  any  purpose  or  purposes  shall  be  called  pursuant  to  a
resolution approved by the Board of Directors and may not be called by any other person or persons. The only business which may be
conducted at a special meeting shall be the matter or matters set forth in the notice of such meeting.

Section  2.04  Adjournments.  Any  meeting  of  the  stockholders,  annual  or  special,  may  be  adjourned  from  time  to  time  to
reconvene at the same or some other place, if any, and notice need not be given of any such adjourned meeting if the time, place, if any,
thereof  and  the  means  of  remote  communication,  if  any,  are  announced  at  the  meeting  at  which  the  adjournment  is  taken.  At  the
adjourned  meeting,  the  Corporation  may  transact  any  business  which  might  have  been  transacted  at  the  original  meeting.  If  the
adjournment is for more than 30 days, a notice of the adjourned meeting shall be given to each stockholder of record entitled to vote at the
meeting.  If  after  the  adjournment  a  new  record  date  is  fixed  for  stockholders  entitled  to  vote  at  the  adjourned  meeting,  the  Board  of
Directors  shall  fix  a  new  record  date  for  notice  of  the  adjourned  meeting  and  shall  give  notice  of  the  adjourned  meeting  to  each
stockholder of record entitled to vote at the adjourned meeting as of the record date fixed for notice of the adjourned meeting.

Section 2.05 Notice of Meetings. Notice of the place, if any, date, hour, the record date for determining the stockholders entitled
to  vote  at  the  meeting  (if  such  date  is  different  from  the  record  date  for  stockholders  entitled  to  notice  of  the  meeting)  and  means  of
remote communication, if any, of every meeting of stockholders shall be given by the Corporation not less than ten days nor more than 60
days before the meeting (unless a different time is specified by law) to every stockholder entitled to vote at the meeting as of the record
date  for  determining  the  stockholders  entitled  to  notice  of  the  meeting.  Notices  of  special  meetings  shall  also  specify  the  purpose  or
purposes  for  which  the  meeting  has  been  called.  Except  as  otherwise  provided  herein  or  permitted  by  applicable  law,  notice  to
stockholders  shall  be  in  writing  and  delivered  personally  or  mailed  to  the  stockholders  at  their  address  appearing  on  the  books  of  the
Corporation. Without limiting the manner by which notice otherwise may be given effectively to stockholders, notice of meetings may be
given to stockholders by means of electronic transmission in accordance with applicable law. Notice of any meeting need not be given to
any stockholder who shall, either before or after the meeting, submit a waiver of notice or who shall attend such meeting, except when the
stockholder attends for the express purpose of objecting, at the beginning of the meeting, to the transaction of any business because the
meeting is not lawfully called or convened. Any stockholder so waiving notice of the meeting shall be bound by the proceedings of the
meeting in all respects as if due notice thereof had been given.

Section 2.06 List of Stockholders. The officer of the Corporation who has charge of the stock ledger shall prepare a complete

list of the stockholders entitled to vote at any meeting

 
 
 
 
 
 
 
 
 
 
 
 
 
of  stockholders  (provided,  however,  if  the  record  date  for  determining  the  stockholders  entitled  to  vote  is  less  than  ten  days  before  the
date  of  the  meeting,  the  list  shall  reflect  the  stockholders  entitled  to  vote  as  of  the  tenth  day  before  the  meeting  date),  arranged  in
alphabetical order, and showing the address of each stockholder and the number of shares of each class of capital stock of the Corporation
registered  in  the  name  of  each  stockholder  at  least  ten  days  before  any  meeting  of  the  stockholders.  Such  list  shall  be  open  to  the
examination of any stockholder, for any purpose germane to the meeting, on a reasonably accessible electronic network if the information
required to gain access to such list was provided with the notice of the meeting or during ordinary business hours, at the principal place of
business of the Corporation for a period of at least ten days before the meeting. If the meeting is to be held at a place, the list shall also be
produced and kept at the time and place of the meeting the whole time thereof and may be inspected by any stockholder who is present. If
the meeting is held solely by means of remote  communication,  the  list  shall  also  be  open  for  inspection  by  any  stockholder  during  the
whole time of the meeting as provided by applicable law. Except as provided by applicable law, the stock ledger of the Corporation shall
be the only evidence as to who are the stockholders entitled to examine the stock ledger and the list of stockholders or to vote in person or
by proxy at any meeting of stockholders.

Section 2.07 Quorum.  Unless  otherwise  required  by  law,  the  Corporation's  Certificate  of  Incorporation  (the  " Certificate  of
Incorporation")  or  these  by-laws,  at  each  meeting  of  the  stockholders,  a  majority  in  voting  power  of  the  shares  of  the  Corporation
entitled to vote at the meeting, present in person or represented by proxy, shall constitute a quorum. If, however, such quorum shall not be
present  or  represented  at  any  meeting  of  the  stockholders,  the  stockholders  entitled  to  vote  thereat,  present  in  person  or  represented  by
proxy, shall have power, by the affirmative vote of a majority in voting power thereof, to adjourn the meeting from time to time, in the
manner provided in Section 2.04, until a quorum shall be present or represented. A quorum, once established, shall not be broken by the
subsequent  withdrawal  of  enough  votes  to  leave  less  than  a  quorum. At  any  such  adjourned  meeting  at  which  there  is  a  quorum,  any
business may be transacted that might have been transacted at the meeting originally called.

Section 2.08 Conduct of Meetings. The Board of Directors may adopt by resolution such rules and regulations for the conduct
of  the  meeting  of  the  stockholders  as  it  shall  deem  appropriate. At  every  meeting  of  the  stockholders,  the  President,  or  in  his  or  her
absence or inability to act, the Vice President, or, in his or her absence or inability to act, the person whom the President shall appoint,
shall  act  as  chairman  of,  and  preside  at,  the  meeting.  The  secretary  or,  in  his  or  her  absence  or  inability  to  act,  the  person  whom  the
chairman of the meeting shall appoint secretary of the meeting, shall act as secretary of the meeting and keep the minutes thereof. Except
to  the  extent  inconsistent  with  such  rules  and  regulations  as  adopted  by  the  Board  of  Directors,  the  chairman  of  any  meeting  of  the
stockholders  shall  have  the  right  and  authority  to  prescribe  such  rules,  regulations  and  procedures  and  to  do  all  such  acts  as,  in  the
judgment of such chairman, are appropriate for the proper conduct of the meeting. Such rules, regulations or procedures, whether adopted
by  the  Board  of  Directors  or  prescribed  by  the  chairman  of  the  meeting,  may  include,  without  limitation,  the  following:  (a)  the
establishment of an agenda or order of business for the meeting; (b) the determination of when the polls shall open and close for any given
matter to be voted on at the meeting; (c) rules and procedures for maintaining order at the meeting and the safety of those present; (d)
limitations on attendance at or participation in

 
 
 
 
 
 
 
 
 
the  meeting  to  stockholders  of  record  of  the  corporation,  their  duly  authorized  and  constituted  proxies  or  such  other  persons  as  the
chairman of the meeting shall determine; (e) restrictions on entry to the meeting after the time fixed for the commencement thereof; and
(f) limitations on the time allotted to questions or comments by participants.

Section 2.09 Voting; Proxies. Unless otherwise required by law or the Certificate of Incorporation the election of directors shall
be decided by a plurality of the votes cast at a meeting of the stockholders by the holders of stock entitled to vote in the election. Unless
otherwise  required  by  law,  the  Certificate  of  Incorporation  or  these  by-laws,  any  matter,  other  than  the  election  of  directors,  brought
before any meeting of stockholders shall be decided by the affirmative vote of the majority of shares present in person or represented by
proxy  at  the  meeting  and  entitled  to  vote  on  the  matter.  Each  stockholder  entitled  to  vote  at  a  meeting  of  stockholders  or  to  express
consent to corporate action in writing without a meeting may authorize another person or persons to act for such stockholder by proxy, but
no such proxy shall be voted or acted upon after three years from its date, unless the proxy provides for a longer period. A proxy shall be
irrevocable  if  it  states  that  it  is  irrevocable  and  if,  and  only  as  long  as,  it  is  coupled  with  an  interest  sufficient  in  law  to  support  an
irrevocable  power. A  stockholder  may  revoke  any  proxy  which  is  not  irrevocable  by  attending  the  meeting  and  voting  in  person  or  by
delivering  to  the  secretary  of  the  Corporation  a  revocation  of  the  proxy  or  a  new  proxy  bearing  a  later  date.  Voting  at  meetings  of
stockholders need not be by written ballot.

Section 2.10 Inspectors at Meetings of Stockholders. The Board of Directors, in advance of any meeting of stockholders, may,
and  shall  if  required  by  law,  appoint  one  or  more  inspectors,  who  may  be  employees  of  the  Corporation,  to  act  at  the  meeting  or  any
adjournment thereof and make a written report thereof. The Board of Directors may designate one or more persons as alternate inspectors
to replace any inspector who fails to act. If no inspector or alternate is able to act at a meeting, the person presiding at the meeting shall
appoint one or more inspectors to act at the meeting. Each inspector, before entering upon the discharge of his or her duties, shall take and
sign  an  oath  faithfully  to  execute  the  duties  of  inspector  with  strict  impartiality  and  according  to  the  best  of  his  or  her  ability.  The
inspectors shall (a) ascertain the number of shares outstanding and the voting power of each, (b) determine the shares represented at the
meeting, the existence of a quorum and the validity of proxies and ballots, (c) count all votes and ballots, (d) determine and retain for a
reasonable  period  a  record  of  the  disposition  of  any  challenges  made  to  any  determination  by  the  inspectors  and  (e)  certify  their
determination of the number of shares represented at the meeting and their count of all votes and ballots. The inspectors may appoint or
retain  other  persons  or  entities  to  assist  the  inspectors  in  the  performance  of  their  duties.  Unless  otherwise  provided  by  the  Board  of
Directors, the date and time of the opening and the closing of the polls for each matter upon which the stockholders will vote at a meeting
shall  be  announced  at  the  meeting.  No  ballot,  proxies,  votes  or  any  revocation  thereof  or  change  thereto,  shall  be  accepted  by  the
inspectors  after  the  closing  of  the  polls  unless  the  Court  of  Chancery  of  the  State  of  Delaware  upon  application  by  a  stockholder  shall
determine otherwise. In determining the validity and counting of proxies and ballots cast at any meeting of stockholders, the inspectors
may consider such information as is permitted by applicable law. No person who is a candidate for office at an election may serve as an
inspector at such election.

 
 
 
 
 
 
 
 
 
Section 2.11 Written Consent of Stockholders Without a Meeting.  Any action to be taken at any annual or special meeting of
stockholders may be taken without a meeting, without prior notice and without a vote, if a consent or consents in writing, setting forth the
action to be so taken, shall be signed by the holders of outstanding stock having not less than the minimum number of votes that would be
necessary to authorize or take such action at a meeting at which all shares entitled to vote thereon were present and voted and shall be
delivered (by hand or by certified or registered mail, return receipt requested) to the Corporation by delivery to its registered office in the
State  of  Delaware,  its  principal  place  of  business  or  an  officer  or  agent  of  the  Corporation  having  custody  of  the  book  in  which
proceedings  of  meetings  of  stockholders  are  recorded.  Every  written  consent  shall  bear  the  date  of  signature  of  each  stockholder  who
signs the consent, and no written consent shall be effective to take the corporate action referred to therein unless, within 60 days of the
earliest dated consent delivered in the manner required by this Section, written consents signed by a sufficient number of holders to take
action are delivered to the Corporation as aforesaid. Prompt notice of the taking of the corporate action without a meeting by less than
unanimous  written  consent  shall,  to  the  extent  required  by  applicable  law,  be  given  to  those  stockholders  who  have  not  consented  in
writing, and who, if the action had been taken at a meeting, would have been entitled to notice of the meeting if the record date for notice
of such meeting had been the date that written consents signed by a sufficient number of holders to take the action were delivered to the
Corporation. Stockholders may act by written consent to elect directors; provided, however, that, if such consent is less than unanimous,
such action by written consent may be in lieu of holding an annual meeting only if all of the directorships to which directors could be
elected at an annual meeting held at the effective time of such action are vacant and are filled by such action.

Section 2.12 Fixing the Record Date.

(a) In  order  that  the  Corporation  may  determine  the  stockholders  entitled  to  notice  of  or  to  vote  at  any  meeting  of
stockholders or any adjournment thereof, the Board of Directors may fix a record date, which record date shall not precede the date upon
which the resolution fixing the record date is adopted by the Board of Directors, and which record date shall not be more than 60 nor less
than  ten  days  before  the  date  of  such  meeting.  If  the  Board  of  Directors  so  fixes  a  date,  such  date  shall  also  be  the  record  date  for
determining the stockholders entitled to vote at such meeting unless the Board of Directors determines, at the time it fixes such record
date, that a later date on or before the date of the meeting shall be the date for making such determination. If no record date is fixed by the
Board of Directors, the record date for determining stockholders entitled to notice of or to vote at a meeting of stockholders shall be at the
close of business on the day next preceding the day on which notice is given, or, if notice is waived, at the close of business on the day
next  preceding  the  day  on  which  the  meeting  is  held. A  determination  of  stockholders  of  record  entitled  to  notice  of  or  to  vote  at  a
meeting  of  stockholders  shall  apply  to  any  adjournment  of  the  meeting; provided, however,   that  the  Board  of  Directors  may  fix  a  new
record date for the determination of stockholders entitled to vote at the adjourned meeting and in such case shall also fix as the record
date  for  stockholders  entitled  to  notice  of  such  adjourned  meeting  the  same  or  an  earlier  date  as  that  fixed  for  the  determination  of
stockholders entitled to vote therewith at the adjourned meeting.

 
 
 
 
 
 
 
 
(b)  In  order  that  the  Corporation  may  determine  the  stockholders  entitled  to  consent  to  corporate  action  in  writing
without a meeting, the Board of Directors may fix a record date, which record date shall not precede the date upon which the resolution
fixing the record date is adopted by the Board of Directors, and which record date shall not be more than ten days after the date upon
which  the  resolution  fixing  the  record  date  is  adopted  by  the  Board  of  Directors.  If  no  record  date  has  been  fixed  by  the  Board  of
Directors, the record date for determining stockholders entitled to consent to corporate action in writing without a meeting: (i) when no
prior action by the Board of Directors is required by law, the record date for such purpose shall be the first date on which a signed written
consent  setting  forth  the  action  taken  or  proposed  to  be  taken  is  delivered  to  the  Corporation  by  delivery  (by  hand,  or  by  certified  or
registered mail, return receipt requested) to its registered office in the State of Delaware, its principal place of business, or an officer or
agent of the Corporation having custody of the book in which proceedings of meetings of stockholders are recorded and (ii) if prior action
by the Board of Directors is required by law, the record date for such purpose shall be at the close of business on the day on which the
Board of Directors adopts the resolution taking such prior action.

(c) In order that the Corporation may determine the stockholders entitled to receive payment of any dividend or other
distribution or allotment of any rights or the stockholders entitled to exercise any rights in respect of any change, conversion or exchange
of stock, or for the purpose of any other lawful action, the Board of Directors may fix a record date, which record date shall not precede
the date upon which the resolution fixing the record date is adopted, and which record date shall be not more than 60 days prior to such
action. If no record date is fixed, the record date for determining stockholders for any such purpose shall be at the close of business on the
day on which the Board of Directors adopts the resolution relating thereto.

ARTICLE III BOARD OF DIRECTORS

Section 3.01 General Powers.  The  business  and  affairs  of  the  Corporation  shall  be  managed  by  or  under  the  direction  of  the
Board of Directors. The Board of Directors may adopt such rules and procedures, not inconsistent with the Certificate of Incorporation,
these by-laws or applicable law, as it may deem proper for the conduct of its meetings and the management of the Corporation.

Section 3.02 Number; Term of Office.  The number of directors of the Corporation shall not be less than three nor more than
seven.  The  number  of  directors  shall,  at  the  date  of  adoption  of  these  Bylaws,  initially  be  fixed  at  four,  and  hereafter,  such  number  of
directors may be fixed or changed at any annual meeting of the stockholders or at any special meeting of the stockholder called for that
purpose  by  the  affirmative  vote  of  the  holders  of  a  majority  or  more  of  the  voting  power  of  the  Corporation.  Each  director  shall  hold
office  for  a  period  of  one  year  and  until  a  successor  is  duly  elected  and  qualified  or  until  the  director's  earlier  death,  resignation,
disqualification or removal.

 
 
 
 
 
 
 
 
 
 
 
Section 3.03 Newly Created Directorships and Vacancies. Any newly created directorships resulting from an increase in the
authorized number of directors and any vacancies occurring in the Board of Directors, may be filled by the affirmative votes of a majority
of the remaining members of the Board of Directors, although less than a quorum, or by a sole remaining director. A director so elected
shall  be  elected  to  hold  office  until  the  earlier  of  the  expiration  of  the  term  of  office  of  the  director  whom  he  or  she  has  replaced,  a
successor is duly elected and qualified or the earlier of such director's death, resignation or removal.

Section 3.04 Resignation. Any director may resign at any time by notice given in writing or by electronic transmission to the
Corporation. Such resignation shall take effect at the date of receipt of such notice by the Corporation or at such later time as is therein
specified.

Section 3.05 Removal.  Except  as  prohibited  by  applicable  law  or  the  Certificate  of  Incorporation,  the  stockholders  entitled  to
vote  in  an  election  of  directors  may  remove  any  director  from  office  at  any  time,  with  or  without  cause,  by  the  affirmative  vote  of  a
majority in voting power thereof.

Section 3.06 Fees and Expenses. Directors shall receive such fees, which may include equity compensation, and expenses as the

Board of Directors shall from time to time prescribe.

Section 3.07 Regular Meetings. Regular meetings of the Board of Directors may be held without notice  at  such  times  and  at

such places as may be determined from time to time by the Board of Directors or its chairman.

Section 3.08 Special Meetings. Special meetings of the Board of Directors may be held at such times and at such places as may
be determined by the chairman or the President on at least 24 hours' notice to each director given by one of the means specified in Section
3.11 hereof other than by mail or on at least three days' notice if given by mail. Special meetings shall be called by the chairman or the
President in like manner and on like notice on the written request of any two or more directors.

Section 3.09 Telephone Meetings.  Board  of  Directors  or  Board  of  Directors  committee  meetings  may  be  held  by  means  of
telephone conference or other communications equipment by means of which all persons participating in the meeting can hear each other
and be heard. Participation by a director in a meeting pursuant to this Section shall constitute presence in person at such meeting.

Section 3.10 Adjourned Meetings. A majority of the directors present at any meeting of the Board of Directors, including an
adjourned meeting, whether or not a quorum is present, may adjourn and reconvene such meeting to another time and place. At least 24
hours' notice of any adjourned meeting of the Board of Directors shall be given to each director whether or not present at the time of the
adjournment, if such notice shall be given by one of the means specified in Section 3.11 hereof other than by mail, or at least three days'
notice if by mail. Any business may be transacted at an adjourned meeting that might have been transacted at the meeting as originally
called.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Section 3.11 Notices. Subject to Section 3.08, Section 3.10 and Section 3.12 hereof, whenever notice is required to be given to
any director by applicable law, the Certificate of Incorporation or these by-laws, such notice shall be deemed given effectively if given in
person or by telephone, mail addressed to such director at such director's address as it appears on the records of the Corporation, facsimile,
e-mail or by other means of electronic transmission.

Section 3.12 Waiver of Notice.  Whenever notice to directors is required by applicable law, the Certificate of Incorporation or
these by-laws, a waiver thereof, in writing signed by, or by electronic transmission by, the director entitled to the notice, whether before or
after such notice is required, shall be deemed equivalent to notice. Attendance by a director at a meeting shall constitute a waiver of notice
of such meeting except when the director attends a meeting for the express purpose of objecting, at the beginning of the meeting, to the
transaction of any business on the ground that the meeting was not lawfully called or convened. Neither the business to be transacted at,
nor the purpose of, any regular or special Board of Directors or committee meeting need be specified in any waiver of notice.

Section 3.13 Organization. At each meeting of the Board of Directors, the chairman or, in his or her absence, another director
selected  by  the  Board  of  Directors  shall  preside.  The  secretary  shall  act  as  secretary  at  each  meeting  of  the  Board  of  Directors.  If  the
secretary is absent from any meeting of the Board of Directors, an assistant secretary shall perform the duties of secretary at such meeting;
and in the absence from any such meeting of the secretary and all assistant secretaries, the person presiding at the meeting may appoint
any person to act as secretary of the meeting.

Section 3.14 Quorum of Directors.  The  presence  of  a  majority  of  the  Board  of  Directors  shall  be  necessary  and  sufficient  to

constitute a quorum for the transaction of business at any meeting of the Board of Directors.

Section 3.15 Action by Majority Vote. Except as otherwise expressly required by these by-laws, the Certificate of Incorporation

or by applicable law, the vote of a majority of the directors shall be the act of the Board of Directors.

Section 3.16 Action  Without  Meeting.  Unless  otherwise  restricted  by  the  Certificate  of  Incorporation  or  these  by-laws,  any
action required or permitted to be taken at any meeting of the Board of Directors or of any committee thereof may be taken without a
meeting if all directors or members of such committee, as the case may be, consent thereto in writing or by electronic transmission, and
the writings or electronic transmissions are filed with the minutes of proceedings of the Board of Directors or committee in accordance
with applicable law.

Section 3.17 Committees  of  the  Board  of  Directors.  The  Board  of  Directors  may  designate  one  or  more  committees,  each
committee to consist of one or more of the directors of the Corporation. The Board of Directors may designate one or more directors as
alternate members of any committee, who may replace any absent or disqualified member at any meeting of the committee. If a member
of a committee shall be absent from any meeting, or disqualified from voting thereat, the remaining member or members present at the
meeting and not disqualified from voting, whether or not such member or members constitute a quorum, may

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
unanimously  appoint  another  member  of  the  Board  of  Directors  to  act  at  the  meeting  in  the  place  of  any  such  absent  or  disqualified
member. Any such committee, to the extent permitted by applicable law, shall have and may exercise all the powers and authority of the
Board of Directors in the management of the business and affairs of the Corporation and may authorize the seal of the Corporation to be
affixed  to  all  papers  that  may  require  it  to  the  extent  so  authorized  by  the  Board  of  Directors.  Unless  the  Board  of  Directors  provides
otherwise, at all meetings of such committee, a majority of the then authorized members of the committee shall constitute a quorum for
the transaction of business, and the vote of a majority of the members of the committee present at any meeting at which there is a quorum
shall  be  the  act  of  the  committee.  Each  committee  shall  keep  regular  minutes  of  its  meetings.  Unless  the  Board  of  Directors  provides
otherwise, each committee designated by the Board of Directors may make, alter and repeal rules and procedures for the conduct of its
business.  In  the  absence  of  such  rules  and  procedures  each  committee  shall  conduct  its  business  in  the  same  manner  as  the  Board  of
Directors conducts its business pursuant to this Article III.

ARTICLE IV OFFICERS

Section 4.01 Positions and Election. The officers of the Corporation shall be elected annually by the Board of Directors and shall
include a president, a treasurer and a secretary. The Board of Directors, in its discretion, may also elect a chairman (who must be a director),
one or more vice chairmen (who must be directors) and one or more vice presidents, assistant treasurers, assistant secretaries and other
officers. Any two or more offices may be held by the same person.

Section 4.02 Term.  Each  officer  of  the  Corporation  shall  hold  office  until  such  officer's  successor  is  elected  and  qualified  or
until such officer's earlier death, resignation or removal. Any officer elected or appointed by the Board of Directors may be removed by
the Board of Directors at any time with or without cause by the majority vote of the members of the Board of Directors then in office. The
removal of an officer shall be without prejudice to his or her contract rights, if any. The election or appointment of an officer shall not of
itself create contract rights. Any officer of the Corporation may resign at any time by giving written notice of his or her resignation to the
president or the secretary. Any such resignation shall take effect at the time specified therein or, if the time when it shall become effective
shall not be specified therein, immediately upon its receipt. Unless otherwise specified therein, the acceptance of such resignation shall not
be necessary to make it effective. Should any vacancy occur among the officers, the position shall be filled for the unexpired portion of
the term by appointment made by the Board of Directors.

Section 4.03 The President. The president shall have general supervision over the business of the Corporation and other duties
incident to the office of president, and any other duties as may be from time to time assigned to the president by the Board of Directors
and subject to the control of the Board of Directors in each case.

Section 4.04 Vice Presidents. Each vice president shall have such powers and perform such duties as may be assigned to him or

her from time to time by the chairman of the Board of Directors or the president.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Section 4.05 The Secretary. The secretary shall attend all sessions of the Board of Directors and all meetings of the stockholders
and record all votes and the minutes of all proceedings in a book to be kept for that purpose, and shall perform like duties for committees
when  required.  He  or  she  shall  give,  or  cause  to  be  given,  notice  of  all  meetings  of  the  stockholders  and  meetings  of  the  Board  of
Directors, and shall perform such other duties as may be prescribed by the Board of Directors or the president. The secretary shall keep in
safe custody the seal of the Corporation and have authority to affix the seal to all documents requiring it and attest to the same.

Section 4.06 The Treasurer.   The  treasurer  shall  have  the  custody  of  the  corporate  funds  and  securities,  except  as  otherwise
provided  by  the  Board  of  Directors,  and  shall  keep  full  and  accurate  accounts  of  receipts  and  disbursements  in  books  belonging  to  the
Corporation and shall deposit all moneys and other valuable effects in the name and to the credit of the Corporation in such depositories as
may be designated by the Board of Directors. The treasurer shall disburse the funds of the Corporation as may be ordered by the Board of
Directors, taking proper vouchers for such disbursements, and shall render to the president and the directors, at the regular meetings of the
Board of Directors, or whenever they may require it, an account of all his or her transactions as treasurer and of the financial condition of
the Corporation.

Section 4.07 Duties  of  Officers  May  Be  Delegated.  In  case  any  officer  is  absent,  or  for  any  other  reason  that  the  Board  of
Directors  may  deem  sufficient,  the  president  or  the  Board  of  Directors  may  delegate  for  the  time  being  the  powers  or  duties  of  such
officer to any other officer or to any director.

ARTICLE V

STOCK CERTIFICATES AND THEIR TRANSFER

Section 5.01 Certificates  Representing  Shares.  The  shares  of  stock  of  the  Corporation  shall  be  represented  by  certificates;
provided that the Board of Directors may provide by resolution or resolutions that some or all of any class or series shall be uncertificated
shares that may be evidenced by a book-entry system maintained by the registrar of such stock. If shares are represented by certificates,
such certificates shall be in the form, other than bearer form, approved by the Board of Directors. The certificates representing shares of
stock of each class shall be signed by, or in the name of, the Corporation by the chairman, any vice chairman, the president or any vice
president,  and  by  the  secretary,  any  assistant  secretary,  the  treasurer  or  any  assistant  treasurer.  Any  or  all  such  signatures  may  be
facsimiles. Although any officer, transfer agent or registrar whose manual or facsimile signature is affixed to such a certificate ceases to be
such officer, transfer agent or registrar before such certificate has been issued, it may nevertheless be issued by the Corporation with the
same effect as if such officer, transfer agent or registrar were still such at the date of its issue.

Section 5.02 Lost,  Stolen  or  Destroyed  Certificates.  The  Board  of  Directors  may  direct  a  new  certificate  or  uncertificated
shares to be issued in place of any certificate theretofore issued by the Corporation alleged to have been lost, stolen or destroyed upon the
making of an affidavit of that fact by the owner of the allegedly lost, stolen or destroyed certificate. When

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
authorizing  such  issue  of  a  new  certificate  or  uncertificated  shares,  the  Board  of  Directors  may ,  in  its  discretion  and  as  a  condition
precedent to the issuance thereof, require the owner of the lost, stolen or destroyed certificate, or the owner's legal representative to give
the Corporation a bond sufficient to indemnify it against any claim that may be made against the Corporation with respect to the certificate
alleged to have been lost, stolen or destroyed or the issuance of such new certificate or uncertificated shares.

ARTICLE VI
GENERAL PROVISIONS

Section 6.01 Seal. The board of directors may adopt and use a corporate seal. The seal of the Corporation shall be  in such form
as shall be approved by the Board of Directors. The seal may  be used by causing it or a facsimile thereof to be impressed or affixed or
reproduced or otherwise, as may be prescribed by law or custom or by the Board of Directors. Failure to affix the corporate seal, if any,
shall not affect the validity of any instrument.

Section 6.02 Fiscal Year. The fiscal year of the Corporation shall be the calendar year.

Section 6.03 Checks, Notes, Drafts, Etc. All checks, notes, drafts or other orders for the payment of money of the Corporation
shall be signed, endorsed or accepted in the name of the Corporation by such officer, officers, person or persons as from time to time may
be designated by the Board of Directors or by an officer or officers authorized by the Board of Directors to make such designation.

Section 6.04 Dividends. Subject to applicable law and the Certificate of Incorporation, dividends upon the shares of capital stock
of the Corporation may be declared by the Board of Directors at any regular or special meeting of the Board of Directors or by consent in
writing.  Dividends  may  be  paid  in  cash,  in  property  or  in  shares  of  the  Corporation's  capital  stock,  unless  otherwise  provided  by
applicable law or the Certificate of Incorporation.

Section  6.05  Conflict  with  Applicable  Law  or  Certificate  of  Incorporation.  These  by-laws  are  adopted  subject  to  any
applicable law and the Certificate of Incorporation. Whenever  these  by-laws  may  conflict  with  any  applicable  law  or  the  Certificate  of
Incorporation, such conflict shall be resolved in favor of such law or the Certificate of Incorporation.

ARTICLE VII
AMENDMENTS

These by-laws may be amended, altered, changed, adopted and repealed or new by-laws adopted at any meeting of the Board of

Directors.

Eff. March 17 2017
/s/ Chandler D. Robinson

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
  [***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
  Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January
8, 2018.

CANCER RESEARCH UK

and

CANCER RESEARCH TECHNOLOGY LIMITED

and

MONOPAR THERAPEUTICS LLC

CLINICAL TRIAL AND OPTION AGREEMENT
(CTOA)

 
 
 
 
 
 
 
 
 
 
  
 
 
 
 
 
 
TABLE OF CONTENTS

DEFINITIONS AND INTERPRETATION
1
CONDITIONS PRECEDENT
2
CONDUCT OF THE CLINICAL TRIAL AND SPONSORSHIP
3
COMPANY’S OBLIGATIONS
4
CONFIDENTIALITY/PUBLICATION
5
INTELLECTUAL PROPERTY RIGHTS
6
OPTION
7
WARRANTIES AND LIMITS OF LIABILITY
8
INDEMNITIES
9
ASSIGNMENT
10
TERM AND TERMINATION
11
CONSEQUENCES OF TERMINATION
12
DISPUTE RESOLUTION
13
14
NOTICES
15 WAIVER
16
17.
18
19
20
21
22
23
24
25.

FORCE MAJEURE
INSOLVENCY
SEVERABILITY
ENTIRE AGREEMENT
AMENDMENT
PUBLIC ANNOUNCEMENTS
PAYMENTS
DATA PROTECTION
THIRD PARTY RIGHTS
EXECUTION

Schedule 1
Schedule 2
Schedule 3
Schedule 4
Schedule 5
Schedule 6
Schedule 7
Schedule 8
Schedule 9
Schedule 10
Schedule 11
Schedule 12
Schedule 13

Company Patent Rights
Report Synopsis Headings
Licence from CRT to Company
No Fault Compensation Scheme
Assignment and Licence from Company to CRT
Protocol
Company Materials
Back-Up Antibodies
XOMA Licence
Progress Reports
Clinical Protocol Summary
Escrow Agreement
Technical Agreement

4
12
12
14
16
19
20
21
22
24
24
25
26
27
28
28
28
28
29
29
29
30
30
30
30

 
 
 
 
 
 
 
 
THIS AGREEMENT is made the 15th day of May 2015

BETWEEN:

CANCER RESEARCH UK a company  limited  by  guarantee  registered  under  number  4325234  and  a charity  registered  under  number
1089464 of Angel Building, 407 St. John Street, London, EC1V 4AD, England (the “Charity”);

CANCER RESEARCH TECHNOLOGY LIMITED a company registered in England and Wales with number 1626049 and registered
office at Angel Building, 407 St. John Street, London, EC1V 4AD, England (“CRT”); and

MONOPAR THERAPEUTICS LLC, a limited liability company registered in/incorporated in/ established under the laws of The State
of Delaware, U.S.A., with registered office/principal place of business at 598 Rockefeller Road, Lake Forest, Illinois, U.S.A., 60045 (the
“Company”).

WHEREAS:

(A) 

(B) 

(C) 

(D) 

(E) 

The Company has the right to conduct research and clinical testing on the Antibody (as defined below). At this time, the Company
does not intend to undertake any further development of the Antibody.

The Charity's charitable objects are to protect and promote the health of the public in particular by research into the nature, causes,
diagnosis, prevention, treatment and cure of cancer, including development of findings of research into practical applications.

The Charity has expertise in the clinical evaluation of novel anti-cancer agents and considers that the Antibody has the potential to
be  a  valuable  drug  that  could  be  applied  for  the  treatment  of  cancer. Accordingly,  the  Charity  is  interested  in  undertaking  the
development  of  the Antibody  at  its  own  cost. As  the  development  is  to  be  undertaken  in  pursuance  of  the  Charity's  charitable
objects, the Charity will have the right to publish the results of such development work.

On completion of the Charity’s development work, the Company will have the option to take a licence to the results thereof with a
view to the Company developing the drug further. If the Company does not wish to take a licence to such results, then CRT shall
have the right to an assignment of rights owned by the Company and a licence to the rights licensed to the Company, in both cases
in and to the Antibody, to enable CRT to find an alternative partner to develop the Antibody further.

CRT  is  a  wholly  owned  subsidiary  of  the  Charity  and  is,  by  arrangement  with  the  Charity,  responsible  for  the  management,
exploitation  and  commercialisation  of  intellectual  property  generated  by  the  Charity  or  using  funding  from  the  Charity  and  the
Charity has assigned and will assign such intellectual property to CRT for such purpose. CRT remits all its taxable profits to the
Charity.

(F) 

The  Company,  CRT  and  the  Charity  have  therefore  agreed  to  enter  into  this Agreement  to  enable  the  Charity  to  undertake  the
development of the Antibody subject to the following terms and conditions:

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
  [***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
  Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

NOW IT IS HEREBY AGREED as follows:

1.

1.1

DEFINITIONS AND INTERPRETATION

In this Agreement the words and phrases set out below shall, unless the context requires otherwise, have the corresponding meaning
attributed to them below. In addition, any words and phrases in this Agreement which are not defined below, but which are defined
in the CTD, shall have the meaning attributed to them in the CTD.

“Additional

Studies”

means  any  biomarker,  manufacturing,  purity,  toxicology,  imaging  or  combination  studies,  or  any  other
exploratory or pre-clinical in vitro or in vivo studies commenced after the Commencement Date and associated
with  any  part  of  the  Antibody,  or  carried  out  in  support  of  the  clinical  trial  conducted  pursuant  to  this
Agreement,  where  such  studies  are  performed  by  or  on  behalf  of  the  Charity  (as  the  same  may  be  amended
from time to time by the Charity).

“Additional
Results”

means  all  Know-How,  data,  information  and  results  Controlled  by  the  Charity  or  CRT  and  arising  from  the
Additional Studies.

“Affiliate”

means an entity that, whether now or in the future, Controls, is Controlled by or is under common Control with
a Party. For the purpose of this definition only, “Control” means the possession (directly or indirectly) of fifty
per cent or more of the voting stock or other equity interest of a subject entity with the power to vote, or the
power  in  fact  to  control  the  management  decisions  of  such  entity  through  the  ownership  of  securities  or  by
contract or otherwise and “Controls” and “Controlled by” shall be construed accordingly.

“Antibody”

means  the  humanised  anti-uPAR  monocolonal  antibody  known  as  HuATN-658  and/or  any  monoclonal
antibody derived directly or indirectly from the Cell Line, including any fragment or conjugated antibody.

“this Agreement”

means this agreement and each of the Schedules to it as amended from time to time in accordance with Clause
20.

“Back-Up
Antibodies”

means  any  and  all  antibodies,  other  than  the anti-uPAR  monocolonal  antibody  known  as  HuATN-658,   that
have been or are discovered, generated or developed by or on behalf of the Company or any of its Affiliates in
the course of the [***] including, but not limited to, the compounds identified in Schedule 8.

“Case 
Forms”

Report

means  a  record  of  the  data  and  other  information  gathered  on  each  Clinical  Trial  Subject  pursuant  to  the
Protocol.

“Cell line”

means [***].

“Charity’s
Standard
Operating
Procedures”

means  the  documents  in  use  by  the  Centre  for  Drug  Development  of  the  Charity  from  time  to  time  that  are
designated  as  standard  operating  procedures  and  which  describe  the  procedures  that  must  be  followed  to
complete various tasks.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
“Chief
Investigator”

means the person who will lead and co-ordinate the work of the Clinical Trial overall where the Clinical Trial
is to be carried out at more than one site.

“Clinical Trial”

means the Phase I clinical trial described in the Protocol to be conducted under the Sponsorship of the Charity
and any Additional Studies.

“Clinical 
Database 
Date”

Trial
Lock

means  the  date  when  the  clinical  research  database  relating  to  the  Clinical  Trial  is  locked  (after  the  Clinical
Trial Results have been cleaned but excluding any Long Term Survival Data) in accordance with the Charity’s
Standard Operating Procedures.

“Clinical 
Legislation”

Trial

means all laws and regulations from time to time in force applicable to the performance of the Clinical Trial,
including the CTD, the Human Rights Act 1998, the Data Protection Act 1998, the Medicines Act 1968, the
Medicines for Human Use (Clinical Trials) Regulations 2004, and the Human Tissue Act 2004.

“Clinical 
LPFV Date”

Trial

means  the  date  when  the  final  Clinical  Trial  Subject  in  the  Clinical  Trial  attends  their  first  study  visit.  The
Clinical Trial LPFV Date may be further defined in the Protocol.

“Clinical 
Results”

Trial

means  all  Know-How,  data,  information,  results  and  improvements  Controlled  by  the  Charity  or  CRT  and
arising from the Clinical Trial, including the contents of each Progress Report, the Final Report, Case Report
Forms and associated Data Listings and any other updates that may be agreed by the Parties from time to time.

“Clinical 
Subject”

Trial

means  any  person  who  is  enrolled  in  the  Clinical  Trial  either  as  a  recipient  or  planned  recipient  of  the
Investigational Medicinal Product or as a control.

“Commencement
Date”

“Company  GMP
Materials”

“Company
Intellectual
Property”
“Company Know-
How”

means the date on which the Conditions Precedent have been satisfied.

means those Company Materials listed in Part 2 of Schedule 7.

means the Company Patent Rights, and all rights in the Company Know-How, the Investigational Medicinal
Product and the Company Materials.

means such Know-How in the Company’s Control relating to the Antibody and/or Investigational Medicinal
Product (and any constituents thereof), including: (i) any safety and toxicological data; (ii) information relating
to  the  manufacturing/production;  (iii)  information  relating  to  quality;  (iv)  information  relating  to  safe  and
proper  handling,  storage  and  use;  (v)  any  other  data  which  is  relevant  to  the  efficient  performance  of  the
Clinical Trial and/or would make the Investigational Medicinal Product in any way easier to make; and (vi) any
other data that would make the Antibody more useful, more valuable or in any way improve its prospects for
development or commercialisation.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
“Company
Materials”

means  the  Cell  Line  and  Materials  identified  in  Schedule  7  that  are  to  be  provided  by  the  Company  to  the
Charity pursuant to this Agreement.

“Company  Patent
Rights”

means  (i)  those  Patent  Rights  listed  in  Schedule  1;  (ii)  those  Patent  Rights  owned  by  or  licensed  to  the
Company which would be infringed by the unauthorised manufacture, use or sale in, or importation into, the
relevant country of the Antibody, Back-Up Antibodies and/or Investigational Medicinal Product; and (iii) all
Patent Rights deriving priority from (i) and (ii).

“Conditions
Precedent”

“Confidential
Information”

have the meaning given to them in Clause 2.1.

means  all  information  designated  as  confidential  by  any  Party  in  writing  together  with  all  other  information
which  relates  to  the  business,  affairs,  technology,  products,  developments,  trade  secrets,  Know-How,
personnel, customers, agents, distributors and suppliers of any Party or information which may reasonably be
regarded as the confidential information of the Disclosing Party. Subject to the terms of any licence agreement
entered into in relation to them, the Clinical Trial Results shall be the Confidential Information of the Charity
and CRT.

“Control”

means,  with  respect  to  Intellectual  Property  Rights,  possession  of  the  ability  (whether  through  ownership  or
licence, other than a licence granted under this Agreement) to access and provide the Know-How and Material
or grant the licences or sublicences or make the assignments as provided herein without violating the terms of
any agreement or other arrangement with any third party.

“Contributors”

means  the  Chief  Investigator,  the  Principal  Investigator(s),  the  Sub-Investigators,  the  Experts,  the  NHS
Trust(s) involved in the Clinical Trial, any sub-contractor of the Charity and/or any academic or not-for-profit
entity involved in the Clinical Trial.

“Costs”

“CTD”

means all actual prepaid and committed costs and expenses incurred from time to time in connection with the
Clinical  Trial,  including,  for  the  avoidance  of  doubt,  the  internal  personnel  costs  of  the  Charity  and  the
Charity’s Biotherapeutics Development Unit (BDU) and Formulation Unit.

means  the  European  Clinical  Trials  Directive  (Directive  2001/20/EC)  and  national  legislation  implementing
such Directive, as the same may be amended from time to time.

“Data Listings”

means  the  computer  generated  data  listings  produced  by  the  Charity  detailing  all  anonymised  patient  data
collected under the Clinical Trial other than the Long Term Survival Data.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
“Declaration 
Helsinki”

“Disclosing
Party”

of

means the 2008 version of the Helsinki Declaration of the World Medical Association.

has the meaning specified in Clause 5.1.

“Escrow Account”

means an investment account established by the Company with the Escrow Agent under the provisions of the
Escrow Agreement.

“Escrow Agent”

means Fifth Third Bank, a United States banking corporation with registered address at Fifth Third Square, 38
Fountain  Square  Plaza,  Cincinnati,  OH,  45263,  or  any  other  substantially  comparable  United  States  banking
corporation selected by mutual agreement of the Parties.

“Escrow
Agreement”

means  a  written  agreement  between  the  Parties  and  the  Escrow Agent  in  substantially  the  form  attached  as
Schedule  12,  and  under  which  the  Company  is  obliged  to  cause  the  Escrow  Agent  to  open  the  Escrow
Account, and deposit the Escrow Amount in the Escrow Account, before the Long Stop Date.

“Escrow Amount”

means a sum of of eight hundred thousand US dollars (US $800,000).

“Ethics
Committee”

“Exclusive
Results”

has the meaning given to it in the CTD.

means those Clinical Trial Results and the Intellectual Property Rights therein that directly relate to and only to
the IMP. Exclusive Results shall not include any assay methodology, formulation-related results or biomarker
results which do not directly relate to and only to the Investigational Medicinal Product.

“Exercise Notice”

has the meaning specified in Clause 7.1.

“Expert”

means  any  member  of  the  Charity’s  expert  committees  or  any  other  person  not  being  an  employee  of  the
Charity whom the Charity may engage from time to time to advise the Charity on the Clinical Trial.

“Final Report”

means  a  Report  Synopsis,  unless,  pursuant  to  Clause  3.10,  a  Full  Clinical  Study  Report  is  prepared  by  the
Charity instead of a Report Synopsis.

“Financial Year”

means the period commencing on January 1 and ending on December 31.

“Full 
Study Report”

Clinical

means  a  full  clinical  study  report  in  relation  to  the  Clinical  Trial  written  by  or  on  behalf  of  the  Charity  in
accordance  with  the  Charity’s  Standard  Operating  Procedures  and  which  meets  the  standards  of  the  ICH
Guidelines for Structure and Content of Clinical Study reports as per ICH Topic E3 dated July 1996 except that
Long Term Survival Data will not be included in the report.

“Full  CS  Report
Fee”

has the meaning given to it in Clause 3.10.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
“Good
Manufacturing
Practice”

means the principles and guidelines of good manufacturing practice in respect of medicinal products for human
use and investigational medicinal products for human use as defined in: (i) the CTD; (ii) European Community
Directive  2003/94/EC;  (iii)  European  Community  Directive  2005/28/EC;  (iv)  Eudralex  Volume  4:  ‘EU
Guidelines to Good Manufacturing Practice, Medicinal Products for Human and Veterinary Use, Part II Basic
Requirements  for  Active  Substances  used  as  Starting  Materials’,  ICHQ7a  Good  Manufacturing  Practice
Guidance  for  Active  Pharmaceutical  Ingredients  and  ‘EU  Guidelines  to  Good  Manufacturing  Practice
Medicinal  Products  for  Human  and  Veterinary  Use, Annex  13:  Investigational  Medicinal  Products’;  and  (v)
any  national  legislation  implementing  the  aforementioned  Directives  and  any  relevant  guidance  relating
thereto.

“ICH GCP”

means the latest version from time to time of the International Conference on Harmonisation (ICH) Tripartite
Guidelines,  Good  Clinical  Practice  (CPMP/ICH/135/95)  together  with  such  other  good  clinical  practice
requirements  as  are  specified  in  the  CTD  and  in  Commission  Directive  2005/28/EC  and  in  any  other
regulations  relating  to  medicinal  products  for  human  use  and  in  any  guidance  published  by  the  European
Commission pursuant to such Directives or regulations.

“Independent
Opinion”

means the opinion of an independent expert in the field of valuation of intellectual property in a similar field to
the  Company  Intellectual  Property,  appointed  by  agreement  between  the  Parties  or  in  default  of  such
agreement within twenty one (21) days of a Party seeking in writing to the others to appoint such expert, by the
President for the time being of the Association of the British Pharmaceutical Industry (ABPI) in England and
Wales, referred to at Clause 13.1.

“Intellectual
Property Rights”

means  all  Patent  Rights,  Know-How,  copyright,  database  rights,  design  rights,  moral  rights,  rights  in  trade
names,  logos  and  trade  and  service  marks,  domain  names,  rights  in  Materials  and  all  rights  or  forms  of
protection of a similar nature or having equivalent or similar effect to any of them which may subsist anywhere
in  the  world,  whether  or  not  any  of  them  are  registered,  including  any  application  for  registration  of  any  of
them.

“Investigational
Medicinal
Product” or
“IMP”

“Investigational
Medicinalor
Product Dossier”
or “IMPD”

means the pharmaceutical formulation of the Antibody suitable for use in the Clinical Trial.

means a dossier relating to the Investigational Medicinal Product which accompanies a request for clinical trial
authorisation to conduct the Clinical Trial from a Regulatory Authority. The Investigational Medicinal Product
Dossier shall include a specification of the IMP.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

“Know-How”

means all technical and other information which is not in the public domain, including information comprising
or  relating  to  concepts,  discoveries,  data,  designs,  formulae,  ideas,  inventions,  methods,  models,  designs  for
experiments  and  tests  and  results  of  experimentation  and  testing,  processes,  specifications  and  techniques,
laboratory  records,  clinical  data,  reports,  manufacturing  data  and  information  contained  in  submissions  to
Regulatory Authorities.

“Licence”

means a licence to the Clinical Trial Results and any Intellectual Property Rights therein in the form attached at
Schedule 3. Such licence shall be exclusive in respect of the Exclusive Results, and non-exclusive in relation to
the Non-Exclusive Results.

“Long Stop Date”

has the meaning given to it in Clause 2.2.

“Long 
Survival Data”

Term

means  any  ongoing  survival  data  for  Clinical  Trial  Subjects  that  the  Charity  collects  after  the  completion  of
the interventional component of the Clinical Trial.

“Losses”

means  losses,  damages,  costs  and  expenses  (including  reasonable  legal  costs  and  expenses),  in  each  case
directly incurred by a Party.

“Materials”

means  any  chemical  or  biological  substances  including  any:  organic  or  inorganic  element  or  compound;
nucleotide  or  nucleotide  sequence  including  DNA  and  RNA  sequences  gene;  vector  or  construct  including
plasmids, phages, bacterial vectors, bacteriophages and viruses; host organism including bacteria, fungi, algae,
protozoa and hybridomas; eukaryotic or prokaryotic cell line or expression system or any development strain
or  product  of  that  cell  line  or  expression  systems;  protein  including  any  peptide  or  amino  acid  sequence,
enzyme, antibody or protein conferring targeting properties and any fragment of a protein or a peptide enzyme
or  antibody;  drug  or  pro-drug;  assay  or  reagent;  any  plasma  or  tissue;  or  any  other  genetic  or  biological
material or micro-organism or any transgenic animal.

“Non-Exclusive
Results”

means those Clinical Trial Results that are not Exclusive Results (and all Intellectual Property Rights therein),
including all assay methodology, formulation-related results or biomarker results.

“Option”

has the meaning specified in Clause 7.1.

“Option Fee”

means  the  sum  of  [***]  less  the  amount  of  any  Full  CS  Report  Fee  actually  paid  by  the  Company  to  CRT
under Clause 3.10 and excluding VAT or other applicable sales tax.

“Option Period”

has the meaning specified in Clause 7.1.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

“Party”

means any party to this Agreement and “Parties” means all of them.

“Patent Rights”

means any patent applications, patents, author certificates, inventor certificates, utility models, and all foreign
counterparts  of  them  and  includes  all  divisionals,  renewals,  continuations,  continuations-in-part,  extensions,
reissues,  substitutions,  confirmations,  registrations,  revalidations  and  additions  of  or  to  them,  as  well  as  any
Supplementary Protection Certificate, or any like form of protection (including any pediatric, orphan drug or
other exclusivity granted by a Regulatory Authority beyond the expiry of the original patent expiration date).

“Principal
Investigator”

“Progress
Report”

means the person who will lead and co-ordinate the work of the Clinical Trial at a particular Clinical Trial site.

means a report on the status of the Clinical Trial in the format set out in Schedule 10, or in such other format as
is the Charity’s standard practice at the relevant time in respect of a clinical trial at the same stage, and of the
same scope, as the Clinical Trial.

“Protocol”

means the clinical trial protocol to be prepared by the Charity and the Chief Investigator as may be amended
from time to time by the Charity in accordance with Clause 3.6.

“Recipient Party”

has the meaning specified in Clause 5.2.

“Regulatory
Authority”

“Report
Synopsis”

means  any  local,  national  or  supra-national  agency,  authority,  department,  inspectorate,  minister,  ministry
official or public or statutory person (whether autonomous or not) or any government of any country as shall
have jurisdiction over the Clinical Trial or any part of it or over any activity of the Parties in connection with
the  Clinical  Trial.  Regulatory Authority  includes,  but  is  not  limited  to,  the  United  Kingdom  Medicines  and
Healthcare  products  Regulatory Agency  (MHRA),  the  United  States  Food  and  Drug Administration  (FDA)
and the European Medicines Agency (EMEA).

a  summary  of  the  results  of  the  Clinical  Trial  written  by  or  on  behalf  of  the  Charity  in  accordance  with  the
Charity’s Standard Operating Procedures in a form substantially similar to the format set out in Schedule 2 and
the  format  of  the  clinical  study  synopsis  set  out  in Annex  I  of  ICH  Topic  E3  of  the  ICH  Guidelines  for
Structure  and  Content  of  Clinical  Study  reports  dated  July  1996.  The  Report  Synopsis  shall  not  include  or
contain  any  additional  documents  or  any  appendices,  exhibits  or  annexes  nor  shall  it  include  or  contain  any
Data  Listings,  Case  Report  Forms  or  any  raw  data  comprised  within  the  Clinical  Trial  Results  or  cover  any
Long Term Survival Data.

“uPAR”

means [***].

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

[***]

means any and all research programmes undertaken by or on behalf of the Company, Tactic Pharma LLC or
by Attenuon, LLC, or any of their Affiliates, and in the course of which the Antibody or the antibody known as
ATN-658  or  any  of  the  Back-Up  Antibodies  were  discovered,  generated  or  developed  (including  but  not
limited to development activities conducted after the Commencement Date).

“Signature

means the period of [***] commencing on:

Period”

(i)  in  the  event  that  the  Charity  does  not  prepare  a  Full  Clinical  Study  Report  pursuant  to  Clause  3.10,  the
Company’s receipt of the Data Listings pursuant to Clause 7.3; or
(ii) in the event that the Charity prepares a Full Clinical Study Report pursuant to Clause 3.10, the date of the
Exercise Notice.

“Sub-
Investigator”

means a clinician appointed and supervised by the Chief Investigator or Principal Investigator to assist in the
carrying out of the Clinical Trial at the same trial site as the Principal Investigator.

“Supplementary  
Protection
Certificate”

means  a  right  based  on  a  patent  pursuant  to  which  the  holder  of  the  right  is  entitled  to  exclude  third  parties
from  using,  making,  having  made,  selling  or  otherwise  disposing  or  offering  to  dispose  of,  importing  or
keeping the product to which the right relates, such as supplementary protection certificates in Europe, and any
similar right anywhere in the world.

“Tactic”

Tactic Pharma LLC, an Illinois limited liability company based at [***].

“Tobacco Party”

means:  (i)  any  entity  who  develops,  sells  or  manufactures  tobacco  products;  and/  or  (ii)  any  entity  which
makes  the  majority  of  its  profits  from  the  importation,  marketing,  sale  or  disposal  of  tobacco  products.
Furthermore, Tobacco Party shall include any entity that is an Affiliate of any entity referred to in (i) or (ii).

“Transfer
Documents”

means the following documents: (i) the asset contribution agreement between the Company and Tactic dated
20 January 2015 (and as amended on 20 January 2015); the assignment and assumption of licence agreement
between the Company and Tactic dated 20 January 2015; and (iii) the letter from Tactic to the Parties dated 12
March 2015 in respect of the Cell Line and related Intellectual Property Rights.

“XOMA IP”

means any and all Intellectual Property Rights licensed to the Company under the XOMA Licence.

“XOMA Licence”

means the agreement entered into between XOMA (US) LLC and Tactic on 24 September 2014 in respect of
the Antibody, which was assigned to the Company by Tactic pursuant to an agreement dated 20 January 2015.
Both agreements are attached in Schedule 9.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

“XOMA  Licence
Payments”

means those milestone payments set out in the XOMA Licence.

1.2

In this Agreement:

1.2.1

unless the context requires otherwise, all references to a particular Clause, paragraph or Schedule shall be references to that
clause, paragraph or schedule, of or to this Agreement;

1.2.2

the table of contents and headings are inserted for convenience only and shall be ignored in construing this Agreement;

1.2.3

1.2.4

1.2.5

1.2.6

unless the contrary intention appears, words importing the masculine gender shall include the feminine and vice versa and
words in the singular include the plural and vice versa;

unless  the  contrary  intention  appears,  words  denoting  persons  shall  include  any  individual,  partnership,  company,
corporation, joint venture, trust, association, organisation or other entity, in each case whether or not having separate legal
personality;

reference to any statute or regulation includes any modification or re-enactment of that statute or regulation, provided that
the modification or re-enactment does not diminish the rights or extend the obligations of any Party; and

references to the words “include” or “including” shall be construed without limitation to  the  generality  of  the  preceding
words.

2.

2.1

CONDITIONS PRECEDENT

Notwithstanding anything to the contrary in this Agreement, the Charity and CRT shall have no obligations, nor have any liability,
of  any  nature  howsoever  arising  under  or  in  connection  with  this Agreement  unless  and  until  the  following  conditions  precedent
have been satisfied:

2.1.1

the valid execution of the Escrow Agreement; and

2.1.2

2.1.3

the Company’s performance of its obligations under the Escrow Agreement to open the Escrow Account and deposit the
Escrow Amount in it; and

the Company’s delivery to the Charity of written evidence to the Charity’s reasonable satisfaction that the Company has
obtained insurance described in Clause 9.5,

(the “Conditions Precedent”).

2.2

If the Conditions Precedent have not been satisfied by 14:00pm (BST) on the date falling [***] after the date of signature of this
Agreement (the “Long Stop Date”), the Agreement shall expire on the Long Stop Date.

2.3

The Company shall use its best endeavours to satisfy the Conditions Precedent before the Long Stop Date.

3.

3.1

CONDUCT OF THE CLINICAL TRIAL AND SPONSORSHIP

Subject  to:  (i)  the  Company’s  compliance  with  its  obligations  hereunder;  and  (ii)  the  Ethics  Committee  and  the  Regulatory
Authority granting consent for the Clinical Trial, the Charity will use its reasonable endeavours to carry out or procure the carrying
out of the Clinical Trial in accordance with the Protocol.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
3.2

3.3

3.4

3.5

Once the Clinical Trial has been opened to Clinical Trial Subjects, the Charity shall use reasonable endeavours to provide to the
Company at least one Progress Report per month (or with the frequency that is the Charity’s standard practice at the relevant time
in respect of a clinical trial at the same stage, and of the same scope, as the Clinical Trial, but no less frequently than quarterly). The
Company may use the Progress Reports for the purpose of determining whether or not to exercise the Option. All Progress Reports
and any supplementary information provided under them shall be the Confidential Information of the Charity and the provisions of
Clause  5  shall  apply.  The  Company  acknowledges  that  information  or  data  provided  under  this  Clause  3.2  may  not  be  verified,
clean or accurate, and is provided “as is”. Without prejudice to the generality of Clause 8.7, neither CRT nor the Charity make any
representation or warranty (express or implied) of any nature in respect of such data or information, including as to its accuracy,
quality, usefulness or comprehensiveness.

The Charity may, at its sole discretion: (i) sub-contract to third parties any part of the Clinical Trial; and (ii) engage such Experts
and such persons to fulfil the roles of Chief Investigator and/or Principal Investigator as the Charity deems appropriate. Company
shall  be  notified  of  any  such  third  parties,  Experts  and  persons  set  forth  in  this  clause  3.3,  and  the  Charity  may  make  such
notification by email.

The Charity shall, at its own expense, be responsible for seeking approval of the Clinical Trial and the Protocol from the Regulatory
Authority and Ethics Committee prior to commencing the Clinical Trial. For the avoidance of doubt, the Charity shall not be held
liable  or  responsible  for  any  failure  and/or  refusal  by  the  Ethics  Committee  or  the  Regulatory Authority  to  grant  consent  for  the
Clinical Trial or any change required therein.

The Charity shall use reasonable endeavours to carry out, or procure the carrying out of, the Clinical Trial in accordance with the
relevant aspects of:

3.5.1

Clinical Trial Legislation; and

3.5.2

ICH GCP and the Declaration of Helsinki.

Any breach of this Clause 3.5 shall be a material breach.

3.6

The Charity shall be free to amend the Protocol or to change the third party undertaking any part of the Clinical Trial as it deems
appropriate, provided that such Protocol or change to the Protocol has first been approved by the Ethics Committee and, if required
by law or regulation, the Regulatory Authority; and further provided that:

3.6.1

3.6.2

prior  to  submission  for  Ethics  Committee  approval,  the  Charity  shall  provide  to  the  Company  a  copy  of  the  first  final
version of the Protocol at least fourteen (14) days before seeking Ethics Committee approval and give due consideration to
any comments received from the Company by the Charity within such time.

the Charity shall notify the Company in writing of any proposed changes to the Protocol at least fourteen (14) days before
seeking Ethics Committee approval for such changes, and shall give due consideration to any comments that the Company
might make within such time. In an emergency (such as patient safety needs) the said fourteen (14) day time period may be
reduced to such time period as the Charity is actually able to give to the Company in the circumstances and the Charity
may,  if  in  its  reasonable  opinion  it  is  required,  submit  such  changes  to  the  Ethics  committee  prior  to  notifying  the
Company of such. The Charity will try to reach a consensus with the Company on all issues arising out of the Company’s
review of any Protocol pursuant to this Clause 3.6.2, but the Charity shall have the final decision.

 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

3.6.3

in the event that the Ethics Committee and/or the Regulatory Authority does not approve the original Protocol and/or agree
to  any  amendment  to  the  Protocol,  the  Charity  shall  have  the  right  to  terminate  this Agreement  forthwith  upon  written
notice to the Company.

3.7

3.8

The Charity shall have sole responsibility for the conduct and control of the Clinical Trial and shall accept the obligations of the
sponsor  of  the  Clinical  Trial  in  accordance  with  the  requirements  of  the  Medicines  for  Human  Use  (Clinical  Trials)  Regulations
2004.

The Charity shall use reasonable endeavours to procure that Clinical Trial Subjects are recruited in accordance with the selection
procedures and criteria set out in the Protocol.

3.9

The Charity shall promptly advise the Company, in writing, of the occurrence of the Clinical Trial LPFV Date.

3.10

The Company may elect to receive a Full Clinical Study Report instead of a Report Synopsis by:

3.10.1

providing the Charity with written notice of its election to receive a Full Clinical Study Report, which written notice must
be received by the Charity before the expiration of thirty (30) days from the date the Charity advised the Company of the
occurrence of the Clinical Trial LPFV Date; and

3.10.2

paying  the  Charity  the  sum  of [***]  excluding  VAT  or  other  applicable  sales  tax  (the  “ Full  CS  Report  Fee”)  within
twenty one (21) days after service of such notice.

If the Company does not serve a written notice and pay the Full CS Report Fee as specified in this Clause 3.10, the Charity shall prepare a

Report Synopsis and shall have no obligation to prepare or provide the Company with a Full Clinical Study Report.

3.11

The Charity shall provide the Final Report to the Company and CRT within [***] after the Clinical Trial Database Lock Date.

3.12

4.

4.1

The Charity shall only use the Investigational Medicinal Product for the purposes of carrying out the Clinical Trial and shall not
permit any third party to use the Investigational Medicinal Product except as required for the purpose of carrying out the Clinical
Trial or as set out in this Agreement.

COMPANY’S OBLIGATIONS

The Company shall at the Company’s sole cost, provide the Charity with:

4.1.1

such  information  and  Know-How  relating  to  the  manufacture  of  the  IMP  as  is  relevant  to  the  efficient  production  of
sufficient quantity of the IMP to conduct the Clinical Trial, as soon as practicable following the Commencement Date;

4.1.2

all Company Know-How and the Company Materials as soon as practicable following the Commencement Date;

4.1.3

any other information in the Company’s Control pertaining to the safety of the IMP or which in the reasonable opinion of
the Company may have a bearing on the conduct of the Clinical Trial as soon as the same comes to the attention of the
Company.

4.1.4

such scientific and technical guidance as the Charity may reasonably request to enable the Charity and the Contributors to
conduct and manage the Clinical Trial in a safe and proper manner; and

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
4.1.5

all  information  (including  information  for  inclusion  in  the  Investigational  Medicinal  Product  Dossier)  and  co-operation
reasonably  requested  by  the  Charity  at  any  time  from  the  Commencement  Date  to  enable  the  Charity  to  compile  an
Investigational Medicinal Product Dossier; provided that such requested information is in the Company’s Control (which
shall include all information transferred, and all information which the Company is entitled to request or Control, under the
Transfer Documents). In the case of co-operation requested under this Clause 4.1.5, the Company shall procure (at its own
cost) that any subcontractor which has performed activities or produced documents on its behalf under this Agreement is
made available to the Charity on such notice, for such time and with such frequency as may be reasonably requested by the
Charity. The Company shall provide information requested by the Charity within fourteen (14)  days  of  request  (or  such
other period as may be reasonable given the nature of the request).

4.2

4.3

The Company shall provide to the Charity any and all data, documentation, information and Know-How described in Clauses 4.1.1
to  4.1.5  on  an  ongoing  basis  within  a  reasonable  time  after  the  same  comes  to  the  attention  of  the  Company  (if  already  in  the
Company’s Control), or into the Company’s Control, after the Commencement Date.

The  Company  will  keep  the  Charity  informed  of  the  scope  and  results  of  any  pre-clinical  or  other  non-clinical  studies  being
undertaken by it or with third parties in relation to the Antibody or Back-Up Antibodies. If the Company is intending to transfer the
Antibody or undertake any new research in relation to the Antibody or a Back-Up Antibody with a third party, it will consult with
the  Charity  on  the  scope  of  the  intended  research  and  the  identity  of  the  third  party  and  take  into  good  faith  consideration  any
comments  the  Charity  may  have  in  respect  to  the  same.  This  Clause  should  not  be  interpreted  to  limit  any  restrictions  on  the
Company’s use of the Antibody or any Back-Up Antibody under Clause 6.1 or elsewhere in this Agreement.

4.4

The Company shall submit to CRT:

4.4.1

4.4.2

a copy of its detailed operating budget for development of the Antibody  (including a quarterly cash flow and expenditure
forecast) in respect of each Financial Year as adopted by the Company’s board (the “ Annual Budget”), at least thirty (30)
days prior to the commencement of the Financial Year to which the Annual Budget relates; and

quarterly  management  accounts  of  the  Company  (to  include,  inter  alia,  a  (consolidated)  profit  and  loss  account,  balance
sheet and cash flow statement and shall indicate where such management accounts differ to any material extent from the
Annual Budget for such period), within sixty (60) days of the end of the period to which they relate; save that the accounts
relating to the final quarter in any calendar year may be provided within ninety five (95) days, rather than sixty (60) days,
of the end of that quarter. Such quarterly management accounts shall be prepared on a basis which is consistent with those
adopted in the preparation of all previous management accounts of the Company.

4.5

4.6

The Company shall generally keep CRT informed of the progress of the Company's business and affairs and shall promptly supply
CRT with written details of any circumstances which will or might cause any actual or prospective material adverse change in the
financial position, prospects or business of the Company.

As between the Parties, the Company will be solely responsible for any and all payments due under the XOMA Licence that may
become due as a result of the grant of rights to the Charity under this Agreement or the carrying out the Clinical Trial in accordance
with this Agreement.

 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

4.7

5.

5.1

Following  its  receipt  of  the  Company  GMP  Material,  the  Charity  will  assess  whether  or  not  it  wishes  to  use  the  Company  GMP
Material to manufacture IMP. At the Charity’s request, the Charity and the Company shall negotiate in good faith the terms of a
technical agreement that sets out the responsibilities of each Party in respect of IMP and the GMP aspects of manufacturing IMP
(the “Technical Agreement”). Negotiations shall take place and be concluded within [***] of the Charity’s request for a Technical
Agreement. If required, the Technical Agreement will be in a form substantially similar to that set out in Schedule 13.

CONFIDENTIALITY/PUBLICATION

Subject to Clause 5.5, each Party shall keep confidential and not disclose to any third party (other than the Experts, Contributors,
Ethics  Committee,  Regulatory  Authority  and  staff  involved  in  carrying  out  the  Clinical  Trial  on  a  need  to  know  basis)  any
Confidential  Information  disclosed  to  it  by  another  Party  (the  “Disclosing  Party”)  without  the  prior  written  consent  of  the
Disclosing Party. For the avoidance of doubt, the Charity shall be permitted to disclose Confidential Information disclosed to it to
CRT  and  CRT  shall  be  permitted  to  disclose  Confidential  Information  disclosed  to  it  to  the  Charity.  Any  party  to  whom
Confidential Information is disclosed in accordance with this Clause 5.1 shall be:

5.1.1

subject to no less onerous obligations than those contained in this Clause 5 to keep such information confidential; and

5.1.2

advised of its confidential nature.

5.2

The  obligations  of  confidence  referred  to  in  Clause  5.1  shall  not  apply  to  any  part  of  the  Confidential  Information  which  can  be
proved by evidence in writing:

5.2.1

was known to the recipient Party (the “Recipient Party”) before its disclosure by the Disclosing Party;

5.2.2

was available to the public before that date or was otherwise in the public domain;

5.2.3

becomes available to the public or enters the public domain after that date otherwise than as a result of an act or default of
the Recipient Party;

5.2.4

is received by the Recipient Party from a third party not bound to the Disclosing Party by any obligation of secrecy;

5.2.5

5.2.6

is independently developed or generated by the Recipient Party in circumstances where it has not been derived directly or
indirectly from the Disclosing Party’s Confidential Information; or

is required to be disclosed by: (i) law, (ii) a Regulatory Authority; or (iii) an order of any court, provided however, that in
each  such  event  the  Recipient  Party  required  to  disclose  the  Confidential  Information  shall  give  prompt  notice  to  the
Disclosing Party of such requirement so that such Disclosing Party may seek a protective order or other appropriate remedy
to the extent of such disclosure.

The obligations of the Parties under Clause 5.1 shall survive the expiry or termination of this Agreement for whatever reason for a
period of ten (10) years from the date of such expiry or termination.

Each of the Parties agrees that the provisions of this Clause 5 are fair and reasonable and that money damages are not a sufficient
remedy for any breach of this Clause 5 and therefore, in addition to all other remedies, all Parties shall be entitled to seek injunctive
or other equitable relief as a remedy for such breach.

Notwithstanding  any  confidentiality  obligations  assumed  by  the  Parties  hereunder,  the  Parties  acknowledge:  i)  the  importance  of
publications  to  the  academic  standing  of  the  Charity  and  the  Contributors;  and  ii)  the  capital  raising,  transactional,  and  licensing
prospects of the Company; and iii) the reporting and disclosure obligations of the Company to its investors and to XOMA under the
XOMA  Licence. Accordingly,  the  Parties  have  agreed  as  follows  as  regards  publication  of  Clinical  Trial  Results  and  Progress
Reports:

5.3

5.4

5.5

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
5.5.1

5.5.2

The  Charity  shall  use  reasonable  endeavours  to  publish,  or  procure  the  publication  by  the  Contributors  of,  the  Clinical
Trial Results in a timely manner in accordance with generally accepted academic practice, whether during the course of or
after completion of the Clinical Trial.

The Company may disclose the content of Progress Reports to XOMA only to the extent it is required to do so under the
XOMA Licence, provided that the disclosure will exclude all information regarding clinical responses and shall be limited
to only information regarding the clinical indication, anticipated timelines of the trial, the number of patients dosed, and
such other information of a similar nature as may be reasonably required by the XOMA Licence.

5.5.3

The Company may disclose:

(a)

(b)

(c)

the content of Progress Reports to a third party in connection with capital raising, financing, transactional, and/or
licensing  activities  or  prospects  for  the  benefit  of  the  Company.  Prior  to  making  such  disclosure,  the  Company
shall  give  notice  to  the  Charity,  including  details  of  the  content  of  the  proposed  disclosure  and  the  reason  for
wishing to make such disclosure, and shall inform the Charity of the identity of the third party in its notice unless
it is prevented from doing so due to express confidentiality restrictions owed to, and requested by, the third party,
in  which  case  the  Company  shall  state  the  main  business  area  within  which  the  third  party  operates.  The
Company may, without the Charity’s prior approval, disclose only the clinical indication, anticipated timelines of
the  trial,  and  the  number  of  patients  dosed,  but  shall  obtain  the  Charity’s  approval  before  proceeding  with  any
other disclosure under this Clause 5.5.3(a);

the Final Report to the Company’s consultants and professional advisors, solely for the purpose of assisting in the
evaluation of the results with a view to exercise of the Option and provided that no patient data shall be disclosed
unless it has been cleansed; and

the content of Progress Reports to persons holding investments in the Company, solely for the purpose of a status
update, such as periodic disclosure of recruitment numbers to investors in the Company by way of demonstration
of progress in the Clinical Trial.

5.5.4

It is further provided that each disclosure of the content of Progress Reports by the Company under this Clause 5.5 shall be
subject to the following conditions:

(a)

(b)

all recipients shall be informed in writing beforehand of the confidential nature of the information being disclosed
and shall have agreed in writing to obligations of confidentiality in favour of the Company no less onerous than
those  contained  in  this  Clause  5  (but  without  any  right  of  further  disclosure)  to  keep  such  information
confidential; and

only the content of the documents containing the relevant information which has been processed into a suitable
format may be disclosed but not copies of the actual documents themselves.

 
 
 
 
 
 
 
 
 
 
 
5.6

5.7

The Charity will include provisions in its contracts with the Contributor(s) that require such Contributor(s) to notify the Charity in
advance of submission of any abstract, presentation or manuscript incorporating Clinical Trial Results that the Contributor(s) wish
to publish or have published or to present or have presented.

Upon receipt of such notification from a Contributor or if the Charity wishes itself to publish or have published or to present or have
presented an abstract, presentation or manuscript incorporating Clinical Trial Results the Charity shall so notify the Company and
CRT and provide (in so far as it is able to do so in the case of a Contributor’s notification) in response to the Company’s and/or
CRT’s reasonable request a copy or summary thereof at least seven (7) days prior to submission for publication of an abstract or
presentation  or  at  least  thirty  (30)  days  prior  to  submission  for  publication  of  a  manuscript  (or  twenty  one  (21)  days  prior  to
submission  for  publication  of  a  manuscript  in  the  case  of  a  Contributor’s  notification).  Any  such  copy  or  summary  shall
provide sufficient details to enable the Company and CRT to ascertain whether it contains Confidential Information of the Company
or CRT respectively or whether Patent Rights or other proprietary protection should be sought.

5.8

The  Company  and  CRT  shall  review  and  make  any  comments  on  such  intended  publication  or  presentation  of  an  abstract  to  the
Charity  within  seven  (7)  days  and/or  shall  review  and  make  any  comments  on  such  intended  publication  or  presentation  of  a
manuscript within thirty (30) days. The Company and/or CRT may request that:

5.8.1

5.8.2

Confidential  Information  of  the  Company  (not  including  Clinical  Trial  Results  nor  information  directly  relating  to  the
Investigational Medicinal Product) or Confidential Information of CRT (not including Clinical Trial Results) be removed
from the proposed publication or presentation; and/or

any such publication or presentation be delayed if in the Company’s or CRT’s reasonable opinion it is necessary to delay
publication or presentation in order to file a patent application or application for other proprietary protection in respect of
any invention made in the course of the Clinical Trial. Any such delay will be kept to the minimum period practicable and
will in no event extend beyond thirty (30) days from the date the proposed publication or presentation was provided to the
Company.

In the event of a request pursuant to Clauses 5.8.1 or 5.8.2, the Company or CRT (as the case may be) shall provide the Charity
with a written explanation of the reasons why it believes information should be removed or a delay is necessary. For the avoidance
of doubt, any Patent Rights filed pursuant to Clause 5.8.2 shall be filed in CRT’s name unless any Company personnel are deemed
inventors on any such filing, in which case such Patent Right shall be filed in both CRT’s and Company’s names. As used herein,
inventorship shall be determined in accordance with English law.

5.9

5.10

The Charity and CRT shall be entitled to publish information in relation to the proposed Clinical Trial, including that it is or will be
a trial conducted by the Clinical Development Partnerships initiative set up by the Charity and CRT, the pre-requisites for patient
recruitment,  a  brief  description  of  the  Clinical  Trial,  including  the  name  of  the  Company,  the  reference  number  and  class  of  the
Investigational Medicinal Product and the location(s) at which the trial is taking place.

In addition to the disclosures under Clause 5.5, the Company may disclose the commercial terms of this Agreement to any actual or
potential  investors,  bankers,  acquirers,  acquirees  or  merger  partners,  in  each  case  under  appropriate  confidentiality  provisions
substantially equivalent to those of this Agreement.

 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

5.11

6.

6.1

Except  as  expressly  permitted  in  Clause  5,  the  Company  shall  not  disclose  the  Clinical  Trial  Results  to  any  potential  investors,
licensees or sub-licensees of the Company (or any other person) until the Company has been granted the Licence.

INTELLECTUAL PROPERTY RIGHTS

The Company hereby grants to the Charity with a right to sub licence to Contributors:

6.1.1

the [***] of the Investigational Medicinal Product;

6.1.2

the [***] relating to the Investigational Medicinal Product;

6.1.3

an [***] under the Company Intellectual Property; and

6.1.4

a [***] under the XOMA IP,

               on a [***] basis for the purpose of preparing for and carrying out (and having prepared or carried out for the Charity) the Clinical
Trial. The Company shall not be entitled to (and shall (i) procure that its Affiliates do not, and (ii) not authorise any other third party
to) conduct any clinical trials in respect of the Antibody or any Back-Up Antibody during the term of this Agreement.

6.2

6.3

6.4

The  Company  shall  use  commercially  reasonable  endeavours  to  continue  to  prosecute  and  maintain,  at  its  own  cost,  all  of  the
Company  Patent  Rights.  If  the  Company  intends  to  substantially  narrow  the  scope  of  the  claims  of  any  Patent  Rights  within  the
Company Patent Rights it will first consult with CRT and take into good faith consideration any concerns or views expressed by
CRT. If the Company elects not to prosecute or maintain any part of the Company Patent Rights, the Company shall notify CRT in
writing within a reasonable period and no less than [***] prior to the expiration of any applicable time bars. After receipt of such
notice, CRT may elect, before the expiry of any such time bars, by written notice to the Company, to take an assignment to any
Company Patent Rights identified in such notice at CRT’s sole discretion and for consideration not exceeding [***]. In the event
that  CRT  elects  to  take  such  an  assignment,  the  Company  shall,  at  CRT’s  expense,  promptly  transfer  to  CRT  (or  any  person
nominated  by  CRT)  copies  of  any  and  all  documents  in  the  Company’s  Control  relating  to  the  filing,  prosecution,  maintenance,
enforcement  and  defence  of  such  Company  Patent  Rights.  The  Company  shall  not  assign,  charge,  encumber  or  dispose  of  any
interest in any of the Company Intellectual Property to a Tobacco Party or in a manner that limits or impairs the Charity’s or CRT’s
rights under the licence (or assignment, where applicable) of Company Intellectual Property pursuant to this Agreement without the
Charity’s or CRT’s prior written consent.

As between the Company and the Charity, [***]. The Charity hereby [***]. CRT hereby [***].

Subject to [***], the Company shall [***].

 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

6.5

6.6

6.7

6.8

6.9

7.

7.1

7.2

7.3

7.4

7.5

Solely in connection with the Charity’s and the Contributors’ activities performed pursuant to the Clinical Trial, where carried out in
accordance with the terms of this Agreement, the Company shall not, and shall procure that its Affiliates shall not, anywhere in the
world,  institute  or  prosecute  (or,  other  than  as  required  by  law,  in  any  way  aid  any  third  party  in  instituting  or  prosecuting)  any
claim,  demand,  action  or  cause  of  action  for  damages,  costs,  expenses  or  compensation,  or  for  an  enjoinment,  injunction,  or  any
other  equitable  remedy,  alleging  the  infringement  by  the  Charity  and/or  any  Contributors  of  any  Patent  Rights  of  the  Company
and/or any Patent Rights of the Company’s Affiliates. For the avoidance of doubt, the foregoing shall not apply in respect of: (i)
development, at any time, of products other than the IMP; or (ii) any activity in relation to the IMP which constitutes a breach of the
terms of this Agreement.

Any  breach  of  Clause  6.5  shall  be  a  material  breach  and  shall  accordingly  entitle  the  Charity  to  terminate  this Agreement  under
Clause 11.2.

CRT hereby reserves and excludes from the Option, the worldwide, perpetual and irrevocable right in and to the Exclusive Results
for the Contributors and the Charity (including scientists funded and/or employed by the Charity) to:

6.7.1

use  the  Exclusive  Results  for  the  purpose  of  non-commercial  scientific  research  carried  out  by  or  for  or  under  their
respective direction in accordance with their respective charitable and/or academic status, whether alone or in collaboration
with a third party or third parties; and

6.7.2

grant licences under, and make available, the Exclusive Results solely to the extent necessary to exercise the rights under
Clause 6.7.1, but not otherwise.

For the avoidance of doubt, CRT shall be entitled, at its discretion, at any time (including during the Option Period) to grant non-
exclusive licences to the Non-Exclusive Results to any person and for any purpose.

Neither Charity nor CRT, or any affiliate or agent of Charity or CRT, shall institute any type of proceeding in a court, governmental
agency, or patent office anywhere throughout the world for the purposes of invalidating, narrowing, or reducing the term of one or
more  claim  in  an  issued  patent  or  pending  patent  application.  The  institution  of  any  such  proceeding  during  the  term  of  this
agreement and afterwards during the term of Company’s Patent Rights shall be a material breach and shall accordingly entitle the
Company to terminate this Agreement under Clause 11.2.

OPTION

CRT  grants  to  the  Company  the  option,  exercisable  by  notice  to  CRT  in  writing  (the  “ Exercise Notice”)  at  any  time  during  the
[***] period after the Company receives the Final Report (the “Option Period”), to enter into the Licence (the “Option”). Subject
to Clause 6.7, the Option shall be [***]
Upon exercise of the Option, the Company shall pay the Option Fee to CRT within the Option Period.

Save  where  the  Charity  has  provided  a  Full  Clinical  Study  Report,  CRT  shall  procure  the  provision  of  the  Data  Listings  to  the
Company following the exercise of the Option and the receipt by CRT of the Option Fee.

If the Company exercises the Option, CRT and the Company shall execute the Licence within the Signature Period.

If:

7.5.1

the Company does not exercise the Option within the Option Period; or

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

7.5.2

following the exercise of the Option, the Company does not enter into the Licence within the Signature Period,  then the
Company shall, within [***] of the expiry of the Option Period or Signature Period (as applicable):

a)

b)

assign the Company Intellectual Property and sub-license the XOMA IP to CRT by executing an agreement in the
form attached at Schedule 5, and CRT shall be free to license or otherwise grant rights in respect of the Clinical Trial
Results and the Intellectual Property Rights in the Clinical Trial Results on such terms and to such third parties as it
shall see fit; and

provide  CRT  with  such  assistance  as  CRT  may  reasonably  request  in  liaising  with  XOMA  for  the  purpose  of
obtaining direct contractual rights with XOMA in respect of the XOMA IP.

8.

8.1

WARRANTIES AND LIMITS OF LIABILITY

The Charity warrants that:

8.1.1

it will procure the discharge of its obligations hereunder with reasonable care and skill; and

8.1.2

it will use its reasonable endeavours to procure that each Contributor that carries out part of the Clinical Trial ensures that
the  relevant  Chief  Investigator  and/or  the  Principal  Investigator  discharge  their  obligations  in  respect  of  that  part  of  the
Clinical Trial in accordance with applicable ICH GCP provisions.

8.2

The Company warrants and represents that:

8.2.1

it is entitled to make the Company Materials available to the Charity for the purposes of this Agreement;

8.2.2

8.2.3

to  the  best  of  its  knowledge  and  belief  the  use  and  possession  of  the  Company  Materials  and/or  the Antibody  by  the
Charity and/or the Contributors shall not infringe the rights (including without limitation any Intellectual Property Rights)
of any third party;

the  Company  Materials  have  been  manufactured,  handled  and  stored  at  all  times  in  compliance  with  relevant  legislation
and, in the case of relevant Company Materials (including the Company Materials identified in Part 2 of Schedule 7), in
accordance with Good Manufacturing Practice;

8.2.4

it is a party to the XOMA Licence, which is in full force and effect;

8.2.5

it  has,  and  will  maintain  throughout  the  Term,  the  full  right,  power  and  authority,  and  has  obtained  all  assignments,
approvals or consents necessary to grant the rights, including under the Transfer Documents and the XOMA Licence, as
provided under this Agreement;

8.2.6

the XOMA Licence is the only third party licence held by the Company in respect of the manufacture, possession and use
of the Antibody, IMP and the rights granted to the Charity under this Agreement;

8.2.7

the XOMA Licence set out in Schedule 9 is a true and correct copy of the XOMA Licence;

8.2.8

to  the  best  of  its  knowledge  and  belief,  there  are  no  outstanding  breaches  of  the  XOMA  Licence  by  any  party  (or  any
predecessor parties) to the XOMA Licence;

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
8.2.9

to  the  best  of  its  knowledge  and  belief  there  are  no  acts,  facts,  circumstances  or  omissions  at  the  Commencement  Date
which would give XOMA the right to terminate the XOMA Licence, either now or at a later date;

8.2.10

it shall maintain, and shall not amend or terminate the XOMA Licence without CRT’s prior written consent; and

8.2.11

it shall notify the Charity and CRT as soon as possible if it becomes aware of any facts, circumstances or omissions which
may give XOMA the right to terminate the XOMA Licence.

References to the “best of its knowledge and belief” in Clause 8.2 shall include any knowledge within the Company or its Affiliates, and,

where relevant, of any predecessor party to the XOMA Licence, having made due and proper enquiries.

8.3

8.4

8.5

8.6

8.7

9.

9.1

The  Company  warrants  and  represents  that  all  information  and  Know-How  supplied  to  the  Charity  and/or  CRT  pursuant  to  this
Agreement (including any safety information) shall be accurate and complete and shall be supplied as soon as practicable following
the Commencement Date to enable the Charity to conduct and manage the Clinical Trial in a safe and proper manner.

Nothing in this Agreement shall exclude or limit the liability of any Party for death or personal injury resulting from its negligence
or the negligence of its employees while acting in the course of their employment or shall exclude or limit the liability of any Party
for fraud.

Subject  to  Clause  8.4,  the  entire  aggregate  liability,  for  any  loss  or  damage  arising  from  any  act  or  omission  relating  to  this
Agreement  regardless  of  the  form  of  action,  whether  in  contract  or  tort  (including  in  each  case  negligence),  strict  liability  or
otherwise:

8.5.1

of the Charity and CRT to the Company shall be limited to £1,000,000 (one million Pounds Sterling) in aggregate;

8.5.2

of the Company to CRT and the Charity shall be limited to US $7,500,000 (7.5 million US dollars) in aggregate. The
Escrow Amount is not, and shall not be deemed to operate in any manner as, a cap or limit on the Company’s liability to
the other Parties.

To  the  fullest  extent  permissible  by  law,  no  Party  shall  under  any  circumstances  be  liable  to  any  other  for  any  loss  of  revenue,
business,  contracts,  anticipated  savings,  profits,  data  or  information,  or  any  indirect  or  consequential  loss  howsoever  arising
whether from negligence, breach of contract or otherwise.

Save  to  the  extent  otherwise  provided  in  this  Agreement,  each  Party  specifically  excludes  to  the  extent  permitted  by  law  all
warranties,  representations,  and  conditions  regarding  the  performance  of  its  obligations  under  this  Agreement  including  those
implied by law, whether as to suitability, quality or fitness for any purpose or otherwise.

INDEMNITIES

Subject  to  Clause  8.5,  the  Charity  shall  indemnify  and  hold  the  Company  its  officers,  and  employees  (the  “Company
Indemnitees”)  harmless  from  and  against all  Losses  arising  from  any  claims  and  proceedings  made  or  brought  (whether
successfully or otherwise) on behalf of Clinical Trial Subjects for personal injury (including death), arising out of the conduct of the
Clinical Trial, save where such claims, proceedings and/or Losses arise as a consequence of (i) any wrongful act or omission and/or
negligence of any of the Company Indemnitees; (ii) a breach of this Agreement by the Company; or (iii) a misrepresentation by the
Company.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
9.2

Notwithstanding the provisions of Clause 9.1 above and any other restrictions on liability contained in this Agreement, but subject
to Clause 8.5 above, the Company shall indemnify and hold the Charity, CRT, the Contributors, the Experts and their respective
officers,  employees  and  agents  (the  “Charity Indemnitees”)  harmless  from  and  against all  Losses  arising  from  any  claims  and
proceedings made or brought (whether successful or otherwise):

9.2.1

9.2.2

9.2.3

on behalf of Clinical Trial Subjects for personal injury (including death), arising out of: (i) any failure or delay on the part
of the Company to provide relevant or accurate Company KnowHow and other information relating to the storage, use and
safety of any of the Company Materials. and/or (ii) any wrongful act or omission and/or negligence of the Company (or
any third party engaged by the Company) in the supply and/or manufacture of any of the Company Materials; and

 alleging infringement of a third party’s Patent Rights or other Intellectual Property Rights resulting from use of Company
Intellectual Property or Company Materials in the course of or in consequence of the performance of the Clinical Trial or
by importation, storage, supply or use of any of the Company Materials and/or Antibody as permitted by this Agreement.
provided always that;

it is a condition of the indemnity that the Charity and CRT hand over or procure the hand over (as the case may be) of
control  of  the  matter  to  the  Company,  and  give  or  procure  (as  the  case  may  be)  such  information  and  assistance  as  the
Company  may  reasonably  request  in  connection  with  the  matter,  and  allow  or  procure,  (as  the  case  may  be)  that  the
Company has exclusive conduct of the matter and any ensuing legal proceedings.

The indemnities set out in Clauses 9.1 and 9.2 shall survive the expiration or termination of this Agreement for whatever reason.
Each Party’s agreement to indemnify, defend, and hold the other Party and its respective indemnitees harmless is conditioned upon
the  indemnified  Party:  (a)  providing  written  notice  to  the  indemnifying  Party  of  any  claim  or  proceeding  arising  out  of  the
indemnified activities within thirty (30) days after the indemnified Party has knowledge of such claim or proceeding; (b) permitting
the indemnifying Party to assume full responsibility and authority to investigate, prepare for, and defend against any such claim or
proceeding;  and  (c)  assisting  the  indemnifying  Party,  at  the  indemnifying  Party's  reasonable  expense,  in  the  investigation  of,
preparation for and defence of any such claim or proceeding. If the indemnifying Party assumes the defence of a third party claim,
the indemnifying Party will not be subject to any liability for any settlement of such claim made by the indemnified Party without
the indemnifying Party’s consent (which consent may not be unreasonably withheld, delayed or conditioned).

The Charity shall ensure that all Clinical Trial Subjects receive the benefit of a no-fault compensation scheme substantially in the
form  attached  at  Schedule  4  hereto.  Subject  to  the  indemnity  in  Clause  9.2,  the  Charity  shall  bear  all  costs  associated  with  the
provision of such compensation scheme including in relation to all claims received pursuant to such scheme.

The Company shall carry insurance coverage on an "occurrence" or "claims made" basis for potential liabilities which the Company
may have under this Agreement, and ensure that the Charity and CRT are each named additional insureds on each such policy and
may  claim  directly  under  them.  The  Company  shall  maintain  such  insurance  in  full  force  throughout  the  term  of  the Agreement
(and in the case of insurance coverage on a "claims made" basis, for a further two years after the term of the Agreement) and shall
upon request of the Charity provide such evidence of compliance as the Charity deems sufficient. The initial insurance policy of the
Company which satisfied the condition under Clause 2.1.3 is agreed to provide the minimum coverage required for the policy to be
carried by the Company under this Clause 9.5. The Company’s obligations, and the Charity’s and CRT’s rights, under this Clause
9.5  shall  apply  in  addition  to,  and  not  instead  of,  the  obligations  of  the  Company,  and  rights  of  the  Charity  and  CRT,  under  the
Escrow Agreement. Neither the existence of the Escrow Agreement nor any of its contents shall limit the obligations imposed or
rights granted under this Clause 9.5.

9.3

9.4

9.5

 
 
 
 
 
 
 
 
 
 
10.

ASSIGNMENT

10.1

No  Party  shall  assign  its  rights  under  this Agreement  or  any  part  thereof.  provided  that  the  Company  may  assign  its  rights  and
obligations  to  a  third  party  in  connection  with  any  merger  or  consolidation  of  the  Company  with  another  business  entity,  or  in
connection  with  the  sale  of  all  or  a  substantial  part  of  its  business  and  related  assets  that  includes  its  business  in  relation  to  the
Licensed Product (including, among other things, all XOMA IP and Intellectual Property licensed under this Agreement), other than
a merger or consolidation with or a sale of assets to a Tobacco Party and provided that the Company obtains a direct covenant from
the  acquiring  party  to  CRT  and  the  Charity  undertaking  to  be  bound  by  the  terms  of  this Agreement.  Save  as  set  out  in  this
Agreement,  no  Party  shall  sub-contract  the  performance  of  all  or  any  of  its  obligations  under  this Agreement  without  the  prior
written consent of the other Parties.

11.

TERM AND TERMINATION

11.1

Unless terminated earlier pursuant to the provisions hereunder, and except as otherwise provided hereunder, this Agreement shall
remain in full force and effect from the Commencement Date until the earlier of the date that:

11.1.1

the Agreement  expires  pursuant  to  Clause  2.2  due  to  a  failure  to  satisfy  the  Conditions  Precedent  before  the  Long  Stop
Date;

11.1.2

the Company enters into the Licence pursuant to Clause 7.4; or

11.1.3

the Company assigns the Company Intellectual Property and sub-licenses the XOMA IP to CRT pursuant to Clause 7.5.

11.2

Any of the Parties hereto may at any time terminate this Agreement, but shall not be obliged to do so, upon written notice to the
other Party (being the Charity and CRT where the terminating Party is the Company, or the Company where the terminating Party is
the Charity or CRT) under the following circumstances:

11.2.1

in  the  event  that  the  other  Party  commits  a  material  breach  of  this Agreement  and  does  not  fully  remedy,  if  capable  of
remedy, the same within sixty (60) days of its receipt of written notice of the breach from any other Party; or

11.2.2

in  the  event,  in  respect  of  a  Party:  that  respective  Party  proposes  a  voluntary  arrangement  for  that  respective  Party  or  a
voluntary  arrangement  is  approved  for  that  respective  Party;  or  an  administration  order  is  made  as  to  such  Party;  or  a
receiver or administrative receiver is appointed of any of such Party’s assets; or undertakings or a winding-up resolution or
petition is passed as to such Party (otherwise than for the purpose of solvent reconstruction or amalgamation); or if any
circumstances  arise  which  entitle  a  court  or  a  creditor  to  appoint  a  receiver,  administrative  receiver  or  administrator  or
make a winding-up order or similar; or equivalent action is taken against or by such Party by reason of its insolvency. A
Party shall notify the other Parties immediately upon becoming aware that any of the events identified in this Clause 11.2.2
has or is likely to take place in relation to it.

11.3

The Charity shall have the right to terminate this Agreement forthwith, upon written notice to the Company:

 
 
 
 
 
 
 
 
 
 
 
 
 
 
11.3.1

if the Charity has an insufficient quantity of IMP of the standard required to perform the activities envisaged under this
Agreement (whether due to a breach by the Company of Clause 8.2 or otherwise);

11.3.2

in accordance with Clause 3.6; or

11.3.3

if the Charity considers in its sole discretion that it would be unethical or otherwise undesirable for any reason to proceed or
continue with the Clinical Trial.

