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Cerecor Inc.

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FY2018 Annual Report · Cerecor Inc.
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UNITED STATES
SECURITIES AND EXCHANGE COMMISSION
Washington, D.C. 20549
FORM 10‑K

(Mark One)

ý ANNUAL REPORT PURSUANT TO SECTION 13 OR 15(d) OF THE SECURITIES EXCHANGE ACT OF 1934

For the fiscal year ended December 31,  2018
OR
☐ TRANSITION REPORT PURSUANT TO SECTION 13 OR 15(d) OF THE SECURITIES EXCHANGE ACT OF 1934

For the transition period from ______to______             
Commission File No. 001‑37590
Cerecor Inc.
(Exact name of registrant as specified in its charter)

Delaware
(State or other jurisdiction of
incorporation or organization)

45‑0705648
(I.R.S. Employer
Identification No.)

540 Gaither Road, Suite 400
Rockville, Maryland 20850
(Address of principal executive offices)
Telephone: (410) 522-8707
(Registrant’s telephone number, including area code)
Securities registered pursuant to Section 12(b) of the Act:

Title of each class
Common Stock, $0.001 par value

Name of each exchange on which registered
NASDAQ Stock Market

Securities registered pursuant to section 12(g) of the Act:  None
Indicate by check mark if the registrant is a well‑known seasoned issuer, as defined in Rule 405 of the Securities Act. Yes ☐  No  ý
Indicate by check mark if the registrant is not required to file reports pursuant to Section 13 or Section 15(d) of the Act. Yes ☐  No  ý
Indicate by check mark whether the registrant (1) has filed reports required to be filed by Section 13 or 15(d) of the Securities Exchange Act of

1934 during the preceding 12 months (or for such shorter period that the registrant was required to file such reports), and
(2) has been subject to such filing requirements for the past 90 days. Yes ý  No ☐

Indicate by check mark whether the registrant has submitted electronically and posted on its corporate web site, if any, every Interactive Data
File required to be submitted and posted pursuant to Rule 405 of Regulation S‑T (§232.405 of this chapter) during the preceding 12 months (or for such
shorter period that the registrant was required to submit and post such files). Yes ý  No ☐

Indicate by check mark if disclosure of delinquent filers pursuant to Item 405 of Regulation S‑K (§299.405 of this chapter) is not contained

herein, and will not be contained, to the best of registrant’s knowledge, in definitive proxy or information statements incorporated by reference in
Part III of this Form 10‑K or any amendment to this Form 10‑K. ☐

Indicate by check mark whether the registrant is a large accelerated filer, an accelerated filer, a non-accelerated filer, a smaller reporting
company, or an emerging growth company. See definitions of “large accelerated filer,” “accelerated filer,” “smaller reporting company,” and "emerging
growth company" in Rule12b-2 of the Exchange Act.

Large accelerated filer ☐

Accelerated filer ☐

Non‑accelerated filer ý

Smaller reporting company ý Emerging growth company ý

If an emerging growth company, indicate by check mark if the registrant has elected not to use the extended transition period for complying

with any new or revised financial accounting standards provided pursuant to Section 13(a) of the Exchange Act. ý

Indicate by check mark whether the registrant is a shell company (as defined in Rule 12b‑2 of the Exchange Act). Yes ☐  No  ý

The aggregate market value of the registrant’s shares of common stock held by non-affiliates of the registrant as of June 30, 2018 (based on
the closing price of $4.34 on June 29, 2018, the last business day of the registrant's most recently completed second fiscal quarter) was $40,821,693.
Shares of common stock held by each officer and directors and by each person known to be the registrant who owned 10% or more of the outstanding
common stock have been excluded in that such person may be deemed to be affiliates. This determination of affiliate status is not necessarily a
conclusive determination for other purposes.

As of March 11, 2019, there were 42,653,659 outstanding shares of the registrant’s common stock, par value $0.001 per share.

Documents Incorporated by Reference: Portions of the registrant’s Definitive Proxy Statement to be filed with the Securities and Exchange
Commission no later than 120 days after the end of the registrant’s fiscal year ended December 31, 2018, are incorporated by reference in Part III of
this Annual Report on Form 10-K.

 
 
 
 
 
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TABLE OF CONTENTS

PART I 
Item 1. Business 
Item 1A. Risk Factors 
Item 1B. Unresolved Staff Comments 
Item 2. Properties 
Item 3. Legal Proceedings 
Item 4. Mine Safety Disclosures 
PART II 
Item 5. Market for Registrant’s Common Equity, Related Stockholder Matters and Issuer Purchases of Equity
Securities 
Item 6. Selected Financial Data 
Item 7. Management’s Discussion and Analysis of Financial Condition and Results of Operations 
Item 7A. Quantitative and Qualitative Disclosures About Market Risk 
Item 8. Financial Statements and Supplementary Data 