11.4

11.5

The Charity shall have the right to terminate this Agreement forthwith, upon written notice to the Company if, by way of merger,
acquisition or otherwise, the Company becomes a Tobacco Party.

The Parties may by mutual written agreement terminate this Agreement for any reason, including, if in their opinion the objectives
of the Clinical Trial cannot be achieved.

12.

CONSEQUENCES OF TERMINATION

12.1

In the event of termination of this Agreement by the Company:

12.1.1 without prejudice to Clause 12.1.4, the Company shall have no obligation to enter into the Option or any other licence with

CRT or the Charity, or to licence or assign its Intellectual Property Rights to CRT;

12.1.2

subject to Clause 12.1.4 and 12.6, the Charity shall, within ninety (90) days after written request of the Company, return to
the Company or destroy (by a method specified by the Company) and at the Company’s cost and expense any remaining
quantities  of  the  Company  Materials  and/or  Confidential  Information  of  the  Company  in  the  Charity’s  possession  or
control;

12.1.3 where  the  Charity  has  commenced  the  Clinical  Trial,  the  Charity  shall  within  thirty  (30)  days  of  finalisation  of  the  last
Case Report Form submit to the Company copies of all completed Case Report Forms and Data Listings for the Clinical
Trial. The Charity shall be entitled to retain the original Case Report Forms for its own records; and

12.1.4 where the Charity has commenced the Clinical Trial, the Charity shall nonetheless be entitled to make (or have made) the
Investigational  Medicinal  Product  and  continue  to  provide  it  to:  (i)  any  particular  Clinical  Trial  Subject  who  has
commenced  treatment;  and/or  (ii)  any  Clinical  Trial  Subject  where  the  Regulatory Authority  and/or  Ethics  Committee
request or require that such provision occurs.

12.2

In the event of any termination of this Agreement pursuant to Clause 11.2 or 11.4 by CRT or the Charity:

12.2.1

the Option shall lapse forthwith;

12.2.2

the Company shall within thirty (30) days of the date of such termination reimburse the Charity all Costs;

12.2.3

the Parties shall within thirty (30) days of the date of such termination execute the agreement set out in Schedule 5; and

12.2.4

the Charity shall be entitled to (as applicable) commence and complete the Clinical Trial and the Company shall provide
the Charity with the necessary assistance to allow the Charity to do so. For the avoidance of doubt, the licence granted by
the Company under Clause 6.1 shall continue to the extent necessary to allow the Charity to commence and complete the
Clinical Trial, provided that upon completion or termination of the Clinical Trial the Charity shall, within thirty (30) days
written  notice  by  the  Company  return  to  the  Company  or  destroy  (by  a  method  specified  by  the  Company)  and  at  the
Company’s cost and expense any remaining quantities of the Company Materials and/or Confidential Information of the
Company in the Charity’s possession or control.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
12.3

In the event of termination of this Agreement pursuant to Clause 11.3 by the Charity or pursuant to Clause 11.5:

12.3.1

subject to Clause 12.3.2 and 12.6, the Charity shall, within thirty (30) days written request by the Company, return to the
Company  or  destroy  (by  a  method  specified  by  the  Company)  and  at  the  Company’s  cost  and  expense  any  remaining
quantities  of  the  Company  Materials  and/or  Confidential  Information  of  the  Company  in  the  Charity’s  possession  or
control;

12.3.2 where  the  Charity  has  commenced  the  Clinical  Trial,  the  Company  shall  nonetheless  continue  to  permit  the  Charity  to
continue to provide such Investigational Medicinal Product to: (i) any particular Clinical Trial Subject who has commenced
treatment;  and/or  (ii)  any  Clinical  Trial  Subject  where  the  Regulatory  Authority  and/or  Ethics  Committee  request  or
require that such provision occurs; and

12.3.3 where the Charity and CRT consider it appropriate to do so in light of the reason for termination, for a period of thirty (30)
days  from  the  date  of  termination  (or  such  longer  period  as  CRT  may  notify)  CRT  shall  offer  the  Company  the  option,
exercisable by written notice to CRT, to enter into the Licence in respect of those Clinical Trial Results in existence at the
date of termination and subject to agreement between CRT and the Company on amended financial and other terms for the
Licence to reflect that the Clinical Trial was not completed. If the Parties are not able to agree amended financial terms
within thirty (30) days of the date CRT receives the Company’s exercise notice, the Parties at their joint cost and expense
shall obtain an Independent Opinion on a fair and reasonable reduction to the financial terms which will be binding on both
Parties.

Termination of this Agreement for whatever reason shall not affect the accrued rights of the Parties arising out of this Agreement as
at the date of its termination.

the 

The  provisions  of 
this  Agreement:  5
(Confidentiality/Publication),  6.3  (Assignment  of  Clinical  Trial  Results  to  CRT),  6.5  (Covenant  not  to  sue),  6.9  (invalidation  of
Company’s IP rights), 8.4 to 8.6 inclusive (Limits or exclusion of liability), 8.7 (Exclusion of other warranties), 9 (Indemnities), 10
(Assignment), 12 (Consequences of termination), 13 to 23 inclusive (Dispute Resolution to Third Party Rights inclusive).

following  Clauses  shall  survive 

the  expiration  or 

termination  of 

12.4

12.5

12.6

The Charity shall retain copies of the Company’s Confidential Information and the Clinical Trial Results in accordance with ICH
GCP and as otherwise required under the Charity’s obligations as Sponsor of the Clinical Trial.

13.

DISPUTE RESOLUTION

13.1

Insofar  as  this  Agreement  provides  that  a  matter  shall  be  resolved  by  Independent  Opinion,  the  opinion  of  the  appointed
independent expert (who shall act as an expert and not as an arbitrator) shall be final and binding on the Parties. In the event of a
Party  seeking  an  Independent  Opinion  under  this Agreement,  each  Party  shall  make  written  submissions  to  the  expert  and  to  the
other  Parties  within  fourteen  (14)  days  of  the  appointment.  Each  Party  shall  have  seven  (7)  days  to  respond  to  the  others’
submissions. The expert shall be requested to deliver his Independent Opinion within a further thirty (30) days. The costs of any
Independent  Opinion  shall  be  borne  in  such  proportions  as  the  expert  may  determine  in  his  Independent  Opinion  to  be  fair  and
reasonable  in  all  the  circumstances  or,  if  no  such  determination  is  made  in  the  Independent  Opinion,  by  the  Parties  in  equal
proportions.

 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

13.2

It  shall  be  a  condition  precedent  to  the  commencement  of  any  action  in  court  or  other  tribunal  (save  an  action  for  an  interim
injunction or an Independent Opinion sought under Clause 13.1) in respect of any dispute relating to this Agreement that the Parties
have sought to resolve the dispute by one Party notifying the others in writing for resolution to the Chief Executive Officer of CRT,
the Director of Drug Development of the Charity and the CEO of the Company (or their express delegates) (the “Representatives”)
who shall meet (whether in person or via teleconference) within twenty one (21) days of such notice to seek resolution in good faith.
If the Representatives are unable to resolve the dispute at such meeting, any Party may pursue any remedy available to such Party at
law or in equity, subject to the terms and conditions of this Agreement and the other agreements expressly contemplated hereunder.

13.3

This Agreement shall be governed by and construed in accordance with English Law and, subject to the provisions of Clause 13.1
and 13.2, each Party agrees to submit to the exclusive jurisdiction of the English Courts (except in respect of disputes under Clause
5 where jurisdiction is non-exclusive).

14.

NOTICES

14.1

Any notice or other document to be given under this Agreement shall be in writing and shall be deemed to have been given:

14.1.1

upon delivery if given in person; or

14.1.2

upon confirmation of receipt if sent by facsimile or email; or

14.1.3

 (if posted to an inland destination) three (3) business days after deposit into First Class post; or

14.1.4

(If posted to an overseas destination) five (5) days after deposit into airmail post; or

14.1.5

upon delivery by air delivery service;

to a Party at the address set out below (or, if provided below or so notified, such facsimile or electronic communication) for such Party or

such other address as the Party may from time to time designate by written notice to the other Parties.

Address of the Company

Monopar Therapeutics LLC

598 Rockefeller Road

Lake Forest, IL USA 60045

Contact: Chief Executive Officer

Email: [***]

Address of the Charity

Cancer Research UK

Angel Building

407 St. John Street

London EC1V 4AD

England

Contact: Director of Drug Development

Fax: +44 (0) 20 7121 6700

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
With a copy to:

Cancer Research UK

Angel Building

407 St. John Street

London EC1V 4AD

England

Contact: Caroline Foxton

Fax: +44 (0) 20 7121 6700

Address of CRT

Cancer Research Technology Limited

Angel Building

407 St. John Street

London

EC1V 4AD

United Kingdom

Contact: Chief Executive Officer

Fax: +44 (0) 20 3014 8633

15.

WAIVER

15.1

No failure or delay on the part of any Party hereto to exercise any right or remedy under this Agreement shall be construed as or
operate as a waiver thereof nor shall any single or partial exercise of any right or remedy under this Agreement preclude the exercise
of any other right or remedy or preclude the further exercise of such right or remedy as the case may be.

16.

FORCE MAJEURE

16.1

No Party shall be liable to any other Party or shall be in default of its obligations hereunder if such default is the result of any cause
beyond  the  reasonable  control  of  the  Party  affected  including  war,  hostilities,  revolution,  civil  commotion,  strike,  epidemic,
accident, fire, wind, flood or because of any act of God . The Party affected by such circumstances shall promptly notify the other
Parties in writing when such circumstances cause a delay or failure in performance (a “Delay”) and where they cease to do so. In the
event of a Delay lasting for twenty six (26) weeks or more either of the non-affected Parties shall have the right to terminate this
Agreement immediately by notice in writing to the affected Party.

17.

INSOLVENCY

17.1

All rights and licenses granted under or pursuant to this Agreement by the Company to CRT and the Charity are for all purposes of
Section  365(n)  of  Title  11  of  the  U.S.  Bankruptcy  Code  (“Title 11”),  licenses  of  rights  to  “intellectual  property”  as  defined  in
Section 101 of Title 11.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
17.2

The  Company  agrees  that  CRT  and  the  Charity  shall  retain  and  may  fully  exercise  all  of  its  rights  and  elections  under  the  U.S.
Bankruptcy Code. If a case under Title 11 is commenced by or against the Company, CRT and the Charity shall have all rights of
licensees set out in Section 365(n) of Title 11.

17.3 Without  limiting  CRT’s  and  the  Charity’s  rights  under  Section  365(n)  of  Title  11,  if  a  case  under  Title  11  is  commenced  by  or
against  the  Company,  and  this Agreement  is  rejected  by  the  Company  in  any  bankruptcy  proceeding  by  or  against  the  Company
under the U.S. Bankruptcy Code, (i) the Company shall provide CRT and the Charity with a complete duplicate of (and complete
access to, as appropriate) any IP and embodiments of IP not already in their possession; and (ii) the Company shall not interfere
with CRT’s and the Charity’s rights to IP and embodiments of IP, and shall facilitate and assist with CRT and the Charity obtaining
IP and embodiments of IP (including from a third party).

17.4

The term “embodiments” of IP includes all tangible, intangible, electronic or other embodiments of rights and licenses, including
antibodies, compounds and products embodying IP and related rights and technology. All rights of CRT and the Charity under this
Clause and under Section 365(n) of Title 11 are in addition to, not in substitution of, any other rights and remedies that they may
have under this Agreement, Title 11 and any other applicable law.

18.

SEVERABILITY

18.1

If  and  to  the  extent  that  any  court  or  tribunal  of  competent  jurisdiction  holds  any  of  the  terms,  provisions  or  conditions  or  parts
thereof  of  this Agreement,  or  the  application  hereof  to  any  circumstances,  to  be  invalid  or  to  be  unenforceable  in  a  final  non-
appealable  order,  the  remainder  of  this Agreement  and  the  application  of  such  term,  provision  or  condition  or  part  thereof  to
circumstances other than those as to which it is held invalid or unenforceable shall not be affected thereby, and each of the other
terms, provisions and conditions of this Agreement shall be valid and enforceable to the fullest extent permissible by law.

19.

ENTIRE AGREEMENT

19.1

This Agreement  embodies  and  sets  forth  the  entire  agreement  and  understanding  of  the  Parties  and  supersedes  all  prior  oral  or
written agreements, understandings or arrangements relating to the subject matter of this Agreement. No Party shall be entitled to
rely on any agreement, understanding or arrangement which is not expressly set forth in this Agreement unless otherwise agreed
between the Parties and recorded in writing. In the event of any inconsistency between this Agreement and the Protocol, the terms
of this Agreement shall govern.

20.

AMENDMENT

20.1

This Agreement shall not be amended, modified, varied or supplemented except in writing signed by duly authorised representatives
of the Parties.

20.2

The Charity shall at all times be free to amend, modify, vary or supplement any of its own Standard Operating Procedures.

21.

PUBLIC ANNOUNCEMENTS

21.1

The text of any press release, shareholders’ report or other communication to be published  or disclosed in any way by or on behalf
of the Company by or in the media concerning the Charity, the Contributors or the Experts, the subject matter of this Agreement or
concerning this Agreement itself, other than as required by law or by any regulatory or government authority, shall be submitted to
the  Charity  and  CRT  at  least  seven  (7)  days  in  advance  of  publication  or  disclosure  for  approval,  such  approval  not  to  be
unreasonably  withheld;  provided  that  insofar  as  a  disclosure  repeats  or  restates  a  prior  public  disclosure  permitted  by  this
Agreement, such disclosure need not be submitted to the Charity or CRT for approval.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
22.

PAYMENTS

22.1

22.2

22.3

All  payments  due  to  CRT  and  the  Charity  under  this Agreement  shall  be  made  in  cleared  funds  in  pounds  sterling  to  the  bank
accounts  nominated  by  CRT  and  the  Charity  respectively  from  time  to  time.  All  costs  of  transmission  shall  be  borne  by  the
Company.

All payments under this Agreement are expressed to be exclusive of value added tax howsoever arising, which the Company shall
pay in addition to those payments.

Save  as  expressly  set  out  in  Clause  7.2,  all  amounts  due  under  this Agreement  shall  be  paid  in  full  without  any  deduction  or
withholding other than as required by law and the Company shall not be entitled to assert any credit, set-off or counterclaim against
CRT or the Charity in order to justify withholding payment of any such amount in whole or in part.

22.4 Where  a  Party  does  not  receive  payment  of  any  sums  due  to  it  by  the  due  date,  interest  shall  accrue  both  before  and  after  any
judgement on the sum due and owing to such Party at the rate equivalent to an annual rate of two percent (2%) over the then current
base  rate  of  Natwest  Bank,  calculated  on  a  daily  basis,  until  the  full  amount  is  paid,  without  prejudice  to  such  Party’s  right  to
receive payment on the due date.

23.

DATA PROTECTION

23.1

23.2

The Parties’ attention is drawn to the Data Protection Act 1998, Directive 95/46/EC of the European Parliament and any national or
European  legislation  and/or  regulations  implementing  them  or  made  in  pursuance  of  them  (all  referred  to  together  as  the  “Data
Protection Requirements”).

Each Party warrants that it will observe all its obligations under the Data Protection Requirements which arise in connection with
the performance of this Agreement and in particular that it will process and use any personal data fairly and lawfully.

24.

THIRD PARTY RIGHTS

24.1

Save  for  the  third  parties  identified  in  Clauses  5.5  (Contributors’  right  to  publish),  6.5  (Covenant  not  to  sue),  9.1  and  9.2
(Indemnities) and 9.3 (No fault compensation scheme), who shall have the benefit of those respective Clauses, this Agreement shall
not create any rights that shall be enforceable by anyone other than the Parties to this Agreement. The rights created in Clauses 5.5,
6.5, 9.1, 9.2 and 9.3 may be altered or extinguished by the Parties without consent of any third party beneficiary of such rights.

25.

EXECUTION

25.1

This Agreement may be executed in any one or more number of counterpart agreements, and as scanned email attachments, and all
signatures and counterparts so exchanged shall be considered as original and shall be deemed to form part of and together constitute
this Agreement.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
IN WITNESS whereof this Agreement has been executed by duly authorised officers of the Parties on the day first above written.

Signed by:
Name:
Title:

/s/ PJ L’Hullier
PJ L’Hullier
Director, Business Management

For and on behalf of
CANCER RESEARCH TECHNOLOGY LIMITED

Signed by:
Name:
Title:

/s/ Dr. Nigel Blackburn
Dr. Nigel Blackburn
Director of Drug Development CRUK Centre for Drug Development

For and on behalf of
CANCER RESEARCH UK

Signed by:
Name:
Title:

/s/ Chandler Robinson
Chandler Robinson
CEO and Manager

For and on behalf of
MONOPAR THERAPEUTICS LLC

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

Schedule 1
Company Patent Rights
(details of company patent rights to be inserted here)

B& N Ref    Country    Status    Comments    Applicaiton #    Filing Date    Patent #    Grant Date

                                                                                                                       [***]         [***]         [***]       [***]              [***]               
[***]            [***]            [***]                                            

 
 
 
 
 
 
 
 
 
 
Name of Sponsor/Company:

Schedule 2
Report Synopsis

Individual Study Table
Referring to Part
of the Dossier

Name of Finished Product:

Volume:

Name of Active Ingredient:

Page:

Title of Study:

Investigators:

Study Centre(s):

Publication (reference):

Studied period (years):

Phase of development:

(date of first enrolment)
(date of last completed)

Objectives:

Methodology:

Number of Patients (planned and analysed):

Diagnosis and main criteria for inclusion:

Test product, dose and mode of administration, batch number:

Duration of treatment:

Reference therapy, dose and mode of administration, batch number:

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Name of Sponsor/Company:

Individual Study Table
Referring to Part
of the Dossier

Name of Finished Product:

Volume:

Name of Active Ingredient:

Page:

Criteria for evaluation:

Efficacy:

[Drafting  Note:  The  sub-heading  of  “Efficacy”  can  be  adapted  to  “Pharmacokinetics”,  “Pharmacodynamics”,  “Immunogenicity”,
“Pharmacogenomics”  etc,  as  dictated  by  the  study  objectives.  If  there  is  more  than  one  major  area  of  evaluation,  further  top-level
headings can be added here.]

Safety:

[Drafting Note: The sub-heading of “Safety” must always be included.]

Statistical methods:

SUMMARY – CONCLUSIONS

EFFICACY RESULTS:

[Drafting  Note:  The  sub-heading  of  “Efficacy  Results”  can  be  adapted  to  “Pharmacokinetics”,  “Pharmacodynamics”,
“Immunogenicity”,  “Pharmacogenomics  Results”  etc,  as  dictated  by  the  study  endpoints.  If  there  is  more  than  one  major  area  of
evaluation, further top-level headings can be added here.

Efficacy (and/or other similar) result CONCLUSIONS ONLY should be summarised. The summaries can be superficial if the study
was uncontrolled, seriously flawed or aborted such that this data cannot be analysed.]

SAFETY RESULTS:

[Drafting Note: The subheading of “Safety Results” must always be included. Safety result CONCLUSIONS ONLY must always be
presented.]

CONCLUSION:

Date of the report:

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Schedule 3
Licence from CRT to Company

THIS AGREEMENT is made the________ day of ____________________20[●●]

BETWEEN:

(1)

(2)

CANCER RESEARCH TECHNOLOGY LIMITED, a company registered in England and Wales under number 1626049 with
registered office at Angel Building, 407 St. John Street, London, EC1V 4AD, England] (“CRT”); and

[MONOPAR THERAPEUTICS LLC, a limited liability company registered in/incorporated in/ established under the laws of The
State of Delaware, U.S.A., with registered office/principal place of business at 598 Rockefeller Road, Lake Forest, Illinois, U.S.A.,
60045] (the “Company”).]

RECITALS

(A) 

(B) 

CRT is a wholly owned subsidiary of Cancer Research UK (the “Charity”) and is, by arrangement with the Charity, responsible for
the  management,  exploitation  and  commercialisation  of  intellectual  property  generated  by  the  Charity  or  using  funding  from  the
Charity.

Pursuant to a Clinical Trial and Option Agreement between CRT, the Charity and the Company dated [●●●] attached at Appendix 2
(the “CTOA”) the Charity has conducted the Clinical Trial (as defined below) and assigned the results of such Clinical Trial and all
intellectual property therein to CRT.

(C) 

CRT  has  agreed  to  grant  the  Company  a  licence  under  the  Licensed  Intellectual  Property  (as  defined  below)  upon  the  terms  and
conditions set out in this Agreement.

OPERATIVE PROVISIONS

1.

1.1

INTERPRETATION

In  this Agreement  except  where  the  context  requires  otherwise,  the  following  words  and  expressions  shall  have  the  following
meanings:

“Accountancy
Opinion”

means  the  opinion  of  an  independent  United  Kingdom  chartered  accountant  appointed  by  agreement  between  the
Parties or in default of such agreement within twenty one (21) days of either Party seeking in writing to the other to
appoint  such  accountant,  at  the  request  of  either  Party,  by  the  President  for  the  time  being  of  the  Institute  of
Chartered Accountants in England and Wales, referred to in Clauses 1, 6.3 and 24.1.

“Affiliate”

has the same meaning as that ascribed to that phrase in the CTOA.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
“Affordable Price”

means in relation to a Licensed Product: (i) a determination by the UK Pricing Authority that such Licensed Product
should  be  used  within  the  NHS;  and/or  (ii)  approval  by  the  UK  Pricing Authority  of  the  price  proposed  by  the
Company or its Sub-Licensee in relation to sales of that Licensed Product in the United Kingdom (or one or more
constituent countries thereof).

“Agreement”

means this agreement and each of the Appendices as amended from time to time in accordance with Clause 21.

“Clinical Trial”

has the same meaning as that ascribed to that phrase in the CTOA.

“Clinical Trial
Results”

“Company
Intellectual
Property”

“Company Patent
Rights”

has the same meaning as that ascribed to that phrase in the CTOA.

has the same meaning as that ascribed to that phrase in the CTOA.

has the same meaning as that ascribed to that phrase in the CTOA.

“Competing
Programme”

means  a  research  and  development  programme  under  which  human  subjects  in  a  clinical  trial  have  or  are  to  be
administered a treatment or compound directed towards the same target molecule as the Antibody.

“Confidential
Information”

means  the  Clinical  Trial  Results  and  all  information  relating  to  the  customers,  suppliers,  business  partners,  clients,
finances, business plans and products (in each case actual or prospective) of a Party which is not in the public domain
and which is acquired by the other Party pursuant to this Agreement.

“Contributors”

has the same meaning as that ascribed to that phrase in the CTOA.

“Control”

means:

a) with respect to corporate ownership, the possession (directly or indirectly) of fifty per cent or

more of the voting stock or other equity interest of a subject entity with the power to vote, or the power in
fact to control the management decisions of such entity through the ownership of securities or by contract
or otherwise; and

b) with respect to Intellectual Property Rights, possession of the ability (whether through ownership

or licence, other than a licence granted under this Agreement) to provide the information or grant the
licences or sublicences or make the assignments as provided herein without violating the terms of any
agreement or other arrangement with any third party,

and “Controls” and “Controlled by” shall be construed accordingly.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
“Currency”

means pounds sterling or such other currency as CRT may reasonably specify from time to time.

“Data Exclusivity
Period”

means any period of clinical trial data or other regulatory exclusivity, together with any such periods under national
implementations in the European Union of Article 10.1 of Directive 2001/EC/83 and all equivalents elsewhere in the
Territory.

“Data Listings”

has the same meaning as that ascribed to that phrase in the CTOA.

“Development
Plan”

means  the  development  plan  at Appendix  1  (as  the  same  shall  be  updated  in  accordance  with  Clause  3.1)  which
describes: (i) the steps to be taken to develop Licensed Products within the Territory; and (ii) the relevant timescales
within which such steps will be taken.

“Effective Date”

means the date this Agreement is made.

“Exclusive
Results”

“Expert Opinion”

has the same meaning as that ascribed to that phrase in the CTOA.

means  the  opinion  of  an  independent  expert  appointed  by  agreement  between  the  Parties  or  in  default  of  such
agreement within twenty one (21) days of either Party seeking in writing to the other to appoint such expert, by the
President for the time being of the Association of the British Pharmaceutical Industry referred to in Clauses 12.3 and
24.1.

“Field”

means the treatment, prophylaxis, diagnosis, prevention and/or cure of human disease and conditions.

“Final Report”

has the same meaning as that ascribed to that phrase in the CTOA.

“First Commercial
Sale”

means, with respect to a Licensed Product, the first transfer or disposition for value of such Licensed Product by or
on  behalf  of  the  Company  or  a  Sub-Licensee  or  an  Affiliate  of  either  of  them,  after  all  relevant  Regulatory
Authorisations for the transfer or disposition of such Licensed Product have been obtained in respect of the relevant
region or country.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

“Indication”

means  a  disease  classification  block  as  defined  within  the  ‘International  Statistical  Classification  of  Diseases  and
Related  Health  Problems’  as  published  from  time  to  time  by  the  World  Health  Organization  (e.g.  “C50  Malignant
neoplasm  of  Breast”,  “C92  Myeloid  leukaemia”,  “B20  Human  immunodeficiency  virus  [HIV]  disease  resulting  in
infectious and parasitic diseases”, “M34 Systemic sclerosis”).

“Investigational
Medicinal
Product” or “IMP”

“Intellectual
Property Rights”

“Licensed
Intellectual
Property”

“Licensed
Product”

has the same meaning as that ascribed to that phrase in the CTOA.

has the same meaning as that ascribed to that phrase in the CTOA.

means the Clinical Trial Results and all Intellectual Property Rights therein.

means any product:

a) whose application for Regulatory Authorisation from a Regulatory Authority in any jurisdiction
included the Clinical Trial Results and/or the Final Report and/or the Data Listings or any part of any of
them, and/or

b) that contains the Antibody or a Back-Up Antibody (or any part of either), in each case whether or

not as the sole active ingredient, and/or

c) the unauthorised manufacture, sale or use of which would infringe a valid claim of the Company

Patent Rights.

“Major Markets”

means [***]

“Milestone Event”

has the meaning specified in Clause 4.1.2.

“Milestone
Payments”

“NDA”

has the meaning specified in Clause 4.1.2.

means, in relation to any Licensed Product, a biologics license application, new drug application, supplementary new
drug application, abbreviated new drug application or any of their equivalents filed with the United States Food and
Drugs Administration (FDA) or any successor to it, a marketing authorisation application or its equivalent filed with
the European Medicines Agency (EMEA) or any successor to it, or a marketing authorisation application or a product
licence application or equivalent filed with the relevant Regulatory Authority in any one or more countries or regions
within the Territory.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

“Net Sales Value”

“New Company
IP”

“Non-Exclusive
Results”

“Oncology
Indication”

means, in relation to Licensed Product the gross amount invoiced by the Company or SubLicensee or Affiliate of the
Company or a SubLicensee [***] to the extent that any of those items are included as separate items in the amount so
invoiced, and [***].
means any Intellectual Property Rights developed by or on behalf of the Company on or after the Effective Date that
directly relate to the IMP and its use.

has the same meaning as that ascribed to that phrase in the CTOA.

means an Indication in the range C00 – D48 (e.g. “C50 Malignant neoplasm of Breast”, “C92 Myeloid leukaemia”).

“Party”

means either party to this Agreement and “Parties” means both of them.

“Patent Rights”

has the same meaning as ascribed to that phrase in the CTOA.

“Phase II Clinical
Trial
Commencement”

means the first dosing of a human subject in a clinical trial of a Licensed Product (or in the adaptation of an existing
clinical trial) in any country that would satisfy the requirements of 21 CFR §312.21(b) and is intended to establish
dose  response  and/or  preliminary  data  on  the  efficacy  of  Licensed  Product  and/or  route  of  administration  of  the
Licensed Product.

“Phase III Clinical
Trial
Commencement”

means the first dosing of a human subject in a clinical trial of a Licensed Product (or the adaptation of an existing
clinical  trial)  to  be  a  larger  scale  (than  Phase  I  or  Phase  II),  usually  multi-centred  trial  in  any  country  that  would
satisfy the requirements of 21 CFR §312.21(c) and is intended to establish the efficacy and safety of the Licensed
Product or any other human clinical trial of the Licensed Product intended as a pivotal trial for regulatory approval
purposes whether or not such trial is a traditional Phase III trial.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

“pound” and “£”

means British pound sterling or if England changes its currency during the Term, then a sum equivalent in the new
currency based on the spot exchange rate at the date of adoption of the new currency.

“Price Approval”

means,  in  those  countries  in  the  Territory  where  Regulatory Authorities  may  approve  or  determine  pricing  and/or
pricing reimbursement for pharmaceutical products, such approval or determination.

“Quarter”

means any of the three-monthly periods commencing on the first day of any of the months of January, April, July,
and October in any year and “Quarterly” has a corresponding meaning.

“Regulatory
Authorisations”

means  all  marketing  authorisations,  approvals,  clearances  and  authorisations  that  may  be  required  by  a  Regulatory
Authority in any country or region within the Territory prior to Phase II Clinical Trial Commencement and/or Phase
III Clinical Trial Commencement and/or commercial sale of the Licensed Product, including any necessary variations
thereto, but excluding always any Price Approvals.

“Regulatory
Authority”

means any local or national agency, court, authority, department, inspectorate, minister, ministry official or public or
statutory person (whether autonomous or not) of, or of any government of, any country having jurisdiction over this
Agreement  or  either  of  the  Parties  or  over  the  development  or  marketing  of  medicinal  products  including,  the
European Medicines Agency and the European Court of Justice.

“Signature Fee”

means the sum of [***].

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

“Sub-Licence
Revenue”

“Sub-Licensee”

means any monies or non-monetary consideration (including securities) receivable from time to time by the Company
or any of its Affiliates in respect of: (i) any sub-licence granted by the Company or any of its Affiliates under this
Agreement; (ii) any licence granted by the Company or any of its Affiliates (whether under the Company Intellectual
Property  or  otherwise)  to  sell  Licensed  Products  anywhere  in  the  Territory;  and/or  (iii)  the  grant  of  the  right  to
acquire  such  a  sub-licence  or  licence,  including,  in  each  case,  option  fees,  licence  issue  fees  or  other  up-front
payments, annual licence fees, milestone or other lump sum payments which are attributable to the grant of the rights
in question, excluding royalties and Net Sales Value as referred to in Clause 4.4 (in the case of non-monetary Sub-
Licence Revenue such as company stocks and shares, such non-monetary consideration shall not form Sub-Licence
Revenue  until  Company  or  relevant Affiliate  has  received  cash  proceeds  from  the  disposal  or  other  realisation  of
such consideration. [***]
means  any  person  who  is  granted:  (i)  a  sub-licence  in  accordance  with  Clause  2.3  in  respect  of  the  rights  granted
under  this  Agreement  (and  any  further  tiers  of  sub-licence  thereunder);  and/or  (ii)  a  licence  by  the  Company
(whether under the Company Intellectual Property or otherwise) to sell Licensed Products anywhere in the Territory,
but  shall  not  mean  distributors,  wholesalers,  and  sales  agents  (sales  to  whom  will  be  sales  for  the  purpose  of  Net
Sales Value).

“Term”

means the term of this Agreement as determined under Clause 12.1.

“Territory”

means worldwide.

“Tobacco Party”

means: (i) any entity who develops, sells or manufactures tobacco products; and/ or (ii) any entity which makes the
majority of its profits from the importation, marketing, sale or disposal of tobacco products. Furthermore, Tobacco
Party shall include any entity that is an Affiliate of any entity referred to in (i) or (ii).

“UK Pricing
Authority”

means any supra-national, national or regional government department, authority, agency or entity (including a non-
departmental  public  body  or  similar  entity)  with  responsibility  for  evaluating  the  cost  effectiveness  of  medicinal
products in the United Kingdom (or one or more constituent countries thereof) or otherwise determining whether the
NHS (or constituent parts thereof) should purchase medicinal products.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

“XOMA”

has the meaning ascribed to that phrase in the CTOA.

“XOMA Licence”

has the same meaning ascribed to that phrase in the CTOA.

“Year”

means a calendar year.

1.2

In this Agreement:

1.2.1

unless the context requires otherwise, all references to a particular Clause, paragraph or Appendix shall be references to
that clause, paragraph or appendix, in or to this Agreement;

1.2.2

the headings are inserted for convenience only and shall be ignored in construing this Agreement;

1.2.3

1.2.4

unless the contrary intention appears, words importing the masculine gender shall include the feminine and vice versa and
words in the singular include the plural and vice versa;

unless  the  contrary  intention  appears,  words  denoting  persons  shall  include  any  individual,  partnership,  company,
corporation, joint venture, trust, association, organisation or other entity, in each case whether or not having separate legal
personality; and

1.2.5

references  to  the  words  ‘include’  or  ‘including’  shall  be  construed  without  limitation  to  the  generality  of  the  preceding
words.

2.

2.1

GRANT OF LICENCE

Subject to the provisions of this Agreement and the surviving provisions of the CTOA, CRT hereby grants to the Company:

2.1.1

[***]; and

2.1.2

[***],

in each case to research, develop, make, have made, import, use and sell Licensed Products for any and all uses in the Territory and to apply

for Regulatory Authorisation for such Licensed Products in any jurisdiction.

2.2

CRT  hereby  reserves  and  excepts  from  the  [***]  under  Clause  2.1.1  the  worldwide,  perpetual  and  irrevocable  right  for  the
Contributors and the Charity (including use by scientists funded and/or employed by the Charity) to:

2.2.1

use the Licensed Intellectual Property for the purpose of non-commercial scientific research carried out by or for or under
their  respective  direction  in  accordance  with  their  respective  charitable  and/or  academic  status,  whether  alone  or  in
collaboration with a third party or third parties and whether sponsored or funded, in whole or in part, by any third party
including any commercial entity; and

2.2.2

make publications in relation to the Licensed Intellectual Property and any results of research using the same in accordance
with generally accepted academic practice.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
2.3

The Company shall be entitled to grant sub-licences in respect of the rights granted under this Agreement, provided that:

2.3.1

2.3.2

2.3.3

any  sub-licence  granted  by  the  Company  shall  be  expressed  to  terminate  automatically  on  the  termination  of  this
Agreement for any reason;

any sub-licence granted by the Company beyond the first tier of sub-licensing shall expressly prohibit further sub-licensing
without CRT’s prior written consent, which consent may not be unreasonably conditioned, delayed, or withheld.

the Company shall ensure that there are included in the terms of any sub-licence like obligations and undertakings on the
part of the Sub-Licensee as are contained in this Agreement (except this Clause 2.3, but including Clause 9 (indemnity)
and Clause 14 (confidentiality)) and shall further ensure that all Sub-Licensees duly comply with the same;

2.3.4

no sub-licence shall be granted to a Tobacco Party;

2.3.5

the sub-licence shall be entered into on an arms-length basis reflecting the market value of the rights granted; and

2.3.6

the Company shall provide CRT with a copy of such sub-licence within thirty (30) days of entering into it.

Any breach of Clause 2.3 shall be deemed to be a material breach.

The grant of any sub-licence shall be without prejudice to the Company’s obligations under this Agreement. Any act or omission of
any  such  Sub-Licensee  which,  if  it  were  the  act  or  omission  of  the  Company  would  be  a  breach  of  any  of  the  provisions  of  this
Agreement, will be deemed to be a breach of this Agreement by the Company who will be liable to CRT accordingly.

CRT will provide the Company with any Long Term Survival Data as and when the Charity has completed collection of the same.

The Company may not publish or publicly disclose any Clinical Trial Results in the one (1) year period beginning on the Effective
Date without the prior written consent of CRT, which will be given at CRT’s sole discretion. All publications by the Company of
the  Clinical  Trial  Results  and  results  of  research  using  the  same  will  be  made  in  accordance  with  generally  accepted  academic
practice, including in respect of the role played by the Contributors. The foregoing provisions of this Clause 2.7 shall not apply to
disclosure  of  Clinical  Trial  Results,  or  any  portion  thereof,  by  the  Company  to  the  extent  required  for  (a)  satisfying  mandatory
reporting and disclosure obligations under United States and other securities laws. or (b) to existing licensors or sublicensors of the
Company  in  order  to  comply  with  reporting  obligations  in  existence  as  at  the  date  of  this  agreement  under  the  XOMA  Licence,
provided that in the case of (b) the disclosure  shall  be  limited  to  only  information  as  may  be  reasonably  required  by  the  XOMA
Licence and subject to XOMA being bound by confidentiality obligations that are no less restrictive than those that the Company is
bound by under this Agreement in respect of confidential information disclosed to it.

The Charity shall, within thirty (30) days written request by the Company, return to the Company or destroy (by a method specified
by  the  Company)  and  at  the  Company’s  cost  and  expense  any  remaining  quantities  of  the  Company  Materials  in  the  Charity’s
possession or control.

PERFORMANCE

The Company shall provide an updated Development Plan to CRT on at least a six-monthly basis before the first approval of an
NDA in respect of a Licensed Product, and on an annual basis thereafter.

2.4

2.5

2.6

2.7

2.8

3.

3.1

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

3.2

3.3

The Company shall procure the achievement of Phase II Clinical Trial Commencement within [***] of the Effective Date.

The Company shall use its commercially reasonable efforts at all times during the Term to:

3.3.1

comply with the most up-to-date version of the Development Plan;

3.3.2

develop and pursue Regulatory Authorisation for a Licensed Product for use in [***] in each of the [***];

3.3.3

3.3.4

3.3.5

introduce  a  Licensed  Product  for  use  in  [***]  into  each  of  the  [***]  as  soon  as  reasonably  and  commercially  practical
following receipt of the corresponding Regulatory Authorisations and subsequently use commercially reasonable efforts to
market  the  Licensed  Product  and  pursue  maximum  market  penetration  throughout  the  Major  Markets  for  such  Licensed
Product;

launch each Licensed Product in the United Kingdom as soon as practicable and in any event no later than [***] after the
date the first Regulatory Authorisation is granted by the European Medicines Agency; and

make  Licensed  Products  that  are  launched  in  the  United  Kingdom  available  at  an  Affordable  Price  if  required  by  a
Regulatory Authority in order to obtain a Price Approval for such Licensed Products in the United Kingdom.

3.4

Subject  to  Clause  3.5.2,  the  Company  shall  provide  CRT  with  reports  as  to  the  progress  of  the  development  of  each  Licensed
Product, the progress of any applications for Regulatory Authorisation and Price Approval, and the progress of and plans for the
marketing and sale of the Licensed Product and its compliance with the Development Plan, in such form and detail as CRT may
reasonably  require.  The  Company  shall  provide  such  reports  on  at  least  a  six-monthly  basis  before  first  approval  of  an  NDA  in
respect of a Licensed Product, and on an annual basis thereafter.

3.5

If, prior to the First Commercial Sale in the United Kingdom and two (2) other Major Markets, the Company undergoes a change of
Control, or acquires or begins (whether independently or with a third party) a Competing Programme:

3.5.1

3.5.2

it  shall  notify  CRT  in  writing  within  thirty  (30)  days  after  the  change  of  Control  occurring,  or  its  commencement  or
acquisition of the Competing Programme; and

for the [***] period following the change of Control, or commencement or acquisition  of  the  Competing  Programme,  it
shall provide CRT with a report described in Clause 3.4 at least once every three (3) months.

3.6

3.7

The Company shall give CRT prompt notice upon the occurrence of any Milestone Event.

The Company shall submit to CRT:

3.7.1

3.7.2

a  copy  of  its  detailed  operating  budget  (including  a  semi-annual  cash  flow  and  expenditure  forecast)  for  the  Licensed
Product in respect of each Financial Year as adopted by the Company’s board (the “ Annual Budget”), at least thirty (30)
days prior to the commencement of the Financial Year to which the Annual Budget relates;

semi-annual management accounts of the Company (to include, inter alia, a (consolidated) profit and loss account, balance
sheet and cash flow statement and shall indicate where such management accounts differ to any material extent from the
Annual Budget for such period), within sixty (60) days of the end of the period to which they relate; save that the accounts
relating to the final quarter in any calendar year may be provided within ninety five (95) days, rather than sixty (60) days,
of the end of that quarter. Such semi-annual management accounts shall be prepared on a basis which is consistent with
those adopted in the preparation of all previous management accounts of the Company.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

3.8

The Company shall generally keep CRT informed of the progress of the Company's business and affairs and shall supply CRT with
written details of any circumstances which will or might cause any actual or prospective material adverse change in the financial
position, prospects or business of the Company.

3.9

Any breach of Clause 3 shall be deemed to be a material breach of this Agreement.

4.

4.1

4.2

CONSIDERATION

The Company shall pay the Signature Fee to CRT within thirty (30) days of the Effective Date.

Subject  to  clause  4.5,  the  Company  shall  pay  the  following  payments  (“Milestone Payments”)  to  CRT  each  time  the  following
events (“Milestone Events”) occur in relation to any Licensed Product:

4.2.1

[***];

4.2.2

[***];

4.2.3

[***];

4.2.4

[***];

4.2.5

[***];

4.2.6

[***];

4.2.7

[***]; and

4.2.8

[***]

Upon the occurrence of each Milestone Event, any Milestone Event listed before it in this Clause 4 which has not occurred shall be
deemed to have occurred. For the avoidance of doubt, a Milestone Event may be triggered by the actions of the Company, a Sub-
Licensee or any third party acting on behalf of the Company or any Sub-Licensee.

4.3

Subject to Clause 4.5, the Company shall pay to CRT:
4.3.1

[***];

4.3.2

[***]; and

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

4.3.3

[***].

For the avoidance of doubt, Sub-Licence Revenue expressly excludes royalty payments due under Clause 4.4 or Net Sales Value.

4.4

The Company shall pay royalties to CRT on a Licensed Product by Licensed Product, and country by country basis until the later of:

4.4.1

[***];

4.4.2

t[***]; and

4.4.3

[***],

4.5

5.

5.1

In the event that any Milestone Event is triggered by any Sub-Licensee, the Company shall pay to CRT the greater of: (i) [***]; and
(ii) [***].

PAYMENT AND STATEMENT

All payments due to CRT under this Agreement shall be made in the Currency in cleared funds to the following bank account:

[***]

[***]

[***]

[***]

[***]

[***]

[***]

[***]

[***]

[***]

[***]

[***]

or such other account as CRT may notify to the Company from time to time.

5.2

The Company shall pay to CRT:

5.2.1

the Signature Fee on the date specified in Clause 4.1;

5.2.2

each of the Milestone Payments within thirty (30) days of the relevant Milestone Event occurring; and

5.2.3

each  payment  that  is  due  under  Clause  4.3  or  4.4,  within  thirty  (30)  days  of  the  Company  or  any  relevant  Affiliate
receiving the corresponding Sub-Licence Revenue or percentage of Net Sales Value. All sums due to CRT under Clause
4.3  or  4.4  shall  belong  to  CRT  upon  the  Company’s  or  its  Affiliate’s  receipt  of  the  revenue  to  which  such  payment
corresponds (and is a percentage of) and such sums shall be held on trust for CRT until paid to CRT in accordance with this
Clause 5.2.3. The Company shall take all steps necessary to ensure, and to procure that any relevant Affiliate ensures, that
sums  held  on  trust  are  separate  and  identifiable  from  other  monies  of  the  Company  or Affiliate,  including  holding  such
sums  in  a  separate  account  to  monies  that  belong  to  the  Company  and/or Affiliate. At  CRT’s  reasonable  request,  the
Company shall provide written evidence of the arrangements required under this Clause 5.2.3.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
5.3

5.4

5.5

5.6

5.7

5.8

Where  Licensed  Products  are  sold  or  Sub-Licence  Revenue  or  royalties  are  received  by  the  Company  (or  a  Sub-Licensee)  in  a
currency other than the Currency, the rate of exchange to be used for converting such other currency into the Currency shall be the
relevant mid-spot rate for the currency quoted by the Financial Times on the last day of the Quarter to which they relate.

All costs of transmission and currency conversion shall be borne by the Company.

All payments to CRT under this Agreement are expressed to be exclusive of value added tax howsoever arising, and the Company
shall pay to CRT in addition to those payments or, if earlier, on receipt of a tax invoice or invoices from CRT, all value added tax
for which CRT is liable to account in relation to any supply made or deemed to be made for value added tax purposes pursuant to
this Agreement.

All sums payable under this Agreement shall be paid without deduction or deferment in respect of any claims whatsoever and of any
taxes except any tax which the Company is required by law to deduct or withhold. If the Company is required by law to make any
such tax deduction or withholding, the Company shall pay to CRT such amount as shall, after deduction, amount to the sum referred
to in this Agreement give reasonable assistance to CRT to claim exemption from or (if that is not possible) a credit for the deduction
or withholding under any applicable double taxation or similar agreement from time to time in force, and shall promptly give CRT
proper evidence as to the deduction or withholding and payment over of the tax deducted or withheld.

Where CRT does not receive payment of any sums due to it by the due date, interest shall accrue both before and after any judgment
on the sum due and owing to CRT at the rate equivalent to an annual rate of two percent (2%) over the then current base rate of the
Bank  of  England,  calculated  on  a  daily  basis,  until  the  full  amount  is  paid  to  CRT,  without  prejudice  to  CRT’s  right  to  receive
payment on the due date.

Within thirty (30) days after the end of each Quarter, the Company shall send to CRT a written statement detailing in respect of that
Quarter (including a nil report if appropriate):

5.8.1

any Milestone Payments which became due to CRT;

5.8.2

5.8.3

for each sub-licence, details of each item of Sub-Licence Revenue received by the Company during that Quarter and the
Sub-Licence Revenue payable to CRT thereon;

the quantity of each type of Licensed Product sold or otherwise disposed of by the Company or any Sub-Licensees in each
country in the Territory;

5.8.4

the Net Sales Value in respect of each such type of Licensed Product in each country of the Territory;

5.8.5

the aggregate Net Sales Value in respect of that Quarter for Licensed Product;

5.8.6

the type and value of deductions made in the calculation of Net Sales Value by type of Licensed Product and country;

5.8.7

any currency conversions, showing the rates used;

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

5.8.8

any further information necessary for the calculation of Sub-Licence Revenue and Net Sales Value of Licensed Products
and/or the royalties due to CRT; and

5.8.9

the amount of the royalties due to CRT in respect of that Quarter.

6.

6.1

ACCOUNTS

The Company shall:

6.1.1

6.1.2

keep  and  notwithstanding  termination  of  this Agreement,  maintain  and  shall  procure  that  each  Sub-Licensee  keeps  and
maintains, for at least six (6) years, true and accurate accounts and records (including any underlying documents supporting
such  accounts  and  records)  in  sufficient  detail  to  enable  the  amount  of  all  sums  payable  under  this Agreement  to  be
determined; and

during the Term and thereafter until the said period of six (6) years relevant to the accounts and records has expired, at the
reasonable  request  of  CRT  and  (subject  to  Clause  6.2)  at  the  expense  of  CRT  from  time  to  time,  permit  or  procure
permission for a qualified accountant nominated by CRT to inspect and audit those accounts and records and, to the extent
that they relate to the calculation of those sums, to take copies of them. Subject to receiving not less than thirty (30) days
written  notice,  the  Company  shall  at  the  request  of  CRT  assemble  in  one  location  that  is  respectively  convenient  to  the
Company and Sub-Licensee(s) all such relevant accounts and records of the Company and all Sub-Licensee(s).

If, following any inspection pursuant to Clause 6.1.2, CRT’s nominated accountant certifies to CRT that the payments in respect of
any Quarter or Year fall short of the sums which were properly payable in respect of that Quarter or Year under this Agreement,
CRT shall send a copy of the certificate to the Company and the Company shall (subject to Clause 6.3) within thirty (30) days of
the date of receipt of the certificate pay the shortfall to CRT [***], the Company shall also reimburse to CRT the reasonable costs
and expenses of CRT in making the inspection.

If  within  fifteen  (15)  days  of  the  date  of  receipt  by  the  Company  any  certificate  produced  pursuant  to  Clause  6.2  the  Company
notifies  CRT  in  writing  that  it  disputes  the  certificate,  the  dispute  shall  be  referred  for  resolution  by Accountancy  Opinion  in
accordance with Clause 24.1.

INTELLECTUAL PROPERTY PROTECTION, PROCEEDINGS AND COSTS

The Company shall throughout the Term continue to use commercially reasonable efforts to prosecute and maintain the Company
Patent Rights. Notwithstanding the foregoing, if the Company elects not to prosecute or maintain any part of the Company Patent
Rights in any of the Major Markets, the Company shall notify CRT in writing at least ninety (90) days prior to the expiration of any
applicable time bars. After receipt of such notice, CRT may elect, before the expiry of any such time bars, by written notice to the
Company, to take an assignment of the relevant Company Patent Rights such that CRT may continue to prosecute and/or maintain
the Company Patent Rights at CRT’s sole discretion and expense.

WARRANTY

Each Party warrants that it has the legal capacity to enter into this Agreement.

Each  Party  acknowledges  that,  in  entering  into  this Agreement,  it  does  not  do  so  in  reliance  on  any  warranty  or  other  provision
except as expressly provided in this Agreement, and any conditions, warranties or other terms implied by statute or common law are
excluded to the fullest extent permitted by law.

6.2

6.3

7.

7.1

8.

8.1

8.2

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
8.3

Without limiting the scope of Clause 8.2, CRT does not give any warranty, representation or undertaking:

8.3.1

as to the efficacy or usefulness or accuracy of the Clinical Trial Results; or

8.3.2

that  the  exercise  of  rights  granted  under  this Agreement  will  not  infringe  the  intellectual  property  or  other  rights  of  any
other person.

9.

9.1

9.2

INDEMNITY

The Company shall indemnify and hold harmless CRT, the Contributors and the Charity and their respective officers, employees
and agents (each, an “Indemnified Party”) from and against any and all third party claims, demands, losses, damages and expenses
(including, without limitation, legal fees) arising from or in connection with the exercise of the rights granted in Clause 2 by the
Company  or  a  Sub-Licensee  or  the  actions  of  any Affiliate  of  any  of  them  in  relation  to  the  Licensed  Product.  This  Clause  9  is
without prejudice to and shall not limit the rights of the Company, and is without prejudice to and shall not limit the liabilities of
the Charity, under Clause 9.1 of the CTOA.

Promptly after receipt by CRT of any written claim or alleged claim or notice of the commencement of any action, administrative or
legal proceeding, or investigation to which the indemnity provided for in this Clause 9 may apply, CRT shall give written notice to
the  Company  of  such  fact  and  specifying  that  the  Company  shall  have  the  option  to  assume  the  defence  thereof  by  election  in
writing  within  seven  (7)  days  of  receipt  of  such  notice.  If  the  Company  fails  to  make  such  election,  the  Indemnified  Party  may
assume such defence and the Company will be liable for the legal and other expenses consequently incurred in connection with such
defence. If CRT fails to notify Company within thirty (30) days of receipt of any written claim or alleged claim or notice of the
relevant commencement, then the Company shall not be liable for the legal and other expenses consequently incurred in connection
with such defence. The Parties will co-operate in good faith in the conduct of any defence, provide such reasonable assistance as
may be required to enable any claim properly to be defended and the Party with conduct of the action shall provide promptly to the
other Party copies of all correspondence and documents and notice in writing of the substance of all oral communications relating to
such action.

9.3

Should the Company assume conduct of the defence:

9.3.1

9.3.2

the Indemnified Party may retain separate legal advisers, at its sole cost and expense save that if the Company denies the
applicability of the indemnity or reserves its position in relation to the same, the indemnity in this Clause 9 shall extend to
the  Indemnified  Party’s  costs  and  expenses  so  incurred  unless  it  is  subsequently  resolved  between  the  Parties  or
determined by a court of competent jurisdiction (after exhaustion or expiration of all rights of appeal) that the indemnity
under this Clause 9 was not available to the Indemnified Party in the terms claimed by the Indemnified Party;

the Company will not, except with the written consent of the Indemnified Party consent to the entry of any judgment or
enter into any settlement provided always, that if the Indemnified Party unreasonably refuses to consent to such entry of
judgment or settlement and the matter proceeds to trial at which a greater amount is ordered by the Court then the amount
which the Indemnified Party shall be entitled to recover from the Company pursuant to this Clause 9 shall be limited to the
amount for which the action would otherwise have been settled or compromised and the Indemnified Party shall assume all
costs of defending the claim or proceeding from the date of the Indemnified Party’s refusal;

 
 
 
 
 
 
 
 
 
 
 
 
9.3.3

CRT shall not admit liability in respect of, or compromise or settle any such action without the prior written consent of the
Company, such consent not to be unreasonably withheld, conditioned or delayed; and

9.3.4

the Company shall not be responsible for or bound by any settlement made by CRT in breach of Clause 9.3.3.

10.

INSURANCE

10.1

The Company shall maintain, at its own cost, comprehensive product liability insurance and general commercial liability insurance,
and shall ensure that each insurance policy maintained under this Clause 10.1 is held in the joint names of the Parties as co-insureds.
Within thirty (30) days of the Effective Date and of the beginning of each policy period, the Company shall provide CRT with a
certificate  evidencing  the  coverage  required  hereby,  and  the  amount  thereof.  Such  insurance  shall  be  with  a  reputable  insurance
company  and  shall  be  maintained  for  not  less  than  six  (6)  years  following  the  expiration/termination  of  this Agreement  for  any
reason or if such coverage is of the ‘claims made’ type, for ten (10) years following the expiration or termination of this Agreement
for any reason.

11.

LIMITATION OF LIABILITY

11.1

11.2

Neither Party nor the Charity, nor their respective officers, employees and agents shall have liability whether under statute or in tort
(including negligence), contract or otherwise to the other Party in respect of any consequential, indirect or pure economic loss nor in
any event for loss of goodwill, opportunity, profit or contract.

Nothing  in  this Agreement  shall  be  construed  as  excluding  or  limiting  the  liability  of  either  Party  or  the  Charity  or  any  of  their
respective officers, employees and agents to the other Party for death or personal injury of any person resulting from the negligence
of such persons.

12.

TERM AND TERMINATION

12.1

This Agreement will become effective on the Effective Date and, subject to the provisions of this Clause 12, will remain effective in
each  country  of  the  Territory  until  expiry  of  the  obligation  of  the  Company  to  pay  royalties  under  Clause  4.4  in  relation  to  that
country pursuant to this Agreement.

12.2 Without prejudice to any other rights of the Parties this Agreement may be terminated by notice in writing:

12.2.1

12.2.2

by either Party forthwith if the other Party shall be in material breach of any of its obligations under this Agreement and in
the  case  of  a  remediable  breach  fails  to  remedy  the  breach  within  ninety  (90)  days  of  written  notice  containing  full
particulars of the breach and requiring it to be remedied;

by  CRT  if  a  voluntary  arrangement  is  proposed  or  approved  or  an  administration  order  is  made,  or  a  receiver  or
administrative receiver is appointed of any of the Company’s assets or undertakings or a winding-up resolution or petition
is passed (otherwise than for the purpose of solvent reconstruction or amalgamation) or if any circumstances arise which
entitle the Court or a creditor to appoint a receiver, administrative receiver or administrator or make a winding-up order or
similar or equivalent action is taken against or by the Company by reason of its insolvency;

12.2.3

by CRT forthwith in the event that, by way of merger, acquisition or otherwise, the Company becomes a Tobacco Party; or

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

12.2.4

by CRT upon ninety (90) days written notice to the Company if the Company:

(a)

(b)

(c)

(d)

(e)

(f)

(g)

discontinues  the  development  (including  prosecuting  application  for  Regulatory Authorisation)  of  all  Licensed
Products; or

discontinues  the  development  (including  prosecuting  application  for  Regulatory  Authorisation)  of  a  Licensed
Product in relation to one or more Oncology Indications (in which case termination shall not apply to the whole
Agreement but shall be limited to such Licensed Product and such Oncology Indications); or

discontinues  the  development  (including  prosecuting  application  for  Regulatory Authorisation)  of  all  Licensed
Products in Oncology Indications (in which case termination shall not apply to the whole Agreement but shall be
limited to Oncology Indications); or

fails  to  use  its  commercially  reasonable  efforts  to  obtain  Regulatory Authorisation  in  all  of  the  Major  Markets
within fifteen (15) years, taking into account the unique aspects of the development and regulatory path for the
Licensed Product, indication and market (in which case termination shall not apply to the whole Agreement but
shall be limited to that Major Market); or

having obtained Regulatory Authorisation for a Licensed Product in a Major Market, ceases to actively market and
sell  such  Licensed  Product  in  such  Major  Market  (in  which  case  termination  shall  not  apply  to  the  whole
Agreement but shall be limited to that Licensed Product in that Major Market); or

ceases to carry on business in the Field; or

without reasonable cause fails to commence sales of any Licensed Product in a Major Market within two (2) years
of obtaining Regulatory Authorization to market such Licensed Product in such market (in which case termination
shall not apply to the whole Agreement but shall be limited to that Licensed Product in that Major Market).

12.3

12.4

The Company shall notify CRT in writing immediately upon any of the events described in Clause 12.2 occurring. However, CRT’s
right to terminate under Clause 12.2 shall not be conditional upon the Company’s such notice.

In the event of disagreement between the Parties as to whether entitlement to terminate has arisen under Clause 12.2.1 or 12.2.4, the
Parties at their joint cost and expense shall obtain an Expert Opinion which shall be final as to whether it has arisen.

13.

EFFECTS OF TERMINATION

13.1

Subject to Clause 13.2, upon the termination of this Agreement for any reason:

13.1.1

other  than  termination  by  CRT  pursuant  to  Clause  12.2.1,  12.2.2,  or  12.2.3  subject  to  all  the  terms  of  this Agreement
(including  without  limitation  payment  of  royalties),  the  Company  shall  be  entitled  for  a  period  not  exceeding  [***]
following such termination to:

(a)

manufacture any of the Licensed Products to the extent necessary to satisfy orders accepted before termination;
and

(b)

sell, use or otherwise dispose of any unsold stocks of the Licensed Products.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
13.1.2

subject to Clause 13.1.1, the Company shall, and shall procure that all Sub-Licensees shall, cease to exploit the Licensed
Intellectual Property in any way, either directly or indirectly;

13.1.3

subject  to  Clause  13.1.1,  the  Company  shall,  at  the  request  and  option  of  CRT,  return  or  destroy  CRT’s  Confidential
Information;

13.1.4

notwithstanding any provision of this Agreement allowing the Company credit, payment of royalties and all other sums to
CRT shall become due and payable to CRT immediately upon notice of termination of this Agreement;

13.1.5

the  Company  shall,  within  thirty  (30)  days  of  notice  of  termination  of  this Agreement  provide  CRT  with  a  final  written
statement detailing, in respect of the time elapsed since the last statement under Clause 5.8, the matters set out in Clause
5.8;

13.1.6

other than termination by the Company pursuant to Clause 12.2.1, the Company:

(a)

(b)

(c)

(d)

hereby grants to CRT an exclusive, perpetual, worldwide, sub-licensable licence under the Company Intellectual
Property, Company Patent Rights and New Company IP to research, develop, make, have made, market, use and
sell Licensed Products, on revenue share and, if appropriate, royalty terms to be agreed; provided that such licence
shall  only  become  effective  upon  termination,  and  not  before.  If,  having  regard  to  the  nature  and  status  of  the
rights licensed, the products to which they relate, the likely market for such products, the nature and standing of
potential  sub-licensees  and  actual  or  potential  competing  products,  the  Parties  cannot  agree  such  revenue  share
and, if appropriate, royalty terms within three (3) months of the date of termination then either Party may refer the
matter, subject to Clause 24.2, for determination by an Accountancy Opinion;

in the case of XOMA IP, hereby grants to CRT a sub-licence to the full extent of the Company‘s rights under the
XOMA Licence; provided that such licence shall only become effective upon termination, and not before;

at CRT’s request, shall promptly transfer to CRT (or any person nominated by CRT) any and all documents and
information  in  the  Company’s  Control  relating  to  the  Patent  Rights  exclusively  licensed  to  CRT  under  clause
13.1.6 above and CRT may assume responsibility for the prosecution, maintenance and enforcement of the same;
and

at CRT’s request, shall transfer to CRT (or its nominee) any Regulatory Authorisations, Price Approvals and other
permits and applications relating to Licensed Products.

13.2

This Clause 13.2 shall not apply in the case of termination of this Agreement under Clause 12.1. In the event that this Agreement is
terminated  solely  in  respect  of  particular  Licensed  Product  and/or  Indication  and/or  Major  Market,  the  provisions  of  Clause  13.1
shall apply, but solely in respect of the relevant Licensed Product, Indication and/or Major Market.

13.3

Insolvency:

13.3.1 All rights and licenses granted under or pursuant to Clause 13.1.6 by the Company to CRT are for all purposes of Section
365(n)  of  Title  11  of  the  U.S.  Bankruptcy  Code  (“Title 11”),  licenses  of  rights  to  “intellectual  property”  as  defined  in
Section 101 of Title 11.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
13.3.2

the Company agrees that CRT shall retain and may fully exercise all of its rights and elections under the U.S. Bankruptcy
Code. If a case under Title 11 is commenced by or against the Company, CRT shall have all rights of licensees set out in
Section 365(n) of Title 11;

13.3.3 without limiting CRT’s rights under Section 365(n) of Title 11, if a case under Title 11 is commenced by or against the
Company, and this Agreement is rejected by the Company in any bankruptcy proceeding by or against the Company under
the U.S. Bankruptcy Code, (i) the Company shall provide CRT with a complete duplicate of (and complete access to, as
appropriate) any IP and embodiments of IP not already in their possession; and (ii) the Company shall not interfere with
CRT’s rights to IP and embodiments of IP, and shall facilitate and assist with CRT obtaining IP and embodiments of IP
(including from a third party); and

13.3.4

the  term  “embodiments”  of  IP  includes  all  tangible,  intangible,  electronic  or  other  embodiments  of  rights  and  licenses,
including antibodies, compounds and products embodying IP and related rights and technology. All rights of CRT under
this Clause and under Section 365(n) of Title 11 are in addition to, not in substitution of, any other rights and remedies that
they may have under this Agreement, Title 11 and any other applicable law.

13.2

The termination of this Agreement howsoever arising will be without prejudice to the rights and duties of either Party accrued prior
to  termination.  The  following  Clauses  will  continue  to  be  enforceable  notwithstanding  termination:  Clauses  1  (Definitions),  6
(Accounts),  7.2  (XOMA  Licence),  9  (Indemnity),  10  (Insurance),  11  (Limitation  of  Liability),  12  (Termination),  13  (Effects  of
Termination), 14 (Confidentiality), 19 (Severability), 24 (Dispute Resolution) and 25 (Law and Jurisdiction).

14.

CONFIDENTIALITY

14.1

Each Party undertakes with the other that it shall keep and it shall procure that its respective directors and employees keep secret
and confidential all Confidential Information belonging to or Controlled by the other Party and shall not disclose the same or any
part of the same to any person whatsoever other than:

14.1.1

in  the  case  of  the  Company:  (i)  to  Sub-Licensees  subject  to  compliance  with  Clause  2.3.3,  (ii)  to  potential  development
partners,  sublicensees,  and  investors  bound  by  terms  of  confidentiality  at  least  as  strict  as  those  herein,  and  (iii)  as
necessary in communications with Regulatory Authorities in the Territory relating to the Licensed Products;

14.1.2

in the case of CRT to the Charity; and

14.1.3

in the case of each Party, to its directors or employees directly or indirectly concerned in the exercise of the rights granted
under this Agreement.

14.2

The provisions of Clause 14.1 shall not apply to Confidential Information which CRT or the Company (as the case may be):

14.2.1

can prove to have been in its possession (other than under an obligation of confidence to the other or to a third party) at the
date of receipt or which enters the public domain otherwise than through a breach of any obligation of confidentiality owed
to the Party communicating such information to the other;

14.2.2

can prove it has independently developed; or

14.2.3

is required to disclose by law or by the order of a competent court, solely to the extent of such disclosure.

14.3

The provisions of this Clause 14 shall remain in force for a period of five (5) years from the expiry or termination of this Agreement

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
15.

ASSIGNMENT

15.1

The  Company  shall  not  without  CRT’s  consent  assign  its  rights  under  this Agreement  except  in  conjunction  with  a  merger  or
consolidation of the Company with another business entity or the sale of all or substantially all or a substantial part of its business
and related assets that includes its business in relation to the Licensed Products other than a merger or consolidation with, or a sale
of assets to, a Tobacco Party and provided that Company obtains a direct covenant from the acquiring party to CRT undertaking to
be bound by the terms of this Agreement.

16.

NOTICES

16.1

Any notice or other document to be given under this Agreement shall be in writing and shall be deemed to have been given:

16.1.1

upon delivery if given in person; or

16.1.2

upon confirmation of receipt if sent by facsimile (or other similar means of electronic communication, such as email); or

16.1.3

(if posted to an inland destination) three (3) business days after deposit into First Class post; or

16.1.4

(If posted to an overseas destination) five (5) days after deposit into airmail post; or

16.1.5

upon delivery by air delivery service,

to a Party at the address set out below (or, if provided below or so notified, such facsimile or electronic communication) for such Party or
such other address as the Party may from time to time designate by written notice to the other Party.  [As  may  be  updated  at  the
Effective Date.]

Address of the Company

Monopar Therapeutics LLC

598 Rockefeller Road

Lake Forest, IL USA 60045

Contact:  Chief Executive Officer

Address of CRT

Angel Building

407 St. John Street

London EC1V 4AD

United Kingdom

Contact: Chief Executive Officer

Fax: +44 (0) 20 3014 8633

17.

WAIVER

17.1

No failure or delay on the part of either Party hereto to exercise any right or remedy under this Agreement shall be construed as or
operate as a waiver thereof nor shall any single or partial exercise of any right or remedy under this Agreement preclude the exercise
of any other right or remedy or preclude the further exercise of such right or remedy as the case may be.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
18.

FORCE MAJEURE

18.1

Except in relation to obligations pursuant to Clauses 4 and/or 5, neither Party shall be liable to the other Party or shall be in default
of its obligations hereunder if such default is the result of war, hostilities, revolution, civil commotion, strike, epidemic, accident,
fire, wind, flood or because of any act of God or other cause beyond the reasonable control of the Party affected. The Party affected
by  such  circumstances  shall  promptly  notify  the  other  Party  in  writing  when  such  circumstances  cause  a  delay  or  failure  in
performance (a “Delay”) and where they cease to do so. In the event of a Delay lasting for twenty six (26) weeks or more the non-
affected Party shall have the right to terminate this Agreement immediately by notice in writing to the affected Party.

19.

SEVERABILITY

19.1

If  and  to  the  extent  that  any  court  or  tribunal  of  competent  jurisdiction  holds  any  of  the  terms,  provisions  or  conditions  or  parts
thereof  of  this Agreement,  or  the  application  hereof  to  any  circumstances,  to  be  invalid  or  to  be  unenforceable  in  a  final  non-
appealable  order,  the  remainder  of  this Agreement  and  the  application  of  such  term,  provision  or  condition  or  part  thereof  to
circumstances other than those as to which it is held invalid or unenforceable shall not be affected thereby, and each of the other
terms, provisions and conditions of this Agreement shall be valid and enforceable to the fullest extent permissible by law.

20.

ENTIRE AGREEMENT

20.1

This Agreement  and  the  surviving  clauses  of  the  CTOA,  embodies  and  sets  forth  the  entire  agreement  and  understanding  of  the
Parties  and  supersedes  all  prior  oral  or  written  agreements,  understandings  or  arrangements  relating  to  the  subject  matter  of  this
Agreement.  Without  prejudice  to  any  liability  for  fraudulent  misrepresentation  or  fraudulent  misstatement  neither  Party  shall  be
entitled to rely on any agreement, understanding or arrangement which is not expressly set forth in this Agreement unless otherwise
agreed between the Parties and recorded in writing.

21.

AMENDMENT

21.1

This Agreement shall not be amended, modified, varied or supplemented except in writing signed by duly authorised representatives
of the Parties.

22.

PUBLIC ANNOUNCEMENTS

22.1

The text of any press release, shareholders’ report or other communication to be published or disclosed to the public in any way by
or in the media concerning CRT or the Charity, the subject matter of this Agreement or concerning this Agreement itself, other than
as required by law or by any Regulatory Authority or the rules of any securities exchange, shall be submitted to CRT at least seven
(7) days in advance of publication for approval, such approval not to be unreasonably withheld, conditioned, or delayed, provided
that insofar as a disclosure repeats or restates a prior public disclosure permitted by this Agreement, such disclosure need not be
submitted to the Charity or CRT for approval.

23.

FURTHER ASSURANCE

23.1

The  Parties  hereby  undertake  to  do  all  such  other  acts  and  things,  and  execute  and  provide  all  such  documents  at  the  requesting
Party’s cost as may be necessary or desirable to give effect to the purposes of this Agreement.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
24.

DISPUTE RESOLUTION

24.1

24.2

Insofar as this Agreement provides that a matter shall be resolved by Accountancy Opinion or Expert Opinion the opinion of such
expert (who shall act as an expert and not as an arbitrator) shall be final and binding on the Parties. In the event of a Party seeking
an Accountancy  Opinion  or  Expert  Opinion  under  this Agreement,  each  Party  shall  make  written  submissions  to  the  expert  so
appointed and to the other Party within fourteen (14) days of the appointment. Each Party shall have seven (7) days to respond to
the other’s submissions. The expert shall be requested to deliver his Accountancy Opinion or Expert Opinion within a further thirty
(30) days. The costs of any Accountancy Opinion or Expert Opinion shall be borne in such proportions as the expert may determine
in his opinion to be fair and reasonable in all the circumstances or, if no such determination is made in the opinion, by the Parties in
equal proportions.

It  shall  be  a  condition  precedent  to  the  commencement  of  any  action  in  court  or  other  tribunal  (save  an  action  for  an  interim
injunction or an Expert Opinion sought under Clause 12.1) in respect of any dispute relating to this Agreement that the Parties have
sought to resolve the dispute by either Party notifying the other Party in writing for resolution to the Chief Executive Officer (in the
case of CRT) and the Chief Executive Officer (in the case of the Company) (or their express delegates) (the “Senior Executives”)
who shall meet (whether in person or via teleconference) within twenty one (21) days of such notice to seek resolution in good faith.
If the Senior Executives are unable to resolve the dispute at such meeting, either Party may pursue any remedy available to such
Party at law or in equity, subject to the terms and conditions of this Agreement and the other agreements expressly contemplated
hereunder.

25.

LAW AND JURISDICTION

25.1

This Agreement shall be governed by and construed in accordance with English Law and, subject to the provisions of Clauses 24.1
and 24.2, each Party agrees to submit to the exclusive jurisdiction of the English Courts (except in respect of disputes under Clause
14 where jurisdiction is non-exclusive).

26.

EXECUTION

26.1

This Agreement may be executed in any one or more number of counterpart agreements, and as scanned email attachments, and all
signatures and counterparts so exchanged shall be considered as original and shall be deemed to form part of and together constitute
this Agreement.

27.

CONTRACTS (RIGHTS OF THIRD PARTIES) ACT 1999

27.1

Save that the Charity, the Contributors and their and CRT’s respective officers, employees and agents in respect of Clauses 9 and 11
may  enforce  those  respective  terms,  no  term  of  this Agreement  is  enforceable  under  the  Contracts  (Rights  of  Third  Parties) Act
1999 by a person who is not a Party to this Agreement. Notwithstanding the provisions of this Clause, the Parties shall be entitled to
amend, suspend, cancel or terminate this Agreement or any part of it in accordance with Clause 21, without the consent of any third
party including those referred to in this Clause.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
The Parties hereby execute this Agreement by their duly authorised representatives:

Signed by:

_____________________________________

Name:

Title:

_____________________________________

_____________________________________

For and on behalf of
CANCER RESEARCH TECHNOLOGY LIMITED

Signed by:

_____________________________________

Name:

Title:

_____________________________________

 _____________________________________

For and on behalf of
MONOPAR THERAPEUTICS LLC

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Appendix 1
Development Plan

Appendix 2
Executed CTOA

 
 
 
 
 
 
 
 
 
 
 
Preamble

Schedule 4
No Fault Compensation Scheme

The  Association  of  the  British  Pharmaceutical  Industry  favours  a  simple  and  expeditious  procedure  in  relation  to  the  provision  of
compensation  for  injury  caused  by  participation  in  clinical  trials.  The  Association  therefore  recommends  that  a  member  company
sponsoring  a  clinical  trial  should  provide  without  legal  commitment  a  written  assurance  to  the  investigator  —  and  through  him  to  the
relevant research ethics committee — that the following Guidelines will be adhered to in the event of injury caused to a patient attributable
to participation in the trial in question.

1      Basic Principles

1.1 

1.2 

1.3 

1.4 

1.5 

1.6 

1.7 

Notwithstanding  the  absence  of  legal  commitment,  the  company  should  pay  compensation  to  patient-volunteers  suffering  bodily
injury (including death) in accordance with these Guidelines.

Compensation should be paid when, on the balance of probabilities, the injury was attributable to the administration of a medicinal
product under trial or any clinical intervention or procedure provided for by the protocol that would not have occurred but for the
inclusion of the patient in the trial.

Compensation should be paid to a child injured in utero through the participation of the subject’s mother in a clinical trial as if the
child were a patient-volunteer with the full benefit of these Guidelines.

Compensation should only be paid for the more serious injury of an enduring and disabling character (including exacerbation of an
existing condition) and not for temporary pain or discomfort or less serious or curable complaints.

Where there is an adverse reaction to a medicinal product under trial and injury is caused by a procedure adopted to deal with that
adverse reaction, compensation should be paid for such injury as if it were caused directly by the medicinal product under trial.

Neither the fact that the adverse reaction causing the injury was foreseeable or predictable, nor the fact that the patient has freely
consented (whether in writing or otherwise) to participate in the trial should exclude a patient from consideration for compensation
under  these  Guidelines,  although  compensation  may  be  abated  or  excluded  in  the  light  of  the  factors  described  in  paragraph  4.2
below.

For the avoidance of doubt, compensation should be paid regardless of whether the patient is able to prove that the company has
been  negligent  in  relation  to  research  or  development  of  the  medicinal  product  under  trial  or  that  the  product  is  defective  and
therefore, as the producer, the company is subject to strict liability in respect of injuries caused by it.

2      Type of Clinical Research Covered

2.1 

2.2 

These Guidelines apply to injury caused to patients involved in Phase II and Phase III trials, that is to say, patients under treatment
and surveillance (usually in hospital) and suffering from the ailment which the medicinal product under trial is intended to treat but
for which a product licence does not exist or does not authorise supply for administration under the conditions of the trial.

These  Guidelines  do  not  apply  to  injuries  arising  from  studies  in  non-patient  volunteers  (Phase  I),  whether  or  not  they  are  in
hospital, for which separate Guidelines for compensation already exist.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
2.3 

2.4

These Guidelines do not apply to injury arising from clinical trials on marketed products (Phase IV) where a product licence exists
authorising supply for administration under the conditions of the trial, except to the extent that the injury is caused to a patient as a
direct  result  of  procedures  undertaken  in  accordance  with  the  protocol  (but  not  any  product  administered)  to  which  the  patient
would not have been exposed had treatment been other than in the course of the trial.

These Guidelines do not apply to clinical trials which have not been initiated or directly sponsored by the company providing the
product  for  research.  Where  trials  of  products  are  initiated  independently  by  doctors  under  the  appropriate  Medicines Act  1968
exemptions, responsibility for the health and welfare of patients rests with the doctor alone (see also paragraph 5.2 below).

3            Limitations

3.1 

3.2 

3.3 

3.4 

No compensation should be paid for the failure of a medicinal product to have its intended effect or to provide any other benefit to
the patient.

No compensation should be paid for injury caused by other licensed medicinal products administered to the patient for the purpose
of comparison with the product under trial.

No compensation should be paid to patients receiving placebo in consideration of its failure to provide therapeutic benefit.

No compensation should be paid (or it should be abated as the case may be) to the extent that the injury has arisen:

3.4.1 

through a significant departure from the agreed protocol;

3.4.2 

through the wrongful act or default of a third party, including a doctor’s failure to deal adequately with an adverse reaction;

3.4.3

through contributory negligence by the patient.

4        Assessment of Compensation

4.1 

4.2 

The amount of compensation paid should be appropriate to the nature, severity and persistence of the injury and should in general
terms be consistent with the quantum of damages commonly awarded for similar injuries by an English Court in cases where legal
liability is admitted.

Compensation may be abated, or in certain circumstances excluded, in the light of the following factors (on which will depend the
level of risk the patient can reasonably be expected to accept):

4.2.1

the seriousness of the disease being treated, the degree of probability that adverse reactions will occur and any warnings
given;

4.2.2

the risks and benefits of established treatments relative to those known or suspected of the trial medicine.

This reflects the fact that flexibility is required given the particular patient’s circumstances. As an extreme example, there may be a
patient suffering from a serious or life-threatening disease who is warned of a certain defined risk of adverse reaction. Participation
in the trial is then based on an expectation that the benefit/risk ratio associated with participation may be better than that associated
with alternative treatment. It is, therefore, reasonable that the patient accepts the high risk and should not expect compensation for
the occurrence of the adverse reaction of which he or she was told.

4.3 

In any case where the company concedes that a payment should be made to a patient but there exists a difference of opinion between
company and patient as to the appropriate level of compensation, it is recommended that the company agrees to seek at its own cost
(and make available to the patient) the opinion of a mutually acceptable independent expert, and that his opinion should be given
substantial weight by the company in reaching its decision on the appropriate payment to be made.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
5       Miscellaneous

5.1 

5.2 

5.3 

5.4 

Claims pursuant to the Guidelines should be made by the patient to the company, preferably via the investigator, setting Out details
of the nature and background of the claim and, subject to the patient providing on request an authority for the company to review
any medical records relevant to the claim, the company should consider the claim expeditiously.

The undertaking given by a company extends to injury arising (at whatever time) from all administrations, clinical interventions or
procedures occurring during the course of the trial but not to treatment extended beyond the end of the trial at the instigation of the
investigator. The use of unlicensed products beyond the trial period is wholly the responsibility of the treating doctor and in this
regard  attention  is  drawn  to  the  advice  provided  to  doctors  in  MAL  3Q2  concerning  the  desirability  of  doctors  notifying  their
protection society of their use of unlicensed products.

The fact that a company has agreed to abide by these Guidelines in respect of a trial does not affect the right of a patient to pursue a
legal remedy in respect of injury alleged to have been suffered as a result of participation. Nevertheless, patients will normally be
asked to accept that any payment made under the Guidelines will be in full settlement of their claims.

A  company  sponsoring  a  trial  should  encourage  the  investigator  to  make  clear  to  participating  patients  that  the  trial  is  being
conducted  subject  to  the ABPI  Guidelines  relating  to  compensation  for  injury  arising  in  the  course  of  clinical  trials  and  have
available copies of the Guidelines should they be requested.

References

1            Guidelines for Medical Experiments in Non-patient Human Volunteers, ABPI March 1988, as amended May 1990.
2            MAL 30— A Guide to the Provisions affecting Doctors and Dentists, DHSS, (Revised June 1985)

The Association of the British Pharmaceutical Industry
12 Whitehall London SW1

 
 
 
 
 
 
 
 
 
 
 
 
 
 
Schedule 5
Assignment and Licence from Company to CRT

THIS AGREEMENT is made the________ day of _______________________20[●●]

BETWEEN:

(1)

(2)

CANCER  RESEARCH  TECHNOLOGY  LIMITED,  a  company  registered  in  England  and  Wales  with  number  1626049  with
registered office at Angel Building, 407 St. John Street, London, EC1V 4AD, England (“CRT”); and

[MONOPAR THERAPEUTICS LLC, a limited liability company registered in/incorporated in/ established under the laws of The
State of Delaware, U.S.A., with registered office/principal place of business at 598 Rockefeller Road, Lake Forest, Illinois, U.S.A.,
60045] (the “Company”).

WHEREAS

(A)

(B)

CRT,  the  Company  and  the  Charity  (as  defined  below)  are  parties  to  a  Clinical  Trial  and  Option Agreement  dated  [●●●]  (the
“CTOA”) relating to the Investigational Medicinal Product (as defined in the CTOA).

Pursuant  to  clause  7.5  of  the  CTOA,  the  Company  has  agreed  to  assign  the  Company  Intellectual  Property  and  sub-license  the
XOMA IP in return for a royalty and a share of any revenue generated by CRT from the commercial exploitation of such intellectual
property rights upon the terms and conditions set out below.

NOW IT IS HEREBY AGREED as follows:

1.

1.1

INTERPRETATION

In  this Agreement  except  where  the  context  requires  otherwise,  the  following  words  and  expressions  shall  have  the  following
meanings:

“Affiliate”

has the same meaning as that ascribed to that phrase in the CTOA.

“Accountancy
Opinion”

means  the  opinion  of  an  independent  United  Kingdom  chartered  accountant  appointed  by  agreement  between  the
Parties or in default of such agreement within twenty one (21) days of either Party seeking in writing to the other to
appoint  such  accountant,  at  the  request  of  either  Party,  by  the  President  for  the  time  being  of  the  Institute  of
Chartered Accountants in England and Wales, referred to in Clauses 6.3 and 12.1.

“Charity”

means  Cancer  Research  UK,  a  charity  registered  under  number  1089464  of Angel  Building,  407  St.  John  Street,
London EC1V 4AD, England.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
“Clinical Trial”
“Company
Intellectual
Property”
“Company  Know-
How”

has the meaning given in the CTOA.
means  the  Company  Patent  Rights  and  all  rights  in  the  Company  Materials,  the  Investigational  Medicinal  Product
and the Company Know-How.

means: (a) any Know How that was disclosed by the Company to the Charity pursuant to the CTOA; (b) any Know
How described in Annex 2; and (c) such other Know How in the Company’s Control relating to the Investigational
Medicinal Product (and any constituents thereof) or any Back-Up Antibody including but not limited to: (i) any safety
and toxicological data; (ii) information relating to manufacturing/production; (iii) information relating to quality; (iv)
information relating to safe and proper handling, storage and use; and (v) any information which would in any way
improve the prospects for its commercialisation.

“Company
Materials”

means Materials Controlled by the Company which include and relate to the Investigational Medicinal Product, the
Antibody and the Back-Up Antibodies, more particularly described in Annex 3.

“Company  Patent
Rights”

means (i) those Patent Rights listed in Annex 1A; (ii) those Patent Rights Controlled by the Company which would
be  infringed  by  the  unauthorised  manufacture,  use  or  sale  in,  or  importation  into,  the  relevant  country  of  the
Investigational Medicinal Product, Antibody or Back-Up Antibodies; and (iii) all Patent Rights deriving priority from
(i) and (ii).

“Control”
“Data Exclusivity
Period”

has the meaning given in the CTOA.
means any period of clinical trial data or other regulatory exclusivity, together with any such periods under national
implementations in the European Union of Article 10.1 of Directive 2001/EC/83 and all equivalents elsewhere in the
Territory.

“Direct Costs”

means XOMA Licence Payments paid by CRT pursuant to Clause 7.2.

“Effective Date” means the date of this Agreement.

“First Commercial
Sale”

means, with respect to a Licensed Product, the first transfer or disposition for value of such Licensed Product by or
on behalf of CRT or a Sub-Licensee or an Affiliate of either of them, after all relevant Regulatory Authorisations for
the transfer or disposition of such Licensed Product have been obtained in respect of the relevant region or country.

 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

“Gross Revenue” means any and all monies or non-monetary consideration (including securities) received by CRT from time to time in
respect of the commercial exploitation of the Investigational Medicinal Product, Antibody, Back-Up Antibodies, or
any  Licensed  Product;  [***].  For  the  avoidance  of  doubt,  any  developmental  and/or  sales  milestone  revenue  shall
constitute Gross Revenue, and not Royalties.

“Investigational
Medicinal
Product” or “IMP”

“Intellectual
Property Rights”

“Know-How”
“Licence”
“Licensed
Product”

has the meaning given in the CTOA.

means  all  Patent  Rights,  Know-How,  copyright,  database  rights,  design  rights,  moral  rights,  rights  in  trade  names,
logos and trade and service marks, domain names, rights in Materials and all rights or forms of protection of a similar
nature or having equivalent or similar effect to any of them which may subsist anywhere in the world, whether or not
any of them are registered including any application for registration of any of them.

has the meaning given in the CTOA.
has the meaning given in the CTOA.
means any product:

a) whose application for a Regulatory Authorisation from a Regulatory Authority in any jurisdiction

included the Clinical Trial Results and/or the Final Report and/or the Data Listings or any part of any of
them, and/or

b) that contains the Antibody or a Back-Up Antibody (or any part of either), in each case whether or

not as the sole active ingredient, and/or

c) the unauthorised manufacture, sale or use of which would infringe a valid claim of the Company

Patent Rights,

where “Clinical Trial Results”, “Final Report” and “Data Listings” have the meaning given to them in the CTOA
and “Regulatory Authorisation” has the meaning given to it in the Licence.

 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

“Materials”
“NDA”

has the meaning given in the CTOA.
means, in relation to any Licensed Product, a biologics license application, new drug application, supplementary new
drug application, abbreviated new drug application or any of their equivalents filed with the United States Food and
Drugs Administration (FDA) or any successor to it, a marketing authorisation application or its equivalent filed with
the European Medicines Agency (EMEA) or any successor to it, or a marketing authorisation application or a product
licence application or equivalent filed with the relevant Regulatory Authority in any one or more countries or regions
within the Territory.

means Gross Revenue less Direct Costs.

“Net Revenue”
“Net Sales Value” means, in relation to Licensed Product, the gross amount invoiced by CRT or Sub-Licensee or Affiliate of CRT or a
Sub-Licensee [***] to the extent that any of those items are included as separate items in the amount so invoiced, and
[***]

“Party”

means either party to this Agreement and “Parties” means both of them.

“Patent Rights”
“Royalties”

has the meaning given in the CTOA.
means any monies that CRT receives from a Sub-Licensee which are a percentage of Net Sales Value only, and are
paid to CRT on a Licensed-Product by Licensed-Product and country-by-country basis.

“Sub-Licensee”

means  any  person  who  is  granted  a  sub-licence  in  respect  of  the  Company  Intellectual  Property  under  this
Agreement;  and/or  any  person  who  is  granted  a  sub-licence  (whether  under  the  Company  Intellectual  Property  or
otherwise) to sell Licensed Products anywhere in the Territory, but shall not mean distributors, wholesalers, and sales
agents (sale to whom will be sales for the purpose of Net Sales Value).

 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

means worldwide.
“Territory”
“XOMA IP”
has the meaning given in the CTOA.
“XOMA Licence” has the meaning given in the CTOA.
has the meaning given in the CTOA.
“XOMA Licence
Payments”

1.2

2.

2.1

2.2

2.3

2.4

2.5

The  headings  in  this  Agreement  are  for  convenience  only  and  shall  not  affect  its  interpretation.  Unless  the  contrary  intention
appears, words denoting persons shall include any individual, partnership, company, corporation, joint venture, trust, association,
organisation  or  other  entity,  in  each  case  whether  or  not  having  separate  legal  personality.  References  to  the  words  “include”  or
“including” shall be construed without limitation to the generality of the preceding words.

ASSIGNMENT AND LICENCE FROM COMPANY TO CRT

Pursuant to clause 7.5 of the CTOA, and in consideration of the provisions of Clause 4, the Company hereby assigns to CRT with
full title guarantee:

2.1.1

[***] the Company Patent Rights (and the inventions disclosed in such Company Patent Rights) and the [***];

2.1.2

[***] the Company Intellectual Property and [***];

2.1.3

[***] the Company Intellectual Property [***];

2.1.4

[***] the Company Patent Rights; and

2.1.5

[***].

Effective only upon a written request from CRT and to the extent it is entitled to do so under the XOMA Licence, the Company
hereby grants to CRT [***] to research, develop, make, have made, import, use and sell the Investigational Medicinal Product and
products incorporating the Antibody or any Back-Up Antibody. The licence granted under this Clause 2.2 shall become effective
upon written notice from CRT to the Company (such notice to be given within thirty (30) days of the Effective Date).

The Company shall disclose to CRT any Company Know-How that was not already disclosed to CRT pursuant to the CTOA within
three (3) months of the Effective Date and agrees that the Company Know-How may be used by CRT and anyone to whom CRT
discloses the Company Know-How, and that the Company shall not disclose the Company Know-How to any third party or use the
Company Know-How in any internal research programme.

The Company either has or shall transfer, or procure the transfer of, the Company Materials and any and all rights therein to CRT
(or any third party nominated by CRT) within three (3) months of the Effective Date and agrees that the Company Materials may be
used by CRT and any third party authorised by CRT and that the Company shall not transfer any Company Materials to any third
party or use the Company Materials in any internal research programme.

At CRT’s request, the Company shall negotiate with CRT in good faith on reasonable commercial terms a [***] the Company and
not  already  licensed  or  assigned  under  this  Agreement  which  may  be  necessary  and/or  useful  for  the  development  and/or
commercial exploitation of the Company Intellectual Property.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
3.

3.1

3.2

3.3

3.4

3.5

ASSISTANCE AND FURTHER ASSURANCE

The  Company  shall  promptly  provide  to  CRT  or  its  nominated  patent  agent  all  documents  relating  to  the  filing,  prosecution  and
maintenance of the Company Patent Rights.

The Company shall execute, sign and do all instruments, applications, documents, acts and things that may reasonably be required
by CRT to enable CRT to enjoy the full benefit of the property and rights hereby assigned or licensed and (if requested to do so by
CRT) to apply for any patents or other forms of protection in respect of the Investigational Medicinal Product throughout the world
and fully and effectively to assign the same to CRT or as CRT shall direct.

The Company shall assist CRT and any third party that CRT may nominate in understanding and using the Company Know-How
and the Company Materials and assist CRT and any such third party in relation to any further development of the Investigational
Medicinal  Product  and  any  regulatory  application  in  relation  thereto  (including  without  limitation  and  to  the  extent  that  the
Company  may  lawfully  do  so  by  the  provision  of  information  that  may  be  requested  from  time  to  time  in  relation  to  the  origin,
development, and distribution by the Company to any third parties of the Licensed Product).

The Company shall maintain the XOMA Licence, and not terminate it without the prior written agreement of CRT.

To the extent it has the rights under the XOMA Licence to Control Patent Rights which are XOMA IP, the Company shall transfer
to CRT control of the filing, prosecution, maintenance, enforcement and defence of any such Patent Rights to CRT.

 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

4.

4.1

4.2

4.3

CONSIDERATION

Subject to Clause 4.5, CRT and the Company shall share Net Revenue in the following proportions:

CRT [***];
Company [***].

In the event that any Gross Revenue is received by CRT as part of the consideration for the grant of rights  which  include  rights
other than those in respect of Company Intellectual Property, CRT shall apportion the consideration as between on the one hand, the
rights granted in respect of the Company Intellectual Property and, on the other, any other rights granted, in such manner as is fair
and reasonable.

If  CRT  receives  any  non-monetary  consideration  in  respect  of  the  commercial  exploitation  of  the  Company  Intellectual  Property
(such as company stocks and shares), such non-monetary consideration shall not form Gross Revenue until CRT has received cash
proceeds  from  the  disposal  or  other  realisation  of  such  consideration.  CRT  shall  not  determine  the  timing  of  and  price  for  any
realisation  of  the  Company’s  share  of  non-monetary  consideration  without  first  having  notified  and  consulted  the  Company,  but
shall  otherwise  seek  to  realise  such  non-monetary  consideration  at  the  earliest  opportunity  that  is  consistent  with  securing  a
reasonable  return.  For  the  avoidance  of  doubt,  any  dividend  or  similar  monetary  consideration  received  in  respect  of  such  non-
monetary consideration shall form Gross Revenue.

4.4

Subject to Clause 4.5, CRT and the Company shall share any Royalties received by CRT in each calendar quarter of the Royalty
Term in the following proportions:

 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

CRT [***];
Company [***],

provided that under no circumstance other than that set out in Clause 4.5 shall CRT pay the Company under this Clause 4.4 [***] in each
such calendar quarter. CRT shall include in any and all sub-licenses granted under this Agreement obligations on its sub-licensee(s)
to  make  timely  payments  (on  not  less  than  a  quarterly  basis)  of  sufficient  royalties  to  CRT  to  ensure  that  CRT  can  meet  its
obligations under this Clause 4.4.

In this Clause 4.4, “Royalty Term” means a period, on a Licensed Product-by-Licensed Product, country-by-country basis, beginning on the

Effective Date and ending upon the later to occur of:

4.4.1

the expiry of any Data Exclusivity Period in respect of the data submitted for the NDA for such Licensed Product in such
country;

4.4.2

the expiry of ten (10) years from the First Commercial Sale; and

4.4.3

the date when unauthorised manufacture, sale or use of the Licensed Product would no longer infringe a valid claim of the
Company Patent Rights in the country of sale or manufacture.

Without restricting or limiting any of the Charity’s or CRT’s rights under the CTOA, CRT may deduct as a first charge and set off
from sums due to the Company under this Clause 4 any and all sums of any nature that are due and payable, but not yet paid, by the
Company to CRT or the Charity under or in connection with the CTOA (including, without limitation, any sums due pursuant to
Clause 9.2 or 12.2 of the CTOA).

PAYMENT AND STATEMENT

All  payments  due  to  the  Company  under  this Agreement  shall  be  made  in  United  States  Dollars  in  cleared  funds  to  such  bank
account as Company may notify to CRT from time to time.

4.5

5.

5.1

5.2

CRT shall pay to Company:

5.3

5.4

5.5

5.6

5.2.1

payments due under Clause 4.1, Clause 4.2, and Clause 4.3 within thirty (30) days of CRT receiving the revenue; and

5.2.2

the  payments  due  pursuant  to  Clause  4.4  Quarterly  within  thirty  (30)  days  of  the  end  of  each  Quarter  in  which  the
corresponding Royalties are received by CRT.

Where  Licensed  Products  are  sold  or  Sub-Licence  Revenue  or  Royalties  are  received  by  CRT  (or  a  Sub-Licensee)  in  a  currency
other than United States Dollars, the rate of exchange to be used for converting such other currency into United States Dollars shall
be the relevant mid-spot rate for the currency quoted by the Financial Times on the last day of the Quarter to which they relate.

All costs of transmission and currency conversion shall be borne by CRT.

All payments to the Company under this Agreement are expressed to be exclusive of value added tax howsoever arising, and CRT
shall pay to the Company in addition to those payments or, if earlier, on receipt of a tax invoice or invoices from the Company, all
value added tax for which the Company is liable to account in relation to any supply made or deemed to be made for value added
tax purposes pursuant to this Agreement.

All sums payable under this Agreement shall be paid without deduction or deferment in respect of any claims whatsoever and of any
taxes except any tax which CRT is required by law to deduct or withhold. If CRT is required by law to make any such tax deduction
or  withholding,  CRT  shall  pay  to  the  Company  such  amount  as  shall,  after  deduction,  amount  to  the  sum  referred  to  in  this
Agreement give reasonable assistance to the Company to claim exemption from or (if that is not possible) a credit for the deduction
or withholding under any applicable double taxation or similar agreement from time to time in force, and shall promptly give the
Company proper evidence as to the deduction or withholding and payment over of the tax deducted or withheld.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
5.7

5.8

Where the Company does not receive payment of any sums due to it by the due date, interest shall accrue both before and after any
judgment  on  the  sum  due  and  owing  to  the  Company  at  the  rate  equivalent  to  an  annual  rate  of  two  percent  (2%)  over  the  then
current  base  rate  of  the  Bank  of  England,  calculated  on  a  monthly  basis,  until  the  full  amount  is  paid  to  the  Company,  without
prejudice to the Company’s right to receive payment on the due date.

Within thirty (30) days after the end of each Quarter, CRT shall send to the Company a written statement detailing in respect of that
Quarter (including a nil report if appropriate):

5.8.1

any payments which became due to Company;

5.8.2

5.8.3

for  each  sub-licence,  details  of  each  item  of  Sub-Licence  Revenue  received  by  CRT  during  that  Quarter  and  the  Sub-
Licence Revenue payable to Company thereon;

the quantity of each type of Licensed Product sold or otherwise disposed of by CRT or any Sub-Licensees in each country
in the Territory;

5.8.4

the Net Sales Value in respect of each such type of Licensed Product in each country of the Territory;

5.8.5

the aggregate Net Sales Value in respect of that Quarter for Licensed Product;

5.8.6

the type and value of deductions made in the calculation of Net Sales Value by type of Licensed Product and country;

5.8.7

any currency conversions, showing the rates used;

5.8.8

any further information necessary for the calculation of Sub-Licence Revenue and Net Sales Value of Licensed Products
and/or the Royalties due to Company; and

5.8.9

the amount of the Royalties due to Company in respect of that Quarter.

6.

6.1

ACCOUNTS

CRT shall:

6.1.1

6.1.2

keep  and  notwithstanding  termination  of  this Agreement,  maintain  and  shall  procure  that  each  Sub-Licensee  keeps  and
maintains,  for  at  least  three  (3)  years,  true  and  accurate  accounts  and  records  (including  any  underlying  documents
supporting such accounts and records) in sufficient detail to enable the amount of all sums payable under this Agreement to
be determined; and

during the Term and thereafter until the said period of three (3) years relevant to the accounts and records has expired, at
the reasonable request of Company and (subject to Clause 6.2) at the expense of the Company from time to time, permit or
procure permission for a qualified accountant nominated by the Company to inspect and audit those accounts and records
and, to the extent that they relate to the calculation of those sums, to take copies of them. Subject to receiving not less than
thirty  (30)  days  written  notice,  CRT  shall  at  the  request  of  the  Company  assemble  in  one  location  that  is  respectively
convenient to CRT and Sub-Licensee(s) all such relevant accounts and records of CRT and all Sub-Licensee(s).

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

6.2

6.3

7.

7.1

7.2

8.

8.1

9.

9.1

If,  following  any  inspection  pursuant  to  Clause  6.1.2,  the  Company’s  nominated  accountant  certifies  to  the  Company  that  the
payments in respect of any Quarter or Year fall short of the sums which were properly payable in respect of that Quarter or Year
under this Agreement, the Company shall send a copy of the certificate to CRT and CRT shall (subject to Clause 6.3) within thirty
(30) days of the date of receipt of the certificate pay the shortfall to the Company and, [***] of the sum properly payable, CRT shall
also reimburse to the Company the reasonable costs and expenses of the Company in making the inspection.

If within fifteen (15) days of the date of receipt by CRT any certificate produced pursuant to Clause 6.2 CRT notifies the Company
in  writing  that  it  disputes  the  certificate,  the  dispute  shall  be  referred  for  resolution  by Accountancy  Opinion  in  accordance  with
Clause 12.1.

XOMA LICENCE

As of the Effective Date and subject to any notices served pursuant to Clause 8.2.11 of the CTOA, the Company hereby restates and
gives  the  warranties  and  representations  set  out  in  Clause  8.2  of  the  CTOA  (save  that  references  in  such  provisions  to:  (i)  the
“Agreement” shall mean this Agreement not the CTOA; (ii) to rights granted to the Charity shall mean rights granted to CRT; and
(iii)  to  the  “Commencement  Date”  shall  mean  the  Effective  Date).  In  addition,  the  Company  shall  give  as  much  notice  as
practicable to CRT if the XOMA Licence is liable to be, or is summarily terminated, and at CRT’s request use its commercially
reasonable endeavours to facilitate a continuance and an assignment of the XOMA Licence to CRT.

CRT will be responsible for paying directly to XOMA (US) LLC any XOMA Licence Payments incurred after the Effective Date,
in each case in accordance with the terms of the XOMA Licence insofar as such XOMA Licence Payments are triggered by, and
only by, CRT or any of its Sub-Licensee(s) or Affiliates. Each XOMA Licence Payment paid by CRT shall be a Direct Cost. The
Company will remain solely responsible for all XOMA Licence Payments incurred prior to the Effective Date.

MANAGEMENT AND EXPLOITATION

The filing, prosecution, maintenance, enforcement and defence of any Company Intellectual Property and further development and
commercial exploitation thereof shall be at the sole discretion of CRT.

CONFIDENTIALITY

Subject to the other provisions of this Clause 9, each Party undertakes that both during and after termination of this Agreement, it
will keep confidential and not disclose to any person other than to its officers, employees or professional advisors whose province it
is  to  know,  any  confidential  proprietary  information  of  the  other  Party  disclosed  to  or  obtained  by  it  in  connection  with  this
Agreement. For these purposes, Company Know-How shall be deemed to be the confidential information of CRT but only to the
extent  such  Company  Know-How  pertains  solely  or  directly  to  the  Licensed  Product  and  the  Field. Additionally,  subject  to  the
provisions of Clause 9.2, any information of the Charity (and any charitable body succeeding to it) disclosed to or obtained by the
Company in connection with this Agreement shall be deemed to be the confidential information of the Charity.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
9.2

With the exception of Company Know-How which the Company shall keep confidential in accordance with Clause 9.1, Clause 9.1
shall not apply to:

9.2.1

9.2.2

9.2.3

information which is or was already known to the receiving Party at the time of disclosure under this Agreement, as shown
by the receiving Party’s written records, without any obligation to keep it confidential;

information which at the time of being disclosed or obtained by the receiving Party under this Agreement or at any time
thereafter, is published or otherwise generally available to the public other than due to default by the receiving Party of its
obligations hereunder; or

information which is required to be disclosed by a competent Court or regulatory authority or otherwise by applicable law
or statute or any rule or regulation of any Regulatory Authority or other government or administrative agency or authority,
to the extent of such disclosure, provided that the receiving Party shall give notice of such disclosure as soon as reasonably
practicable.

Clause 9.1 above shall not apply to the use or disclosure of any information by any Party for the purpose of exercising or enforcing
its rights under this Agreement.

Each  Party  will  ensure  that  all  personnel  and  third  parties  to  whom  confidential  information  of  another  Party  is  disclosed  are
informed of the provisions of this Clause 9.

So long as this Agreement remains in effect, as between CRT and the Company only, clause 5 of the CTOA shall cease to operate
and this Clause 9 shall replace and supersede the obligations and rights of CRT and the Company only under such clause 5 of the
CTOA.

9.3

9.4

9.5

10

WARRANTIES

10.1

The Company represents and warrants to CRT that to the best of its knowledge and belief:

10.1.1

it is not aware of any inventors of the Company Patent Rights other than the inventors named therein;

10.1.2

it is the legal and beneficial owner of the Company Intellectual Property free of any third party rights or encumbrances;

10.1.3

it has not and will not enter into any Agreement which prevents it fulfilling its obligations under this Agreement;

10.1.4

it has not done anything whereby the whole or any part of the rights assigned or licensed under the Agreement might be
invalidated or registration of them refused;

10.1.5

the manufacture, use and possession of the Investigational Medicinal Product by CRT or any person authorised by CRT
shall not infringe the rights (including without limitation any Intellectual Property Rights) of any third party; and

10.1.6

it  has  not  done  or  omitted  to  do  anything  with  respect  to  the  Investigational  Medicinal  Product  which  may  materially
prejudice the further development of the Investigational Medicinal Product or adversely affect any application which may
be made to any regulatory authority concerned with the approval of medicinal products and their sale.

10.2

Nothing in this Agreement shall be treated as imposing on CRT any liability to the Company in relation to the further development
and commercial exploitation of the Investigational Medicinal Product or the Company Intellectual Property.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
11.

DURATION

11.1

This Agreement shall come into force on the Effective Date and shall extend for so long as CRT has the potential to receive Gross
Revenue and/or Royalties.

12.

DISPUTE RESOLUTION

12.1

12.2

Insofar as this Agreement provides that a matter shall be resolved by Accountancy Opinion or Expert Opinion the opinion of such
expert (who shall act as an expert and not as an arbitrator) shall be final and binding on the Parties. In the event of a Party seeking
an Accountancy  Opinion  or  Expert  Opinion  under  this Agreement,  each  Party  shall  make  written  submissions  to  the  expert  so
appointed and to the other Party within fourteen (14) days of the appointment. Each Party shall have seven (7) days to respond to
the other’s submissions. The expert shall be requested to deliver his Accountancy Opinion or Expert Opinion within a further thirty
(30) days. The costs of any Accountancy Opinion or Expert Opinion shall be borne in such proportions as the expert may determine
in his opinion to be fair and reasonable in all the circumstances or, if no such determination is made in the opinion, by the Parties in
equal proportions.

It  shall  be  a  condition  precedent  to  the  commencement  of  any  action  in  court  or  other  tribunal  (save  an  action  for  an  interim
injunction or an Expert Opinion sought under Clause 12.1) in respect of any dispute relating to this Agreement that the Parties have
sought to resolve the dispute by either Party notifying the other Party in writing for resolution to the Chief Executive Officer (in the
case of CRT) and the Chief Executive Officer (in the case of the Company) (or their express delegates) (the “Senior Executives”)
who shall meet (whether in person or via teleconference) within twenty one (21) days of such notice to seek resolution in good faith.
If the Senior Executives are unable to resolve the dispute at such meeting, either Party may pursue any remedy available to such
Party at law or in equity, subject to the terms and conditions of this Agreement and the other agreements expressly contemplated
hereunder.

13.

GENERAL

13.1

The surviving terms and conditions of the CTOA shall, in accordance with its terms, continue in full force and effect.

13.2

13.3

This Agreement shall be governed by and construed in accordance with English law and each Party agrees to submit to the exclusive
jurisdiction of the English courts (except in respect of disputes under Clause 9 where jurisdiction is non-exclusive).

This Agreement  may  be  executed  in  any  one  or  more  number  of  counterpart  agreements,  as  scanned  email  attachments,  and  all
signatures and counterparts so exchanged shall be considered as original and shall be deemed to form part of and together constitute
this Agreement.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
IN  WITNESS  whereof  this  document  is  executed  by  the  parties  on  the  date  stated  at  the  beginning  of  this Agreement  through  their
authorised signatories

Signed by:

Name:
Title:

Signed by:

Name:

Title:

_____________________________________  

_____________________________________  
_____________________________________  

For and on behalf of
CANCER  RESEARCH  TECHNOLOGY
LIMITED

_____________________________________  

_____________________________________  

 _____________________________________  

For and on behalf of
MONOPAR THERAPEUTICS LLC

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
ANNEX 1A
COMPANY PATENT RIGHTS

[Drafting note – Annex 1A to include those patents identified in schedule 1 of the CTOA and any applications made during the term of the
CTOA relating to the Investigational Medicinal Product and its use (e.g. formulation, manufacturing, etc.)]

PATENT/
APPLICATION NUMBER

TITLE

TERRITORY

FILING
DATE

PATENT/
APPLICATION NUMBER

ANNEX 1B
COMPANY COMBINATION PATENT RIGHTS

TITLE

TERRITORY

FILING
DATE

ANNEX 2
COMPANY KNOW-HOW

ANNEX 3
COMPANY MATERIALS

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Schedule 6
Protocol
(copy of protocol to be inserted here)

 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

Schedule 7
Company Materials
(insert list of materials to be provided by the Company to the Charity)

[***]; purified huATN-658 reference material.

Schedule 7 - Part 2
Company GMP Materials
(insert list of GMP materials to be provided by the Company to the Charity)

[***].
Schedule 8
Back-Up Antibodies

The  [***]  known  as  [***],  each  of  which  is  owned  by  the  Company  but,  as  at  the  Commencement  Date,  are  held  by  XOMA  at  its
premises.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Schedule 9
XOMA Licence
(copy of XOMA Licence to be inserted here)

 
 
 
 
Schedule 10
Progress Reports

 
 
 
 
 
Schedule 11
Clinical Protocol Summary
(To be added to this Agreement within 3 months of signing)

 
 
 
Schedule 12
Escrow Agreement

 
 
 
ESCROW AGREEMENT

THIS AGREEMENT is made the ________ day of ________ 2015 (the “Effective Date”)

AMONG:

CANCER RESEARCH UK  a  company  limited  by  guarantee  registered  under  number  4325234  and  a  charity  registered  under  number
1089464 of Angel Building, 407 St. John Street, London, EC1V 4AD, England (the “Charity”);

CANCER RESEARCH TECHNOLOGY LIMITED a company registered in England and Wales with number 1626049 and registered
office at Angel Building, 407 St. John Street, London, EC1V 4AD, England (“CRT”);

MONOPAR THERAPEUTICS LLC, a limited liability company registered in/incorporated in/ established under the laws of The State of
Delaware,  U.S.A.,  with  registered  office/principal  place  of  business  at  598  Rockefeller  Road,  Lake  Forest,  Illinois,  U.S.A.,  60045  (the
“Company”); and

[NAME], as the escrow agent (the “Escrow Agent”).

WHEREAS:

(A)  The  Charity,  CRT  and  the  Company  have  entered  into  that  certain  CLINICAL  TRIAL  AND  OPTION  AGREEMENT   (the
“CTOA”), a true copy of which (as executed) is attached hereto as Exhibit A , incorporated herein by reference and made a part of this
Agreement;

(B)  The  Charity,  CRT  and  the  Company  further  intend  that  the  Company  shall  hold  in  escrow,  throughout  the  Escrow  Period,  Eight
Hundred  Thousand  Dollars  ($800,000.00  USD)  as  collateral  for  the  liabilities  of  the  Company  under  the  CTOA  (“Escrow
Consideration”);

NOW IT IS HEREBY AGREED as follows:

1. Escrow.

1.1 Escrow Fund.  The  Escrow Agent  shall  immediately  establish  and  open  an  account  to  receive,  invest,  hold  and  disburse  the
funds  that  constitute  (i)  the  Escrow  Consideration  (the  “Escrow Fund”)  and  (ii)  the  Escrow  Earnings  (defined  below).  That  account  is
referred to as the “Escrow Account”.

1.2 Appointment.  CRT,  the  Charity,  and  the  Company  hereto  hereby  appoint,  and  the  Escrow  Agent  hereby  accepts  such
appointment as, and agrees to act throughout the Escrow Period as, the escrow agent to hold, safeguard and disburse the Escrow Fund and
the Escrow Earnings (defined below) pursuant to the terms and conditions hereof.

1.3 Deposit. Within fourteen (14) days of the Effective Date, the Company shall deposit the Escrow Consideration in the Escrow

Account and provide written evidence of the same to CRT and the Charity.

1.4 Investment of the Escrow Consideration.

(a) The Escrow Agent agrees to invest and reinvest funds in the Escrow Account, but only upon written instruction signed
by an authorized agent of the Company, and only in one or more of the following investments (the “Permitted Investments”) from time to
time:  (i)  bank  accounts;  (ii)  bank  money-market  accounts;  (iii)  short-term  certificates  of  deposit;  or  (iv)  short-term  securities  issued  or
guaranteed by the United States government.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

(b)  The  Company,  the  Charity,  and  CRT  recognize  and  agree  that  the  Escrow  Agent  will  not  provide  supervision,
recommendations or advice relating to either the investment of moneys held in the Escrow Account or the purchase, sale, retention or other
disposition of any Permitted Investment. Interest and other earnings on Permitted Investments shall be added to the Escrow Account and
disbursed  in  accordance  with  Sections  4  and  5  hereof.  Without  prejudice  to  Section  2,  any  loss  or  expense  incurred  as  a  result  of  an
investment will be borne by the Escrow Account. In the event that the Escrow Agent does not receive directions to invest funds held in the
Escrow Account, the Escrow Agent shall invest such funds in bank money-market accounts.

(c) The Escrow Agent is hereby authorized to execute purchases and sales of Permitted Investments through the facilities
of its own trading or capital markets operations or those of any affiliated entity. The Escrow Agent shall send statements to the Company
hereto on a monthly basis reflecting activity in the Escrow Account for the preceding month. Although the Company recognizes that it may
obtain a broker confirmation or written statement containing comparable information at no additional cost, the Company hereby agrees that
confirmations of Permitted Investments are not required to be issued by the Escrow Agent for each month in which a monthly statement is
rendered.  No  statement  need  be  rendered  for  the  Escrow  Account  if  no  activity  occurred  for  such  month.  The  Company  shall  send
statements to CRT hereto on a quarterly basis stating the balance of funds in the Escrow Account for the preceding quarter.

(d) The Escrow Agent shall sell or redeem any Permitted Investments as necessary to make any payments or distributions
required  under  this  Agreement.  The  Escrow  Agent  shall  have  no  responsibility  or  liability  for  any  loss  which  may  result  from  any
investment made pursuant to, and in accordance with, this Agreement, or for any loss resulting from the authorized sale of such investment.

(e) Proceeds of the sale of investments will be delivered on the business day on which the appropriate instructions are
received by the Escrow Agent if received prior to the deadline for same day sale of such permitted investments. If such instructions are
received after the applicable deadline, proceeds will be delivered on the next succeeding business day.

(f)  Investments  will  be  made  promptly  following  the  availability  of  such  funds  to  the  Escrow  Agent  taking  into
consideration  the  regulations  and  requirements  (including  investment  cut-off  times)  of  the  Federal  Reserve  wire  system,  any  investment
provider and the Escrow Agent.

applicable.

(g) The Company, the Charity, and CRT shall furnish the Escrow Agent with a completed Form W-8 or Form W-9, as

1.5 Purpose of the Escrow Fund. The Escrow Fund shall be held by the Escrow Agent to provide a source of collateral for the

liabilities of the Company under the CTOA.

1.6 Escrow Period. The “Escrow Period” shall mean the period commencing on the Effective Date and ending on the earlier of:

(i) the date that [***];

reason; or

(ii)  by  mutual  written  agreement  between  the  Company,  CRT,  and  the  Charity  to  terminate  this Agreement  for  any

 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

(iii) five (5) years from the Effective Date of the CTOA;

(the “Claim Expiration Date”); provided that if there are any Claims that are not Resolved at the end of such period, the
Escrow  Period  shall  extend  automatically  beyond  the  Claim  Expiration  Date  and  continue  until  such  time  as  all  Claims  have  been
Resolved.

Period, unless it has been five (5) years since the Effective Date of the CTOA, in which case no notice is required.

The  Company,  CRT,  and  the  Charity  shall  jointly  deliver  to  Escrow Agent  written  notice  upon  the  end  of  the  Escrow

“Resolved” shall mean, in respect of a Claim, that the Claim has been (i) agreed in writing between the Company, the
Charity  and  CRT  as  to  both  liability  and  quantum;  (ii)  finally  determined  (as  to  both  liability  and  quantum)  pursuant  to  Section  5  or,  if
applicable,  by  a  court  of  competent  jurisdiction  from  which  there  is  no  right  of  appeal,  or  from  whose  judgment  the  relevant  Party  is
debarred (by passage of time or otherwise) from making an appeal, including in situations where the Claim relates to a third party claim
brought against the Charity, CRT or a Charity Indemnitee; or (iii) unconditionally withdrawn by the Charity and CRT in writing; and, in
each case, all sums due to the Charity or CRT under this Agreement in respect of such Claim have been paid.

1.7 Instructions. All instructions required under this Agreement will be delivered to Escrow Agent in writing, in either original or
facsimile  form,  executed  by  an  authorized  person  of  each  of  the  Company,  CRT,  and  the  Charity.  Escrow Agent  reserves  the  right  to
telephone an authorized person to confirm the details of such instructions or documents.

1.8 Taxes and Income Distributions.

be treated as owning the funds in the Escrow Fund.

(a) Ownership of Funds in Escrow. For U.S. federal income tax purposes, the parties hereto agree that the Company shall

(b) Treatment  of  Escrow  Fund  Earnings.  The  Company  shall  include  in  its  taxable  income  all  interest,  dividends  and
other income earned on the amounts in the Escrow Fund (the “Escrow Earnings”), and the Escrow Agent shall make distributions to the
Company (“Income Distributions”),  at  the  end  of  each  calendar  quarter  and  upon  the  final  distribution  out  of  the  Escrow  Fund,  [***];
provided that in no circumstance shall Income Distributions result in the Escrow Fund falling below eight hundred thousand US dollars
($800,000 USD).

2. Maintenance of Escrow Fund.

2.1 Minimum.  The  Company  shall  ensure  at  all  times  during  the  Escrow  Period  that  the  Escrow  Fund  is  at  least  equal  to  the
difference between (i) the amount of eight hundred thousand US dollars ($800,000 USD), and (ii) [***] in connection with Claims made
under Section 5.1 (the “Escrow Balance”). The Company shall also ensure at all times during the Escrow Period that the Escrow Balance
is available for payment to the Charity or CRT in connection with Claims allowed under Section 5.

2.2 Additional Deposits. If, for any reason, at any time during the Escrow Period the Escrow Fund is less than the Escrow Balance,
the  Company  shall  immediately  make  any  additional  deposits  in  the  Escrow Account,  and  take  any  other  steps,  needed  to  ensure  that  it
meets its obligations under Section 2.1.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
3. Fees. The Escrow Agent shall be entitled to receive a fee for its services under this agreement. The fee shall be ____________________.
Fees are payable by the Company and shall not be paid out of or deducted from the Escrow Fund.

4. Disbursement.  Promptly  after  the  Escrow  Period,  the  Escrow Agent  shall  deliver  to  the  Company  all  funds  remaining  in  the  Escrow
Fund.

5. Claims Upon the Escrow Fund; Objections to Claims; Resolution of Conflicts.

5.1 Claims Upon Escrow Fund. By written notice to the Escrow Agent and the Company, CRT and the Charity shall have the right
to  make  a  Claim  upon  the  Escrow  Fund  at  any  time  during  the  Escrow  Period  before  5:00  p.m.  Eastern  Standard  Time  on  the  Claim
Expiration Date upon any failure by the Company to fully discharge any of its obligations under, or fully meet its liabilities arising under or
in connection with, the CTOA (each, a “Claim”), including if:

(a)  the  Company  fails  to  fully  discharge  its  obligations  under  Clause  9.2  of  the  CTOA.  Subject  to  Clause  13  of  the
CTOA, CRT or the Charity, but not both, shall have the right to receive from the Escrow Agent an amount out of the Escrow Fund equal to
the amount the Company has failed to cover to fully discharge its obligations under Clause 9.2 of the CTOA. Such right shall include the
right of the Charity or CRT to make Claims on behalf of Charity Indemnitees, and receive from the Escrow Agent an amount out of the
Escrow Fund equal to the amount payable by the Company to Charity Indemnitees, under the CTOA; and

(b)  the  Company  fails  to  pay  amounts  owed  to  the  Charity  under  Clause  12.2.2  of  the  CTOA  upon  termination  of  the
CTOA by CRT or the Charity pursuant to Clause 11.2 or 11.4. Subject to Clause 13 of the CTOA, CRT or the Charity, but not both, shall
have the right to receive from the Escrow Agent an amount out of the Escrow Fund equal to the amount the Company owes the Charity.

The Charity’s and CRT’s rights under this Section 5.1 are subject to Section 5.4.

5.2 Objections to Claims.

(a) At the time of delivery of a written notice of a Claim to the Escrow Agent and the Company by CRT or the Charity,
and for a period of twenty (20) days after such delivery is made to the Company, the Escrow Agent shall make no delivery to CRT, the
Charity, or the Charity Indemnitees of any amount from the Escrow Fund pursuant to Section 5.1 hereof unless the Escrow Agent shall
have  received  written  authorization  from  the  Company  to  make  such  delivery. After  the  expiration  of  such  twenty  (20)  day  period,  the
Escrow Agent shall pay and deliver funds (in US dollars) claimed by the Charity or CRT from the Escrow Fund to an account designated by
the Charity or CRT; provided, however, that no such payment or delivery may be made if the Company shall object in a written statement
to the Claim made in the written notice, and such statement shall have been delivered to the Escrow Agent, the Charity and CRT prior to
the expiration of such twenty (20) day period.

delivers its objection to any Claim.

(b) The Company shall furnish CRT and the Charity with detailed written reason(s) for its objection at the same time as it

by making any objection that has no reasonable prospect of being upheld if referred to arbitration.

(c) The Company shall not unreasonably object to any Claim made to the Escrow Agent by CRT or the Charity, including

 
 
 
 
 
 
 
 
 
 
 
 
 
5.3 Resolution of Conflicts; Arbitration.

(a) In case the Company shall object in writing to any Claim or Claims made in any written notice by CRT or the Charity,
the Company, CRT, and the Charity shall attempt in good faith to agree upon the rights of the respective parties with respect to each of
such Claims. If the Company, CRT, and the Charity should so agree, a memorandum setting forth such agreement shall be prepared and
signed by the parties and shall be furnished to the Escrow Agent. The Escrow Agent shall be entitled to rely on any such memorandum and
distribute funds or withhold payments from the Escrow Fund in accordance with the terms thereof.

(b)  If  no  such  agreement  can  be  reached  within  twenty  (20)  business  days  after  delivery  of  the  Company’s  written
objection  to  CRT  or  the  Charity’s  Claim  in  the  written  notice  notwithstanding  good  faith  negotiation,  any  of  the  Company,  CRT  or  the
Charity may demand arbitration of the matter. The Company, CRT, or the Charity shall, within twenty (20) days of the demand, mutually
select one independent arbitrator with at least five (5) years relevant experience; provided, however, that if the Company, CRT, and the
Charity cannot agree upon one arbitrator during such twenty (20) day period, the Company, on the one hand, and CRT and the Charity, on
the other, shall, within five (5) days following such twenty (20) day period, each select one arbitrator and the two arbitrators so selected
shall  select  a  third  arbitrator,  each  of  which  arbitrators  shall  be  independent  and  have  at  least  five  (5)  years  relevant  experience.  The
arbitrator(s) shall set a limited time period and establish procedures designed to reduce the cost and time for discovery to the extent possible
while  allowing  the  parties  an  opportunity,  adequate  in  the  sole  judgment  of  the  arbitrators,  to  discover  relevant  information  from  the
opposing parties about the subject matter of the dispute. The arbitrator(s) shall rule upon motions to compel or limit discovery and shall
have  the  authority  to  impose  sanctions,  including  attorneys’  fees  and  costs,  should  the  arbitrator(s)  determine  that  discovery  was  sought
without substantial justification or that discovery was refused or objected to without substantial justification. The decision of the arbitrator
(or, in the case of three arbitrators, a majority of the three arbitrators) as to the validity and amount of any Claim in such written notice shall
be binding and conclusive upon the parties to this Agreement, and notwithstanding anything in Section 5.2 hereof, the Escrow Agent shall
act in accordance with such decision and make or withhold payments out of the Escrow Fund in accordance therewith. Such decision shall
be written and shall be supported by written findings of fact and conclusions which shall set forth the award, judgment, decree or order
awarded  by  the  arbitrator(s).  The  arbitrator(s)  shall  also  have  the  authority  to  award  additional  sums  to  the  Charity  and  CRT,  and
reimbursement  of  attorneys’  fees  and  costs,  should  the  arbitrator(s)  determine  that  the  objection  had  no  reasonable  prospect  of  being
upheld.

(c)  Judgement  upon  any  award  rendered  by  the  arbitrators  may  be  entered  in  any  court  having  jurisdiction. Any  such
arbitration shall be held in London, England, under the International Arbitration Rules of the International Centre for Dispute Resolution
then in effect.

(d) Each party shall bear its own fees and costs in connection with the arbitration. The fees, costs and expenses of the
arbitrator(s), if any, shall be apportioned between the Company, on the one hand, and CRT and the Charity, on the other, based upon the
inverse proportion of the amount of disputed items resolved in favor of such party (i.e., so that the prevailing party bears a lesser amount of
such fees and expenses).

5.4 Limit. The maximum aggregate amount that the Charity and CRT may claim, and that is payable to them, from the Escrow
Account to satisfy any and all Claims made under this Agreement shall be eight hundred thousand US dollars ($800,000 USD). The rights
granted  under  this Agreement  are  in  addition  to,  and  not  instead  of,  any  rights  of  the  Charity  and  CRT  under  or  in  connection  with  the
CTOA, whether under contract, statute or tort. Nothing in this Agreement shall, or is intended to, limit such rights, including where sums
paid under this Agreement do not fully discharge the Company’s liabilities.

 
 
 
 
 
 
 
 
 
6. Limitation on Escrow Agent’s Liability. The Escrow Agent’s responsibilities and liabilities shall be limited as follows:

6.1 The Escrow Agent shall not be responsible for or be required to enforce any of the terms or conditions of the CTOA or any
other  agreement  between  the  parties  thereto.  The  Escrow  Agent  shall  not  be  responsible  or  liable  in  any  manner  whatsoever  for  the
performance by the Company, CRT, or the Charity of their respective obligations under the CTOA or this Agreement, nor shall the Escrow
Agent be responsible or liable in any manner whatsoever for the failure of any party to the CTOA to honor any of the provisions of the
CTOA.

6.2  The  duties  and  obligations  of  the  Escrow Agent  shall  be  limited  to  and  determined  solely  by  the  express  provisions  of  this
Agreement and the CTOA, and no implied duties or obligations shall be read into this Agreement against the Escrow Agent. The Escrow
Agent shall neither be responsible for, nor chargeable with, knowledge of the terms and conditions of any other agreement, instrument or
document  other  than  this  Escrow Agreement  or  the  CTOA,  whether  or  not  a  copy  and/or  original  of  such  agreement  is  held  by  Escrow
Agent; and, the Escrow Agent shall have no duty to know or inquire as to the performance or nonperformance of any provision of any such
agreement, instrument or document. This Escrow Agreement sets forth all matters pertinent to the escrow contemplated hereunder, and no
additional obligations of the Escrow Agent shall be inferred from the terms of this Escrow Agreement or any other agreement, instrument
or document. All references in this Escrow Agreement to any other agreement (other than the CTOA) are for the convenience of the parties
other than the Escrow Agent, and the Escrow Agent has no duties or obligations with respect thereto.

6.3  The  Escrow Agent  shall  be  entitled  to  rely  upon  and  shall  be  protected  in  acting  in  reliance  upon  any  instruction,  notice,
information, certificate, instrument or other document which is submitted to it in connection with its duties under, and in accordance with,
this Agreement and which the Escrow Agent in good faith believes to have been signed or presented by the proper party or parties. The
Escrow Agent shall have no liability with respect to the form, execution, validity or authenticity thereof.

6.4 The Escrow Agent shall be entitled to consult, at its own cost, with independent counsel of its own selection and the opinion of
such counsel shall be full and complete authorization and protection to the Escrow Agent in respect of any action taken or omitted by the
Escrow Agent hereunder in good faith and in accordance with the opinion of such counsel, unless caused by or arising from its own fraud,
gross negligence or willful misconduct.

6.5 The Escrow Agent shall have no responsibility or liability for any diminution in value of any assets held under this agreement
which may result from any investments or reinvestments made in accordance with any provision which may be contained in this agreement.

6.6 The Escrow Agent shall not be liable for any action taken or omitted under this Agreement while acting in good faith, unless

caused by or arising from its own fraud, negligence or misconduct.

6.7 The Escrow Agent shall have the right to perform any of its duties hereunder through custodians or nominees, and shall be

liable for all acts and omissions of such custodians or nominees as if they were acts or omissions of the Escrow Agent.

 
 
 
 
 
 
 
 
 
 
6.8 Any banking association or corporation into which the Escrow Agent may be merged, converted or with which the Escrow
Agent may be consolidated, or any corporation resulting from any merger, conversion or consolidation to which the Escrow Agent shall be
a party, or any banking association or corporation to which all or substantially all of the corporate trust business of the Escrow Agent shall
be transferred, shall succeed to all of the Escrow Agent’s rights, obligations and immunities hereunder without the execution or filing of
any paper or any further act on the part of any of the parties hereto, anything herein to the contrary notwithstanding.

6.9 The Escrow Agent shall have the right at any time to resign for any reason and be discharged of its duties as Escrow Agent
hereunder by giving written notice of its resignation to the parties hereto at least thirty (30) calendar days prior to the date specified for such
resignation to take effect. In addition, the Company, the Charity and CRT may remove the Escrow Agent as escrow agent at any time with
or without cause, by an instrument given to the Escrow Agent, which instrument shall be signed by each of the Company, the Charity and
CRT  and  shall  designate  the  effective  date  of  such  removal.  In  the  event  of  any  such  resignation  or  removal,  a  successor  escrow  agent
which, unless the Company, CRT, and the Charity otherwise agree in writing, shall be a bank or trust company organized under the laws of
the United States of America or of the State of Illinois shall be appointed by Company with the approval of CRT and the Charity, which
approval shall not be unreasonably delayed, conditioned, or withheld. Any such successor escrow agent shall deliver to Company, CRT and
the Charity a written instrument accepting such appointment, and thereupon it shall succeed to all the rights and duties of the Escrow Agent
hereunder and shall be entitled to receive the Escrow Fund. All responsibilities of the Escrow Agent hereunder shall cease and terminate on
the effective date of its resignation or removal and its sole responsibility thereafter shall be to hold the Escrow Fund for a period of thirty
(30) calendar days following the effective date of resignation or removal, at which time:

(1)  if  a  successor  Escrow  Agent  shall  have  been  appointed  and  written  notice  thereof  shall  have  been  given  to  the
resigning or removed Escrow Agent by parties hereto and the successor Escrow Agent, then the resigning Escrow Agent shall deliver the
remaining Escrow Fund to the successor Escrow Agent; or

(2)  if  a  successor  Escrow Agent  shall  not  have  been  appointed,  for  any  reason  whatsoever,  the  resigning  or  removed
Escrow Agent shall deliver the Escrow Fund to a court of competent jurisdiction in the County of New York, New York and give written
notice of the same to Company, CRT, and the Charity.

6.10 In the event that the Escrow Agent shall  be  uncertain  as  to  its  duties  or  rights  hereunder  or  shall  receive  instructions  with
respect to the Escrow Fund, which, in its sole discretion, are in conflict either with other instructions received by it or with any provision of
this Agreement, the Escrow Agent shall have the absolute right to suspend all further performance under this Agreement (except for the
safekeeping and investment of the Escrow Fund) until such uncertainty or conflicting instructions have been resolved by alternative dispute
resolution, to the Escrow Agent’s sole satisfaction, pursuant to Section 7 hereof or by final judgment of a court of competent jurisdiction,
joint written instructions executed by all parties hereto, or otherwise. In the event that any controversy arises between one or more of the
parties  hereto  or  any  other  party  with  respect  to  this Agreement  and/or  the  Escrow  Fund,  the  Escrow Agent  shall  not  be  required  to
determine the proper resolution of such controversy or the proper disposition of the Escrow Fund.  In such event, and without the consent
or approval of any other party, (i) the Escrow Agent shall have the absolute right, in its sole discretion, to deposit; and (ii) the Company
shall have the absolute right, in its sole discretion, to require the Escrow Agent to deposit, the cash remaining in the Escrow Fund with the
clerk of a court of competent jurisdiction specified in Section 6 hereof, file a suit in interpleader in that court and obtain an order from that
court requiring all parties involved to resolve their respective claims to the Escrow Fund pursuant to Section 6. Upon the deposit by the
Escrow Agent of the Escrow Fund with the clerk of that court in accordance with this provision, the Escrow Agent shall be relieved of all
further obligations, and the Company shall have no obligation to restore the Escrow Balance under Section 2.

 
 
 
 
 
 
 
6.11 The Company shall indemnify and hold the Escrow Agent harmless from and against all liabilities, causes of action, claims,
demands, judgments, damages, reasonable costs and expenses that may arise out of or in connection with the Escrow Agent’s good faith
acceptance of and performance of its duties and obligations under this Agreement, except to the extent related to acts or omissions of the
Escrow  Agent  in  bad  faith  constituting  fraud,  gross  negligence  or  willful  misconduct  or  otherwise  in  breach  of  this  Agreement.  The
provisions of this Section 6.11 shall survive the resignation or removal of the Escrow Agent and the termination of this Agreement.

7. Dispute Resolution/Governing Law.

7.1  This Agreement  shall  be  governed  by  and  construed  in  accordance  with  the  laws  of  the  State  of  New  York  without  giving

effect to the principles of conflicts of laws (other than Section 5-1401 of the New York General Obligations Law).

7.2  Subject  to  Section  5.3(c),  the  parties  hereto  intend  that  all  disputes  between  the  parties  arising  out  of  or  related  to  this

Agreement shall be settled by the parties amicably through good-faith discussions upon the written request of any party.

7.3 In the event that any such dispute cannot be resolved thereby within a period of twenty (20) days after such notice has been
given, such dispute shall be resolved by binding arbitration, which shall take place in the County of New York, New York, administered by
and in accordance with the then-existing International Arbitration Rules of the International Centre for Dispute Resolution.

7.4 An award rendered in connection with an arbitration pursuant to this Section 7 shall be final and binding upon the parties, and
the parties agree and consent that the arbitral award shall be conclusive proof of the validity of the determinations of the arbitrations set
forth in the award, and judgment upon any award rendered by the arbitrators may be entered by any state or federal court having jurisdiction
thereof.

7.5 This Section 7 is subject to the terms of Section 10 hereof.

8. Notices. All notices and other communications given or made pursuant hereto shall be in writing and shall be deemed to have been duly
given  or  made  as  of  the  date  delivered,  mailed  or  transmitted,  and  shall  be  effective  upon  receipt,  if  delivered  personally,  mailed  by
registered  or  certified  mail  (postage  prepaid,  return  receipt  requested)  or  sent  by  fax  (with  immediate  confirmation)  or  internationally
recognized overnight courier service, as follows:

If to the Company, to:

Monopar Therapeutics LLC

598 Rockefeller Road

Lake Forest, IL USA 60045

Contact: Chief Executive Officer

If to the Charity or CRT, to:

Angel Building

407 St. John Street

London EC1V 4AD

United Kingdom

Contact: Chief Executive Officer and Director of Centre for Drug Development

Fax: +44 (0) 20 3014 8633

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
If to the Escrow Agent, to:

[]

[]

[]

Attn:

Fax:

9. Interpretation and Construction of Agreement.

9.1  Unless  the  context  shall  otherwise  require,  any  pronoun  herein  shall  include  the  corresponding  masculine,  feminine,  and
neuter  forms,  and  words  using  the  singular  or  plural  number  shall  also  include  the  plural  or  singular  number,  respectively.  The  words
“include,” “includes” and “including” herein shall be deemed to be followed by the phrase “without limitation” and the word “or” shall
include the meaning “either or both.” All references herein to sections, exhibits, and schedules shall be deemed to be references to sections
of,  and  exhibits  and  schedules  to,  this Agreement  unless  the  context  shall  otherwise  require.  The  headings  of  the  sections  herein  are
inserted for convenience of reference only and are not intended to be a part of or to affect the meaning or interpretation of this Agreement.
Unless  the  context  shall  otherwise  require,  any  reference  herein  to  any  agreement,  other  instrument,  statute  or  regulation  is  to  such
agreement, instrument, statute or regulation as amended and supplemented from time to time (and, in the case of a statute or regulation, to
any successor provision).

9.2 The Company, CRT, and the Charity acknowledge that each has participated in the drafting of this Agreement and that any
rule of construction to the effect that ambiguities are to be resolved against the drafting party shall not be applied in the construction or
interpretation of this Agreement.

9.3 Any reference herein to a “day” or a number of “days” (without the explicit qualification of “business”) shall be interpreted as
a reference to a calendar day or number of calendar days. If any action or notice is to be taken or given on or by a particular calendar day,
and  such  calendar  day  is  not  a  business  day,  then  such  action  or  notice  shall  be  deferred  until,  or  may  be  taken  or  given  on,  the  next
business day.

10. Specific Performance. Each party agrees that irreparable harm, for which there may be no adequate remedy at law and for which the
ascertainment  of  damages  would  be  difficult,  would  occur  in  the  event  any  of  the  provisions  of  this Agreement  were  not  performed  in
accordance  with  its  specific  terms  or  were  otherwise  breached.  Each  party  accordingly  agrees  that  the  other  parties  shall  be  entitled  to
specifically enforce this Agreement and to obtain an injunction or injunctions to prevent breaches of the provisions of this Agreement and to
enforce specifically the terms and provisions hereof or thereof, in each instance without being required to post bond or other security and in
addition to, and without having to prove the adequacy of, other remedies at law.

11. Counterpart  Signatures,  Electronic  Communication  Delivery.  This  Agreement  may  be  executed  in  one  or  more  counterparts  and
delivered by electronic communication, all of which shall be considered one and the same agreement, and shall become effective when one
or more counterparts have been signed by each of the parties and delivered to the other parties, it being understood that all parties need not
sign the same counterpart.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
12. Entire Agreement.  This Agreement  and  the  documents,  instruments  and  other  agreements  specifically  referred  to  herein  or  delivered
pursuant hereto (a) constitute the entire agreement among the parties with respect to the subject matter hereof and (b) supersede all prior
agreements and understandings, both written and oral, among the parties with respect to the subject matter hereof.

13. Amendment; Waiver; Requirement of Writing. This Agreement may be amended, modified, superseded, rescinded, or canceled only by
a written instrument executed by the Company, CRT, the Charity, and the Escrow Agent. Any term or condition of this Agreement may be
waived at any time by the party hereto entitled to the benefit thereof, and any such term or condition may be modified at any time by an
agreement in writing executed by each of the parties hereto entitled to the benefit thereof. No delay or failure on the part of any party in
exercising  any  rights  hereunder,  and  no  partial  or  single  exercise  thereof,  will  constitute  a  waiver  of  such  rights  or  of  any  other  rights
hereunder.

14. Expenses.  Each  of  the  parties  hereto  shall  bear,  without  right  of  reimbursement  from  any  other  party,  all  the  costs  incurred  by  it
incident to the preparation, execution, and delivery of this Agreement or the performance of its obligations hereunder, whether or not the
transactions contemplated by this Agreement shall be consummated.

15. No Third-Party Beneficiaries. Nothing in this Agreement will be construed as giving any person, other than the parties, their successors
and permitted assigns, any right, remedy, or claim under or in respect of this Agreement or any provision hereof; it being acknowledged
that (i) this Section 15 is without prejudice to the rights of the Charity Indemnitees under the CTOA; (ii) the Charity and CRT may make
Claims under this Agreement on behalf of the Charity Indemnitees in respect of Claims made by the Charity Indemnitees under the CTOA;
and (iii) the Escrow Agent may make payments to the Charity and/or CRT on behalf of such Charity Indemnitees in respect of such Claims,
but only after the Escrow Agent has received written confirmation from such Charity Indemnitees of the authority of the Charity and/or
CRT to receive such payments on behalf of such Charity Indemnitees..

16. Disclaimer of Agency . Except for any provisions herein expressly authorizing one party to act for  another,  this Agreement  shall  not
constitute any party as a legal representative or agent of any other party, nor shall a party have the right or authority to assume, create, or
incur any liability of any kind, expressed or implied, against or in the name or on behalf of any other party or any of such other party’s
affiliates.

17. Relationship of the Parties .  Nothing  contained  in  this Agreement  is  intended  to,  or  shall  be  deemed  to,  create  a  partnership  or  joint
venture relationship among the parties hereto or any of their affiliates for any purpose, including tax purposes.

18. Assignment. This Agreement and the rights and obligations of each party hereunder or thereunder shall be binding upon, and inure to
the  benefit  of,  the  parties  hereto  and  their  respective  successors  and  permitted  assigns.  None  of  the  Company,  CRT  or  the  Charity  shall
assign  this Agreement  without  the  prior  written  consent  of  each  other,  which  consent  may  not  be  unreasonably  conditioned,  delayed,  or
withheld. Assignment by Escrow Agent shall be governed by Section 6 hereof.

19. Severability.  In  the  event  that  any  provision  of  this  Agreement,  or  the  application  thereof,  becomes  or  is  declared  by  a  court  of
competent jurisdiction to be illegal, void or unenforceable, the remainder of this Agreement will continue in full force and effect, and the
application of such provision to other persons or circumstances will be interpreted so as reasonably to effect the intent of the parties hereto.
The parties further agree to replace such void or unenforceable provision of this Agreement with a valid and enforceable provision that will
achieve, to the extent possible, the economic, business and other purposes of such void or unenforceable provision.

 
 
 
 
 
 
 
 
 
 
20. Several Liability. The obligations and liabilities of each party under this Agreement are several, not joint.

[Signatures on following page]

 
 
 
 
 
 
 
 
IN WITNESS whereof this Agreement has been executed by duly authorised officers of the parties on the day first above written.

Signed
by:                                 

_____________________________________

Name:                                 _____________________________________

Title:                                  _____________________________________

For and on behalf of

CANCER RESEARCH TECHNOLOGY LIMITED

Signed
by:                                 

_____________________________________

Name:                                 _____________________________________

Title:                                  _____________________________________

For and on behalf of

CANCER RESEARCH UK

Signed
by:                                 

_____________________________________

Name:                                 _____________________________________

Title:                                  _____________________________________

For and on behalf of

MONOPAR THERAPEUTICS LLC

Signed
by:                                 

_____________________________________

Name:                                 _____________________________________

Title:                                  _____________________________________

For and on behalf of

[ESCROW AGENT]

Signature Page to Escrow Agreement

Exhibit A

Clinical Trial and Option Agreement

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Schedule 13

Technical Agreement (Standard Form)

 
 
 
 
 TECHNICAL AGREEMENT

between

Cancer Research UK

and

MONOPAR THERAPEUTICS LLC

The Cancer Research UK Centre for Drug Development is the Sponsor of clinical trials where the investigational medicinal product
(IMP, including the master cell bank and bulk drug substance where applicable) is manufactured, and/or analysed, and/or labelled, and/or
stored, and/or shipped by Cancer Research UK The Sponsor has obligations with respect to all aspects of the management of the IMP in
the clinical trial.This document is a technical agreement that meets the requirements of European Good Manufacturing Practice (GMP)
legislation 2003/94/EC. This document should also be interpreted with respect to the European Clinical Trials legislation 2001/20/EC and
Eudralex Volume 4, Annex 13, paragraph 36 and 37 regarding reference and retention samples.

The technical agreement takes the form of a detailed check list of all the activities associated with manufacturing, packaging, storage and
distribution of the huATN-658 master cell bank  It defines the individual responsibilities of  Monopar Therapeutics and of Cancer
Research UK and in particular defines who is responsible for the GMP aspects of the activities listed. Responsibility for each activity is
assigned to either party in the appropriate tick box. If any element of the check list does not apply, it should be clearly crossed through
not left blank. More detail may be added as necessary to clarify particular points to ensure that only one party is responsible for each
point.

Technical Agreement Signatures

Contract Giver

Company
Name

Cancer Research UK Biotherapeutics Development Unit

Address

Clare Hall

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Position
Name
Authorised
signatory
Date

Company
Name
Address

Position
Name
Authorised
signatory
Date

Company
Name
Address

Position
Name
Authorised
signatory
Date

Authorised
signatory
Date

Purpose

Potters Bar
Hertfordshire
EN6 3LD
Qualified Person
Dr Robert Scott

Cancer Research UK Centre of Drug Development (Contract Giver)

Angel Building
407 St John Street
London EC1V 4AD

Drug Supply Manager
Dr Nigel Westwood

CONTRACT ACCEPTOR

MONOPAR THERAPEUTICS LLC

598 Rockefeller Road
Lake Forest, Illinois
U.S.A., 60045

This Technical Agreement assigns the responsibilities of Monopar Therapeutics and Cancer Research UK with respect to
the huATN-658 master cell bankNote: Monopar Therapeutics has outsourced the manufacture and storage of the master
cell bank. Therefore, some aspects of these activities may be delegated by Monopar Therapeutics to third parties. However,
Monopar Therapeutics remains responsible for oversight of those functions as outlined in the Technical Agreement.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

BDU
CA
CG
GMP
EU

EU GMP

IMP
MCB
QP
Retention
sample

Reference
sample

Definitions and Acronyms

Biotherapeutics Development Unit
Contract Acceptor
Contract Giver
Good Manufacturing Practice
European Union
European Union current Good Manufacturing Practice as defined in directive
2003/94/EC
Investigational Medicinal Product = drug product (unless otherwise stated IMP means
manufactured to EU cGMP or its equivalent)
[***]
Qualified Person
A sample of a packaged unit from a batch of finished
product for each packaging run/trial period. It is stored for
identification purposes
A sample of a batch in its primary packaging or finished
product container which is stored for the purpose of being analysed
should the need arise

1.00

1.01

1.02

1.03

1.04

1.05

1.06

1.07

Strikethrough text where responsibility is not applicable to either party

RESPONSIBILITIESMaster Cell Bank (MCB)

Monopar (CA)

Cancer Research
UK (CG)

Supply to the CG copies of audit reports plus associated corrective/preventative actions
and close out documentation for the CA's GMP contract manufacturer used to
manufacture and store the MCB
Supply to the CG a statement from QA confirming what GMP standard the MCB was
produced in compliance with including reference to EU GMP if appropriate
Supply to the CG a Certificates of Analysis for the MCB approved, signed and dated
by QA
CA confirms that ≥200 of sealed vials have been stored at -140°C (LN) that form the
QA approved MCB CG provides documentation to confirm that the vials have been
stored in an area dedicated to GMP appropriately documented and secure and
completely separate from any non tested cell banks
Supply copies of completed QA reviewed batch manufacturing records used in the
manufacture of the MCB
Supply copies to the CG of all deviations recorded during the manufacture and storage
of the MCB and any associated corrective/preventative actions taken and
documentation closing out the deviation
Supply copies to CG of storage records for the MCB demonstrating that the MCB has
been stored correctly at all times since it was frozen

X

X

X

X

X

X

X

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted information, pursuant to an Order dated January 8, 2018.

1.08

1.09

1.10

1.11

1.12

1.13

1.14

1.15

Supply copies to the CG of all out of specifications reported either during the
manufacture, testing or storage of the MCB and related corrective/preventative and/or
close out documentation
Supply to the CG a material Safety Data Sheet (if applicable) to the CG including
biological safety classification of the [***]
Shipment of packaged, MCB to sponsor's licenced facility as notified by the CG with
temperature monitoring of the MCB using a suitably qualified shipper
Supply to the CG data to confirm that the MCB is both mycoplasma free and sterile
when tested using validated pharmacopoieal methods
Supply to the CG data on the stability and recovery of the MCB. Trended stability data
generated from the MCB shall be supplied to the CG if available
Confirm receipt of the MCB on delivery to the CG and notify the CA immediately of
any breakages, packaging issues, temperature alarms or documentation discrepancies
CG confirms that ≥100 of sealed vials received will be stored at -140°C (LN) which
form the QA approved CA supplied MCB CG will store the vials in an area dedicated
to GMP, which is appropriately documented and secure and completely separate from
any non tested cell banks
CA will notify the CG of any Competent Authority inspection findings directly related
to the MCB when stored at the CA's contractor

X

X

X

X

X

X

X

X

Distribution List
Cancer Research UK Formulation Unit

Name/Title/Duties

Dr Robert Scott - QA/QC Manager Cancer Research UK Biotherapeutics Development Unit, Responsible for quality assurance at the
BDU and quality control of biologicals QP certification and release of IMP
Dr Heike Lentfer - Head of BDU. Responsible for delivering the development and manufacture of biological IMPs
Dr Nigel Westwood - Drug Supply ManagerAccountable for ensuring API and IMP are available for the clinical trials Sponsored by
Cancer Research UK

Please add names here

Monopar Therapeutics

Name/Title/Duties

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

AMENDED AND RESTATED LICENSE AGREEMENT

THIS AMENDED AND RESTATED LICENSE AGREEMENT (this “Agreement”), effective as of September 24, 2014 (the

“Effective Date”), is entered into between Tactic Pharma, LLC, a limited liability company (“TACTIC”), having offices at 1062 Princeton
Avenue, Highland Park, IL 60035 and XOMA (US) LLC, a Delaware limited liability company (“XOMA”), having offices at 2910
Seventh Street, Berkeley, California 94710. Each of XOMA and TACTIC are sometimes referred to herein separately as a “Party” and
together as “Parties.”

WHEREAS TACTIC was formed upon the dissolution of Attenuon, LLC, San Diego, California, 92121 (“ATTENUON”), such

that TACTIC can be considered a successor of ATTENUON;

WHEREAS TACTIC is the successor and rightful owner of certain IP rights developed by ATTENUON, including, but not limited

to, ATN-658;

WHEREAS ATTENUON and XOMA had entered into a certain HUMAN ENGINEERING™ LICENSE AGREEMENT,
effective September 29, 2006, (the “Prior Agreement”) in which, among other things, Attenuon, LLC obtained a license to certain HUMAN
ENGINEERING PATENT RIGHTS as described in the Prior Agreement for the purposes of developing and commercializing human
engineered ATN-658;

WHEREAS for the good and valuable consideration set forth in this agreement, the Parties agree that all rights, claims, and
obligations under the Prior Agreement between Attenuon, LLC, its successors, and XOMA are now null and void unless expressly restated
herein. Accordingly, the Parties agree that there are no outstanding payments, liabilities, or other obligations owed by TACTIC to XOMA
under the Prior Agreement.

For good and valuable consideration, the receipt and sufficiency of which are hereby acknowledged, the Parties agree as follows:

ARTICLE 1

DEFINITIONS

For purposes of this Agreement, the terms defined in this Article 1 shall have the respective meanings set forth below:

1.1 “Affiliate” shall mean, with respect to any Person, any other Person which, presently or in the future, directly or indirectly

controls, is controlled by, or is under common control with, such Person.

1.2 “Antibody” shall mean any immunoglobulin molecule (such as IgG), whether in monospecific or any other form, and shall

include, without limitation, any immunoglobulin fragment (such as Fv, Fab, F(ab') or F(ab')2), any fusion protein of an immunoglobulin or
immunoglobulin fragment and any single chain antibody (such as scFv), as well as any derivative of any of the foregoing.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

1.3 “TACTIC Antibody” shall mean the non-human Antibody directed to the TACTIC Target, referred to by TACTIC as “ATN-

658”

1.4  “TACTIC Patent Rights” shall have the meaning set forth in Section 1.6.

1.5 “TACTIC Program Inventions” shall have the meaning set forth in Section 1.6.

1.6  “TACTIC Program Inventions and Patent Rights” shall mean any and all (a) Program Inventions, whether or not patentable,

that (i) comprise or embody (A) [***], (B) [***], (C) [***], (D) [***], (E) [***] and (F) any uses of any and all of the foregoing, or (ii) do
not meet the definition of [***] by virtue of the preceding clause (i) or the definition of [***] by virtue of clause (i) thereof and were [***]
(collectively, the “TACTIC Program Inventions”); and (b) Patent Rights arising out of the conduct of activities under the Prior Agreement
that claim or cover such TACTIC Program Inventions (the “TACTIC Patent Rights”). Notwithstanding the foregoing, TACTIC Program
Inventions and Patent Rights do not include any [***] and Patent Rights; provided that the foregoing shall not apply to [***] (I) [***] (II)
[***] (III) [***] (IV) [***] (V) [***] and (VI) any uses of any and all of the foregoing, each of which shall be included in the [***] and
[***].

1.7 “TACTIC Target” shall mean the target antigen known as urokinase-type plasminogen activator receptor (uPAR).

1.8 “Combination Product” shall have the meaning set forth in Section 1.22.

1.9 “Composition of Matter” shall mean any composition of matter or article of manufacture.

1.10 “Confidential Information” shall mean any proprietary or confidential information or material disclosed by a Party to the

other Party pursuant to the Prior Agreement or this Agreement which is (a) disclosed in tangible form and is designated thereon as
“Confidential” at the time it is delivered to the receiving Party, or (b) disclosed orally and identified as confidential or proprietary when
disclosed and such disclosure of confidential information is confirmed in writing within thirty (30) days by the disclosing Party.
Notwithstanding the foregoing, Confidential Information shall not include information which the receiving Party can establish by written
documentation (i) to have been publicly known prior to disclosure of such information by the disclosing Party to the receiving Party, (ii) to
have become publicly known, without fault on the part of the receiving Party, subsequent to disclosure of such information by the
disclosing Party to the receiving Party, (iii) to have been received by the receiving Party at any time from a source, other than the
disclosing Party, rightfully having possession of and the right to disclose such information, other than under an obligation of

 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

confidentiality, (iv) to have been otherwise rightfully known by the receiving Party prior to disclosure of such information by the
disclosing Party to the receiving Party, other than under an obligation of confidentiality, or (v) to have been independently developed by
employees or agents of the receiving Party without access to or use of such information disclosed by the disclosing Party to the receiving
Party without violating any obligation of confidentiality or non-use.

1.11 “Control,” “Controls” and “Controlled” shall mean, with respect to a particular item of information or Intellectual Property

Right, that the applicable Party or any of its Affiliates owns (whether solely or jointly with the other Party or any Third Party), or has a
license to, such item or right and has the ability to grant to the other Party access to, and a license or sublicense (as applicable) under, such
item or right as provided for herein without violating the terms of any agreement with any Third Party.

1.12  “CPR” shall have the meaning set forth in Section 9.2.

1.13 “Dispute” shall have the meaning set forth in Section 9.1.

1.14 “Human Engineer™,” “Human Engineered™” and “Human Engineering™” shall mean, for purposes of this Agreement, with

respect to a particular Antibody, resulting from, or otherwise practicing, the methods of the Human Engineering™ Patent Rights or any
other proprietary protein engineering methods used by XOMA for modifying non-human Antibodies with the intended purpose of making
them suitable for medical purposes in humans.

1.15 “Human Engineered™ TACTIC Antibodies” shall mean the Human Engineered™ versions of the TACTIC Antibodies

provided by XOMA under the Prior Agreement.

1.16 “Human Engineering™ Patent Rights” shall mean the Patent Rights listed on Schedule 1.16 hereto and all patents issuing on

any of the applications so listed, including extensions, reissues and re-examinations.

1.17 “Indemnitee” shall have the meaning set forth in Section 8.2.

1.18 “Indemnitor” shall have the meaning set forth in Section 8.2.

1.19 “Intellectual Property Rights” shall mean Patent Rights, copyrights, trademarks, service marks, know-how, trade secrets, and

applications and registrations for the foregoing, in any country, supranational organization or territory of the world.

1.20  "Joint Program Inventions" shall mean any and all Program Inventions, whether or not patentable, that are invented jointly by

employees, agents, consultants or contractors of both [***], but [***].

1.21 "Major Market Country" shall mean any of the United States of America, Japan or any of the top five (5) countries (measured

by pharmaceutical sales for the most recently com​ pleted calendar year for which such information is available at the time of
determination) of the European Union.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

1.22  “Milestone Payment” shall have the meaning set forth in Section 3.1.

1.23 “Net Sales” shall mean the gross amount invoiced by TACTIC, its Affiliates, assignees or sublicensees for sales of Products to

Third Parties, less the following items, as allocable to such Products:

(a) trade discounts, rebates or allowances actually allowed and taken directly with respect to such sales;

(b) credits or allowances additionally granted upon returns, rejections, recalls or retroactive price reductions;

(c) freight, shipping and insurance charges;

(d) [***];

(e) taxes, duties or other governmental tariffs (other than income taxes); and

(f) government mandated rebates.

In the event that a Product is sold as part of a Combination Product (as defined below) in any country, the Net Sales of the Product as part
of a Combination Product in that country for the purposes of determining royalty payments shall be determined by multiplying the Net
Sales of the Combination Product in that country by the fraction (A/A+B) where A is the average sale price in the relevant quarterly
period of the Product in that country when sold separately in finished form and B is the average sale price in the relevant quarterly period
of the Other Element (as defined below) in that country sold separately in finished form. In the event that the average sale price of the
Product in that country can be determined but the average sale price of the Other Element in that country cannot be determined, Net Sales
of the Product in that country for the purposes of determining royalty payments shall be calculated by multiplying the Net Sales of the
Combination Product in that country by the fraction (C/D) where C is the selling Party's average sales price in the relevant quarterly
period of the Product and D is the average selling price in the relevant quarterly period of the Combination Product in that country. If the
average sale price of the Other Element in that quarterly period can be determined but the average price of the Product in that country
cannot be determined, Net Sales of the Combination Product in that country for the purposes of determining royalty payments shall be
calculated by multiplying the Net Sales of the Combination Product in that country by the following formula: one (1) minus E/D where E
is the average selling price in the relevant quarterly period of the Other Element in that country and D is the average selling price of the
Combination Product in that country in the relevant quarterly period. If the average sale price of both the Product and the Other Element
cannot be deter​ mined, the Net Sales of the Product shall be reasonably agreed upon by the Parties. As used herein, the term
"Combination Product" shall mean a product which contains or comprises a Product as an active component and at least one other active
compound (an "Other Element").

Provision of Products free of charge for clinical trials, for promotional or sampling purposes or as donations (for example to non-profit
institutions or government agencies for a non-commercial purpose) at levels not in excess of industry norms, shall not be considered in
determining Net Sales.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

1.24 “Patent Prosecution” shall mean, with respect to particular Patent Rights, (a) preparing, filing and prosecuting patent
applications (including, but not limited to, provisional, non-provisional, reissue, reexamination, continuing, continuation, continuation-in-
part, divisional, and substitute applications and any foreign counterparts thereof) of such Patent Rights; (b) maintaining such Patent Rights;
and (c) managing or conducting any interference or opposition or similar proceedings relating to the foregoing.

1.25 “Patent Rights” shall mean any of the following, whether existing now or in the future anywhere in the world: (a) patents and

patent applications; (b) continuations, continuations-in-part, divisionals and substitute applications with respect to any such patent
application; (c) any patents issued based on or claiming priority to any such patent applications; (d) any reissue, reexamination, renewal or
extension (including any supplemental patent certificate) of any such patents; and (e) any confirmation patent or registration patent or patent
of addition based on any such patents.

1.26 “Person” shall mean an individual, corporation, partnership, limited liability company, trust, business trust, association, joint
stock company, joint venture, pool, syndicate, sole proprietorship, unincorporated organization, governmental authority or any other form
of entity or organization not specifically listed herein.

1.27 “Product” shall mean any Composition of Matter that comprises or contains the Human Engineered™ Tactic Antibodies or

any derivatives, conjugates and/or fragments thereof.

1.28 "Program Invention" shall mean any invention (whether or not patentable), discovery, Composition of Matter, improvement,

enhancement, technology, data or information made or conceived in connection with the conduct of activities pursuant to the Prior
Agreement.

1.29 “PTO” shall have the meaning set forth in Section 5.4(c).

1.30 “Term” shall have the meaning set forth in Section 7.1.

1.31 “Third Party” shall mean any Person other than XOMA or TACTIC or their Affiliates.

1.32 “Title XI” shall have the meaning set forth in Section 11.2.

1.33  “Valid Claim” shall mean (a) a claim of an issued and unexpired patent which has not been held permanently revoked,
unenforceable or invalid by a decision of a court or other governmental agency of competent jurisdiction, unappealable or unappealed
within the time allowed for appeal and that is not admitted to be invalid or unenforceable through reissue, disclaimer or otherwise, or (b) a
claim (including amendments) of a pending patent application that has neither (i) been abandoned or finally rejected without the possibility
of appeal or refiling nor (ii) been pending for more than [***], provided that any claim excluded from this definition in reliance on this
clause (b)(ii) that subsequently issues shall constitute a Valid Claim so long as it meets the requirements of clause (a) above.

 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

1.34 "XOMA Deliverables" shall mean the XOMA materials and information delivered to ATTENUON under the Prior

Agreement.

1.35 “XOMA Patent Rights” shall have the meaning set forth in Section 1.37.

1.36 “XOMA Program Inventions” shall have the meaning set forth in Section 1.37.

1.37 “XOMA Program Inventions and Patent Rights” shall mean any and all (a) Program Inventions, whether or not patentable,
that (i) comprise or embody (A) [***] (B) methods that are generally applicable to the [***] or (ii) do not [***] and were invented solely
by employees, agents, consultants or contractors of [***] (collectively, the “XOMA Program Inventions”); and (b) all Patent Rights arising
out of the conduct of activities under the Prior Agreement that claim or cover such XOMA Program Inventions (the “XOMA Patent
Rights”).

ARTICLE 2

2.1 License Grants to TACTIC. XOMA hereby grants to TACTIC:

INTELLECTUAL PROPERTY RIGHTS

(a) a worldwide, non-exclusive license, with the right to sublicense in its sole discretion, under any and all

Intellectual Property Rights Controlled by XOMA at any time during the Term covering, claiming or relating to Program Inventions, and/or
XOMA’s Human Engineering™ technology utilized in XOMA's performance of work under the Prior Agreement including, without
limitation, the Human Engineering™ Patent Rights), to make, have made, use, offer for sale, sell and import Human Engineered™ TACTIC
Antibodies and any Product.

2.2 Ownership of Intellectual Property.

2.2.1 Inventorship for Program Inventions shall be determined in accordance with U.S. patent laws.

2.2.2 TACTIC reserves and shall retain all right, title and interest in and to the TACTIC Antibody and all Intellectual

Property Rights therein.

2.2.3 Subject to the rights and licenses granted under this Agreement, ownership of all Program Inventions, irrespective of

inventorship, shall be as follows: (a) TACTIC shall own TACTIC Program Inventions and Patent Rights; (b) XOMA shall own all XOMA
Program Inventions and Patent Rights; and (c) TACTIC and XOMA shall jointly own, in equal undivided shares, any Joint Program
Inventions.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

2.2.4 XOMA hereby assigns, and agrees to assign, to TACTIC all of XOMA’s right, title and interest in and to any and all

TACTIC Program Inventions and Patent Rights, including, without limitation, the right to sue for past, present and future infringement.
XOMA agrees, without further consideration, to execute all documents, certificates and other instruments, and to do all acts reasonably
necessary to vest and confirm in TACTIC, its successors and assigns, the legal title to all such Program Inventions and Patent Rights;
provided that, if such requests require more than de minimis out-of-pocket expenditures by XOMA, TACTIC will reimburse XOMA for
such expenditures, to the extent previously approved by TACTIC in writing (which approval shall not be unreasonably withheld or
delayed).

2.2.5 TACTIC hereby assigns, and agrees to assign, to XOMA all of TACTIC’s right, title and interest in and to any and

all XOMA Program Inventions and Patent Rights, including, without limitation, the right to sue for past, present and future infringement.
TACTIC agrees, without further consideration, to execute all documents, certificates and other instruments, and to do all acts reasonably
necessary to vest and confirm in XOMA, its successors and assigns, the legal title to all such Program Inventions and Patent Rights;
provided that, if such requests require more than de minimis out-of-pocket expenditures by TACTIC, XOMA will reimburse TACTIC for
such expenditures, to the extent previously approved by XOMA in writing (which approval shall not be unreasonably withheld or delayed).

2.3 No Implied Rights. Only the rights and licenses granted pursuant to the express terms of this Agreement shall be of any legal

force. Without limiting the foregoing and subject to the license granted by XOMA in Section 2.1, neither the grants provided in Section 2.1
nor the assignment from XOMA to TACTIC provided in Section 2.2.4 provide TACTIC with any right to practice the methods of the
Human Engineering™ technology (including, without limitation, the Human Engineering™ Patent Rights) or, subject to the grants made in
Section 2.1, to receive from XOMA or use information received from XOMA related to its Human Engineering™ technology, and in no
event shall XOMA be required to disclose such methods or information.

2.4 Sublicenses. Any sublicense permitted hereunder shall be set forth in a written agreement containing provisions relating to

ownership of intellectual property that are substantially consistent with, and with respect to audits and confidentiality that are substantially
consistent with, and at least as stringent as, those contained herein and shall be subject and subordinate to the terms and conditions of this
Agreement.

ARTICLE 3

FINANCIAL TERMS

3.1 Milestone Payments. In full consideration of the rights and licenses granted to TACTIC herein, TACTIC shall pay to XOMA

the applicable payments below (each, a “Milestone Payment”)

Event

1. [***]

Payment

[***]

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

2. [***]

3. [***]

4. [***]

5. [***]

6. [***]

[***]

[***]

[***]

[***]

[***]

Each Milestone Payment shall be due [***] days from the achievement of the corresponding milestone event. Each Milestone Payment
[***], and [***] (a) [***] or (b) [***].

3.2 Third Party Payments. TACTIC will be responsible for all financial obligations due Third Parties.

3.3 Payments; Currency. All payments due under this Article 3 shall be paid in United States dollars in immediately available

funds to an account designated by XOMA.

3.4 Payment Reports and Timing.

3.4.1 TACTIC shall make a written report to XOMA within thirty (30) days of the achievement of each of the milestones

set forth in Section 3.1 with respect to Product

3.5 Payment Records and Audits.

3.5.1 TACTIC shall, and shall contractually require all Third Parties selling Products on its behalf to, keep complete and
accurate books of account for, and records of Net Sales of, Product in sufficient detail to enable the milestone payments payable under this
Agreement to be determined

3.5.2 Upon the written request of XOMA, TACTIC shall permit an independent auditor appointed by XOMA and

reasonably acceptable to TACTIC to have access during normal business hours to such of the records of TACTIC and its Affiliates as may
be reasonably necessary to verify the accuracy of the Net Sales under this Agreement. The auditor shall only disclose to XOMA whether
the Net Sales reported are correct or incorrect and the amount of any discrepancy. No other information shall be provided to XOMA
without the prior consent of TACTIC unless disclosure is required by law, regulation or judicial order. If XOMA determines that disclosure
is required by law, regulation or judicial order, it shall give TACTIC reasonable prior notice thereof in order for TACTIC to seek a
protective order against or limiting such disclosure. TACTIC is entitled to require the auditor to execute a reasonable confidentiality
agreement prior to commencing any such audit. Any agreement between TACTIC and/or any of its Affiliates, on the one hand, and one or
more Third Parties, on the other hand, pursuant to which such Third Party may market and/or sell Product shall contain provisions for
access and inspection of records substantially similar to the foregoing.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

3.5.3 Audits conducted under this Section 3.5 shall be at the expense of XOMA unless an unpaid amount for the full

period covered by the audit is identified, in which case all reasonable out-of-pocket costs incurred by the auditor to perform the audit will
be paid promptly by TACTIC. Any unpaid amounts discovered by such inspections or otherwise will be paid promptly by TACTIC, with
interest on such amounts from the date(s) such amount(s) were due, at a rate equal to the lesser of the prime rate reported by the Bank of
America plus [***] per annum, or the highest interest rate permitted under applicable New York law.

ARTICLE 4

CONFIDENTIALITY

4.1 Confidential Information. Except as expressly provided herein, the Parties agree that, for the Term and for [***] thereafter,

each of them shall keep completely confidential and shall not publish or otherwise disclose and shall not use for any purpose except for the
purposes contemplated by this Agreement any Confidential Information furnished to it by the other Party. Each Party also agrees to cause
its Affiliates with access to any Confidential Information to comply with all terms of this Agreement relating to such Confidential
Information and the treatment thereof, and each Party shall remain primarily liable for any breach of any such provision by any of its
Affiliates.

4.2 Permitted Use and Disclosures. The receiving Party may use or disclose Confidential Information to the extent such use or
disclosure is reasonably necessary in complying with any applicable law, regulation or court order or in conducting clinical trials or in
connection with seeking, enforcing or defending Patent Rights covering Program Inventions; provided that if the receiving Party is required
to make any such disclosure of Confidential Information, other than pursuant to a confidentiality agreement, it will give reasonable advance
notice to the disclosing Party of such disclosure and will use its reasonable efforts to secure confidential treatment of such Confidential
Information prior to its disclosure (whether through protective orders or otherwise). Notwithstanding the foregoing, TACTIC may use and
disclose the Confidential Information of XOMA as reasonably necessary in connection with the exercise of TACTIC’s rights under Section
2.1(a) and otherwise with respect to the development or exploitation of TACTIC Program Inventions and Patent Rights, including, without
limitation, to actual or prospective business partners, investors, contractors, and sublicensees of TACTIC, in each case, pursuant to a
confidentiality agreement with terms substantially consistent with, and at least as stringent as, those set forth in this Agreement.

4.3 Confidential Terms. Except as expressly provided herein, each Party agrees not to disclose any terms of this Agreement to any

Third Party without the consent of the other Party; provided that disclosures may be made as required by securities or other applicable
laws, or as reasonably necessary to actual or prospective business partners, investors and Tactic's sublicensees under this Agreement
pursuant to a confidentiality agreement with terms at least as stringent as those in this Agreement, or to a Party's accountants, attorneys and
other professional advisors owing a contractual or other duty of confidentiality to such Party. Upon the reasonable written request of the
disclosing Party, the receiving Party shall promptly return or destroy, and certify the same in writing, all Confidential Information of the
other Party; provided that the receiving Party may retain one (1) copy of any such Confidential Information in its files for purposes of
maintaining appropriate records of its activities in connection with this Agreement.

 
 
 
 
 
 
 
 
 
 
 
4.4 Use of Name. Neither Party shall use the name or trademarks of the other Party, except to the extent that a Party is permitted to

use the Confidential Information of the other Party or required to do so pursuant to this Article 4, without the prior written consent of such
other Party, such consent not to be unreasonably withheld or delayed.

4.5 Previous Agreements. The parties acknowledge and understand that the Prior Agreement is now void and superseded by this

Agreement.

ARTICLE 5

PATENT RIGHTS

5.1 Prosecution and Maintenance of TACTIC and XOMA Patent Rights. TACTIC shall have sole and exclusive responsibility for

Patent Prosecution of all TACTIC Patent Rights. XOMA shall have sole and exclusive responsibility for Patent Prosecution of XOMA
Patent Rights. In each such case, the non-prosecuting Party will provide the prosecuting Party with such assistance and execute such
documents as are reasonably necessary to permit or continue such Patent Prosecution by the prosecuting Party. The prosecuting Party shall
bear all Patent Prosecution expenses, including attorneys’ fees, incurred by such Party, or by the other Party at the request of the
prosecuting Party, in the performance of Patent Prosecution.

5.2 Enforcement of TACTIC and XOMA Patent Rights.

5.2.1                      Notifications. Each Party shall provide to the other Party copies of (a) any written notices it receives

from any Third Party regarding any patent nullity action, declaratory judgment action, alleged invalidity, unenforceability,
infringement or non-infringement with respect to or alleged misappropriation of intellectual property with respect to Program
Inventions, or the TACTIC Patent Rights, and (b) any written allegations it receives from a Third Party that the manufacture, use,
sale, offer for sale or import of Product infringes the Intellectual Property Rights of such Third Party, in each case promptly
following receipt thereof.

5.2.2                      Infringement Proceedings Against Third Parties . TACTIC shall have the sole and exclusive right, but

not the obligation, to institute and direct legal proceedings against any Third Party believed to be infringing the TACTIC Patent
Rights. XOMA shall have the sole and exclusive right, but not the obligation, to institute and direct legal proceedings against any
Third Party believed to be infringing any XOMA Patent Rights. Each Party will bear all of its own costs, including attorneys’ fees,
relating to such legal proceedings; provided that the Party directing such legal proceedings shall bear the other Party’s out-of-pocket
expenses, including attorneys’ fees, incurred in complying with requests for cooperation made by the directing Party. Without
limiting the foregoing, any recovery in connection with such suit or proceeding will be retained solely by the Party directing such
suit or proceeding.

 
 
 
 
 
 
 
 
 
 
 
 
5.3 Infringement Proceedings by Third Parties . In the event that a Party receives written notice that it or any of its Affiliates have
been individually named as a defendant in a legal proceeding by a Third Party alleging infringement or misappropriation of a Third Party
Intellectual Property Right as a result of the manufacture, use, sale, offer for sale or import of a Product or the XOMA Materials, such Party
shall promptly notify the other Party in writing. Such written notice shall include a copy of any summons or complaint (or the equivalent
thereof) received regarding the foregoing.

5.4 Cooperation. Each Party hereby agrees:

(a) 

(b) 

(c) 

to cooperate in the Patent Prosecution of any inventions within the Program Inventions ;

to take all reasonable additional actions and execute such agreements, instruments and documents as may be
reasonably required to perfect the other Party’s ownership interest in the XOMA Materials and the Program
Inventions in accordance with the intent of this Agreement;

to provide comments and suggestions, as reasonably requested by the other Party, with respect to copies of drafts
of material filings with or other submissions to the U.S. Patent and Trademark Office or any foreign counterpart
(the “PTO”) relating to Patent Prosecution, or the court or other tribunal relating to any infringement claims
against Third Parties under the TACTIC Patent Rights or the defense of infringement or misappropriation claims
by Third Parties relating to Product;

(d) 

to cooperate, as reasonably necessary, with the other Party in gaining patent term extensions, supplemental
protection certificates or their equivalents wherever applicable to TACTIC Patent Rights;

5.5 No Other Technology Rights. Except as otherwise provided in this Agreement, under no circumstances shall a Party, as a result

of this Agreement, obtain any ownership interest or other right in any invention, discovery, Composition of Matter or other technology, or
in any other Intellectual Property Right, of the other Party (including without limitation those owned, controlled or developed by the other
Party at any time pursuant to this Agreement).

ARTICLE 6

6.1 Each Party hereby represents and warrants to the other Party as follows:

REPRESENTATIONS AND WARRANTIES

which it is organized.

6.1.1 Existence. Such Party is duly organized, validly existing and in good standing under the laws of the jurisdiction in

6.1.2 Authorization and Enforcement of Obligations. Such Party (a) has the requisite power and authority and the legal

right to enter into this Agreement and to perform its obligations hereunder, and (b) has taken all necessary action on its part to authorize the
execution and delivery of this Agreement and the performance of its obligations hereunder. This Agreement has been duly executed and
delivered on behalf of such Party, and constitutes a legal, valid, binding obligation, enforceable against such Party in accordance with its
terms.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
required to be obtained by such Party in connection with this Agreement have been obtained.

6.1.3 Consents. All necessary consents, approvals and authorizations of all governmental authorities and other Persons

6.1.4 No Conflict. The execution and delivery of this Agreement and the performance of such Party’s obligations

hereunder (a) do not conflict with or violate any requirement of applicable laws or regulations and (b) do not conflict with, or constitute a
default under, any contractual obligation of such Party.

6.1.5 Additional Representations of TACTIC. TACTIC further represents and warrants that (a) TACTIC was formed upon the
dissolution of ATTENUON, such that TACTIC can be considered a lawful successor of ATTENUON; (b) TACTIC is the successor and
rightful owner of certain IP rights developed by ATTENUON, including, but not limited to, ATN-658; (c) TACTIC will have in place by
the start of a Phase I clinical trial general liability and product liability insurance with respect to the research, development and
commercialization of the TACTIC Target, the TACTIC Antibody and Human Engineered™ TACTIC Antibodies in such amounts as are
reasonable and customary in the biopharmaceutical industry and covenants that it shall maintain appropriate general liability and product
liability insurance with respect thereto in such amounts for so long as such research, development and commercialization continues and
thereafter for so long as is reasonable and customary in the biopharmaceutical industry, and (d) TACTIC and its Affiliates will have in
place by the start of a Phase I clinical trial appropriate policies and procedures intended to assure that Confidential Information of XOMA,
or other material non-public information of XOMA, delivered or otherwise made available to TACTIC will not be used by TACTIC or its
officers, directors, employees or agents in connection with any activity that would constitute a criminal or civil violation of United States
securities laws and/or the regulations of the U.S. Securities and Exchange Commission and, for so long as any provision of this Agreement
remains in effect, TACTIC covenants that it shall maintain and enforce such policies and procedures and shall not disclose any such
Confidential Information of XOMA, or other material non-public information of XOMA, to TACTIC's Affiliates who do not then
maintain and enforce such policies.

6.2 DISCLAIMER OF WARRANTIES. EXCEPT AS OTHERWISE SET FORTH IN SECTION 6.1 OF THIS AGREEMENT,

NEITHER PARTY MAKES ANY REPRESENTATIONS OR WARRANTIES, EXPRESS OR IMPLIED, WITH RESPECT TO THE
ANTIBODIES AND OTHER INFORMATION DELIVERED OR TO BE DELIVERED PURSUANT TO THE PRIOR AGREEMENT
OR THE PROGRAM INVENTIONS, INCLUDING WITHOUT LIMITATION ANY WARRANTY OF MERCHANTABILITY,
FITNESS FOR A PARTICULAR PURPOSE OR NON-INFRINGEMENT OF THE PATENT RIGHTS OR OTHER INTELLECTUAL
PROPERTY RIGHTS OF ANY OTHER PERSON.

 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

ARTICLE 7

TERM AND TERMINATION

7.1 Term. Subject to Sections 7.5 and 7.6 hereof, the term of this Agreement will commence on the Effective Date and shall

remain in full force and effect until the expiration of all obligations of TACTIC under Article 3, unless earlier terminated pursuant to 7.2 or
7.3 (the period from the Effective Date through such expiration or earlier termination being referred to herein as the “Term”). Upon such
expiration, TACTIC shall be deemed to have a fully paid-up license to the rights set forth in Section 2.1.

7.2 Termination for Material Breach. This Agreement may be terminated by the non-breaching Party if the other Party is in breach

of its material obligations under this Agreement and after receiving notice describing such breach in reasonable detail and requesting its
cure has not cured such breach within [***] days (in the case of a payment breach with respect to any amount not being disputed in good
faith) or [***] days (in the case of a non-payment breach). Notwithstanding the foregoing sentence of this Section 7.2: (a) if such breach is
cured or shown to be non-existent within the aforesaid [***] days or [***] day period, the notice shall be deemed automatically withdrawn
and of no effect and the notifying Party shall provide written notice to the breaching Party of the withdrawal; and (b) without limiting the
effects of the following sentence of this Section 7.2, in the event of a good faith dispute with respect to the existence of a material breach,
the [***] day or [***] day cure period shall be tolled until such time as the dispute is resolved pursuant to Article 10. The Parties
acknowledge that any failure by XOMA to provide a Human EngineeredTM TACTIC Antibody that meets the Success Criteria or that meets
any other technical objectives shall not in and of itself be deemed a material breach of this Agreement.

7.3 Termination For Convenience. This Agreement may be terminated without cause at any time upon sixty (60) days prior written

notice by TACTIC to XOMA, at TACTIC’s discretion.

7.4 Contested Validity. If TACTIC, a TACTIC successor, a TACTIC sublicensee of the rights granted hereunder, or a person or
entity Controlled by any of the preceding entities, intends to challenge the validity or enforceability of any of the XOMA Patent Rights,
whether through a declaratory judgment action, opposition, post-grant proceeding or otherwise, then such entity shall: (a) [***] and (b)
[***].

7.5 Effect of Termination.

7.5.1 Termination of this Agreement shall not release either Party hereto from any liability (including, without limitation,

any payment obligation) which, at the time of such termination, has already accrued to the other Party or which is attributable to a period
prior to such termination nor preclude either Party from pursuing any rights and remedies it may have hereunder or at law or in equity with
respect to any breach of this Agreement.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

7.5.2 Upon any termination of this Agreement, TACTIC and XOMA shall (a) promptly return to the other Party all

Confidential Information received from the other Party (except that each Party may retain one copy for its files solely for the purpose of
determining its rights and obligations hereunder) or (b) destroy all such Confidential Information with the other Party’s consent.

Notwithstanding the survival of Article 2 as set forth in Section 7.6 below, (a) the rights and licenses of TACTIC

under Section 2.1 shall terminate and be of no further force or effect, and (b) TACTIC (on behalf of itself, its Affiliates, and its successors
and assigns) shall not (i) practice or exercise any invention claimed in, or license, authorize or otherwise allow any Third Party to practice
or exercise such invention claimed in, any XOMA Patent Rights or (ii) except as reasonably necessary to comply with applicable law,
regulation or court order as provided in Section 4.2, use or disclose, or authorize or otherwise allow the use or disclosure of, the XOMA
Deliverables, upon (A) termination of this Agreement by TACTIC pursuant to Section 7.3; (B) termination of this Agreement by XOMA
pursuant to Section 7.2 based on TACTIC 's failure to pay any amount due under Article 3 hereof and not being disputed in good faith; or
(C) TACTIC 's failure to pay a sum that had been disputed in good faith by the Parties (together with all accrued interest due thereon
under this Agreement) within [***] days after a final determination by an arbitrator pursuant to Section 9.3 that such amount is due under
this Agreement..

7.5.3 Nothing herein shall in any way limit or restrict XOMA’s ability to seek and obtain money damages, injunctive

relief or any other remedy, whether at law or in equity, that may be available from or awarded by a court of competent jurisdiction based
on, arising out of or relating to any breach of this Agreement by TACTIC.

or authorize or otherwise allow the use of any Human Engineered™ TACTIC Antibody.

7.5.4  Notwithstanding anything to the contrary herein, XOMA shall not, at any time during the Term or thereafter, use,

7.6 Survival. Sections 3.5, 7.5 and 7.6, and Articles 1, 2 (including, subject to Section 7.5.2, all rights and licenses therein), 4, 5, 6,

8, 9, 10 and 11 of this Agreement shall survive any termination hereof.

ARTICLE 8

INDEMNITY

8.1 Indemnity.

8.1.1 By XOMA. XOMA shall indemnify and hold TACTIC harmless, and hereby forever releases and discharges

TACTIC, from and against all losses, liabilities, damages and expenses (including reasonable attorneys’ fees and costs) resulting from all
claims, demands, actions and other proceedings by any Third Party to the extent arising from (a) the breach of any representation, warranty
or covenant of XOMA under this or the Prior Agreement, (b)  a claim that the processes or technologies used by XOMA in the
performance of its activities under the Prior Agreement (other than any such claim with respect to the CMV promoter), including, without
limitation, Human Engineering™ activities, infringe the Intellectual Property Rights of such Third Party (other than Intellectual Property
Rights to the TACTIC Target, any Antibody to the TACTIC Target (including any Product), or (c) the gross negligence or willful
misconduct of XOMA, its Affiliates or sublicensees in the performance of its obligations, and its permitted activities, under this or the Prior
Agreement; in each case except to the extent arising from the gross negligence or willful misconduct of ATTENUON or TACTIC

 
 
 
 
 
 
 
 
 
 
 
 
 
 
8.1.2 By TACTIC. TACTIC shall indemnify and hold XOMA harmless, and hereby forever releases and discharges

XOMA, from and against all losses, liabilities, damages and expenses (including reasonable attorneys’ fees and costs) resulting from all
claims, demands, actions and other proceedings by any Third Party to the extent arising from (a) the breach of any representation, warranty
or covenant of ATTENUON or TACTIC under this or the Prior Agreement, (b) excluding losses, liabilities, damages and expenses covered
by XOMA pursuant to Section 8.1.1(b), the making, having made, using, offering for sale, selling or importing of any Antibody to the
TACTIC Target (including without limitation any Human Engineered™ TACTIC Antibody or Product) by ATTENUON, TACTIC, its
Affiliates or licensees or by XOMA pursuant to the terms of this Agreement, (c) the use of the TACTIC Target or the ATTENUON
Deliverables by XOMA pursuant to the terms of the Prior Agreement or (d) the gross negligence or willful misconduct of ATTENUON,
TACTIC, their Affiliates or licensees in the performance of its obligations, and its permitted activities, under this or the Prior Agreement; in
each case except to the extent arising from (i) a claim that the processes used by XOMA in the performance of Human Engineering™
infringe the Intellectual Property Rights of such Third Party (other than Intellectual Property Rights to the TACTIC Target, any Antibody to
the TACTIC Target, or (ii) the gross negligence or willful misconduct of XOMA.

8.2 Procedure. A Party (the “Indemnitee”) that intends to claim indemnification under this Article 8 shall promptly notify the other
Party (the “Indemnitor”) of any claim, demand, action or other proceeding for which the Indemnitee intends to claim such indemnification.
The Indemnitor shall have the right to participate in, and to the extent the Indemnitor so desires, to assume the defense thereof with counsel
selected by the Indemnitor; provided, however, that the Indemnitee shall have the right to retain its own counsel, with the fees and
expenses to be paid by the Indemnitor, if representation of the Indemnitee by the counsel retained by the Indemnitor would be inappropriate
due to actual or potential differing interests between the Indemnitee and any other Party represented by such counsel in such proceeding.
The indemnity obligations under this Article 8 shall not apply to amounts paid in settlement of any claim, demand, action or other
proceeding if such settlement is effected without the prior express written consent of the Indemnitor, which consent shall not be
unreasonably withheld or delayed. The failure to deliver notice to the Indemnitor within a reasonable time after notice of any such claim or
demand, or the commencement of any such action or other proceeding, if prejudicial to its ability to defend such claim, demand, action or
other proceeding, shall relieve such Indemnitor of any liability to the Indemnitee under this Article 8 with respect thereto, but the omission
so to deliver notice to the Indemnitor shall not relieve it of any liability that it may have to the Indemnitee otherwise than under this Article
8. The Indemnitor may not settle or otherwise consent to an adverse judgment in any such claim, demand, action or other proceeding that
diminishes the rights or interests of the Indemnitee without the prior express written consent of the Indemnitee, which consent shall not be
unreasonably withheld or delayed. The Indemnitee, its employees and agents shall reasonably cooperate with the Indemnitor and its legal
representatives in the investigation and defense of any claim, demand, action or other proceeding covered by this Article 8.

 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

ARTICLE 9

DISPUTE RESOLUTION

9.1 Attempts to Amicably Resolve Disputes. If any dispute, controversy or claim is initiated by either Party arising out of,

resulting from or relating in any way to this Agreement, the performance by either Party of its obligations under this Agreement or the
subject matter of this Agreement (a “Dispute”), then the Parties shall attempt to resolve such Dispute as follows. The Party initiating the
Dispute shall give written notice to the other Party specifying in reasonably specific detail the basis for such Dispute. Following receipt of
such notice, the Parties shall refer the Dispute to their respective chief executive officers (or their designees) for resolution. The Parties’
respective chief executive officers (or their designees) shall meet (in person, by videoconference or by telephone as mutually agreed upon
by the Parties) to attempt to reach a mutually acceptable resolution of the Dispute.

9.2 Mediation. Subject to Section 9.4, if a Dispute is not resolved in the manner set forth in Section 9.1 within [***] days after
receipt of notice under Section 9.1, the Parties agree to try in good faith to resolve such dispute in an expeditious manner by mediation
administered by the CPR Institute for Dispute Resolution or its successor organization (“CPR”) in accordance with its mediation procedure.
The mediation proceeding shall be conducted at the location of the Party not originally requesting the resolution of the Dispute. The Parties
agree that they shall share equally the cost of the mediation filing and hearing fees and the cost of the mediator. Each Party must bear its
own attorney’s fees and associated costs and expenses. For the avoidance of doubt, nothing in connection with such mediation shall be
binding on either Party, except for the provisions regarding sharing of costs set forth in this Section 9.2.

9.3 Arbitration.

referral to mediation under Section 9.2 shall be finally resolved by binding arbitration, as set forth in this Section 9.3.

9.3.1 Subject to Section 9.4, any Dispute that is not resolved in the manner set forth in Section 9.2 within [***] days after

9.3.2 Whenever a Party shall decide to institute arbitration proceedings, it shall give written notice to that effect to the

other Party. Any such arbitration shall be conducted under the Commercial Arbitration Rules of the American Arbitration Association by a
panel of one (1) arbitrator appointed in accordance with such rules to be appointed within [***] days of such notice. Such arbitrator shall
have no less than [***] of experience directly in the field of biotechnology licensing, and shall be available to serve under the geographic
and time constraints set forth herein and in Section 9.3.3. Any such arbitration shall be held in New York, New York.

 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

9.3.3 The arbitrator shall be jointly instructed by the Parties in writing to set a schedule that will enable them to complete

all proceedings and render their award within [***] days from the date of appointment of the arbitrator in accordance with Section 9.3.2.
For good cause shown, the arbitrator may extend this schedule for up to, but in no event more than, [***] additional days. The failure of the
arbitrator to render a final award within the foregoing time frame shall not give rise to a jurisdictional defect, but this fact shall not be
disclosed to the arbitrators until after the expiration of such [***] day period. The arbitrator shall have the authority to grant specific
performance in such equitable manner as they determine. The prevailing Party in any such arbitration (as determined by the arbitrator) shall
be entitled to recover its reasonable attorneys’ fees and expenses incurred in connection with such arbitration. Judgment upon the award so
rendered may be entered in any court having jurisdiction as provided in Section 9.5 or application may be made to such court for judicial
acceptance of any award and an order of enforcement, as the case may be.

based upon such claim, dispute or other matter in question would be barred by the applicable statute of limitations.