Item 9. Changes in and Disagreements with Accountants on Accounting and Financial Disclosure 
Item 9A. Controls and Procedures 
Item 9B. Other Information 
PART III 
Item 10. Directors, Executive Officers and Corporate Governance 
Item 11. Executive Compensation 
Item 12. Security Ownership of Certain Beneficial Owners and Management and Related Stockholder Matters 
Item 13. Certain Relationships and Related Transactions, and Director Independence 
Item 14. Principal Accountant Fees and Services 
PART IV. 
Item 15. Exhibits; Financial Statement Schedules
Item 16. Form 10-K Summary

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SPECIAL NOTE REGARDING FORWARD‑LOOKING STATEMENTS

PART I

This  report  and  the  information  incorporated  herein  by  reference  contain  forward-looking  statements  that  involve  a  number  of
risks and uncertainties, as well as assumptions that, if they never materialize or prove incorrect, could cause our results to differ materially
from  those  expressed  or  implied  by  such  forward-looking  statements. Although  our  forward-looking  statements  reflect  the  good  faith
judgment  of  our  management,  these  statements  can  only  be  based  on  facts  and  factors  currently  known  by  us.  Consequently,  forward-
looking statements are inherently subject to risks and uncertainties, and actual results and outcomes may differ materially from results and
outcomes discussed in the forward-looking statements.

Forward-looking statements can be identified by the use of forward-looking words such as “believes,” “expects,” “may,” “will,”
“plans,” “intends,” “estimates,” “could,” “should,” “would,” “continue,” “seeks,” “aims,” “projects,” “predicts,” “pro forma,” “anticipates,”
“potential” or other similar words (including their use in the negative), or by discussions of future matters such as results of operations,
cash flows, market position, sales efforts, the development of product candidates or products, the timing and results of clinical trials, the
potential  attributes  and  benefits  of  our  product  candidates,  the  use  and  sufficiency  of  capital  resources  and  other  statements  that  are  not
historical. These statements include but are not limited to statements under the captions  “Business,”  “Risk  Factors”  and  “Management’s
Discussion and Analysis of Financial Condition and Results of Operations” as well as other sections in this report. You should be aware
that the occurrence of any of the events discussed under the caption “Risk Factors” and elsewhere in this report could substantially harm
our business, results of operations and financial condition and cause our results to differ materially from those expressed or implied by our
forward-looking statements. If any of these events occurs, the trading price of our common stock could decline and you could lose all or a
part of the value of your shares of our common stock.

The  cautionary  statements  made  in  this  report  are  intended  to  be  applicable  to  all  related  forward-looking  statements  wherever
they may appear in this report. We urge you not to place undue reliance on these forward-looking statements, which speak only as of the
date of this report.

As used in this report, the terms "Cerecor," "Company," "we," "us," and "our" mean Cerecor Inc. and its subsidiaries unless the

context indicates otherwise.

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Item 1. Business.

Overview

Cerecor  Inc.  (the  Company  or  "Cerecor")  is  a  fully  integrated  biopharmaceutical  company  with  commercial  operations  and
research  and  development  capabilities. The  Company  is  building  a  robust  pipeline  of  innovative  therapies  in  neurology,  pediatric
healthcare, and orphan rare diseases.

The Company's neurology pipeline is led by CERC-301, which is currently in a Phase I safety study for Neurogenic Orthostatic
Hypotension ("nOH"). The Company is also developing two other neurological clinical and preclinical stage compounds. The Company's
pediatric  orphan  rare  disease  pipeline  is  led  by  CERC-801,  CERC-802  and  CERC-803. All three  of  these  compounds  are  preclinical
therapies for inherited metabolic disorders known as Congenital Disorders of Glycosylation ("CDGs") by means of substrate replacement
therapy. The  U.S.  Food  and  Drug Administration  ("FDA")  has  granted  Rare  Pediatric  Disease  designation  ("RPDD")  and  Orphan  Drug
Designation ("ODD") to all three compounds. Under the FDA’s Rare Pediatric Disease Priority Review Voucher ("PRV") program, upon
the  approval  of  a  new  drug  application  ("NDA")  for  the  treatment  of  a  rare  pediatric  disease,  the  sponsor  of  such  application  would  be
eligible for a PRV that can be used to obtain priority review for a subsequent new drug application or biologics license application. The
PRV may be sold or transferred an unlimited number of times. The Company plans to leverage the 505(b)(2) NDA pathway for all  three
compounds  to  accelerate  development  and  approval. The  Company  is  also  in  the  process  of  developing one  other  preclinical  pediatric
orphan rare disease compound, CERC-913.

The  Company  also  has  a  diverse  portfolio  of  marketed  products. Our  marketed  products  are  led  by  our  prescribed  dietary
supplements and prescribed drugs. Our prescribed dietary supplements include Poly-Vi-Flor and Tri-Vi-Flor which are prescription vitamin
and fluoride supplements used in infants and children to treat or prevent deficiency of essential vitamins and fluoride. The Company also
markets  a  number  of  prescription  drugs  that  treat  a  range  of  pediatric  diseases,  disorders  and  conditions. Cerecor's  prescription  drugs
include  Millipred®,  Ulesfia®,  Karbinal™  ER, AcipHex®  Sprinkle™  and  Cefaclor  for  Oral  Suspension.  Finally,  the  Company  has  one
marketed medical device, Flexichamber™.