9.3.4 In no event shall a demand for arbitration be made after the date when institution of a legal or equitable proceeding

9.3.5 Notwithstanding the foregoing, either Party shall have the right, without waiving any right or remedy available to

such Party under this Agreement or otherwise, to seek and obtain from any court of competent jurisdiction any interim or provisional relief
that is necessary or desirable to protect the rights or property of such Party, pending, the selection of the arbitrators hereunder or pending
the arbitrators’ determination of any dispute, controversy or claim hereunder.

9.4 Disputes Regarding Patents. Notwithstanding any provision hereof to the contrary, any Dispute relating to the determination of

ownership, validity, enforceability or infringement by the other Party of a Party’s patents shall, if not resolved in the manner set forth in
Section 9.1 within [***] days after receipt of notice under Section 9.1, be submitted exclusively to the federal courts located in New York,
New York , and the Parties hereby consent to the jurisdiction and venue of such court.

9.5 Venue; Jurisdiction.

9.5.1 Any action or proceeding brought by either Party seeking to enforce any provision of, or based on any right arising

out of, this Agreement must be brought against either Party in the courts of the State of New York. Each Party (i) hereby irrevocably
submits to the jurisdiction of the state courts of the State of New York and to the jurisdiction of any United States District Court in the
State of New York , for the purpose of any suit, action, or other proceeding arising out of or based upon this Agreement or the subject
matter hereof brought by any Party or its successors or assigns, (ii) hereby waives, and agrees not to assert, by way of motion, as a defense,
or otherwise, in any such suit, action, or proceeding, any claim that it is not subject personally to the jurisdiction of the above-named courts,
that its property is exempt or immune from attachment or execution, that the suit, action or proceeding is brought in an inconvenient forum,
that the venue of the suit, action, or proceeding is improper or that this Agreement or the subject matter hereof may not be enforced in or by
such court, and (iii) hereby waives and agrees not to seek any review by any court of any other jurisdiction that may be called upon to grant
an enforcement of the judgment of any such Illinois state or federal court.

 
 
 
 
 
 
 
 
 
9.5.2 Process in any action or proceeding seeking to enforce any provision of, or based on any right arising out of, this

Agreement may be served on any Party anywhere in the world. Each Party consents to service of process by registered mail at the address to
which notices are to be given pursuant to Section 11.4. Nothing herein shall affect the right of a Party to serve process in any other manner
permitted by applicable law. Each Party further agrees that final judgment against it in any such action or proceeding arising out of or
relating to this Agreement shall be conclusive and may be enforced in any other jurisdiction within or outside the United States of America
by suit on the judgment, a certified or exemplified copy of which shall be conclusive evidence of the fact and of the amount of its liability.

9.5.3 Each Party agrees that it shall not, and that it shall instruct those in its control not to, take any action to frustrate or

prevent the enforcement of any writ, decree, final judgment, award (arbitral or otherwise) or order entered against it with respect to this
Agreement, and shall agree to be bound thereby as if issued or executed by a competent judicial tribunal having personal jurisdiction
situated in its country of residence or domicile.

ARTICLE 10

SUCCESSORS AND ASSIGNS

10.1 Limited Right to Assign. Neither TACTIC nor XOMA may transfer or assign this Agreement or any of its rights hereunder

without the written consent of the other; provided, however, that (a) XOMA may, without such consent, assign this Agreement and its
rights and obligations hereunder to a Third Party only in connection with the transfer or sale of all or substantially all of its business relating
to Human Engineering™, or in the event of a merger, consolidation or other transaction resulting in a change in control of XOMA, and (b)
TACTIC may, without such consent, assign this Agreement and its rights and obligations hereunder to a Third Party only in connection with
the transfer or sale of a Human Engineered™ version of a TACTIC Antibody or all or substantially all of its assets relating to its anti-uPAR
monoclonal antibodies or in the event of a merger, consolidation or other transaction resulting in a change in control of TACTIC. Any
attempted transfer or assignment in violation of this Section 10.1 shall be void. Nothing herein shall prohibit any transfer or assignment by
either TACTIC or XOMA to or among any of their respective Affiliates.

10.2 Permitted Successors and Assigns. This Agreement shall be binding upon and inure to the benefit of the Parties and their

successors and assigns as permitted in Section 10.1.

ARTICLE 11

MISCELLANEOUS

11.1 Governing Law. This Agreement and any dispute arising from the performance or breach hereof shall be governed by and

construed and enforced in accordance with the laws of the State of New York, without reference to conflicts of laws principles.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

11.2 Bankruptcy. All rights and licenses granted under or pursuant to this Agreement by one Party to the other are, for all purposes

of Section 365(n) of Title XI of the United States Code (“Title XI”), licenses of rights to “intellectual property” as defined in Title XI.
During the Term each Party shall create and maintain current copies to the extent practicable of all such intellectual property. If a
bankruptcy proceeding is commenced by or against one Party under Title XI, the other Party shall be entitled to a copy of any and all such
intellectual property and all embodiments of such intellectual property, and the same, if not in the possession of such other Party, shall be
promptly delivered to it (a) upon such Party’s written request following the commencement of such bankruptcy proceeding, unless the
Party subject to such bankruptcy proceeding, or its trustee or receiver, elects within [***] days to continue to perform all of its obligations
under this Agreement, or (b) if not delivered as provided under clause (a) above, upon such other Party’s request following the rejection of
this Agreement by or on behalf of the Party subject to such bankruptcy proceeding. If a Party has taken possession of all applicable
embodiments of the intellectual property of the other Party pursuant to this Section 11.2 and the trustee in bankruptcy of the other Party
does not reject this Agreement, the Party in possession of such intellectual property shall return such embodiments upon request. If a Party
seeks or involuntarily is placed under Title XI and the trustee rejects this Agreement as contemplated under 11 U.S.C. 365(n)(1), the other
Party hereby elects, pursuant to Section 365(n) of Title XI, to retain all rights granted to it under this Agreement to the extent permitted by
law.

11.3 Waiver. No waiver of any rights shall be effective unless consented to in writing by the Party to be charged and the waiver of

any breach or default shall not constitute a waiver of any other right hereunder or any subsequent breach or default.

11.4 Notices. All invoices, notices, requests and other communications hereunder shall be in writing and shall be delivered or sent

in each case to the respective address specified below, or such other address as may be specified in writing to the other Party hereto, and
shall be effective on receipt.

If to TACTIC: 

Tactic Pharma, LLC

                                                                          [***]

                                                                        Attention: Andrew Mazar, CSO.

With a copy to: 

Baker & Hostetler, LLP 2929 Arch Street

Cira Centre – 12th Floor

Philadelphia, PA 19004

Attention: Tactic Pharma Legal Counsel, Dr. Jeffrey H. Rosedale

If to XOMA: 

XOMA (US) LLC

                                                                         2910 Seventh Street

                                                                        Berkeley, California 94710

                                                                        Attention: Legal Department

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
with a copy to: 

XOMA (US) LLC

                                                                          2910 Seventh Street

                                                                          Berkeley, California 94710

                                                                          Attention: Legal Department

11.5 Independent Contractors. The Parties are independent contractors under this Agreement. Nothing contained in this Agreement

is intended nor is to be construed so as to constitute TACTIC or XOMA as partners or joint venturers with respect to this Agreement.
Except as expressly provided for by this Agreement, no Party shall have any express or implied right or authority to assume or create any
obligations on behalf of or in the name of any other Party or to bind any other Party to any other contract, agreement or undertaking with
any Third Party.

11.6 Force Majeure. A Party shall neither be held liable or responsible to the other Party, nor be deemed to have defaulted under or

breached this Agreement, for failure or delay in fulfilling or performing any obligation under this Agreement (other than an obligation for
the payment of money) to the extent, and for so long as, such failure or delay is caused by or results from causes beyond the reasonable
control of such Party, including but not limited to fire, floods, embargoes, war, acts of war (whether war be declared or not), insurrections,
riots, civil commotions, strikes, lockouts or other labor disturbances, acts of God or acts, omissions or delays in acting by any governmental
authority or other Party.

11.7 Other Activities. Except as otherwise expressly provided in this Agreement, nothing in this Agreement shall preclude either
Party from conducting other programs (either for its own benefit or with or for the benefit of any other Person) to conduct research, or to
develop or commercialize products or services, for use in any field.

11.8 Headings. The captions to the several sections hereof are not a part of this Agreement, but are included merely for

convenience of reference only and shall not affect its meaning or interpretation.

11.9 Entire Agreement; Amendment.

11.9.1 This Agreement constitutes the entire and exclusive agreement between the Parties with respect to the subject

matter hereof and supersedes and cancels all previous discussions, agreements, representations, commitments and writing in respect
thereof.

authorized representatives of the Parties.

11.9.2 No amendment or addition to this Agreement shall be effective unless reduced to writing and executed by the

11.10 Illegality; Unenforceability. In the event that any provision of this Agreement shall be determined to be illegal or
unenforceable, that provision will be limited or eliminated to the minimum extent necessary so that this Agreement shall otherwise remain
in full force and effect and enforceable.

11.11 Counterparts. This Agreement may be executed in counterparts, each of which shall be deemed to be an original and together

shall be deemed to be one and the same agreement.

[SIGNATURE PAGE FOLLOWS ]

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
IN WITNESS WHEREOF, the Parties have executed this Agreement as of the date first set forth above.

         TACTIC PHARMA, LLC

XOMA (US) LLC

By: /s/ Andrew Mazar
Andrew Mazar

            Chief Scientific Officer

By: /s/ James Neal
James R. Neal
VP, Business Development & Program Leadership

 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

Schedule 1.16

Title: 

[***]
Inventors:                                Studnicka, Little, Fishwild, Kohn

Human Engineering™ Patent Rights

Based on [***].

COUNTRY
[***]

[***]

SERIAL NO.
[***]

PATENT NO.
[***]

EXPIRES
[***]

-1-

 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

VALIDIVE® OPTION AND LICENSE AGREEMENT

BY AND BETWEEN

MONOPAR THERAPEUTICS INC.

AND

ONXEO S.A.

 
 
 
 
 
 
 
 
 
 
 
  
            
 
 
 
 
 
 
 
TABLE OF CONTENTS

1.
2,
3
4
5
6
7
8
9
10
11

DEFINITIONS AND INTERPRETATION
MONOPAR VALIDIVE OPTION; MONOPAR DEVELOPMENT AND COMMERCIALIZATION
LICENSES; TECHNOLOGY TRANSFER; EXCLUSIVITY
FINANCIAL TERMS
INTELLECTUAL PROPERTY
WARRANTIES AND LIMITATION OF LIABILITY
INDEMNITY AND INSURANCE
CONFIDENTIALITY
TERM AND TERMINATION
DISPUTE RESOLUTION
MISCELLANEOUS

2
11
16
18
22
25
27
29
31
37
38

SCHEDULE
1
SCHEDULE
2
SCHEDULE
3
SCHEDULE
4
SCHEDULE
5

Licensed Patents

Licensed Know-How

Licensed Trademarks

Validive Materials

Confirmatory Patent License

 
 
 
 
 
 
 
OPTION AND LICENSE AGREEMENT

THIS OPTION AND LICENSE AGREEMENT  (together with any Schedules attached hereto, this “Agreement”) is made and entered
into  as  of  June  17,  2016  (the “Effective  Date”),  by  and  between  Monopar  Therapeutics  Inc.,  a  Delaware  corporation  located  at  598
Rockefeller Rd, Lake Forest, Illinois 60201, United States of America (“Monopar”), and Onxeo S.A., a French société anonyme à Conseil
d’administration located at 49, boulevard du Général Martial Valin, 75015 Paris, France (“ Onxeo”). Monopar and Onxeo are sometimes
referred to herein individually as a “Party” and collectively as the “Parties.”

WHEREAS:

RECITALS

(A) 

(B) 

(C) 

(D) 

Onxeo owns Patents, Trademark registrations and other proprietary rights relating to Validive® (as  defined  below). At  this  time,
Onxeo does not intend to undertake any further development of Validive®.

Monopar has expertise in research, development, and commercialization of pharmaceutical products.

Onxeo desires to grant, and Monopar desires to obtain, an exclusive option to take a license to research, develop, and commercialize
Validive® on  an  exclusive  basis  for  any  and  all  uses  in  the  Field  in  the  Territory  (each,  as  defined  below),  all  on  the  terms  and
conditions set forth herein.

Upon exercise by Monopar of the option for the license for Validive ®, Onxeo desires to grant Monopar, and Monopar desires to
obtain, an exclusive license in the Field in the Territory to use, sell, offer for sale, import, and make or have made Licensed Products
(as defined below) in the Field in the Territory on the terms and conditions set forth herein.

 
 
 
 
 
 
 
 
 
 
 
 
NOW IT IS HEREBY AGREED as follows:

AGREEMENT

1.

1.1

DEFINITIONS AND INTERPRETATION

In this Agreement the words and phrases set out below shall, unless the context requires otherwise, have the corresponding meaning
attributed to them below.

“Active Party” has the meaning set forth in Section 5.3.5.

“Affiliate” means with respect to a given entity, any person, corporation, partnership or other entity, that Controls, is Controlled by,
or is under common Control with such entity.

“Agreement” means this agreement and each of the Schedules as amended from time to time in accordance with Section 11.3.

“Arising Intellectual Property”  means  all  Intellectual  Property,  including  Know-How,  conceived,  created  or  invented  after  the
Effective Date by or on behalf of either Party; and any Patents which claim any inventions described or comprised in such Know-
How, but excluding Intellectual Property, including Know-How, comprised in the Licensed Intellectual Property.

“Audit for Cause” has the meaning set forth in Section 2.2.3.

“Bankruptcy Code” has the meaning set forth in Section 9.4.

“Breaching Party” has he meaning set forth in Section 9.2.1.

“Business Day” means a day other than a Saturday, Sunday or any public holiday in Paris, France or New York, New York, United
States.

“Clinical Data” means any Know-How that is included in, or supports, a regulatory submission for approval of the testing of drugs
in man or for approval for the placing of medicinal products on the market (including submissions to the FDA, the EMA or other
competent Regulatory Authorities).

“Combination Product” means any product that comprises a Licensed Product sold in conjunction with another active component
so as to be a combination product (whether packaged together or in the same therapeutic formulation).

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
“Commencement” means, in relation to a clinical trial, the date upon which a Licensed Product is first administered to a human
subject, whether such subject is a healthy volunteer or a patient.

“Commercialization”  or “Commercialize”  means  activities  directed  to  obtaining  pricing  and  reimbursement  approvals,
marketing,  promoting,  distributing,  offering  for  sale,  or  selling  a  Licensed  Product.  For  clarity,  “Commercialization”  shall  not
include manufacturing activities, but shall include importation, exportation and use related to offering for sale or selling a Licensed
Product.

“Commercially Reasonable Efforts” means efforts of a Party to carry out its obligations in a diligent and sustained manner using
such  effort  and  employing  such  resources  normally  used  by  an  established  biopharmaceutical  company  in  the  exercise  of  its
reasonable business discretion relating to the research, development or commercialization of a similar product owned by such Party
or to which such Party has exclusive rights, with similar product characteristics, that is of similar market potential at a similar stage
in  its  development  or  product  life,  taking  into  account  issues  of  market  exclusivity  (including  Patent  coverage  and  Regulatory
Exclusivity), safety and efficacy, product profile, the competitiveness of the marketplace, the proprietary position of the compound
or product, the regulatory structure involved, the profitability of the applicable products (including pricing and reimbursement status
achieved), and other relevant factors, including technical, legal, scientific, and/or medical factors.

“Confidential Information” means any information, in tangible or non-tangible form (including oral disclosure) including Know-
How, research and development plans, information relating to the customers, suppliers, business partners, clients, finances, business
plans and products (in each case actual or prospective) of a Party, the terms of this Agreement, and any other technical or business
information, which is obtained by either Party from the other (or its representatives) pursuant to this Agreement and is marked as
confidential, or indicated by notice as being confidential no more than five (5) Business Days after its disclosure. Licensed Know-
How shall be deemed the Confidential Information of Onxeo.

“Control” means:

(a) 

(b) 

the  possession  (directly  or  indirectly)  of  fifty  per  cent  (50%)  or  more  of  the  voting  stock  or  other  equity  interest  of  a
subject entity with the power to vote, or the power in fact to control the management decisions of such entity through the
ownership of securities or by contract or otherwise;

in respect of any Patent Rights, Know-How or other Intellectual Property whether owned by or licensed to an entity, the
possession  of  the  legal  right  and  ability  to  grant  the  respective  licenses  or  sublicenses  as  provided  in  this Agreement
without violating the terms of any agreement or other arrangement with any Third Party;

 
 
 
 
 
 
 
 
 
 
and “Controlling” and “Controlled by” shall be construed accordingly.

“Cure Period” has the meaning set forth in Section 9.2.1.

 “Development” means pre-clinical and clinical drug development activities reasonably relating to the discovery and development
of pharmaceutical compounds and submission of information to a Regulatory Authority, including toxicology, pharmacology, and
other  discovery  and  pre-clinical  studies,  test  method  development  and  stability  testing,  manufacturing  process  development
(including validation test methods and procedures), formulation development, delivery system development, quality assurance and
quality  control  development,  statistical  analysis,  clinical  trials  and  activities  relating  to  obtaining  Regulatory  Approval,  but
excluding Commercialization activities. When used as a verb, “Develop” means to engage in Development.

“Disclosing Party” has the meaning set forth in Section 8.1.

“Effective Date” means the date this Agreement is made.

“EMA” means the European Medicines Agency or any successor to it.

“Executive  Officers”  means  a  representative  of  Onxeo  authorized  by  notice  to  Monopar,  and  the  Chief  Executive  Officer  of
Monopar or such other authorized senior manager of a Party as may be substituted from time to time upon the giving of written
notice to the other Party.

“Extended Exclusivity Period”  means  any  period  during  which  one  of  the  following  subsists  in  respect  of  a  Licensed  Product:
orphan  drug  designation  or  exclusivity,  pediatric  designation  or  exclusivity,  new  chemical  entity  exclusivity,  or  other  exclusivity
(excluding a Patent) granted by a Regulatory Authority beyond the expiry of the relevant Patent.

“FDA” means the United States Food and Drug Administration or any successor to it.

“Field” means any and all uses.

“First  Commercial  Sale”  means  the  first  transfer  of  a  Licensed  Product  by  Monopar  to  the  first  Third  Party  (other  than  a
Sublicensee or a distributor) in any country in the Territory, in exchange for cash or some equivalent to which value can be assigned
for the purpose of determining Net Sales, after Regulatory Approval of such Licensed Product has been granted, or such marketing
and sale is otherwise permitted, by the Regulatory Authority of such country, excluding registration samples, compassionate use,
and use in Phase IV Trials.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
“Force Majeure” means in relation to either Party any event or circumstance which is beyond the reasonable control of that Party,
which event or circumstance that Party could not reasonably be expected to have taken into account at the Effective Date and which
results in or causes the failure of that Party to perform any or all of its obligations under this Agreement including an act of God,
lightning, fire, storm, flood, earthquake, strike, lockout or other industrial disturbance, war, a terrorist act, blockade, revolution, riot,
insurrection, civil commotion, public demonstration, sabotage, act of vandalism, explosion, provided that lack of funds shall not be
interpreted as a cause beyond the reasonable control of that Party.

“GAAP”  shall  mean  generally  accepted  accounting  principles  as  applicable  in  the  United  States,  consistently  applied;  provided
that,  to  the  extent  that  a  Party  adopts  International  Financial  Reporting  Standards  (IFRS),  then  “GAAP”  means  International
Financial Reporting Standards (IFRS), consistently applied.

“Inactive Party” has the meaning set forth in Section 5.3.5.

“IND” means an investigational new drug application filed with the FDA, or an application filed with any Regulatory Authority
outside the United States of America (including any supranational agency such as the EMA) necessary to commence human clinical
trials in such jurisdiction.

“Indemnified Party” has the meaning set forth in Section 7.1.3.

“Indemnifying Party” has the meaning set forth in Section 7.1.3.

“Indication”  means  a  disease  classification  block  as  defined  within  the  International  Statistical  Classification  of  Diseases  and
Related  Health  Problems  as  published  from  time  to  time  by  the  World  Health  Organization  (e.g.  “C50  Malignant  neoplasm  of
Breast”,  “C92  Myeloid  leukemia”,  “B20  Human  immunodeficiency  virus  [HIV]  disease  resulting  in  infectious  and  parasitic
diseases”, “M34 Systemic sclerosis”). For the avoidance of doubt, therapeutic indications having the same histology (such as first-
line to second-line therapies) do not constitute a different Indication.

“Intellectual Property” means Patents, Know-How and Trademarks.

“Intellectual Property Rights” means all Patent Rights, rights to Know-How, copyrights, database rights, design rights, rights in
Trademarks and domain names, and all rights or forms of protection of a similar nature or having equivalent or similar effect to any
of  them  which  may  subsist  anywhere  in  the  world,  whether  or  not  any  of  them  are  registered  including  any  application  for
registration of any of them.

 
 
 
 
 
 
 
 
 
 
 
 
“Know-How” means any unpatented, technical and other information which is not in the public domain including, ideas, concepts,
inventions  (whether  or  not  patentable),  discoveries,  data,  designs,  formulae,  algorithms,  methods,  models,  specifications,  clinical
data,  information  relating  to  biological  and  chemical  structures,  properties  and  functions  as  well  as  methods  for  synthesizing
chemical  compounds,  procedures  for  experiments  and  tests  (including  diagnostic  tests),  results  of  experimentation  and  testing,
results of research and development including laboratory records and data analyses. Information in a compilation or a compilation of
information may be Know-How notwithstanding that some or all of its individual elements are in the public domain.

“Laws” means all applicable laws, statutes, rules, regulations, ordinances and other pronouncements having the effect of law in any
federation,  nation,  multinational  governmental  entity,  state,  province,  county,  city  or  other  political  subdivision,  domestic  or
foreign.

“License Fee” has the meaning set forth in Section 4.2.

“Licensed Intellectual Property” means the Licensed Know-How, Licensed Patents and Licensed Trademarks.

“Licensed Know-How” means the Know-How directly and solely relating to the Licensed Product that is Controlled by Onxeo or
its Affiliates at the Effective Date as further described in SCHEDULE 2.

“Licensed Patents” means Patents further described in SCHEDULE 1.

“Licensed  Product”  means  all  products  containing  clonidine  or  its  analogues,  salts,  prodrugs,  and  any  derivatives  thereof,
formulated using Onxeo’s Lauriad® technology, including the product referred to as Validive® or Clonidine Lauriad®.

“Licensed Trademarks” means Trademarks further described in SCHEDULE 3.

“Losses” means any cost, expense or loss actually suffered resulting from any or all claims, causes of action or demands made by a
Third Party, including reasonable attorneys' fees.

“Material”  means  any  chemical  or  biological  material  and  any  property  rights  relating  to  any  of  the  foregoing  other  than
Intellectual Property Rights.

“Milestone Event” has the meaning given in Section 4.3.1.

“Milestone Payment” has the meaning given in Section 4.3.1

“Monopar Indemnified Parties” means Monopar and its Affiliates and their respective directors, officers, employees and agents.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

“Monopar Validive Option” has the meaning specified in Section 2.1.

“Monopar Validive Option Period” has the meaning specified in Section 2.1.1.

“NDA” means an application for approval to market a product commercially such as a New Drug Application filed pursuant to the
requirements of the FDA, as more fully defined in 21 CFR § 314.3 et seq, or a Biologics License Application filed pursuant to the
requirements  of  the  FDA,  as  more  fully  defined  in  21  CFR  §  601,  or  a  marketing  authorization  application  filed  pursuant  to  the
requirements of European Directive 2001/83/EC, or any equivalent or similar application filed with any other Regulatory Authority
in any country or region in the Territory, together, in each case, with all additions, deletions or supplements thereto.

“Net Sales” means the aggregate gross invoice prices of all Licensed Products sold by Monopar, its Affiliates or its Sublicensees to
Third Parties (that are not Sublicensees) anywhere within the Territory, including wholesale distributors, less deductions from such
amounts calculated in accordance with GAAP so as to arrive at net sales under GAAP, and further reduced by [***] or increased for
[***].

Any  and  all  set-offs  against  gross  invoice  prices  shall  be  calculated  in  accordance  with  GAAP.  Sales  or  other  commercial
dispositions of Licensed Products between Monopar and its Affiliates and its Sublicensees, and Licensed Products provided to Third
Parties without charge, in connection with research and development, clinical trials, compassionate use, humanitarian and charitable
donations, or indigent programs or for use as samples shall be excluded from the computation of Net Sales, and no payments will be
payable on such sales or such other commercial dispositions, except where such an Affiliate or Sublicensee is an end user of the
Licensed Product.

If a Licensed Product is sold or otherwise commercially disposed of for consideration other than cash or in a transaction that is not
at arm’s length between the buyer and the seller, then the gross amount to be included in the calculation of Net Sales shall be the
amount that would have been invoiced had the transaction been conducted at arm’s length and for cash. Such amount that would
have  been  invoiced  shall  be  determined,  wherever  possible,  by  reference  to  the  average  selling  price  of  the  relevant  Licensed
Product in arm’s length transactions in the relevant country.

Notwithstanding the foregoing, in the event a Licensed Product is sold as a Combination Product, Net Sales shall be calculated by
multiplying the Net Sales of the Combination Product by the fraction A/(A+B), where A is the gross invoice price of the Licensed
Product if sold separately in a country and B is the gross invoice price of the other product(s) included in the Combination Product if
sold separately in such country. If no such separate sales are made by Monopar, its Affiliates or Sublicensees in a country, Net Sales
of the Combination Product shall be calculated in a manner to be negotiated and agreed upon by the Parties, reasonably and in good
faith,  prior  to  any  sale  of  such  Combination  Product,  which  shall  be  based  upon  the  respective  cost  of  goods  sold  of  the  active
components of such Combination Product. In the event that the Parties are not able to so agree on the calculation of Net Sales of the
Combination Product within three (3) months after commencement of such negotiations, the dispute shall be submitted to final and
binding arbitration, as provided in Section 10.3

 
 
 
 
 
 
 
 
 
 
 
“Non-Breaching Party” has the meaning set forth in Section 9.2.1.

“Onxeo Indemnified Parties” means Onxeo and its Affiliates and their respective directors, officers, employees and agents.

“Parties” means Monopar and Onxeo and “Party” shall mean any of them.

“Patents” and “Patent Rights” means any patent applications, patents, author certificates, inventor certificates, utility models, and
all  foreign  counterparts  of  them  and  includes  all  divisionals,  renewals,  continuations,  continuations-in-part,  extensions,  reissues,
reexaminations, substitutions, confirmations, registrations, revalidations and additions of or to them, as well as any Supplementary
Protection Certificate, or any like form of protection.

“Person”  means  any  individual,  firm,  corporation,  partnership,  limited  liability  company,  trust,  business  trust,  joint  venture,
Regulatory Authority, association, or other entity.

“Phase III Trial”  means  a  human  clinical  trial  of  a  Licensed  Product,  which  trial  is  designed:  (a)  to  establish  that  the  Licensed
Product is safe and efficacious for its intended use; (b) to define warnings, precautions and adverse reactions that are associated with
the Licensed Product in the dosage range to be prescribed; and (c) consistent with 21 CFR § 312.21(c).

“Phase III Clinical Trial Report” means a full clinical study report in relation to a Phase III Trial which is written by or on behalf
of Monopar.

“Phase IV Trial” means (i) any clinical trial in humans conducted to satisfy a requirement of a Regulatory Authority in order to
maintain  a  Regulatory Approval  and  (ii)  any  clinical  trial  in  humans  conducted  after  the  first  Regulatory Approval  in  the  same
disease state for which the Licensed Product received Regulatory Approval in the Territory.

 
 
 
 
 
 
 
 
 
 
 
“Price Approval”   means,  in  those  countries  in  the  Territory  where  a  Regulatory Authority  may  approve  or  determine  pricing
and/or pricing reimbursement for pharmaceutical products, such approval or determination.

“Progress Report” means a written report produced by Monopar setting out brief details of: (i) the progress of development of the
Licensed Product; (ii) the progress of any applications for Regulatory Authorization and (where relevant) Price Approvals; and (iii)
the progress of and plans for marketing and sale of the Licensed Product.

“Prosecution”  means  the  preparation,  filing,  procuring,  and  maintenance  of  Patents,  such  as  before  national,  international,  and
regional  patent  offices,  including  any  interferences,  derivation  proceedings,  reissue  proceedings,  reexaminations,  and  post-grant
proceedings (such as inter partes reviews, post-grant reviews, and oppositions). When used as a verb, “Prosecute” means to engage
in Prosecution.

“Quarter” means any of the three (3) monthly periods commencing on the first day of any of the months of January, April, July,
and October in any year and “Quarterly” has a corresponding meaning.

“Receiving Party” has the meaning set forth in Section 8.1.

“Regulatory  Approval”  means,  with  respect  to  any  Licensed  Product  in  any  jurisdiction,  all  approvals  (including  Pricing
Approvals)  from  any  Regulatory Authority  necessary  for  the  development,  commercial  manufacture,  marketing  and  sale  of  the
Licensed Product in such jurisdiction in accordance with Laws.

“Regulatory Authority”  means  any  national  or  supranational  governmental  authority,  including  the  FDA,  EMEA,  or  Koseisho
(i.e.,  the  Japanese  Ministry  of  Health  and  Welfare,  or  any  successor  agency  thereto),  that  has  responsibility  in  countries  in  the
Territory over the Development and/or Commercialization of a Licensed Product.

“Regulatory Filings” means any and all regulatory applications and filings and associated correspondence made in order to obtain
Regulatory Approvals.

“Sublicensee” means a person to whom a sublicense is granted in accordance with Section 3.2 in respect of the whole or any part of
the rights granted under this Agreement or any person to whom such Sublicensee grants a sublicense in accordance with Section 3.2.

“Supplementary Protection Certificate” means a right based on a patent pursuant to which the holder of the right is entitled to
exclude  Third  Parties  from  using,  making,  having  made,  selling  or  otherwise  disposing  or  offering  to  dispose  of,  importing  or
keeping  the  product  to  which  the  right  relates,  such  as  supplementary  protection  certificates  in  Europe,  and  any  similar  right
anywhere in the world.

 
 
 
 
 
 
 
 
 
 
 
 
 
“Term” means the term of this Agreement determined in accordance with Section 9.1.4.

“Territory” means any and all countries in the world.

“Third Party” means any Person other than Monopar, Onxeo and their respective Affiliates and Sublicensees.

“Trademark”  means  any  word,  name,  symbol,  color,  designation,  or  device  or  any  combination  thereof,  whether  registered  or
unregistered,  including  any  trademark,  trade  dress,  service  mark,  service  name,  brand  mark,  trade  name,  brand  name,  logo,  or
business symbol.

“United States” or “U.S.” means the United States of America and all its territories and possessions.

“Valid Claim”  means  a  claim  within  an  issued  United  States  Patent  or  any  foreign  Patent  that  has  not  expired,  lapsed,  or  been
cancelled or abandoned, and that has not been dedicated to the public, disclaimed, or held unenforceable, invalid, or been cancelled
by a court or administrative agency of competent jurisdiction in an order or decision from which no appeal has been or can be taken,
including,  without  limitation,  through  opposition,  reexamination,  reissue  or  disclaimer;  provided  that,  on  a  country-  by-country
basis, a patent application or subject matter of a claim thereof pending for more than five (5) years from the earliest filing date to
which such patent application or claim is entitled shall not be considered to have any Valid Claim for purposes of this Agreement
unless and until a patent with respect to such application issues with such claim.

“Validive” or “Validive®” means the Licensed Product when used in association with the Trademark “Validive®” or “Clonidine
Lauriad®.”

“Validive Materials” means the Materials further described in SCHEDULE 4.

“Year” means a calendar year.

1.2

In this Agreement:

1.2.1

unless the context requires otherwise, all references to a particular Article, Section or Schedule shall be references to
that article, section or schedule, of or to this Agreement;

1.2.2

the table of contents and headings are inserted for convenience only and shall be ignored in construing this Agreement;

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission.
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

1.2.3

1.2.4

1.2.5

1.2.6

1.2.7

unless the contrary intention appears, words importing the masculine gender shall include the feminine and vice versa
and words in the singular include the plural and vice versa;

unless  the  contrary  intention  appears,  words  denoting  persons  shall  include  any  individual,  partnership,  company,
corporation, joint venture, trust, association, organization or other entity, in each case whether or not having separate
legal personality;

reference to any statute or regulation includes any modification or re-enactment of that statute or regulation, provided
that the modification or re-enactment does not diminish the rights or extend the obligations of any Party;

references  to  the  words  “include”  or  “including”  shall  be  construed  without  limitation  to  the  generality  of  the
preceding words;

where  either  Party’s  approval  or  consent  is  required  hereunder,  except  as  otherwise  specified  herein,  such  Party’s
approval or consent shall be a prior written consent which may be granted or withheld in such Party’s discretion, but
shall not be unreasonably conditioned, delayed or denied; and

1.2.8

all references to “dollars” shall be to the lawful currency of the United States of America.

2.

2.1

MONOPAR VALIDIVE OPTION; MONOPAR DEVELOPMENT AND COMMERCIALIZATION

Monopar Validive Option. Subject to the terms and conditions of this Agreement, including the payment of amounts to Onxeo as
and  when  such  amounts  become  due  under  this Agreement,  Onxeo  hereby  grants  to  Monopar  the  exclusive  right,  exercisable  at
Monopar’s sole discretion, in accordance with Sections 2.1.1 through 2.1.7, to elect to obtain an exclusive worldwide license under
Section 3.1  to  Develop,  Commercialize,  and  manufacture  Licensed  Products  under  the  terms  and  conditions  set  forth  in  this
Agreement (the “Monopar Validive Option”).

2.1.1 Monopar Validive Option Period. As from the Effective Date, Monopar shall:

(a)

have [***] to submit a new application for orphan drug designation in the United States;

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

(b)

from  the  time  of  receiving  feedback  from  the  orphan  drug  office  of  the  FDA,  have  [***]  to  prepare  the
materials for and request a meeting with the FDA;

(c)

from the date of the FDA meeting, have [***] to exercise the Monopar Validive Option.

The periods described in Sections 2.1.1(a), 2.1.1(b), and 2.1.1(c) shall together be known as the “Monopar Validive
Option Period”.

2.1.2 Monopar Validive Option Termination; Expiration. The Monopar Validive Option shall terminate or expire if:

(a)

Monopar  fails  timely  to  achieve  2.1.1(a),  2.1.1(b),  or  2.1.1(c)  without  first  having  exercised  the  Monopar
Validive  Option,  and  with  Onxeo  having  promptly  responded  to  information  requests  during  the  Monopar
Validive Option Period (any such period of delay by Onxeo shall cause an automatic equivalent time period
extension to the Monopar Validive Option Period); or

(b)

Monopar voluntarily terminates the Monopar Validive Option at any time and for any reason;

If  one  of  2.1.1(a),  2.1.1(b),  or  2.1.1(c)  is  not  satisfied,  or  if  Monopar  voluntarily  terminates  the  Monopar  Validive
Option at any time and for any reason:

(c)

(d)

the Monopar Validive Option shall terminate, and all rights to the Licensed Product shall remain with Onxeo
unencumbered by Monopar’s option; and

Onxeo shall have the right to request from Monopar a copy of all documents and correspondence exchanged
with the FDA, at no cost. Such documents shall be delivered within thirty (30) days of such request.

2.1.3 Monopar  Validive  Option  Exercise .  The  Monopar  Validive  Option  shall  only  be  exercisable  during  the  Monopar
Validive  Option  Period.  Monopar  shall  exercise  its  Monopar  Validive  Option,  if  at  all,  by  written  notice  to  Onxeo,
which notice shall make reference to this Agreement and Validive.

2.1.4 Monopar Rights on Exercise of the Monopar Validive Option. Following exercise of the Monopar Validive Option,
Monopar  shall  have  responsibility  for  Development  and  Commercialization  of  Licensed  Products,  subject  to  its
obligations  under  this Agreement.  Upon  Monopar’s  exercise  of  the  Monopar  Validive  Option,  Onxeo  shall  provide
Monopar with all information and data for Licensed Products and the Validive Materials, and Onxeo shall cooperate
with  Monopar  to  provide  a  smooth  transfer  of  such  information  and  data  and  the  Validive  Materials  as  soon  as
reasonably practical after exercise of the Monopar Validive Option.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
2.1.5

2.1.6

Early  Exercise  of  Monopar  Validive  Option.   Monopar  may  exercise  the  Monopar  Validive  Option  at  any  time
during the Monopar Validive Option Period upon written notice to Onxeo.

Onxeo’s  obligations  during  the  Monopar  Validive  Option  Period .  Onxeo  shall  authorize  Monopar  to  reference
Onxeo’s Validive IND as filed with the FDA, to submit a new orphan designation dossier for Validive, and to organize
a  meeting  with  the  FDA  regarding  Validive,  all  in  Monopar’s  Name.  Onxeo  shall  provide  Monopar  with  all
authorizations,  consents  and  rights  of  reference  that  Monopar  may  reasonably  request  in  order  to  (a)  facilitate  the
submission  of  the  new  orphan  designation  dossier  for  Validive,  and  (b)  request  for  and  conduct  a  meeting  with  the
FDA regarding Validive in Monopar’s name. Onxeo shall provide reasonable support to Monopar in connection with
the meeting with the FDA, without (except as the Parties may otherwise agree) any obligation for Onxeo to incur any
expenses. Onxeo shall not initiate any further Development efforts during this Monopar Validive Option Period.

2.1.7 Monopar’s obligations during the Monopar Validive Option Period . Monopar shall, at its own cost and expense,
re-file for orphan drug designation for Validive, and prepare all required materials, request and lead a meeting with the
FDA  regarding  development  of  Validive  in  the  Field  and  Territory  as  specifically  related  to  the  treatment  of  oral
mucositis. Without Onxeo’s permission, or unless required by applicable law, rules or regulations or request from a
stock  exchange  on  which  shares  are  listed,  Monopar  shall  make  no  public  statement  mentioning  Onxeo  and/or
Validive until the results of the FDA meeting are known.

2.1.8 Monopar’s Failure to Exercise the Monopar Validive Option . If Monopar does not exercise the Monopar Validive
Option during the Monopar Validive Option Period, then the Monopar Validive Option shall expire. All rights granted
to Monopar hereunder shall terminate, and Onxeo will thereafter have all such rights previously granted to Monopar,
for  Onxeo  to  Develop  and  Commercialize  Validive  at  Onxeo’s  sole  expense.  Monopar’s  rights  and  licenses  granted
hereunder to Validive shall terminate.

 
 
 
 
 
 
 
2.2

Monopar Development and Regulatory Responsibilities.

2.2.1

2.2.2

2.2.3

Development Responsibilities and Costs. Monopar, at its sole cost and expense, shall have responsibility for conducting,
and shall use Commercially Reasonable Efforts to conduct, all Development activities with respect to Licensed Products
following exercise of the Monopar Validive Option.

Regulatory Responsibilities and Costs. Promptly after Monopar’s exercise of the Monopar Validive Option, Onxeo shall
(a) assign to Monopar all Regulatory Filings for Licensed Products and, (b) upon Monopar’s request, assign to Monopar all
clinical  trial  or  other  subcontractor  agreements  relating  solely  to  Licensed  Products.  Following  exercise  of  the  Monopar
Validive Option, Monopar shall prepare, file, maintain, and own all Regulatory Filings and related submissions relating to
Licensed Products. Monopar shall have responsibility for, and shall prepare, all Regulatory Filings and related submissions
with respect to Licensed Products. At Monopar’s election, following exercise of the Monopar Validive Option, Monopar
shall be responsible for all safety reporting obligations globally with respect to such Licensed Products, and to take over
and maintain the global safety database for Licensed Products.

Record  Keeping;  Audit  for  Cause.  Each  Party  shall  maintain,  or  cause  to  be  maintained,  records  of  its  respective
Development and regulatory activities with respect to the Licensed Product in the Field in the Territory in sufficient detail
and in good scientific manner appropriate for patent and regulatory purposes, which shall  be  complete  and  accurate  and
shall  fully  and  properly  reflect  all  work  done  and  results  achieved  in  the  performance  of  its  respective  development
activities, and which shall be retained by such Party for at least ten (10) years after the termination of this Agreement, or
for such longer period as may be required by applicable law. Each Party shall have the right, during normal business hours,
upon at least ten (10) Business Days prior notice and without charge, to inspect and copy any such records, except in the
event of an audit for safety reason; provided, however, that, except in the event of an “audit for cause,” neither Party shall
have the right to conduct more than one such inspection in any twelve (12) month period. “Audit for cause” shall mean
any audit conducted by Onxeo in reason of any material deficiencies of Monopar or its Affiliates or Sublicensees relating to
the activities contemplated hereunder. 

 
 
 
 
 
 
 
2.3

2.4

Monopar  Commercialization  Responsibilities  and  Costs.  Monopar,  at  its  sole  cost  and  expense,  shall  have  responsibility  for
conducting, and shall use Commercially Reasonable Efforts to conduct, all Commercialization activities with respect to Licensed
Products following exercise of the Monopar Validive Option.

Manufacture  and  Supply.  Monopar,  at  its  sole  option  and  expense,  may  choose  to  continue  with  Onxeo’s  current  contract
manufacturing  partners  for  part  or  all  presently  sourced  manufacturing  or  manufacturing  related  activities,  including  API  and
Licensed  Product  manufacture,  for  part  or  all  of  the  Term.  In  such  event,  Monopar  shall  be  solely  responsible  for  negotiating
agreements with such manufacturing partners, it being understood and agreed that Onxeo’s sole obligation in this respect shall be to
introduce Monopar to such manufacturing partners. Under all circumstances, Monopar reserves the exclusive right to manufacture
and supply any and all Licensed Products.

2.5

Reporting and Right of Inspection.

2.5.1 Monopar  shall  provide  Onxeo  upon  Monopar’s  exercise  of  the  Monopar  Validive  Option  with  a  copy  of  an  initial
Development and Commercialization plan for the Licensed Products. Thereafter, Monopar shall provide Onxeo with
an  updated  Development  and  Commercialization  plan  for  each  Year  no  later  than  December  1  of  the  Year  for  each
Year. Additionally, every Year within thirty (30) days after Monopar’s annual financial reports have been completed,
but in no event later than April 1, the Parties shall meet by teleconference to discuss the progress in and results of the
Development and Commercialization of the Licensed Products during the previous year.

2.5.2

During the Term, Monopar shall also keep (and shall cause its Affiliates and Sublicensees to keep), and shall make
available  to  Onxeo  for  inspection  on  Onxeo’s  reasonable  demand  once  per  year  complete  and  accurate  records
pertaining  to  the  progress  in  and  results  of  the  Development  and  Commercialization  activities  in  the  Territory,  in
sufficient detail to permit Onxeo to ensure the satisfaction of Monopar’s contractual obligations hereunder.

 
 
 
 
 
 
 
 
2.6

Subcontracting

Monopar may have performed by subcontractors any activities required of Monopar hereunder. Monopar shall be solely responsible
for the performance by any of its subcontractors of Monopar’s obligations hereunder.

2.7

No Onxeo Financial Obligation

Except  as  expressly  provided  herein,  all  costs  relating  to  the  Development  and  Commercialization  of  the  Licensed  Product  after
Monopar’s exercise of the Monopar Validive Option shall be borne solely by Monopar, and Onxeo shall not be obligated to take any
action which may subject Onxeo to any cost, expense or liability with respect to other matters.

3.

3.1

LICENSES; TECHNOLOGY TRANSFER; EXCLUSIVITY

License to Monopar for Validive and Licensed Products.

3.1.1

3.1.2

Licensed  Intellectual  Property.  Subject  to  the  terms  and  conditions  of  this  Agreement,  Onxeo  hereby  grants  to
Monopar and its Affiliates the exclusive (even as to Onxeo and its Affiliates), worldwide license, with the right to grant
sublicenses under the Licensed Intellectual Property as described in Section 3.2 below, to use, sell, offer to sell, import,
make and have made, and otherwise Develop, Commercialize or manufacture Licensed Products during the Term, in
the  Territory  and  in  the  Field,  and  to  apply  for  Regulatory Approval  in  its  own  name  for  Licensed  Products  in  any
jurisdiction, such license to be effective upon Monopar’s exercise of the Monopar Validive Option and payment of the
License Fee.

License to Trademark . Subject to the terms and conditions of this Agreement, and at no additional cost to Monopar
or its Affiliates, Onxeo hereby grants to Monopar and its Affiliates an exclusive right and license during the Term, with
the  right  to  grant  sublicenses  as  described  in  Section 3.2  below,  to  the  Licensed  Trademarks,  such  Licensed
Trademarks  to  be  used  by  Monopar  solely  in  connection  with  the  Development  and  Commercialization  of  Licensed
Products  and  in  Monopar’s  corporate  communications  with  respect  thereto.  A  complete  list  of  such  Licensed
Trademarks, and existing registrations thereof, is attached as SCHEDULE 3. Monopar shall be in charge of securing
and maintaining the registration(s) of the Licensed Trademarks in the Territory in the name of Monopar and at its sole
cost and expense. Onxeo shall provide upon request, and at no cost to Onxeo, any assistance reasonably required by
Monopar.

 
 
 
 
 
 
 
 
 
 
 
 
3.2

3.3

3.4

3.5

Sublicenses.  Monopar  shall  have  the  right  to  grant  sublicenses  to  Third  Parties  without  the  prior  written  consent  of  Onxeo.
Monopar shall ensure that there are included in the terms of any sublicense substantially equivalent obligations and undertakings on
the part of the Sublicensee to those applying to Monopar in this Agreement. Any such sublicenses shall be without limitation on
Monopar’s  obligations  hereunder  and  Monopar  shall  be  solely  responsible  for  the  performance  by  any  of  its  Sub-Licenses  of
Monopar’s obligations hereunder.

Use of Names; Logo. Monopar, at its sole cost and expense, shall be responsible for the selection, registration, and maintenance of
all Trademarks which it employs in connection with its activities conducted pursuant to this Agreement, including those licensed
hereunder.

No other licenses. No license to use any Intellectual Property is granted to Monopar, or any Sublicensee, except the rights expressly
granted in this Agreement.

Technology Transfer by Onxeo after Exercise by Monopar of the Monopar Validive Option.  As soon as reasonably practical
after Monopar exercises its Monopar Validive Option, Onxeo shall transfer to Monopar, at no cost to Monopar, all Onxeo Licensed
Know-How and other information in Onxeo’s possession and Control or reasonably available to Onxeo that are necessary or useful
for  the  exercise  by  Monopar  and  its Affiliates  of  the  rights  granted  under  Section  3.1  with  respect  to  Licensed  Products  and  the
Validive Materials. Onxeo shall provide all reasonable assistance, including making its personnel reasonably available for meetings
or  teleconferences,  to  support  and  assist  Monopar,  at  no  cost  to  Onxeo,  in  the  Development  and  Commercialization  of  Licensed
Products, for a period of one (1) year after Monopar exercises its Monopar Validive Option. Within thirty (30) days of receiving the
License Fee, Onxeo shall:

3.5.1

transfer title to all IND’s for Licensed Products to Monopar;

3.5.2

assign Licensed Patents to Monopar;

3.5.3

assign Licensed Trademarks to Monopar;

3.5.4

3.5.5

submit  to  the  appropriate  authorities  the  necessary  paperwork  to  transfer  title  to  all  orphan  drug  designations  for
Licensed Products to Monopar;

transfer title in the Validive Materials to Monopar. Such materials are purchased ‘as is’ and “where is” and it shall be
Monopar’s responsibility to check the quality of such materials and that they are suitable for Monopar’s use thereof;
and

 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

3.5.6

provide Monopar with such information and Know-How relating to the manufacture of Validive as is relevant to the
efficient production of a sufficient quantity of Validive for clinical trials.

Exclusivity. During the Term, Onxeo will not engage in the research, discovery, optimization, development or commercialization
of  any  products  that  would  be  considered  a  Licensed  Product.  Notwithstanding  the  foregoing,  following  termination  of  this
Agreement, Onxeo shall be free to research, optimize, develop or commercialize, either on its own or with or through a Third Party,
any Licensed Product.

Acquisition of Rights. Should Monopar  wish,  at  any  time  during  the  Term,  to  acquire  all  right,  title,  and  interest  in  and  to  the
Licensed Intellectual Property, then held by Onxeo or any successor or permitted assignee, it may by giving notice to Onxeo request
that  Onxeo  enter  into  negotiations  in  this  regard. Any  such  acquisition  on  terms  and  conditions  (including  financial  terms  and
conditions) acceptable to each Party in its sole discretion.

FINANCIAL TERMS

Option Fee. [***] for entering into this Agreement.

License Fee.

3.6

3.7

4.

4.1

4.2

4.2.1 Monopar shall pay to Onxeo within ten (10) Business Days of exercising the Monopar Validive Option the sum of one
million  dollars  ($1,000,000.00),  the  “License Fee”.  The  License  Fee  is  a  one-time,  non-refundable,  non-creditable
payment.

4.3

Development and Sales Milestones.

4.3.1 Monopar shall pay the following payments (each, a “Milestone Payment”) to Onxeo upon the first occurrence only of

the following events (each, a “Milestone Event”) in relation to Licensed Product:

(a)

[***] upon [***] for a Licensed Product;

 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

(b)

(c)

(d)

(e)

(f)

(g)

(h)

(i)

(j)

t[***] upon [***] for a Licensed Product;

[***] upon [***] for a Licensed Product;

[***] upon [***] for a Licensed Product;

[***] upon [***];

[***] upon [***];

[***] upon [***];

[***] upon [***];

[***] upon [***]; and

[***] upon [***].

4.4

Royalty. Monopar shall pay royalties to Onxeo on a Licensed Product-by-Licensed Product and country-by-country basis until the
later of (1) the date when the Licensed Product is no longer within the scope of a Valid Claim of a Licensed Patent in the country of
sale or manufacture, (2) the expiry of any Extended Exclusivity Period in the relevant country, or [***] after the First Commercial
Sale of the Licensed Product in such country. The rate shall be [***] of Net Sales ex-US. For the United States, the rate shall be
[***] of Net Sales for the [***] starting from the First Commercial Sale of Licensed Product [***] of Net Sales for [***] after the
First Commercial Sale of Licensed Product, and [***] of Net Sales from [***] onward after the First Commercial Sale of Licensed
Product.  The  otherwise  applicable  rate  shall  be  reduced  by  [***]  on  a  Licensed  Product-by-Licensed  Product  and  country-by-
country basis if a royalty payment is due solely by reason of subparagraph (3) above.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
4.5

Payments.  All  payments  due  to  Onxeo  under  this  Agreement  shall  be  made  in  dollars  by  bank  wire  transfer  of  immediately
available  funds,  with  fees  of  the  transmitting  bank  paid  by  Monopar,  to  such  bank  account  as  Onxeo  may  notify  to  Monopar  in
writing from time to time.

4.6

Timings of Payments.

4.6.1

The payments due under Section 4.3 shall be payable within sixty (60) Business Days after when they are due.

4.6.2

4.6.3

Any royalties due pursuant to Section 4.4 shall be paid Quarterly within sixty (60) days of the end of each Quarter with
respect to Net Sales in such Quarter; and

After Monopar exercises the Monopar Validive Option, any costs or expenses related to the Prosecution, registration
or maintenance of Licensed Patents or Licensed Trademarks shall be paid by Monopar.

4.7

4.8

Taxes. All payments to Onxeo under this Agreement are expressed to be inclusive of value added tax (or any other sale goods tax)
howsoever arising.

Withholding. In the event that Monopar is required by law to withhold or pay to any government authority any taxes on behalf of
Onxeo, with respect to any payments to it hereunder, the amount payable to Onxeo shall not be increased such that the amount that
Onxeo  actually  receives  is  equal  to  the  amount  that  Onxeo  would  have  received  had  no  withholding  been  made.  Monopar  shall
furnish Onxeo with proper evidence of the taxes so paid and Onxeo shall be responsible for reclaiming such tax. Each Party shall
furnish  the  other  Party  with  appropriate  documents  to  secure  application  of  the  most  favorable  rate  of  withholding  tax  under
applicable Law. Notwithstanding the above, in the event that Monopar, by reason of an assignment of its rights hereunder or other
actions, causes Onxeo to be subject to withholding to which Onxeo is not subject as of the Effective Date, if Onxeo is unable to
reclaim such withholding tax payments, Monopar shall increase such payments made hereunder such that the amount that Onxeo
actually receives is equal to the amount that Onxeo would have received had no withholding been made.

 
 
 
 
 
 
 
 
 
 
4.9

Quarterly Report.  Within  forty-five  (45)  days  after  the  end  of  each  Quarter,  Monopar  shall  send  to  Onxeo  a  written  statement
detailing in respect of that Quarter (including a nil report if appropriate):

4.9.1

any Milestone Event achieved by it or any Sublicensee and any Milestone Payment which became due to Onxeo;

4.9.2

4.9.3

the  quantity  of  Licensed  Products  sold  or  otherwise  disposed  of  by  Monopar  at  the  wholesale  and  retail  levels,  its
Affiliates or any Sublicensees in the Territory;

the Net Sales in respect of Licensed Products in each country of the Territory in sufficient detail to allow Onxeo to
calculate  all  payments  due  under  Section 4.3  and  Section 4.4,  including,  without  limitation,  the  numbers  of  units  of
Licensed Products sold, the aggregate gross sales price for such units (in its native currency), and a description of the
amount  and  justification  for  an  any  deductions  made  to  such  aggregate  gross  sales  in  determining  the  reported  Net
Sales;

4.9.4

the aggregate Net Sales in respect of that Quarter for Licensed Product;

4.9.5

any currency conversions, showing the rates used; and

4.9.6

the amount of the royalties due to Onxeo in respect of that Quarter.

4.10

Interest. Where the payee does not receive payment within the relevant period of any sums that are finally determined to be due
and payable to it under this Agreement, interest shall accrue on the sum due and payable from the date payment was first due to the
date payment is made at the rate equivalent to an annual rate of two percent (2%) over the then current base rate of one (1) month
LIBOR,  calculated  on  a  daily  basis,  without  prejudice  to  payee’s  right  to  receive  payment  within  the  relevant  period,  provided
always  the  provisions  of  this  Section 4.10  shall  not  apply  to  the  extent  and  for  the  period  that  a  Force  Majeure  event  prevents
payment.

4.11

Accounts.

4.11.1 Monopar shall:

(a)

keep and, notwithstanding the expiry or termination of this Agreement, maintain for at least six (6) years, true
and  accurate  accounts  and  records  (including  any  underlying  documents  supporting  such  accounts  and
records) in sufficient detail to enable the amount of all sums payable under this Agreement to be determined;
and

 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

(b)

during the Term and thereafter until the said period of six (6) years relevant to the accounts and records has
expired, at the reasonable request of Onxeo and (subject to Section 4.11.2) at the expense of Onxeo from time
to  time,  permit  or  procure  permission  for  a  qualified  accountant  nominated  by  Onxeo  and  reasonably
acceptable to Monopar to inspect and audit those accounts and records.

4.11.2

If, following any inspection pursuant to Section 4.11.1(b), Onxeo's nominated accountant confirms to Onxeo that the
payments in respect of any Year fall short of the sums which were properly payable in respect of that Year under this
Agreement,  Onxeo  shall  send  a  copy  of  the  certificate  to  Monopar  and  Monopar  shall  (subject  to  Section 4.11.3)
within [***] of the date of receipt of the certificate pay the shortfall to Onxeo and, if the shortfall exceeds the greater
of  [***]  of  the  sum  properly  payable  or  [***],  Monopar  shall  also  reimburse  to  Onxeo  the  reasonable  costs  and
expenses of Onxeo in making the inspection, provided that costs and expenses so reimbursed shall not exceed [***] of
the shortfall so determined.

4.11.3

If  within  thirty  (30)  days  of  the  date  of  receipt  by  Monopar  of  any  certificate  produced  pursuant  to  Section 4.11.2
Monopar  notifies  Onxeo  in  writing  that  it  disputes  the  certificate,  the  dispute  shall  be  referred  for  resolution  by  an
independent expert jointly appointed by the Parties. If the Parties fail to jointly appoint an independent expert, shall be
finally resolved as provided in Article 10 (Dispute Resolution).

5.

5.1

INTELLECTUAL PROPERTY

Ownership of Arising Intellectual Property. All right, title and interest in and to any data, Patents, and extensions thereof, Know-
How and other information created, developed, or arising on or after the Effective Date and pertaining to Licensed Products shall be
solely  owned  by  Monopar.  For  the  avoidance  of  doubt, Arising  Intellectual  Property  generated  through  CMC,  Quality,  data,  or
clinical  observations  will  be  owned  by  Monopar.  As  of  the  Effective  Date,  at  its  own  cost,  Monopar  shall  have  the  full  and
exclusive benefit of, and right to apply for and obtain, patents or other similar forms of protection in respect of any part or parts of
the subject-matter of the Licensed Patents throughout the world, and the right to claim priority from the Licensed Patents.

5.2

Ownership of Clinical Data. Any Clinical Data generated by or on behalf of Monopar will be owned by Monopar.

 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

5.3

Intellectual Property Management.

5.3.1

Upon Monopar exercising its Monopar Validive Option, Monopar shall be responsible for, and shall bear or pay all
costs  and  expenses  related  to,  the  Prosecution  and  maintenance,  of  the  Licensed  Patents  and  Patents  claiming  any
Arising  Intellectual  Property,  and  the  registration,  renewal  and  maintenance  of  the  Licensed  Trademarks,  until  the
termination of this agreement. The Parties shall hold all information they know or acquire under this Section 5.3.1 that
is related to all such Patents as confidential, subject to the provisions of this Agreement.

5.3.2 Monopar  shall  keep  Onxeo  reasonably  informed  in  writing  as  to  the  Prosecution,  registration  and/or  maintenance
status of the Licensed Patents and Licensed Trademarks, and shall at Onxeo's request promptly provide Onxeo with a
copy  of  all  submissions  made  to  or  responses  received  from  the  relevant  patent  and  trademark  offices  and  all
correspondence  to  and  responses  received  from  the  relevant  patent  and  trademark  agents  in  relation  to  the  Licensed
Patents and Licensed Trademarks in each country of the Territory.

5.3.3

If Monopar elects not to file an application or otherwise not prosecute, register and/or maintain a Licensed Patent or
Licensed Trademark in any country of the Territory, Monopar shall notify Onxeo in writing promptly of its decision
and shall use its reasonable efforts to provide Onxeo with at least [***] notice prior to the expiration of any applicable
time bars. During the aforementioned [***] notice period, Monopar shall retain the responsibility for the Prosecution,
registration  and  maintenance  of  the  relevant  Licensed  Patent  or  Licensed  Trademark.  On  the  expiry  of  such  notice
period:

(a)

(b)

(c)

the  license  granted  pursuant  to  Section 3.1.1  shall  terminate  in  respect  of  that  country  and  that  relevant
Licensed  Product  for  any  relevant  Licensed  Patent  or  Licensed  Trademark  which  is  the  subject  of  such  a
notice;

Monopar shall, at Onxeo's request, promptly transfer to Onxeo (or any person nominated by Onxeo) any and
all  documents  and  information  in  Monopar's  control  relating  to  such  relevant  Licensed  Patent  or  Licensed
Trademark; and

Onxeo shall be free to Prosecute, register or abandon such relevant Licensed Patent or Licensed Trademark at
its  sole  discretion  and  to  grant  rights  thereunder  to  any  Person  without  further  reference  to  Monopar,  and
Onxeo shall thereafter be responsible for the expense of filing, prosecuting, registering and maintaining the
relevant Patents and Trademarks.

 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

5.3.4

Infringement.  Each  Party  will  promptly  notify  the  other  Party  in  writing  within  [***]  of  it  becoming  aware  of  any
infringement or suspected infringement by a Third Party of any of the Licensed Patents or Licensed Trademarks, or
any  unauthorized  use  of  the  Licensed  Know-How.  In  respect  of  the  Licensed  Patents,  Patents  claiming  Arising
Intellectual  Property  or  Licensed  Trademarks,  Monopar  may  (a)  at  its  own  cost  and  expense  and  subject  to  Section
5.3.5, bring proceedings in its own name or, if required by law, jointly with Onxeo, for infringement of the Licensed
Patents, Patents claiming Arising Intellectual Property or Licensed Trademarks; and (b) in any such proceedings settle
any  claim  for  infringement  of  the  Licensed  Patents,  Patents  claiming  Arising  Intellectual  Property  or  Licensed
Trademarks, provided that Monopar shall not, without the consent of Onxeo (which consent shall not be unreasonably
withheld, conditioned or delayed), enter into any settlement that (a) imposes any liability or obligation on Onxeo, or
(b) unreasonably reduces (i) the scope of the subject matter claimed in any Licensed Patent or (ii) the right to use any
Licensed Trademark. Should Monopar fail to initiate such infringement proceedings within ten (10) Business Days of
a demand therefor from Onxeo, Onxeo may do so at its own cost and subject to Section 5.3.5.

Monopar  shall  be  solely  responsible  for  the  defense  of  any  claims  that  its  activities  with  respect  to  Licensed  Products
infringe the Intellectual Property Rights of any Third Parties and shall bear and pay the costs and expenses thereof.

5.3.5

Entitlement  to  Proceeds.  Any  damages,  profits  and  awards  of  whatever  nature  recovered  by  a  Party  in  any
proceedings  referred  to  in  this  Section 5.3  shall  be  retained  solely  by  the  Party  directing  or  defending  such  suit  or
proceeding.  In  any  such  proceedings,  the  Party  bringing  or  defending  the  proceedings  (the  “Active Party”)  and  the
other  Party  (the  “Inactive  Party”)  will  bear  all  of  its  own  costs,  including  attorneys’  fees,  relating  to  such  legal
proceedings; provided that the Active Party shall bear the Inactive Party’s out-of-pocket expenses, including attorneys’
fees, incurred in complying with requests for cooperation made by the Active Party. The Inactive Party shall promptly
provide the Active Party with all documents and assistance as the Active Party  may  reasonably  require.  The Active
Party shall promptly provide the Inactive Party with notice of such proceedings and keep the Inactive Party regularly
informed  of  progress  and  promptly  provide  the  Inactive  Party  with  such  information  as  the  Inactive  Party  may
reasonably require including copies of all documents filed at court in the proceedings.

 
 
 
 
 
 
 
5.3.6

Confirmatory Patent Licenses. The Parties shall, at the request of either of them and at the expense of the requesting
Party  but  for  no  further  consideration,  enter  into  such  confirmatory  patent  licenses  relating  to  the  Licensed  Patents,
substantially in the form set out in SCHEDULE 5, as may be necessary or desirable in accordance with the relevant
Law and practice in each country in the Territory for registration at the relevant patent offices so that this Agreement
need  not  be  registered  or  recorded  unless  the  Parties  are  required  to  do  so  by  law.  If  there  are  any  inconsistencies
between the terms of any such confirmatory patent license and the provisions of this Agreement, this Agreement shall
prevail.

5.3.7

Patent Term Extension. With respect to Licensed Products, Onxeo grants Monopar the exclusive right to apply for, in
its  own  name  where  possible,  a  Supplementary  Protection  Certificate,  patent  term  extension  and/or  any  other
exclusivity in respect of any Licensed Product. At Monopar's reasonable request, Onxeo shall provide, at no cost to
itself, reasonable assistance to Monopar in connection with any such applications.

WARRANTIES AND LIMITATION OF LIABILITY

Warranty.

6.1.1

No reliance on warranties not in the Agreement.  Each Party acknowledges that, in entering into this Agreement, it
does not do so in reliance on any warranty or other provision except as expressly provided in this Agreement, and all
conditions, warranties, terms and undertakings implied by statute or otherwise are excluded from this Agreement to the
fullest extent permissible by law.

6.

6.1

6.1.2 Warranties. Each Party hereby warrants to the other Party that, as of the Effective Date:

(a)

it is duly organized and validly existing under the laws of its place of incorporation;

 
 
 
 
 
 
 
 
 
 
(b)

(c)

(d)

(e)

it has legal power, authority and right to enter into this Agreement;

the execution and performance by it of its obligations hereunder will not constitute a breach of, or conflict
with, its organizational documents nor any other material agreement or arrangement, whether written or oral,
by which it is bound;

it  has  full  corporate  power  and  authority  and  has  taken  all  corporate  action  necessary  to  enter  into  and
perform this Agreement, and that this Agreement has been duly authorized, executed, and delivered by that
Party; and

that this Agreement is a valid, binding, and legally enforceable obligation of that Party (subject to applicable
Laws  of  insolvency  and  bankruptcy  and  customary  conditions  and  limitations  as  concerns  equitable
remedies).

6.1.3

Additional Warranties of Onxeo. Onxeo warrants to Monopar at the Effective Date that:

(a)

(b)

(c)

(d)

(e)

(f)

it does not Control any Intellectual Property which is required for the use, import, development or sale of the
Licensed Product in the Territory which is not included in the licenses granted under this Agreement;

as  far  as  it  is  aware  there  is  no  pending  or  existing,  nor  has  Onxeo  received  notice  of  any  threatened,
litigation, actions, suits or claims against it before any court or governmental agency or other tribunal with
regard to the Licensed Intellectual Property;

as far as it is aware there are no oppositions, inter partes reviews, post grant reviews, derivation proceedings,
or interferences concerning the Licensed Patents pending before any governmental agency or other tribunal;

as far as it is aware there are no inventors of the Licensed Patents other than the inventors named therein;

it  is  the  legal  and  beneficial  owner  of  the  Licensed  Intellectual  Property  free  of  any  third  party  rights  or
encumbrances,

as far as it is aware all maintenance fees and annual payments due in respect of the Licensed Patents have
been paid;

 
 
 
 
 
 
 
 
 
 
 
 
 
 
(g)

(h)

(i)

(j)

as far as it is aware the use and possession of Validive or Validive Materials by Monopar shall not infringe
the rights (including without limitation any Intellectual Property Rights) of any third party;

it has not done anything whereby the whole or any part of the rights assigned or licensed under the Agreement
might be invalidated or registration of them refused;

it  has  not  and  will  not  enter  into  any  agreement  which  prevents  it  fulfilling  its  obligations  under  this
Agreement; and

as  far  as  it  is  aware  there  is  no  material  Know-How  that  is  necessary  or  useful  to  the  Development,
Commercialization or manufacturing of the Product that is not included in the Licensed Know-How.

6.1.4

No Further Representations or Warranties.  No director, officer, employee or agent of any Party or its Affiliates is
authorized to make any further representation or warranty to the other Party which is not contained in this Agreement,
and each Party acknowledges that it has not relied on any such oral or written representations or warranties.

Limitation of Liability. Neither Party, nor any Onxeo Indemnified Party, nor any Monopar Indemnified Party, nor their respective
directors, officers, employees and agents shall have any liability under or in connection with this Agreement whether under statute
or in tort (including but not limited to negligence), contract or otherwise in respect of: (i) any consequential or indirect loss; and/or
(ii) any loss of goodwill, profit, opportunity or contract, in either case even if advised in advance of the possibility of such losses.
However, nothing in this Agreement shall be construed as excluding or limiting the liability of any person for any liability which
cannot be limited or excluded by law, such as for personal injury or death. This Section 6.2 in no way shall be construed to limit the
liability of one Party to the other Party for milestones and royalties payable under the terms of this Agreement.

INDEMNITY AND INSURANCE

Indemnity.

7.1.1

Indemnification by Monopar.   Monopar  shall  indemnify,  defend  and  hold  harmless  the  Onxeo  Indemnified  Parties
against any and all Losses incurred or suffered by the Onxeo Indemnified Parties to the extent any Loss arises out of or
was caused by an act or omission of Monopar arising from or in connection with: (a) the exercise of the rights granted
in  Section 3.1  or  the  actions  of  Monopar  in  relation  to  its  Development,  Commercialization  or  manufacture  of  a
Licensed Product; or (b) in the performance of its obligations under this Agreement; except, in all cases, to the extent
that such Loss arises out of or was caused by the violation by Onxeo of a legal or contractual duty owed to Monopar.

6.2

7.

7.1

 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

7.1.2

7.1.3

Indemnification  by  Onxeo.  Onxeo  shall  indemnify,  defend  and  hold  harmless  the  Monopar  Indemnified  Parties
against any and all Losses incurred or suffered by the Monopar Indemnified Parties to the extent such Loss arises out
of or was caused by an act or omission of Onxeo in the performance of its obligations under this Agreement except, in
all cases, to the extent that such Loss arises out of or was caused by the violation by Monopar of a legal or contractual
duty owed to Onxeo.

Notification  of  Liabilities/Losses.  A  person  or  entity  entitled  to  indemnification  under  this  Section  7.1  (an
“Indemnified Party”) shall give prompt written notification [***] to the Party from whom indemnification is sought
(the “Indemnifying Party”) of the commencement or notice of any claim or proceeding relating to a Loss for which
indemnification may be sought or, if earlier, upon the assertion of any such Loss, (it being understood and agreed that
the failure by an Indemnified Party to give notice of a Loss of which it has knowledge as provided in this Section 7.1.3
within  [***]  shall  relieve  the  Indemnifying  Party  of  its  indemnification  obligation  under  this  Agreement).  The
Indemnifying Party shall be liable for any reasonable legal fees and expenses subsequently incurred in connection with
the defense of such Loss after receiving such notice. The Parties shall thereafter keep the other Party informed of any
Losses.

(a)

In  the  case  of  a  Loss  for  which  Onxeo  seeks  indemnification  under  Section 7.1.1,  Onxeo  shall  permit
Monopar  to  direct  and  control  the  defense  of  the  Loss  and  shall  provide  such  reasonable  assistance  as  is
reasonably  requested  by  Monopar  (at  Monopar’s  cost)  in  the  defense  of  the  Loss;  provided  that  nothing  in
this Section 7.1.3(a) shall permit Monopar to make any admission on behalf of Onxeo, or to settle any claim
or  litigation  which  would  impose  any  financial  obligations  on  Onxeo  without  the  prior  written  consent  of
Onxeo, such consent not to be unreasonably conditioned, withheld, or delayed.

 
 
 
 
 
 
 
7.2

8.

8.1

(b)

In  the  case  of  a  Loss  for  which  Monopar  seeks  indemnification  under  Section 7.1.2,  Monopar  shall  permit
Onxeo  to  direct  and  control  the  defense  of  the  Loss  and  shall  provide  such  reasonable  assistance  as  is
reasonably requested by Onxeo (at Onxeo’s cost) in the defense of the Loss, provided always that nothing in
this Section 7.1.3(b) shall permit Onxeo to make any admission on behalf of Monopar, to settle any claim or
litigation  which  would  impose  any  financial  obligations  on  Monopar  without  the  prior  written  consent  of
Monopar, such consent not to be unreasonably conditioned, withheld or delayed.

Insurance. Each Party, at its own expense, and reasonably prior to Commencement of any human being dosed with the Licensed
Product,  shall  put  in  place  and  thereafter  maintain,  at  its  own  cost,  insurance  through  a  reputable  insurance  company.  For
clarification,  such  insurance  shall  be  maintained  for  an  amount  within  the  range  that  is  customary  for  similar  products  in  the
Territory, on a country-by-country basis, where they are sold.

CONFIDENTIALITY

Nondisclosure.  Each  Party  agrees  that,  during  the  Term  and  for  a  period  of  seven  (7)  years  thereafter,  a  Party  (the  “Receiving
Party”) receiving Confidential Information of the other Party (the “Disclosing Party”) (or that has received any such Confidential
Information from the other Party prior to the Effective Date) shall (a) maintain in confidence such Confidential Information using
not less than the efforts such Receiving Party uses to maintain in confidence its own proprietary industrial information of similar
kind and value, (b) not disclose such Confidential Information to any Third Party without the prior written consent of the Disclosing
Party, except for disclosures expressly permitted below, and (c) not use such Confidential Information for any purpose except those
permitted by this Agreement (it being understood that this clause (c) shall not create or imply any rights or licenses not expressly
granted under this Agreement).

8.2

Exceptions.  The  obligations  in  Section 8.1  shall  not  apply  with  respect  to  any  portion  of  the  Confidential  Information  that  the
Receiving Party can show by competent written proof:

8.2.1

is publicly disclosed by the Disclosing Party, either before or after it is disclosed to the Receiving Party hereunder;

 
 
 
 
 
 
 
 
 
 
8.2.2

8.2.3

8.2.4

8.2.5

was  known  to  the  Receiving  Party  or  any  of  its  Affiliates,  without  any  obligation  to  keep  it  confidential  or  any
restriction on its use, prior to disclosure by the Disclosing Party;

is subsequently disclosed to the Receiving Party or any of its Affiliates by a Third Party lawfully in possession thereof
and without any obligation to keep it confidential or any restriction on its use;

is  published  by  a  Third  Party  or  otherwise  becomes  publicly  available  or  enters  the  public  domain,  either  before  or
after it is disclosed to the Receiving Party; or

is  independently  developed  by  or  for  the  Receiving  Party  or  its Affiliates  without  reference  to  or  reliance  upon  the
Disclosing Party’s Confidential Information.

8.3

Authorized  Disclosure.  The  Receiving  Party  may  disclose  Confidential  Information  belonging  to  the  Disclosing  Party,  and
Confidential Information deemed to belong to both Parties under the terms of this Agreement, to the extent (and only to the extent)
such disclosure is reasonably necessary in the following instances:

(a)

(b)

(c)

(d)

Prosecuting Patents;

Regulatory Filings and obtaining Regulatory Approvals;

Prosecuting or defending litigation, including responding to a subpoena in a third party litigation;

Subject  to  Section 8.4,  complying  with  Laws  (including  the  rules  and  regulations  of  the  Securities  and
Exchange Commission or any securities exchange) and with judicial process, if in the reasonable opinion of
the Receiving Party’s counsel, such disclosure is necessary for such compliance; and

(e)

Disclosure, solely on a “need to know basis,” to Affiliates.

8.4

Securities  Filings.  In  the  event  either  Party  proposes  to  file  with  the  Securities  and  Exchange  Commission  or  the  securities
regulators of any state or other jurisdiction a registration statement or any other disclosure document which describes or refers to the
terms  and  conditions  of  this Agreement  under  the  Securities Act  of  1933,  as  amended,  the  Securities  Exchange Act  of  1934,  as
amended, or any other applicable securities Law, the Party shall notify the other Party of such intention and shall provide such other
Party with a copy of relevant portions of the proposed filing prior to such filing (and any revisions to such portions of the proposed
filing  a  reasonable  time  prior  to  the  filing  thereof),  including  any  exhibits  thereto  relating  to  the  terms  and  conditions  of  this
Agreement,  and  shall  use  reasonable  and  diligent  efforts  to  obtain  confidential  treatment  of  the  terms  and  conditions  of  this
Agreement that such other Party requests be kept confidential, and shall only disclose Confidential Information that it is advised by
counsel  that  it  legally  is  required  to  disclose.  No  such  notice  shall  be  required  under  this  Section 8.4  if  the  description  of  or
reference to this Agreement contained in the proposed filing has been included in any previous filing made by either Party hereunder
or otherwise approved by the other Party.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
8.5

8.6

8.7

9.

9.1

Publications. After  exercise  of  the  Monopar  Validive  Option,  Monopar  shall  have  the  exclusive  right  to  publish  or  present  data
and/or results relating to Licensed Products.

Effect of Disclosure. The Receiving Party agrees that the disclosure of the Disclosing Party's Confidential Information without the
express  written  consent  of  the  Disclosing  Party  may  cause  irreparable  harm  to  the  Disclosing  Party,  and  that  any  breach  or
threatened breach of this Agreement by the Receiving Party may entitle the Disclosing Party to injunctive relief, in addition to any
other legal remedies available to it, in any court of competent jurisdiction.

Relationship to Confidentiality Agreement.  This Agreement supersedes the Mutual Confidential Disclosure Agreement between
the  Parties  executed  as  of  January  19,  2016;  provided  that  all  “Confidential  Information”  disclosed  or  received  by  the  Parties
thereunder  shall  be  deemed  “Confidential  Information”  hereunder  and  shall  be  subject  to  the  terms  and  conditions  of  this
Agreement.

TERM AND TERMINATION

Term; Expiration.  This Agreement  shall  become  effective  as  of  the  Effective  Date  and  shall  continue  in  force  and  effect  until
expiration as described in this Section 9.1, unless earlier terminated pursuant to Section 9.2, 9.3, or 9.4, and shall expire as follows:

9.1.1

9.1.2

on  a  Licensed  Product-by-Licensed  Product  and  country-by-country  basis,  on  the  date  of  expiration  of  all  payment
obligations of Monopar under this Agreement with respect to each Licensed Product in each country, as applicable;

in its entirety upon the expiration of all payment obligations under this Agreement with respect to the last Licensed
Product Commercialized in the last country in the Territory; or

 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

9.1.3

9.1.4

if Monopar does not exercise the Monopar Validive Option in accordance with Section 2.1, then this Agreement will
terminate in its entirety upon the expiration of the Monopar Validive Option.

The period beginning on the Effective Date and ending on expiration or termination of this Agreement, or as the case
may be, until the date of expiration or termination of a Licensed Product, shall be the “Term” of this Agreement in its
entirety or with respect to a given Licensed Product, as applicable.

9.2

Termination for cause.

9.2.1 Material Breach. Either Party (the “Non-Breaching Party”) may, without prejudice to any other remedies available
to it at law or in equity, terminate this Agreement in its entirety, or terminate any Licensed Product in any portion of
the Territory that is affected by a material breach, in its sole discretion, in the event the other Party (the “Breaching
Party”)  has  materially  breached  this Agreement,  and  such  breach,  if  curable,  has  continued  for  [***]  (the  “Cure
Period”)  after  written  notice  thereof  is  provided  to  the  Breaching  Party  by  the  Non-Breaching  Party,  such  notice
describing the alleged material breach in sufficient detail to put the Breaching Party on notice; provided that, if such
breach is not susceptible to cure within the Cure Period, then, the Non-Breaching Party’s right to termination shall be
suspended only if and for so long as the Breaching Party has provided to the Non-Breaching Party a written plan that is
reasonably  calculated  to  effect  a  cure  and  such  plan  is  reasonably  acceptable  to  the  Non-Breaching  Party,  and  the
Breaching Party commits to and does carry out such plan. In all circumstances, if within the Cure Period the Breaching
Party pays the Non-Breaching Party an amount equal to the costs, damages, expenses and losses incurred as a result of
the material breach, the material breach shall be considered cured.

9.2.2

Disagreement  as  to  Material  Breach;  Cure  Period.   If  the  Parties  reasonably  and  in  good  faith  disagree  as  to
whether there has been a material breach, the Party that disputes that there has been a material breach may contest the
allegation  in  accordance  with  Article 10  (Dispute  Resolution).  Notwithstanding  the  preceding  sentence,  the  Cure
Period for any allegation made in good faith as to a material breach under this Agreement will run from the date that
written notice thereof was first provided to the Breaching Party by the Non-Breaching Party. The right of either Party
to terminate this Agreement, in whole or in part, as provided in this Section 9.2, shall not be affected in any way by
such Party’s waiver or failure to take action with respect to any previous default. It is understood and acknowledged
that, during the pendency of such a dispute, all of the terms and conditions of this Agreement shall remain in effect,
and the Parties shall continue to perform all of their respective obligations under this Agreement.

 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

9.3

Monopar Unilateral Termination Rights.

9.4

9.3.1

9.3.2

Termination of Agreement in Its Entirety.  Monopar may, in its sole discretion, exercisable at any time during the
Term, terminate this Agreement in its entirety for any reason or no reason at all, upon [***] written notice to Onxeo.

Termination on a Licensed Product-by-Licensed Product basis. Monopar may, in its sole discretion, exercisable at
any time during the Term, terminate this Agreement on a Licensed Product-by-Licensed Product basis for any reason or
no reason at all, upon [***] written notice to Onxeo.

Termination for Insolvency. To the extent permitted under Law, either Party may terminate this Agreement, (a) if, at any time, the
other  Party  files  in  any  court  or  agency  pursuant  to  any  statute  or  regulation  of  any  state  or  country,  a  petition  in  bankruptcy  or
insolvency or for reorganization or for an arrangement or for the appointment of a receiver or trustee of the Party or of substantially
all of its assets, or (b) if the other Party is served with an involuntary petition against it, filed in any insolvency proceeding, and such
petition  shall  not  be  dismissed  within  [***]  after  the  filing  thereof,  or  (c)  if  the  other  Party  shall  propose  or  be  a  party  to  any
dissolution  or  liquidation,  or  (d)  if  the  other  Party  shall  make  an  assignment  of  substantially  all  of  its  assets  for  the  benefit  of
creditors.  Each  Party  agrees  to  give  the  other  Party  prompt  notice  of  the  foregoing  events  giving  rise  to  termination  under  this
Section 9.4. All rights and licenses granted under or pursuant to any section of this Agreement are and shall otherwise be deemed to
be  for  purposes  of  Section  365(n)  of  Title  11,  United  States  Code  (the  “Bankruptcy  Code”)  licenses  of  rights  to  “intellectual
property”  as  defined  in  Section  101(35A)  of  the  Bankruptcy  Code.  The  Parties  shall  retain  and  may  fully  exercise  all  of  their
respective rights and elections under the Bankruptcy Code. All materials required to be delivered by the non-bankrupt Party under
this Agreement (including all manufacturing information), and all materials relating to the Licensed Intellectual Property that, in the
course  of  dealing  between  the  Parties  under  this Agreement,  are  or  would  be  customarily  delivered,  shall  be  considered  to  be
“embodiments” of such intellectual property for purposes of Section 365(n) of the Bankruptcy Code. Upon the bankruptcy of any
Party, the non-bankrupt Party shall further be entitled to a complete duplicate of, or complete access to, any Intellectual Property
licensed to the non-bankrupt Party, and such, if not already in its possession, shall be promptly delivered to the non-bankrupt Party,
unless  the  bankrupt  Party  elects  to  continue,  and  continues,  to  perform  all  of  its  obligations  under  this Agreement. All  written
agreements entered into in connection with the Parties’ performance under this Agreement from time to time shall be considered
agreements “supplementary” to this Agreement for purposes of Section 365(n) of the Bankruptcy Code.

 
 
 
 
 
 
 
 
9.5

Consequences  of  Expiration  or  Termination.  All  of  the  following  effects  of  expiration  or  termination,  as  applicable,  are  in
addition to the other rights and remedies that may be available to the Parties at law or in equity.

9.5.1

9.5.2

Consequences of Expiration of the Term.  Upon expiration of the  Term,  as  determined  on  a  Licensed  Product-by-
Licensed  Product  and  country-by-country  basis,  Monopar  shall  have  an  exclusive,  fully-paid,  royalty-free,  perpetual
right and license, with the right to grant sublicenses, under all Licensed Patents and Licensed Know-How to use, sell,
offer to sell, import, make and have made any Licensed Product in the Field and in the Territory.

Consequences of Termination of this Agreement by Monopar Pursuant to Section  9.3.1 or by Onxeo Pursuant
to Section 9.1.3, 9.2.1, or 9.4. In the event of a termination of this Agreement in its entirety by Monopar pursuant to
Section 9.3.1 or a termination of this Agreement in its entirety by Onxeo pursuant to Section 9.1.3 (failure to exercise
the Monopar Validive Option) or 9.2.1 (for cause) or 9.4 (insolvency):

(a)

(b)

(c)

notwithstanding anything contained in this Agreement to the contrary, all rights and licenses granted herein to
Monopar with respect to any Licensed Products shall terminate;

all  payment  obligations  hereunder  shall  terminate,  other  than  those  that  are  accrued  and  unpaid  as  of  the
effective date of such termination;

should Onxeo so demand, Monopar shall assign to Onxeo any Patents or Know-How (other than the Licensed
Patents and Licensed Know-How) Controlled by Monopar that Monopar both actually uses and are necessary
to Develop or Commercialize Licensed Products and shall negotiate in good faith with Onxeo the amount of
contingent milestone and/or royalty payments which shall be the sole consideration for such assignment. The
transfer of such rights to Onxeo shall be automatically effective upon Onxeo’s demand even if the amount of
each milestone and/or royalty payments are not determined. In the event that the Parties are not able to agree
amount  of  milestone  and/or  royalty  payments  within  three  (3)  months  after  commencement  of  such
negotiations, the dispute shall be submitted to final and binding arbitration, as provided in Section 10.3

 
 
 
 
 
 
 
 
 
(d)

(e)

(f)

Monopar  shall  promptly  either,  at  Onxeo’s  election,  return  to  Onxeo  or  destroy,  at  no  cost  to  Onxeo,  all
Onxeo  Licensed  Know-How,  Materials,  and  other  data  and  information  transferred  by  Onxeo  to  Monopar,
including all Onxeo Licensed Know-How, Validive Materials, and other information transferred to Monopar
pursuant to Section 3.5; and Onxeo, except as provided in Section 9.5.2(e) or 9.5.2(f) shall promptly either, at
Monopar’s  election,  return  to  Monopar  or  destroy,  at  no  cost  to  Monopar,  all  Monopar  Confidential
Information;

Monopar will provide, as soon as reasonably practical after Monopar’s notice of such termination, to Onxeo,
to the extent permitted under any applicable Third Party contract, (i) any information, Validive Materials, and
data  for,  including  copies  of  all  clinical  study  data  and  results,  and  all  other  information,  and  the  like
developed by or for the benefit of Monopar directly and solely relating to Licensed Products, and (ii) other
documents  to  the  extent  directly  and  solely  related  to  the  Licensed  Products  that  are  necessary  in  the
the  Territory.
continued  Development  and  Commercialization  of  Licensed  Products 
Notwithstanding  the  foregoing,  this  Section 9.5.2(e)  shall  not  apply  in  the  case  of  a  termination  of  this
Agreement  in  its  entirety  by  Onxeo  pursuant  to  Section 9.1.3  (failure  to  exercise  the  Monopar  Validive
Option); and

throughout 

should Onxeo so demand, Monopar shall assign to Onxeo any and all title to Regulatory Approvals directly
and solely related to Licensed Products (including orphan drug designations), all title to Licensed Intellectual
Property  or  registrations  thereof,  and  Regulatory  Filings  directly  and  solely  related  to  Licensed  Products;
provided that this Section 9.5.2(f) shall also apply in the case of a termination of this Agreement in its entirety
by Onxeo pursuant to Section 9.1.3 (failure to exercise the Monopar Validive Option).

 
 
 
 
 
 
9.5.3

Consequences  of  Termination  by  Monopar  Pursuant  to  Section   9.2.1  or  9.4.  In  the  event  of  termination  by
Monopar of this Agreement in its entirety or with respect to a Licensed Product pursuant to Section  9.2 (for cause) or
pursuant to Section 9.4 (insolvency):

(a)

(b)

(c)

all licenses granted to Monopar with respect to Licensed Products shall continue in full force in perpetuity;

all  future  milestones  and  royalties  payable  by  Monopar  under  this  Agreement  shall  be  reduced  by  a
percentage agreed to by Monopar and Onxeo. In the event the Parties are not able to agree on the percentage
amount within three (3) months after commencement of such negotiations, the dispute shall be submitted to
final and binding arbitration as provided in Section 10.3; and

Onxeo shall promptly either, at Monopar’s election, return to Monopar or destroy, at no cost to Monopar, all
Monopar  Confidential  Information,  materials,  and  other  data  and  information  transferred  by  Monopar  to
Onxeo.

9.5.4

Sell-Down. If Monopar, its Affiliates or Sublicensees at termination of this Agreement possess Licensed Product, have
started the manufacture thereof or have accepted orders therefor, Monopar, its Affiliates or Sublicensees shall have the
right,  for  up  to  one  (1)  year  following  the  date  of  termination,  to  sell  their  inventories  thereof,  complete  the
manufacture  thereof  and  Commercialize  such  fully-manufactured  Licensed  Product,  in  order  to  fulfill  such  accepted
orders or distribute such fully-manufactured Licensed Product, but only in the ordinary course of business and on the
same terms and conditions of sale as previously applied and subject to the obligation of Monopar to pay Onxeo any
and all payments as provided in this Agreement.

9.6

Provisions  to  continue  on  termination.  The  termination  of  this Agreement  howsoever  arising  will  be  without  prejudice  to  the
rights and duties of either Party accrued prior to termination. The following Articles will continue to be enforceable notwithstanding
termination: Articles 6, 8, 10 and 11 and Sections 4.5, 4.6, 4.7, 4.8, 4.9, 4.10, 4.11, 5.1, 5.2, 7.1 and 9.5 inclusive.

 
 
 
 
 
 
 
 
 
10.

DISPUTE RESOLUTION

10.1

10.2

The Parties recognize that disputes as to certain matters arising under this Agreement may arise from time-to-time. It is the objective
of the Parties to seek to resolve any disputes arising under this Agreement in an expedient manner and, if at all possible, without
resort  to  litigation,  and  to  that  end  the  Parties  agree  to  abide  by  the  procedures  set  forth  in  this  Section 10  to  resolve  any  such
disputes. The Parties initially shall attempt to resolve any issues through good faith negotiations in the spirit of mutual cooperation
between senior managers of the Parties with authority to resolve the dispute, for a period of thirty (30) days after receipt of the first
notice by either Party requesting negotiations. Should any issue not be timely resolved by good faith negotiations, any dispute with
respect thereto shall be submitted to final and binding arbitration, as provided below.

Any controversy or claim arising out of or relating to this Agreement, or the interpretation or breach thereof, shall be resolved by
final  and  binding  arbitration  administered  by  the  International  Centre  for  Dispute  Resolution  in  accordance  with  its  International
Arbitration Rules as then in force. The number of arbitrators shall be three (3), or one (1) if the amount in controversy is less than
one million dollars ($1,000,000), and the place of arbitration shall be New York County, New York. When three (3) arbitrators are
required  based  on  the  amount  in  controversy,  each  Party  shall  appoint  an  arbitrator  and  the  Parties  shall  mutually  agree  on  the
appointment  of  the  third  arbitrator.  When  one  (1)  arbitrator  is  required  based  on  the  amount  in  the  controversy,  the  Parties  shall
mutually agree on the appointment of an arbitrator within one (1) month of submission of the request for arbitration, failing which
the  sole  arbitrator  shall  be  selected  by  the  International  Centre  for  Dispute  Resolution.  The  language  of  the  arbitration  shall  be
English. The arbitrator(s) shall be entitled to award interim and conservatory relief to the fullest extent permitted by New York law,
shall apply the International Bar Association Rules on the Taking of Evidence in International Commercial Arbitration as now in
effect, and shall otherwise apply New York procedural law.

10.3

In the event that the Parties are unable to complete negotiations as described in the definition of “Net Sales”, in Section  9.5.2(c) or
in Section 9.5.3(b) within the time period there indicated, each Party shall, no later than the last day of such period, submit its final
and  best  offer  to  the  other  Party,  and  a  single  arbitrator  appointed  pursuant  to  Section 10.2  (and  without  further  negotiations  as
provided in Section 10.1), whose sole authority shall be to select one of the final offers so submitted.

 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

11.

MISCELLANEOUS

11.1

11.2

11.3

11.4

Severability. If any one or more of the provisions of this Agreement is held to be invalid or unenforceable, the provision shall be
considered severed from this Agreement and shall not serve to invalidate any remaining provisions hereof. The Parties shall make a
good  faith  effort  to  replace  any  invalid  or  unenforceable  provision  with  a  valid  and  enforceable  one  such  that  the  objectives
contemplated by the Parties when entering this Agreement may be realized.

Notices. All notices shall be in writing and sent by hand, email, or recorded delivery and shall be deemed to be properly served: (i) if
sent by hand, when delivered at the relevant address; (ii) if sent by recorded delivery, three (3) Business Days after posting; (iii) if
sent by email, when transmitted, provided a confirmatory copy is sent by post within twenty four (24) hours of transmission, and
shall be sent to the following addresses or email address as may be amended by the relevant Party in writing:

If to Onxeo:

Onxeo S.A.
49, boulevard du Général Martial Valin, 1st Floor
75015 Paris, France
Attention: Judith Greciet
email: [***]

If to Monopar:

Monopar Therapeutics Inc.
598 Rockefeller Rd
Lake Forest, IL 60045
Attention: Chandler Robinson
email: [***]

Variation.  No  variation,  modification,  amendment,  extension  or  release  from  any  provision  of  this Agreement  shall  be  effective
unless it is in writing, signed by both Parties.

Force Majeure. Except for the payment of money, neither Party shall be liable for delay or failure in the performance of any of its
obligations  hereunder  if  such  delay  or  failure  is  due  to  causes  beyond  its  reasonable  control,  including  acts  of  God,  fires,
earthquakes, acts of war, terrorism, or civil unrest (“Force Majeure”); provided, however, that the affected Party promptly notifies
the other Party and further provided that the affected Party shall use its Commercially Reasonable Efforts to avoid or remove such
causes of non-performance and to mitigate the effect of such occurrence, and shall continue performance with the utmost dispatch
whenever such causes are removed. When such circumstances arise, the Parties shall negotiate in good faith any modifications of
the terms of this Agreement that may be necessary or appropriate in order to arrive at an equitable solution.

 
 
 
 
 
 
 
 
 
 
 
 
 
11.5

11.6

Entire Agreement.   This Agreement  and  the  attached  Schedules  constitutes  the  entire  agreement  between  the  Parties  as  to  the
subject  matter  of  this  Agreement,  and  supersedes  and  merges  all  prior  and  contemporaneous  negotiations,  representations,
agreements and understandings regarding the same.

Further Assurance. Each Party hereby undertakes to do all such other acts and things, and execute and provide all such documents
at the other Party's request and cost as may be necessary or desirable to give effect to the purposes of this Agreement.

11.7 Waiver.  No  relaxation,  forbearance,  waiver  or  indulgence  by  either  Party  in  enforcing  any  of  the  terms  or  conditions  of  this
Agreement or the granting of time by either Party to the other shall prejudice, affect or restrict the rights and powers of such Party,
unless contained in a writing signed by the Party charged with such waiver. The waiver of any breach of any term or any condition
of this Agreement shall not be construed as a waiver of any subsequent breach of a term or condition of the same or of a different
nature.

11.8

11.9

Relationship of the Parties. Each Party is an independent contractor under this Agreement. Nothing contained herein is intended or
is to be construed so as to constitute Onxeo and Monopar as partners, agents or joint venturers. Neither Party shall have any express
or implied right or authority to assume or create any obligations on behalf of or in the name of the other Party or to bind the other
Party  to  any  contract,  agreement  or  undertaking  with  any  Third  Party.  There  are  no  express  or  implied  third  party  beneficiaries
hereunder.

Execution.  This  Agreement  may  be  executed  in  any  one  or  more  number  of  counterpart  agreements,  and  as  scanned  email
attachments, and all signatures and counterparts so exchanged shall be considered as original and shall be deemed to form part of
and together constitute this Agreement.

11.10 Assignment.  Neither  Party  may,  without  the  consent  of  the  other  Party,  assign  or  transfer  any  of  its  rights  and  obligations
hereunder; provided that no such consent is required for an assignment or transfer to an Affiliate of or to a successor in interest by
reason of merger or consolidation or sale of all or substantially all of the assets of such Party relating to the subject matter of this
Agreement; provided further that (a) with respect to an assignment to a successor in interest, such assignment includes all rights and
obligations under this Agreement, (b) such successor in interest or Affiliate shall have agreed as of such assignment or transfer to be
bound by the terms of this Agreement in a writing provided to the non-assigning Party, and (c) where this Agreement is assigned or
transferred to an Affiliate, the assigning Party remains responsible for the performance of this Agreement. Subject to the foregoing,
this Agreement shall inure to the benefit of and be binding on the Parties’ successors and assigns. Any assignment or transfer in
violation of the foregoing shall be null and void and wholly invalid, the assignee or transferee in any such assignment or transfer
shall  acquire  no  rights  whatsoever,  and  the  non-assigning,  non-transferring  Party  shall  not  recognize,  nor  shall  it  be  required  to
recognize, such assignment or transfer.

 
 
 
 
 
 
 
 
 
11.11

Public Announcements. The text of any press release, shareholders’ report or other communication to be published or disclosed in
any way naming the other Party or this Agreement, other than as required by law or by any regulatory or government authority, shall
be submitted to the other Party at least seven (7) days in advance of publication or disclosure for approval, such approval not to be
unreasonably  withheld;  provided  that  insofar  as  a  disclosure  repeats  or  restates  a  prior  public  disclosure  permitted  by  this
Agreement, such disclosure need not be submitted to the other Party for approval.

11.12 Governing Law.   This Agreement  shall  be  governed  by  and  construed  in  accordance  with  the  laws  of  the  State  of  New  York

without giving effect to the principles of conflicts of laws (other than Section 5-1401 of the New York General Obligations Law).

[Signature Page Follows]

 
 
 
 
 
 
 
 
 
IN WITNESS whereof this Agreement has been executed by duly authorized officers of the Parties on the day first above written.

For and on behalf of ONXEO S.A.

Signed by:    

/s/ Judith Greciet

Name:                                 Judith Greciet

Title:                                  CEO

For and on behalf of MONOPAR THERAPEUTICS INC.

Signed by:

/s/ Chandler D. Robinson

Name:     

Title:    

Chandler D. Robinson

CEO

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

SCHEDULE 1

LICENSED PATENTS

                                                                         Validive patent status 26/04/20

 Onxeo's Reference
 [***]

 Country/Region 
[***] 

 Application Number
[***] 

 Grant Date
[***] 

 Patent Number
[***] 

  Onxeo's Reference
 [***]

  Country/Region 
 [***]

 Application Number
 [***]

 Grant Date
 [***]

  Patent Number
 [***]

 Status
[***] 

Status
 [***]

 
 
 
 
 
 
 
 
 
 
 
SCHEDULE 2

LICENSED KNOW-HOW

The Licensed Know-How shall include all regulatory and technical documents that the personnel of Onxeo responsible for Development
and Commercialization of Onxeo’s products maintain in the ordinary course of business with respect to the Licensed Products, including:

(1) a copy of the submissions to and correspondence to and from the regulatory authorities;

(2) the list of the composition thereof;

(3) reports and filings concerning complaints and adverse incidents not otherwise provided; and

(4) marketing and promotional materials, if any.

 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

SCHEDULE 3

LICENSED TRADEMARKS

ONXEO-Ref

Title

Jurisdiction

Filing Number

Filing Date

Registration
Number

Registration Date

[***]

[***]

[***]

[***]

[***]

[***]

[***]

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

SCHEDULE 4

VALIDIVE MATERIALS

[***]

[***]

[***]

[***]

Raw materials

Description
[***]
[***] (development)

Stability Study

Description
Clinical Batches

[***]

Technical Batches

Expiry
[***]
[***]

Study point ongoing

Location

[***]

[***]

  [***]                                                                                       [***]                                                                        [***]

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
SCHEDULE 5

CONFIRMATORY PATENT LICENSE

THIS DEED is made the ___________day of______________________201[●]

1) 

2) 

MONOPAR  THERAPEUTICS  INC ,  whose  principal  office  is  598  Rockefeller  Road,  Lake  Forest,  Illinois,  USA,  60045
(“Monopar”); and

ONXEO  S.A.,  with  its  principal  place  of  business  located  at  49,  boulevard  du  Général  Martial  Valin,  75015  Paris,  France
(hereinafter “Onxeo”).

RECITALS:

By  an  agreement  (the “Main Agreement”)  dated  __________________  and  made  between  Monopar  and  Onxeo.  Onxeo  agreed  for  the
consideration  therein  contained,  among  other  things,  to  grant  to  Monopar  a  license  under  [Country/region  Patent  No.__________]  (the
“Patent”) of which this Agreement is a confirmatory license.

OPERATIVE PROVISIONS:

1. 

2. 

In pursuance of the Main Agreement and for the consideration referred to in the Main Agreement Onxeo hereby grants to Monopar
the exclusive license from the ________ day of_____________ 20___ to research, develop, use, keep, make, have made, import,
sell and otherwise dispose of Licensed Products (as defined in the Main Agreement) in the Field (as defined in the Main Agreement)
in the Territory (as defined in the Main Agreement) for the life of the Patent and subject to the provisions of the Main Agreement.

Subject to the provisions of the Main Agreement this Agreement shall terminate without notice in the event of the termination of the
Main Agreement in accordance with its terms.

IN WITNESS of which this Agreement has been executed as a deed and delivered the day and year first above written.

EXECUTED as a deed

For and on behalf of

ONXEO S.A.

acting by a Director and its Secretary / two Directors

EXECUTED as a deed

For and on behalf of

MONOPAR THERAPEUTICS INC

acting by a Director and its Secretary / two Directors

)

)

)

)

)

)

)

)

)

)

)

)

)

)

)

)

Name (PRINT):                                                            

Title (PRINT):                                                            

Signature:                                                            

Date:                                                            

Name (PRINT)                                                            

Title (PRINT)                                                            

Signature:                                                            

Date:                                                            

Name (PRINT):                                                            

Title (PRINT):                                                            

Signature:                                                            

Date:                                                            

Name (PRINT)                                                            

Title (PRINT)                                                            

Signature:                                                            

Date:                                                            

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
AMENDMENT No. 1 to VALIDIVE OPTION AND LICENSE AGREEMENT

This  amendment  number  one  (“Amendment”)  to  the  Validive  Option  and  License  Agreement  dated  June  17,  2016  (the
“Agreement”) is by and between Monopar Therapeutics Inc., a Delaware corporation having a place of business at 5 Revere Drive, Suite
200,  Northbrook,  Illinois  60062  (“Monopar”),  and  Onxeo  S.A.,  a  French  société  anonyme  à  Conseil  d’administration  located  at  49,
boulevard du Général Martial Valin, 75015 Paris, France (“ Onxeo”). Monopar and Onxeo shall also hereinafter be referred to as a Party or
collectively as the Parties.

WHEREAS, the Parties entered into the Agreement effective June 17, 2016 (“Effective Date”);

RECITALS

WHEREAS, Monopar has exercised the licensing option and paid the License Fee as provided in the Agreement; and

WHEREAS, the Parties now wish to amend the Agreement as more particularly set forth below.

NOW, THEREFORE, in consideration of the covenants contained herein the Parties hereto, intending to be legally bound hereby,

agree to and hereby do amend the Agreement as follows:

1.  All capitalized terms used herein and not otherwise defined shall have the same meaning as defined in the Agreement.

2.  Schedule 3 of the Agreement is replaced in its entirety with the attached Schedule 3.

3.  For  the  avoidance  of  doubt,  the  Trademarks  added  to  Schedule  3  by  this Amendment  (“ Additional Trademarks ”)  shall  be  deemed
Licensed  Trademarks  under  the Agreement  as  of  the  Effective  Date  and  within  the  rights  granted  by  Onxeo  to  Monopar  including
assignment upon Monopar’s exercise of the Monopar Validive Option.

4.  Onexo  agrees  to  execute  and  deliver  documents  as  may  be  necessary  or  desirable  to  give  effect  to  the  assignment  of  the Additional

Trademarks.

5.  Except  as  otherwise  amended  hereby,  the Agreement  shall  remain  in  full  force  and  effect  as  presently  written,  and  the  rights,  duties,

liabilities and obligations of the Parties thereto will continue in full effect.

IN  WITNESS  WHEREOF,  the  Parties  have  caused  this Amendment  to  be  executed  by  their  duly  authorized  representatives,

effective of the Effective Date.

MONOPAR THERAPEUTICS INC.
Signature: /s/ Chandler D. Robinson
Print Name: Chandler Robinson 
Title: CEO

ONXEO S.A.
Signature: /s/ Judith Greciet
Print Name: Judith Greciet 
Title: CEO

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

Schedule 3 Licensed Trademarks

Title
[***]

Jurisdiction
[***]

Filing Number
[***]

Filing Date
[***]

Registration Number Registration Date
[***]

[***]

 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

CONTRIBUTION AGREEMENT (351)

             This  Contribution Agreement  (this  “Agreement”)  is  entered  into  as  of August  25,  2017  (the  “ Effective Date”),  among  TacticGem  LLC,  a
Delaware  limited  liability  company  (the  “Company”),  Monopar  Therapeutics  Inc.,  a  Delaware  corporation  (“Monopar”),  Gem
Pharmaceuticals,  LLC,  an  Alabama  limited  liability  company  (“Gem”)  and  Tactic  Pharma,  LLC,  an  Illinois  limited  liability  company
(“Tactic”, and collectively with Gem, the owners of 100% of the issued and outstanding limited liability company interests of the Company).
The  Company,  Monopar,  Tactic,  and  Gem  are  sometimes  hereinafter  referred  to  collectively  as  the  “ Parties”,  and  each  individually  as  a
“Party”.

BACKGROUND INFORMATION

A.           The parties have entered into that certain Contribution Agreement by and among the Company, Tactic, and Gem, dated as of
August 24, 2017 (the “721 Contribution Agreement”) whereby Gem contributed to the Company all of Gem’s right, title and interest in and to the
property and assets described on Exhibit A attached hereto (collectively, the “ Gem Contributed Assets”) and Tactic contributed to the Company the
Tactic Contributed Assets (as defined in the 721 Contribution Agreement).

B.           Pursuant to this Agreement and subsequent to the contributions contemplated by the 721 Contribution Agreement, the Company
will contribute (the “Company Contribution”)  to  Monopar  all  of  the  Company’s  right,  title  and  interest  in  and  to  the  Gem  Contributed Assets  in
exchange for 3,055,394.12 shares of Monopar’s common stock. Subsequent to the transactions contemplated by the 721 Contribution Agreement and
this Agreement,  the  Company  will  own  7,166,667  shares  of  Monopar  common  stock,  which  will  constitute  79.70%  of  the  total  number  of  shares
outstanding  of  Monopar.  By  a  separate  agreement  (the  “Investor  Contribution  Agreement”),  entered  into  on  or  before  this Agreement,  between
Monopar and a third party investor (the “Investor”), the Investor will contribute $2,000,004 to Monopar in exchange for 333,334 shares of common
stock  (the  “Investor  Contribution”,  and  together  with  the  Company  Contribution,  the  “351  Transaction”).  The  Company  and  the  Investor,
collectively, will own at least 80% of the total combined voting power of all classes of stock entitled to vote and at least 80% of the total number of
shares of all classes of stock of Monopar subsequent to the 351 Transaction.

C.           It is the intent of the Parties hereto that the 351 Transaction constitutes a tax-free transfer pursuant to Section 351 of the Internal

Revenue Code of 1986, as amended.

 
 
 
 
 
 
 
 
 
NOW, THEREFORE, in consideration of the mutual covenants herein contained and for other good and valuable consideration, the receipt

and adequacy of which are hereby acknowledged, the Parties agree as follows:

STATEMENT OF AGREEMENT

ARTICLE I
COMPANY CONTRIBUTION

§1.1           Contribution. As of the Effective Date, (a) the Company hereby contributes the Gem Contributed Assets to Monopar, and (b) Monopar
hereby  accepts  the  Gem  Contributed Assets,  and   assumes  and  agrees  to  perform  all  obligations,  restrictions  and  conditions  which  are
applicable  to  the  Gem  Contributed Assets  to  the  extent  such  obligations  arise  or  accrue  from  and  after  the  Effective  Date  (except  as
otherwise provided in this Agreement). Monopar does not assume or otherwise accept responsibility for any Liabilities (as defined in the
721 Agreement) or obligations of Gem, Tactic, or the Company, provided that Monopar will assume the obligations of Gem accruing or
arising  after  the  Effective  Date  under  the  agreements  listed  on  the  attached Exhibit  B  (the  “Assigned  Contracts”),  with  Gem  being
responsible for all such liabilities and obligations accruing or arising prior to the Effective Date.

§1.2            Shares Issued. In exchange for the Gem Contributed Assets, Monopar shall issue 3,055,394.12 shares of its common stock (the
“Issued Stock”) to the Company. The Company shall hold such shares as a separate block of stock that may be specifically indentified as separate
from the other 4,111,272.88 shares of Monopar common stock held by the Company.

ARTICLE II
REPRESENTATIONS AND WARRANTIES

§2.1           Representations and Warranties of the Company, Tactic, and Gem.  The representations and warranties of the Company, Tactic, and
Gem set forth in Article 5 of the 721 Agreement are hereby made by them to Monopar and incorporated by reference in this Agreement as if
fully rewritten herein.

§ 2.2                      Representations and Warranties of Monopar. Monopar hereby represents and warrants to each of the other Parties hereto  that the
statements contained in this §2.2 are, except as would not be reasonably expected to have a material adverse effect, true and correct
as of the Effective Date.

(a)           Organization; Authority; Enforceability . Monopar is a corporation duly organized, validly existing and in good standing under the
laws  of  the  State  of  Delaware,  and  has  full  corporate  power  and  authority  to  execute  and  deliver  this Agreement  and  perform  its
obligations hereunder. This Agreement constitutes the legal, valid, and binding obligation of Monopar, enforceable against Monopar
in accordance with its terms, subject to the effects of bankruptcy, insolvency, fraudulent conveyance, reorganization, moratorium,
and other similar laws relating to and/or affecting creditors’ rights generally and to general equitable principles. The Issued Stock,
when  issued  pursuant  to  the  terms  and  conditions  of  this Agreement,  will  be  duly  authorized,  validly  issued,  fully  paid,  and  non-
assessable, and issued in compliance with all applicable federal and state securities laws.

 
 
 
 
 
 
 
 
 
 
 
(b)           Non-Contravention. Neither the execution and delivery of this Agreement, nor the consummation of the transactions contemplated
hereby,  will  (i)  violate  any  constitution,  statute,  regulation,  rule,  injunction,  judgment,  order,  decree,  ruling,  charge,  or  other  restriction  of  any
government,  governmental  agency,  or  court  to  which  Monopar is  subject  or  any  provision  of  Monopar’s Organizational  Documents  or  any  other
governing document of Monopar or (ii) conflict with, result in a breach of, constitute a default under, result in the acceleration of, create in any party
the  right  to  accelerate,  terminate,  modify,  or  cancel,  or  require  any  notice  under  any  agreement,  contract,  lease,  license,  instrument,  or  other
arrangement to which any assets of Monopar are subject (or result in the imposition of any Encumbrance upon any assets of Monopar).

( c )           Private Placement Memorandum of Monopar. The Private Placement Memorandum of Monopar dated August 22, 2017, which
includes the private placement memorandum dated March 25, 2017 (the “PPM”) contains information about Monopar. The PPM was prepared for an
offering limited to accredited investors and does not contain all of the information that would be included in a registration statement filed with the
SEC. Monopar is not aware of any inaccurate statements of fact in the PPM.

(d)            Capitalization. (i) The authorized capital of Monopar as of July 31, 2017 consisted of 40,000,000 shares of common stock, $0.001
par  value  per  share,  and  8,675,919.61  shares  of  common  stock  outstanding  (non-dilutive);  (ii)  on  a  fully  diluted  basis,  accounting  for  all  issued
options,  there  were  9,231,439.61  shares  of  common  stock  outstanding  as  of  July  31,  2017;  (iii)  following  the  surrender  of  2,888,727.12  shares  of
Tactic’s Monopar common stock back to Monopar, Monopar would have shares outstanding of 5,787,192.5 shares of common stock (non-dilutive),
and 6,342,712.5 shares of common stock on a fully-diluted basis; and (iv) 700,000 shares of Common Stock have been reserved for issuance under
Monopar’s  2016  Stock  Incentive  Plan,  of  which  555,520  shares  are  subject  to  issued  and  outstanding  options. All  outstanding  shares  of  Monopar
common stock have been duly authorized and validly issued, are fully paid and non-assessable, and to Monopar’s knowledge, issued in compliance
with all applicable federal and state securities laws.

(e)           Disclosure. No representation or warranty or other statement made by Monopar in this Agreement, or otherwise in connection with
the transactions contemplated hereby contains any material untrue statement or omits to state a material fact necessary to make any
of them, in light of the circumstances in which it was made, not misleading in any adverse respect.

( f )           No Other Representations and Warranties . Except for the representations and warranties set forth in this Agreement, each of the
Company,  Tactic,  and  Gem  acknowledges  and  agrees  that  no  representation  or  warranty  of  any  kind  whatsoever,  express  or  implied,  at  law  or  in
equity, is made or shall be deemed to have been made by or on behalf of Monopar to the Company, Tactic, or Gem, and Monopar hereby disclaims
any such representation or warranty, whether by or on behalf of Monopar. 

 
 
 
 
 
 
 
 
 
 
ARTICLE III
POST-CLOSING MATTERS

§3.1            Tax Matters. Each Party shall cooperate fully, as and to the extent reasonably requested by any other Party, in connection with
the preparation and filing of any Tax Return (as defined in the 721 Agreement) and any audit with respect to Tax (as defined in the 721 Agreement),
with respect to the Gem Contributed Assets. Such cooperation shall include the retention and, upon request, the provision of records and information
which are reasonably relevant to any such Tax Return or audit or any tax planning and shall also include making employees available on a mutually
convenient basis to provide additional information and explanation of any material provided hereunder. Each Party further agrees, upon request, to
use its commercially reasonable efforts to obtain any certificate or other document from any taxing authority or any other individual, corporation,
partnership, limited liability company, association, trust or any other entity or organization as may be necessary to mitigate, reduce or eliminate any
Tax that could be imposed (including any sales, use, documentary, stamp, gross receipts, registration, transfer, conveyance, excise, recording, license,
stock transfer stamps and other similar taxes and fees arising out of or in connection with or attributable to the transactions effected pursuant to this
Agreement (collectively, “Transfer Taxes”; but for purposes of clarification, Transfer Taxes do not include any income taxes incurred by or allocable
to  any  party  in  connection  with  or  attributable  to  the  transfer  of  the  Gem  Contributed  Assets,  and  the  transactions  affected  pursuant  to  this
Agreement). The Company shall bear and be responsible for the timely payment of, and to such extent shall indemnify and hold harmless Monopar
against  any  Transfer  Taxes,  and  Gem  and  Tactic  shall  each  in  turn  bear  and  be  responsible  for  the  timely  payment  of,  and  to  such  extent  shall
indemnify and hold harmless the Company against, fifty percent (50%) of such Transfer Taxes so paid.

§3.2            Consulting Relationship with Gem Personnel.  Each of Gerald M. Walsh and Richard D. Olson shall become consultants of
Monopar  at  the  Effective  Date  and  Monopar  will  execute  a  consulting  agreement  with  such  individuals  in  substantially  the  form  of  the  attached
Exhibit C.

§ 3.3                      Indemnification.

(a) Notwithstanding any investigation conducted at any time with regard thereto, by or on behalf of the Company, Tactic, Gem or Monopar,
all  representations,  warranties,  covenants  and  agreements  of  the  Parties  in  this Agreement  (including  those  incorporated  by  reference)  and  in  any
other  documents  executed  or  delivered  by  any  of  them  pursuant  to  this Agreement  or  in  connection  with  the  transactions  contemplated  by  this
Agreement (collectively, the “Additional Documents”) shall survive the execution, delivery, and performance of this Agreement and the Additional
Documents.

 
 
 
 
 
 
 
(b) (i) Each Party shall defend, indemnify and hold harmless the other Parties, and their directors, officers, employees and representatives
from and against any and all Damages asserted against, resulting to, imposed upon, or incurred or suffered by such Party, directly or indirectly, as a
result of or arising from any Indemnifiable Claims as set forth in Sections 9.2, 9.3, 9.4, 9.5, 9.7, 9.8 and 9.9 of the 721 Contribution Agreement (the
“Indemnification Provisions”), which are hereby incorporated by reference; and (ii) Monopar shall  defend, indemnify and hold harmless each of the
Parties from and against any and all Damages asserted against, resulting to, imposed upon, or incurred or suffered by Gem, directly or indirectly, as a
result of or arising from any material breaches of the representations and warranties of Monopar in §2.2 pursuant to the Indemnification Provisions.
Indemnification by any Party to this Agreement shall be governed by the Indemnification Provisions. References to the “Agreement” in such Sections
shall be interpreted to refer to this Agreement in the context of Indemnifiable Claims under this Agreement.

§3.4. Tax Treatment .  Each  of  the  Parties  acknowledges  and  agrees  that  the  contribution  of  the  Gem  Contributed Assets  to  Monopar  is
intended to qualify for treatment as an exchange described in Section 351(a) of the Internal Revenue Code of 1986, as amended (the "Code"). All
Parties agree to prepare or cause to be prepared their Tax Returns in accordance with the immediately preceding sentence, including complying with
the record keeping requirements of Treasury Regulation Section 1.351-3.

§ 4.1 Registration Rights.

ARTICLE IV
REGISTRATION RIGHTS

(a)  Monopar  shall,  upon  direction  by  the  Company  at  any  time  after  Monopar  has  been  subject  to  the  reporting  requirements  of  the
Securities and Exchange Act of 1934 for at least 12 months (the “Initial Holding Period”), file with the U.S. Securities and Exchange Commission
(“SEC”) a Form S-3 or other appropriate form of registration statement, covering the resale of any Monopar common stock by the Company, Gem,
or Tactic and shall use its best efforts to have such registration statement declared effective as soon as practical thereafter. During the period that the
registration statement is effective, Monopar shall make all public filings required in the normal course of its business and necessary to maintain the
effectiveness of the registration statement during the period of resale of any Monopar common stock by the Company, Gem, or Tactic; provided that
the  Company,  Gem,  and  Tactic  agree  that  Monopar  may,  from  time  to  time,  inform  the  Company,  Gem,  and  Tactic  that  it  may  not  sell  Monopar
common stock until further notice if circumstances exist which have not been disclosed publicly and the omission of which, in the reasonable opinion
of Monopar, would result in a material omission of fact in the registration statement. The Company, Gem, and Tactic agree that upon receipt of such
notice and until otherwise informed by Monopar, the Company, Gem, and Tactic shall not sell, or permit to be

 
 
 
 
 
 
 
sold, the Monopar common stock. The Company, Gem, and Tactic acknowledge that Monopar cannot guarantee receipt of approval from the SEC,
and in the event that approval is not granted, the Company, Gem, and/or Tactic, as applicable, must hold the Monopar common stock until such time
as  the  Company,  Gem,  and/or  Tactic  may  be  permitted  to  sell  the  Monopar  common  stock  pursuant  to  applicable  securities  laws  or  exemptions
therefrom. Monopar shall pay the costs to prepare and file the registration statement, including the registration fee due to the SEC and all legal and
accounting expenses and the cost of compliance with the securities or blue sky laws in the State of Delaware or any other state. The Company, Gem,
or Tactic, as applicable (the party which is the seller of such Monopar common stock) shall pay all other costs of sale of the Monopar common stock,
including any underwriting fees, commissions on sale or stock transfer taxes resulting from the sale of the Monopar common stock. In the event that
a  registration  statement  for  the  resale  of  the  Monopar  common  stock  is  not  approved  by  the  SEC,  Monopar  shall,  upon  written  request  of  the
Company, prepare and file a registration statement on Form S-1 registering for sale any of the common stock and use its best efforts to have such
registration statement declared effective as soon as practical thereafter. Monopar shall pay the costs to prepare and file such registration statement,
including the registration fee due to the SEC and all legal and accounting expenses and the cost of compliance with the securities or blue sky laws in
the State of Delaware or any other State. Additionally, the Company, Gem, and Tactic shall receive the piggyback registration rights set forth in (b)
below.

 (b)           At any time following the Effective Date (but without obligation to do so) if Monopar proposes to register any of its common
stock under the Securities Act of 1933, as amended (the “Securities Act”) in connection with the public offering of such securities solely for cash
(other than a registration effected solely to implement an employee benefit plan or a transaction to which Rule 145 of the Securities Act is applicable
or  a  registration  using  any  form  that  does  not  permit  secondary  sales  of  securities),  Monopar  will  give  written  notice  to  the  Company,  Gem,  and
Tactic  of  its  intention  to  do  so  and,  upon  written  request  of  the  Company,  Gem,  or  Tactic,  delivered  to  Monopar  within  15  days  after  receipt  of
notice, Monopar will use its best efforts at its own expense (but excluding any underwriting commissions and stock transfer taxes accruing to any
common stock registered by the Company, Gem, or Tactic) to cause to be registered under the Securities Act the shares of common stock specified by
the Company, Gem, or Tactic, subject to (1) the right of other holders of restricted stock to include their stock in any such registration prior to the
inclusion of the common stock, including but not limited to rights of parties acquiring shares of common stock under any agreement that Monopar
will register the resale thereof, (2) the Company’s acceptance of the terms of any underwriting agreement entered into or proposed to be entered into
between Monopar and any underwriter of such offering, and (3) if the sole or managing underwriter of such offering determines that the aggregate
number of shares of common stock which have been requested by the Company, Gem, or Tactic to be included in the registration should be limited to
a lesser number or not included due to market conditions, then Monopar may only sell the lesser portion, if any. If a limitation is imposed on the
number of common stock includable by Monopar in any such offering, Monopar shall give the Company, Gem, and Tactic, as applicable, prompt
written notice thereof.

§4.2               Form 10. Monopar shall exert its commercially reasonable best efforts to cause to be filed with the Securities and Exchange
Commission (the “SEC”), under the Securities Exchange Act of 1934 (the “1934 Act”), a registration statement on Form 10 (or another appropriate
form), to register Monopar’s shares of common stock, $0.001 par value per share, within ninety (90) days after the Effective Date.

ARTICLE V
MISCELLANEOUS PROVISIONS

§5.1            Severability. Any term or provision of this Agreement that is invalid or unenforceable in any situation in any jurisdiction (as
determined by a court) shall not affect the validity or enforceability of the remaining terms and provisions hereof or the validity or enforceability of
the offending term or provision in any other situation or in any other jurisdiction.

 
 
 
 
 
 
 
 
§5.2           Notices. All notices, requests, demands, claims, and other communications hereunder shall be made as set forth in Section 11.1 of

the 721 Contribution Agreement.

§5.3            Construction. The parties have participated jointly in the negotiation and drafting of this Agreement. In the event an ambiguity
or question of intent or interpretation arises, this Agreement shall be construed as if drafted jointly by the parties and no presumption or burden of
proof  shall  arise  favoring  or  disfavoring  any  party  by  virtue  of  the  authorship  of  any  of  the  provisions  of  this Agreement. Any  reference  to  any
federal,  state,  local,  or  foreign  statute  or  law  shall  be  deemed  also  to  refer  to  all  rules  and  regulations  promulgated  thereunder,  unless  the  context
requires otherwise.

§5.4            Entire Agreement; Amendment; Waivers, etc.  This Agreement (including its  schedules  and  exhibits),  along  with  the  721
Agreement  and  the  Investor  Contribution Agreement  constitutes  the  entire  agreement  among  the  Parties  and  supersedes  all  prior  agreements  and
understandings,  agreements  or  representations  by  or  among  the  Parties,  written  and  oral,  with  respect  to  their  subject  matter.  No  amendment,
supplement, waiver or termination of this Agreement is binding unless executed in writing by the Party to be bound thereby. No waiver of any of the
provisions  of  this Agreement  constitutes  a  waiver  of  any  other  provision  of  this Agreement,  whether  or  not  similar,  unless  otherwise  expressly
provided.

§5.5           

Successors  and Assigns .  Except  as  otherwise  expressly  permitted  in  this Agreement,  the  Parties  agree  not  to  assign  this
Agreement  or  any  of  the  rights,  interests,  or  obligations  hereunder  to  any  other  person  or  entity  (whether  in  whole  or  in  part,  whether  directly  or
indirectly, and whether voluntarily or, to the fullest extent permitted by applicable law, involuntarily), except with the prior written consent of the
other Party, which consent such Party may grant or withhold in its sole discretion, and which consent, if granted, does not imply any other consent in
the future. Any purported assignment in violation of this Section will be void and of no legal effect. This Agreement will inure to the benefit of and
be binding upon each Party to this Agreement and each Party’s successors, heirs, permitted assigns, and legal representatives.

§5.6           Captions. The headings of the Sections and Articles of this Agreement are inserted for convenience only and shall not constitute

a part hereof or affect in any way the meaning or interpretation of this Agreement.

§5.7            Counterparts. This Agreement may be executed in any number of separate counterparts (including facsimile and electronic

transmission), each of which upon execution and delivery will constitute an original and all of which taken together will constitute one agreement.

§5.8           Governing Law; Consent to Jurisdiction and Venue.

(a)           THIS AGREEMENT SHALL BE GOVERNED BY, AND CONSTRUED IN ACCORDANCE WITH, THE LAWS OF THE
STATE OF DELAWARE, WITHOUT GIVING EFFECT TO ANY CHOICE OF LAW OR CONFLICTING PROVISION OR RULE (WHETHER
OF THE STATE OF DELAWARE OR ANY OTHER JURISDICTION) THAT WOULD CAUSE THE LAWS OF ANY JURISDICTION OTHER
THAN THE STATE OF DELAWARE TO BE APPLIED.

 
 
 
 
 
 
 
 
 
 
(b)           Each of the Parties hereto irrevocably submits itself to the exclusive jurisdiction of the United States District Court of the Northern
District of Illinois (unless such court lacks jurisdiction under Applicable Law, in which case each Party submits itself exclusively to the jurisdiction
of the state courts of Illinois sitting in Cook County) for the purpose of any Action arising out of or relating to this Agreement and/or the transactions
contemplated hereby.

(c)                      Each  of  the  Parties  hereto  irrevocably  agrees  that  all  claims  with  respect  to  any  such Action  arising  out  of  or  relating  to  this
Agreement and/or the transactions contemplated hereby shall be heard and determined exclusively in United States District Court of the Northern
District of Illinois (unless such court lacks jurisdiction under Applicable Law, in which case each Party submits itself exclusively to the jurisdiction
of the state courts of Illinois sitting in Cook County).

§  5.9                      WAIVER OF JURY TRIAL. AS A SPECIFICALLY BARGAINED INDUCEMENT FOR EACH OF THE PARTIES
TO  ENTER  INTO  THIS  AGREEMENT  (EACH  PARTY  HAVING  HAD  OPPORTUNITY  TO  CONSULT  COUNSEL),  EACH  PARTY
EXPRESSLY WAIVES THE RIGHT TO TRIAL BY JURY IN ANY LAWSUIT, ACTION OR PROCEEDING RELATING TO OR ARISING IN
ANY WAY FROM THIS AGREEMENT OR ANY TRANSACTIONS RELATED HERETO OR CONTEMPLATED HEREBY.

§ 
Agreement.

5.10                      Defined Terms. Any  terms  not  defined  in  this Agreement  shall  have  the  meanings  assigned  to  them  in  the  721

The Parties have duly executed this Agreement as of the date first above written.

MONOPAR THERAPEUTICS, INC.

By:/s/ Chandler Robinson
Chandler Robinson, CEO

TACTIC PHARMA, LLC

By: /s/ Chandler Robinson
Its: Manager

TACTICGEM LLC

By: CDR Pharma LLC
Its: Manager

By: /s/ Chandler Robinson
Its: Member of the Manager

GEM PHARMACEUTICALS, LLC

By: /s/ Arthur Klausner
Arthur Klausner, CEO

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
EXHIBIT A

Gem Contributed Assets

See Attached.

 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

“Gem Contributed Assets” means, collectively, the following (each as defined herein):

1.            $5,000,000 in cash.
2.            All right, title and interest, tangible and intangible, in and to the following (individually and collectively, the “Compounds”):
a.            GPX-100
b.            GPX-150
c.            GPX-160
d.            GPX-170
e.            GPX-180
3.            The Related Assets
4.            All of the Gem Contributed Intellectual Property
5.            All of the Gem Contracts including:
a.            License Agreements
b.            Research and Collaboration Agreements
c.            Manufacturing, Clinical Research and Compound Storage Agreements
6.            All inventory of product, including raw materials, work in process and finished product
7.            All works-made-for hire agreements relating to the Compounds.
8.            After Closing, Gem will use reasonable good faith efforts to cause Monopar and the Company to be added as additional insureds to its product

liability and comprehensive general liability insurance policies (the “Gem Insurance Policies”). Such rights as additional insureds shall be
transferred to each of Monopar and the Company and shall be considered Gem Contributed Assets.

B.            “GPX-150” means:

1. [***]
2. [***]
3. Any [***]
4. [***]
5. Any formulation of [***]
6. Any uses of [***]

C.            “GPX-160” means:

1.            [***]
2.            [***]
3.            [***]
4.            Any formulation of [***]
5.            Any uses of [***]

D.            “GPX-100” means:

1. [***]
2. [***]
3. [***]
4. [***]
5. Any formulation of [***]
6. Any uses of [***]

 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

E.            “GPX-170” means:

1. [***]
2. [***]
3. Any [***]
4. [***]
5. Any formulation of [***]
6. Any uses and formulations of [***] and

F.            “GPX-180” means:

1. [***]
2. [***] and [***].
3. Any [***]
4. [***]
5. Any formulation of [***]
6. Any uses and formulations of [***]

G.            “Related Assets” means:

1.            All assets related to Gem’s use and development of the Compounds (including without limitation [***] for any purpose, all assets used by

Gem, and necessary or useful to Gem as of Closing, in conducting research, development, testing, marketing, selling, manufacturing and/or
distributing the Compounds and any other analogs derived from them and their use (including without limitation [***] or any other analogs
derived from GPX-100, GPX-150, GPX-160, GPX-170, or GPX-180)) as such activity is presently conducted and as such activity is presently
planned to be conducted, including, but not limited to, all inventory of Compounds, all other inventory, agreements, contracts, licenses,
Intellectual Property related to or useful for the Business, intellectual property assignments, , orphan drug or other regulatory designations,
pending orphan drug or other regulatory applications, trademarks, service marks and all goodwill associated therewith, pre-clinical and
clinical data, manufacturing equipment; anthracycline molecules that, [***].

2.            The [***].
3.            Manufacturing agreements.
4.            Written reports, regulatory documents, case reports, and manufacturing methods.
5.            All FDA and other regulatory authorities filings and scientific studies relating to the Compounds and the Related Assets including the

following:

a.            Orphan drug designation [***]
b.            [***] GPX-150 [***]. All relevant filings and approvals in the US for GPX-150 have been made to this IND and are part of the IND record.

[Date February 7, 2007]

 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

H.            “Gem Contributed Intellectual Property” has the meaning set forth in Section 10 of the Agreement. “Intellectual Property” means:

All domestic and foreign (1) patents and patent applications, and all patents issuing thereon, including without limitation utility, model and design
patents and certificates of invention, together with all reissue patents, patents of addition, divisionals, provisional applications, renewals,
continuations, continuations-in-part, substitutions, additions, extensions, confirmations, re-examinations, and all foreign counterparts of the forgoing
which are in the process of being prepared, and all inventions and improvements disclosed therein including the right to claim priority benefit of or to
any of the foregoing (collectively, “Patents”); (2) trademarks, service marks, trade dress, trade names, brand names, designs, logos, commercial
symbols and corporate names, and all registrations, applications and goodwill associated therewith (collectively, “Trademarks”); (3) copyrights and
all works of authorship, whether or not registered or copyrightable, and all applications, registrations, and renewals in connection therewith
(collectively, “Copyrights”); (4) confidential and proprietary information, including without limitation, trade secrets, know-how, formulae, ideas,
concepts, discoveries, innovations, improvements, results, reports, information and data, research, laboratory and programmer notebooks, methods,
procedures, proprietary technology, operating and maintenance manuals, engineering and other drawings and sketches, customer lists, supplier lists,
pricing information, cost information, business manufacturing and production processes and techniques, designs, specifications, and blueprints
(collectively, “Trade Secrets”); and (5) all other intellectual property and proprietary rights in any form or medium known or later devised, all copies
and tangible embodiments of the foregoing, and all goodwill associated with any of the foregoing; and (6) the right to bring suit, the right to claim
and retain all damages and/or seek other remedies for the past, present, and future infringement and/or misappropriation of and the right to collect
royalties and other payments under or on account of any of the foregoing; in each case whether registered or unregistered.

U.S. patents and patent applications within the Gem Contributed Intellectual Property:

1.            [***].
2.            [***].
3.            [***].
4.            [***].
5.            [***].
6.            [***].
7.            [***].
8.            Patent pending [***], filed [***]: covers the composition of [***] and the [***].
9.            [***]

 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

Foreign patents and patent applications within the within the Gem Contributed Intellectual Property:

Country
 [***]

Patent #
 [***]

Based on U.S. Patent No.
 [***]

 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

 [***]

[***]

[***]

    Copyrights and Trade Secrets within the Gem Contributed Intellectual Property:

1.            Analysis of [***] for GPX-150
2.            Analysis of [***]for GPX-150
3.            Analysis of [***] for GPX-100

           Unpatented inventions within the Gem Contributed Intellectual Property:

           1. GPX-160, GPX-170 and GPX-180

           Trademarks within the Gem Contributed Intellectual Property:

           1.            Gem Pharmaceuticals (unregistered

2.            On [***], Gem submitted an International Non-Proprietary Name (INN)request to the World Health Organization for GPX-150,  [***]

I.            Gem Contracts

License Agreements (no active license agreements)

1.            Non-binding term sheet with Vitel Laboratories, expired on August 1, 2017.
2.            Coronado Biosciences agreement, expired on October 8, 2010.
3.            [AOI, expired on February 5, 2003]

Assigned Research and Collaboration Agreements (no active agreements other than [***])

1. [***]:
-- two Service Agreements, each expired April 30, 2016; fully completed and fully paid
-- Service Agreement expired August 14, 2017; work complete but final report due to be delivered soon after Closing. Gem agrees to promptly
deliver to Monopar said report upon receipt, to pay in full all amounts owed under said Agreement, and if requested, to use reasonable good faith
efforts to obtain a consent from BSU in substantially the same form as Exhibit E to the Contribution Agreement.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

--Service Agreement expiring August 31, 2017; work complete and final report has been delivered. Gem agrees to pay in full all amounts owed under
said Agreement.
2. [***], expired on June 24, 2015.
3. Agreements with [***] as reflected in proposals of [***] dated April 21, 2016, June 24, 2016, July 5, 2016, and December 6, 2016.
Assigned Manufacturing, Clinical Research and Compound Storage Agreements
1.            Manufacturing (All manufacturing agreements other than [***] have expired)

a.            Tetrionics, expired January, 2005.
b.            SAFC, expired August, 2015.
c.            [***], dated May 31, 2017.
d.            Bioserv, expired January, 2016.

2.            Clinical Research Organizations (no active agreements)

a.            Premier Research , expired on May 14, 2014.
b.            Clinical Trial Data Services, expired on March 26, 2017.

3.            Compound Storage
a.            Clinical Supplies Management, Inc., dated October 16, 2014.

 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

Other Gem Contracts

1.            Renewal Service Agreement between Gem Pharmaceuticals, LLC and CPAGlobaldated August 31, 2016.

J.            All inventory of product, including raw materials, work in process and finished product

1.            Inventory of GPX-150 and GPX-100 located in [***]
●            200 vials of GPX-150 product (about 50 mg/vial = about 10 grams of GPX-150 mixed with lactose)
●            6.8 grams of GPX-150 from a batch made in 2006
2.            Inventory of clinical-grade GPX-150 located at CSM in [***]
●            GPX-150 Powder 14.11 grams – expired 17 Nov 2016
●            GPX-150 50mg vial 406 vials – expired 31 Oct 2016
3.            Inventory of GPX-150 (approximately 15 grams) located at [***]

 
 
 
 
 
 
 
 
EXHIBIT B

Assigned Contracts

1. Master Services Agreement by and between Gem and Clinical Supplies Management, Inc., dated October 1, 2014

2. Renewal Service Agreement between Gem Pharmaceuticals, LLC and CPA Global dated August 31, 2016

 
 
 
 
 
 
 
 
 
EXHIBIT C

Form of Consulting Agreement

See attached.

 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

CONSULTING AGREEMENT

This Consulting Agreement (herein referred to as “Agreement”) is made and entered into as of this day of , 2017 (the “Effective Date”), by
and between Monopar Therapeutics, Inc. (herein referred to as “Monopar”), a Delaware corporation, located at 5 Revere Dr., Suite 200, Northbrook,
IL  60062,  and  Gerald  M.  Walsh  (herein  referred  to  as  “Jerry”)  who  resides  at  [***]  (each  herein  referred  to  as  “Party”  and  collectively  as
“Parties”).

RECITALS

WHEREAS, Jerry specializes in the fields of pharmacology, toxicology, intellectual property, and pharmaceutical management.

WHEREAS, Monopar desires to contract with Jerry to provide certain consultation services, as requested by Monopar, and Jerry wishes to

provide such services to Monopar, upon the terms and conditions set forth below.

NOW, THEREFORE, in consideration of the premises and mutual covenants contained herein, the Parties agree as follows:

Consulting Arrangement. Jerry agrees to perform consulting services as described herein upon the terms and conditions herein set forth.

Term  of Agreement .  Subject  to  the  provision  for  early  termination  set  forth  below  in Section 5  of  this Agreement,  this Agreement  shall
commence as of the Effective Date and shall continue from the Effective Date through one year later (the “Term”).

Duties of Jerry.

1. 

2.

3.

3.1 

3.2 

Specific Duties. Jerry shall provide consulting services to Monopar, such duties to include: See Appendix A (herein referred to as the
“Services”).

Obligations. Jerry shall be diligent in the performance of Services, and be professional in his commitment to meeting his obligations
hereunder. Jerry represents and warrants that he is not party to any other existing agreement, which would prevent him from entering
into  this Agreement  or  which  would  adversely  affect  this Agreement.  Jerry  may  be  engaged  or  employed  in  any  other  business,
profession,  or  other  activity  but  Jerry  shall  not  perform  Services  for  any  other  individuals  or  entities  in  direct  competition  with
Monopar,  within  the  scope  of  Services  under  this  Agreement,  during  the  Term  of  this  Agreement,  and  for  two  years  after  its
termination, except as provided for by mutual written agreement of the Parties. Jerry shall not perform services for any party which
would require or facilitate the unauthorized disclosure of any confidential or proprietary information of Monopar.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

3.3 

Reporting.  Jerry  will  report  to Andrew  P.  Mazar,  Ph.D.  and  liase  with  Chandler  Robinson,  M.D.,  Patrice  Rioux,  M.D.  and/or  any
other assigned Monopar employee or consultant as may be designated in writing by Monopar.

3.4            Compensation. Monopar shall pay Jerry as follows:

a. [***] per month payable within thirty (30) days of the end of each month.

b. [***] per hour for consulting work that exceeds fifteen (15) hours per month, and has been approved by Monopar. Jerry will document all
hours, including the initial fifteen (15) hours, and invoice Monopar monthly for the hours above the first fifteen (15) hours.

Jerry shall not be reimbursed, and is responsible for the facilities and equipment necessary to perform Services required under this

Agreement.

4.

5.

6.

Reimbursement of Expenses. Monopar shall promptly reimburse Jerry for all direct expenses incurred in providing the Services to Monopar
pursuant to this Agreement, including travel, meals and lodging as long as Monopar’s prior approval has been obtained. Invoices submitted by
Jerry pursuant to this Section 4 shall also include a detail of all reimbursable expenses incurred during the period covered by such invoice as
well as receipts. Per diem for food will be reimbursed as per IRS specified rates in effect at that time.

Termination of Agreement - Failure to perform . In the event that Jerry ceases to perform the Services or breaches his obligations as required
hereunder for any reason and such cessation or breach remains uncured for ten (10) business days following Monopar’s written notice thereof
to  Jerry,  Monopar  shall  have  the  right  to  immediately  terminate  this Agreement  upon  notice  to  Jerry  and  to  enforce  such  other  rights  and
remedies under this Agreement as it may have as a result of said breach.

In the event that Monopar breaches its obligations under this Agreement and such breach remains uncured for ten (10) business days
following Jerry’s written notice thereof to Monopar, Jerry shall have the right to immediately terminate this Agreement upon notice to
Monopar and to enforce such other rights and remedies under this Agreement as it may have as a result of said breach.

Certain Liabilities. It is understood and agreed that Jerry shall be acting as an independent contractor and not as an agent or employee of, or
partner, joint venturer or in any other relationship with Monopar. Jerry will be solely responsible for all insurance, employment taxes, FICA
taxes and all obligations to governments or other organizations for its employees arising out of this consulting assignment. Jerry acknowledges
that no income, social security or other taxes shall be withheld or accrued by Monopar for Jerry’s benefit. Jerry assumes all risks and hazards
encountered in the performance of duties under this Agreement. Unless Monopar has provided prior written approval, Jerry shall not use any
sub-contractors to perform obligations hereunder. Jerry shall be solely responsible for any and all injuries, including death, to all persons and
any and all loss or damage to property, which may result from performance under this Agreement.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
7.

8.

9.

10.

11. 

Indemnities.  Jerry  hereby  agrees  to  indemnify  Monopar  and  hold  Monopar  harmless  from  and  against  all  claims  (whether  asserted  by  a
person, firm, entity or governmental unit or otherwise), liabilities, losses, damages, expenses, charges and fees which Monopar may sustain or
incur  arising  out  of  or  attributable  to  any  gross  negligence  or  willful  misconduct  by  Jerry,  as  applicable,  in  the  performance  under  this
Agreement.  Monopar  hereby  agrees  to  indemnify  Jerry  and  hold  Jerry  harmless  from  and  against  all  liabilities,  losses,  damages,  expenses,
charges and fees which Jerry may sustain or incur by reason of any claim which may be asserted against Jerry by any person, firm, corporation
or governmental unit and which may arise out of or be attributable to any gross negligence or willful misconduct by Monopar or its employees
or contractors, as applicable, in the performance of this Agreement.

Warranties. The Services shall be performed in a professional manner, consistent with industry standards. In performing the Services under
this Agreement, Jerry shall not make any unauthorized use of any confidential or proprietary information of any other party or infringe the
intellectual property rights of any other party. Monopar represents and warrants that it has full right, power, and authority to enter into this
Agreement and to perform its obligations hereunder.

Arbitration. Any controversy or claim between Monopar and Jerry arising out of or relating to this Agreement, or the breach thereof, shall be
submitted to arbitration in accordance with the rules of the American Arbitration Association. The site of the arbitration shall be Chicago, IL,
and  except  as  provided  herein  the  arbitration  shall  be  conducted  in  accordance  with  the  Rules  of  the American Arbitration Association
prevailing at the time the demand for arbitration is made hereunder. At least one member of the arbitration panel shall be a financial expert
knowledgeable in the area of biopharmaceutical corporate compliance. Judgment upon any award rendered by the arbitrator(s) may be entered
in any court of competent jurisdiction and shall be binding and final. The cost of arbitration shall be borne by the losing Party, as determined
by the arbitrator(s).

Confidential  Information.  Jerry  has  executed  the  attached  confidential  disclosure  agreement  referenced  herein  as  Appendix  B  prior  to
commencement of the Services. Jerry hereby represents and warrants that the obligations thereunder shall be binding.

Inventions.  Jerry  agrees  that  all  ideas,  developments,  suggestions  and  inventions  conceived  or  reduced  to  practice,  as  a  result  of  Services
provided  by  Jerry  under  this Agreement,  shall  be  the  exclusive  property  of  Monopar  and  shall  be  promptly  communicated  and  assigned  to
Monopar.  Jerry  shall  require  any  other  parties  contracted  by  Jerry  to  disclose  the  same  to  Jerry  and  to  be  bound  by  the  provisions  of  this
paragraph.  During  the  period  of  this Agreement  and  thereafter  at  any  reasonable  time  when  called  upon  to  do  so  by  Monopar,  Jerry  shall
require  any  employees  of  or  other  parties  contracted  by  Jerry  to  execute  patent  applications,  assignments  to  Monopar  (or  any  designee  of
Monopar) and other papers and to perform acts which Monopar believes necessary to secure to Monopar full protection and ownership of the
rights  in  and  to  the  services  performed  by  Jerry  and/or  for  the  preparation,  filing  and  prosecution  of  applications  for  patents  or  inventions
made by any employees of or other parties contracted by Jerry hereunder. The decision to file patent applications on inventions made by any
employees of or other parties contracted by Jerry shall be made by Monopar and shall be for such countries, as Monopar shall elect. Monopar
agrees to bear all the expense in connection with the preparation, filing and prosecution of applications for patents and for all matters provided
in  this  paragraph  requiring  the  time  and/or  assistance  of  Jerry  as  to  such  inventions.  Notwithstanding  the  foregoing,  ideas,  developments,
suggestions,  and  inventions  conceived  or  reduced  to  practice  by  Jerry  that  do  not  directly  arise  from  Jerry’s  performance  under  this
Agreement, shall be owned by Jerry.

 
 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

12. 

Miscellaneous.

12.1 

Notice. Any  notices  to  be  given  hereunder  by  either  Party  to  the  other  may  be  effectuated,  in  writing,  by  personal  delivery,  by
electronic  mail,  or  by  mail,  registered  or  certified,  postage  prepaid,  with  return  receipt  requested  or  by  Federal  Express.  Mailed
notices shall be addressed to the parties at the following addresses:

If to Monopar:                                    Monopar Therapeutics, Inc

5 Revere Dr.
Suite 200
Northbrook, IL, 60062
Attention: Chandler Robinson, M.D.
Email: [***]

If to
Jerry:                                                      
                                                                            [***]

Gerald M.Walsh

or at such other addresses as either Monopar or Jerry may designate by written notice to each other. Notices delivered personally shall be deemed
duly given on the date of actual receipt, mailed notices shall be deemed duly given as of the fourth day after the date so mailed, and electronic mail
shall be deemed duly given upon confirmation of receipt by recipient.

12.2  Waiver of Breach. The waiver by either Party to a breach of any provision in this Agreement cannot operate or be construed as a

waiver of any subsequent breach by either Party.

12.3 

Severability. If any provision of this Agreement is determined by a court of competent jurisdiction to be invalid or unenforceable, that
provision  shall  be  deemed  modified  to  the  extent  necessary  to  make  it  valid  or  enforceable,  or  if  it  cannot  be  so  modified,  then
severed,  and  the  remainder  of  the Agreement  shall  continue  in  full  force  and  effect  as  if  the Agreement  had  been  signed  with  the
invalid portion so modified or severed.

 
 
 
 
 
           
 
 
 
 
 
 
12.4 

12.5 

Choice of Law.  This Agreement  has  been  made  and  entered  into  in  the  State  of  Illinois,  and  the  laws  of  such  state,  excluding  its
choice of law rules, shall  govern  the  validity  and  interpretation  of  this Agreement  and  the  performance  due  hereunder.  The  losing
party in any dispute hereunder shall pay the attorneys’ fees and disbursements of the prevailing party.

Integration.  The  drafting,  execution  and  delivery  of  this  Agreement  by  the  Parties  have  been  induced  by  no  representations,
statements,  warranties  or  agreements  other  than  those  expressed  herein.  This Agreement  embodies  the  entire  understanding  of  the
Parties, and there are no further or other agreements or understandings, written or oral, in effect between the Parties relating to the
subject matter hereof unless expressly referred to herein.

12.6  Modification. This Agreement may not be modified unless such is in writing and signed by both Parties to this Agreement.

12.7 

12.8 

12.9 

Assignment. Jerry shall not be permitted to assign this Agreement to any other person or entity without the prior written consent of
Monopar. Jerry hereby agrees that Monopar shall be permitted to assign this Agreement to any affiliate of Monopar. This Agreement
shall be binding upon and shall inure to the benefit of the successors and permitted assigns of the parties.

Survival.  The  provisions  of Sections 7, 8, 9, 10,  and 11  shall  survive  expiration  or  termination  of  this Agreement  for  any  reason.
Expiration or termination of this Agreement shall not affect Monopar’s obligations to pay any amounts that may then be due to Jerry.

Force Majeure. If Jerry’s performance of his obligations under this Agreement is prevented or delayed due to a flood, earthquake,
war, terrorist act, revolution, riot, or insurrection, Jerry shall not be deemed in breach of his obligations under this Agreement or
otherwise liable for any costs, charges or losses sustained or incurred by Monopar, to the extent arising directly from such force
majeure event.

IN WITNESS WHEREOF, the Parties hereto have executed this Agreement as of the day and year first above written.

ACCEPTED AND AGREED TO:

Gerald M. Walsh

By: Individual

Monopar Therapeutics Inc

By: Chandler Robinson

Its: Chief Executive Officer

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Services include, but are not limited to, assisting the Monopar Management team with the following:

APPENDIX A

1.            Near and long term planning of product development for existing Monopar drugs such as Validive, ATN-658, GPX-150, GPX-160, GPX-

170, and GPX-180.

2.            Developing near and long term budgets for product development programs: preclicnal, clinical, manufacturing, and related regulatory affairs.

3.            Designing, managing, evaluating, and reporting for preclinical and clinical studies and for manufacturing API and drug product.

4.            Data storage and retrieval for preclinical, clinical, manufacturing, and regulatory programs.

5.            Identifying and evaluating suitable in-licensing drug products, including evaluation of strength and scope of patent protection.

6.            Identifying patentable IP based on data from Monopar’s preclinical, clinical, and manufacturing programs.

7.            Creating presentation content for Board Meetings, fund raising, and M&A activities.

8.            Evaluating qualifications of employment candidates for Monopar.

9.            Any other Services required by Monopar.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Appendix B

See executed CDA attached

 
 
 
 
 
 
  
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

MONOPAR THERAPEUTICS INC.
CONFIDENTIAL DISCLOSURE AGREEMENT

AGREEMENT between the individual Gerald M. Walsh (“Recipient”) and Monopar Therapeutics Inc. (“Monopar”).

In consideration for the mutual agreements contained herein and the other provisions of this Agreement, the receipt of which is hereby
acknowledged by the parties, the parties hereto agree as follows:

1. Scope of Confidential Information

“Confidential Information” means, subject to the other provisions of this Section:

(a) all information, whether oral or written, disclosed by Monopar that is described in Schedule A under “Description of Confidential Information”.
Confidential Information may relate to the activities or property of Monopar or any of Monopar’s members, directors, officers, employees,
consultants, agents, representatives or affiliated entities (collectively, “Associated Persons”); and

(b) any written material prepared by Recipient or Recipient’s partners, directors, officers, employees, agents, representatives or affiliated entities
(collectively, “Associated Persons”) containing any Monopar Confidential Information.

“Confidential Information” does not include information that: (i) was available to Recipient (free of any confidentiality obligation in favor of
Monopar) prior to disclosure of such information by Monopar to Recipient; (ii) is made available to Recipient from a third party which (at the time
of such availability) was not, to Recipient’s knowledge, subject to a confidentiality obligation with respect to such information; (iii) is made
available to third parties by Monopar without restriction on the disclosure of such information, (iv) is or becomes available to the public on or after
the date of this Agreement (other than as a result of disclosure prohibited by any confidentiality obligation contained herein); or (v) is developed
independently by Recipient or its Associated Persons without reference to the Confidential Information.

Recipient agrees that it will not disclose to Monopar or to any of its employees or consultants any confidential, proprietary, or trade secret
information, or any other form of confidential protectable intellectual property, regardless of whether such information is the property of Recipient
itself or of some other individual or organization.

2. Use and Disclosure of Confidential Information

(a) Recipient agrees: (i) to preserve the confidentiality of Confidential Information for [***] from the date of signing this Agreement; (ii) to use
and/or permit the use of Confidential Information only for the purposes of, and to the extent necessary for, evaluating a business relationship
between the parties and, if such a relationship is consummated, carrying out such relationship; (iii) to disclose Confidential Information to, and to
permit the use of Confidential Information by, only such persons within Recipient who Recipient reasonably determines need to know such
information in connection with the activities described in (ii) above; and (iv) to use reasonable care to maintain the confidentiality of Confidential
Information, provided that such care shall be at least as great as the precautions taken by Recipient to protect its own confidential and/or proprietary
information.

(b) Notwithstanding anything to the contrary herein, Recipient is free to make (and this Agreement does not restrict) disclosure of any Confidential
Information in a judicial, legislative, or administrative investigation or proceeding or to a government or other regulatory agency; provided that, to
the extent permitted by, and practicable under, the circumstances, Recipient provides to Monopar (i) prior notice of the intended disclosure or (ii) if
prior notice is not permitted or practicable under the circumstances, prompt notice of such disclosure.

3. Certain Rights and Limitations

(a) All Confidential Information shall remain the property of Monopar. The provision of Confidential Information hereunder shall not transfer any
right, title or interest in such information to Recipient. Monopar does not grant any express or implied right to Recipient to or under Monopar’s
patents, copyrights, trademarks, trade secret information or other proprietary rights.

(b) Recipient agrees to adhere to all applicable laws and regulations relating to the export of technical data received hereunder.

(c) This Agreement imposes no obligations on either party to purchase, sell, license, transfer or otherwise transact in any technology, services or
products. This Agreement does not create any agency or partnership relationship between the parties hereto.

(d) All information disclosed hereunder is without representation or warranty of any kind whatsoever, including without limitation, any
representation or warranty as to accuracy or completeness, whether express or implied.

4. Remedies

(a) Upon Monopar’s reasonable request, Recipient agrees to return promptly to Monopar all Confidential Information that is in writing and in the
possession of Recipient and, upon written request, to certify the return or destruction (at Monopar’s option) of all Confidential Information.

(b) Recipient agrees that monetary damages may not be an adequate remedy for improper disclosure or use of Confidential Information, that
Monopar, upon breach of this contract, shall be entitled to such injunctive or equitable relief as may be deemed proper by a court of competent
jurisdiction, without waiving any other right or remedy, and that Recipient shall not resist an application for such relief on the ground that Monopar
has an adequate remedy at law.

5. Miscellaneous

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 (a) Except where expressly indicated otherwise, the words “written” or “in writing” shall include, but not be limited to, written or printed
documents, electronic and facsimile transmissions and computer disks or tapes (whether machine or user readable).

(b) In the event that any one or more of the provisions of this Agreement will for any reason be held to be invalid, illegal or unenforceable by a
court of competent jurisdiction, the remaining provisions of this Agreement will be unimpaired, and the invalid, illegal or unenforceable provisions
will be replaced by a mutually acceptable provision, which being valid, legal or enforceable, comes closest to the intention of the parties underlying
the invalid, illegal or unenforceable provision.

(c) No amendment or alteration of the terms of this Agreement shall be effective unless made in writing and executed by both parties hereto.

(d) A failure or delay in exercising any right in respect of this Agreement will not be presumed to operate as a waiver, and a single or partial
exercise of any right will not be presumed to preclude any subsequent or further exercise of that right or the exercise of any other right. Any
modification or waiver of any provision of this Agreement shall not be effective unless made in writing. Any such waiver shall be effective only in
the specific instance and for the purpose given.

(e) This Agreement and its enforcement shall be governed by, and construed in accordance with, the laws of the State of Illinois, without
regard to conflicts-of-law principles.

 
 
 
 
 
 
[***] = Confidential Information has been omitted and filed separately with the Securities and Exchange Commission. 
Confidential treatment has been approved with respect to the omitted informatio n, pursuant to an Order dated January 8, 2018.

[SIGNATURE PAGE FOLLOWS]

IN WITNESS WHEREOF, the parties hereto have executed this Agreement.

“RECIPIENT”

“MONOPAR”

Monopar Therapeutics Inc.

By:_______________________________________

By:_______________________________________

Name: Gerald M. Walsh
Title: Consultant

Name: Chandler D. Robinson
 Title: CEO

Date:_____________________________________

Date: _____________________________________

Notices hereunder shall be sent to:
Gerald M. Walsh
[***]

Notices hereunder shall be sent to:

[***]

SCHEDULE A

Description of Confidential Information Disclosed by Monopar:

(a) The identity of the particular compound or compounds under investigation by Monopar; (b) the medical indication and/or other purpose for which
any of these compounds are being investigated by Monopar; (c) the (known or putative) mechanism of action of any of these compounds; (d) any
techniques used by Monopar to discover, develop, produce, or test any of these compounds; and (e) any non-public business, financial, regulatory,
clinical or scientific information pertaining to Monopar or the compound or compounds that Monopar identifies as confidential when disclosed.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
MONOPAR THERAPEUTICS INC. 2016 STOCK INCENTIVE PLAN

1. Purpose of the Plan.

The purpose of this Plan is to enhance shareholder value by linking the compensation of officers, directors, key employees and
consultants  of  the  Company  to  increases  in  the  price  of  Monopar  Therapeutics  Inc.  common  stock  and  the  achievement  of  other
performance objectives, and to encourage ownership in the Company by key personnel and consultants whose long-term employment and
retention is considered essential to the Company’s continued progress and success. The Plan is also intended to assist the Company in the
recruitment of new employees and consultants and to motivate, retain and encourage such employees, directors and consultants to act in
the shareholders’ interest and share in the Company’s success.

2. Definitions.

As used herein, the following definitions shall apply:

(a) “Administrator” means the Board, any Committee or such delegates as shall be administering the Plan in

accordance with Section 4 of the Plan.

(b) “Affiliate” means any Subsidiary or other entity that is directly or indirectly controlled by the Company or

any entity in which the Company has a significant ownership interest as determined by the Administrator. The Administrator
shall, in its sole discretion, determine which entities are classified as Affiliates and designated as eligible to participate in this
Plan.

(c) “Applicable Law” means the requirements relating to the administration of stock option plans under U.S.

federal and state laws, any stock exchange or quotation system on which the Company has listed or submitted for quotation the
Common Shares to the extent provided under the terms of the Company’s agreement with such exchange or quotation system and,
with respect to Awards subject to the laws of any foreign jurisdiction where Awards are, or will be, granted under the Plan, the
laws of such jurisdiction.

(d) “Award” means a Stock Award, Option, Stock Appreciation Right, or Other Stock-Based Award granted in

accordance with the terms of the Plan, or any other property (including cash) granted pursuant to the provisions of the Plan.

(e) “Awardee” means an Employee, Director or Consultant who has been granted an Award under the Plan.

(f) “Award Agreement” means a Stock Award Agreement, Option Agreement, Stock Appreciation Right

Agreement, or Other Stock-Based Award Agreement, which may be in written or electronic format, in such form and with such
terms as may be specified by the Administrator, evidencing the terms and conditions of an individual Award. Each Award
Agreement is subject to the terms and conditions of the Plan. The effectiveness of an Award shall not be subject to the Award
Agreement’s being signed by

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
the Company and/or the Participant receiving the Award unless specifically so provided in the Award Agreement.

(g) “Board” means the Board of Directors of the Company.

(h) “Change of Control” shall mean, except as otherwise provided in an Award Agreement, one of the following shall

have taken place after the date of this Plan:

(i) any “person” (as such term is used in Sections 13(d) or 14(d) of the Exchange Act) (other than the Company,

any majority controlled subsidiary of the Company, or the fiduciaries of any Company benefit plans) becomes the beneficial
owner (as defined in Rules 13d-3 and 13d-5 under the Exchange Act), directly or indirectly, of 30% or more of the total voting
power of the voting securities of the Company then outstanding and entitled to vote generally in the election of directors of the
Company; provided, however, that no Change of Control shall occur upon the acquisition of securities directly from the
Company;

(ii) individuals who, as of the beginning of any 24 month period, constitute the Board (as of the date hereof, the
“Incumbent Board”) cease for any reason during such 24 month period to constitute at least a majority of the Board, provided
that any individual becoming a Director subsequent to the date hereof whose election, or nomination for election by the
Company’s shareholders, was approved by a vote of at least a majority of the Directors then comprising the Incumbent Board
shall be considered as though such individual were a member of the Incumbent Board, but excluding for this purpose any such
individual whose initial assumption of office is in connection with an actual or threatened election contest relating to the election
of the Directors of the Company; or

(iii) consummation of (A) a merger, consolidation or reorganization of the Company, in each case, with respect to

which all or substantially all of the individuals and entities who were the respective beneficial owners of the voting securities of
the Company immediately prior to such merger, consolidation or reorganization do not, following such merger, consolidation or
reorganization, beneficially own, directly or indirectly, at least 65% of the combined voting power of the then outstanding voting
securities entitled to vote generally in the election of directors of the entity or entities resulting from such merger, consolidation
or reorganization, (B) a complete liquidation or dissolution of the Company, or (C) a sale or other disposition of all or
substantially all of the assets of the Company, unless at least 65% of the combined voting power of the then outstanding voting
securities entitled to vote generally in the election of directors of the entity or entities that acquire such assets are beneficially
owned by individuals or entities who or that were beneficial owners of the voting securities of the Company immediately before
such sale or other disposition.

Notwithstanding the foregoing, if any payment or distribution event applicable to an Award is subject to the requirements of Section
409A(a)(2)(A) of the Code, the determination of the occurrence of a Change of Control shall be governed by applicable

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
provisions of Section 409A(a)(2)(A) of the Code and regulations and rulings issued thereunder for purposes of determining whether
such payment or distribution may then occur.

(i) “Code” means the United States Internal Revenue Code of 1986, as amended, and any successor thereto, the Treasury
Regulations thereunder and other relevant interpretive guidance issued by the Internal Revenue Service or the Treasury Department.
Reference to any specific section of the Code shall be deemed to include such regulations and guidance, as well as any successor
provision of the Code.

(j) “Committee” means a committee of Directors appointed by the Board in accordance with Section 4 of the Plan or, in

the absence of any such special appointment, the Compensation Committee of the Board.

(k) “Common Shares” means the common shares, $0.001 par value, of the Company, or any security of the Company

issued in substitution, exchange or lieu thereof.

(l) “Company” means Monopar Therapeutics Inc., a Delaware corporation, or, except as utilized in the definition of

Change of Control, its successor.

(m) “Consultant” means an individual providing services to the Company or any of its Affiliates as an independent

contractor, and includes prospective consultants who have accepted offers of consultancy for the Company or any of its Affiliates, so
long as such person (i) renders bona fide services that are not in connection with the offer and sale of the Company’s securities in a
capital-raising transaction, (ii) does not directly or indirectly promote or maintain a market for the Company’s securities, and (iii)
otherwise qualifies as a consultant under the applicable rules of the SEC for registration of shares of stock on a Form S-8 registration
statement

(n) “Conversion Award” has the meaning set forth in Section 4(b)(xii) of the Plan.

(o) “Director” means a member of the Board. Any Director who does not serve as an employee of the Company is

referred to herein as a “Non-employee Director.”

(p) “Disability” means (i) “Disability” as defined in any employment, consulting or similar agreement to which the

Participant is a party, or (ii) if there is no such agreement or it does not define “Disability,” (A) permanent and total disability as
determined under the Company’s long-term disability plan applicable to the Participant, or (B) if there is no such plan applicable to
the Participant or the Committee determines otherwise in an applicable Award Agreement, “Disability” shall mean the Participant’s
continuous illness, injury or incapacity for a period of six consecutive months, as determined by the Administrator in its discretion.
Notwithstanding the above, with respect to an Incentive Stock Option, Disability shall mean permanent and total disability as defined
in Section 22(e)(3) of the Code and, with respect to any Award that constitutes “nonqualified deferred compensation” within the
meaning of Section 409A of the Code, the foregoing definition shall apply for purposes of vesting of such Award, provided that such
Award shall not be settled until the earliest of: (x) the Participant’s “disability” within the meaning of Section 409A of the Code, (y)
the Participant’s “separation from service”

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
within the meaning of Section 409A of the Code and (z) the date such Award would otherwise be settled pursuant to the terms of the
Award Agreement.

(q) “Disaffiliation” means a Subsidiary’s or Affiliate’s ceasing to be a Subsidiary or Affiliate for any reason (including,

without limitation, as a result of a public offering, or a spin-off or sale by the Company, of the stock of the Subsidiary or Affiliate) or
a sale of a division of the Company and its Affiliates.

(r) “Employee” means a regular, active employee of the Company or any Affiliate, including an Officer or Director who

is also a regular, active employee of the Company or any Affiliate. The Administrator shall determine whether the Chairman of the
Board qualifies as an “Employee.” For any and all purposes under the Plan, the term “Employee” shall not include a person hired as an
independent contractor, leased employee, consultant or a person otherwise designated by the Administrator, the Company or an
Affiliate at the time of hire as not eligible to participate in or receive benefits under the Plan or not on the payroll, even if such
ineligible person is subsequently determined to be a common law employee of the Company or an Affiliate or otherwise an employee
by any governmental or judicial authority. Unless otherwise determined by the Administrator in its sole discretion, for purposes of the
Plan, an Employee shall be considered to have terminated employment and to have ceased to be an Employee if his or her employer
ceases to be an Affiliate, even if he or she continues to be employed by such employer.

(s) “Exchange Act” means the United States Securities Exchange Act of 1934, as amended, and any successor thereto.

(t) “Fair Market Value” means a valuation performed by a qualified independent appraiser within the previous twelve

months, taking into consideration all available information.

(u) “Grant Date” means, with respect to each Award, the date upon which the Award is granted to an Awardee pursuant to

this Plan, which may be a designated future date as of which such Award will be effective, as determined by the Committee.

(v) “Incentive Stock Option” means an Option that is identified in the Option Agreement as intended to qualify as an

incentive stock option within the meaning of Section 422 of the Code and the regulations promulgated thereunder, and that actually
does so qualify.

(w) “Nonqualified Stock Option” means an Option that is not an Incentive Stock Option.

(x) “Officer” means a person who is an officer of the Company within the meaning of Section 16 of the Exchange Act and

the rules and regulations promulgated thereunder.

(y) “Option” means a right granted under Section 8 of the Plan to purchase a number of Shares at such exercise price, at
such times, and on such other terms and conditions as are specified in the agreement or other documents evidencing the Award (the
“Option

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Agreement”).  Both Incentive Stock Options and Nonqualified Stock Options may be granted under the Plan.

(z) “Other Stock-Based Award” means an Award granted pursuant to Section 12 of the Plan on such terms and conditions as

are specified in the agreement or other documents evidencing the Award (the “Other Stock-Based     Award Agreement ”).

(aa) “Participant”  means  the  Awardee  or  any  person  (including  any  estate)  to  whom  an  Award  has  been  assigned  or

transferred as permitted hereunder.

(bb) “Plan” means this 2016 Stock Incentive Plan, as set forth herein and as hereafter amended from time to time.

(cc) “Qualifying Performance Criteria” shall have the meaning set forth in Section 13(b) of the Plan.

( d d ) “Retirement”  means,  unless  the  Administrator  determines  otherwise,  Termination  of  Employment,  voluntary  or
involuntary, by a Participant from the Company and its Affiliates, other than a Termination for Cause, after attaining age fifty-five
(55)  and  having  at  least  five  (5)  years  of  service  with  the  Company  and  its Affiliates,  excluding  service  with  an Affiliate  of  the
Company prior to the time that such Affiliate became an Affiliate of the Company. For Plan purposes, a “voluntary” Termination of
Employment  is  a  Termination  of  Employment  where  the  Participant  does  not  qualify  for  severance  benefits,  whether  under  a
severance agreement or the Company’s or any of its Affiliate’s severance policy, plan or other arrangement.

   (ee) “Securities Act” means the United States Securities Act of 1933, as amended. (ff) “Share” means a Common Share, as
adjusted in accordance with Section 15 of

the Plan.

(gg) “Stock Appreciation Right”   means  a  right  granted  under  Section  10  of  the  Plan  on  such  terms  and  conditions  as  are

specified in the agreement or other documents evidencing the Award (the “Stock Appreciation Right Agreement”).

(hh) “Stock Award”   means  an  award  or  issuance  of  Shares  or  Stock  Units  made  under  Section  11  of  the  Plan,  the  grant,
issuance, retention, vesting and/or transferability of which is subject during specified periods of time to such conditions (including,
without  limitation,  continued  employment  or  performance  conditions)  and  terms  as  are  expressed  in  the  agreement  or  other
documents evidencing the Award (the “Stock Award Agreement”).

(ii) “Stock  Unit”  means  a  bookkeeping  entry  representing  an  amount  equivalent  to  the  Fair  Market  Value  of  one  Share,
payable in cash, property or Shares. Stock Units represent an unfunded and unsecured obligation of the Company, except as otherwise
provided for by the Administrator.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
(jj) “Subsidiary”  means  any  company  (other  than  the  Company)  in  an  unbroken  chain  of  companies  beginning  with  the
Company,  provided  each  company  in  the  unbroken  chain  (other  than  the  Company)  owns,  at  the  time  of  determination,  stock
possessing 50% or more of the total combined voting power of all classes of stock in one of the other companies in such chain.

(kk) “Termination for Cause”  means,  unless  otherwise  provided  in  an Award Agreement,  Termination  of  Employment  on
account  of  any  act  of  fraud  or  intentional  misrepresentation  or  embezzlement,  misappropriation  or  conversion  of  assets  of  the
Company or any Affiliate, or the intentional and repeated violation of the written policies or procedures of the Company, provided
that,  for  an  Employee  who  is  party  to  an  individual  severance  or  employment  agreement  defining  Cause,  “Cause”  shall  have  the
meaning  set  forth  in  such  agreement  except  as  may  be  otherwise  provided  in  such  agreement.  For  purposes  of  this  Plan,  a
Participant’s Termination of Employment shall be deemed to be a Termination for Cause if, after the Participant’s employment has
terminated,  facts  and  circumstances  are  discovered  that  would  have  justified,  in  the  opinion  of  the  Committee,  a  Termination  for
Cause.

(ll) “Termination  of  Employment”   means  for  purposes  of  this  Plan,  unless  otherwise  determined  by  the  Administrator,
ceasing  to  be  an  Employee  (as  determined  in  accordance  with  Section  3401(c)  of  the  Code  and  the  regulations  promulgated
thereunder) of the Company or one of its Subsidiaries or Affiliates. Unless otherwise determined by the Committee in the terms of an
Award Agreement or otherwise, if a Participant’s employment with the Company and its Affiliates terminates but such Participant
continues to provide services to the Company and its Affiliates in a Non-employee Director capacity, such change in status shall be
deemed  a  Termination  of  Employment. A  Participant  employed  by,  or  performing  services  for,  a  Subsidiary  or  an Affiliate  or  a
division of the Company and its Affiliates shall be deemed to incur a Termination of Employment if, as a result of a Disaffiliation,
such Subsidiary, Affiliate, or division ceases to be a Subsidiary, Affiliate or division, as the case may be, and the Participant does not
immediately  thereafter  become  an  Employee  of  (or  service  provider  for),  or  member  of  the  board  of  directors  of,  the  Company  or
another Subsidiary or Affiliate. Temporary absences from employment because of illness, vacation or leave of absence and transfers
among  the  Company  and  its  Subsidiaries  and  Affiliates  shall  not  be  considered  Terminations  of  Employment.  In  addition,
Termination  of  Employment  shall  mean  a  “separation  from  service”  as  defined  in  regulations  issued  under  Code  Section  409A
whenever necessary to ensure compliance therewith for any payment or settlement of a benefit conferred under this Plan that is subject
to such Code section, and, for such purposes, shall be determined based upon a reduction in the bona fide level of services performed
to a level equal to twenty percent (20%) or less of the average level of services performed by the Employee during the immediately
preceding  36-month  period.  For  the  purposes  of  this  Plan,  Termination  of  Employment  shall  also  mean  the  termination  of  a
Consultant’s  services  to  the  Company  and  the  termination  of  a  Director’s  position  as  a  member  of  the  Board  of  Directors  of  the
Company.

 
 
 
 
 
 
 
 
 
 
3. Stock Subject to the Plan.

(a) Aggregate Limit. Subject to the provisions of Section 15(a) of the Plan, the maximum aggregate number of Shares

which may be subject to Awards granted under the Plan is 10,000 Shares, less one Share for every one Share that was subject to an
option or stock appreciation right granted under any prior plan, and one share for every one Share that was subject to an award other
than an option or stock appreciation right granted under any prior plan. Any Shares that are subject to Options or Stock Appreciation
Rights shall be counted against this limit as one Share for every one Share granted, and any Shares that are subject to Awards other
than Options or Stock Appreciation Rights shall be counted against this limit as one Share for every one Share granted. After the
Effective Date of the Plan (as provided in Section 6), no awards may be granted under any prior plan. Shares subject to or delivered
under Conversion Awards shall not reduce the aggregate number of Shares which may be subject to or delivered under Awards
granted under this Plan. The Shares issued under the Plan may be either Shares reacquired by the Company, including Shares
purchased in the open market, or authorized but unissued Shares.

Notwithstanding any other provision of this Plan, the Company has no prior plans.

(b) Code Section 162(m) and 422 Limits; Other Share Limitations. Subject to the provisions of Section 15(a) of the Plan,
no Employee may be granted under this Plan (i) Options or Stock Appreciation Rights during any calendar year with respect to more
than 1,000 Shares, and (ii) Stock Awards and Other Stock-Based Awards that are intended to comply with the performance-based
exception under Code Section 162(m) and are denominated in Shares under which more than 1,000 Shares may be earned for each
calendar year (or other 12 month period) in the vesting or performance period. During any calendar year, no Participant may be
granted an Award that is intended to comply with the performance-based exception under Code Section 162(m) and is denominated in
cash under which more than one million dollars ($1,000,000.00) may be earned for each calendar year (or other 12 month period) in
the performance period. The foregoing limitations in this section shall be multiplied by two with respect to Awards granted to a
Participant during the first calendar year in which the Participant commences employment with the Company and its Affiliates.
Subject to the provisions of Section 15(a) of the Plan, the aggregate number of Shares that may be subject to all Incentive Stock
Options granted under the Plan shall not exceed 10,000 Shares. Notwithstanding anything to the contrary in the Plan, the limitations
set forth in this Section 3(b) shall be subject to adjustment under Section 15(a) of the Plan only to the extent that such adjustment will
not affect the status of any Award intended to qualify as “performance-based compensation” under Section 162(m) of the Code.

(c) Limit on Awards to Directors. Notwithstanding any other provision of the Plan to the contrary, the aggregate Grant
Date Fair Market Value (computed as of the date of grant in accordance with applicable financial accounting rules) of all Awards
granted to any Non-employee Director during any single calendar year (excluding Awards made at the election of the Non-employee
Director in lieu of all or a portion of annual and committee cash retainers) shall not exceed one million dollars ($1,000,000.00).

 
 
 
 
 
 
 
 
 
 
 
 
(d) Share Counting Rules.

(i) For purposes of this Section 3 of the Plan, Shares subject to Awards that have been canceled, expired, settled in

cash, or forfeited for any reason (in whole or in part) shall not reduce the aggregate number of Shares which may be subject to
Awards granted under this Plan and shall be available for future Awards granted under this Plan in accordance with Section 3(d)
(iii). In addition, if any Shares subject to an award under any prior plan are canceled, expired, settled in cash, or forfeited for any
reason (in whole or in part) after December 31, 2015, then such Shares subject to an award under any prior plan shall, to the extent
of such cancellation, expiration, settlement in cash, or forfeiture, again be available for grant under this Plan in accordance with
Section 3(d)(iii). Notwithstanding the foregoing, Shares added back under the provisions of this subsection (d) shall not be
counted when determining the limit on Shares that may be granted as Incentive Stock Options under subsection (b), above.

(ii) Notwithstanding anything to the contrary contained herein, the following Shares shall not be added to the

Shares authorized for grant under paragraph (i) of this Section: (a) Shares tendered by the Participant or withheld by the Company
in payment of the purchase price of an Option or, after December 31, 2015, an option under any prior plan, (b) Shares tendered by
the Participant or withheld by the Company to satisfy any tax withholding obligation with respect to Options or Stock
Appreciation Rights or, after December 31, 2015, options or stock appreciation rights under any prior plan, (c) Shares subject to a
Stock Appreciation Right or, after December 31, 2015, a stock appreciation right under any prior plan, that are not issued in
connection with its stock settlement on exercise thereof, and (d) Shares reacquired by the Company on the open market or
otherwise using cash proceeds from the exercise of Options or, after December 31, 2015, options under any prior plan. Shares
subject to Awards that have been retained by the Company in payment or satisfaction of the tax withholding obligation of an
Awardee, other than for an Option or Stock Appreciation Right as described above, and Shares that have been delivered (either
actually or constructively by attestation) to the Company in payment or satisfaction of the tax withholding obligation of an
Awardee, other than for an Option or Stock Appreciation Right as described above, shall again be available for grant under the
Plan. Similarly, if any Shares subject to an award under any prior plan are, after December 31, 2015, either retained by the
Company in payment or satisfaction of the tax withholding obligation of an awardee, other than for an option or a stock
appreciation right as described above, or if Shares are delivered (either actually or constructively by attestation) to the Company
in payment or satisfaction of the tax withholding obligation of an awardee under a prior plan, other than for an option or stock
appreciation right, as described above, then such Shares subject to an award under any prior plan shall, to the extent of such
tendering or withholding, again be available for grant under this Plan.

(iii) Any Shares that again become available for grant pursuant to this Section shall be added back as (i) one Share
for every one Share subject to Options or Stock Appreciation Rights granted under the Plan or options or stock appreciation rights

 
 
 
 
 
 
 
 
 
 
 
 
granted  under  any  prior  plan,  and  (ii)  as  one  Share  for  every  one  Share  subject  to  Awards  other  than  Options  or  Stock
Appreciation  Rights  granted  under  the  Plan  or  awards  other  than  options  or  stock  appreciation  rights  granted  under  any  prior
plan.

(iv) Conversion Awards shall not reduce the Shares authorized for grant under the Plan or the limitations on

Awards to a Participant under subsection (b), above, nor shall Shares subject to a Conversion Award again be available for an
Award under the Plan as provided in this subsection (d).

4. Administration of the Plan.

(a) Procedure.

(i) Multiple Administrative Bodies.  The Plan shall be administered by the Board, a Committee designated by the

Board to so administer this Plan and/or their respective delegates.

(ii) Section 162(m). To the extent that the Administrator determines it to be desirable to qualify Awards granted
hereunder as “performance-based compensation” within the meaning of Code Section 162(m), Awards to “covered employees”
(within the meaning of Code Section 162(m)) or to Employees that the Committee determines may be “covered employees” in the
future shall be made by a Committee of two or more “outside directors” within the meaning of Section 162(m) of the Code.
References herein to the Administrator in connection with Awards intended to qualify as “performance-based compensation” shall
mean a Committee meeting the “outside director” requirements of Code Section 162(m). Notwithstanding any other provision of
the Plan, the Administrator shall not have any discretion or authority to make changes to any Award that is intended to qualify as
“performance-based compensation” to the extent that the existence of such discretion or authority would cause such Award not to
so qualify.

(iii) Rule 16b-3. To the extent desirable to qualify transactions hereunder as exempt under Rule 16b-3

promulgated under the Exchange Act (“Rule 16b-3”), Awards to Officers and Directors shall be made by the entire Board or a
Committee of two or more “non-employee directors” within the meaning of Rule 16b-3.

(iv) Other Administration. To the extent required by the rules of the principal

U.S.  national  securities  exchange  on  which  the  Shares  are  traded,  the  members  of  the  Committee  shall  also  qualify  as
“independent directors” as set forth in such rules. Except to the extent prohibited by Applicable Law, the Board or a Committee
may delegate to a Committee of one or more Directors or to authorized officers of the Company the power to approve Awards to
persons eligible to receive Awards under the Plan who are not (A) subject to Section 16 of the Exchange Act or (B) at the time of
such approval, “covered employees” under Section 162(m) of the Code.

(v) Awards to Directors. The Board shall have the power and authority to grant Awards to Non-employee

Directors, including the authority to determine the number and type of awards to be granted; determine the terms and conditions,
not

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
inconsistent with the terms of this Plan, of any award; and to take any other actions the Board considers appropriate in connection
with the administration of the Plan.

(vi) Delegation of Authority for the Day-to-Day Administration of the Plan. Except to the extent prohibited by

Applicable Law, the Administrator may delegate to one or more individuals the day-to-day administration of the Plan and any of
the functions assigned to it in this Plan. Such delegation may be revoked at any time.

(b) Powers of the Administrator. Subject to the provisions of the Plan and, in the case of a Committee or delegates acting as

the Administrator, subject to the specific duties delegated to such Committee or delegates, the Administrator shall have the authority,
in its discretion:

(i) to select the Non-employee Directors, Consultants and Employees of the Company or its Affiliates to whom

Awards are to be granted hereunder;

(ii) to determine the number of Common Shares to be covered by each Award granted hereunder;

(iii) to determine the type of Award to be granted to the selected Employees and Non-employee Directors;

(iv)

to approve forms of Award Agreements;

(v) to determine the terms and conditions, not inconsistent with the terms of the Plan, of any Award granted

hereunder. Such terms and conditions include, but are not limited to, the exercise and/or purchase price, the time or times when an
Award may be exercised (which may or may not be based on performance criteria), the vesting schedule, any vesting and/or
exercisability provisions, terms regarding acceleration of Awards or waiver of forfeiture restrictions, the acceptable forms of
consideration for payment for an Award, the term, and any restriction or limitation regarding any Award or the Shares relating
thereto, based in each case on such factors as the Administrator, in its sole discretion, shall determine and may be established at
the time an Award is granted or thereafter;

(vi)

to correct administrative errors;

(vii) to construe and interpret the terms of the Plan (including sub-plans and Plan addenda) and Awards granted

pursuant to the Plan;

(viii) to adopt rules and procedures relating to the operation and administration of the Plan to accommodate the

specific requirements of local laws and procedures. Without limiting the generality of the foregoing, the Administrator is
specifically authorized (A) to adopt rules and procedures regarding the conversion of local currency, the shift of tax liability from
employer to employee (where legally permitted) and withholding procedures and handling of stock certificates which vary with
local requirements, and (B) to adopt sub-plans and Plan addenda as the

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Administrator deems desirable, to accommodate foreign laws, regulations and practice;

(ix) to prescribe, amend and rescind rules and regulations relating to the Plan, including rules and regulations

relating to sub-plans and Plan addenda;

(x) to modify or amend each Award, including, but not limited to, the acceleration of vesting and/or exercisability,
provided, however, that any such modification or amendment (A) is subject to the plan amendment provisions set forth in Section
16 of the Plan, and (B) may not materially impair any outstanding Award unless agreed to in writing by the Participant, except
that such agreement shall not be required if the Administrator determines in its sole discretion that such modification or
amendment either (Y) is required or advisable in order for the Company, the Plan or the Award to satisfy any Applicable Law or
to meet the requirements of any accounting standard, or (Z) is not reasonably likely to significantly diminish the benefits provided
under such Award, or that adequate compensation has been provided for any such diminishment, except following a Change of
Control;

(xi) to allow or require Participants to satisfy withholding tax amounts by electing to have the Company withhold

from the Shares to be issued upon exercise of a Nonqualified Stock Option or vesting of a Stock Award that number of Shares
having a Fair Market Value equal to the amount required to be withheld. The Fair Market Value of the Shares to be withheld shall
be determined in such manner and on such date that the Administrator shall determine or, in the absence of provision otherwise,
on the date that the amount of tax to be withheld is to be determined. All elections by a Participant to have Shares withheld for
this purpose shall be made in such form and under such conditions as the Administrator may provide;

(xii) to authorize conversion or substitution under the Plan of any or all stock options, stock appreciation rights or

other stock awards held by awardees of an entity acquired by the Company (the “Conversion Awards”). Any conversion or
substitution shall be effective as of the close of the merger or acquisition. The Conversion Awards may be Nonqualified Stock
Options or Incentive Stock Options, as determined by the Administrator, with respect to options granted by the acquired entity;

(xiii) to authorize any person to execute on behalf of the Company any instrument required to effect the grant of

an Award previously granted by the Administrator;

(xiv) to impose such restrictions, conditions or limitations as it determines appropriate as to the timing and manner

of any resale by a Participant or of other subsequent transfers by the Participant of any Shares issued as a result of or under an
Award or upon the exercise of an Award, including, without limitation, (A) restrictions under an insider trading policy, (B)
restrictions as to the use of a specified brokerage firm for such resale or other transfers, and (C) institution of “blackout” periods
on exercises of Awards;

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
(xv) to provide, either at the time an Award is granted or by subsequent action, that an Award shall contain as a
term thereof, a right, either in tandem with the other rights under the Award or as an alternative thereto, of the Participant to receive,
without payment to the Company, a number of Shares, cash or a combination thereof, the amount of which is determined by reference
to the value of the Award; and

granted hereunder.

(xvi) to make all other determinations deemed necessary or advisable for administering the Plan and any Award

(c) Effect of Administrator’s Decision. All questions arising under the Plan or under any Award shall be decided

by the Administrator in its total and absolute discretion. All decisions, determinations and interpretations by the Administrator
regarding the Plan, any rules and regulations under the Plan and the terms and conditions of any Award granted hereunder, shall
be final and binding on all Participants. The Administrator shall consider such factors as it deems relevant, in its sole and absolute
discretion, to making such decisions, determinations and interpretations, including, without limitation, the recommendations or
advice of any officer or other employee of the Company and such attorneys, consultants and accountants as it may select.

(d) Indemnity. To the extent allowable under Applicable Law, each member of the Committee or of the Board and

any person to whom the Board or Committee has delegated any of its authority under the Plan shall be indemnified and held
harmless by the Company from any loss, cost, liability, or expense that may be imposed upon or reasonably incurred by such
person in connection with or resulting from any claim, action, suit, or proceeding to which he or she may be a party or in which he
or she may be involved by reason of any action or failure to act pursuant to the Plan, and against and from any and all amounts
paid by him or her in satisfaction of judgment in such action, suit, or proceeding against him or her; provided he or she gives the
Company an opportunity, at its own expense, to handle and defend the same before he or she undertakes to handle and defend it
on his or her own behalf. The foregoing right of indemnification shall not be exclusive of any other rights of indemnification to
which such persons may be entitled pursuant to the Company’s Articles of Incorporation or By-laws, as a matter of law, or
otherwise, or any power that the Company may have to indemnify them or hold them harmless.

5. Eligibility.

Awards  may  be  granted  only  to  Directors,  Employees  and  Consultants  of  the  Company  or  any  of  its  Affiliates;  provided,
however, that Incentive Stock Options may be granted only to Employees of the Company and its Subsidiaries (within the meaning of
Section 424(f) of the Code).

6. Term of Plan.

The Plan shall become effective upon its approval by shareholders of the Company. It shall continue in effect for a term of ten

(10) years from the date the Plan is approved by the

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
shareholders of the Company (the “ Effective Date”) unless terminated earlier under Section 16 of the Plan.

7. Term of Award.

Subject to the provisions of the Plan, the term of each Award shall be determined by the Administrator and stated in the Award
Agreement, and may extend beyond the termination of the Plan. In the case of an Option or a Stock Appreciation Right, the term shall be
ten (10) years from the Grant Date or such shorter term as may be provided in the Award Agreement. Notwithstanding the foregoing, the
term  of  Awards  other  than  Awards  that  are  structured  to  qualify  as  Incentive  Stock  Options  under  Section  9  shall  be  extended
automatically if the Award would expire at a time when trading in Common Shares is prohibited by law or the Company’s insider trading
policy to the 30th day after the expiration of the prohibition.

8. Options.

The Administrator may grant an Option or provide for the grant of an Option, either from time to time in the discretion of the
Administrator  or  automatically  upon  the  occurrence  of  specified  events,  including,  without  limitation,  the  achievement  of  performance
goals.

(a) Option Agreement. Each Option Agreement shall contain provisions regarding (i) the number of Shares that

may be issued upon exercise of the Option, (ii) the type of Option, (iii) the exercise price of the Option and the means of payment
of such exercise price, (iv) the term of the Option, (v) such terms and conditions regarding the vesting and/or exercisability of an
Option as may be determined from time to time by the Administrator, (vi) restrictions on the transfer of the Option and forfeiture
provisions, and
(vii) such further terms and conditions, in each case not inconsistent with this Plan, as may be determined from time to time by
the Administrator.

(b) Exercise Price. The per share exercise price for the Shares to be issued upon exercise of an Option shall be

determined by the Administrator, except that the per Share exercise price shall be no less than 100% of the Fair Market Value per
Share on the Grant Date, except with respect to Conversion Awards.

(c) No Option Repricings. Subject to Section 15 of the Plan, the exercise price of an Option may not be reduced
without shareholder approval, nor may outstanding Options be cancelled in exchange for cash, other Awards or Options with an
exercise price that is less than the exercise price of the original Option without shareholder approval.

(d) No Reload Grants. Options shall not be granted under the Plan in consideration for and shall not be

conditioned upon the delivery of Shares to the Company in payment of the exercise price and/or tax withholding obligation under
any other employee stock option.

(e) Vesting Period and Exercise Dates. Options granted under this Plan shall vest and/or be exercisable at such
time and in such installments during the period prior to the expiration of the Option’s term as determined by the Administrator
and as specified in the Option Agreement. The Administrator shall have the right to make the timing of the

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
ability to exercise any Option granted under this Plan subject to continued active employment (or retention in the case of a consultant
or  Director),  the  passage  of  time  and/or  such  performance  requirements  as  deemed  appropriate  by  the Administrator. At  any  time
after the grant of an Option, the Administrator may reduce or eliminate any restrictions surrounding any Participant’s right to exercise
all or part of the Option.

(f) Form of Consideration. The Administrator shall determine the acceptable form of consideration for exercising

an Option, including the method of payment, either through the terms of the Option Agreement or at the time of exercise of
an Option. Acceptable forms of consideration may include:

    (i) cash;

(ii) check or wire transfer (denominated in U.S. Dollars);

(iii) subject to any conditions or limitations established by the Administrator, other Shares which were held for a

period of more than six (6) months on the date of surrender and which have a Fair Market Value on the date of surrender equal
to or greater than the aggregate exercise price of the Shares as to which said Option shall be exercised (it being agreed that the
excess of the Fair Market Value over the aggregate exercise price, if any, shall be refunded to the Awardee in cash);

(iv) subject to any conditions or limitations established by the Administrator, the Company withholding Shares

otherwise issuable upon exercise of an Option;

(v) consideration received by the Company under a broker-assisted sale and remittance program acceptable to

the Administrator and in compliance with Applicable Law;

(vi) such other consideration and method of payment for the issuance of Shares to the extent permitted by

Applicable Law; or

(vii)

any combination of the foregoing methods of payment.

(g) Procedure for Exercise; Rights as a Shareholder.

(i) Any Option granted hereunder shall be exercisable according to the terms of the Plan and at such times and

under such conditions as determined by the Administrator and set forth in the applicable Option Agreement.

(ii) An Option shall be deemed exercised when (A) the Company receives (1) written or electronic notice of

exercise (in accordance with the Option Agreement or procedures established by the Administrator) from the person entitled to
exercise the Option and (2) full payment for the Shares with respect to which the related Option is exercised, and (B) with respect
to Nonqualified Stock Options, provisions acceptable to the Administrator have been made for payment of all applicable
withholding taxes.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
(iii) Unless provided otherwise by the Administrator or pursuant to this Plan, until the Shares are issued (as

evidenced by the appropriate entry on the books of the Company or of a duly authorized transfer agent of the Company), no right
to vote or receive dividends or any other rights as a shareholder shall exist with respect to the Shares subject to an Option,
notwithstanding the exercise of the Option.

(iv) The Company shall issue (or cause to be issued) such Shares as soon as administratively practicable after the

Option is exercised. An Option may not be exercised for a fraction of a Share.

(h) Termination of Employment, Consultancy or Board Membership.

(i) The Administrator shall determine as of the Grant Date (subject to modification subsequent to the Grant Date)

the effect a Termination of Employment due to (A) Disability, (B) Retirement, (C) death, or (D) otherwise (including Termination
for Cause) shall have on any Option.

(ii) Unless otherwise provided in the Award Agreement:

(A) Upon termination from membership on the Board by a Non- employee Director for reasons other than

Retirement as set forth in subparagraph (D) below, any Option held by such Director that (1) has not vested and is not
exercisable as of the effective date of such termination from membership on the Board shall be subject to immediate
cancellation and forfeiture or (2) is vested and exercisable as of the effective date of such termination shall remain
exercisable for five (5) years thereafter, or the remaining term of the Option, if less;

(B) Upon Termination of Employment, excluding termination from membership on the Board by a Non-employee
Director, due to death or Disability, any Option held by such Employee that is vested and exercisable as of the effective date
of  such  Termination  of  Employment  shall  remain  exercisable  for  one  year  after  such  Termination  of  Employment  due  to
death or Disability or the remaining term of the Option, if less;

(C) Upon Termination of Employment, excluding termination from membership on the Board by a Non-employee
Director, due to death or Disability, any Option held by such Employee that is not yet vested shall vest in full as of the date
of  death  or  Disability,  and  any  such  vested  Options  shall  remain  exercisable  for  one  year  after  such  Termination  of
Employment due to death or Disability or the remaining term of the Option, if less;

(D) Upon Termination of Employment due to Retirement, (1) any Option held by such Awardee shall, to the extent
not already vested, become ratably vested (rounded up or down to the nearest whole Share) based upon the full months of the
applicable vesting period elapsed as of the end of the month in which the Termination of Employment due to Retirement
occurs over the total number of months in such period; provided, however, that, in the case of a

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Retirement  due  to  a  voluntary  Termination  of  Employment,  the  terms  of  this  Section  8(h)(ii)(D)(1)  shall  not  apply  with
respect to any Option granted less than six (6) months prior to the effective date of such Termination of Employment; and (2)
any  Option  held  by  an  Awardee  at  Retirement,  to  the  extent  vested  and  exercisable  as  of  the  effective  date  of  such
Retirement  (including,  without  limitation,  any  Options  that  have  ratably  vested  pursuant  to  the  preceding  clause  (1)),  will
remain outstanding for the lesser of five (5) years or the remaining term of the Option; and

(E)"  Any  other  Termination  of  Employment,  termination  from  membership  on  the  Board  by  a  Non-employee
Director,  shall  result  in  immediate  cancellation  and  forfeiture  of  all  outstanding  Options  that  have  not  vested  as  of  the
effective  date  of  such  Termination  of  Employment,  and  any  vested  and  exercisable  Options  held  at  the  time  of  such
Termination of Employment shall remain exercisable for ninety (90) days thereafter, or the remaining term of the Option, if
less. Notwithstanding the foregoing, all outstanding and unexercised Options shall be immediately cancelled in the event of a
Termination for Cause.

9. Incentive Stock Option Limitations/Terms.

(a) Eligibility. Only employees (as determined in accordance with Section 3401(c) of the Code and the regulations

promulgated thereunder) of the Company or any of its Subsidiaries may be granted Incentive Stock Options. No Incentive Stock
Option shall be granted to any such employee who as of the Grant Date owns stock possessing more than 10% of the total combined
voting power of the Company, except in compliance with Section 422 of the Code regarding 10 – percent shareholders.

(b) $100,000 Limitation. Notwithstanding the designation “Incentive Stock Option” in an Option Agreement, if and to the

extent that the aggregate Fair Market Value of the Shares with respect to which Incentive Stock Options are exercisable for the first
time by the Awardee during any calendar year (under all plans of the Company and any of its Subsidiaries) exceeds U.S. $100,000,
such Options shall be treated as Nonqualified Stock Options. For purposes of this Section 9(b) of the Plan, Incentive Stock Options
shall be taken into account in the order in which they were granted. The Fair Market Value of the Shares shall be determined as of the
Grant Date.

(c) Transferability. The Option Agreement must provide that an Incentive Stock Option is not transferable by the Awardee

otherwise than by will or the laws of descent and distribution, and, during the lifetime of such Awardee, must not be exercisable by
any other person. If the terms of an Incentive Stock Option are amended to permit transferability, the Option will be treated for tax
purposes as a Nonqualified Stock Option.

(d) Exercise Price. The per Share exercise price of an Incentive Stock Option shall in no event be inconsistent with the

requirements for qualification of the Incentive Stock Option under Section 422 of the Code.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
(e) Other Terms. Option Agreements evidencing Incentive Stock Options shall contain such other terms and

conditions as may be necessary to qualify, to the extent determined desirable by the Administrator, with the applicable provisions
of Section 422 of the Code. If any such terms and conditions, as of the Grant Date or any later date, do not so comply, the Option
will be treated thereafter for tax purposes as a Nonqualified Stock Option.

10. Stock Appreciation Rights.

A “Stock Appreciation Right” is a right that entitles the Awardee to receive, in cash or Shares (as determined by the

Administrator), value equal to or otherwise based on the excess of

(i) the Fair Market Value of a specified number of Shares at the time of exercise over (ii) the aggregate exercise price of the right, as
established by the Administrator on the Grant Date. Stock Appreciation Rights may be granted to Awardees either alone (“freestanding”)
or in addition to or in tandem with other Awards granted under the Plan and may, but need not, relate to a specific Option granted under
Section 8 of the Plan. Any Stock Appreciation Right granted in tandem with an Option may be granted at the same time such Option is
granted or at any time thereafter before exercise or expiration of such Option, and shall be based on the Fair Market Value of one Share on
the Grant Date or, if applicable, on the Grant Date of the Option with respect to a Stock Appreciation Right granted in exchange for or in
tandem with, but subsequent to, the Option (subject to the requirements of Section 409A of the Code). All Stock Appreciation Rights under
the Plan, other than Conversion Awards, shall be granted subject to the same terms and conditions applicable to Options as set forth in
Section 8 of the Plan. Subject to the provisions of Section 8 of the Plan, the Administrator may impose such other conditions or restrictions
on any Stock Appreciation Right as it shall deem appropriate.

11.  Stock Awards.

(a) Stock Award Agreement. Each Stock Award Agreement shall contain provisions regarding (i) the number of
Shares subject to such Stock Award or a formula for determining such number, (ii) the purchase price of the Shares, if any, and
the means of payment for the Shares, (iii) the performance criteria, if any, and level of achievement versus these criteria that shall
determine the number of Shares granted, issued, retainable and/or vested, (iv) such terms and conditions on the grant, issuance,
vesting and/or forfeiture of the Shares as may be determined from time to time by the Administrator, (v) restrictions on the
transferability of the Stock Award, and (vi) such further terms and conditions, in each case not inconsistent with this Plan, as may
be determined from time to time by the Administrator. The Committee may, in its sole discretion, waive the vesting restrictions
and any other conditions set forth in any Award Agreement under such terms and conditions as the Committee shall deem
appropriate, subject to the limitations imposed under Code Section 162(m) and the regulations thereunder in the case of an Award
intended to comply with the performance-based exception under Code Section 162(m), unless determined otherwise under the
circumstances by the Committee.

(b) Restrictions and Performance Criteria. The grant, issuance, retention and/or vesting of Stock Awards issued

to Employees may be subject to such performance criteria and level of achievement versus these criteria as the Administrator
shall determine, which

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
criteria  may  be  based  on  financial  performance,  personal  performance  evaluations  and/or  completion  of  service  by  the Awardee.
Notwithstanding  anything  to  the  contrary  herein,  the  performance  criteria  for  any  Stock  Award  that  is  intended  to  satisfy  the
requirements for “performance-based compensation” under Section 162(m) of the Code (a “Performance Stock Award ”)  shall  be
established by the Administrator based on one or more Qualifying Performance Criteria selected by the Administrator and specified in
writing  not  later  than  ninety  (90)  days  after  the  commencement  of  the  period  of  service  (or,  if  earlier,  the  elapse  of  25%  of  such
period) to which the performance goals relate or otherwise within the time period required by the Code or the applicable Treasury
Regulations, provided that the outcome is substantially uncertain at that time. Stock Awards for which vesting is not based on the
attainment of performance criteria are referred to as “Restricted Stock Awards.”

(c) Termination of Employment or Board Membership.

(i) The Administrator shall determine as of the Grant Date (subject to modification subsequent to the Grant Date)
the effect a Termination of Employment due to (A) Disability, (B) Retirement (C) death, or (D) otherwise (including Termination
for Cause) shall have on any Stock Award.

(ii) Unless otherwise provided in the Award Agreement:

(A) A Termination of Employment due to Disability or death shall result in immediate full vesting of any as yet
unvested Stock Award, and in the case of a Stock Award that vests upon the achievement of performance goals, the vested
amount shall be based upon the target award amount;

(B) A  Termination  of  Employment  due  to  Retirement  shall  result  in  vesting  of  a  prorated  portion  of  any  Stock
Award (rounded up or down to the nearest whole Share), based upon the full months of the applicable performance period,
vesting period or other period of restriction elapsed as of the end of the month in which the Termination of Employment due
to Retirement occurs over the total number of months in such period; provided, however, that, in the case of a Retirement due
to  voluntary  Termination  of  Employment,  the  terms  of  this  Section  11(c)(ii)(B)  shall  not  apply  with  respect  to  any  Stock
Award granted less than six (6) months prior to the effective date of such Termination of Employment; and

(C) Any other Termination of Employment shall result in immediate cancellation and forfeiture of all outstanding,

unvested Stock Awards.

If clause (B) of this Section 11(c)(ii) applies to a Stock Award under which vesting is based on the attainment of
performance criteria over a performance period, the ratable vesting percentage determined by the portion of the performance
period during which the Awardee was an Employee of the Company or an Affiliate shall be applied to determine the portion
of the Stock

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Award that is vested based upon actual performance results after the completion of the performance period.

(d) Rights as a Shareholder. Unless otherwise provided for by the Administrator, the Participant shall have the rights

equivalent to those of a shareholder and shall be a shareholder only after Shares are issued (as evidenced by the appropriate entry on
the books of the Company or of a duly authorized transfer agent of the Company) to the Participant.

12. Other Stock-Based Awards.

(a) Other Stock-Based Awards. An “Other Stock-Based Award” means any other type of equity-based or equity-related
Award not otherwise described by the terms of this Plan (including the grant or offer for sale of unrestricted Shares), as well as any
cash bonus based on the attainment of Qualifying Performance Criteria as described in Section 13(b), in such amount and subject to
such terms and conditions as the Administrator shall determine. Such Awards may involve the transfer of actual Shares to
Participants, or payment in cash or otherwise of amounts based on the value of Shares or pursuant to attainment of a performance
goal. Each Other Stock-Based Award will be evidenced by an Award Agreement containing such terms and conditions as may be
determined by the Administrator.

(b) Value of Other Stock-Based Awards. Each Other Stock-Based Award shall be expressed in terms of Shares or units

based on Shares or a target amount of cash, as determined by the Administrator. The Administrator may establish performance goals
in its discretion. If the Administrator exercises its discretion to establish performance goals, the number and/or value of Other Stock-
Based Awards that will be paid out to the Participant will depend on the extent to which the performance goals are met.
Notwithstanding anything to the contrary herein, the performance criteria for any Other Stock-Based Award that is intended to satisfy
the requirements for “performance-based compensation” under Section 162(m) of the Code shall be established by the Administrator
based on one or more Qualifying Performance Criteria selected by the Administrator and specified in writing not later than ninety (90)
days after the commencement of the period of service (or, if earlier, the elapse of 25% of such period) to which the performance goals
relate and otherwise within the time period required by the Code and the applicable Treasury Regulations, provided that the outcome
is substantially uncertain at that time.

(c) Payment of Other Stock-Based Awards. Payment, if any, with respect to Other Stock-Based Awards shall be made in

accordance with the terms of the Award, in cash or Shares or a combination thereof, as the Administrator determines.

(d) Termination of Employment, Consultancy, or Board Membership.

(i) The Administrator shall determine as of the Grant Date (subject to modification subsequent to the Grant Date)

the effect a Termination of Employment

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
due to (A) Disability, (B) Retirement, (C) death, or (D) otherwise (including Termination for Cause) shall have on any Other
Stock-Based Award.

(ii) Unless otherwise provided in the Award Agreement:

(A) A Termination of Employment due to Disability or death shall result in immediate full vesting of any as yet
unvested Other Stock-Based Award, and in the case of an Other Stock-Based Award which vests on the basis of attainment
of a performance goal, the vested amount shall be based upon the target award amount;

(B) A  Termination  of  Employment  due  to  Retirement  shall  result  in  vesting  of  a  prorated  portion  of  any  Other
Stock-Based Award (rounded up or down to the nearest whole Share or unit based on Shares, as applicable), based upon the
full months of the applicable performance period, vesting period or other period of restriction elapsed as of the end of the
month in which the Termination of Employment due to Retirement occurs over the total number of months in such period;
provided, however, that, in the case of a Retirement due to voluntary Termination of Employment, the terms of this Section
12(d)(ii)(B)  shall  not  apply  with  respect  to  any  Other  Stock-Based Award  granted  less  than  six  (6)  months  prior  to  the
effective date of such Termination of Employment; and

(C) Any other Termination of Employment shall result in immediate cancellation and forfeiture of all outstanding,

unvested Other Stock-Based Awards.

If clause (B) of this Section 12(d)(ii) applies to an Other Stock-Based Award under which vesting is based on the
attainment of performance criteria over a performance period, the ratable vesting percentage determined by the portion of
the  performance  period  during  which  the Awardee  was  an  Employee  of  the  Company  or  an Affiliate  shall  be  applied  to
determine  the  portion  of  the  Other  Stock-Based  Award  that  is  vested  based  upon  actual  performance  results  after  the
completion of the performance period.

13. Other Provisions Applicable to Awards.

(a) Non-Transferability of Awards. Unless determined otherwise by the Administrator, an Award may not be sold, pledged,
assigned, hypothecated, transferred or disposed of in any manner other than by beneficiary designation, will or by the laws of descent
or distribution, including but not limited to any attempted assignment or transfer in connection with the settlement of marital property
or other rights incident to a divorce or dissolution, and any such attempted sale, assignment or transfer shall be of no effect prior to the
date an Award is vested and settled. The Administrator may only make an Award transferable to an Awardee’s family member or any
other person or entity provided the Awardee does not receive consideration for such transfer. If the Administrator makes an Award
transferable, either as of the Grant Date or thereafter, such Award shall contain

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
such additional terms and conditions as the Administrator deems appropriate, and any transferee shall be deemed to be bound by such
terms upon acceptance of such transfer.

(b) Qualifying Performance Criteria. For purposes of this Plan, the term “Qualifying Performance Criteria” shall mean any

one or more of the following performance criteria, either individually, alternatively or in any combination, on a basis consistent with
U.S. Generally Accepted Accounting Principles (“GAAP”) or on a non-GAAP or adjusted GAAP basis, applied to either the
Company as a whole or to a Subsidiary, business unit, Affiliate or business segment, either individually, alternatively or in any
combination, and measured either annually or cumulatively over a period of years, on an absolute basis or relative to a pre-established
target, to previous years’ results or to a designated comparison group, in each case as specified by the Committee in the Award or by
duly adopted resolution: (i) sales or cash return on sales; (ii) cash flow or free cash flow or net cash from operating activity; (iii)
earnings (including gross margin, earnings before or after interest and taxes, earnings before taxes, and net earnings); (iv) basic or
diluted earnings per share; (v) growth in earnings or earnings per share; (vi) stock price; (vii) return on equity or average shareholders’
equity; (viii) total shareholder return; (ix) return on capital; (x) return on assets or net assets; (xi) return on investments; (xii) revenue
or gross profits; (xiii) income before or after interest, taxes, depreciation and amortization, or net income; (xiv) pretax income before
allocation of corporate overhead and bonus; (xv) operating income or net operating income; (xvi) operating profit or net operating
profit (whether before or after taxes); (xvii) operating margin; (xviii) return on operating revenue; (xix) working capital or net
working capital; (xx) market share; (xxi) asset velocity index; (xxii) contract awards or backlog; (xxiii) overhead or other expense or
cost reduction; (xxiv) growth in shareholder value relative to the moving average of the S&P 500 Index or a peer group index; (xxv)
credit rating; (xxvi) strategic plan development and implementation; (xxvii) improvement in workforce diversity; (xxviii) customer
satisfaction; (xxvix) employee satisfaction; (xxx) management succession plan development and implementation; and (xxxi) employee
or customer retention. With respect to any Award that is intended to satisfy the requirements for “performance-based compensation”
under Section 162(m) of the Code, the performance criteria must be Qualifying Performance Criteria, and the Administrator will
(within the first quarter of the performance period, but in no event more than ninety (90) days into that period) establish the specific
performance targets (including thresholds and whether to exclude certain extraordinary, non-recurring, or similar items) and Award
amounts (subject to the right of the Administrator to exercise discretion to reduce payment amounts following the conclusion of the
performance period). Extraordinary, non-recurring items that may be the basis of adjustment include acquisitions or divestitures,
restructurings, discontinued operations, extraordinary items, and other unusual or non-recurring charges, an event either not directly
related to the operations of the Company, Subsidiary, division, business segment or business unit or not within the reasonable control
of management, the cumulative effects of tax or accounting changes in accordance with U.S. GAAP, and foreign exchange gains or
losses.

(c) Certification. Prior to the payment of any compensation under an Award intended to qualify as “performance-based

compensation” under Section 162(m) of the Code, the Administrator shall certify in writing the extent to which any Qualifying
Performance

 
 
 
 
 
 
 
Criteria and any other material terms under such Award have been satisfied (other than in cases where such criteria relate solely
to the increase in the value of the Common Shares).

(d) Discretionary Adjustments Pursuant to Section 162(m). Notwithstanding satisfaction or completion of any Qualifying

Performance Criteria, to the extent specified as of the Grant Date, the number of Shares, Options or other benefits granted, issued,
retainable and/or vested under an Award on account of satisfaction of such Qualifying Performance Criteria may be reduced (but not
increased) by the Administrator on the basis of such further considerations as the Administrator in its sole discretion shall determine.

(e) Six Month Holding Period for Purposes of Rule 16b-3. If the Company is subject to the reporting requirements of

Section 13 of the Exchange Act, the Plan Administrator shall ensure that transactions between the Company and an Officer or Director
under this Plan are exempt from Section 16(b) of the Exchange Act pursuant to one of the exemptions available under 17 C.F.R. 240.16b-3.
If the Administrator determines that the exemption pursuant to 17 C.F.R. 240.16b-3(d)(3) is to be used, then (i) shares purchased upon
exercise of an Option or another derivative security (as defined in Exchange Act Rule 16a-1(c)) issued under this Plan by an Officer or
Director may not be sold before at least six months have elapsed from the date the Option or other derivative security was granted; and (ii)
any other equity securities of the Company acquired by an Officer or Director under this Plan other than as described in subparagraph (i)
above may not be sold before at least six months have elapsed from the date they equity security was acquired.

14. Dividends and Dividend Equivalents.

Awards other than Options and Stock Appreciation Rights may provide the Awardee with the right to receive dividend payments
or  dividend  equivalent  payments  on  the  Shares  subject  to  the  Award,  whether  or  not  such  Award  is  vested.  Notwithstanding  the
foregoing, dividends or dividend equivalents shall not be paid with respect to Stock Awards or Other Stock-Based Awards that, in either
case, vest based on the achievement of performance goals prior to the date the performance goals are satisfied and the Award is earned,
and then shall be payable only with respect to the number of Shares or Stock Units actually earned under the Award. Such payments may
be made in cash, Shares or Stock Units or may be credited as cash or Stock Units to an Awardee’s account and later settled in cash or
Shares or a combination thereof, as determined by the Administrator. Such payments and credits may be subject to such conditions and
contingencies as the Administrator may establish.

15. Adjustments upon Changes in Capitalization, Organic Change or Change of Control.

(a) Adjustment Clause. In the event of (i) a stock dividend, extraordinary cash dividend, stock split, reverse stock

split, share combination, or recapitalization or similar event affecting the capital structure of the Company (each, a “Share
Change”), or (ii) a merger, consolidation, acquisition of property or shares, separation, spin-off, reorganization, liquidation,
Disaffiliation, or similar event affecting the Company or any of its Subsidiaries (each, an “Organic Change”), the Administrator
or the Board may in its discretion make such substitutions or adjustments as it deems appropriate and equitable

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
to (i) the Share limitations set forth in Section 3 of the Plan, (ii) the number and kind of Shares covered by each outstanding Award,
and (iii) the price per Share subject to each such outstanding Award. In the case of Organic Changes, such adjustments may include,
without limitation, (x) the cancellation of outstanding Awards in exchange for payments of cash, property or a combination thereof
having an aggregate value equal to the value of such Awards, as determined by the Administrator or the Board in its sole discretion (it
being understood that in the case of an Organic Change with respect to which shareholders receive consideration other than publicly
traded equity securities of the ultimate surviving entity, any such determination by the Administrator that the value of an Option or
Stock Appreciation Right shall for this purpose be deemed to equal the excess, if any, of the value of the consideration being paid for
each Share pursuant to such Organic Change over the exercise price of such Option or Stock Appreciation Right shall conclusively be
deemed  valid);  (y)  the  substitution  of  other  property  (including,  without  limitation,  cash  or  other  securities  of  the  Company  and
securities  of  entities  other  than  the  Company)  for  the  Shares  subject  to  outstanding  Awards;  and  (z)  in  connection  with  any
Disaffiliation, arranging for the assumption of Awards, or replacement of Awards with new awards based on other property or other
securities (including, without limitation, other securities of the Company and securities of entities other than the Company), by the
affected  Subsidiary,  Affiliate,  or  division  or  by  the  entity  that  controls  such  Subsidiary,  Affiliate,  or  division  following  such
Disaffiliation (as well as any corresponding adjustments to Awards that remain based upon Company securities). The Committee may
adjust  in  its  sole  discretion  the  Qualifying  Performance  Criteria  applicable  to  any Awards  to  reflect  any  Share  Change  and  any
Organic  Change  and  any  unusual  or  non-recurring  events  and  other  extraordinary  items,  impact  of  charges  for  restructurings,
discontinued operations, and the cumulative effects of accounting or tax changes, each as defined by GAAP or as identified in the
Company’s  financial  statements,  notes  to  the  financial  statements,  management’s  discussion  and  analysis  or  the  Company’s  other
SEC filings, provided that in the case of Qualifying Performance Criteria applicable to any performance-based Awards intended to
qualify under Code Section 162(m), such adjustment does not violate Section 162(m) of the Code. Any adjustment under this Section
15(a) need not be the same for all Participants.

(b) Change of Control. In the event of a Change of Control, unless otherwise determined by the Administrator as of
the Grant Date of a particular Award (or subsequent to the Grant Date), the following acceleration, exercisability and valuation
provisions shall apply:

(i) On the date that such Change of Control occurs, any or all Options and Stock Appreciation Rights awarded

under this Plan not previously exercisable and vested shall become fully exercisable and vested.

(ii) Except as may be provided in an individual severance or employment agreement (or severance plan) to which
an Awardee is a party, in the event of an Awardee’s Termination of Employment within two (2) years after a Change of Control
for any reason other than because of the Awardee’s death, Retirement, Disability or Termination for Cause, each Option and
Stock Appreciation Right held by the Awardee (or a transferee) that is vested shall remain exercisable until the

 
 
 
 
 
 
 
 
 
 
 
earlier  of  the  third  (3 rd)  anniversary  of  such  Termination  of  Employment  (or  any  later  date  until  which  it  would  remain
exercisable  under  such  circumstances  by  its  terms)  or  the  expiration  of  its  original  term.  In  the  event  of  an  Awardee’s
Termination  of  Employment  more  than  two  (2)  years  after  a  Change  of  Control,  or  within  two  (2)  years  after  a  Change  of
Control because of the Awardee’s death, Retirement, Disability or Termination for Cause, the provisions of Sections 8(h) and 10
of the Plan shall govern (as applicable).

(iii) On the date that such Change of Control occurs, the restrictions and conditions applicable to any or all Stock

Awards and Other Stock-Based Awards shall lapse and such Awards shall be fully vested. Unless otherwise provided in an
Award at the Grant Date, upon the occurrence of a Change of Control, any performance based Award shall be deemed fully
earned at the target amount as of the date on which the Change of Control occurs. All Stock Awards, Other Stock-Based Awards
and cash Awards shall be settled or paid within thirty (30) days of vesting hereunder. Notwithstanding the foregoing, if the
Change of Control would not qualify as a permissible date of distribution under Section 409A(a)(2)(A) of the Code, and the
regulations thereunder, the Awardee shall be entitled to receive the payment of cash or settlement of Shares under the Award, as
applicable, from the Company on the date that would have applied absent this provision.

(iv) The Administrator, in its discretion, may determine that, upon the occurrence of a Change of Control of the

Company, each Option and Stock Appreciation Right outstanding shall terminate within a specified number of days after notice to
the Participant, and/or that each Participant shall receive, with respect to each Share subject to such Option or Stock Appreciation
Right, an amount equal to the excess of the Fair Market Value of such Share immediately prior to the occurrence of such Change
of Control over the exercise price per Share of such Option and/or Stock Appreciation Right; such amount to be payable in cash,
in one or more kinds of stock or property (including the stock or property, if any, payable in the transaction) or in a combination
thereof, as the Committee, in its discretion, shall determine, and if there is no excess value, the Committee may, in its discretion,
cancel such Awards.

(c) Section 409A. Notwithstanding the foregoing: (i) any adjustments made pursuant to Section 15(a) of the Plan to Awards

that are considered “deferred compensation” within the meaning of Section 409A of the Code shall be made in compliance with the
requirements of Section 409A of the Code; (ii) any adjustments made pursuant to Section 15(a) of the Plan to Awards that are not
considered “deferred compensation” subject to Section 409A of the Code shall be made in such a manner as to ensure that after such
adjustment, the Awards either continue not to be subject to Section 409A of the Code or comply with the requirements of Section
409A of the Code; (iii) the Administrator shall not have the authority to make any adjustments pursuant to Section 15(a) of the Plan to
the extent that the existence of such authority would cause an Award that is not intended to be subject to Section 409A of the Code to
be subject thereto; and (iv) if any Award is subject to Section 409A of the Code, Section 15(b) of the Plan shall be applicable only to
the extent specifically provided in the Award Agreement and permitted pursuant to

 
 
 
 
 
 
 
 
 
 
 
 
Section 24 of the Plan in order to ensure that such Award complies with Code Section 409A.

16. Amendment and Termination of the Plan.

(a) Amendment and Termination. The Board may amend, alter or discontinue the Plan or any Award Agreement, but any

such amendment shall be subject to approval of the shareholders of the Company in the manner and to the extent required by
Applicable Law. In addition, without limiting the foregoing, unless approved by the shareholders of the Company and subject to
Section 16(b), no such amendment shall be made that would:

(i) increase the maximum aggregate number of Shares which may be subject to Awards granted under the Plan;

(ii) reduce the minimum exercise price for Options or Stock Appreciation Rights granted under the Plan; or

(iii) reduce the exercise price of outstanding Options or Stock Appreciation Rights, as prohibited by Section 8(c)

without shareholder approval.

(b) Effect of Amendment or Termination. No amendment, suspension or termination of the Plan shall materially impair the

rights of any Participant with respect to an outstanding Award, unless mutually agreed otherwise between the Participant and the
Administrator, which agreement must be in writing and signed by the Participant and the Company, except that no such agreement
shall be required if the Administrator determines in its sole discretion that such amendment either (i) is required or advisable in order
for the Company, the Plan or the Award to satisfy any Applicable Law or to meet the requirements of any accounting standard, or (ii)
is not reasonably likely to significantly diminish the benefits provided under such Award, or that any such diminishment has been
adequately compensated, except that this exception shall not apply following a Change of Control. Termination of the Plan shall not
affect the Administrator’s ability to exercise the powers granted to it hereunder with respect to Awards granted under the Plan prior to
the date of such termination.

(c) Effect of the Plan on Other Arrangements. Neither the adoption of the Plan by the Board or a Committee nor the

submission of the Plan to the shareholders of the Company for approval shall be construed as creating any limitations on the power of
the Board or any Committee to adopt such other incentive arrangements as it or they may deem desirable, including without
limitation, the granting of restricted shares or restricted share units or stock options otherwise than under the Plan, and such
arrangements may be either generally applicable or applicable only in specific cases.

17. Designation of Beneficiary.

(a) An Awardee may file a written designation of a beneficiary who is to receive the Awardee’s rights pursuant to

Awardee’s Award or the Awardee may include his or her Awards in an omnibus beneficiary designation for all benefits under the
Plan. To the extent that Awardee has completed a designation of beneficiary while employed with the

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Company, such beneficiary designation shall remain in effect with respect to any Award hereunder until changed by the Awardee
to the extent enforceable under Applicable Law.

(b) Such designation of beneficiary may be changed by the Awardee at any time by written notice. In the event of the

death of an Awardee and in the absence of a beneficiary validly designated under the Plan who is living at the time of such Awardee’s
death, the Company shall allow the legal representative of the Awardee’s estate to exercise the Award.

18. No Right to Awards or to Employment.

No person shall have any claim or right to be granted an Award and the grant of any Award shall not be construed as giving an
Awardee the right to continue in the employ of the Company or its Affiliates. Further, the Company and its Affiliates expressly reserve the
right,  at  any  time,  to  dismiss  any  Employee  or Awardee  at  any  time  without  liability  or  any  claim  under  the  Plan,  except  as  provided
herein or in any Award Agreement entered into hereunder.

19. Legal Compliance.

Shares shall not be issued pursuant to an Option, Stock Appreciation Right, Stock Award or Other Stock-Based Award unless
such  Option,  Stock Appreciation  Right,  Stock Award  or  Other  Stock-Based Award  and  the  issuance  and  delivery  of  such  Shares  shall
comply with Applicable Law, specifically including without limitation all applicable federal and state securities laws and regulations, and
shall  be  further  subject  to  the  approval  of  counsel  for  the  Company  with  respect  to  such  compliance.  Unless  the Awards  and  Shares
covered by this Plan have been registered under the Securities Act or the Company has determined that such registration is unnecessary,
each person receiving an Award and/or Shares pursuant to any Award may be required by the Company (a) to give a representation in
writing  that  such  person  is  acquiring  such  Shares  for  his  or  her  own  account  for  investment  and  not  with  a  view  to,  or  for  sale  in
connection  with,  the  distribution  of  any  part  thereof,  and  (b)  to  make  such  additional  representations,  warranties,  and  agreements  with
respect to the investment intent of such person or persons as the Company may request.

All certificates for Shares or certificates, agreements, or other documents evidencing securities delivered under the Plan shall be
subject  to  such  stop-transfer  orders  and  other  restrictions  as  the  Company  may  deem  advisable  under  the  rules,  regulations,  and  other
requirements of the Securities and Exchange Commission, any securities law, and the Company may cause a legend or legends to be put
on any such certificates, agreements or other documents to make appropriate reference to such restrictions.

In the case of the exercise of an Option by a person or estate acquiring the right to exercise such Option by bequest or inheritance,
the Administrator  may  require  reasonable  evidence  as  to  the  ownership  of  such  Option  and  may  require  such  consents  and  releases  of
taxing authorities as the Administrator deems advisable.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
20. Inability to Obtain Authority.

To the extent the Company is unable to or the Administrator deems it unfeasible to obtain authority from any regulatory body
having jurisdiction, which authority is deemed by the Company’s counsel to be advisable or necessary to the lawful issuance and sale of
any Shares hereunder, the Company shall be relieved of any liability with respect to the failure to issue or sell such Shares as to which
such requisite authority shall not have been obtained.

21. Reservation of Shares.

The  Company,  during  the  term  of  this  Plan,  will  at  all  times  reserve  and  keep  available  such  number  of  Shares  as  shall  be

sufficient to satisfy the requirements of the Plan.

22. Notice.

Any written notice to the Company required by any provisions of this Plan shall be addressed to the Secretary of the Company
and  shall  be  effective  when  received. Any  notice  to  a  Participant  hereunder  shall  be  addressed  to  the  last  address  of  record  with  the
Company and shall be effective when sent via first class mail, courier service, or electronic mail to such last address of record.

23. Governing Law; Interpretation of Plan and Awards.

(a) This Plan and all determinations made and actions taken pursuant hereto shall be governed by the substantive

laws, but not the choice of law rules, of the state of Delaware, except as to matters governed by U.S. federal law.

(b) In the event that any provision of the Plan or any Award granted under the Plan is declared to be illegal,

invalid or otherwise unenforceable by a court of competent jurisdiction, such provision shall be reformed, if possible, to the extent
necessary to render it legal, valid and enforceable, or otherwise deleted, and the remainder of the terms of the Plan and/or Award
shall not be affected except to the extent necessary to reform or delete such illegal, invalid or unenforceable provision.

(c) The headings preceding the text of the sections hereof are inserted solely for convenience of reference, and

shall not constitute a part of the Plan, nor shall they affect its meaning, construction or effect.

(d) The terms of the Plan and any Award shall inure to the benefit of and be binding upon the parties hereto and

their respective permitted heirs, beneficiaries, successors and assigns.

24. Section 409A.

It is the intention of the Company that no Award shall be “deferred compensation” subject to Section 409A of the Code, unless
and to the extent that the Administrator specifically determines otherwise, and the Plan and the terms and conditions of all Awards shall be
interpreted accordingly. The terms and conditions governing any Awards that the Administrator

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
determines will be subject to Section 409A of the Code, including any rules for elective or mandatory deferral of the delivery of cash or
Shares pursuant thereto and any rules regarding treatment of such Awards in the event of a Change of Control, shall be set forth in the
applicable Award Agreement, deferral election forms and procedures, and rules established by the Administrator, and shall comply in all
respects with Section 409A of the Code. The following rules will apply to Awards intended to be subject to Section 409A of the Code
(“409A Awards”):

(a) If a Participant is permitted to elect to defer an Award or any payment under an Award, such election will be

permitted only at times in compliance with Code Section 409A.

(b) The Company shall have no authority to accelerate distributions relating to 409A Awards in excess of the

authority permitted under Section 409A.

(c) Any distribution of a 409A Award following a Termination of Employment that would be subject to Code

Section 409A(a)(2)(A)(i) as a distribution following a separation from service of a “specified employee” as defined under Code
Section 409A(a)(2)(B)(i), shall occur no earlier than the expiration of the six-month period following such Termination of
Employment.

(d) In the case of any distribution of a 409A Award, if the timing of such distribution is not otherwise specified in

the Plan or an Award Agreement or other governing document, the distribution shall be made not later than the end of the
calendar year during which the settlement of the 409A Award is specified to occur.

(e) In the case of an Award providing for distribution or settlement upon vesting or the lapse of a risk of

forfeiture, if the time of such distribution or settlement is not otherwise specified in the Plan or an Award Agreement or other
governing document, the distribution or settlement shall be made not later than March 15 of the year following the year in which
the Award vested or the risk of forfeiture lapsed.

(f) Notwithstanding anything herein to the contrary, in no event shall the Company or the Administrator be liable
for the payment of, or any gross up payment in connection with, any taxes or penalties owed by the Participant pursuant to Code
Section 409A.

25. Limitation on Liability.

The Company and any Affiliate which is in existence or hereafter comes into existence shall not be liable to a Participant, an

Employee, an Awardee or any other persons as to:

(a) The Non-Issuance of Shares. The non-issuance or sale of Shares as to which the Company has been unable to

obtain from any regulatory body having jurisdiction the authority deemed by the Company’s counsel to be necessary to the lawful
issuance and sale of any shares hereunder; and

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
(b) Tax or Exchange Control Consequences. Any tax consequence or any exchange control obligation owed, by

any Participant, Employee, Awardee or other person due to the receipt, exercise or settlement of any Option or other Award
granted hereunder.

26. Unfunded Plan.

Insofar as it provides for Awards, the Plan shall be unfunded. Although bookkeeping accounts may be established with respect to
Awardees  who  are  granted  Stock Awards  or  Other  Stock-Based Awards  under  this  Plan,  any  such  accounts  will  be  used  merely  as  a
bookkeeping convenience. The Company shall not be required to segregate any assets which may at any time be represented by Awards,
nor shall this Plan be construed as providing for such segregation. Neither the Company nor the Administrator shall be deemed to be a
trustee of stock or cash to be awarded under the Plan. Any liability of the Company to any Participant with respect to an Award shall be
based solely upon any contractual obligations which may be created by the Plan; no such obligation of the Company shall be deemed to be
secured  by  any  pledge  or  other  encumbrance  on  any  property  of  the  Company.  Neither  the  Company  nor  the Administrator  shall  be
required to give any security or bond for the performance of any obligation which may be created by this Plan.

27. Foreign Employees.

Awards may be granted hereunder to Employees and Consultants who are foreign nationals, who are located outside the United
States or who are not compensated from a payroll maintained in the United States, or who are otherwise subject to (or could cause the
Company  to  be  subject  to)  legal  or  regulatory  provisions  of  countries  or  jurisdictions  outside  the  United  States,  on  such  terms  and
conditions different from those specified in the Plan as may, in the judgment of the Administrator, be necessary or desirable to foster and
promote achievement of the purposes of the Plan, and, in furtherance of such purposes, the Administrator may make such modifications,
amendments, procedures, or subplans as may be necessary or advisable to comply with such legal or regulatory provisions.

28. Tax Withholding.

Each Participant shall pay to the Company, or make arrangements satisfactory to the Company regarding the payment of, any
federal, state, local or foreign taxes of any kind required by law to be withheld with respect to any Award under the Plan no later than the
date as of which any amount under such Award first becomes includible in the gross income of the Participant for any tax purposes with
respect to which the Company has a tax withholding obligation. Unless otherwise determined by the Company, withholding obligations
may be settled with Shares, including Shares that are part of the Award that gives rise to the withholding requirement; provided, however,
that not more than the legally required minimum withholding may be settled with Shares that are part of the Award. The obligations of
the Company under the Plan shall be conditional on such payment or arrangements, and the Company and its Affiliates shall, to the extent
permitted by law, have the right to deduct any such taxes from any vested Shares or any other payment due to the participant at that time
or at any future time. The Administrator may establish such procedures as it deems appropriate, including making irrevocable elections,
for the settlement of withholding obligations with Shares.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
29. Cancellation of Award; Forfeiture of Gain.

Notwithstanding anything to the contrary contained herein, an Award Agreement may provide that the Award will be cancelled
and the Participant will forfeit the Shares or cash received or payable on the vesting or exercise of the Award, and that the amount of any
proceeds of the sale or gain realized on the vesting or exercise of the Award must be repaid to the Company, under such conditions as
may be required by Applicable Law or established by the Committee in its sole discretion.

30. Data Privacy and Transfer

As  a  condition  of  acceptance  of  an Award,  the  Participant  explicitly  thereby  consents  to  the  collection,  use  and  transfer,  in
electronic  or  other  form,  of  personal  data  by  and  among,  as  applicable,  the  Company  and  its Affiliates  for  the  exclusive  purpose  of
implementing, administering and managing the Participant’s participation in the Plan. The Participant understands that the Company and
its  Affiliates  hold  certain  personal  information  about  the  Participant,  including  the  Participant’s  name,  home  address  and  telephone
number,  date  of  birth,  social  security  or  other  identification  number,  salary,  nationality,  job  title,  Shares  held  in  the  Company  or  any
Subsidiary, details of all Awards or any other entitlement to Shares awarded, canceled, exercised, vested, unvested or outstanding in the
Participant’s  favor,  for  the  purpose  of  implementing,  managing  and  administering  the  Plan  (the  “Data”).  The  Participant  further
understands that the Company and its Affiliates may transfer the Data among themselves as necessary for the purpose of implementation,
management and administration of the Plan, and that the Company and its Affiliates may each further transfer the Data to any third parties
assisting  the  Company  in  the  implementation,  management,  and  administration  of  the  Plan.  The  Participant  understands  that  these
recipients may be located in the Participant’s country, or elsewhere, and that the recipient’s country may have different data privacy laws
and protections than the Participant’s country. The Participant understands that he or she may request a list with the names and addresses
of any potential recipients of the Data by contacting his or her local human resources representative. The Participant, through participation
in the Plan and acceptance of an Award under the Plan, authorizes such recipients to receive, possess, use, retain and transfer the Data, in
electronic or other form, for the purposes of implementing, administering and managing the Plan, including any requisite transfer of such
Data  as  may  be  required  to  a  broker  or  other  third  party  with  whom  the  Participant  may  elect  to  deposit  any  Shares.  In  addition,  by
accepting an Award under the Plan, each Participant agrees and acknowledges (i) that the Data will be held only as long as is necessary to
implement,  manage,  and  administer  the  Plan;  (ii)  that  the  Participant  may,  at  any  time,  view  the  Data,  request  additional  information
about the storage and processing of the Data, require any necessary amendments to the Data, or refuse or withdraw consent to the use and
transfer  of  the  Data,  without  cost,  by  delivering  such  revocation  or  withdrawal  of  consent  in  writing  to  a  designated  human  resources
representative; and (iii) that refusal or withdrawal of consent may affect the Participant’s ability to participate in the Plan thereafter.

 
 
 
 
 
 
 
 
 
 
 
This Plan was adopted by the Board of Directors of the Company on April 4, 2016.

This Plan was approved by the stockholders of the Company on April 4, 2016.

MONOPAR THERAPEUTICS INC.

  04/04/2016

By: /s/ Chandler D. Robinson

Name: Chandler D. Robinson
Title: CEO

.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
EXECUTIVE EMPLOYMENT AGREEMENT

This Executive Employment Agreement (the "Agreement") is entered into as of January 1, 2017, by and between Chandler D. Robinson
("Executive") and Monopar Therapeutics Inc. (the "Company").

Whereas, the Company desires to employ Executive as its Chief Executive Officer effective as of January 1, 2017 (the "Effective Date"),
and Executive desires to serve in such capacity, pursuant to the terms and conditions set forth in this Agreement; and

Now, Therefore, in consideration of the mutual promises and covenants contained herein, it is hereby agreed by and between the parties
hereto as follows:

ARTICLE I

DEFINITIONS

For purposes of the Agreement, the following terms are defined as follows:

1.1. "Board" means the Board of Directors of the Company.

1.2.  "Cause" means any of the following events described below:

   (a) Executive's conviction of a felony or other crime involving moral turpitude;

   (b) any willful act or acts of dishonesty undertaken by Executive and intended to result in substantial gain or personal enrichment of
Executive, Executive's family or any third party at the expense of the Company;

   (c) any willful act of gross misconduct which is materially and demonstrably injurious to the Company; and/or

   (d) Executive's inability under applicable law to continue to work lawfully in the United States.

For the purpose of this Agreement, no act, or failure to act, by Executive shall be considered "willful" if done, or omitted to be done, by him
in good faith and in the reasonable belief that his act or omission was in the best interest of the Company and/or required by applicable law.

1.3. "Change in Control" means the occurrence of any of the following events: (i) any sale or exchange of the capital stock by the
stockholders of the Company in one transaction or series of related transactions where more than fifty percent (50%) of the outstanding

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
voting  power  of  the  Company  is  acquired  by  a  person  or  entity  or  group  of  related  persons  or  entities;  or  (ii)  any  reorganization,
consolidation  or  merger  of  the  Company  where  the  outstanding  voting  securities  of  the  Company  immediately  before  the  transaction
represent  or  are  converted  into  less  than  fifty  percent  (50%)  of  the  outstanding  voting  power  of  the  surviving  entity  (or  its  parent
corporation) immediately after the transaction; or (iii) the consummation of any transaction or series of related transactions that results in
the sale of all or substantially all of the assets of the Company; or (iv) any "person" or "group" (as defined in the Securities Exchange Act
of 1934, as amended (the "Exchange Act") becoming the "beneficial owner" (as defined in Rule 13d-3 under the Exchange Act) directly or
indirectly of securities representing more than fifty percent (50%) of the voting power of the Company then outstanding. Except that any
change in the beneficial ownership of the securities of the Company as a result of a private financing of the Company that is approved by
the Board, shall not be deemed to be a Change in Control.

1.4.     "Change in Control Multiple" shall mean one and a half (1.5).

1.5. "Change in Control Period" means that period commencing on the consummation of a Change in Control and ending on the first
anniversary thereof.

1.6. "COBRA" means the Consolidated Omnibus Budget Reconciliation Act of 1985, as amended.

1.7.     "Code" means the Internal Revenue Code of 1986, as amended.

1.8.     "Company" means Monopar Therapeutics Inc. or any successor thereto.

 1.9. "Confidential Disclosure Agreement" means the Confidential Disclosure Agreement entered into between Executive and the
Company.

1.10.   "Covered Termination" means (a) an Involuntary Termination Without Cause or (b) a voluntary termination for Good Reason,
provided that the termination constitutes a Separation from Service.

1.11. "Good Reason" means Executive's resignation as a result of a Good Reason Condition. In order to resign for Good Reason,
Executive must provide written notice to the Company of the existence of the Good Reason Condition within thirty (30) days of the initial
existence of such Good Reason Condition. Upon receipt of such notice of the Good Reason Condition, the Company will be provided with
a period of thirty (30) days during which it may remedy the Good Reason Condition and not be required to provide for the payments and
benefits described in Section 4 as a result of such proposed resignation due to the Good Reason Condition specified in the notice. If the
Good Reason Condition is not remedied within the period specified in the preceding sentence, Executive may resign for Good Reason
based on the Good Reason Condition specified in the notice, provided that

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
such resignation must occur within sixty (60) days after the initial existence of such Good Reason Condition.

1.12. "Good Reason Condition" means that any of the following are undertaken without Executive's express written consent:

    (a)     a material reduction in Executive's Base Salary;

    (b)    a material diminution in Executive's responsibilities;

    (c)    the Company's material breach of any material term of this Agreement; or

   (d) a requirement that Executive relocate to an office that would increase Executive's one-way commute distance by more than fifty (50)
miles based on Executive's primary residence at the time such relocation is announced.

1.13. "Involuntary Termination Without Cause" means Executive's dismissal or discharge by the Company other than for Cause. The
termination of Executive's employment as a result of Executive's death or inability to perform the essential functions of his job due to
disability will not be deemed to be an Involuntary Termination Without Cause.

1.14. "Separation from Service" means Executive's termination of employment or service where such termination of employment or
service constitutes a "separation from service" within the meaning of Treasury Regulation Section l.409A-l(h).

ARTICLE II

EMPLOYMENT BY THE COMPANY

2.1. Position and Duties. Subject to terms set forth herein, as of the Effective Date, Executive shall serve as the Company's Chief
Executive Officer and perform such duties as are customarily associated with the position of Chief Executive Officer and such other duties
as are assigned to Executive by the Board. During the term of Executive's employment with the Company, Executive will devote
Executive's best efforts and substantially all of Executive's business time and attention (except for vacation periods and reasonable periods
of illness or other incapacities permitted by the Company's general employment policies, if any, or as otherwise set forth in this Agreement)
to the business of the Company.

2.2. Employment at Will. Both the Company and Executive shall have the right to terminate Executive's employment with the Company
at any time, with or without Cause, and without prior notice. If Executive's employment with the Company is terminated, Executive will be
eligible to receive severance benefits to the extent provided in this

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Agreement.

      2.3. Employment Policies. The employment relationship between the parties shall also be governed by the general employment
policies and practices of the Company, if any, including those relating to protection of confidential information and assignment of
inventions, except that when the terms of this Agreement differ from or are in conflict with the Company's general employment policies or
practices, this Agreement shall control.

ARTICLE ID
COMPENSATION

      3.1. Base Salary. As of the Effective Date, Executive shall receive for services to be rendered hereunder an annual base salary of
$300,000 ("Base Salary"), payable on the regular payroll dates of the Company, subject to increase in the sole discretion of the Board.

     3.2. Annual Bonus. Executive is subject to an annual bonus at the discretion of the Board.

     3.3. Standard Company Benefits. Executive shall be entitled to all rights and benefits for which Executive is eligible under the terms
and conditions of the standard Company benefits and compensation practices, if any, that may be in effect from time to time and are
provided by the Company to its executive employees generally. Executive shall be entitled each year to four (4) weeks leave for vacation at
full pay, provided, that the maximum amount Executive may have accrued at any point in time is four (4) weeks (meaning that once
Executive has accrued four (4) weeks, Executive will not accrue any additional vacation time until he takes vacation and falls below the
four (4) week accrual cap). Executive shall also be entitled to reasonable holidays and illness days with full pay in accordance with the
policies applicable to the Company and its affiliates, if any, from time to time in effect. Employee acknowledges and agrees that in order to
maintain flexibility, the Company and its affiliates have the right to amend or terminate any employee benefit plan at any time. Until the
Company obtains both retirement and healthcare benefits for eligible employees, Executive shall be entitled to an additional cash payment
of at least
$6,250 per month or such greater amount as determined by the Board; reduced, however, for any given month by any employer
contributions made for that month by the company to a qualified retirement plan/account established by the company for Executive.

     3.4. Stock Options. Subject to approval by the Board, Executive may be granted options to purchase shares of the Company's common
stock with an exercise price per share as determined by the Compensation Committee or similar function of the Board.

     3.5. Expenses. The Company will reimburse  Executive for all reasonable and necessary expenses incurred by Employee in connection
with the Company's business, provided at such expenses incurred and are properly documented and accounted for m accordance with

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
the policy of the Company and requirements of the Internal Revenue Service.

ARTICLE IV
SEVERANCE AND CHANGE IN CONTROL BENEFITS

    4.1. Severance Benefits. Upon Executive's termination of employment, Executive shall receive any accrued but unpaid Base Salary and
other accrued and unpaid compensation, including any Annual Bonus that has been earned with respect to a prior year, but remains unpaid
as of the date of the termination. If the termination is due to a Covered Termination or permanent disability, provided that Executive first
returns all Company property in his possession and, within sixty (60) days following the Covered Termination, executes and does not
revoke an effective general release of all claims against the Company and its affiliates in a form reasonably acceptable to the Company and
Executive (a "Release of Claims"), Executive shall also be entitled to receive the following severance benefits described in this Section
4.1.

    (a) Covered Termination Not Related to a Change in Control. If Executive's employment terminates due to a Covered Termination
which occurs outside of a Change in Control Period, Executive shall receive the following:

    (i) An amount equal to twelve (12) months of Executive's Base Salary payable in substantially equal installments in accordance with the
Company's normal payroll policies, if any, less applicable withholdings, with such installments to commence as soon as administratively
practicable following the date the Release of Claims is not subject to revocation and, in any event, within sixty (60) days following the date
of the Covered Termination.

    (ii) If Executive elects to receive continued healthcare coverage pursuant to the provisions of COBRA, the Company shall directly pay,
or reimburse Executive for, the premium for Executive and Executive's covered dependents through the earlier of (i) the first anniversary of
the date of Executive's termination of employment and (ii) the date Executive and Executive's covered dependents, if any, become eligible
for healthcare coverage under another employer's plan(s). Notwithstanding the foregoing, (i) if any plan pursuant to which such benefits are
provided is not, or ceases prior to the expiration of the period of continuation coverage to be, exempt from the application of Section 409A
of the Code under Treasury Regulation Section 1.409A-l(a)(5), or (ii) the Company is otherwise unable to continue to cover Executive
under its group health plans without penalty under applicable law (including without limitation, Section 2716 of the Public Health Service
Act), then, in either case, an amount equal to each remaining Company subsidy shall thereafter be paid to Executive in substantially equal
monthly installments. After the Company ceases to pay premiums pursuant to this Section 4.l(a)(ii), Executive may, if eligible, elect to
continue healthcare coverage at Executive's expense in accordance with the

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
provisions of COBRA.

    (iii) All of Employee's vested options or stock appreciation rights with respect to the Company's common stock shall remain exercisable
until the first anniversary of Executive's termination of employment (or, if earlier, the maximum period specified in the award documents
and plans governing such options or stock appreciation rights, as applicable, assuming Executive's employment had not terminated).

    (b) Covered Termination Related to a Change in Control. If Executive's employment terminates due to a Covered Termination that
occurs during a Change in Control Period, Executive shall receive the following:

    (i) Executive shall be entitled to receive an amount equal to the Change in Control Multiplier multiplied by the sum of: (i) Executive's
Base Salary and (ii) Executive's target Annual Bonus for the fiscal year of Executive's termination, in each case, at the rate equal to the
higher of (x) the rate in effect immediately prior to Executive's termination of employment or (y) the rate in effect immediately prior to the
Change in Control payable in a cash lump sum, less applicable withholdings, as soon as administratively practicable following the date the
Release of Claims is not subject to revocation and, in any event, within sixty (60) days following the date of the Covered Termination.

    (ii) If Executive elects to receive continued healthcare coverage pursuant to the provisions of COBRA, the Company shall directly pay,
or reimburse Executive for, the premium for Executive and Executive's covered dependents through the earlier of (i) the date that is that
number of years equal to the Change in Control Multiplier following the date of Executive's termination of employment and (ii) the date
Executive and Executive's covered dependents, if any, become eligible for healthcare coverage under another employer's plan(s).
Notwithstanding the foregoing, (i) if any plan pursuant to which such benefits are provided is not, or ceases prior to the expiration of the
period of continuation coverage to be, exempt from the application of Section 409A of the Code under Treasury Regulation Section l.409A-
l(a)(5), or (ii) the Company is otherwise unable to continue to cover Executive under its group health plans without penalty under
applicable law (including without limitation, Section 2716 of the Public Health Service Act), then, in either case, an amount equal to each
remaining Company subsidy shall thereafter be paid to Executive in substantially equal monthly installments. After the Company ceases to
pay premiums pursuant to this Section 4.l(b)(ii), Executive may, if eligible, elect to continue healthcare coverage at Executive's expense in
accordance with the provisions of COBRA.

    (iii) Each outstanding equity award, including, without limitation, each stock option and restricted stock award, held by Executive shall
automatically become vested and, if applicable, exercisable and any forfeiture restrictions or rights of repurchase thereon shall immediately
lapse, in each case, with respect to one hundred percent (100%) of the shares subject thereto. To the extent vested after giving effect to the
acceleration provided in the

 
 
 
 
 
 
 
 
 
 
 
 
 
 
preceding sentence, each stock option held by Executive shall remain exercisable until the earlier of the original expiration date for such
stock option or the second anniversary of Executive's Covered Termination.

    (c) Termination for Death or Disability. If Executive's employment is terminated due to death or permanent disability where the
Company makes a determination in good faith that, due to a mental or physical incapacity, Executive has been unable to perform his duties
under this Agreement for a period of not less than six (6) consecutive months or 180 days in the aggregate in any 12-month period,
Executive shall receive the following:

    (i) An amount equal to three (3) months of Executive's Base Salary payable in substantially equal installments in accordance with the
Company's normal payroll policies, less applicable withholdings, with such installments to commence as soon as administratively
practicable following the date the Release of Claims is not subject to revocation and, in any event, within sixty (60) days following the date
of the Covered Termination.

    (ii) If Executive (or in the event of death, his designee) elects to receive continued healthcare coverage pursuant to the provisions of
COBRA, the Compan:Y shall directly pay, or reimburse Executive for, the premium for Executive and Executive's covered dependents
through the earlier of (i) the three (3) month anniversary of the date of Executive's termination of employment and (ii) the date Executive
and Executive's covered dependents, if any, become eligible for healthcare coverage under another employer's plan(s). Notwithstanding the
foregoing, (i) if any plan pursuant to which such benefits are provided is not, or ceases prior to the expiration of the period of continuation
coverage to be, exempt from the application of Section 409A of the Code under Treasury Regulation Section l.409A-l(a)(5), or (ii) the
Company is otherwise unable to continue to cover Executive under its group health plans without penalty under applicable law (including
without limitation, Section 2716 of the Public Health Service Act), then, in either case, an amount equal to each remaining Company
subsidy shall thereafter be paid to Executive in substantially equal monthly installments. After the Company ceases to pay premiums
pursuant to this Section 4.l(b)(ii), Executive may, if eligible, elect to continue healthcare coverage at Executive's expense in accordance the
provisions of COBRA.

    4.2. 280G Provisions. Notwithstanding anything in this Agreement to the contrary, if any payment or distribution Executive would
receive pursuant to this Agreement or otherwise ("Payment") would (a) constitute a "parachute payment" within the meaning of Section
280G of the Code, and (b) but for this sentence, be subject to the excise tax imposed by Section 4999 of the Code (the "Excise Tax"), then
such Payment shall either be (i) delivered in full, or (ii) delivered as to such lesser extent which would result in no portion of such Payment
being subject to the Excise Tax, whichever of the foregoing amounts, taking into account the applicable federal, state and local income
taxes and the Excise Tax, results in the receipt by Executive on an after-tax basis, of the largest payment, notwithstanding

 
 
 
 
 
 
 
 
 
 
 
 
that all or some portion the Payment may be taxable under Section 4999 of the Code. The accounting firm engaged by the Company for
general audit purposes as of the day prior to the effective date of the Change in Control shall perform the foregoing calculations. The
Company shall bear all expenses with respect to the determinations by such accounting firm required to be made hereunder. The
accounting firm shall provide its calculations to the Company and Executive within fifteen (15) calendar days after the date on which
Executive's right to a Payment is triggered (if requested at that time by the Company or Executive) or such other time as requested by the
Company or Executive. Any good faith determinations of the accounting firm made hereunder shall be final, binding and conclusive upon
the Company and Executive. Any reduction in payments and/or benefits pursuant to this Section 4.2 will occur in the following order: (1)
reduction of cash payments; (2) cancellation of accelerated vesting of equity awards other than stock options; (3) cancellation of
accelerated vesting of stock options; and (4) reduction of other benefits payable to Executive.

    4.3. Section 409A.

    (a) Notwithstanding any provision to the contrary in this Agreement, if Executive is deemed at the time· of his Separation from Service to
be a "specified employee" for purposes of Section 409A(a)(2)(B)(i) of the Code, to the extent delayed commencement of any portion of the
benefits to which Executive is entitled under this Agreement is required in order to avoid a prohibited distribution under Section 409A(a)(2)
(B)(i) of the Code which would subject Executive to a tax obligation under Section 409A of the Code, such portion of Executive's benefits
shall not be provided to Executive prior to the earlier of (i) the expiration of the six- month period measured from the date of the
Executive's Separation from Service or (ii) the date of Executive's death. Upon the expiration of the applicable Code Section 409A(a)(2)(B)
(i) period, all payments deferred pursuant to this Section 4.3(a) shall be paid in a lump sum to Executive, and any remaining payments due
under the Agreement shall be paid as otherwise provided herein.

    (b) Any reimbursements payable to Executive pursuant to the Agreement shall be paid to Executive no later than 30 days after Executive
provides the Company with a written request for reimbursement, and to the extent that any such reimbursements are deemed to constitute
"nonqualified deferred compensation" within the meaning of Section 409A of the Code (i) such amounts shall be paid or reimbursed to
Executive promptly, but in no event later than December 31 of the year following the year in which the expense is incurred,  (ii) the amount
of any such payments eligible for reimbursement in one year shall not affect the payments or expenses that are eligible for payment or
reimbursement in any other taxable year, and (iii) Executive's right to such payments or reimbursement shall not be subject to liquidation or
exchange for any other benefit.

    (c) For purposes of Section 409A of the Code (including, without limitation, for purposes of Treasury Regulation Section l.409A-2(b)(2)
(iii)), Executive's right to receive

 
 
 
 
 
 
 
 
 
 
 
installment payments under the Agreement shall be treated as a right to receive a series of separate payments and, accordingly, each
installment payment hereunder shall at all times be considered a separate and distinct payment.

    4.4. Mitigation. Executive shall not be required to mitigate damages or the amount of any payment provided under this Agreement by
seeking other employment or otherwise, nor shall the amount of any payment provided for under this Agreement be reduced by any
compensation earned by Executive as a result of employment by another employer or by any retirement benefits received by Executive
after the date of the Covered Termination, or otherwise.

ARTICLEV

PROPRIETARY INFORMATION OBLIGATIONS

    5.1. Agreement. Executive agrees to continue to abide by the Confidential Disclosure Agreement

    5.2. Remedies. Executive's duties under the Confidential Disclosure·Agreementshall survive termination of Executive's employment
with the Company and the termination of this Agreement. Executive acknowledges that a remedy at law for any breach or threatened breach
by Executive of the provisions of the Confidential Disclosure Agreement, as well as Executive's obligations pursuant to Section 6.2 and
Article 7 below, would be inadequate, and Executive therefore agrees that the Company shall be entitled to seek injunctive relief in case of
any such breach or threatened breach.

ARTICLE VI OUTSIDE ACTIVITIES

    6.1. Other Activities.

    (a) Executive shall not, during the term of this Agreement undertake or engage in any other employment, occupation or business
enterprise, other than ones in which Executive is a passive investor, unless he obtains the prior written consent of the Board.

    (b) Executive may engage in civic and not-for-profit activities so long as such activities do not materially interfere with the performance
of Executive's duties hereunder. In addition, Executive shall be allowed to serve as a member of the board of directors of up to two (2) other
for profit entities at any time during the term of this Agreement, which service shall not materially interfere with the performance of
Executive's duties hereunder; provided, however, that the Board may require that Executive resign from one or both of such director
positions if it can reasonably and in good faith demonstrate that such resignation(s) would be in the best interests of the Company in a
significant and material way.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
    6.2. Competition. Executive agrees that, from the date hereof until a period of twelve  (12) months following the date of termination of
Executive's employment with the Company, Executive will not directly or indirectly, either as an employee, employer, consultant, agent,
principal, partner, corporate officer, director, or in any other individual or representative capacity, engage or participate in any "Competitive
Business" anywhere in the United States of America. As used herein, a "Competitive Business" is defined as any business developing
uPAR antibodies to treat cancer, or clonidine to treat oral mucositis.

ARTICLE VII NONINTERFERENCE

In addition to Executive's obligations under the Confidential Disclosure Agreement, Executive shall not for a period of one (1) year
following Executive's termination of employment for any reason, either on Executive's own account or jointly with or as a manager, agent,
officer, employee, consultant, partner, joint venturer, owner or stockholder or otherwise on behalf of any other person, firm or corporation,
directly or indirectly solicit or attempt to solicit away from the Company any of its officers or employees or offer employment to any person
who is an officer or employee of the Company;provided, however, that a general advertisement to which an employee of the Company
responds shall in no event be deemed to result in a breach of this Article 7. Executive also agrees not to harass or disparage the Company or
its employees, clients, directors or agents or divert or attempt to divert any actual or potential business of the Company. The provisions of
this Article 7 shall survive the termination or expiration of the applicable Executive's employment with the Company and shall be fully
enforceable thereafter. If it is determined by a court of competent jurisdiction in any state that any restriction in this Article 7 is excessive in
duration or scope or is unreasonable or unenforceable under the laws of that state, it is the intention of the parties that such restriction may
be modified or amended by the court to render it enforceable to the maximum extent permitted by the law of that state.

ARTICLE VIII GENERAL PROVISIONS

    8.1. Notices. Any notices provided hereunder must be in writing and shall be deemed effective upon the earlier of personal delivery
(including personal delivery by facsimile) or the third day after mailing by first class mail, to the Company at its primary office location
and to Executive at Executive's address as listed on the Company payroll.

    8.2. Tax Withholding. Executive acknowledges that all amounts and benefits payable under this Agreement are subject to deduction and
withholding to the extent required by applicable law.

Severability. Whenever possible, each prov1s1on of this Agreement will be interpreted in such manner as to be effective and valid under
applicable law, but if any

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
provision of this Agreement is held to be invalid, illegal or unenforceable in any respect under any applicable law or rule in any jurisdiction,
such invalidity, illegality or unenforceability will not affect any other provision or any other jurisdiction, but this Agreement will be
reformed, construed and enforced in such jurisdiction as if such invalid, illegal or unenforceable provisions had never been contained
herein.

    8.3. Waiver. If either party should waive any breach of any prov1s1ons of this Agreement, they shall not thereby be deemed to have
waived any preceding or succeeding breach of the same or any other provision of this Agreement. ·

    8.4. Complete Agreement. This Agreement constitutes the entire agreement between Executive and the Company and is the complete,
final, and exclusive embodiment of their agreement with regard to this subject matter, and will supersede all prior agreements,
understandings, discussions, negotiations and undertakings, whether written or oral, between the parties with respect to the subject matter
hereof, including without limitation, the Prior Agreement. This Agreement is entered into without reliance on any promise or representation
other than those expressly contained herein or therein. and cannot be modified or amended except in a writing signed by an officer·-of the.
Company and Executive.

    8.5. Counterparts. This Agreement may be executed in separate counterparts, any one of which need not contain signatures of more than
one party, but all of which taken together will constitute one and the same Agreement.

    8.6. Headings. The headings of the sections hereof are inserted for convenience only and shall not be deemed to constitute a part hereof
nor to affect the meaning thereof.

    8.7. Successors and Assigns. This Agreement is intended to bind and inure to the benefit of and be enforceable by Executive and the
Company, and their respective successors, assigns, heirs, executors and administrators, except that Executive may not assign his rights or
delegate his duties or obligations hereunder without the prior written consent of the Company.

    8.8. Arbitration. Unless otherwise prohibited by law or specified below, all disputes, claims and causes of action, in law or equity,
arising from or relating to this Agreement or its enforcement, performance, breach, or interpretation shall be resolved solely and
exclusively by final and binding arbitration held in Illinois in conformity with the then​ existing employment arbitration rules and Illinois
law. The arbitrator shall: (a) provide adequate discovery for the resolution of the dispute; and (b) issue a written arbitration decision, to
include the arbitrator's essential findings and conclusions and a statement of the award. However, nothing in this section is intended to
prevent either party from obtaining injunctive relief in court to prevent irreparable harm pending the conclusion of any such arbitration. The
Company shall bear the costs of any such arbitration.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
    8.9. Executive Acknowledgement. Executive acknowledges that (a) he has consulted with or has had the opportunity to consult with
independent counsel of his own choice concerning this Agreement, and has been advised to do so by the Company, and (b) that he has read
and understands the Agreement, is fully aware of its legal effect and has entered into it freely based on his own judgment.

    8.10. Choice of Law. All questions concerning the construction, validity and interpretation of this Agreement will be governed by the law
of the State of Illinois without regard to the conflicts of law provisions thereof.

In Witness Whereof, the parties have executed this Agreement as of the date first written

above.

On behalf of Monopar Therapeutics Inc.

  /s/ Christopher M. Starr
  Christopher M. Starr, Ph.D.
  Executive Chairman

Accepted and Agreed:

/s/ Chandler D. Robinson
Chandler D. Robinson

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
AMENDED AND RESTATED EXECUTIVE EMPLOYMENT AGREEMENT

This Amended and Restated Executive Employment Agreement (the “ Agreement”) is entered into as of November 1,
2017,  by  and  between  Chandler  D.  Robinson  (“Executive”)  and  Monopar  Therapeutics  Inc.  (the  “ Company”)  and
replaces  in  its  entirety  the  Executive  Employment Agreement  by  and  between  Executive  and  the  Company  dated
January 1, 2017.

Whereas, the Company desires to retain the employment of Executive as its Chief Executive Officer effective as of
November 1, 2017 (the “Effective Date”), and Executive desires to serve in such capacity, pursuant to the terms and
conditions set forth in this Agreement; and

Now, Therefore, in consideration of the mutual promises and covenants contained herein, it is hereby agreed by and
between the parties hereto as follows:

ARTICLE I DEFINITIONS

For purposes of the Agreement, the following terms are defined as follows:

1.1. “Board” means the Board of Directors of the Company.

1.2. “Cause” means any of the following events described below:

(a) Executive’s conviction of a felony or other crime involving moral turpitude;

(b) any willful act or acts of dishonesty undertaken by Executive and intended to result in substantial gain or personal

enrichment of Executive, Executive’s family or any third party at the expense of the Company;

(c) any willful act of gross misconduct which is materially and demonstrably injurious to the Company; and/or

(d) Executive’s inability under applicable law to continue to work lawfully in the United States.

For  the  purpose  of  this Agreement,  no  act,  or  failure  to  act,  by  Executive  shall  be  considered  “willful”  if  done,  or
omitted to be done, by him in good faith and in the reasonable belief that his act or omission was in the best interest of
the Company and/or required by applicable law.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
1.3. “Change  in  Control ”  means  the  occurrence  of  any  of  the  following  events:  (i)  any  sale  or  exchange  of  the
capital stock by the stockholders of the Company in one transaction or series of related transactions where more than
fifty  percent  (50%)  of  the  outstanding  voting  power  of  the  Company  is  acquired  by  a  person  or  entity  or  group  of
related persons or entities; or (ii) any reorganization, consolidation or merger of the Company where the outstanding
voting  securities  of  the  Company  immediately  before  the  transaction  represent  or  are  converted  into  less  than  fifty
percent (50%) of the outstanding voting power of the surviving entity (or its parent corporation) immediately after the
transaction; or (iii) the consummation of any transaction or series of related transactions that results in the sale of all or
substantially all of the assets of the Company; or (iv) any “person” or “group” (as defined in the Securities Exchange
Act of 1934, as amended (the “Exchange Act”) becoming the “beneficial owner” (as defined in Rule 13d-3 under the
Exchange Act) directly or indirectly of securities representing more than fifty percent (50%) of the voting power of the
Company then outstanding. Except that any change in the beneficial ownership of the securities of the Company as a
result  of  a  private  financing  of  the  Company  that  is  approved  by  the  Board,  shall  not  be  deemed  to  be  a  Change  in
Control.

1.4. “Change in Control Multiple ” shall mean one and a half (1.5).

1.5. “Change in Control Period ” means that period commencing on the consummation of a Change in Control and

ending on the first anniversary thereof.

1.6. “COBRA” means the Consolidated Omnibus Budget Reconciliation Act of 1985, as amended.

1.7. “Code” means the Internal Revenue Code of 1986, as amended.

1.8. “Company” means Monopar Therapeutics Inc. or any successor thereto.

1.9. “Confidential Disclosure Agreement” means the Confidential Disclosure Agreement entered into between

Executive and the Company.

    1.10.    “Covered Termination” means (a) an Involuntary Termination Without Cause or

(b) a voluntary termination for Good Reason, provided that the termination constitutes a Separation from Service.

1.11. “Good Reason” means Executive’s resignation as a result of a Good Reason Condition. In order to resign for
Good Reason, Executive must provide written notice to the Company of the existence of the Good Reason Condition
within  thirty  (30)  days  of  the  initial  existence  of  such  Good  Reason  Condition.  Upon  receipt  of  such  notice  of  the
Good Reason Condition, the Company will be provided with a period of thirty (30) days during which it may remedy
the Good Reason Condition and not be required to provide for the

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
payments  and  benefits  described  in  Section  4  as  a  result  of  such  proposed  resignation  due  to  the  Good  Reason
Condition  specified  in  the  notice.  If  the  Good  Reason  Condition  is  not  remedied  within  the  period  specified  in  the
preceding  sentence,  Executive  may  resign  for  Good  Reason  based  on  the  Good  Reason  Condition  specified  in  the
notice,  provided  that  such  resignation  must  occur  within  sixty  (60)  days  after  the  initial  existence  of  such  Good
Reason Condition.

1.12. “Good Reason Condition ” means that any of the following are undertaken without Executive’s express written

consent:

(a) 

 a material reduction in Executive’s Base Salary;

(b)

(c)

a material diminution in Executive’s responsibilities;

the Company’s material breach of any material term of this Agreement; or

(d)      a requirement that Executive relocate to an office that would increase Executive’s one-way commute distance

by more than fifty (50) miles based on Executive’s primary residence at the time such relocation is announced.

1.13. “Involuntary Termination Without Cause ” means Executive’s dismissal or discharge by the Company other
than for Cause. The termination of Executive’s employment as a result of Executive’s death or inability to perform the
essential functions of his job due to disability will not be deemed to be an Involuntary Termination Without Cause.

1.14. “Separation from Service” means Executive’s termination of employment or service where such termination
of employment or service constitutes a “separation from service” within the meaning of Treasury Regulation Section
1.409A-1(h).

ARTICLE II EMPLOYMENT BY THE COMPANY

2.1. Position  and  Duties.   Subject  to  terms  set  forth  herein,  as  of  the  Effective  Date,  Executive  shall  serve  as  the
Company’s Chief Executive Officer and perform such duties as are customarily associated with the position of Chief
Executive  Officer  and  such  other  duties  as  are  assigned  to  Executive  by  the  Board.  During  the  term  of  Executive’s
employment  with  the  Company,  Executive  will  devote  Executive’s  best  efforts  and  substantially  all  of  Executive’s
business  time  and  attention  (except  for  vacation  periods  and  reasonable  periods  of  illness  or  other  incapacities
permitted by the Company’s general employment policies, if any, or as otherwise set forth in this Agreement) to the
business of the Company.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
2.2.  Employment  at  Will.  Both  the  Company  and  Executive  shall  have  the  right  to  terminate  Executive’s
employment  with  the  Company  at  any  time,  with  or  without  Cause,  and  without  prior  notice.  If  Executive’s
employment  with  the  Company  is  terminated,  Executive  will  be  eligible  to  receive  severance  benefits  to  the  extent
provided in this Agreement.

2.3. Employment Policies. The employment relationship between the parties shall also be governed by the general
employment  policies  and  practices  of  the  Company,  if  any,  including  those  relating  to  protection  of  confidential
information and assignment of inventions, except that when the terms of this Agreement differ from or are in conflict
with the Company’s general employment policies or practices, this Agreement shall control.

ARTICLE III COMPENSATION

  3.1.  Base Salary.  As of the Effective Date, Executive shall receive for services to be rendered hereunder an annual
base salary of $375,000 (“Base Salary”), payable on the regular payroll dates of the Company, subject to increase in
the sole discretion of the Board.

  3.2    Retention Bonus. Executive shall be paid a one-time retention bonus of $3,813.97 (gross before taxes) payable
with Executive’s next regular paycheck.

3.3. Annual Bonus. Executive is subject to an annual bonus at the discretion of the Board, which bonus is initially

being targeted for up to 50% of the annualized amount of Base Salary.

3.4. Standard Company Benefits. Executive shall be entitled to all rights and benefits for which Executive is eligible
under the terms and conditions of the standard Company benefits and compensation practices, if any, that may be in
effect  from  time  to  time  and  are  provided  by  the  Company  to  its  executive  employees  generally.  Executive  shall  be
entitled each year to four (4) weeks leave for vacation at full pay, provided, that the maximum amount Executive may
have accrued at any point in time is four (4) weeks (meaning that once Executive has accrued four (4) weeks, Executive
will  not  accrue  any  additional  vacation  time  until  he  takes  vacation  and  falls  below  the  four  (4)  week  accrual  cap).
Executive  shall  also  be  entitled  to  reasonable  holidays  and  illness  days  with  full  pay  in  accordance  with  the  policies
applicable to the Company and its affiliates, if any, from time to time in effect. Employee acknowledges and agrees that
in  order  to  maintain  flexibility,  the  Company  and  its  affiliates  have  the  right  to  amend  or  terminate  any  employee
benefit  plan  at  any  time.  Until  such  time  as  the  Company  obtains  healthcare  benefits  for  eligible  employees  and
Executive elects to opt in to such benefits, Executive shall be entitled to an additional salary of at least $4,583.33 per
month or such greater amount as determined by the Board.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
3.5. Stock Options. Subject to approval by the Board, Executive may be granted options to purchase shares of the
Company’s common stock with an exercise price per share as determined by the Compensation Committee or similar
function of the Board.

3.6.  Expenses.  The  Company  will  reimburse  Executive  for  all  reasonable  and  necessary  expenses  incurred  by
Employee  in  connection  with  the  Company’s  business,  provided  that  such  expenses  incurred  and  are  properly
documented and accounted for in accordance with the policy of the Company and requirements of the Internal Revenue
Service.

ARTICLE IV
SEVERANCE AND CHANGE IN CONTROL BENEFITS

4.1.  Severance  Benefits.  Upon  Executive’s  termination  of  employment,  Executive  shall  receive  any  accrued  but
unpaid  Base  Salary  and  other  accrued  and  unpaid  compensation,  including  any Annual  Bonus  that  has  been  earned
with respect to a prior year, but remains unpaid as of the date of the termination. If the termination is due to a Covered
Termination or permanent disability, provided that Executive first returns all Company property in his possession and,
within sixty (60) days following the Covered Termination, executes and does not revoke an effective general release of
all  claims  against  the  Company  and  its  affiliates  in  a  form  reasonably  acceptable  to  the  Company  and  Executive  (a
“Release  of  Claims”),  Executive  shall  also  be  entitled  to  receive  the  following  severance  benefits  described  in  this
Section 4.1.

(a) Covered  Termination  Not  Related  to  a  Change  in  Control.   If  Executive’s  employment  terminates  due  to  a

Covered Termination which occurs outside of a Change in Control Period, Executive shall receive the following:

(i) An amount equal to twelve (12) months of Executive’s Base Salary payable in substantially equal installments in
accordance with the Company’s normal payroll policies, if any, less applicable withholdings, with such installments to
commence as soon as administratively practicable following the date the Release of Claims is not subject to revocation
and, in any event, within sixty (60) days following the date of the Covered Termination.

(ii) If Executive elects to receive continued healthcare coverage pursuant to the provisions of COBRA, the Company
shall directly pay, or reimburse Executive for, the premium for Executive and Executive’s covered dependents through
the earlier of (i) the first anniversary of the date of Executive’s termination of employment and (ii) the date Executive
and Executive’s covered dependents, if any, become eligible for healthcare coverage under another employer’s plan(s).
Notwithstanding the foregoing, (i) if any plan pursuant to which such benefits are provided is not, or ceases prior to the
expiration of the period of continuation coverage to be, exempt from the application of Section 409A of the

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Code under Treasury Regulation Section 1.409A-1(a)(5), or (ii) the Company is otherwise unable to continue to cover
Executive  under  its  group  health  plans  without  penalty  under  applicable  law  (including  without  limitation,  Section
2716 of the Public Health Service Act), then, in either case, an amount equal to each remaining Company subsidy shall
thereafter  be  paid  to  Executive  in  substantially  equal  monthly  installments.  After  the  Company  ceases  to  pay
premiums  pursuant  to  this  Section  4.1(a)(ii),  Executive  may,  if  eligible,  elect  to  continue  healthcare  coverage  at
Executive’s expense in accordance with the provisions of COBRA.

(iii) All of Employee’s vested options or stock appreciation rights with respect to the Company’s common stock shall
remain exercisable until the first anniversary of Executive’s termination of employment (or, if earlier, the maximum
period specified in the award documents and plans governing such options or stock appreciation rights, as applicable,
assuming Executive’s employment had not terminated).

(b)  Covered  Termination  Related  to  a  Change  in  Control.   If  Executive’s  employment  terminates  due  to  a

Covered Termination that occurs during a Change in Control Period, Executive shall receive the following:

(i) Executive shall be entitled to receive an amount equal to the Change in Control Multiplier multiplied by the sum
of: (i) Executive’s Base Salary and (ii) Executive’s target Annual Bonus for the fiscal year of Executive’s termination,
in  each  case,  at  the  rate  equal  to  the  higher  of  (x)  the  rate  in  effect  immediately  prior  to  Executive’s  termination  of
employment  or  (y)  the  rate  in  effect  immediately  prior  to  the  Change  in  Control  payable  in  a  cash  lump  sum,  less
applicable withholdings, as soon as administratively practicable following the date the Release of Claims is not subject
to revocation and, in any event, within sixty (60) days following the date of the Covered Termination.

(ii) If Executive elects to receive continued healthcare coverage pursuant to the provisions of COBRA, the Company
shall directly pay, or reimburse Executive for, the premium for Executive and Executive’s covered dependents through
the earlier of (i) the date that is that number of years equal to the Change in Control Multiplier following the date of
Executive’s  termination  of  employment  and  (ii)  the  date  Executive  and  Executive’s  covered  dependents,  if  any,
become  eligible  for  healthcare  coverage  under  another  employer’s  plan(s).  Notwithstanding  the  foregoing,  (i)  if  any
plan pursuant to which such benefits are provided is not, or ceases prior to the expiration of the period of continuation
coverage to be, exempt from the application of Section 409A of the Code under Treasury Regulation Section 1.409A-
1(a)(5), or (ii) the Company is otherwise unable to continue to cover Executive under its group health plans without
penalty  under  applicable  law  (including  without  limitation,  Section  2716  of  the  Public  Health  Service Act),  then,  in
either case, an amount equal to each remaining Company subsidy shall thereafter be paid to Executive in substantially
equal monthly installments. After the Company ceases to pay premiums pursuant to this Section 4.1(b)(ii), Executive
may, if eligible, elect to continue

 
 
 
 
 
 
 
 
 
 
 
 
healthcare coverage at Executive’s expense in accordance with the provisions of COBRA.

(iii) Each outstanding equity award, including, without limitation, each stock option and restricted stock award, held
by Executive shall automatically become vested and, if applicable, exercisable and any forfeiture restrictions or rights
of repurchase thereon shall immediately lapse, in each case, with respect to one hundred percent (100%) of the shares
subject  thereto.  To  the  extent  vested  after  giving  effect  to  the  acceleration  provided  in  the  preceding  sentence,  each
stock option held by Executive shall remain exercisable until the earlier of the original expiration date for such stock
option or the second anniversary of Executive’s Covered Termination.

(c)  Termination  for  Death  or  Disability .  If  Executive’s  employment  is  terminated  due  to  death  or  permanent
disability  where  the  Company  makes  a  determination  in  good  faith  that,  due  to  a  mental  or  physical  incapacity,
Executive has been unable to perform his duties under this Agreement for a period of not less than six (6) consecutive
months or 180 days in the aggregate in any 12-month period, Executive shall receive the following:

(i) An  amount  equal  to  three  (3)  months  of  Executive’s  Base  Salary  payable  in  substantially  equal  installments  in
accordance  with  the  Company’s  normal  payroll  policies,  less  applicable  withholdings,  with  such  installments  to
commence as soon as administratively practicable following the date the Release of Claims is not subject to revocation
and, in any event, within sixty (60) days following the date of the Covered Termination.

(ii) If Executive (or in the event of death, his designee) elects to receive continued healthcare coverage pursuant to
the provisions of COBRA, the Company shall directly pay, or reimburse Executive for, the premium for Executive and
Executive’s covered dependents through the earlier of (i) the three (3) month anniversary of the date of Executive’s
termination of employment and (ii) the date Executive and Executive’s covered dependents, if any, become eligible for
healthcare coverage under another employer’s plan(s). Notwithstanding the foregoing, (i) if any plan pursuant to which
such benefits are provided is not, or ceases prior to the expiration of the period of continuation coverage to be, exempt
from  the  application  of  Section  409A  of  the  Code  under  Treasury  Regulation  Section  1.409A-1(a)(5),  or  (ii)  the
Company  is  otherwise  unable  to  continue  to  cover  Executive  under  its  group  health  plans  without  penalty  under
applicable law (including without limitation, Section 2716 of the Public Health Service Act), then, in either case, an
amount equal to each remaining Company subsidy shall thereafter be paid to Executive in substantially equal monthly
installments. After the Company ceases to pay premiums pursuant to this Section 4.1(b)(ii), Executive may, if eligible,
elect to continue healthcare coverage at Executive’s expense in accordance the provisions of COBRA.

4.2. 280G Provisions. Notwithstanding anything in this Agreement to the contrary, if any payment or distribution

Executive would receive pursuant to this Agreement or

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
otherwise (“Payment”) would (a) constitute a “parachute payment” within the meaning of Section 280G of the Code,
and (b) but for this sentence, be subject to the excise tax imposed by Section 4999 of the Code (the “Excise  Tax”),
then such Payment shall either be (i) delivered in full, or (ii) delivered as to such lesser extent which would result in no
portion of such Payment being subject to the Excise Tax, whichever of the foregoing amounts, taking into account the
applicable federal, state and local income taxes and the Excise Tax, results in the receipt by Executive on an after-tax
basis, of the largest payment, notwithstanding that all or some portion the Payment may be taxable under Section 4999
of  the  Code.  The  accounting  firm  engaged  by  the  Company  for  general  audit  purposes  as  of  the  day  prior  to  the
effective date of the Change in Control shall perform the foregoing calculations. The Company shall bear all expenses
with respect to the determinations by such accounting firm required to be made hereunder. The accounting firm shall
provide  its  calculations  to  the  Company  and  Executive  within  fifteen  (15)  calendar  days  after  the  date  on  which
Executive’s right to a Payment is triggered (if requested at that time by the Company or Executive) or such other time
as  requested  by  the  Company  or  Executive. Any  good  faith  determinations  of  the  accounting  firm  made  hereunder
shall be final, binding and conclusive upon the Company and Executive. Any reduction in payments and/or benefits
pursuant  to  this  Section  4.2  will  occur  in  the  following  order:  (1)  reduction  of  cash  payments;  (2)  cancellation  of
accelerated vesting of equity awards other than stock options; (3) cancellation of accelerated vesting of stock options;
and (4) reduction of other benefits payable to Executive.

4.3.

Section 409A.

(a)  Notwithstanding  any  provision  to  the  contrary  in  this  Agreement,  if  Executive  is  deemed  at  the  time  of  his
Separation  from  Service  to  be  a  “specified  employee”  for  purposes  of  Section  409A(a)(2)(B)(i)  of  the  Code,  to  the
extent delayed commencement of any portion of the benefits to which Executive is entitled under this Agreement is
required in order to avoid a prohibited distribution under Section 409A(a)(2)(B)(i) of the Code which would subject
Executive  to  a  tax  obligation  under  Section  409A  of  the  Code,  such  portion  of  Executive’s  benefits  shall  not  be
provided to Executive prior to the earlier of (i) the expiration of the six- month period measured from the date of the
Executive’s Separation from Service or (ii) the date of Executive’s death. Upon the expiration of the applicable Code
Section 409A(a)(2)(B)(i) period, all payments deferred pursuant to this Section 4.3(a) shall be paid in a lump sum to
Executive, and any remaining payments due under the Agreement shall be paid as otherwise provided herein.

(b) Any reimbursements payable to Executive pursuant to the Agreement shall be paid to Executive no later than 30
days after Executive provides the Company with a written request for reimbursement, and to the extent that any such
reimbursements are deemed to constitute “nonqualified deferred compensation” within the meaning of Section 409A of
the Code (i) such amounts shall be paid or reimbursed to Executive promptly, but in no event later than December 31
of the year following the year in which the expense is incurred, (ii)

 
 
 
 
 
 
 
 
 
 
the amount of any such payments eligible for reimbursement in one year shall not affect the payments or expenses that
are eligible for payment or reimbursement in any other taxable year, and (iii) Executive’s right to such payments or
reimbursement shall not be subject to liquidation or exchange for any other benefit.

(c) For  purposes  of  Section  409A  of  the  Code  (including,  without  limitation,  for  purposes  of  Treasury  Regulation
Section 1.409A-2(b)(2)(iii)), Executive’s right to receive installment payments under the Agreement shall be treated as
a right to receive a series of separate payments and, accordingly, each installment payment hereunder shall at all times
be considered a separate and distinct payment.

4.4. Mitigation. Executive shall not be required to mitigate damages or the amount of any payment provided under
this Agreement by seeking other employment or otherwise, nor shall the amount of any payment provided for under
this Agreement be reduced by any compensation earned by Executive as a result of employment by another employer
or by any retirement benefits received by Executive after the date of the Covered Termination, or otherwise.

ARTICLE V
PROPRIETARY INFORMATION OBLIGATIONS

5.1. Agreement. Executive agrees to continue to abide by the Confidential Disclosure Agreement.

5.2.  Remedies.  Executive’s  duties  under  the  Confidential  Disclosure  Agreement  shall  survive  termination  of
Executive’s  employment  with  the  Company  and  the  termination  of  this Agreement.  Executive  acknowledges  that  a
remedy  at  law  for  any  breach  or  threatened  breach  by  Executive  of  the  provisions  of  the  Confidential  Disclosure
Agreement, as well as Executive’s obligations pursuant to Section 6.2 and Article 7 below, would be inadequate, and
Executive therefore agrees that the Company shall be entitled to seek injunctive relief in case of any such breach or
threatened breach.

ARTICLE VI OUTSIDE ACTIVITIES

6.1.

Other Activities.

(a) Executive shall not, during the term of this Agreement undertake or engage in any other employment, occupation
or  business  enterprise,  other  than  ones  in  which  Executive  is  a  passive  investor,  unless  he  obtains  the  prior  written
consent of the Board.

(b) Executive may engage in civic and not-for-profit activities so long as such activities do not materially interfere

with the performance of Executive’s duties

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
hereunder. In addition, Executive shall be allowed to serve as a member of the board of directors of up to two (2) other
for profit entities at any time during the term of this Agreement, which service shall not materially interfere with the
performance  of  Executive’s  duties  hereunder;  provided,  however,  that  the  Board  may  require  that  Executive  resign
from one or both of such director positions if it can reasonably and in good faith demonstrate that such resignation(s)
would be in the best interests of the Company in a significant and material way.

6.2.

Competition. Executive agrees that, from the date hereof until a period of twelve  (12) months following the
date of termination of Executive’s employment with the Company, Executive will not directly or indirectly,
either  as  an  employee,  employer,  consultant,  agent,  principal,  partner,  corporate  officer,  director,  or  in  any
other individual or representative capacity, engage or participate in any “Competitive Business” anywhere in
the  United  States  of  America.  As  used  herein,  a  “Competitive  Business”  is  defined  as  any  business
developing uPAR antibodies to treat cancer, or clonidine to treat oral mucositis.

ARTICLE VII NONINTERFERENCE

In addition to Executive’s obligations under the Confidential Disclosure Agreement, Executive shall not for a period
of one (1) year following Executive’s termination of employment for any reason, either on Executive’s own account
or jointly with or as a manager, agent, officer, employee, consultant, partner, joint venturer, owner or stockholder or
otherwise on behalf of any other person, firm or corporation, directly or indirectly solicit or attempt to solicit away
from the Company any of its officers or employees or offer employment to any person who is an officer or employee
of  the  Company; provided, however,  that  a  general  advertisement  to  which  an  employee  of  the  Company  responds
shall in no event be deemed to result in a breach of this Article 7. Executive also agrees not to harass or disparage the
Company or its employees, clients, directors or agents or divert or attempt to divert any actual or potential business of
the Company. The provisions of this Article 7 shall survive the termination or expiration of the applicable Executive’s
employment with the Company and shall be fully enforceable thereafter. If it is determined by a court of competent
jurisdiction  in  any  state  that  any  restriction  in  this Article  7  is  excessive  in  duration  or  scope  or  is  unreasonable  or
unenforceable under the laws of that state, it is the intention of the parties that such restriction may be modified or
amended by the court to render it enforceable to the maximum extent permitted by the law of that state.

ARTICLE VIII GENERAL PROVISIONS

8.1. Notices. Any notices provided hereunder must be in writing and shall be deemed effective upon the earlier of
personal delivery (including personal delivery by facsimile) or the third day after mailing by first class mail, to the
Company at its primary office location and to Executive at Executive’s address as listed on the Company payroll.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
8.2. Tax Withholding. Executive acknowledges that all amounts and benefits payable under this Agreement are

subject to deduction and withholding to the extent required by applicable law.

8.3. Severability. Whenever possible, each provision of this Agreement will be interpreted in such manner as to be
effective  and  valid  under  applicable  law,  but  if  any  provision  of  this  Agreement  is  held  to  be  invalid,  illegal  or
unenforceable  in  any  respect  under  any  applicable  law  or  rule  in  any  jurisdiction,  such  invalidity,  illegality  or
unenforceability  will  not  affect  any  other  provision  or  any  other  jurisdiction,  but  this Agreement  will  be  reformed,
construed  and  enforced  in  such  jurisdiction  as  if  such  invalid,  illegal  or  unenforceable  provisions  had  never  been
contained herein.

8.4. Waiver. If either party should waive any breach of any provisions of this Agreement, they shall not thereby be

deemed to have waived any preceding or succeeding breach of the same or any other provision of this Agreement.

8.5. Complete Agreement.  This Agreement constitutes the entire agreement between Executive  and  the  Company
and  is  the  complete,  final,  and  exclusive  embodiment  of  their  agreement  with  regard  to  this  subject  matter,  and  will
supersede  all  prior  agreements,  understandings,  discussions,  negotiations  and  undertakings,  whether  written  or  oral,
between the parties with respect to the subject matter hereof, including without limitation, the Prior Agreement. This
Agreement  is  entered  into  without  reliance  on  any  promise  or  representation  other  than  those  expressly  contained
herein  or  therein,  and  cannot  be  modified  or  amended  except  in  a  writing  signed  by  an  officer  of  the  Company  and
Executive.

8.6. Counterparts.  This Agreement  may  be  executed  in  separate  counterparts,  any  one  of  which  need  not  contain

signatures of more than one party, but all of which taken together will constitute one and the same Agreement.

8.7. Headings. The headings of the sections hereof are inserted for convenience only and shall not be deemed to

constitute a part hereof nor to affect the meaning thereof.

8.8. Successors and Assigns.  This Agreement is intended to bind and inure to the benefit of and be enforceable by
Executive and the Company, and their respective successors, assigns, heirs, executors and administrators, except that
Executive may not assign his rights or delegate his duties or obligations hereunder without the prior written consent of
the Company.

8.9. Arbitration. Unless otherwise prohibited by law or specified below, all disputes, claims and causes of action, in
law  or  equity,  arising  from  or  relating  to  this Agreement  or  its  enforcement,  performance,  breach,  or  interpretation
shall be resolved solely and

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
exclusively by final and binding arbitration held in Illinois in co onnity with the then existing employment arbitration
rules  and  Illinois  law.  The  arbitrator  shall:  (a)  provide  adequate  discovery  for  the  resolution  of  the  dispute;  and  (b)
issue a written arbitration decision,  to include the arbitrator's essential findings and conclusion and a statement of the
award. However, nothing in  this section is intended to prevent either party from obtaining injunctive relief in court to
prevent irreparable harm pending the inclusion of any such arbitration. The Company shall bear the costs of any such
arbitration. I

8.10.  Eiecutive  Acknowledgement.   Executive  acknowledges  that  (a)  he  has  consulted  with  or   has  had  the
opportunity to consult with independent counsel of his own choice concerning this Agreement, and has been advised to
do so by the Company, and (b) that he has read and understands the Agreement, is fully aware of its legal effect, and
has entered into it freely based on his own judgment.

8.11. Choice of Law. All questions concerning the construction, validity and interpretation of this Agreement will be

governed by the law of the State of Illinois without regard to the conflicts of law provisions thereof.

In Witness Whereof, the parties have executed this Agreement as  of the date first written above.

On behalf of Monopar Therapeutics Inc.

/s/ Christopher M. Starr
Christopher M. Starr
Executive Chairman

Accepted and Agreed:

/s/ Chandler D. Robinson
Chandler D. Robinson

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
  
 
 
 
 
 
 
  
 
CONSULTING AGREEMENT

This Consulting Agreement (herein referred to as "Agreement") is  made  and  entered  into  as  of  this  December  15,  2016  (the
"Effective  Date"),  by  and  between  Monopar  Therapeutics  Inc.  (herein  referred  to  as  "Monopar"),  a  Delaware  limited  liability
corporation, located at corporation, located at 5 Revere Dr., Suite 200, Northbrook, IL 60062, and Kim.R. Tsuchimoto (herein referred to
as "TSUCHIMOTO") who resides at # (each herein referred to as "Party" and collectively as "Parties").

RECITALS

WHEREAS,  TSUCHIMOTO  specializes  in  the  field  of  finance  and  strategy,  including  but  not  limited  to:  pre-IPO  readiness,

internal and external financial reporting, SEC and Nasdaq compliance, internal controls , forecasting/budgeting; and

WHEREAS,  Monopar  desires  to  contract  with  TSUCHIMOTO  to  provide  certain  consultation  services,  as  requested  by

Monopar, and TSUCHIMOTO wishes to provide such services to Monopar, upon the terms and conditions set forth below.

NOW, TIIEREFORE, in consideration of the premises and mutual covenants contained herein, the Parties agree as follows :

1. 

2. 

Consulting  Arrangement.  TSUCHIMOTO  agrees  to  perform  consulting  services  as  described  herein  upon  the  terms  and
conditions herein set forth.

Term of Agreement. Subject to the provision for early termination set forth below in Section 5 of this Agreement, this Agreement
shall  commence  as  of  the  Effective  Date  and  shall  continue  for  a  period  of  twelve  (12)  months  from  the  Effective  Date  (the
"Term"). Either Party may terminate this Agreement without cause with 10-days' prior written notice.

3. 

Duties of TSUCHIMOTO.

3.1 

3.2 

Specific  Duties.  TSUCHIMOTO  shall  provide  consulting  services  to  Monopar,  such  duties  to  include,  managing
finances and accounting, investor and public relations, financial reporting, preparation and management of public trading
or  listing,  SEC  or  other  regulatory  body  financial  reporting  and  compliance,  with  such  other  specific  requirements  as
Monopar may specify from time to time during the Term (herein referred to as the "Services").

TSUCHIMOTO's Obligations. TSUCHIMOTO shall be diligent in the performance of Services , and be professional in
her commitment to meeting her obligations hereunder. TSUCHIMOTO represents and warrants that TSUCHIMOTO is
not party to any other existing agreement, which any of them would prevent her from entering into this Agreement or
which would adversely affect this Agreement. TSUCHIMOTO shall not perform Services for any other individuals or
entities  in  direct  competition  with  Monopar,  except  as  provided  for  by  mutual  written  agreement  of  the  Parties.
TSUCHIMOTO shall not perform

- 1 -

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
                                                                                         
 
services for any party which would require or facilitate the unauthorized disclosure of any confidential or proprietary
information of Monopar.

3.3 

3.4 

Reporting.  TSUCHIMOTO  will  report  to  and  liaise  with  Chandler  Robinson,  M.D.,  and  Christopher  M.  Starr,  Ph.D.
and/or any other assigned Monopar employee or consultant as may be designated in writing by Monopar.

Compensation. Monopar shall pay TSUCHIMOTO a cash retainer of $5,000 per month not to exceed $60,000 for the
period of this Agreement, unless modified in writing by mutual agreement amongst the Parties.

TSUCHIMOTO shall not be reimbursed, and is responsible for the facilities and equipment necessary to perform
Services required under this Agreement.

Reimbursement of Other Expenses. So long as Monopar's prior approval has been obtained, Monopar shall promptly reimburse
TSUCHIMOTO  for  all  direct  expenses  incurred  in  providing  the  Services  to  Monopar  pursuant  to  this Agreement,  including
travel, meals and lodging. The invoice submitted by TSUCHIMOTO pursuant to this Section 4 shall also include a detail of all
reimbursable expenses incurred during the period covered by such invoice.

Termination of Agreement - Failure to perform . In the event that TSUCHIMOTO ceases to perform the Services or breaches its
obligations  as  required  hereunder  for  any  reason,  Monopar  shall  have  the  right  to  immediately  terminate  this Agreement  upon
notice to TSUCHIMOTO and to enforce such other rights and remedies as it may have as a result of said breach.

Certain Liabilities. It is understood and agreed that TSUCHIMOTO shall be acting as an independent contractor and not as an
agent  or  employee  of,  or  partner,  joint  venturer  or  in  any  other  relationship  with  Monopar.  TSUCHIMOTO  will  be  solely
responsible for all her insurance, employment taxes, FICA taxes and all obligations to governments or other organizations arising
out of this consulting assignment. TSUCHIMOTO acknowledges that no income, social security or other taxes shall be withheld
or  accrued  by  Monopar  for  TSUCHIMOTO's  benefit.  TSUCHIMOTO  assumes  all  risks  and  hazards  encountered  in  the
performance of duties under this Agreement. Unless Monopar has provided prior written approval, TSUCHIMOTO shall not use
any sub-contractors to perform TSUCHIMOTO's obligations hereunder. TSUCHIMOTO shall be solely responsible for any and
all injuries, including death, to all persons and any and all loss or damage to property, which may result from performance under
this Agreement.

Indemnities.  TSUCHIMOTO  hereby  agrees  to  indemnify  Monopar  and  hold  Monopar  harmless  from  and  against  all  claims
(whether asserted by a person, firm, entity or governmental unit or otherwise), liabilities, losses, damages, expenses, charges and
fees which Monopar may sustain or incur arising out of or attributable to any breach, gross negligence or willful misconduct by
TSUCHIMOTO, as applicable, in the performance under this Agreement. Monopar hereby agrees to indemnify TSUCHIMOTO
and  hold  TSUCHIMOTO  harmless  from  and  against  all  liabilities,  losses,  damages,  expenses,  charges  and  fees  which
TSUCHIMOTO may sustain or incur by reason of any claim which

4.

5. 

6. 

7. 

- 2 -

 
 
 
 
 
 
 
 
 
 
 
 
 
                                                                                             
 
may be asserted against TSUCHIMOTO by any person, firm, corporation or governmental unit and which may arise out of or be
attributable to any  gross  negligence  or  willful  misconduct  by  Monopar  or  its  employees  or  contractors,  as  applicable,  in  the
performance of this Agreement.

8. 

9. 

10. 

11. 

Warranties.  The  Services  shall  be  performed  in  a  professional  manner,  consistent  with  industry  standards.  In  performing  the
Services, TSUCHIMOTO shall not make any unauthorized use of any confidential or proprietary information of any other party
or infringe the intellectual property rights of any other party. ·

Arbitration. Any controversy or claim between Monopar and TSUCHIMOTO arising out of or relating to this Agreement, or the
breach thereof, shall be submitted to arbitration in accordance with the rules of the American Arbitration Association. The site of
the arbitration shall be Chicago, Illinois, and except as provided herein the arbitration shall be conducted in accordance with the
Rules of the American Arbitration Association prevailing at the time the demand for arbitration is made hereunder. At least one
member of the arbitration panel shall be a financial expert knowledgeable in the area of biopharmaceutical corporate compliance.
Judgment upon any award rendered by the arbitrator(s) may be entered in any court of competent jurisdiction and shall be binding
and final. The cost of arbitration shall be borne by the losing Party, as determined by the arbitrator(s).

Confidential  Information.  TSUCHIMOTO  has  executed  the  attached  confidential  disclosure  agreement  referenced  herein  as
Appendix A   prior  to  commencement  of  the  Services.  TSUCHIMOTO  hereby  represents  and  warrants  that  the  obligations
thereunder shall be binding.

Inventions.  TSUCHIMOTO  agrees  that  all  ideas,  developments,  suggestions  and  inventions  conceived  or  reduced  to  practice
arising out of or during the course of performance under this Agreement shall be the exclusive property of Monopar and shall be
promptly communicated and assigned to Monopar. TSUCHIMOTO shall require any employees of or other parties contracted by
TSUCHIMOTO to disclose the same to TSUCHIMOTO and to be bound by the provisions of this paragraph. During the period
of this Agreement and thereafter at any reasonable time when called upon to do so by Monopar, TSUCHIMOTO shall require any
employees  of  or  other  parties  contracted  by  TSUCHIMOTO  to  execute  patent  applications,  assignments  to  Monopar  (or  any
designee  of  Monopar  )  and  other  papers  and  to  perform  acts  which  Monopar  believes  necessary  to  secure  to  Monopar  full
protection and ownership of the rights in and to the services performed by TSUCHIMOTO and/or for the preparation, filing and
prosecution of applications for patents or inventions made by any employees of or  other  parties  contracted  by  TSUCHIMOTO
hereunder.  The  decision  to  file  patent  applications  on  inventions  made  by  any  employees  of  or  other  parties  contracted  by
TSUCHIMOTO shall be made by Monopar and shall be for such countries, as Monopar shall elect. Monopar agrees to bear all
the expense in connection with the preparation, filing and prosecution of applications for patents and for all matters provided in
this paragraph requiring the time and/or assistance of TSUCHIMOTO as to such inventions.

12. 

Miscellaneous.

- 3 -

 
 
 
 
 
 
 
 
 
 
 
 
 
                                                  
 
12.l Notice. Any notices to be given hereunder by either Party to the other may be effectuated, in writing, by personal delivery or
by mail, registered or certified, postage prepaid, with return receipt requested. Mailed notices shall be addressed to the
parties at the following addresses:

If to Monopar:                                            Monopar Therapeutics Inc.

                                                                                         5 Revere Dr., Suite 200
                                                                                         Northbrook, IL, 60062

        Attention: Chandler Robinson, MD MBA MSc

            Email: #

If to TSUCHIMOTO:                                Kim R. Tsuchimoto

#

  Email: #

or  at  such  other  addresses  as  either  Monopar  or  TSUCHIMOTO  may  designate  by  written  notice  to  each  other.  Notices
delivered personally shall be deemed duly given on the date of actual receipt; mailed notices shall be deemed duly given as of
the fourth day after the date so mailed.

12.2  Waiver  of  Breach.  The  waiver  by  either  Party  to  a  breach  of  any  provision  in  this Agreement  cannot  operate  or  be

construed as a waiver of any subsequent breach by either Party. ·

12.3 

12.4 

12.5 

Severability. If  any  provision  of  this Agreement  is  determined  by  a  court  of  competent  jurisdiction  to  be  invalid  or
unenforceable, that provision shall be deemed modified to the extent necessary to make it valid or enforceable, or if it
cannot be so modified, then severed, and the remainder of the Agreement shall continue in full force and effect as if the
Agreement had been signed with the invalid portion so modified or severed.

Choice  of  Law.  This Agreement  has  been  made  and  entered  into  in  the  State  of  Illinois,  and  the  laws  of  such  state,
excluding its choice of law rules, shall govern the validity and interpretation of this Agreement and the performance due
hereunder. The losing party in any dispute hereunder shall pay the attorneys' fees and  disbursements  of  the  prevailing
party.

Integration.  The  drafting,  execution  and  delivery  of  this  Agreement  by  the  Parties  have  been  induced  by  no
representations, statements, warranties or agreements other than those expressed herein. This Agreement embodies the
entire  understanding  of  the  Parties,  and  there  are  no  further  or  other  agreements  or  understandings,  written  or  oral,  in
effect between the Parties relating to the subject matter hereof unless expressly referred to herein.

- 4 -

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
                                                                                                     
 
12.6  Modification. This Agreement may not be modified unless such is in writing and signed by both Parties

to this Agreement.

12.7  Assignment.  TSUCHIMOTO  shall  not  be  permitted  to  assign  this Agreement  to  any  other  person  or
entity without the prior written consent of Monopar. TSUCHIMOTO hereby agrees that Monopar shall
be permitted to assign this Agreement to any affiliate of Monopar. This Agreement shall be binding upon
and shall inure to the benefit of the successors and permitted assigns of the parties.

12.8  Survival. The provisions of Sections 7, 8, 9, 10, and 11 shall  survive  expiration  or  termination  of  this
Agreement  for  any  reason.  Expiration  or  termination  of  this  Agreement  shall  not  affect  Monopar's
obligations to pay any amounts that may then be due to TSUCHIMOTO.

IN WITNESS WHEREOF, the Parties hereto have executed this Agreement as of the day and year first above

written.

ACCEPTED AND AGREED TO:

Kim R. Tsuchimoto

/s/ Kim R. Tsuchimoto

   Kim R. Tsuchimoto

MONOPAR THERAPEUTICS INC.

/s/ Chandler Robinson
BY: CHANDLER ROBINSON
ITS: CHIEF EXECUTIVE OFFICER

-5-

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
APPENDIX A

See executed CDA attached

 -6-

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
                    
 
MONOPARTHERAPEUTICS LLC
CONFIDENTIAL DISCLOSURE AGREEMENT

AGREEMENT between Kim Tsuchimoto ('' Recipient”) ) and Monopar Therapeutics LLC (“Monopar").

For purposes of this Agreement, the term "Recipient'' shall include, individually and/or collectively the partners, directors. officers,
employees, agents, and/or representatives of Kim Tsuchimoto.

In consideration for the mutual agreements contained herein and the other provisions of this Agreement, the receipt of which is

hereby acknowledged by the parties. the parties hereto agree as follows:

I. Scope of Confidential Information

·'Confidential Information" means, subject to the other provisions of this Section:

(a) all information, whether oral or written, disclosed by Monopar that is described in Schedule A under "Description of Confidential
Information” Confidential Information may relate to the activities or property of Monopar or any of Monopar's members. directors,
officers, employees, consultants, agents, representatives or affiliated entities (collectively, ·'Associated Persons"); and

( ) any written material prepared by Recipient or Recipient's partners,

directors, officers, employees, agents, representatives or affiliated entities (collectively, ''Associated Persons") containing any other
Monopar Confidential Information.

·'Confidential Information'' does not include information that: (i) was available to Recipient (free of any confidentiality obligation in
favor of Monopar) prior to disclosure of such information by Monopar to Recipient; (ii) is made available to Recipient from a third party
which (at the time of such availability) was not, to Recipient's knowledge, subject to a confidentiality obligation with respect to such
information; (iii) is made available to third parties by Monopar without restriction on the disclosure of such information, (iv) is or
becomes available to the public on or after the date of this Agreement (other than as a result of disclosure prohibited by any
confidentiality obligation contained herein): or (v) is developed independently by Recipient or its Associated Persons without
intended disclosure or (ii) if prior notice is not permitted or practicable under the circumstances, prompt notice of such disclosure.

3.Certain Right s and Limitations

(a)            All Confidential Information shall remain the property of Monopar. The provision of Confidential Information hereunder

shall not transfer any right, title or interest in such information to Recipient. Monopar does not gram any express or implied right to
Recipient to or under Monopar's patents, copyrights, trademarks. trade secret information or other proprietary rights.

(b)            Recipient agrees to adhere to all applicable laws and regulations relating to the export of technical data received hereunder.

(c)            This Agreement imposes no obligations on either party to purchase, sell, license, transfer or otherwise transact in any
technology, services or products. This Agreement does not create any agency or partnership relationship between the parties hereto.

4. Remedies

(a)            Upon Monopar's reasonable request, Recipient agrees to return promptly to Monopar all Confidential Information that is in

writing and in the possession of Recipient and, upon written request, to certify the return or destruction (at Monopar's option) of all
Confidential Information.

(b)            Recipient agrees that monetary damages may not be an adequate remedy for improper disclosure or use of Confidential
Information, that Monopar, upon breach of this contract, shall be entitled to such injunctive or equitable relief as may be deemed proper
by a court of competent jurisdiction, without waiving any other right or remedy, and that Recipient shall not resist an application for such
relief on the ground that Monopar has an adequate remedy at law.

5. Miscellane o us

(a) Except where expressly indicated otherwise, the words  "written" or
reference to the Confidential Information.

Recipient agrees that it will not disclose to Monopar or to any of its employees or consultants any confidential. proprietary, patented.

copyrighted, or trade secret information, or any other form of protectable intellectual property, regardless of whether such information is
the property of Recipient itself or of some other individual or organization.

2. Use and Disclosure of Confidential Information

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
(a)          Recipient agrees: (i) to preserve the confidentiality of Confidential Information; (ii) to use and/or permit the use of

Confidential information onyr for the purpose of, and to the extent necessary for, evaluating a business relat1onsh1p between the parties
and, if such a relationship is consummated, carrying out such relationship: (iii) to disclose Confidential Information to, and to permit the
use of Confidential Information by, only such persons within Recipient who Recipient reasonably determines need to know such
information in connection with the activities described in (ii) above; and (iv) to use reasonable care to maintain the confidentiality of
Confidential (information, provided that such care hall be at least as great as the precautions taken by Recipient to protect its own
confidential and/or proprietary information.

(b)            Notwithstanding anything to the contrary herein, Recipient is free to make (and this Agreement does not restrict) disclosure

of any Confidential Information in a judicial, legislative, or administrative investigation .or proceeding or to a government or other
regulatory agency; provided that, to the extent permitted by, and practicable under, the circumstances, Recipient provides to Monopar (i)
prior notice of the

  "in writing" shall include, but not be limited to, written or printed

documents, electronic and facsimile transmissions and computer disks or tapes (whether machine or user readable).

(b) In the event that any one or more of the provisions of this Agreement will for any reason be held to be invalid, illegal or

unenforceable by a court of competent jurisdiction, the remaining provisions of this

Agreement will be unimpaired, and the invalid, illegal or unenforceable pr?v1s1on will be replaced by a mutually acceptable provision,
which being valid, legal or enforceable, comes closest to the intention of the parties underlying the invalid, illegal or unenforceable
provision.

(c) No amendment or alteration of the terms of this Agreement shall be
effective unless made in writing and executed by both parties hereto.

(d)            A failure or delay in exercising any right in respect of this Agreement will not be presumed to operate as a waiver, and a
single or partial exercise of any right will! not be presumed to preclude any subsequent or further exercise of that right or the exercise of
any other right. Any

modification or waive of any provision of this Agreement shall not be effective unless made in writing. Any such waiver shall be
effective only in the specific instance and for the purpose given.

This Agreement and its enforcement shall be governed by and construed in accordance with, the laws of the State of Illinois
without regard to conflicts-of-law principles.

(SIGNATURE PAGE FOLLOWS]

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
IN WITNESS WHEREOF. the parties hereto have executed this Agreement.

·'RECIPIENT'"                                                                                                                                                                                                      '
MONOPAR"

/s/ Kim R. Tsuchimoto
By Kim R. Tsuchimoto
Title: Individual

Date: April 21, 2015

Notices hereunder shall be sent to: #

Monopar Therapeutics LLC

By: /s/ Chandler D. Robinson
Name: Chandler D. Robinson
Date: April 21, 2015

Notices hereunder shall be sent to: #

SCHEDULE A

Description of Confidential Information Disclosed by Monopar:

(a) The identity of the projects and compounds that Monopar is researching; (b) the methods of research and research collaborators being
used to pursue these projects and compounds; (c) the (known or putative) mechanism of action of any of these compounds; (d) any
techniques used by Monopar to discover, develop, produce, purify, or test any of these compounds; and (e) any non-public scientific,
business, or financial information pertaining to Monopar, its projects, or compounds, including all documents and agreements already
signed or currently being negotiated with Cancer Research UK and Cancer Research Technology).

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
EXECUTIVE EMPLOYMENT AGREEMENT

This Executive Employment Agreement (the “ Agreement”) is entered into as of November 1, 2017, by and between
Kim R. Tsuchimoto (“Executive”) and Monopar Therapeutics Inc. (the “ Company”).

Whereas, the Company desires to employ Executive as its Chief Financial Officer effective as of November 1, 2017
(the “Effective Date”), and Executive desires to serve in such capacity, pursuant to the terms and conditions set forth in
this Agreement; and

Now, Therefore, in consideration of the mutual promises and covenants contained herein, it is hereby agreed by and
between the parties hereto as follows:

ARTICLE I
DEFINITIONS

For purposes of the Agreement, the following terms are defined as follows:

1.1.              “Board” means the Board of Directors of the Company.

1.2.              “Cause” means any of the following events described below:

(a)  Executive’s commission of a felony or other crime involving moral turpitude;

(b)  any willful act or acts of dishonesty undertaken by Executive and intended to result in substantial gain or personal
enrichment of Executive, Executive’s family or any third party at the expense of the Company;

(c)  any willful act of gross misconduct which is materially and demonstrably injurious to the Company; and/or

(d)  Executive’s inability to lawfully work in the United States.

For  the  purpose  of  this Agreement,  no  act,  or  failure  to  act,  by  Executive  shall  be  considered  “willful”  if  done,  or
omitted to be done, by Executive in good faith and in the reasonable belief that Executive’s act or omission was in the
best interest of the Company and/or required by applicable law.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
1.3.               “Change in Control ” means the occurrence of any of the following events: (i) any sale or exchange of the
capital stock by the stockholders of the Company in one transaction or series of related transactions where more than
fifty  percent  (50%)  of  the  outstanding  voting  power  of  the  Company  is  acquired  by  a  person  or  entity  or  group  of
related persons or entities; or (ii) any reorganization, consolidation or merger of the Company where the outstanding
voting  securities  of  the  Company  immediately  before  the  transaction  represent  or  are  converted  into  less  than  fifty
percent (50%) of the outstanding voting power of the surviving entity (or its parent corporation) immediately after the
transaction; or (iii) the consummation of any transaction or series of related transactions that results in the sale of all or
substantially all of the assets of the Company; or (iv) any “person” or “group” (as defined in the Securities Exchange
Act of 1934, as amended (the “Exchange Act”) becoming the “beneficial owner” (as defined in Rule 13d-3 under the
Exchange Act) directly or indirectly of securities representing more than fifty percent (50%) of the voting power of the
Company then outstanding. Except that any change in the beneficial ownership of the securities of the Company as a
result  of  a  private  financing  of  the  Company  that  is  approved  by  the  Board,  shall  not  be  deemed  to  be  a  Change  in
Control.

1.4.              “Change in Control Multiple ” shall mean one-quarter (0.25).

1.5.               “Change in Control Period ” means that period commencing on the consummation of a Change in Control
and ending on the first anniversary thereof.

1.6.              “COBRA” means the Consolidated Omnibus Budget Reconciliation Act of 1985, as amended.

1.7.              “Code” means the Internal Revenue Code of 1986, as amended.

1.8.              “Company” means Monopar Therapeutics Inc. or any successor thereto.

1.9.               “Confidential Disclosure Agreement” means the Confidential Disclosure Agreement entered into between
Executive and the Company.

1.10.         
termination for Good Reason, provided that the termination constitutes a Separation from Service.

  “Covered  Termination ”  means  (a)  an  Involuntary  Termination  Without  Cause  or  (b)  a  voluntary

1.11.            “Good Reason” means Executive’s resignation as a result of a Good Reason Condition.  In order to resign
for  Good  Reason,  Executive  must  provide  written  notice  to  the  Company  of  the  existence  of  the  Good  Reason
Condition within thirty (30) days of the initial existence of such Good Reason Condition.  Upon receipt of such notice
of the Good Reason Condition, the Company will be provided with a period of thirty (30) days during which it may
remedy the Good Reason Condition and not be required to provide for the payments and benefits described in Section 4
as a result of such proposed resignation due to the Good Reason Condition specified in the notice.  If the Good Reason
Condition  is  not  remedied  within  the  period  specified  in  the  preceding  sentence,  Executive  may  resign  for  Good
Reason based on the Good Reason Condition specified in the notice, provided that such resignation must occur within
sixty (60) days after the initial existence of such Good Reason Condition.

 
 
 
 
 
 
 
 
 
 
 
1.12.            “Good Reason Condition ” means that any of the following are undertaken without Executive’s express
written consent:

(a)                  a material reduction in Executive’s Base Salary (other than as part of a reduction in the base salary of at
least a majority of the Company’s executives of the same or greater percentage);

(b)                 the Company’s material breach of any material term of this Agreement (a change in job title or role does not
constitute a material breach); or

a  requirement  that  Executive  relocate  to  an  office  that  would  increase  Executive’s  one-way  commute
(c)                
distance by more than fifty (50) miles based on Executive’s primary residence at the time such relocation is announced.

1.13.            “Involuntary Termination Without Cause ” means Executive’s dismissal or discharge by the Company
other  than  for  Cause.    The  termination  of  Executive’s  employment  as  a  result  of  Executive’s  death  or  inability  to
perform  the  essential  functions  of  his  job  due  to  disability  will  not  be  deemed  to  be  an  Involuntary  Termination
Without Cause.

1.14.           
“separation from service” within the meaning of Treasury Regulation Section 1.409A-1(h).

“Separation  from  Service”  means  Executive’s  termination  of  employment  or  service  constitutes  a

ARTICLE II
EMPLOYMENT BY THE COMPANY

2.1.              Position and Duties.  Subject to terms set forth herein, as of the Effective Date, Executive shall serve as the
Company’s  Chief  Financial  Officer  and  perform  such  duties  as  are  customarily  associated  with  the  position  of  Chief
Financial Officer and such other duties as are assigned to Executive by the Chief Executive Officer.  During the term of
Executive’s  employment  with  the  Company,  Executive  will  devote  Executive’s  best  efforts  and  25%  of  Executive’s
business time and attention (except for vacation periods and reasonable periods of illness or other incapacities permitted
by  the  Company’s  general  employment  policies  or  as  otherwise  set  forth  in  this Agreement)  to  the  business  of  the
Company.

2.2.               Employment  at  Will.   Both the Company and Executive shall have the right to terminate Executive’s
employment  with  the  Company  at  any  time,  with  or  without  Cause,  and  without  prior  notice.    If  Executive’s
employment  with  the  Company  is  terminated,  Executive  will  be  eligible  to  receive  severance  benefits  to  the  extent
provided in this Agreement.

 
 
 
  
 
 
 
 
 
 
 
2.3.               Employment  Policies.  The employment relationship between the parties shall also be governed by the
general  employment  policies  and  practices  of  the  Company,  including  those  relating  to  protection  of  confidential
information and assignment of inventions, except that when the terms of this Agreement differ from or are in conflict
with the Company’s general employment policies or practices, this Agreement shall control.

ARTICLE III
COMPENSATION

3.1.               Base Salary.   As of the Effective Date,  Executive shall receive for services to be rendered hereunder an
annual base salary of $68,750 (“Base Salary”), payable on the regular payroll dates of the Company, subject to increase
in the sole discretion of the Board. Base salary represents a part-time salary (25% of full-time) as noted in section 2.1
above.

3.2.              Annual Bonus.  Executive is subject to an annual bonus at the discretion of the Board.

3.3.              Standard Company Benefits.  Upon reaching full-time status (over 30 hours per week of employment with
the Company) Executive shall be entitled to all rights and benefits for which Executive is eligible under the terms and
conditions of the standard Company benefits and compensation practices that may be in effect from time to time and
are provided by the Company to its executive employees generally. Based on 25% service, Executive shall be entitled
each  year  to  one  (1)  week  leave  for  vacation  at  full  pay,  provided,  that  the  maximum  amount  Executive  may  have
accrued at any point in time is one (1) week (meaning that once Executive has accrued one (1) week, Executive will not
accrue  any  additional  vacation  time  until  Executive  takes  vacation  and  falls  below  the  one  (1)  week  accrual  cap).
Executive  shall  also  be  entitled  to  reasonable  holidays  and  illness  days  with  full  pay  in  accordance  with  the  policies
applicable  to  the  Company  and  its  affiliates  from  time  to  time  in  effect.  Employee  acknowledges  and  agrees  that  in
order to maintain flexibility, the Company and its affiliates have the right to amend or terminate any employee benefit
plan at any time.

3.4.               Stock Options. Subject to approval by the Board, Executive may be granted options to purchase shares of
the  Company’s  common  stock  with  an  exercise  price  per  share  as  determined  by  the  Compensation  Committee  or
similar function of the Board.

3.5.               Expenses. The Company will reimburse Executive for all reasonable and necessary expenses incurred by
Employee  in  connection  with  the  Company’s  business,  provided  that  such  expenses  incurred  and  are  properly
documented and accounted for in accordance with the policy of the Company and requirements of the Internal Revenue
Service.

 
 
 
 
 
 
 
 
 
 
ARTICLE IV
SEVERANCE AND CHANGE IN CONTROL BENEFITS

4.1.               Severance Benefits.  Upon Executive’s termination of employment, Executive shall receive any accrued
but unpaid Base Salary and other accrued and unpaid compensation, including any Annual Bonus that has been earned
with respect to a prior bonus year, but remains unpaid as of the date of the termination.  If the termination is due to a
Covered  Termination  or  permanent  disability,  provided  that  Executive  first  returns  all  Company  property  in  his
possession and, within sixty (60) days following the Covered Termination, executes and does not revoke an effective
general release of all claims against the Company and its affiliates in a form reasonably acceptable to the Company (a
“Release  of  Claims”),  Executive  shall  also  be  entitled  to  receive  the  following  severance  benefits  described  in  this
Section 4.1.

(a)                Covered Termination Not Related to a Change in Control.   If Executive’s employment terminates due to
a Covered Termination which occurs outside of a Change in Control Period, Executive shall receive the following:

(i)                An amount equal to three (3) months of Executive’s Base Salary payable in substantially equal installments
in  accordance  with  the  Company’s  normal  payroll  policies,  less  applicable  withholdings,  with  such  installments  to
commence as soon as administratively practicable following the date the Release of Claims is not subject to revocation
and, in any event, within sixty (60) days following the date of the Covered Termination.

(ii)             
If Executive is a full time employee at the time, then if Executive elects to receive continued healthcare
coverage  pursuant  to  the  provisions  of  COBRA,  the  Company  shall  directly  pay,  or  reimburse  Executive  for,  the
premium for Executive and Executive’s covered dependents through the earlier of (i) the first anniversary of the date of
Executive’s termination of employment and (ii) the date Executive and Executive’s covered dependents, if any, become
eligible  for  healthcare  coverage  under  another  employer’s  plan(s).    Notwithstanding  the  foregoing,  (i)  if  any  plan
pursuant  to  which  such  benefits  are  provided  is  not,  or  ceases  prior  to  the  expiration  of  the  period  of  continuation
coverage to be, exempt from the application of Section 409A of the Code under Treasury Regulation Section 1.409A-
1(a)(5),  or  (ii)  the  Company  is  otherwise  unable  to  continue  to  cover  Executive  under  its  group  health  plans  without
penalty  under  applicable  law  (including  without  limitation,  Section  2716  of  the  Public  Health  Service Act),  then,  in
either case, an amount equal to each remaining Company subsidy shall thereafter be paid to Executive in substantially
equal monthly installments. After the Company ceases to pay premiums pursuant to this Section 4.1(a)(ii), Executive
may, if eligible, elect to continue healthcare coverage at Executive’s expense in accordance the provisions of COBRA.

 
 
 
 
 
 
 
(iii)            All of Employee’s vested options or stock appreciation rights with respect to the Company’s common stock
shall  remain  exercisable  until  the  first  anniversary  of  Executive’s  termination  of  employment  (or,  if  earlier,  the
maximum period specified in the award documents and plans governing such options or stock appreciation rights, as
applicable, assuming Executive’s employment had not terminated).

(b)                Covered Termination Related to a Change in Control.   If Executive’s employment terminates due to a
Covered Termination that occurs during a Change in Control Period, Executive shall receive the following:

(i)                Executive shall be entitled to receive an amount equal to the Change in Control Multiplier multiplied by the
sum  of:  (i)  Executive’s  Base  Salary  and  (ii)  Executive’s  target  Annual  Bonus  for  the  fiscal  year  of  Executive’s
termination,  in  each  case,  at  the  rate  equal  to  the  higher  of  (x)  the  rate  in  effect  immediately  prior  to  Executive’s
termination of employment or (y) the rate in effect immediately prior to the Change in Control payable in a cash lump
sum, less applicable withholdings, as soon as administratively practicable following the date the Release of Claims is
not subject to revocation and, in any event, within sixty (60) days following the date of the Covered Termination.

(ii)           
  If  Executive  is  a  full  time  employee  at  the  time,  then  if  Executive  elects  to  receive  continued  healthcare
coverage  pursuant  to  the  provisions  of  COBRA,  the  Company  shall  directly  pay,  or  reimburse  Executive  for,  the
premium  for  Executive  and  Executive’s  covered  dependents  through  the  earlier  of  (i)  the  date  that  is  that  number  of
years equal to the Change in Control Multiplier following the date of Executive’s termination of employment and (ii)
the date Executive and Executive’s covered dependents, if any, become eligible for healthcare coverage under another
employer’s plan(s).  Notwithstanding the foregoing, (i) if any plan pursuant to which such benefits are provided is not,
or ceases prior to the expiration of the period of continuation coverage to be, exempt from the application of Section
409A  of  the  Code  under  Treasury  Regulation  Section  1.409A-1(a)(5),  or  (ii)  the  Company  is  otherwise  unable  to
continue  to  cover  Executive  under  its  group  health  plans  without  penalty  under  applicable  law  (including  without
limitation,  Section  2716  of  the  Public  Health  Service Act),  then,  in  either  case,  an  amount  equal  to  each  remaining
Company subsidy shall thereafter be paid to Executive in substantially equal monthly installments. After the Company
ceases  to  pay  premiums  pursuant  to  this  Section  4.1(b)(ii),  Executive  may,  if  eligible,  elect  to  continue  healthcare
coverage at Executive’s expense in accordance with the provisions of COBRA.

 Each outstanding equity award, including, without limitation, each stock option and restricted stock award,
(iii)           
held  by  Executive  shall  automatically  become  vested  and,  if  applicable,  exercisable  and  any  forfeiture  restrictions  or
rights of repurchase thereon shall immediately lapse, in each case, with respect to one hundred percent (100%) of the
shares subject thereto.  To the extent vested after giving effect to the acceleration provided in the preceding sentence,
each stock option held by Executive shall remain exercisable until the earlier of the original expiration date for such
stock option or the second anniversary of Executive’s Covered Termination.

 
 
 
 
 
 
 
(c)                  Termination for Death or Disability. If Executive’s employment is terminated due to death or permanent
disability  where  the  Company  makes  a  determination  in  good  faith  that,  due  to  a  mental  or  physical  incapacity,
Executive has been unable to perform his duties under this Agreement for a period of not less than one-and-a-half (1.5)
consecutive months or 45 days in the aggregate in any 12-month period, Executive shall receive the following:

(i)                An amount equal to three (3) months of Executive’s Base Salary payable in substantially equal installments
in  accordance  with  the  Company’s  normal  payroll  policies,  less  applicable  withholdings,  with  such  installments  to
commence as soon as administratively practicable following the date the Release of Claims is not subject to revocation
and, in any event, within sixty (60) days following the date of the Covered Termination.

(ii)               If Executive (or in the event of death, his designee) elects to receive continued healthcare coverage pursuant
to the provisions of COBRA, the Company shall directly pay, or reimburse Executive for, the premium for Executive
and Executive’s covered dependents through the earlier of (i) the three (3) month anniversary of the date of Executive’s
termination of employment and (ii) the date Executive and Executive’s covered dependents, if any, become eligible for
healthcare coverage under another employer’s plan(s).  Notwithstanding the foregoing, (i) if any plan pursuant to which
such benefits are provided is not, or ceases prior to the expiration of the period of continuation coverage to be, exempt
from  the  application  of  Section  409A  of  the  Code  under  Treasury  Regulation  Section  1.409A-1(a)(5),  or  (ii)  the
Company  is  otherwise  unable  to  continue  to  cover  Executive  under  its  group  health  plans  without  penalty  under
applicable  law  (including  without  limitation,  Section  2716  of  the  Public  Health  Service Act),  then,  in  either  case,  an
amount equal to each remaining Company subsidy shall thereafter be paid to Executive in substantially equal monthly
installments. After the Company ceases to pay premiums pursuant to this Section 4.1(b)(ii), Executive may, if eligible,
elect to continue healthcare coverage at Executive’s expense in accordance with the provisions of COBRA.

4.2.              
280G  Provisions.   Notwithstanding  anything  in  this Agreement  to  the  contrary,  if  any  payment  or
distribution  Executive  would  receive  pursuant  to  this  Agreement  or  otherwise  (“Payment”)  would  (a)  constitute  a
“parachute payment” within the meaning of Section 280G of the Code, and (b) but for this sentence, be subject to the
excise tax imposed by Section 4999 of the Code (the “Excise Tax”), then such Payment shall either be (i) delivered in
full,  or  (ii)  delivered  as  to  such  lesser  extent  which  would  result  in  no  portion  of  such  Payment  being  subject  to  the
Excise  Tax,  whichever  of  the  foregoing  amounts,  taking  into  account  the  applicable  federal,  state  and  local  income
taxes and the Excise Tax, results in the receipt by Executive on an after-tax basis,

 
 
 
 
 
 
of the largest payment, notwithstanding that all or some portion the Payment may be taxable under Section 4999 of the
Code. The accounting firm engaged by the Company for general audit purposes as of the day prior to the effective date
of the Change in Control shall perform the foregoing calculations.  The Company shall bear all expenses with respect to
the  determinations  by  such  accounting  firm  required  to  be  made  hereunder.    The  accounting  firm  shall  provide  its
calculations to the Company and Executive within fifteen (15) calendar days after the date on which Executive’s right
to a Payment is triggered (if requested at that time by the Company or Executive) or such other time as requested by the
Company or Executive.  Any good faith determinations of the accounting firm made hereunder shall be final, binding
and conclusive upon the Company and Executive.  Any reduction in payments and/or benefits pursuant to this Section
4.2 will occur in the following order: (1) reduction of cash payments; (2) cancellation of accelerated vesting of equity
awards  other  than  stock  options;  (3)  cancellation  of  accelerated  vesting  of  stock  options;  and  (4)  reduction  of  other
benefits payable to Executive.

4.3.              Section 409A.

(a)                  Notwithstanding any provision to the contrary in this Agreement, if Executive is deemed at the time of his
Separation  from  Service  to  be  a  “specified  employee”  for  purposes  of  Section  409A(a)(2)(B)(i)  of  the  Code,  to  the
extent  delayed  commencement  of  any  portion  of  the  benefits  to  which  Executive  is  entitled  under  this Agreement  is
required  in  order  to  avoid  a  prohibited  distribution  under  Section  409A(a)(2)(B)(i)  of  the  Code  which  would  subject
Executive  to  a  tax  obligation  under  Section  409A  of  the  Code,  such  portion  of  Executive’s  benefits  shall  not  be
provided to Executive prior to the earlier of (i) the expiration of the six- month period measured from the date of the
Executive’s Separation from Service or (ii) the date of Executive’s death.  Upon the expiration of the applicable Code
Section 409A(a)(2)(B)(i) period, all payments deferred pursuant to this Section 4.3(a) shall be paid in a lump sum to
Executive, and any remaining payments due under the Agreement shall be paid as otherwise provided herein.

(b)                Any reimbursements payable to Executive pursuant to the Agreement shall be paid to Executive no later
than 30 days after Executive provides the Company with a written request for reimbursement, and to the extent that any
such  reimbursements  are  deemed  to  constitute  “nonqualified  deferred  compensation”  within  the  meaning  of  Section
409A  of  the  Code  (i)  such  amounts  shall  be  paid  or  reimbursed  to  Executive  promptly,  but  in  no  event  later  than
December  31  of  the  year  following  the  year  in  which  the  expense  is  incurred,  (ii)  the  amount  of  any  such  payments
eligible  for  reimbursement  in  one  year  shall  not  affect  the  payments  or  expenses  that  are  eligible  for  payment  or
reimbursement  in  any  other  taxable  year,  and  (iii)  Executive’s  right  to  such  payments  or  reimbursement  shall  not  be
subject to liquidation or exchange for any other benefit.

  For  purposes  of  Section  409A  of  the  Code  (including,  without  limitation,  for  purposes  of  Treasury
(c)                
Regulation Section 1.409A-2(b)(2)(iii)), Executive’s right to receive installment payments under the Agreement shall
be treated as a right to receive a series of separate payments and, accordingly, each installment payment hereunder shall
at all times be considered a separate and distinct payment.

 
 
 
 
 
 
 
4.4.               Mitigation.  Executive shall not be required to mitigate damages or the amount of any payment provided
under this Agreement by seeking other employment or otherwise, nor shall the amount of any payment provided for
under  this Agreement  be  reduced  by  any  compensation  earned  by  Executive  as  a  result  of  employment  by  another
employer or by any retirement benefits received by Executive after the date of the Covered Termination, or otherwise.

ARTICLE V
PROPRIETARY INFORMATION OBLIGATIONS

5.1.              Agreement.  Executive agrees to continue to abide by the Confidential Disclosure Agreement.

5.2.                  Remedies.   Executive’s  duties  under  the  Confidential  Disclosure Agreement  shall  survive  termination  of
Executive’s  employment  with  the  Company  and  the  termination  of  this Agreement.    Executive  acknowledges  that  a
remedy  at  law  for  any  breach  or  threatened  breach  by  Executive  of  the  provisions  of  the  Confidential  Disclosure
Agreement, as well as Executive’s obligations pursuant to Section 6.2 and Article 7 below, would be inadequate, and
Executive  therefore  agrees  that  the  Company  shall  be  entitled  to  seek  injunctive  relief  in  case  of  any  such  breach  or
threatened breach.

6.1.                Other Activities.

ARTICLE VI
OUTSIDE ACTIVITIES

(a)                
  Except  for  activities  disclosed  in  Exhibit A  attached,  Executive  shall  not,  during  the  term  of  this
Agreement undertake or engage in any other employment, occupation or business enterprise, other than ones in which
Executive is a passive investor, unless Executive obtains the prior written consent of the Board.

(b)                
 Executive may engage in civic and not-for-profit activities so long as such activities do not materially
interfere with the performance of Executive’s duties hereunder.  In addition, Executive shall be allowed to serve as a
member of the board of directors of up to two (2) other for profit entities at any time during the term of this Agreement,
which service shall not materially interfere with the performance of Executive’s duties hereunder; provided, however,
that  the  Board,  in  its  discretion,  may  require  that  Executive  resign  from  one  or  both  of  such  director  positions  if  it
determines that such resignation(s) would be in the best interests of the Company.

 
 
 
 
 
 
 
 
 
 
6.2.               Competition/Investments.  During the term of Executive’s employment by the Company, except on behalf
of  the  Company,  Executive  shall  not  directly  or  indirectly,  whether  as  an  officer,  director,  stockholder,  partner,
proprietor, associate, representative, consultant, or in any capacity whatsoever engage in, become financially interested
in, be employed by or have any business connection with any other person, corporation, firm, partnership or other entity
whatsoever which were known by Executive to compete directly with the Company, throughout the world, in any line
of business engaged in (or planned to be engaged in) by the Company; provided, however, that anything above to the
contrary notwithstanding, Executive may own, as a passive investor, securities of any competitor corporation, so long
as Executive’s direct holdings in any one such corporation shall not in the aggregate constitute more than 1% of the
voting stock of such corporation.

ARTICLE VII
NONINTERFERENCE

In addition to Executive’s obligations under the Confidential Disclosure Agreement, Executive shall not for a period of
one (1) year following Executive’s termination of employment for any reason, either on Executive’s own account or
jointly  with  or  as  a  manager,  agent,  officer,  employee,  consultant,  partner,  joint  venturer,  owner  or  stockholder  or
otherwise on behalf of any other person, firm or corporation, directly or indirectly solicit or attempt to solicit away from
the Company any of its officers or employees or offer employment to any person who is an officer or employee of the
Company; provided, however, that a general advertisement to which an employee of the Company responds shall in no
event be deemed to result in a breach of this Article 7.  Executive also agrees not to harass or disparage the Company or
its employees, clients, directors or agents or divert or attempt to divert any actual or potential business of the Company.
The provisions of this Article 7 shall survive the termination or expiration of the applicable Executive’s employment
with the Company and shall be fully enforceable thereafter.  If it is determined by a court of competent jurisdiction in
any state that any restriction in this Article 7 is excessive in duration or scope or is unreasonable or unenforceable under
the laws of that state, it is the intention of the parties that such restriction may be modified or amended by the court to
render it enforceable to the maximum extent permitted by the law of that state.

ARTICLE VIII
GENERAL PROVISIONS

8.1.                Notices.  Any notices provided hereunder must be in writing and shall be deemed effective upon the earlier
of personal delivery (including personal delivery by facsimile) or the third day after mailing by first class mail, to the
Company at its primary office location and to Executive at Executive’s address as listed on the Company payroll.

 
 
 
 
 
 
 
 
8.2.               Tax Withholding.  Executive acknowledges that all amounts and benefits payable under this Agreement
are subject to deduction and withholding to the extent required by applicable law.

8.3.              Severability.  Whenever possible, each provision of this Agreement will be interpreted in such manner as to
be  effective  and  valid  under  applicable  law,  but  if  any  provision  of  this Agreement  is  held  to  be  invalid,  illegal  or
unenforceable  in  any  respect  under  any  applicable  law  or  rule  in  any  jurisdiction,  such  invalidity,  illegality  or
unenforceability  will  not  affect  any  other  provision  or  any  other  jurisdiction,  but  this Agreement  will  be  reformed,
construed  and  enforced  in  such  jurisdiction  as  if  such  invalid,  illegal  or  unenforceable  provisions  had  never  been
contained herein.

8.4.                              Waiver.    If  either  party  should  waive  any  breach  of  any  provisions  of  this Agreement,  they  shall  not
thereby  be  deemed  to  have  waived  any  preceding  or  succeeding  breach  of  the  same  or  any  other  provision  of  this
Agreement.

8.5.                               Complete  Agreement.   This Agreement  constitutes  the  entire  agreement  between  Executive  and  the
Company and is the complete, final, and exclusive embodiment of their agreement with regard to this subject matter,
and will supersede all prior agreements, understandings, discussions, negotiations and undertakings, whether written or
oral, between the parties with respect to the subject matter hereof, including without limitation, the Prior Agreement. 
This Agreement is entered into without reliance on any promise or representation other than those expressly contained
herein  or  therein,  and  cannot  be  modified  or  amended  except  in  a  writing  signed  by  an  officer  of  the  Company  and
Executive.

8.6.               Counterparts.  This Agreement may be executed in separate counterparts, any one of which need not
contain signatures of more than one party, but all of which taken together will constitute one and the same Agreement.

8.7.                 Headings.  The headings of the sections hereof are inserted for convenience only and shall not be deemed
to constitute a part hereof nor to affect the meaning thereof.

8.8.               Successors and Assigns.   This Agreement is intended to bind and inure to the benefit of and be enforceable
by Executive and the Company, and their respective successors, assigns, heirs, executors and administrators, except that
Executive may not assign his rights or delegate his duties or obligations hereunder without the prior written consent of
the Company.

 
 
 
 
 
 
 
 
 
 
 
8.9.            
  Arbitration.  Unless otherwise prohibited by law or specified below, all disputes, claims and causes of
action,  in  law  or  equity,  arising  from  or  relating  to  this  Agreement  or  its  enforcement,  performance,  breach,  or
interpretation  shall  be  resolved  solely  and  exclusively  by  final  and  binding  arbitration  held  in  Illinois  in  conformity
with  the  then-existing  employment  arbitration  rules  and  Illinois  law.    The  arbitrator  shall:  (a)  provide  adequate
discovery  for  the  resolution  of  the  dispute;  and  (b)  issue  a  written  arbitration  decision,  to  include  the  arbitrator’s
essential findings and conclusions and a statement of the award.  However, nothing in this section is intended to prevent
either  party  from  obtaining  injunctive  relief  in  court  to  prevent  irreparable  harm  pending  the  conclusion  of  any  such
arbitration.  The Company shall bear the costs of any such arbitration.

8.10.             Executive Acknowledgement.  Executive acknowledges that (a) Executive has consulted with or has had
the  opportunity  to  consult  with  independent  counsel  of  Executive’s  own  choice  concerning  this Agreement,  and  has
been advised to do so by the Company, and (b) that Executive has read and understands the Agreement, is fully aware
of its legal effect, and has entered into it freely based on his own judgment.

8.11.             Choice of Law.   All questions concerning the construction, validity and interpretation of this Agreement
will be governed by the law of the State of Illinois without regard to the conflicts of law provisions thereof.

In Witness Whereof, the parties have executed this Agreement as of the date first written above.

On behalf of Monopar Therapeutics Inc.

/s/ Chandler D. Robinson
Chandler D. Robinson
Chief Executive Officer

Accepted and Agreed:

/s/ Kim R. Tsuchimoto
 Kim R. Tsuchimoto

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
6.1(a) Other Activities.

Exhibit A

50% of full-time employment plus benefits at Mercaptor Discoveries Inc. as Chief Financial Officer, Secretary,
Treasurer and Co-Founder

25% of full-time employment (paid and unpaid) at DNAcheckup (nonprofit) as Chief Financial Officer, Secretary and
Treasurer

 
 
 
 
 
 
 
 
 
 
 
CONSULTING AGREEMENT

This  Consulting Agreement  (herein  referred  to  as "Agreement") is  made  and  entered  into  as  of  this  December  1,  2016  (the
"Effective  Date"),  by  and  between  Monopar  Therapeutics  Inc.  (herein  referred  to  as  "Monopar"),  a  Delaware  limited  liability
corporation. located at corporation, located at 5 Revere Dr., Suite 200, Northbrook, IL 60062, and Andrew P. Mazar (herein referred  to as
"MAZAR") who resides at # (each herein referred to as "Party" and collectively as "Parties'').

RECITALS

WHEREAS, MAZAR specializes in the field of pre-clinical and clinical development, including but not limited to: pre-clinical
study  design,  clinical  trial  design,  clinical  operations,  manufacturing  operations,  regulatory  strategy,  drug  candidate  evaluation,  and
investor due diligence; and

WHEREAS, Monopar desires to contract with MAZAR to provide certain consultation services, as requested by Monopar, and

MAZAR wishes to provide such services to Monopar, upon the terms and conditions set forth below.

NOW, THEREFORE, in consideration of the premises and mutual covenants contained herein, the Parties agree as follows:

1. 

2.

Consulting Arrangement.  MAZAR  agrees  to  perform  consulting  services  as  described  herein  upon  the  terms  and  conditions
herein set forth.

Term of Agreement Subject to the provision for early termination set forth below in Section S of this Agreement, this Agreement
shall  commence  as  of  the  Effective  Date  and  shall  continue  for  a  period  of  twelve  (12)  months  from  the  Effective  Date  (the
"Term"). Either Party may terminate this Agreement without cause with 10-days’ prior written notice.

3. 

Duties of MAZAR.

3.1 

3.2 

Specific Duties. MAZAR shall provide consulting services to Monopar, such duties to include pre-clinical study design,
clinical  trial  design,  clinical  operations  oversight,  manufacturing  oversight,  regulatory  strategy,  drug  candidate
evaluation, and investor due diligence with such other specific requirements as Monopar may specify from time to time
during the Term (herein referred to as the "Services").

MAZAR's Obligations. MAZAR shall be diligent in the performance of Services, and be professional in his commitment
to meeting his obligations hereunder. MAZAR represents and warrants that MAZAR is not party to any other existing
agreement, which any of them would prevent him from entering into this Agreement or which would adversely affect this
Agreement. MAZAR shall not perform Services for any other individuals or entities in direct competition with Monopar,
except  as  provided  for  by  mutual  written  agreement  of the Parties. MAZAR  shall  not  perform  services  for  any  party
which would require or facilitate

 
 
 
 
 
 
 
 
 
 
 
 
 
 
the unauthorized disclosure of any confidential or proprietary information of Monopar.

3.3 

3.4 

Reporting. MAZAR will report to and liaise with Chandler Robinson, M.D., and Christopher M. Starr, Ph.D. and/or any
other assigned Monopar employee or consultant as may be designated in writing by Monopar.

Compensation. Monopar shall pay MAZAR a cash retainer of $25,000 per month not to exceed $300,000 for the period
of this Agreement, unless modified in writing by mutual agreement amongst the Parties.

MAZAR  shall  not  be  reimbursed,  and  is  responsible  for  the  facilities  and  equipment  necessary  to  perform
Services required under this Agreement.

4.

5. 

6. 

7. 

Reimbursement  of  Other  Expenses.  So  long  as  Monopar's  prior  approval has been  obtained,  Monopar  shall  promptly  reimburse
MAZAR for all direct expenses incurred in providing the Services to Monopar pursuant to this Agreement, including travel, meals
and lodging. The invoice submitted by MAZAR pursuant to this Section 4 shall also include a detail of all reimbursable expenses
incurred during the period covered by such invoice.

Termination of Agreement - Failure to perform. In the event that MAZAR ceases to perform the Services or breaches its obligations
as required hereunder for any reason, Monopar shall have the right to immediately terminate this Agreement upon notice to MAZAR
and to enforce such other rights and remedies as it may have as a result of said breach.

Certain Liabilities.  It  is  understood  and  agreed  that  MAZAR shall be acting as an independent  contractor  and  not  as  an  agent  or
employee  of,  or  partner,  joint venturer or in  any  other  relationship  with  Monopar  MAZAR  will  be  solely  responsible for  all  his
insurance, employment taxes, FICA taxes and all obligations to governments or other  organizations  arising  out  of  this  consulting
assignment.  MAZAR  acknowledges that no income,  social  security  or  other  taxes  shall  be  withheld  or  accrued  by  Monopar  for
MAZAR' s benefit. MAZAR assumes all risks and hazards encountered in the performance of duties under this Agreement. Unless
Monopar  has  provided  prior  written  approval,  MAZAR  shall  not  use  any  sub-contractors  to  perform  MAZAR's  obligations
hereunder.  MAZAR  shall  be  solely  responsible  for  any  and  all  injuries,  including  death,  to  all  persons  and  any  and  all  loss  or
damage to property, which may result from performance under this Agreement.

Indemnities.  MAZAR  hereby  agrees  to  indemnify  Monopar  and  hold  Monopar  harmless  from  and  against  all  claims  (whether
asserted by a person, firm, entity or governmental unit or otherwise). liabilities, losses, damages, expenses, charges and fees which
Monopar may sustain or incur arising out of or attributable to any breach, gross negligence or willful misconduct by MAZAR, as
applicable, in the performance under this Agreement. Monopar hereby  agrees  to  indemnify  MAZAR  and  hold MAZAR  harmless
from and against all liabilities losses, damages, expenses, charges and fees which MAZAR may sustain or incur by reason of any
claim which may be asserted against MAZAR by any person, firm, corporation or governmental unit and which may arise out of or
be attributable to any gross

 
 
 
 
 
 
 
 
 
 
 
 
negligence or willful misconduct by Monopar or its employees or contractors, as applicable, in the performance of this Agreement.

8.

9.

10.

11.

Warranties.  The  Services  shall  be  performed  in  a  professional  manner,  consistent  with  industry  standards.  In  performing  the
Services, MAZAR shall not make any unauthorized use of any confidential or proprietary information of any other party or infringe
the intellectual property rights of any other party.

Arbitration. Any controversy or claim between Monopar and MAZAR ari sing out of or relating to this Agreement, or the breach
thereof, shall  be  submitted  to  arbitration  in  accordance  with  the  rules  of  the American Arbitration Association.  The  s ite  of  the
arbitration shall be Chicago, Illinois, and except as provided herein the arbitration shall be conducted in accordance with the Rules
of the American Arbitration Association prevailing at the time the demand for arbitration is made hereunder . At least one member
of the arbitration panel shall be an expert knowledgeable in the area of biopharmaceutical clinical development. Judgment upon any
award rendered by the arbitrator(s) may be entered in any court of competent jurisdiction and shall be binding and final. The cost of
arbitration shall be borne by the losing Party, as determined by the arbitrator(s).

Confidential Information. MAZAR has executed the attached confidential disclosure agreement referenced herein as  Appendix A
prior to commencement of the Services. MAZAR hereby represents and warrants that the obligations thereunder shall be binding.

Inventions. MAZAR agrees that all ideas, developments, suggestions and inventions conceived or reduced to practice arising out of
or  during  the  course  of  performance  under  this Agreement  shall  be  the  exclusive  property  of  Monopar  and  shall  be  promptly
communicated and assigned to Monopar. MAZAR shall require any employees of or other parties contracted by MAZAR to disclose
the same to MAZAR and to be bound by the provisions of this paragraph. During the period of this Agreement and thereafter at any
reasonable  time  when  called  upon  to  do  so  by  Monopar, MAZAR  shall  require  any employees  of  or  other  parties  contracted  by
MAZAR to execute patent applications, assignments to Monopar (or any designee of Monopar) and other papers and to perform acts
which Monopar believes necessary to secure to Monopar full protection and ownership of the rights in and to the services performed
by MAZAR and/or for the preparation, filing and prosecution of applications for patents or inventions made by any employees of or
other parties contracted by MAZAR hereunder. The decision to file patent applications on inventions made by any employees of or
other parties contracted by MAZAR shall be made by Monopar and shall be for such countries, as Monopar shall elect. Monopar
agrees  to  bear  all  the  expense  in  connection  with  the  preparation, filing  and  prosecution  of  applications  for  patents  and  for  all
matters provided in this paragraph requiring the time and/or assistance of MAZAR as to such inventions.

12. Miscellaneous.

12.1 Notice. Any notices to be given hereunder by either Party to the other may be effectuated, in writing, by  personal  delivery  or  by

mail, registered or certified,

 
 
 
 
 
 
 
 
 
 
postage prepaid, with return receipt requested. Mailed notices shall be addressed to the parties at the following addresses:

If to Monopar:

If to MAZAR:

Monopar Therapeutics Inc. 5 Revere Dr., Suite 200
Northbrook, IL, 60062

Attention: Chandler Robinson, MD MBA MSc

Email: #

Andrew P. MAZAR
#
Email: #

or at such other addresses as either Monopar or MAZAR may designate by written notice to each other. Notices delivered personally
shall be deemed duly given on the date of actual receipt; mailed notices shall be deemed duly given as of the fourth day after the date
so mailed.

12.2  Waiver  of  Breach.  The  waiver  by  either  Party  to  a  breach  of  any  provision  in  this  Agreement  cannot  operate  or  be

construed as a waiver of any subsequent breach by either Party.

12.3  Severability.  If  any  provision  of  this  Agreement  is  determined  by  a  court  of  competent  jurisdiction  to  be  invalid  or
unenforceable,  that  provision  shall  be  deemed  modified  to  the  extent  necessary  to  make  it  valid  or  enforceable, or  if  it
cannot be so modified, then severed, and the remainder of the Agreement shall continue in full force and effect as if the
Agreement had been signed with the invalid portion so modified or severed.

12.4 Choice  of  Law.  This  Agreement  has  been  made  and  entered  into  in  the  State  of  Illinois,  and  the  laws  of  such  state,
excluding its choice of law rules, shall govern the validity and interpretation of this Agreement and the performance due
hereunder. The  losing  party  in  any  dispute  hereunder  shall  pay  the  attorneys' fees  and  disbursements  of  the  prevailing
party.

12.5 

Integration.  The  drafting,  execution  and  delivery  of  this  Agreement  by  the  Parties  have  been  induced  by  no
representations, statements, warranties or agreements other than those expressed herein. This Agreement embodies the
entire  understanding  of  the  Parties, and  there  are  no  further  or  other  agreements  or  understandings,  written  or  oral,  in
effect between the Parties relating to the subject matter hereof unless expressly referred to herein.

12.6  Modification. This Agreement may not be modified unless such is in writing and signed by both Parties to this Agreement.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
12.7 

12.8 

Assignment. MAZAR shall not be permitted  to  assign  this Agreement  to  any  other  person  or  entity  without  the  prior
written consent of Monopar. MAZAR hereby agrees that Monopar shall be permitted  to assign  this Agreement to  any
affiliate of Monopar. This Agreement shall be binding upon and shall inure to the benefit of the successors and permitted
assigns of the parties.

Survival. The provisions of Sections 7, 8, 9, 10, and 11 shall survive expiration or termination of this Agreement for any
reason. Expiration or termination of this Agreement shall not affect Monopar's obligations to pay any amounts that may
then be due to MAZAR

IN WITNESS WHEREOF, the Parties hereto  have executed this Agreement as of the day and year first above written.

ACCEPTED AND AGREED TO:                                                                                       ..

Andrew P. Mazar                                                                             MONOPAR THERAPEUTICS INC.

/s/ Andrew P. Mazar                                                                        /s/ Chandler D. Robinson

BY: ANDREW P. MAZAR                                                            BY: CHANDLER D. ROBINSON
                          ITS: CHIEF EXECUTIVE OFFICER

 
 
 
 
 
 
 
 
 
 
 
 
 
APPENDIX A

See executed CDA attached

 
 
 
 
 
EXECUTIVE EMPLOYMENT AGREEMENT

This  Executive  Employment Agreement  (the   "Agreement")  is  entered  into  as  of  November  1,  2017,  by  and
between Andrew P. Mazar ("Executive") and Monopar Therapeutics Inc. (the "Company").

Whereas, the Company desires to employ Executive as its Executive Vice President, Research and Development
and Chief Scientific Officer, effective as of November 1, 2017 (the "Effective Date"), and Executive desires to
serve in such capacity, pursuant to the terms and conditions set forth in this Agreement; and

Now, Therefore, in consideration of the mutual promises and covenants contained herein, it is hereby agreed by
and between the parties hereto as follows:

ARTICLE I

DEFINITIONS

For purposes of the Agreement, the following terms are defined as follows:

1.1. "Board" means the Board of Directors of the Company.

1.2. "Cause" means any of the following events described below:

(a) Executive's conviction of a felony or other crime involving moral turpitude;

(b) any willful act or acts of dishonesty undertaken by Executive and intended to result in substantial gain or personal

enrichment of Executive, Executive's family or any third party at the expense of the Company;

(c) any willful act of gross misconduct which is materially and demonstrably injurious to the Company; and/or

(d) Executive's inability under applicable law to continue to work lawfully in the United States.

For the purpose of this Agreement, no act, or failure to act, by Executive shall be considered "willful" if done, or
omitted  to  be  done,  by  him  in  good  faith  and  in  the  reasonable  belief  that  his  act  or  omission  was  in  the  best
interest of the Company and/or required by applicable law.

1.3. "Change in Control" means the occurrence of any of the following events: (i) any sale or exchange of the

capital stock by the stockholders of the Company in one transaction

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
or  series  of  related  transactions  where  more  than  fifty  percent  (50%)  of  the  outstanding  voting  power  of  the
Company  is  acquired  by  a  person  or  entity  or  group  of  related  persons  or  entities;  or  (ii)  any  reorganization,
consolidation or merger of the Company where the outstanding voting securities of the Company immediately
before  the  transaction  represent  or  are  converted  into  less  than  fifty  percent  (50%)  of  the  outstanding  voting
power  of  the  surviving  entity  (or  its  parent  corporation)  immediately  after  the  transaction;  or  (iii)  the
consummation of any transaction or series of related transactions that results in the sale of all or substantially all
of  the  assets  of  the  Company;  or  (iv)  any  "person"  or  "group"  (as  defined  in  the  Securities  Exchange Act  of
1934, as amended (the "Exchange Act") becoming the "beneficial owner" (as defined in Rule 13d-3 under the
Exchange Act) directly or indirectly of securities representing more than fifty percent (50%) of the voting power
of the Company then outstanding. Except that any change in the beneficial ownership of the securities of the
Company as a result of a private financing of the Company that is approved by the Board, shall not be deemed
to be a Change in Control.

1.4.

"Change in Control Multiple"  shall mean one and a half (1.5).

1.5.  "Change in Control Period"  means that period commencing on the consummation of a Change in Control and

ending on the first anniversary thereof.

1.6.  COBRA" means the Consolidated Omnibus Budget Reconciliation Act of 1985, as amended.

1.7.

"Code" means the Internal Revenue Code of 1986, as amended.

1.8.

"Company" means Monopar Therapeutics Inc. or any successor thereto.

1.9.  "Confidential Disclosure Agreement" means the Confidential Disclosure Agreement entered into between

Executive and the Company.

     1.10.       "Covered Termination" means (a) an Involuntary Termination Without Cause or  (b) a voluntary
termination for Good Reason, provided that the termination constitutes a Separation
   from Service.

1.11. "Good Reason" means Executive' s resignation as a result of a Good Reason Condition. In order to resign for
Good Reason, Executive must provide written notice to the Company of the existence of the Good Reason Condition
within  thirty  (30)  days  of  the  initial  existence  of  such  Good  Reason  Condition.  Upon  receipt  of  such  notice  of  the
Good Reason Condition, the Company will be provided with a period of thirty (30) days during which it may remedy
the Good Reason Condition and not be required to provide for the payments and benefits described in Section 4 as a
result  of  such  proposed  resignation  due  to  the  Good  Reason  Condition  specified  in  the  notice.  If  the  Good  Reason
Condition is not remedied within the period specified in the preceding sentence, Executive may resign for

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Good Reason based on the Good Reason Condition specified in the notice, provided that such resignation must
occur within sixty (60) days after the initial existence of such Good Reason Condition.

1.12. "Good Reason Condition"  means that any of the following are undertaken without Executive's express written

consent:

(a) a material reduction in Executive's Base Salary;

(b)

(c)

a material diminution in Executive's responsibilities;

the Company's material breach of any material term of this Agreement; or

(d) a requirement that Executive relocate to an office that would increase Executive's one-way commute distance by

more than fifty (50) miles based on Executive's primary residence at the time such relocation is announced.

1.13. "Involuntary Termination Without Cause" means Executive's dismissal or discharge by the Company other
than for Cause. The termination of Executive's employment as a result of Executive's death or inability to perform the
essential functions of his job due to disability will not be deemed to be an Involuntary Termination Without Cause.

1.14. "Separation from Service" means Executive's termination of employment or service where such termination

of employment or service constitutes a "separation from service" within the meaning of Treasury Regulation Section
1.409A-l(h).

ARTICLE II

EMPLOYMENT BY THE COMPANY

2.1. Position  and  Duties.   Subject  to  terms  set  forth  herein,  as  of  the  Effective  Date,  Executive  shall  serve  as  the
Company's  Executive  Vice  President,  Research  and  Development  and  Chief  Scientific  Officer,  and  perform  such
duties  as  are  customarily  associated  with  the  position  of  Executive  Vice  President,  Research  and  Development  and
Chief  Scientific  Officer,  and  such  other  duties  as  are  assigned  to  Executive  by  the  Chief  Executive  Officer  or  the
Board. During the term of Executive's employment with the Company, Executive will devote Executive's best efforts
and substantially all of Executive's business time and attention (except for vacation periods and reasonable periods of
illness or other incapacities permitted by the Company's general employment policies, if any, or as otherwise set forth
in this Agreement) to the business of the Company.

2.2. Employment at Will. Both the Company and Executive shall have the right to terminate Executive's

employment with the Company at any time, with or without Cause,

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
and without prior notice. If Executive's employment with the Company is terminated, Executive will be eligible
to receive severance benefits to the extent provided in this Agreement.

2.3. Employment Policies. The employment relationship between the parties shall also be governed by the general

employment policies and practices of the Company, if any, including those relating to protection of confidential
information and assignment of inventions, except that when the terms of this Agreement differ from or are in conflict
with the Company's general employment policies or practices, this Agreement shall control.

ARTICLE III
COMPENSATION

3.1. Base Salary. As of the Effective Date, Executive shall receive for services to be rendered hereunder an annual
base salary of $350,000 ("Base Salary"), payable on the regular payroll dates of the Company, subject to increase in
the sole discretion of the Board.

3.2. Sign-on Bonus. Executive shall be paid a one-time sign-on bonus of $8,750 (gross before taxes) payable with

Executive's first regular paycheck.

3.3. Annual Bonus. Executive is subject to an annual bonus at the discretion of the Board, which bonus is initially

being targeted for up to 40% of the annualized amount of Base Salary.

3.4.  Standard  Company  Benefits.  Executive  shall  be  entitled  to  all  rights  and  benefits  for  which  Executive  is
eligible under the terms and conditions of the standard Company benefits and compensation practices, if any, that may
be in effect from time to time and are provided by the Company to its executive employees generally. Executive shall
be entitled each year to four (4) weeks leave for vacation at full pay, provided, that the maximum amount Executive
may  have  accrued  at  any  point  in  time  is  four  (4)  weeks  (meaning  that  once  Executive  has  accrued  four  (4)  weeks,
Executive will not accrue any additional vacation time until he takes vacation and falls below the four (4) week accrual
cap).  Executive  shall  also  be  entitled  to  reasonable  holidays  and  illness  days  with  full  pay  in  accordance  with  the
policies applicable to the Company and its affiliates, if any, from time to time in effect. Employee acknowledges and
agrees  that  in  order  to  maintain  flexibility,  the  Company  and  its  affiliates  have  the  right  to  amend  or  terminate  any
employee benefit plan at any time. Until such time as the Company obtains healthcare benefits for eligible employees
and Executive elects to opt in to such benefits, Executive shall be entitled to an additional salary of at least $4,583.33
per month or such greater amount as determined by the Board.

3.5. Stock Options. Subject to approval by the Board, Executive may be granted options to purchase shares of the

Company's common stock with an exercise price per share

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
as determined by the Compensation Committee or similar function of the Board.

3.6. Expenses. The Company will reimburse Executive for all reasonable and necessary expenses incurred by

Employee in connection with the Company's business, provided that such expenses incurred and are properly
documented and accounted for in accordance with the policy of the Company and requirements of the Internal Revenue
Service.

ARTICLE IV
SEVERANCE AND CHANGE IN CONTROL BENEFITS

4.1.  Severance  Benefits.  Upon  Executive's  termination  of  employment,  Executive  shall  receive  any  accrued  but
unpaid  Base  Salary  and  other  accrued  and  unpaid  compensation,  including  any Annual  Bonus  that  has  been  earned
with respect to a prior year, but remains unpaid as of the date of the termination. If the termination is due to a Covered
Termination or permanent disability, provided that Executive first returns all Company property in his possession and,
within sixty (60) days following the Covered Termination, executes and does not revoke an effective general release of
all  claims  against  the  Company  and  its  affiliates  in  a  form  reasonably  acceptable  to  the  Company  and  Executive  (a
"Release of Claims"),   Executive  shall  also  be  entitled  to  receive  the  following  severance  benefits  described  in  this
Section 4.1.

(a) Covered Termination Not Related to a Change in Control.  If Executive's employment terminates due to a

Covered Termination which occurs outside of a Change in Control Period, Executive shall receive the following:

(i) An amount equal to twelve (12) months of Executive's Base Salary payable in substantially equal installments in
accordance with the Company's normal payroll policies, if any, less applicable withholdings, with such installments to
commence as soon as administratively practicable following the date the Release of Claims is not subject to revocation
and, in any event, within sixty (60) days following the date of the Covered Termination.

(ii) If Executive elects to receive continued healthcare coverage pursuant to the provisions of COBRA, the Company
shall directly pay, or reimburse Executive for, the premium for Executive and Executive's covered dependents through
the earlier of (i) the first anniversary of the date of Executive's termination of employment and (ii)  the date Executive
and Executive's covered dependents, if any, become eligible for healthcare coverage under another employer's plan(s).
Notwithstanding the foregoing, (i) if any plan pursuant to which such benefits are provided is not, or ceases prior to the
expiration  of  the  period  of  continuation  coverage  to  be,  exempt  from  the  application  of  Section  409A  of  the  Code
under  Treasury  Regulation  Section  l.409A-l(a)(5),  or  (ii)  the  Company  is  otherwise  unable  to  continue  to  cover
Executive under its group health plans without penalty under

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
applicable law (including without limitation, Section 2716 of the Public Health Service Act), then, in either case,
an amount equal to each remaining Company subsidy shall thereafter be paid to Executive in substantially equal
monthly installments. After the Company ceases to pay premiums pursuant to this Section 4.l(a)(ii), Executive
may, if eligible, elect to continue healthcare coverage at Executive's expense in accordance with the provisions
of COBRA.

(iii) All of Employee's vested options or stock appreciation rights with respect to the Company's common stock shall

remain exercisable until the first anniversary of Executive's termination of employment (or, if earlier, the maximum
period specified in the award documents and plans governing such options or stock appreciation rights, as applicable,
assuming Executive's employment had not terminated).

(b) Covered Termination Related to a Change in Control.  If Executive's employment terminates due to a Covered

Termination that occurs during a Change in Control Period, Executive shall receive the following:

     (i)     Executive shall be entitled to receive an amount equal to the Change in Control Multiplier multiplied by the
sum  of:  (i)  Executive's  Base  Salary  and  (ii)  Executive '  s  target  Annual  Bonus  for  the  fiscal  year  of  Executive's
termination,  in  each  case,  at  the  rate  equal  to  the  higher  of  (x)  the  rate  in  effect  immediately  prior  to  Executive's
termination of employment or (y) the rate in effect immediately prior to the Change in Control payable in a cash lump
sum, less applicable withholdings, as soon as administratively practicable following the date the Release of Claims is
not subject to revocation and, in any event, within sixty (60) days following the date of the Covered Termination.

          (ii)     If  Executive  elects  to  receive  continued  healthcare  coverage  pursuant  to  the  provisions  of  COBRA,  the
Company shall directly pay, or reimburse Executive for, the premium for Executive and Executive's covered dependents
through the earlier of (i) the date that is that number of years equal to the Change in Control Multiplier following the
date of Executive's termination of employment and (ii) the date Executive and Executive's covered dependents, if any,
become  eligible  for  healthcare  coverage  under  another  employer's  plan(s).  Notwithstanding  the  foregoing,  (i)  if  any
plan pursuant to which such benefits are provided is not, or ceases prior to the expiration of the period of continuation
coverage to be, exempt from the application of Section 409A of the Code under Treasury Regulation Section 1.409A-
l(a)(5),  or  (ii)  the  Company  is  otherwise  unable  to  continue  to  cover  Executive  under  its  group  health  plans  without
penalty  under  applicable  law  (including  without  limitation,  Section  2716  of  the  Public  Health  Service Act),  then,  in
either case, an amount equal to each remaining Company subsidy shall thereafter be paid to Executive in substantially
equal monthly installments. After the Company ceases to pay premiums pursuant to this Section 4.l(b)(ii), Executive
may,  if  eligible,  elect  to  continue  healthcare  coverage  at  Executive's  expense  in  accordance  with  the  provisions  of
COBRA.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
    (iii)     Each outstanding equity award, including, without limitation, each stock option and restricted stock award,
held  by  Executive  shall  automatically  become  vested  and,  if  applicable,  exercisable  and  any  forfeiture  restrictions  or
rights of repurchase thereon shall immediately lapse, in each case, with respect to one hundred percent (100%) of the
shares subject thereto. To the extent vested after giving effect to the acceleration provided in the preceding sentence,
each stock option held by Executive shall remain exercisable until the earlier of the original expiration date for such
stock option or the second anniversary of Executive's Covered Termination.

(c) Termination for Death or Disability.  If Executive's employment is terminated due to death or permanent

disability where the Company makes a determination in good faith that, due to a mental or physical incapacity,
Executive has been unable to perform his duties under this Agreement for a period of not less than six (6) consecutive
months or 180 days in the aggregate in any 12-month period, Executive shall receive the following:

(i) An  amount  equal  to  three  (3)  months  of  Executive's  Base  Salary  payable  in  substantially  equal  installments  in
accordance  with  the  Company's  normal  payroll  policies,  less  applicable  withholdings,  with  such  installments  to
commence as soon as administratively practicable following the date the Release of Claims is not subject to revocation
and, in any event, within sixty (60) days following the date of the Covered Termination.

(ii) If Executive (or in the event of death, his designee) elects to receive continued healthcare coverage pursuant to the
provisions  of  COBRA,  the  Company  shall  directly  pay,  or  reimburse  Executive  for, the  premium  for  Executive  and
Executive's  covered  dependents  through  the  earlier  of  (i)  the  three  (3)  month  anniversary  of  the  date  of  Executive's
termination of employment and (ii) the date Executive and Executive's covered dependents, if any, become eligible for
healthcare coverage under another employer's plan(s). Notwithstanding the foregoing, (i) if any plan pursuant to which
such benefits are provided is not, or ceases prior to the expiration of the period of continuation coverage to be, exempt
from  the  application  of  Section  409A  of  the  Code  under  Treasury  Regulation  Section  l.409A-l(a)(5),  or  (ii)  the
Company  is  otherwise  unable  to  continue  to  cover  Executive  under  its  group  health  plans  without  penalty  under
applicable law (including without limitation, Section 2716 of the Public Health Service Act), then, in either case, an
amount equal to each remaining Company subsidy shall thereafter be paid to Executive in substantially equal monthly
installments. After the Company ceases to pay premiums pursuant to this Section 4.l(b)(ii), Executive may, if eligible,
elect to continue healthcare coverage at Executive's expense in accordance the provisions of COBRA.

4.2. 280G Provisions.  Notwithstanding anything in this Agreement to the contrary ,  if any payment or dis tribution
Executive  would  receive  pursuant  to  this Agreement  or   otherwise  ("Payment")  would  (a)  constitute  a  "parachute
paymen"t within the meaning of  Section 280G of the Code, and  (b) but for this sentence, be subject to the excise tax
imposed

 
 
 
 
 
 
 
 
 
 
 
by Section 4999 of the Code (the  "Excise Tax"), then such Payment shall either be  (i) delivered in full, or   (ii)
delivered as to such lesser extent which would result in no portion of such Payment being subject to the Excise
Tax,  whichever  of  the  foregoing  amounts,  taking  into  account  the  applicable  federal,  state  and  local  income
taxes  and  the  Excise  Tax,  results  in  the  receipt  by  Executive  on  an  after-tax  basis,  of  the  largest  payment,
notwithstanding  that  all  or  some  portion  the  Payment  may  be  taxable  under  Section  4999  of  the  Code.  The
accounting firm engaged by the Company for general audit purposes as of the day prior to the effective date of
the  Change  in  Control  shall  perform  the  foregoing  calculations.  The  Company  shall  bear  all  expenses  with
respect to the determinations by such accounting firm required to be made hereunder. The accounting firm shall
provide its calculations to the Company and Executive within fifteen (15) calendar days after the date on which
Executive's right to a Payment is triggered (if requested at that time by the Company or Executive) or such other
time as requested by the Company or Executive. Any good faith determinations of the accounting firm made
hereunder shall be final, binding and conclusive upon the Company and Executive. Any reduction in payments
and/or benefits pursuant to this Section 4.2 will occur in the following order:  (1)  reduction of cash payments;
(2) cancellation of accelerated vesting of equity awards other than stock options; (3) cancellation of accelerated
vesting of stock options; and (4) reduction of other benefits payable to Executive.

4.3.

Section 409A.

(a)  Notwithstanding  any  provision  to  the  contrary  in  this  Agreement,  if  Executive  is  deemed  at  the  time  of  his
Separation  from  Service  to  be  a  "specified  employee"  for  purposes  of  Section  409A(a)(2)(B)(i)  of  the  Code,  to  the
extent delayed commencement of any portion of the benefits to which Executive is entitled under this Agreement is
required in order to avoid a prohibited distribution under Section 409A(a)(2)(B)(i) of the Code which would subject
Executive  to  a  tax  obligation  under  Section  409A  of  the  Code,  such  portion  of  Executive's  benefits  shall  not  be
provided to Executive prior to the earlier of  (i)  the expiration of the six- month period measured from the date of the
Executive's Separation from Service or (ii)  the date of  Executive's  death. Upon the expiration of the applicable Code
Section 409A(a)(2)(B)(i) period, all payments deferred pursuant to this Section 4.3(a) shall be paid in a lump sum to
Executive, and any remaining payments due under the Agreement shall be paid as otherwise provided herein.

(b) Any reimbursements payable to Executive pursuant to the Agreement shall be paid to  Executive no later than 30
days after Executive provides the Company with a written request for reimbursement, and to the extent that any such
reimbursements are deemed to constitute "nonqualified deferred compensation" within the meaning of Section 409A of
the Code (i) such amounts shall be paid or reimbursed to Executive promptly , but in no event later than December 31
of  the  year  following  the  year  in  which  the  expense  is  incurred,  (ii)  the  amount  of  any  such  payments  eligible  for
reimbursement in one year shall not affect the payments or expenses that are eligible for payment or reimbursement in
any other taxable

 
 
 
 
 
 
 
 
 
 
 
 
 
 
year,  and  (iii)  Executive's  right  to  such  payments  or  reimbursement  shall  not  be  subject  to  liquidation  or
exchange for any other benefit.

(c) For  purposes  of  Section  409A  of  the  Code  (including,  without  limitation,  for  purposes  of  Treasury  Regulation
Section 1.409A-2(b)(2)(iii)), Executive's right to receive installment payments under the Agreement shall be treated as
a right to receive a series of separate payments and, accordingly, each installment payment hereunder shall at all times
be considered a separate and distinct payment.

4.4. Mitigation. Executive shall not be required to mitigate damages or the amount of any payment provided under
this Agreement by seeking other employment or otherwise, nor shall the amount of any payment provided for under
this Agreement be reduced by any compensation earned by Executive as a result of employment by another employer
or by any retirement benefits received by Executive after the date of the Covered Termination, or otherwise.

ARTICLE V

PROPRIETARY INFORMATION OBLIGATIONS

5.1. Agreement. Executive agrees to continue to abide by the Confidential Disclosure Agreement.

5.2.  Remedies.  Executive's  duties  under  the  Confidential  Disclosure  Agreement  shall  survive  termination  of
Executive's  employment  with  the  Company  and  the  termination  of  this Agreement.  Executive  acknowledges  that  a
remedy  at  law  for  any  breach  or  threatened  breach  by  Executive  of  the  provisions  of  the  Confidential  Disclosure
Agreement, as well as Executive's obligations pursuant to Section 6.2 and Article 7 below , would be inadequate, and
Executive therefore agrees that the Company shall be entitled to seek injunctive relief in case of any such breach or
threatened breach.

ARTICLE VI OUTSIDE ACTIVITIES

6.1.

Other Activities.

(a) Executive shall not, during the term of this Agreement undertake or engage in any other employment, occupation
or  business  enterprise,  other  than  ones  in  which  Executive  is  a  passive  investor,  unless  he  obtains  the  prior  written
consent of the Board.

(b) Executive may engage in civic and not-for-profit activities so long as such activities do not materially interfere
with the performance of Executive's duties hereunder. In addition, Executive shall be allowed to serve as a member of
the board of directors of up to two (2) other for profit entities at any time during the term of this

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Agreement, which service shall not materially interfere with the performance of Executive's duties hereunder;
provided, however, that the Board may require that Executive resign from one or both of such director positions
if it can reasonably and in good faith demonstrate that such resignation(s) would be in the best interests of the
Company in a significant and material way.

   6.2.         Competition.  Executive agrees that, from the date hereof until a period of twelve  (12) months following the
date of termination of Executive's employment with the Company, Executive will not directly or indirectly, either as an
employee,  employer,  consultant,  agent,  principal,  partner,  corporate  officer,  director,  or  in  any  other  individual  or
representative capacity, engage or participate in any "Competitive Business" anywhere in the United States of America.
As  used  herein,  a  "Competitive  Business"  is  defined  as  any  business  developing  uPAR  antibodies  to  treat  cancer,  or
clonidine to treat oral mucositis.

ARTICLE VII NONINTERFERENCE

In  addition  to  Executive's  obligations  under  the  Confidential  Disclosure Agreement,  Executive  shall  not  for  a
period  of  one  (1)  year  following  Executive's  termination  of  employment  for  any  reason,  either  on  Executive's
own account or jointly with or as a manager, agent, officer, employee, consultant, partner, joint venturer, owner
or stockholder or otherwise on behalf of any other person, firm or corporation, directly or indirectly solicit or
attempt to solicit away from the Company any of its officers or employees or offer employment to any person
who  is  an  officer  or  employee  of  the  Company;  provided, however,   that  a  general  advertisement  to  which  an
employee of the Company responds shall in no event be deemed to result in a breach of this Article 7. Executive
also  agrees  not  to  harass  or  disparage  the  Company  or  its  employees,  clients,  directors  or  agents  or  divert  or
attempt to divert any actual or potential business of the Company. The provisions of this Article 7 shall survive
the  termination  or  expiration  of  the  applicable  Executive's  employment  with  the  Company  and  shall  be  fully
enforceable thereafter. If it is determined by a court of competent jurisdiction in any state that any restriction in
this Article 7 is excessive in duration or scope or is unreasonable or unenforceable under the laws of that state, it
is  the  intention  of  the  parties  that  such  restriction  may  be  modified  or  amended  by  the  court  to  render  it
enforceable to the maximum extent permitted by the law of that state.

ARTICLE VIII GENERAL PROVISIONS

8.1. Notices. Any notices provided hereunder must be in writing and shall be deemed effective upon the earlier of
personal delivery (including personal delivery by facsimile) or the third day after mailing by first class mail, to the
Company at its primary office location and to Executive at Executive's address as listed on the Company payroll.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
8.2. Tax Withholding. Executive acknowledges that all amounts and benefits payable under this Agreement are

subject to deduction and withholding to the extent required by applicable law.

8.3. Severability. Whenever possible, each prov1s1on of this Agreement will be interpreted in such manner as to be
effective  and  valid  under  applicable  law,  but  if  any  provision  of  this  Agreement  is  held  to  be  invalid,  illegal  or
unenforceable  in  any  respect  under  any  applicable  law  or  rule  in  any  jurisdiction,  such  invalidity,  illegality  or
unenforceability  will  not  affect  any  other  provision  or  any  other  jurisdiction,  but  this Agreement  will  be  reformed,
construed  and  enforced  in  such  jurisdiction  as  if  such  invalid,  illegal  or  unenforceable  provisions  had  never  been
contained herein.

8.4. Waiver. If either party should waive any breach of any provisions of this Agreement , they shall not thereby be

deemed to have waived any preceding or succeeding breach of the same or any other provision of this Agreement.

8.5. Complete Agreement.   This Agreement  constitutes  the  entire  agreement  between  Executive  and  the  Company
and  is  the  complete,  final,  and  exclusive  embodiment  of  their  agreement  with  regard  to  this  subject  matter,  and  will
supersede  all  prior  agreements,  understandings,  discussions,  negotiations  and  undertakings,  whether  written  or  oral,
between the parties with respect to the subject matter hereof, including without limitation, the Prior Agreement. This
Agreement  is  entered  into  without  reliance  on  any  promise  or  representation  other  than  those  expressly  contained
herein  or  therein,  and  cannot  be  modified  or  amended  except  in  a  writing  signed  by  an  officer  of  the  Company  and
Executive.

8.6. Counterparts.  This Agreement  may  be  executed  in  separate  counterparts,  any  one  of  which  need  not  contain

signatures of more than one party, but all of which taken together will constitute one and the same Agreement.

8.7. Headings. The headings of the sections hereof are inserted for convenience only and shall not be deemed to

constitute a part hereof nor to affect the meaning thereof.

8.8. Successors and Assigns.  This Agreement is intended to bind and inure to the benefit of and be enforceable by
Executive and the Company, and their respective successors, assigns, heirs,  executors and administrators, except that
Executive may not assign his rights or delegate his duties or obligations hereunder without the prior written consent of
the Company.

8.9. Arbitration. Unless otherwise prohibited by law or specified below, all disputes, claims and causes of action, in
law  or  equity,  arising  from  or  relating  to  this Agreement  or  its  enforcement,  performance,  breach ,  or  interpretation
shall be resolved solely and exclusively by final and binding arbitration held in Illinois in conformity with the then-

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
existing employment arbitration rules and Illinois law. The arbitrator shall: (a) provide adequate discovery for
the  resolution  of  the  dispute;  and  (b)  issue  a  written  arbitration  decision,  to  include  the  arbitrator's  essential
findings and conclusions and a statement of the award. However, nothing in this section is intended to prevent
either party from obtaining injunctive relief in court to prevent irreparable harm pending the conclusion of any
such arbitration. The Company shall bear the costs of any such arbitration.

8.10.  Executive  Acknowledgement.   Executive  acknowledges  that  (a)  he  has  consulted  with  or  has  had  the
opportunity to consult with independent counsel of his own choice concerning this Agreement, and has been advised to
do so by the Company, and (b) that he has read and understands the Agreement, is fully aware of its legal effect, and
has entered into it freely based on his own judgment.

8.11. Choice of Law. All questions concerning the construction, validity and interpretation of this Agreement will be

governed by the law of the State of Illinois without regard to the conflicts of law provisions thereof.

In Witness Whereof, the parties have executed this Agreement as of the date first written above.

On behalf of Monopar Therapeutics Inc.

      /s/ Chandler D. Robinson

      Chandler D. Robinson

      Chief Executive Officer

   Accepted and Agreed:

/s/ Andrew P. Mazar
Andrew P. Mazar

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
CONSULTING AGREEMENT

This Consulting Agreement (herein referred to as "'Agreement'') is made and entered into as of this December 15,  2016  (the
"Effective Date"), by and between Monopar Therapeutics, Inc. (herein referred to as "Monopar'·). a Delaware corporation, located at 5
Revere Dr., Suite 200, Northbrook, IL 60062, and pRx Consulting, LLC (herein referred to as pRx), a Delaware corporation located at #
(each herein referred to as 'Party' and collectively as "Parties'').

                                                           RECITALS

WHEREAS. pRx specializes in the field of clinical  development,  including  but  not  limited  to:  clinical  trial  design,  statistical

modeling, clinical operations, regulatory strategy and investor due diligence.

WHEREAS. Monopar desires to contract with pRx to provide certain consultation services, as requested by Monopar, and pRx

wishes to provide such services to Monopar, upon the terms and conditions set forth below.

1.

2. 

NOW, THEREFORE, in consideration of the premises and mutual covenants contained herein. the Parties agree as follows:

Consulting Arrangement. pRx agrees to perform consulting services as described herein upon the terms and conditions herein set
forth.

Term of Agreement. Subject to the provision for early termination set forth below in Section 5 of this Agreement, this Agreement
shall commence as of the Effective Date and shall continue for a period of six (6) months from the Effective Date (the "Term").
Either Party may terminate this Agreement without cause with 10-days' prior written notice.

3. 

Duties of pRx.

3.1 

3.2 

Specific Duties. pRx shall provide consulting services to Monopar, such duties to include clinical trial design, statistical
modeling  ,  clinical  operations  oversight,  regulatory  strategy  and  investor  due  diligence  with  such  other  specific
requirements as Monopar may specify from time to time during the Term (herein referred to as the "Services ").

pRx's  Obligations.  pRx  shall  be  diligent  in  the  performance  of  Services,  and  be  professional  in  its  commitment  to
meeting its obligations hereunder. pRx represent s and warrants that pRx is not  party  to any other  existing  agreement,
which  any  of  them  would  prevent  pRx  from  entering  into  this  Agreement  or  which  would  adversely  affect  this
Agreement. pRx shall not  perform  Services  for any other individuals  or  entities  in  direct  competition  with  Monopar,
except as provided for by mutual written agreement of the Parties. pRx shall not perform services for any party which
would require or facilitate the unauthorized disclo sure of any confidential or proprietary information of Monopar.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
3.3

Reporting. pRx will report to  and  liaise  with Andrew  P.  Mazar , Ph.D., Chandler Robinson,  M.D.,  and/or  any  other
assigned Monopar employee or consultant as may be designated in writing by Monopar.

3.4 

Compensation. Monopar shall pay pRx as follows:

a.          Five thousand dollars ($5,000) per month in arrears payable on 15-Jan-2017, 15-Feb- 2017, 15-Mar-

201,715-Apr-2017. 15-May-2017 and 15-Jun-2017.

b.          Upon approval of the Monopar Board of Directors, Dr. P. Rioux. president of pRx  Consulting, LLC shall
be granted stock options to purchase up to 100 shares of Monopar's common stock at an exercise price of $0.001 (representing
Monopar's par value of its common stock). Such stock option shall vest as follows: on January 15, 2017, options to purchase up
to 17 shares; on February 15, 2017, options to purchase up to 16 shares; on March 15, 2017, options to purchase up to 17 shares;
on April 15, 2017, options to purchase up to 16 shares; on May 15, 2017, options to purchase up to 17 shares; and on June 15,
2017 options to purchase up to 17 shares of Monopar's common stock. Such vesting shall terminate upon the termination of this
Agreement.  The  number  of  shares,  the  exercise  price  thereof  and  the  rights  granted  under  this  Agreement  are  subject  to
adjustment and modification as provided in the Monopar Therapeutics Inc. 2016 Stock Incentive Plan.

pRx shall not be reimbursed, and is responsible for the facilities and equipment necessary to perform Services required under this
Agreement.

4. 

5. 

6. 

Reimbursement of Other Expenses. So long as Monopar's prior approval has been obtained, Monopar shall promptly reimburse
pR.x for all direct expenses incurred in providing the Services to Monopar pursuant to this Agreement, including travel, meals and
lodging. The invoice submitted by pR.x pursuant to this Section 4 shall also include a detail of all reimbursable expenses incurred
during the period covered by such invoice.

Termination of Agreement  - Failure to perform. In the event that pR.x ceases to perform the Services or breaches its obligations
as required hereunder for any reason, Monopar shall have the right to immediately terminate this Agreement upon  notice to pRx
and to enforce such other rights and remedies as it may have as a result of said breach.

Certain Liabilities. It  is  understood  and  agreed  that  pRx  shall  be  acting  as  an  independent  contractor  and  not  as  an  agent  or
employee of, or partner, joint venturer or in any other relationship with Monopar. pRx will be solely responsible for all insurance,
employment taxes, FICA taxes and all obligations to governments or other organizations for it and  its employees arising out of
this consulting assignment. pRx acknowledges that  no  income,  social  security  or  other  taxes  shall   be  withheld  or  accrued  by
Monopar for pRx' s or its employees' benefit. pRx assumes all risks and hazards encountered in the performance of duties by it or
its employees under this Agreement. Unless Monopar has provided prior written approval, pRx shall not use any sub-contractors
to perform pRx' s obligations hereunder. pRx shall be solely responsible for any and all injuries, including death, to all

- 2 -

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
7. 

8. 

9. 

10. 

11. 

persons and any and all loss or damage to property, which may result from performance under this Agreement.

Indemnities. pRx hereby agrees to indemnify Monopar and hold Monopar harmless from and against all claims (whether asserted
by  a  person,  firm,  entity  or  governmental  unit  or  otherwise),  liabilities,  losses,  damages,  expenses,  charges  and  fees  which
Monopar may sustain or incur arising out of or attributable to any breach, gross negligence or willful misconduct by pRx or its
employees or contractors, as applicable, in the performance under this Agreement. Monopar hereby  agrees to indemnify pRx and
hold pRx. harmless from and against all liabilities , losses. damages, expenses, charges and fees which pRx may sustain or incur
by reason of any claim which may be asserted against pRx by any person, firm, corporation or governmental unit and which may
arise out of  or  be  attributable  to  any  gross  negligence  or  willful  misconduct  by  Monopar  or  its  employees  or  contractors,  as
applicable, in the performance of this Agreement.

Warranties. The  Services  shall  be  performed  in  a  professional  manner,  consistent  with  industry  standards.  In  performing  the
Services, neither pR.x nor any of its employees shall make any unauthorized use of any confidential or proprietary information of
any other party or infringe the intellectual property rights of any other party.

Arbitration. Any  controversy  or  claim  between  Monopar  and  pRx  arising  out  of or  relating  to  this Agreement,  or  the  breach
thereof, shall be submitted to  arbitration  in  accordance  with  the  rules  of  the American Arbitration Association.  The  site of  the
arbitration shall be Chicago, IL, and except as provided herein the arbitration shall be conducted in accordance with the Rules of
the American Arbitration Association prevailing at the time the demand for arbitration is made hereunder. At least one member of
the arbitration panel shall be an expert knowledgeable in the area of biopharmaceutical clinical development. Judgment upon any
award rendered by the arbitrator(s) may be entered in any court of competent jurisdiction and shall be binding and final. The cost
of arbitration shall be borne by the losing Party, as determined by the arbitrator(s).

Confidential  Information.  pRx  has  executed  the  attached  confidential  disclosure  agreement  referenced  herein  as   Appendix A
prior to commencement of the Services. pRx hereby represents and warrants that the obligations thereunder shall be binding upon
it and its employees, and that it shall obtain written commitments from such employees thereto.

Inventions. pRx agrees that all ideas, developments,  suggestions and inventions which an  employee  or  other  parties  contracted
conceive  or  reduce  to  practice  arising  out  of  or  during  the  course  of  performance  under  this Agreement  shall  be  the  exclusive
property of Monopar and shall be promptly communicated and assigned to Monopar. pRx shall require any employees of or other
parties contracted by pRx to disclose the same to pRx and to be bound by the provisions of this paragraph. During the period of
this Agreement and thereafter at any reasonable time when called upon to do so by Monopar , pRx shall require any employees of
or  other  parties  contracted  by  pRx  to  execute  patent applications, assignments  to  Monopar  (or  any  designee  of  Monopar)  and
other papers and to perform acts which Monopar believes necessary to secure to Monopar full protection and ownership of the
rights in and to the services performed by pRx and/or for the preparation,

                                                                                                                                                                                        - 3 -

 
 
 
 
 
 
 
 
 
 
 
 
 
 
filing and prosecution of applications for patents  or  inventions  made  by any employees of or other  parties  contracted  by  pRx
hereunder. The decision to  file patent applications on inventions made by any employees of or other parties contracted by pRx
shall be made by Monopar and shall be for such countries as Monopar shall elect. Monopar agrees to bear  all  the  expense  in
connection with the preparation, filing and prosecution of applications for patents and for all matters provided in this paragraph
requiring the time and/or assistance of pRx as to such inventions.

12. 

Miscellaneous.

12.1 

Notice.  Any  notices  to  be  given  hereunder  by  either  Party  to  the  other  may  be  effectuated,  in  writing,  by  personal
delivery  or  by  mail,  registered  or  certified,  postage  prepaid,  with  return  receipt  requested.  Mailed  notices   shall  be
addressed to the parties at the following addresses:

If to Monopar:                                           Monopar Therapeutics Inc
                                                                   5 Revere Dr., Suite200
                                                                   Northbrook, IL, 60062
                                                                   Attention: Chandler Robinson, MD MBA MSc
                                                                   Email: #

If to pRx:                                                  pRx Consulting
                                                                    #
                                                                   Attention: Patrice Rioux, MD, PhD
                                                                   Email: #

or at such other addresses as either Monopar or pRx may designate by written notice to each other. Notices delivered personally shall be
deemed duly given on the date of actual receipt; mailed notices shall be deemed duly given as of the fourth day after the date so mailed.

12.2  Waiver  of  Breach.  The  waiver  by  either  Party  to  a  breach  of  any  provision  in  this Agreement  cannot  operate  or  be

construed as a waiver of any subsequent breach by either Party.

12.3 

Severability.  If  any  provision  of  this Agreement  is  determined  by  a  court  of  competent  jurisdiction  to  be  invalid  or
unenforceable, that provision shall be deemed modified to the extent necessary to make it valid or enforceable, or if it
cannot be so modified, then severed, and the remainder of the Agreement  shall continue in full force and effect as if the
Agreement had been signed with the invalid portion so modified or severed.

12.4 

Choice  of  Law.  This Agreement  has  been  made  and  entered  into  in  the  State  of  Illinois,  and  the  laws  of  such  state,
excluding its choice of law rules, shall govern the validity and interpretation of this Agreement and the performance due

                                                                                        - 4 -

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
hereunder. The losing party in any dispute hereunder shall pay the attorneys· fees and disbursements of the prevailing
party.

12.5 

Integration.  The  drafting,  execution  and  delivery  of  this  Agreement  by  the  Parties  have  been  induced  by  no
representations, statements, warranties or agreements other than those expressed herein. This Agreement embodies the
entire understanding of the Parties, and there are no further or other agreements  or  understandings,  written or oral,  in
effect between the Parties relating to the  subject matter hereof unless expressly referred to herein.

12.6  Modification.  This  Agreement  may  not  be  modified  unless  such  is  in  writing  and  signed  by  both  Parties  to  this

Agreement.

12.7 

Assignment. pRx shall not be permitted to assign this Agreement to any other person or entity without the prior written
consent  of  Monopar.  pRx  hereby  agrees  that  Monopar  shall  be  permitted  to  assign  this Agreement  to any  affiliate  of
Monopar. This Agreement shall be binding upon and shall inure to the benefit of the successors and permitted assigns of
the parties.

12.8 

Survival. The provisions of Sections 7, 8, 9, 10, and 11 shall survive expiration or termination of this Agreement for any
reason. Expiration or termination of this Agreement  shall not affect Monopar's obligations to pay any amounts that may
then be due to pRx.

IN WITNESS WHEREOF, the Parties hereto have executed this Agreement as of the day and  year first above written.

ACCEPTED AND AGREED TO:

PRx CONSULTING, LLC

    /s/ Patrice Rioux

BY: PATRICE RIOUX, MD, PhD

    ITS: PRESIDENT

MONOPAR THERAPEUTICS INC.

/s/ Chandler Robinson
BY:CHANDLER ROBINSON
ITS: CHIEF EXECUTIVE OFFICER

- 5 -

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
                                                        APPENDIX A

See executed CDA attached

- 6 -

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
EXECUTIVE EMPLOYMENT AGREEMENT

This Executive  Employment  Agreement  (the  "Agreement")  is  entered  into  as  of  October  4,  2017,  by  and  between
Kirsten Anderson ("Executive") and Monopar Therapeutics Inc. (the "Company").

Whereas, the Company desires to employ Executive as its Senior Vice P resident, Clinical Development effective as of
November 1, 2017 (the "Effective Date"), and Executive desires to  serve  in  such capacity,  pursuant  to  the  terms  and
conditions set forth in this Agreement; and

Now, Therefore, in consideration of the mutual promises  and  covenants  contained  herein,  it  is  hereby  agreed  by  and
between the parties hereto as follows:

ARTICLE I
DEFINITIONS

For purposes of the Agreement, the following terms are defined  as follows:

1.1.      "Board" means the Board of Directors of the Company.

1.2       "Cause" means any of the following events described below:

(a) Executive's commission of a felony or other crime involving moral turpitude;

(b) any willful act or acts of dishonesty undertaken by Executive and intended to result in substantial gain or
personal enrichment of Executive, Executive's family or any third party at the expense of the
Company;

(c)     any willful act of gross misconduct which is materially and demonstrably injurious to the Company;
and/or

(d)   Executive's inability to lawfully work in the United States.

For the purpose of this Agreement, no act, or failure to act, by Executive shall be considered " willful" if done, or omitted
to be  done,  by  her  in  good  faith  and  in  the  reasonable  belief  that  her  act  or  omission  was  in  the  best  interest  of  the
Company and/or required by applicable law.

1.3. "Change in Control" means the occurrence of any of the following events: (i) any sale or exchange of the capital
stock by the stockholders of the Company in one transaction or series of related transactions where more than fifty percent (50%) of the
outstanding

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
voting  power  of  the  Company  is  acquired  by  a  person  or  entity  or  group  of  related  persons  or  entities;  or  (ii)  any
reorganization,  consolidation  or  merger  of  the  Company  where  the  outstanding  voting  securities  of  the  Company
immediately before the transaction represent or are converted into less than fifty percent (50%) of  the outstanding voting
power of the surviving entity (or its parent corporation) immediately after the transaction; or (iii) the consummation of
any  transaction  or  series  of  related  transactions  that  results  in  the  sale  of  all  or  substantially  all  of  the  assets  of  the
Company; or (iv) any "person" or "group" (as defined in the Securities Exchange Act of 1934, as amended (the "Exchange
Act")  becoming  the  "beneficial  owner"  (as  defined  in  Rule  13d-3  under  the  Exchange  Act)  directly  or  indirectly  of
securities representing more than fifty percent (50%) of the voting power of the Company then outstanding. Except that
any change in the beneficial ownership of the securities of the Company as a result of a private financing of the Company
that is approved by the Board, shall not be deemed to be a Change in Control.

1.4.

"Change in Control Multiple" shall mean one-half (0.5).

1.5.          "Change in Control Period" means that period commencing on the  consummation of a Change in Control
and ending on the six month anniversary thereof.

1.6.       "COBRA" means the Consolidated Omnibus Budget Reconciliation Act of 1985, as amended.

1.7.

1.8.

"Code" means the Internal Revenue Code of 1986, as amended.

"Company" means Monopar Therapeutics Inc. or any successor thereto.

Executive and the Company.

1.9. 

"Confidential Disclosure Agreement" means the Confidential Disclosure Agreement entered into between

1.10.

"Covered Termination" means (a) an Involuntary Termination Without Cause or (b) a voluntary termination
for Good Reason, provided that the termination constitutes a Separation from Service.

1.11. "Good Reason" means Executive's resignation as a result of a Good Reason Condition. In order to resign for Good
Reason, Executive must provide written notice to the Company of the existence of the Good Reason Condition within thirty (30) days of
the initial existence of such Good  Reason  Condition.  Upon  receipt  of such notice  of  the  Good  Reason Condition, the  Company  will  be
provided with a period of thirty (30) days during which it may remedy the Good Reason Condition and not be required to provide for the
payments and benefits described in Section 4 as a result of such proposed resignation due to the Good Reason Condition specified in the
notice. If the Good Reason Condition is not remedied within the period specified  in the preceding sentence, Executive may resign for Good
Reason based on the Good Reason Condition specified in the notice, provided that

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
such resignation must occur within sixty (60) days after the initial existence of such Good Reason Condition.

consent:

1.12. "Good Reason Condition" means that any of the following are undertaken without Executive's express written

salary of at least a majority of the Company's executives of the same or greater percentage);

(a) 

    a material reduction in Executive's Base Salary (other than as part of a reduction in the base

(b)

(c)

a material diminution in Executive's responsibilities;

the Company's material breach of any material term of this Agreement; or

1.13. "Involuntary Termination Without Cause" means Executive's dismissal or discharge by the Company other

than for Cause. The termination of Executive's employment as a result of Executive' s death or inability to perform the essential functions
of her job due to disability will not be deemed to be an Involuntary Termination Without Cause.

from service" within the meaning of Treasury Regulation Section l.409A-l(h).

1.14. "Separation from Service" means Executive' s termination of employment or service constitutes a "separation

ARTICLE II
EMPLOYMENT BY THE COMPANY

2.1.  Position  and  Duties.  Subject  to  terms  set  forth  herein,  as  of  the  Effective  Date,  Executive  shall  serve  as  the
Company's Senior Vice President, Clinical Development and perform  such duties as are customarily associated with the position of  Senior
Vice President, Clinical Development as  well as any other duties as are assigned to Executive by either the Chief Scientific Officer or other
officer designated by the Chief Executive Officer. During the  term of Executive's employment with the Company,  Executive will devote
Executive's best efforts and substantially all of Executive's business time and attention (except for vacation periods and reasonable periods
of illness or other incapacities permitted by the Company' s general employment policies or as otherwise set forth in this Agreement) to the
business of the Company.

2.2. Employment at Will. Both the Company and Executive shall have the right to terminate Executive's employment
with  the  Company  at  any  time,  with  or  without  Cause,  and  without  prior  notice.  If  Executive's  employment  with  the  Company  is
terminated, Executive will be eligible lo receive severance benefits to the extent provided in this Agreement.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
2.3. Employment Policies. The employment relationship between the parties shall also be governed by the general

employment policies and practices of the Company, including those relating to protection of confidential information and assignment of
inventions, except that when the terms of this Agreement differ from or are in conflict with the Company' s general employment policies or
practices, this Agreement shall control.

ARTICLE III
COMPENSATION

3.1.      Base Salary. As of the Effective Date, Executive  shall  receive  for  services  to  be  rendered  hereunder  an  annual
base  salary  of  $260,000 ("Base Salary"),  payable  on  the  regular  payroll  dates  of  the  Company,  which  are  currently
bi-weekly, subject to increase in the sole discretion of the Board.

3.2     Sign-on Bonus. Executive shall be paid a one-time sign-on bonus of $25,000  (gross  before  taxes)  payable  with
Executive's first regular paycheck.

3.3. Annual Bonus. Executive is eligible for an annual bonus which is at the discretion of the Board.

3.4. Standard Company Benefits. Executive shall be entitled to all  rights  and  benefits  for  which Executive is  eligible
under the terms and conditions of the standard Company benefits and compensation practices that may be in effect from time to time and
are  provided  by  the  Company  to its  executive  employees  generally.  Executive  shall  be  entitled  each  year  to  four  (4)  weeks  leave  for
vacation at full pay, provided , that the maximum amount Executive may have accrued at any point in time is four (4) weeks (meaning that
once Executive has accrued four (4) weeks, Executive will not accrue any additional vacation time until she takes vacation and falls below
the four (4) week accrual cap). Executive shall also be entitled to reasonable holidays and illness days with full pay in accordance with the
policies  applicable  to  the  Company  and  its  affiliates  from  time  to  time  in  effect.  Employee  acknowledges  and  agrees  that  in  order  to
maintain flexibility, the Company and its affiliates have the right to amend or terminate any employee benefit plan at any time.

3.5. Stock Options. Subject to approval by the Board, Executive will be granted options to purchase up to 40,000 shares
of the Company's common stock with an exercise price per share as determined by the Compensation Committee or similar function of the
Board. Such options shall vest 6/48ths upon the six-month anniversary of grant date and l/48lh per month thereafter and shall expire ten
years from the grant date.

in connection with the Company's business, provided that

3.6. Expenses. The Company will reimburse Executive for all reasonable and necessary expenses incurred by Employee

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
such expenses incurred and are properly documented and accounted for in accordance with the policy of the Company and requirements of
the Internal Revenue Service.

ARTICLE IV
SEVERANCE AND CHANGE IN CONTROL BENEFITS

                       4.1.    Severance Benefits. Upon Executive's termination of employment Executive shall receive any accrued but unpaid
Base Salary and other accrued and unpaid compensation, including any Annual Bonus that has been earned with respect to a prior year, but
remains unpaid as of the date of the termination. If the termination is due to a Covered Termination or permanent disability, provided that
Executive first returns all Company property in her possession and, within sixty (60) days following the Covered Termina tion, executes
and does not revoke an effective general release of all claims against the Company and its affiliates in a form reasonably acceptable to the
Company (a "Release of Claims"), Executive shall also be entitled to receive the following severance benefits described in this Section
4.1.

(a) Covered Termination Not Related to a Change in Control. If Executive’s employment terminates
due to a Covered Termination which occurs outside of a Change in Control Period, Executive shall receive the following:

(i) An amount equal to three (3) months of Executive's Base Salary payable in substantially equal

installments in accordance with the Company's normal payroll policies, less applicable withholdings, with such
installments to commence as soon as administratively practicable following the date the Release of Claims is not subject to
revocation and, in any event, within sixty (60) days following the date of the Covered Termination.

(ii) If Executive elects to receive continued healthcare coverage pursuant to the provisions of COBRA,
the  Company  shall  directly  pay,  or  reimburse  Executive  for,  the  premium  for  Executive  and  Executive'  s  covered
dependents through the earlier of (i) the six month anniversary of the date of Executive's termination of employment and
(ii) the date Executive and Executive's covered dependents, if any, become eligible for healthcare coverage under another
employer's plan(s). Notwithstanding the foregoing, (i) if any plan pursuant to which such benefits are provided is not, or
ceases prior to the expiration of the period of continuation coverage to be, exempt from the application of Section 409A of
the Code under Treasury Regulation Section I .409 A- l(a)(S), or (ii) the Company is otherwise unable to continue to cover
Executive under its group health plans without penalty under applicable law (including without limitation, Section 2716 of
the Public Health Service Act), then, in either case, an amount equal to each remaining Company subsidy shall thereafter
be paid to Executive in substantially equal monthly installments. After the Company ceases to pay premiums pursuant to
this Section 4.l(a)(ii), Executive may, if  eligible, elect to continue healthcare coverage at Executive's expense in accordance
the provisions of COBRA.

                        (iii)  All of Employee's vested options or stock appreciation rights with respect to the Company
'  s  common  stock  shall  remain  exercisable  until  the  six  month  anniversary  of  Executive's  termination  of
employment (or, if earlier, the maximum period specified in the award documents and plans governing such
options or stock appreciation rights, as applicable, assuming Executive' s employment had not terminated).

to a Covered Termination that occurs during a Change in Control Period, Executive shall receive the following:

(b) Covered Termination Related to a Change in Control. If Executive's employment terminates due

(i) Executive shall be entitled to receive an amount equal to the Change in Control Multiplier multiplied

by the Executive's Base Salary, at the rate equal to the higher of (x) the rate in effect immediately prior to Executive's
termination of employment or (y) the rate in effect immediately prior to the Change in Control payable in a cash lump sum,
less applicable withholdings, as soon as administratively practicable following the date the Release of Claims is not subject
to revocation and, in any event, within sixty (60) days following the date of the Covered Termination.

(ii) If Executive elects to receive continued healthcare coverage pursuant to the provisions of COBRA,
the  Company  shall  directly  pay,  or  reimburse  Executive  for,  the  premium  for  Executive  and  Executive's  covered
dependents  through  the  earlier  of  (i)  the  date  that  is  that  number  of  years  equal  to  the  Change  in  Control  Multiplier
following  the  date  of  Executive's  termination  of  employment  and  (ii)  the  date  Executive  and  Executive'  s  covered
dependents,  if  any,  become  eligible  for  healthcare  coverage  wider  another  employer'  s  plan(s).  Notwithstanding  the
foregoing, (i) if any plan pursuant to which such benefits are provided is not, or ceases prior to the expiration of the period
of  continuation  coverage  to  be,  exempt  from  the  application  of  Section  409A  of  the  Code  under  Treasury  Regulation
Section l. 409A-l (a)(5), or (ii) the Company is otherwise unable to continue to cover Executive under its group health plans
without penalty under applicable law (including without limitation, Section 2716 of the Public Health Service Act), then, in

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
either case, an  amount  equal to  each  remaining  Company  subsidy  shall  thereafter  be  paid  to  Executive  in  substantially
equal monthly installments. After the Company ceases to pay p remiums pursuant to this Section 4.l (b)(ii), Executive may,
if eligible, elect to continue healthcare coverage at Executive's expense in accordance with the provisions of COBRA.

(iii) Each outstanding equity award, including, without limitation, each stock option and restricted stock
award, held by Executive shall automatically become vested and, if applicable, exercisable and any forfeiture restrictions or
rights of repurchase thereon shall immediately lapse, in each case, with respect to one hundred percent (100%) of the shares
subject thereto. To the extent vested after giving effect to the acceleration provided in the

 
 
 
preceding  sentence,  each  stock  option  held  by  Executive  shall  remain  exercisable  un  til  the  earlier  of  the
original expiration date for such stock option or the second anniversary of Executive's Covered Termination  .

(c)  Termination  for  Death  or  Disability.  If  Executive's  employment  is  terminated  due  to  death  or
permanent disability w here the Company makes a determination in good faith that, due to a mental or physical incapacity,
Executive has been unable to perform her duties under this Agreement for a period of not less than three (3) consecutive
months or 90 days in the aggregate in any 12-month period, Executive shall receive the following:

(i)  An  amount  equal  to  two  (2)  months  of  Executive's  Base  Salary  payable  in  substantially  equal
installments  in  accordance  with  the  Company'  s  normal  payroll  policies,  less  applicable  withholdings,  with  such
installments to commence as soon as administratively practicable following the date the Release of Claims is not subject to
revocation and, in any event, within sixty (60) days following the date of the Covered Termination.

(ii) If Executive (or in the event of death, her designee) elects to receive continued healthcare coverage
pursuant  to  the  provisions  of  COBRA,  the  Company  shall  directly  pay,  or  reimburse  Executive  for,  the  premium  for
Executive  and  Executive' s  covered  dependents  through  the  earlier  of  (i)  the  two  (2)  month  anniversary  of  the  date  of
Executive' s termination of employment and (ii) the date Executive and Executive's covered dependents, if  any,  become
eligible for healthcare coverage under another employer' s plan(s). Notwithstanding the foregoing, (i) if any plan pursuant
to which such benefits are provided is not, or ceases prior to the expiration of the period of continuation coverage to be,
exempt from the application of Section 409A of the Code under Treasury Regulation Section l. 409A-l (a)(5), or (ii) the
Company is otherwise unable to continue to cover Executive under its group health plans without penalty under applicable
law (including without limitation, Section 2716 of the Public Health Service Act), then, in either case , an amount equal to
each remaining Company subsidy shall thereafter be paid to Executive in substantially equal monthly installments. After
the  Company  ceases  to  pay  premiums  pursuant  to  this  Section  4.l  (b)(ii),  Executive  may,  if  eligible,  elect  to  continue
healthcare coverage at Executive's expense in accordance with the provisions of COBRA.

4.2. 280G Provisions. Notwithstanding anything in this Agreement to the contrary, if any payment or distribution
Executive would receive pursuant to this Agreement or otherwise ("Payment") would (a) constitute a "parachute payment" within the
meaning of Section 280G of the Code, and (b) but for this sentence, be subject to the excise tax imposed by Section 4999 of the Code
(the "Excise Tax"), then such Payment shall either be (i) delivered in full, or (ii) delivered as to such lesser extent which would result
in  no  portion  of  such  Payment  being  subject  to  the  Excise  Tax ,  whichever  of  the  foregoing  amounts,  taking  into  account  the
applicable federal, state and local income taxes and the Excise Tax , results in the receipt by Executive on an after-tax basis, of  the
largest payment, notwithstanding

 
 
 
 
 
 
 
 
 
 
 
 
 
 
that all or some portion of the Payment may be taxable under Section 4999 of the Code. The accounting firm  engaged by the Company for
general  audit  purposes  as  of  the  day  prior  to  the  effective  date  of  the  Change  in  Control  shall  perform  the  foregoing  calculations.  The
Company shall bear all expenses with respect to the determinations by such accounting firm required to be made hereunder. The accounting
firm shall provide its calculations to the Company and Executive within thirty (30) calendar days after the date on which Executive's right
to  a  Payment  is  triggered  (if  requested  at  that time by  the  Company  or  Executive)  or  such  other  time  as requested by  the  Company  or
Executive. Any good faith determinations of the accounting firm made hereunder shall be final, binding and conclusive upon the Company
and Executive. Any reduction in payments and/or benefits pursuant to this Section 4.2 will occur in the following order:  ( l) reduction of
cash payments; (2) cancellation of accelerated vesting of equity awards other than stock options; (3) cancellation of accelerated vesting of
stock options; and (4) reduction of other benefits payable to Executive.

4.3.

Section 409A.

(a)  Notwithstanding  any  provision  to  the  contrary  in  this  Agreement,  if  Executive  is  deemed  at  the  time  of  her
Separation from Service to be a "specified employee" for purposes of Section 409A(a)(2)(B)(i) of the Code, to the extent delayed
commencement of any portion of the benefits to which Executive is entitled under this Agreement is required in order to avoid a
prohibited  distribution  under  Section  409A(a)(2)(B)(i)  of  the  Code  which  would  subject  Executive  to  a  tax  obligation  under
Section 409A of the Code , such portion of Executive's benefits shall not be provided to Executive prior to the earlier of (i) the
expiration  of  the  six-  month  period  measured   from  the  date  of  the  Executive's  Separation  from  Service  or  (ii)  the  date  of
Executive's death. Upon the expiration of the applicable Code Section 409A(a)(2)(B)(i) period, all payments deferred pursuant to
this Section 4.3(a) shall be paid in a lump sum to Executive, and any remaining payments due under the Agreement shall be paid
as otherwise provided herein.

(b) Any reimbursements payable to Executive pursuant to the Agreement shall be paid  to Executive no later than 30
days  after  Executive  provides  the  Company  with  a  written  request  for  reimbursement,  and  to  the  extent  that  any  such
reimbursements are deemed to constitute " nonqualified deferred compensation" within the meaning of Section 409A of the Code
(i) such amounts shall be paid or reimbursed to Executive promptly, but in no event later than December 31 of the year following
the year in which the expense is incurred, (ii)  the amount of any such payments eligible for reimbursement in one year shall not
affect the payments or expenses that are eligible for payment or reimbursement in any other taxable year, and (iii)  Executive's
right to such payments or reimbursement shall not be subject to liquidation or exchange for any other benefit.

(c) For purposes of Section 409A of the  Code (including, without limitation, for purposes of Treasury Regulation

Section l. 409A-2(b)(2)(iii)), Executive's right to receive

 
 
 
 
 
 
 
 
 
 
 
 
 
installment payments under the Agreement shall be treated as a right to receive a series of separate payments and, accordingly,
each installment payment hereunder shall at all times be considered a separate and distinct payment.

4.4. Mitigation. Executive shall not be required to mitigate damages or the amount of any payment provided under this
Agreement by seeking other employmen t or otherwise, nor shall the amount of any payment provided for under this Agreement be reduced
by  any  compensation  earned  by  Executive  as  a  result  of  employment  by  another  employer  or  by  any  retirement  benefits  received  by
Executive after the date of the Covered Termination , or otherwise.

ARTICLE V
PROPRIETARY INFORMATION OBLIGATIONS

5.1. Agreement. Executive agrees to continue to abide by the Confidential Disclosure Agreement.

5.2. Remedies. Executive's duties under the Confidential Disclosure Agreement shall survive termination of Executive 's
employment with the Company  and  the  termination  of  this Agreement.  Executive  acknowledges  that  a  remedy  at  law  for  any breach  or
threatened breach by Executive of the provisions of the Confidential Disclosure Agreement , as well as Executive's obligations pursuant to
Section 6.2 and Article 7 below, would be inadequate, and Executive therefore agrees that the Company shall be entitled to seek injunctive
relief in case of any such breach or threatened breach.

ARTICLE VI
OUTSIDE ACTIVITIES

6.1. Other Activities.

(a) Executive shall not, during the term of this Agreement undertake or engage in any other employment,
occupation or business enterprise, other than ones in which  Executive  is a passive  investor,  unless  she  obtains  the  prior
written consent of the Board.

(b) Executive may engage in civic and not-for-profit activities so long as such activities do not materially
interfere  with  the  performance  of  Executive's  duties  hereunder .  In  addition,  Executive  shall  be  allowed  to  serve  as  a
member of the board of directors of up to two (2) other for profit entities at any time during the term of this Agreement,
which service shall not materially interfere with the performance of Executive's duties hereunder; provided, however, that
the Board, in its discretion, may require that Executive resign from one or both of such director positions if it determines
that such resignation(s) would be in the best interests of the Company.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
6.2.  Competition/Investments.  Executive  agrees  that,  from  the  date  hereof  until  a  period  of  twelve  (12)  months
following the date of  termination  of  Executive's  employment  with  the  Company,  Executive  w ill not directly  or  indirectly,  either  as  an
employee, employer, consultant, agent, principal, partner, corporate officer, director, or in any other individual or representative capacity,
engage or participate in any "Competitive Business" anywhere in the world. As used herein , a "Competitive Business" is defined as any
business developing uPAR  antibodies  to  treat  cancer, clonidine  to  treat  oral  mucositis,  non  cardiotoxic  forms  of  anthracyclines  to  treat
cancer,  or  any  other  drug  programs  which  are  deemed  by  Monopar,  at  that  point  in  time  in  the  future,  to  be  directly  competitive  to
Monopar' s drug programs in development at that point in time in the future.

ARTICLE VII
NONINTERFERENCE

In  addition  to  Executive's  obligations  under  the  Confidential  Disclosure Agreement  ,  Executive  shall  not  for  a  period  of  one  (I)  year
following Executive's termination of employment for any reason, either on Executive's own account or jointly with or as a manager, agent,
officer, employee, consultant, partner, joint venturer, owner or stockholder or otherwise on behalf of any other person, firm or corporation,
directly or indirectly solicit or attempt to solicit away from the Company any of its officers or employees or offer employment to any person
who is an officer or employee of the Company; provided, however, that a general  advertisement  to  which  an  employee of the  Company
responds shall in no event be deemed to result in a breach of this Article 7. Executive also agrees not to harass or disparage the Company or
its employees, clients, directors or agents or divert or attempt to divert any actual or potential business of the  Company. The provisions of
this Article 7 shall survive the termination or expiration of the applicable Executive' s Employment with the Company and shall be fully
enforceable thereafter. If it is determined by a court of competent jurisdiction in any state that any restriction in this Article 7 is excessive in
duration or scope or is unreasonable or unenforceable under the laws of that state, it is the intention of the parties that such restriction may
be modified or amended by the court to render it enforceable to the maximum extent permitted by the law of that state.

ARTICLE VIII
GENERAL PROVISIONS

8.1. Notices. Any notices provided hereunder must be in writing and will be given and will be deemed to have been duly
given (a) on the business day sent, when delivered by hand or facsimile transmission (with confirmation) during normal business hours, (b)
upon confirmation of receipt by recipient if sent by electronic mail, or (c) on the business day following the business day of sending, if
delivered by a nationally recognized overnight courier, in each case to the Company at  its primary office location and to Executive at

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Executive's address as listed on the Company payroll.

to deduction and withholding to the extent required by applicable law.

8.2. Tax Withholding. Executive acknowledges that all amounts and benefits payable under this Agreement are subject

8.3. Severability. Whenever  possible,  each  prov1s1on  of  this Agreement  will  be  interpreted  in  such  manner  as  to  be
effective and valid under applicable law, but if any provision of this Agreement  is held to be invalid, illegal or unenforceable in any respect
under any applicable law or rule in any jurisdiction, such invalidity, illegality or unenforceability will not affect any other provision or any
other  jurisdiction,  but  this  Agreement  will  be  reformed,  construed  and  enforced  in  such  jurisdiction  as  if  such  invalid,  illegal  or
unenforceable provisions had never been contained herein.

deemed to have waived any preceding or succeeding breach of the same or any other provision of this Agreement.

8.4. Waiver. If either party should waive any breach of any provisions of this Agreement, they shall not thereby be

8.5. Complete Agreement. This Agreement constitutes the entire agreement between Executive and the Company and is
the  complete,  final,  and  exclusive  embodiment  of  their  agreement  with  regard  to  this  subject  matter,  and  will  supersede  all  prior
agreements, understandings, discussions, negotiations and undertakings, whether written  or  oral, between  the  parties  with  respect  to  the
subject matter hereof, including without limitation, the Prior Agreement. This Agreement is entered into without reliance on any promise or
representation oilier than those expressly contained herein or therein, and cannot be modified or amended except in a writing signed by an
officer of the Company and Executive.

signatures of more than one party, but all of which taken together will constitute one and the same Agreement.

8.6.  Counterparts.  This  Agreement  may  be  executed  in  separate  counterparts,  any  one  of  which  need  not  contain

constitute a part hereof nor to affect the meaning thereof.

8.7. Headings. The headings of the sections  hereof are inserted for convenience only and shall not be deemed to

8.8. Successors  and Assigns.  This Agreement  is  intended  to  bind  and  inure  to  the  benefit  of  and  be  enforceable  by
Executive and the Company, and  their respective successors, assigns, heirs, executors and administrators, except that Executive may not
assign her rights or delegate her duties or obligations hereunder without the prior written consent of the Company.

8.9.     Arbitration. Unless otherwise prohibited by law or specified below, all disputes,

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
claims  and  causes  of  action,  in  law  or  equity,  arising  from  or  relating  to  this Agreement  or  its  enforcement,  performance,  breach,  or
interpretation shall be resolved solely and exclusively by final and binding arbitration held in Illinois in conformity with the then existing
employment arbitration rules and Illinois law. The arbitrator shall: (a) provide adequate discovery for the resolution of the dispute; and (b)
issue a written arbitration decision, to include the arbitrator's essential findings and conclusions  and  a  statement  of  the award.  However,
nothing in this section is intended to prevent either party from obtaining injunctive relief in court to prevent irreparable harm pending the
conclusion of any such arbitration. The arbitrator shall determine who shall bear the costs of any such arbitration.

8.10. Executive Acknowledgement. Executive acknowledges that (a) she has consulted with or has had the opportunity to
consult with independent counsel of her own choice concerning this Agreement, and has been advised to do so by the Company, and (b)
that  she  has  read  and  understands  the Agreement,  is  fully  aware  of  its  legal  effect,  and  bas  entered  into  it  freely  based  on  her  own
judgment.

governed by the law of the State of Illinois without regard to the conflicts of law provisions thereo£

8.11. Choice of Law. All questions concerning the construction, validity and interpretation of this Agreement will be

In Witness Whereof, the parties have executed this Agreement as of the date first written above.

On behalf of Monopar Therapeutics Inc.

                             /s/ Chandler D. Robinson

Chandler D. Robinson, MD MBA MSc
Chief Executive Officer

Accepted and Agreed

                            /s/ Kirsten Anderson                                                                             October 6, 2017
                            Kirsten Anderson

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
CONSULTING AGREEMENT

This Consulting Agreement (herein referred to as “Agreement”) is made and entered into on December 8, 2017, effective as of
January  1,  2018  (the  “Effective Date”),  by  and  between  Monopar  Therapeutics,  Inc.  (herein  referred  to  as  “Monopar”),  a  Delaware
corporation, located at 5 Revere Dr., Suite 200, Northbrook, IL 60062, and pRx Consulting, LLC (herein referred to as pRx), a Delaware
corporation located at # (each herein referred to as “Party” and collectively as “Parties”).

RECITALS

WHEREAS, pRx specializes in the field of clinical development, including but not limited  to:  clinical  trial  design,  statistical

modeling, clinical operations, regulatory strategy, investor due diligence, and the duties of a Chief Medical Officer.

WHEREAS, Monopar desires to contract with pRx to provide certain consultation services as requested by Monopar, and pRx

wishes to provide such services to Monopar, upon the terms and conditions set forth below.

NOW, THEREFORE, in consideration of the premises and mutual covenants contained herein, the Parties agree as follows:

1. 

2. 

Consulting Arrangement. pRx agrees to perform consulting services as described herein upon the terms and conditions herein set
forth.

Term of Agreement. Subject to the provision for early termination set forth below in Section 5 of this Agreement, this Agreement
shall  commence  as  of  the  Effective  Date  and  shall  continue  for  a  period  of  twelve  (12)  months  from  the  Effective  Date  (the
“Term”). Either Party may terminate this Agreement without cause with 10-days’ prior written notice.

3. 

Duties of pRx.

3.1 

3.2 

Specific Duties. pRx shall provide consulting services to Monopar, such duties to include the general duties of a Chief
Medical Officer, clinical trial design, statistical modeling, clinical operations oversight, regulatory strategy, and investor
due diligence, with such other specific requirements as Monopar may specify from time to time during the Term (herein
referred to as the “Services”).

pRx’s Obligations. The president of pRx, Dr. P. Rioux, shall spend on the average over the course of the Term one-and-
a-half  (1.5)  work  days  per  week  working  on  Monopar  matters,  be  diligent  in  the  performance  of  Services,  and  be
professional in its commitment to meeting its obligations hereunder. pRx represents and warrants that pRx is not party to
any other existing agreement, which any of them would prevent pRx from entering into this Agreement or which would
adversely affect this Agreement. pRx shall not perform Services for any other individuals or entities in direct competition
with Monopar, except as provided for by mutual written agreement of the Parties. pRx shall not perform services for any
party

- 1 -

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
which would require or facilitate the unauthorized disclosure of any confidential or proprietary information of
Monopar.

3.3 

Reporting.  pRx  will  report  to  and  liaise  with Andrew  P.  Mazar,  Ph.D.,  Chandler  Robinson,  M.D.,  and/or  any  other
assigned Monopar employee or consultant as may be designated in writing by Monopar.

3.4 

Compensation. Monopar shall pay pRx as follows:

a.            Four thousand dollars ($4,000) per month payable within thirty (30) days of the end of each month.

b.           

 Dr. P. Rioux, president of pRx Consulting, LLC shall be granted stock options to purchase up to 32,004
shares of Monopar’s common stock at an exercise price of $6.00. Such stock option shall vest as follows: on January 1, 2018,
options  to  purchase  up  to  12,000  shares;  and  options  to  purchase  up  to  1,667  shares  on  the  1st  of  each  subsequent  month
thereafter. Such vesting shall terminate upon the termination of this Agreement. The number of shares, the exercise price thereof
and the rights granted under this Agreement are subject to adjustment and modification as provided in the Monopar Therapeutics
Inc. 2016 Stock Incentive Plan.

pRx shall not be reimbursed, and is responsible for the facilities and equipment necessary to perform Services required under this
Agreement.

4. 

5. 

6. 

Reimbursement of Other Expenses. So long as Monopar’s prior approval has been obtained, Monopar shall promptly reimburse
pRx for all direct expenses incurred in providing the Services to Monopar pursuant to this Agreement, including travel, meals and
lodging. The invoice submitted by pRx pursuant to this Section 4 shall also include a detail of all reimbursable expenses incurred
during the period covered by such invoice.

Termination of Agreement - Failure to perform. In the event that pRx ceases to perform the Services or breaches its obligations as
required hereunder for any reason, Monopar shall have the right to immediately terminate this Agreement upon notice to pRx and
to enforce such other rights and remedies as it may have as a result of said breach.

Certain Liabilities.  It  is  understood  and  agreed  that  pRx  shall  be  acting  as  an  independent  contractor  and  not  as  an  agent  or
employee of, or partner, joint venturer or in any other relationship with Monopar. pRx will be solely responsible for all insurance,
employment taxes, FICA taxes and all obligations to governments or other organizations for it and its employees arising out of
this  consulting  assignment.  pRx  acknowledges  that  no  income,  social  security  or  other  taxes  shall  be  withheld  or  accrued  by
Monopar for pRx’s or its employees’ benefit. pRx assumes all risks and hazards encountered in the performance of duties by it or
its employees under this Agreement. Unless Monopar has provided prior written approval, pRx shall not use any sub-contractors
to perform pRx’s obligations hereunder. pRx shall be solely responsible for any and all injuries, including death, to all persons
and any and all loss or damage to property, which may result from performance under this Agreement.

- 2 -

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
7.

8. 

9. 

10. 

11. 

Indemnities. pRx hereby agrees to indemnify Monopar and hold Monopar harmless from and against all claims (whether asserted
by  a  person,  firm,  entity  or  governmental  unit  or  otherwise),  liabilities,  losses,  damages,  expenses,  charges  and  fees  which
Monopar may sustain or incur arising out of or attributable to any breach, gross negligence or willful misconduct by pRx or its
employees or contractors, as applicable, in the performance under this Agreement. Monopar hereby agrees to indemnify pRx and
hold pRx harmless from and against all liabilities, losses, damages, expenses, charges and fees which pRx may sustain or incur by
reason of any claim which may be asserted against pRx by any person, firm, corporation or governmental unit and which may
arise  out  of  or  be  attributable  to  any  gross  negligence  or  willful  misconduct  by  Monopar  or  its  employees  or  contractors,  as
applicable, in the performance of this Agreement.

Warranties.  The  Services  shall  be  performed  in  a  professional  manner,  consistent  with  industry  standards.  In  performing  the
Services, neither pRx nor any of its employees shall make any unauthorized use of any confidential or proprietary information of
any other party or infringe the intellectual property rights of any other party.

Arbitration. Any  controversy  or  claim  between  Monopar  and  pRx  arising  out  of  or  relating  to  this Agreement,  or  the  breach
thereof,  shall  be  submitted  to  arbitration  in  accordance  with  the  rules  of  the American Arbitration Association.  The  site  of  the
arbitration shall be Chicago, IL, and except as provided herein the arbitration shall be conducted in accordance with the Rules of
the American Arbitration Association prevailing at the time the demand for arbitration is made hereunder. At least one member of
the arbitration panel shall be an expert knowledgeable in the area of biopharmaceutical clinical development. Judgment upon any
award rendered by the arbitrator(s) may be entered in any court of competent jurisdiction and shall be binding and final. The cost
of arbitration shall be borne by the losing Party, as determined by the arbitrator(s).

Confidential Information.  pRx  has  executed  the  attached  confidential  disclosure  agreement  referenced  herein  as  Appendix A
prior to commencement of the Services. pRx hereby represents and warrants that the obligations thereunder shall be binding upon
it and its employees, and that it shall obtain written commitments from such employees thereto.

Inventions.  pRx  agrees  that  all  ideas,  developments,  suggestions  and  inventions  which  an  employee  or  other  parties  contracted
conceive  or  reduce  to  practice  arising  out  of  or  during  the  course  of  performance  under  this Agreement  shall  be  the  exclusive
property of Monopar and shall be promptly communicated and assigned to Monopar. pRx shall require any employees of or other
parties contracted by pRx to disclose the same to pRx and to be bound by the provisions of this paragraph. During the period of
this Agreement and thereafter at any reasonable time when called upon to do so by Monopar, pRx shall require any employees of
or  other  parties  contracted  by  pRx  to  execute  patent  applications,  assignments  to  Monopar  (or  any  designee  of  Monopar  )  and
other papers and to perform acts which Monopar believes necessary to secure to Monopar full protection and ownership of the
rights  in  and  to  the  services  performed  by  pRx  and/or  for  the  preparation,  filing  and  prosecution  of  applications  for  patents  or
inventions made by any employees of or other parties contracted by pRx hereunder. The decision to file patent applications on
inventions made by any employees of or other parties contracted by pRx shall be made by

- 3 -

 
 
 
 
 
 
 
 
 
 
 
 
Monopar and shall be for such countries as Monopar shall elect. Monopar agrees to bear all the expense in connection with the
preparation, filing and prosecution of applications for patents and for all matters provided in this paragraph requiring the time
and/or assistance of pRx as to such inventions.

12. 

Miscellaneous.

12.1 

Notice. Any  notices  to  be  given  hereunder  by  either  Party  to  the  other  may  be  effectuated,  in  writing,  by  personal
delivery or by mail, registered or certified, postage prepaid, with return receipt requested, or by electronic mail. Mailed
notices shall be addressed to the Parties at the following addresses:

If to Monopar:  

Monopar Therapeutics Inc.

5 Revere Dr., Suite 200
Northbrook, IL, 60062
Attention: Chandler Robinson, MD MBA MSc
Email: #

If to pRx:   pRx Consulting, LLC
                   #

Attention: Patrice Rioux, MD, PhD
Email: #

or at such other addresses as either Monopar or pRx may designate by written notice to each other. Notices delivered
personally shall be deemed duly given on the date of actual receipt; mailed notices shall be deemed duly given as of
the fourth day after the date so mailed. If sent by electronic mail, such notice will be deemed given upon confirmation
of receipt by recipient.

12.2  Waiver  of  Breach.  The  waiver  by  either  Party  to  a  breach  of  any  provision  in  this Agreement  cannot  operate  or  be

construed as a waiver of any subsequent breach by either Party.

12.3 

Severability.  If  any  provision  of  this Agreement  is  determined  by  a  court  of  competent  jurisdiction  to  be  invalid  or
unenforceable, that provision shall be deemed modified to the extent necessary to make it valid or enforceable, or if it
cannot be so modified, then severed, and the remainder of the Agreement shall continue in full force and effect as if the
Agreement had been signed with the invalid portion so modified or severed.

12.4 

Choice  of  Law.  This Agreement  has  been  made  and  entered  into  in  the  State  of  Illinois,  and  the  laws  of  such  state,
excluding its choice of law rules, shall govern the validity and interpretation of this Agreement and the performance due

- 4 -

 
 
 
 
 
 
 
 
                                           
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
hereunder. The losing party in any dispute hereunder shall pay the attorneys' fees and disbursements of the prevailing
party.

12.5 

integration.  The  drafting,  execution  and  delivery  of  this  Agreement  by  the  Parties  have  been  induced  by  no
representations, statements, warranties or agreements other than those expressed herein. This Agreement embodies the
entire  understanding  of  the  Parties,  and  there  are  no  further  or  other  agreements  or  understandings,  written  or  oral,  in
effect between the Parties relating to the subject matter hereof unless expressly referred to herein.

12.6  Modification.  This  Agreement  may  not  be  modified  unless  such  is  in  writing  and  signed  by  both  Parties  to  this

Agreement.

12.7 

12.8 

Assignment. pRx shall not be permitted to assign this Agreement to any other person or entity without the prior written
consent of Monopar. pRx hereby agrees that Monopar shall be permitted to assign this Agreement to any affiliate of
Monopar. This Agreement shall be binding upon and shall inure to the benefit of the successors and permitted assigns
of the parties.

Survival. The provisions of Sections 7, 8, 9, 10, and 11 shall survive expiration or termination of this Agreement for
any reason. Expiration or termination of this Agreement shall not affect Monopar's obligations to pay any amounts that
may then be due to pRx.

IN WITNESS WHEREOF, the Parties hereto have executed this Agreement as of the day and year first above written.

  ACCEPTED AND AGREED TO:

  pRx Consulting LLC                                                                                    Monopar Therapeutics Inc.

  /s/ Patrice Rioux                                                                                        /s/ Chandler Robinson

  BY: PATRICE RIOUX. MD, PHD                                                             BY: CHANDLER ROBINSON
  ITS: PRESIDENT                                                                                       ITS: CHIEF EXECUTIVE OFFICER

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
  
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
                 
 
 
 
 
 
 
 
 
 
 
 
APPENDIX A

See executed CDA attached

- 6 -

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
First Amendment  to  Employment Agreement  between  Kim  R.  Tsuchimoto  (“Executive”)  and
Monopar Therapeutics Inc. (“Company”) dated November 1, 2017. The following amendments
are made effective March 1, 2018. All other unrevised sections remain in full force.

2.1  Position  and  Duties ,  Executive  will  devote  Executive’s  best  efforts  and  50%  of  Executive’s
business  time  and  attention  (except  for  vacation  periods  and  reasonable  periods  of  illness  or  other
incapacities permitted by the Company’s general employment policies or as otherwise set forth in this
Agreement) to the business of the Company.

3.1 Base Salary , Executive shall receive for services to be rendered hereunder an annual base salary of
$137,500 representing 50% of full-time.

3.3 Standard Company Benefits , Executive shall be entitled to all benefits offered by the Company
so long as Executive devotes 50% or more time to the business of the Company. In lieu of benefits,
Executive shall be reimbursed up to $1,800 per month for out-of-pocket expenses for medical, dental
and vision benefits until such time the Company has benefit plans in place. Based upon 50% service,
Executive shall be entitled each year to two (2) weeks leave for vacation at full pay, provided, that the
maximum  amount  Executive  may  have  accrued  at  any  point  in  time  is  two  (2)  weeks  (meaning  that
once Executive has accrued two (2) weeks, Executive will not accrue any additional vacation time until
she takes vacation and falls below the two (2) week accrual cap).

Pursuant to section  6.1(a) Other Activities, Exhibit A

25%  of  full-time  employment  with  no  benefits  at  Mercaptor  Discoveries  Inc.  as  Chief  Financial
Officer, Secretary, Treasurer and Co-Founder

Minimal  time,  as  needed,  at  DNAcheckup  as  a  volunteer  Chief  Financial  Officer,  Secretary  and
Treasurer

Requested by:

/s/ Kim R. Tsuchimoto

Kim R.
Tsuchimoto                                                                            

Date

February 26, 2018

Approved by:

/s/ Chandler D. Robinson

March 1, 2018

Chandler D.
Robinson                                                                            
Monopar Therapeutics Inc.

Date

Co-Founder, Chief Executive Officer and Director

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
                                                                          
 
 
 
Chandler Robinson Chief Executive Officer
Monopar Therapeutics LLC 598 Rockefeller Road
Lake Forest, IL USA 60045

2ist March 2018

Dear Chandler,

Cancer Research UK

Angel Building 407 St John Street London EClV 4AD United Kingdom

020 7242 0200

cruk.org

Clinical Tri.al and Option Agreement between Monopar Therapeutics LLC, Cancer Research UK and Cancer Research Technology
Limited dated 15th May 2015 ("the Agreement")

As part of a recent portfolio reprioritisation, Cancer Research UK and Cancer Research Technology have decided to close the project
Which is the subject of the Agreement. We will be working with Monopar Therapeutics over the coming months to formalise the
arrangements necessary to effect termination of the Agreement.

Yours faithfully,

 /s/ Nigel Blackburn
Nigel Blackburn

Director of Drug Development CRUK Centre for Drug Development

 
 
 
 
 
 
 
 
 
          
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Patron Her Majesty The Queen

Presidents HRH The Duke of Gloucester KG GCVO and HRH Princess Alexandra, the Hon Lady Ogilvy KG
GCVO Chief Executive Sir Harpal S Kumar
Regist ered Charity in England and Wales (1089464), Scotland (SC041666) and the Isle of Man (1103)

Regi stered Company limited by guarantee in England and Wales (4325234) and registered rn the Isle of Man
(5713F) Registered Address Angel Building, 407 St John Street, London EC1V· 4AD

 
 
 
 
 
 
 
Exhibit 11

Statement Regarding Computation of Per Share Earnings

The statement regarding computation of per share earnings is set forth in Note 2 of the Notes to the Financial Statements of the

Company for the years ended December 31, 2017 and 2016.

 
 
 
 
MONOPAR THERAPEUTICS INC.

CODE OF BUSINESS CONDUCT AND ETHICS

Introduction

Monopar Therapeutics Inc. and its subsidiaries (the “Company”) are committed to maintaining the highest standards of business conduct
and ethics. This Code of Business Conduct and Ethics (the “Code”) reflects the business practices and principles of behavior that support
this commitment. We expect every employee, officer and non-employee director to read and understand this Code and its application to
the  performance  of  his  or  her  business  responsibilities.  References  in  this  Code  to  employees  are  intended  to  cover  staff,  supervisors,
managers, officers and, as applicable, non-employee directors.

Officers, managers and other supervisors are expected to develop in staff a sense of commitment to the spirit, as well as the letter, of this
Code. Supervisors are also expected to ensure that all agents and contractors conform to Code standards when working for or on behalf of
the  Company.  The  compliance  environment  within  each  supervisor’s  assigned  area  of  responsibility  will  be  a  factor  in  evaluating  the
quality of that individual’s performance. In addition, any employee who makes an exemplary effort to implement and uphold our legal
and  ethical  standards  will  be  recognized  for  that  effort  in  his  or  her  performance  review.  Nothing  in  this  Code  alters  the  at-will
employment policy of the Company.

This  Code  addresses  conduct  that  is  particularly  important  to  proper  dealings  with  the  people  and  entities  with  whom  we  interact,  but
reflects only a part of our commitment. From time to time we may adopt additional policies and procedures with which our employees,
officers and non-employee directors are expected to comply, if applicable to them. However, it is the responsibility of each employee to
apply  common  sense,  together  with  his  or  her  own  highest  personal  ethical  standards,  in  making  business  decisions  where  there  is  no
stated guideline in this Code.

Action by members of your immediate family, significant others or other persons who live in your household (referred to in this Code as
“family  members”)  also  may  potentially  result  in  ethical  issues  to  the  extent  that  they  involve  the  Company’s  business.  For  example,
acceptance of inappropriate gifts by a family member from one of our suppliers could create a conflict of interest and result in a Code
violation attributable to you. Consequently, in complying with this Code, you should consider not only your own conduct, but also that of
your immediate family members, significant others and other persons who live in your household.

YOU  SHOULD  NOT  HESITATE  TO  ASK  QUESTIONS  ABOUT  WHETHER  ANY  CONDUCT  MAY  VIOLATE  THIS  CODE,
VOICE  CONCERNS  OR  CLARIFY  GRAY  AREAS.  SECTION  20  BELOW  DETAILS  THE  COMPLIANCE  RESOURCES
AVAILABLE TO YOU. IN ADDITION, YOU SHOULD BE ALERT TO POSSIBLE VIOLATIONS OF THIS CODE BY OTHERS
AND REPORT SUSPECTED VIOLATIONS, WITHOUT FEAR OF ANY FORM OF RETALIATION, AS FURTHER DESCRIBED
IN SECTION 20. Violations of this Code will not be tolerated. Any employee who violates the standards in this Code may be subject to
disciplinary  action,  which,  depending  on  the  nature  of  the  violation  and  the  history  of  the  employee,  may  range  from  a  warning  or
reprimand to and including termination of employment and, in appropriate cases, civil legal action or referral for regulatory or criminal
prosecution.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
1.

Honest and Ethical Conduct

It is the policy of the Company to promote high standards of integrity by conducting our affairs in an honest and  ethical  manner.  The
integrity and reputation of the Company depends on the honesty, fairness and integrity brought to the job by each person associated with
us. Unyielding personal integrity is the foundation of corporate integrity.

2.

Legal Compliance

Obeying the law, both in letter and in spirit, is the foundation of this Code. Our success depends upon each employee’s operating within
legal  guidelines  and  cooperating  with  local,  national  and  international  authorities.  We  expect  employees  to  understand  the  legal  and
regulatory requirements applicable to their business units and areas of responsibility. We hold periodic training sessions to ensure that all
employees  comply  with  the  relevant  laws,  rules  and  regulations  associated  with  their  employment,  including  laws  prohibiting  insider
trading (which are discussed in further detail in Section 3 below). While we do not expect you to memorize every detail of these laws,
rules and regulations, we want you to be able to determine when to seek advice from others. If you do have a question in the area of legal
compliance, it is important that you not hesitate to seek answers from your supervisor or the Compliance Officer (as further described in
Section 20).

Disregard of the law will not be tolerated. Violation of domestic or foreign laws, rules and regulations may subject an individual, as well
as the Company, to civil and/or criminal penalties. You should be aware that conduct and records, including emails, are subject to internal
and external audits and to discovery by third parties in the event of a government investigation or civil litigation. It is in everyone’s best
interests to know and comply with our legal obligations.

3.

Insider Trading

Employees who have access to confidential (or “inside”) information are not permitted to use or share that information for stock trading
purposes or for any other purpose except to conduct our business. All non- public information about the Company or about companies
with which we do business is considered confidential information. To use material non-public information in connection with buying or
selling  securities,  including  “tipping”  others  who  might  make  an  investment  decision  on  the  basis  of  this  information,  is  not  only
unethical, it is illegal. Employees must exercise the utmost care when handling material inside information.

4.

International Business Laws

Our employees are expected to comply with the applicable laws in all countries to which they travel, in which they operate and where we
otherwise do business, including laws prohibiting bribery, corruption or the conduct of business with specified individuals, companies or
countries. The fact that, in some countries, certain laws are not enforced or that violation of those laws is not subject to public criticism
will not be accepted as an excuse for noncompliance. In addition, we expect employees to comply with U.S. laws, rules and regulations
governing the conduct of business by its citizens and corporations outside the U.S.

These U.S. laws and regulations, which extend to all our activities outside the U.S., include:

●

●

The Foreign Corrupt Practices Act, which prohibits directly or indirectly giving anything of value to a government official to obtain
or retain business or favorable treatment and requires the maintenance of accurate books of account, with all company transactions
being properly recorded;

U.S.  Embargoes,  which  generally  prohibit  U.S.  companies,  their  subsidiaries  and  their  employees  from  doing  business  with
countries, or traveling to, subject to sanctions imposed by the U.S. government (including, for example, Belarus, Cuba, Eritrea, Iran,
North Korea, Syria and Venezuela), as well as specific companies and individuals identified on lists published by the U.S. Treasury
Department;

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
●

●

U.S. Export Controls, which restrict exports from the U.S. and re-exports from other countries of goods, software and technology to
many countries, and prohibits transfers of U.S.-origin items to denied persons and entities; and

Anti-boycott Regulations, which prohibit U.S. companies from taking any action that has the effect of furthering or supporting a
restrictive trade practice or boycott imposed by a foreign country against a country friendly to the U.S. or against any U.S. person.

If you have a question as to whether an activity is restricted or prohibited, seek assistance before taking any action, including giving any
verbal assurances that might be regulated by international laws.

5.

Antitrust

Antitrust laws are designed to protect the competitive process. These laws are based on the premise that the public interest is best served
by vigorous competition and will suffer from illegal agreements or collusion among competitors. Antitrust laws generally prohibit:

●

●

●

agreements,  formal  or  informal,  with  competitors  that  harm  competition  or  customers,  including  price  fixing  and  allocations  of
customers, territories or contracts;

agreements, formal or informal, that establish or fix the price at which a customer may resell a product; and

the acquisition or maintenance of a monopoly or attempted monopoly through anti-competitive conduct.

Certain  kinds  of  information,  such  as  pricing,  production  and  inventory,  should  not  be  exchanged  with  competitors,  regardless  of  how
innocent  or  casual  the  exchange  may  be  and  regardless  of  the  setting,  whether  business  or  social. In addition,  the  U.S.  Federal  Trade
Commission Act declares "unfair methods of competition in commerce, and unfair or deceptive acts or practices in commerce" unlawful.
It is a violation of that Act to engage in deceptive, unfair or unethical practices and to make misrepresentations in connection with sales
activities.

Antitrust  laws  impose  severe  penalties  for  certain  types  of  violations,  including  criminal  penalties  and  potential  fines  and  damages  of
millions of dollars, which may be tripled under certain circumstances. Understanding the requirements of antitrust and unfair competition
laws of the various jurisdictions where we do business can be difficult, and you are urged to seek assistance from your supervisor or the
Compliance Officer whenever you have a question relating to these laws.

6.

Environmental Compliance

Federal law imposes criminal liability on any person or company that contaminates the environment with any hazardous substance that
could cause injury to the community or environment. Violation of environmental laws can involve monetary fines and imprisonment. We
expect employees to comply with all applicable environmental laws.

It is our policy to conduct our business in an environmentally responsible way that minimizes environmental impacts. We are committed
to minimizing and, if practicable, eliminating the use of any substance or material that may cause environmental damage, reducing waste
generation  and  disposing  of  all  waste  through  safe  and  responsible  methods,  minimizing  environmental  risks  by  employing  safe
technologies and operating procedures, and being prepared to respond appropriately to accidents and emergencies.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
7.

Workplace

We are committed to the following:

●

●

●

●

●

Providing a safe, violence-free workplace. Violent or threatening behavior is strictly prohibited by anyone on Company premises or
engaged in a Company-related activity. This behavior includes, but is not limited to, threats of any kind; intimidating or physically
aggressive actions; excessive arguing or swearing; defacing Company property; sabotage; demonstrated pattern of refusing to follow
Company policies; and possession of weapons or firearms on Company premises. All reports of workplace violence will be taken
with the upmost seriousness and will be investigated promptly and thoroughly.

Providing a workplace that is free from unlawful harassment, bullying and discrimination. Harassment is unwelcome conduct that is
based on race, color, sex, pregnancy, age, national origin, religion, disability, genetic information, sexual orientation, veteran status,
gender reassignment or other classes protected by applicable law. We will not tolerate  conduct that is severe or pervasive enough to
create  a  work  environment  that  a  reasonable  person  would  consider  intimidating,  hostile,  or  abusive.  No  employee  will  be
disadvantaged for reporting this type of conduct in good faith to Human Resources or the Compliance Officer.

Providing an environment free from combative, verbally abusive or disrespectful behavior. These behaviors can create a climate of
fear,  hostility,  distraction  and  unproductivity.  Such  incidents  should  be  reported  to  your  Supervisor  or  to  Human  Resources. All
reports will be investigated thoroughly and, if found to be valid, may lead to disciplinary action including termination.

Providing equal employment opportunity for all applicants and employees. We do not discriminate on any basis prohibited under
federal, state or local law. This applies to all areas of employment, including recruitment, hiring, training, promotion, compensation,
benefits, transfer, disciplinary action, and social and recreational programs.

Creating a fully inclusive and stimulating environment in which our workforce is free to innovate to meet the needs of our customers
around  the  world.  We  respect  employment  laws  wherever  we  operate  in  the  world,  including  international  labor  standards,  laws
governing freedom of expression and rights of association, privacy and equal opportunities.

8.

Conflicts of Interest

We respect the rights of our employees to manage their personal affairs and investments and do not wish to impinge on their personal
lives. At the same time, employees should avoid conflicts of interest that occur when their personal interests may interfere in any way
with the performance of their duties or the best interests of the Company. A conflicting personal interest could result from an expectation
of personal gain now or in the future or from a need to satisfy a prior or concurrent personal obligation. We expect our employees to be
free  from  influences  that  conflict  with  the  best  interests  of  the  Company  or  might  deprive  the  Company  of  their  undivided  loyalty  in
business  dealings.  Even  the  appearance  of  a  conflict  of  interest  where  none  actually  exists  can  be  damaging  and  should  be  avoided.
Whether or not a conflict of interest exists or will exist can be unclear. Conflicts of interest are prohibited unless specifically authorized as
described below.

If you have any questions about a potential conflict or if you become aware of an actual or potential conflict, and you are not an officer or
director of the Company, you should discuss the matter with your supervisor or the Compliance Officer. Supervisors may not authorize
conflict of interest matters or make determinations as to whether a problematic conflict of interest exists without first seeking the approval
of the Compliance Officer and providing the Compliance Officer with a written description of the activity. If the supervisor is involved in
the  potential  or  actual  conflict,  you  should  discuss  the  matter  directly  with  the  Compliance  Officer.  Officers  and  directors  may  seek
authorizations and determinations from the Audit Committee of the Board of Directors.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Factors that may be considered in evaluating a potential conflict of interest are, among others:

●
●

●

●

●

●
●

●

●

whether it may interfere with the employee’s job performance, responsibilities or morale;
whether the employee has access to confidential information;

whether it may interfere with the job performance, responsibilities or morale of others within the organization;

any potential adverse or beneficial impact on our business;

any potential adverse or beneficial impact on our relationships with our customers or suppliers or other service providers;

whether it would enhance or support a competitor’s position;
the extent to which it would result in financial or other benefit (direct or indirect) to the employee;

the extent to which it would result in financial or other benefit (direct or indirect) to one of our customers, suppliers or other service
providers; and

the extent to which it would appear improper to an outside observer.

Although no list can include every possible situation in which a conflict of interest could arise, the following are examples of situations
that may, depending on the facts and circumstances, involve problematic conflicts of interests:

●

●

●

●

●

●

●

●

●

Employment by (including consulting for) or service on the board of a competitor, customer or supplier or other service provider.
Activity that enhances or supports the position of a competitor to the detriment of the Company is prohibited, including employment
by  or  service  on  the  board  of  a  competitor.  Employment  by  or  service  on  the  board  of  a  customer  or  supplier  or  other  service
provider is generally discouraged and you must seek authorization in advance if you plan to take such a position.

Owning, directly or indirectly, a significant financial interest in any entity that does business, seeks to do business or competes with
us. In addition to the factors described above, persons evaluating ownership in other entities for conflicts of interest will consider
the  size  and  nature  of  the  investment;  the  nature  of  the  relationship  between  the  other  entity  and  the  Company;  the  employee’s
access to confidential information and the employee’s ability to influence the Company’s decisions. If you would like to acquire a
financial interest of that kind, you must seek approval in advance.

Soliciting  or  accepting  gifts,  favors,  loans  or  preferential  treatment  from  any  person  or  entity  that  does  business  or  seeks  to  do
business with us. See Section 12 for further discussion of the issues involved in this type of conflict.

Soliciting  contributions  to  any  charity  or  for  any  political  candidate  from  any  person  or  entity  that  does  business  or  seeks  to  do
business with us.

Taking  personal  advantage  of  corporate  opportunities.  See  Section  9  for  further  discussion  of  the  issues  involved  in  this  type  of
conflict.

Moonlighting without permission.

Conducting  our  business  transactions  with  your  family  member  or  a  business  in  which  you  have  a  significant  financial  interest.
Material related-party transactions approved by the Audit Committee of the Board of Directors and involving any executive officer
or director will be publicly disclosed as required by applicable laws and regulations.

Exercising supervisory or other authority on behalf of the Company over a co-worker who is also a family member. The employee’s
supervisor  and/or  the  Compliance  Officer  will  consult  with  the  Human  Resources  department  to  assess  the  advisability  of
reassignment.

Loans to, or guarantees of obligations of, employees or their family members by the Company could constitute an improper personal
benefit to the recipients of these loans or guarantees, depending on the facts and circumstances. Some loans are expressly prohibited
by law and applicable law requires that our Board of Directors approve all loans and guarantees to employees. As a result, all loans
and guarantees by the Company must be approved in advance by the Audit Committee of the Board of Directors.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
9.

Corporate Opportunities

You may not take personal advantage of opportunities for the Company that are presented to you or discovered by you as a result of your
position with us or through your use of corporate property or information, unless authorized by your supervisor, the Compliance Officer
or the Audit Committee of the Board of Directors, as described in Section 8. Even opportunities that are acquired privately by you may be
questionable if they are related to our existing or proposed lines of business. Significant participation in an investment or outside business
opportunity that is directly related to our lines of business must be pre- approved. You may not use your position with us or corporate
property or information for improper personal gain, nor should you compete with us in any way.

10.

Maintenance of Corporate Books, Records, Documents and Accounts; Financial Integrity; Public Reporting

The integrity of our records and public disclosure depends upon the validity, accuracy and completeness of the information supporting
the  entries  to  our  books  of  account.  Therefore,  our  corporate  and  business  records  should  be  completed  accurately  and  honestly.  The
making  of  false  or  misleading  statements  and  entries,  whether  they  relate  to  financial  results  or  test  results,  is  strictly  prohibited.  Our
records  serve  as  a  basis  for  managing  our  business  and  are  important  in  meeting  our  obligations  to  customers,  suppliers,  creditors,
employees and others with whom we do business. As a result, it is important that our books, records and accounts accurately and fairly
reflect,  in  reasonable  detail,  our  assets,  liabilities,  revenues,  costs  and  expenses,  as  well  as  all  transactions  and  changes  in  assets  and
liabilities. We require that:

● no  entry  be  made  in  our  books  and  records  that  intentionally  hides  or  disguises  the  nature  of  any  transaction  or  of  any  of  our

liabilities, or misclassifies any transactions as to accounts or accounting periods;

●    transactions be supported by appropriate documentation and internal approval;

●    the terms of sales and other commercial transactions be accurately and timely reflected in the documentation for those transactions

and all such documentation be reflected accurately in our books and records;

●   employees comply with our system of internal controls; and

●   no cash or other assets be maintained for any purpose in any unrecorded or “off-the-books” fund.

Our accounting records are also relied upon to produce reports for our management, stockholders and creditors, as well as for governmental
agencies. In particular, we rely upon our accounting and other business and corporate records in preparing the periodic and current reports
that we file with the SEC. Securities laws require that these reports provide full, fair, accurate, timely and understandable disclosure and
fairly  present  our  financial  condition  and  results  of  operations.  Employees  who  collect,  provide  or  analyze  information  for  or  otherwise
contribute in any way in preparing or verifying these reports should strive to ensure that our financial disclosure is accurate and transparent
and  that  our  reports  contain  all  of  the  information  about  the  Company  that  would  be  important  to  enable  stockholders  and  potential
investors to assess the soundness and risks of our business and finances and the quality and integrity of our accounting and disclosures.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
In addition:

●    no employee may take or authorize any action that would cause our financial records or financial disclosure to fail to comply with

generally accepted accounting principles, the rules and regulations of the SEC or other applicable laws, rules and regulations;

●    all employees must cooperate fully with our Finance Department, as well as our independent registered public accounting firm
and legal counsel, respond to their questions with candor and provide them with complete and accurate information to help ensure
that our books and records, as well as our reports filed with the SEC, are accurate and complete; and

●    no employee should knowingly make (or cause or encourage any other person to make) any false or misleading statement in any
of our reports filed with the SEC or knowingly omit (or cause or encourage any other person to omit) any information necessary to
make the disclosure in any of our reports accurate in all material respects.

Any employee who becomes aware of any departure from these standards has a responsibility to report his or her knowledge promptly to
a supervisor, the Compliance Officer or one of the other compliance resources described in Section 20.

11.

Fair Dealing

We  strive  to  outperform  our  competition  fairly  and  honestly.  Advantages  over  our  competitors  are  to  be  obtained  through  superior
performance  of  our  products  and  services,  not  through  unethical  or  illegal  business  practices. Acquiring  proprietary  information  from
others  through  improper  means,  possessing  trade  secret  information  that  was  improperly  obtained,  or  inducing  improper  disclosure  of
confidential information from past or present employees of other companies is prohibited, even if motivated by an intention to advance
our interests. If information is obtained by mistake that may constitute a trade secret or other confidential information of another business,
or if you have any questions about the legality of proposed information gathering, you must consult your supervisor or the Compliance
Officer, as further described in Section 20.

You are expected to deal fairly with our customers, suppliers, employees and anyone else with whom you have contact in the course of
performing your job. Be aware that the Federal Trade Commission Act (the “FTC Act”) provides that “unfair methods of competition in
commerce, and unfair or deceptive acts or practices in commerce, are declared unlawful.” It is a violation of the FTC Act to engage in
deceptive, unfair or unethical practices and to make misrepresentations in connection with sales activities.

Employees involved in procurement have a special responsibility to adhere to principles of fair competition in the purchase of products
and services by selecting suppliers based exclusively on normal commercial considerations, such as quality, cost, availability, service and
reputation, and not on the receipt of special favors.

12.

Gifts and Other Benefits

Gifts,  hospitality  and  other  benefits  may  not  be  offered,  provided  or  accepted  by  any  employee  in  the  course  of  business  without  the
express permission of the Compliance Officer, the Chief Executive Officer, or the Audit Committee of the Board of Directors and must
be consistent with customary business practices and not (a) of more than token or nominal monetary value, (b) in cash or cash equivalent,
(c) susceptible of being construed as a bribe or kickback, (d) made or received on a regular or frequent basis, (e) pose a potential conflict
of interest, or (f) in violation of any laws, regulations, or industry guidance. This principle applies to our transactions everywhere in the
world, even where the practice is widely considered “a way of doing business.” Employees should not accept gifts or entertainment that
may reasonably be deemed to affect their judgment or actions in the performance of their duties. Our customers, suppliers and the public
at large should know that our employees’ judgment is not for sale.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
The Company is further committed to interacting with healthcare professionals in an ethical and professional manner, in compliance with
all  applicable  laws,  rules  and  regulations.  Offering  anything  of  value  to  a  healthcare  professional  intended  to  influence  that  person  to
recommend or purchase a product or service that may be reimbursed through a government-funded system is strictly prohibited by law and
Company policy. Employees must avoid engaging in any activity that would inappropriately influence a healthcare professional’s medical
judgment  or  treatment  decisions.  Meals  and  other  nominally-valued  items  allowable  under  Company  policy  must  be  entered  into  our
expense management system for accurate tracking and reporting purposes.

Under  some  statutes,  such  as  the  U.S.  Foreign  Corrupt  Practices Act  (further  described  in  Section  4),  giving  anything  of  value  to  a
government official to obtain or retain business or favorable treatment is a criminal act subject to prosecution and conviction. Discuss with
your supervisor or the Compliance Officer any proposed entertainment or gifts if you are uncertain about their appropriateness.

13.

Political Contributions & Activity

Political contributions are highly regulated and violations are subject to serious penalties. Accordingly, employees should not make any
political contributions on behalf of the Company anywhere in the world. This includes financial and in-kind contributions made by the
Company. If you engage in personal political activity, you must do so on your own time with your own resources. Be careful to separate
your own political activities from those of the Company and do not use Company property or equipment for personal political purposes,
because even the appearance of a Company contribution of time or resources could be viewed as a violation.

14.

Quality

The  Company  is  committed  to  quality  and  integrity  in  all  its  research,  development,  and  manufacturing  operations.  Each  employee  is
responsible  for  knowing  and  abiding  by  the  laws  and  regulations  that  apply  to  these  activities,  including  without  limitation,  good
laboratory  practices,  good  clinical  practices,  good  manufacturing  practices,  good  distribution  practices,  and  applicable  country-specific
regulation. The Company will not tolerate the falsification or fabrication of research, clinical or manufacturing data.

15.

Product Promotion & Advertising

The Company is committed to complying with all applicable laws, rules and regulation for the countries in which it markets products. No
employee, or consultant acting on behalf of the Company, may promote a product for use before the product is approved for such use.
This  limitation  however,  does  not  restrict  the  appropriate  exchange  of  scientific  information  in  medical  forums  and  upon  specific
unsolicited  request  for  such  information.  The  promotion  of  approved  Company  products  shall  be  done  in  a  factually  accurate  and
balanced manner, shall not be false nor misleading in any way, and facilitated by only those unaltered materials reviewed and approved
by an internal cross-functional committee.

16.

Protection and Proper Use of Company Assets

All  employees  are  expected  to  protect  our  assets  and  ensure  their  efficient  use.  Theft,  carelessness  and  waste  have  an  effect  on  our
profitability. Our property, such as office supplies, lab equipment, computer equipment, buildings and products, are expected to be used
only  for  legitimate  business  purposes,  although  incidental  personal  use  may  be  permitted.  You  may  not,  however,  use  our  corporate
name, any brand name or trademark owned or associated with the Company or any letterhead stationery for any personal purpose.

You may not, while acting on behalf of the Company or while using our computing or communications equipment or facilities, either:

●    access confidential systems (also known as “hacking”) or other resource of another entity without express written authorization

from the entity responsible for operating that resource; or

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
●    commit any unlawful or illegal act, including harassment, libel, fraud, sending of unsolicited bulk email (also known as “spam”) in

violation of applicable law, trafficking in contraband of any kind or espionage.

If you receive authorization to access another entity’s internal computer system or other resource, you must make a permanent record of
that authorization so that it may be retrieved for future reference, and you may not exceed the scope of that authorization.

Unsolicited bulk email is regulated by law in a number of jurisdictions. If you intend to send unsolicited bulk email to persons outside of
the Company, either while acting on our behalf or using our computing or communications equipment or facilities, you should contact
your supervisor or the Compliance Officer for approval.

All  data  residing  on  or  transmitted  through  our  computing  and  communications  facilities,  including  email  and  word  processing
documents,  is  the  property  of  the  Company  and  subject  to  inspection,  retention  and  review  by  the  Company,  with  or  without  an
employee’s or third party’s knowledge, consent or approval, in accordance with applicable law. Any misuse or suspected misuse of our
assets must be immediately reported to your supervisor or the Compliance Officer.

17.

Confidentiality

One of our most important assets is our confidential information. As an employee of the Company, you may learn of information about
the Company that is confidential and proprietary. You also may learn of information before that information is released to the general
public. Employees who have received or have access to confidential information should take care to keep this information confidential.
Confidential information includes non-public information that might be of use to competitors or harmful to the Company or its customers
if disclosed, such as business, marketing and service plans, financial information, product architecture, source codes, inventions, chemical
structures,  designs,  databases,  customer  lists,  pricing  strategies,  personnel  data,  personally  identifiable  information  pertaining  to  our
employees, customers or other individuals (including, for example, names, addresses, telephone numbers and social security numbers),
and similar types of information provided to us by our customers, suppliers and partners. This information may be protected by patent,
trademark, copyright and trade secret laws.

In  addition,  because  we  interact  with  other  companies  and  organizations,  there  may  be  times  when  you  learn  confidential  information
about other companies before that information has been made available to the public. You must treat this information in the same manner
as you are required to treat our confidential and proprietary information. There may even be times when you must treat as confidential the
fact that we have an interest in, or are involved with, another company.

You are expected to keep confidential and proprietary information confidential unless and until that information is released to the public
through  approved  channels  (usually  through  a  press  release,  an  SEC  filing  or  a  formal  communication  from  a  member  of  senior
management,  as  further  described  in  Section  18).  Every  employee  has  a  duty  to  refrain  from  disclosing  to  any  person  confidential  or
proprietary information about us or any other company learned in the course of employment here, until that information is disclosed to
the  public  through  approved  channels.  This  policy  requires  you  to  refrain  from  discussing  confidential  or  proprietary  information  with
outsiders  and  even  with  other  Company  employees,  unless  those  fellow  employees  have  a  legitimate  need  to  know  the  information  in
order  to  perform  their  job  duties.  Unauthorized  use  or  distribution  of  this  information  could  also  be  illegal  and  result  in  civil  liability
and/or criminal penalties.

You should also take care not to inadvertently disclose confidential information. Materials that contain confidential information, such as
memos,  notebooks,  computer  disks  and  laptop  computers,  should  be  stored  securely.  Unauthorized  posting  or  discussion  of  any
information  concerning  our  business,  information  or  prospects  on  the  Internet  is  prohibited.  You  may  not  discuss  our  business,
information  or  prospects  in  any  non-Company  hosted  public  “chat  room,”  web  log  (“blog”),  or  other  similar  electronic  environment,
regardless of whether you use your own name or a pseudonym. Be cautious when discussing sensitive information in public places like
elevators, airports, restaurants and “quasi-public” areas within the Company. All Company emails, voicemails and other communications
are presumed confidential and

should not be forwarded or otherwise disseminated outside of the Company except where required for legitimate business purposes.

In addition to the above responsibilities, if you are handling information protected by any privacy policy published by us, then you must
handle that information in accordance with the applicable policy.

18.

Media/Public Discussions

It is our policy to disclose material information concerning the Company to the public only through specific limited channels to avoid
inappropriate publicity and to ensure that all those with an interest in the Company will have equal access to information. All inquiries or
calls from the press and financial analysts should be referred to the Chief Executive Officer, Chief Scientific Officer or Chief Financial
Officer. We have designated these individuals as our official spokespersons for financial matters, marketing, technical and other related
information. Unless they have made a specific exception, these designees are the only people who may communicate with the press on
behalf of the Company. You also may not provide any information to the media about us off the record, for background, confidentially or
secretly.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
19.

Waivers

Any waiver of this Code for executive officers (including, where required by applicable laws, our principal executive officer, principal
financial officer, principal accounting officer or controller (or persons performing similar functions)) or directors may be authorized only
by our Board of Directors or, to the extent permitted by the rules of Nasdaq, a committee of the Board of Directors and will be disclosed
to stockholders as required by applicable laws, rules and regulations.

20.

Compliance Standards and Procedures

Compliance Resources

To facilitate compliance with this Code, we have established the position of Compliance Officer to oversee this program. The Compliance
Officer is a person to whom you can address any questions or concerns. Our Chief Financial Officer serves as our Compliance Officer. In
addition to fielding questions or concerns with respect to potential violations of this Code, the Compliance Officer is responsible for:

●       investigating  possible  violations  of  this  Code,  both  autonomously  and  in  partnership  with  other  functions  as  needed  (e.g.,

supporting Human Resources on matters of workplace violence, harassment or discrimination);

●    training new employees on the Code and supporting policies;

●    maintaining access to an electronic version of the Code and ensuring that each employee receives annual refresher training and

certifies to their understanding of and compliance with the Code;

●       distributing  copies  of  this  Code  annually  via  email  to  each  employee  with  a  reminder  that  each  employee  is  responsible  for

reading, understanding and complying with this Code;

●    collaborating with Human Resources, management, and other departments as needed on corrective actions to ensure consistent

enforcement of disciplinary measures;

●    updating this Code as needed and alerting employees to any updates, with appropriate approval of the Audit Committee of the
Board  of  Directors,  to  reflect  changes  in  the  law,  Company  operations  and  in  recognized  best  practices,  and  to  reflect  Company
experience; and otherwise promoting an atmosphere of responsible and ethical conduct.

Your most immediate resource for any matter related to this Code is your supervisor. He or she may have the information you need or
may  be  able  to  refer  the  question  to  another  appropriate  source.  There  may,  however,  be  times  when  you  prefer  not  to  go  to  your
supervisor.  In  these  instances,  you  should  feel  free  to  discuss  your  concern  with  the  Compliance  Officer.  If  you  are  uncomfortable
speaking with the Compliance Officer because he or she works in your department or is one of your supervisors, please contact the Chief
Executive Officer. Of course, if your concern involves potential misconduct by another person and relates to questionable accounting or
auditing matters, you may report that violation directly to the Audit Committee of the Board of Directors.

Clarifying Questions and Concerns; Reporting Possible Violations

If you encounter a situation or are considering a course of action and its appropriateness is unclear, discuss the matter promptly with your
supervisor or the Compliance Officer; even the appearance of impropriety can be very damaging and should be avoided.

If you are aware of a suspected or actual violation of Code standards by others, you have a responsibility to report it. You are expected to
promptly  provide  a  compliance  resource  with  a  specific  description  of  the  violation  that  you  believe  has  occurred,  including  any
information you have about the persons involved and the time of the violation. Whether you choose to speak with your supervisor or the
Compliance  Officer,  you  should  do  so  without  fear  of  any  form  of  retaliation.  We  will  take  prompt  disciplinary  action  against  any
employee who retaliates against you, including termination of employment.

Supervisors  must  promptly  report  any  complaints  or  observations  of  Code  violations  to  the  Compliance  Officer.  If  you  believe  your
supervisor has not taken appropriate action, you should contact the Compliance Officer directly. The Compliance Officer will investigate
all  reported  possible  Code  violations  promptly  and  with  the  highest  degree  of  confidentiality  that  is  possible  under  the  specific
circumstances. Neither you nor your supervisor may conduct any preliminary investigation, unless authorized to do so by the Compliance
Officer.  Your  cooperation  in  the  investigation  will  be  expected.  As  needed,  the  Compliance  Officer  will  consult  with  the  Human
Resources  department  and/or  the Audit  Committee  of  the  Board  of  Directors.  It  is  our  policy  to  employ  a  fair  process  by  which  to
determine violations of this Code.

With  respect  to  any  complaints  or  observations  of  violations  that  may  involve  accounting,  internal  accounting  controls  and  auditing
concerns, the Compliance Officer shall promptly inform the Audit Committee of the Board of Directors, and the Audit Committee of the
Board of Directors shall be responsible for supervising and overseeing the inquiry and any investigation that is undertaken.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
If any investigation indicates that a violation of this Code has probably occurred, we will take such action as we believe to be appropriate
under the circumstances. If we determine that an employee is responsible for a Code violation, he or she will be subject to disciplinary
action  up  to,  and  including,  termination  of  employment  and,  in  appropriate  cases,  civil  action  or  referral  for  criminal  prosecution.
Appropriate action may also be taken to deter any future Code violations.

 
Exhibit 31.1

CERTIFICATION

I, Chandler D. Robinson, certify that:

I have reviewed this Annual Report on Form 10-K of Monopar Therapeutics Inc.;

1.
2. Based on my knowledge, this report does not contain any untrue statement of a material fact or omit to state a material fact necessary to
make  the  statements  made,  in  light  of  the  circumstances  under  which  such  statements  were  made,  not  misleading  with  respect  to  the
period covered by this report;

3. Based on my knowledge, the financial statements, and other financial information included in this report, fairly present in all material
respects the financial condition, results of operations and cash flows of the registrant as of, and for, the periods presented in this report;
4. The registrant’s other certifying officer(s) and I are responsible for establishing and maintaining disclosure controls and procedures (as

defined in Exchange Act Rules 13a-15(e) and 15d-15(e)) for the registrant and have:
a) designed  such  disclosure  controls  and  procedures,  or  caused  such  disclosure  controls  and  procedures  to  be  designed  under  our
supervision,  to  ensure  that  material  information  relating  to  the  registrant  is  made  known  to  us  by  others  within  those  entities,
particularly during the period in which this report is being prepared;

b) designed such internal control over financial reporting, or caused such internal control over financial reporting to be designed under
our  supervision,  to  provide  reasonable  assurance  regarding  the  reliability  of  financial  reporting  and  the  preparation  of  financial
statements for external purposes in accordance with generally accepted accounting principles;
evaluated the effectiveness of the registrant’s disclosure controls and procedures and presented in this report our conclusions about
the  effectiveness  of  the  disclosure  controls  and  procedures,  as  of  the  end  of  the  period  covered  by  this  report  based  on  such
evaluation; and

c)

5. The registrant’s other certifying officer(s) and I have disclosed, based on our most recent evaluation of internal control over financial
reporting, to the registrant’s auditors and the audit committee of the registrant’s board of directors (or persons performing the equivalent
functions):
a)

all significant deficiencies and material weaknesses in the design or operation of internal control over financial reporting which are
reasonably likely to adversely affect the registrant’s ability to record, process, summarize and report financial information; and
any  fraud,  whether  or  not  material,  that  involves  management  or  other  employees  who  have  a  significant  role  in  the  registrant’s
internal control over financial reporting.

b)

Date: March 26, 2018

/s/ CHANDLER D. ROBINSON

Chandler D. Robinson

Chief Executive Officer

 
 
 
 
 
 
 
 
 
 
 
  
Exhibit 31.2

CERTIFICATION

I, Kim R. Tsuchimoto, certify that:

I have reviewed this Annual Report on Form 10-K of Monopar Therapeutics Inc.;

1.
2. Based on my knowledge, this report does not contain any untrue statement of a material fact or omit to state a material fact necessary to
make  the  statements  made,  in  light  of  the  circumstances  under  which  such  statements  were  made,  not  misleading  with  respect  to  the
period covered by this report;

3. Based on my knowledge, the financial statements, and other financial information included in this report, fairly present in all material
respects the financial condition, results of operations and cash flows of the registrant as of, and for, the periods presented in this report;
4. The registrant’s other certifying officer(s) and I are responsible for establishing and maintaining disclosure controls and procedures (as

defined in Exchange Act Rules 13a-15(e) and 15d-15(e)) for the registrant and have:
a) designed  such  disclosure  controls  and  procedures,  or  caused  such  disclosure  controls  and  procedures  to  be  designed  under  our
supervision,  to  ensure  that  material  information  relating  to  the  registrant  is  made  known  to  us  by  others  within  those  entities,
particularly during the period in which this report is being prepared;

b) designed such internal control over financial reporting, or caused such internal control over financial reporting to be designed under
our  supervision,  to  provide  reasonable  assurance  regarding  the  reliability  of  financial  reporting  and  the  preparation  of  financial
statements for external purposes in accordance with generally accepted accounting principles;
evaluated the effectiveness of the registrant’s disclosure controls and procedures and presented in this report our conclusions about
the  effectiveness  of  the  disclosure  controls  and  procedures,  as  of  the  end  of  the  period  covered  by  this  report  based  on  such
evaluation; and

c)

5. The registrant’s other certifying officer(s) and I have disclosed, based on our most recent evaluation of internal control over financial
reporting, to the registrant’s auditors and the audit committee of the registrant’s board of directors (or persons performing the equivalent
functions):
a)

all significant deficiencies and material weaknesses in the design or operation of internal control over financial reporting which are
reasonably likely to adversely affect the registrant’s ability to record, process, summarize and report financial information; and
any  fraud,  whether  or  not  material,  that  involves  management  or  other  employees  who  have  a  significant  role  in  the  registrant’s
internal control over financial reporting.

b)

Date: March 26, 2018

/s/ KIM R. TSUCHIMOTO

Kim R. Tsuchimoto

Chief Executive Officer

 
 
 
 
 
 
 
 
Exhibit 32.1

CERTIFICATION PURSUANT TO
18 U.S.C. SECTION 1350,
AS ADOPTED PURSUANT TO
SECTION 906 OF THE SARBANES-OXLEY ACT OF 2002

In connection with the Annual Report on Form 10-K of Monopar Therapeutics Inc. (the Company) for the year ended December 31, 2017,
as filed with the Securities and Exchange Commission on the date hereof (the Report), we, Chandler D. Robinson, and Kim R. Tsuchimoto,
hereby certify, pursuant to 18 U.S.C. §1350, as adopted pursuant to §906 of the Sarbanes-Oxley Act of 2002, that:

(1) the Report fully complies with the requirements of Section 13(a) or 15(d) of the Securities Exchange Act of 1934; and
(2) the information contained in the Report fairly presents, in all material respects, the financial condition and results of operations of

the Company.

/s/ CHANDLER D. ROBINSON

Chandler D. Robinson

Chief Executive Officer

March 26, 2018

/s/ KIM R. TSUCHIMOTO

Kim R. Tsuchimoto

Chief Executive Officer

March 26, 2018

This certification accompanies the Form 10-K to which it relates, is not deemed filed with the Securities and Exchange Commission and is
not to be incorporated by reference into any filing of Monopar Therapeutics Inc. under the Securities Act of 1933, as amended, or the
Securities Exchange Act of 1934, as amended (whether made before or after the date of the Form 10-K), irrespective of any general
incorporation language contained in such filing.