Recent Developments

Ichorion Asset Acquisition

On September 24, 2018, we acquired Ichorion Therapeutics, Inc. for approximately 5.8 million shares of the Company’s Common
Stock, par value $0.001 per share, as adjusted for estimated working capital.  Consideration for the Ichorion asset acquisition also includes
certain development milestones worth up to an additional $15 million, payable either in shares of the Company's common stock or in cash,
at the election of the Company. Substantially all of the value of Ichorion was related to one group of similar identifiable assets, which was
the in-process research and development ("IPR&D") for the three preclinical therapies for CDGs (CERC-801, CERC-802 and CERC-803)
and as such the Company accounted for this transaction as an asset acquisition.

Acquisition of Avadel Products

On February 16, 2018, we acquired all rights in the Avadel U.S. Holdings, Inc’s marketed pediatric products for a nominal cash
payment  and  assumption  of  certain  of Avadel’s  financial  obligations  to  Deerfield  CSF,  LLC,  which  include  a  $15  million  loan  due  in
January  2021  and  certain  royalty  obligations  through  February  2026.  The  acquired  products  consist  of  Karbinal™  ER,  AcipHex®
Sprinkle™, Cefaclor for Oral Suspension, and Flexichamber™.

Research and Development Updates

During the third quarter of 2018, the Company enrolled its first patient in the Phase 1 trial for nOH in Parkinson’s Disease. The

purpose of this study is to evaluate the single-dose safety, tolerability and pharmacokinetics of CERC-301 in the relevant patient population
from the study, as well as explore the effects on blood pressure of nOH during an orthostatic challenge at escalating dose levels. Data is
expected in the first half of 2019. In early 2019, a patent was issued for CERC-301, which provides Cerecor with intellectual property rights
to CERC-301 until 2035.

During the fourth quarter of 2018, the FDA awarded RPDD for CERC-801, CERC-802, and CERC-803. Additionally, the FDA

granted ODD to each of the three compounds in early 2019, thus granting eligibility for receipt of a PRV upon approval of an NDA. In
addition to PRV eligibility, there are numerous benefits associated with receipt of both ODD and RPDD which include 7-year marketing
exclusivity (upon approval) in the United States, tax credits (up to 25% of clinical development costs) and waiver of Prescription Drug
User Fee Act ("PDUFA") application fees (filing fees).

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The Company also filed an Investigational New Drug ("IND") application with the FDA for CERC-801 in the fourth quarter of

2018 and received a may proceed letter in early 2019. Additionally, the FDA designated Fast Track Designation for CERC-801. Fast Track
Designation is granted to drugs being developed for the treatment of serious or life-threatening diseases or conditions where there is an
unmet medical need. The purpose of the Fast Track Designation provision is to help facilitate development and expedite the review of
drugs to treat serious and life-threatening conditions so that an approved product can reach the market expeditiously. The clinical
development program for CERC-801 will commence in 2019 with a Phase 1 study in healthy volunteers. The goals of the study will be to
assess the single dose tolerability and pharmacokinetics of CERC-801. Cerecor seeks to leverage existing clinical and nonclinical data in
conjunction with sponsor-initiated studies, such as this Phase 1 study, to accelerate development and approval of CERC-801 via the 505(b)
(2) pathway.

Additionally, the Company expects to file an IND application with the FDA for CERC-802 in 2019 and expects to file an IND

application with the FDA for CERC-803 in 2020.

Recent Financings

During the first quarter of 2019, the Company closed on an underwritten public offering of common stock for 1,818,182 shares of
common  stock  of  the  Company,  at  a  price  to  the  public  of  $5.50  per  share  ("public  price").  Armistice  Capital  Master  Fund  Ltd.
("Armistice")  participated  in  the  offering  by  purchasing  363,637  shares  of  common  stock  of  the  Company  from  the  underwriter  at  the
public  price. The  gross  proceeds  to  the  Company,  before  deducting  underwriting  discounts  and  commissions  and  estimated  offering
expenses and assuming no exercise of the option to purchase additional shares of common stock, were approximately $10.0 million. The
net proceeds were approximately $9.0 million.

During the fourth quarter of 2018, Armistice exercised warrants and acquired an aggregate of 2,857,143 shares of the Series B

Convertible Preferred Stock, which can be converted to 14,285,715 shares of common stock, for net proceeds of approximately $5.7
million. Additionally, as part of this transaction, the Company issued warrants for 4,000,000 shares of common stock (see "December 2018
Armistice Private Placement" in Note 13 below for a description of this transaction).

During the third quarter of 2018, the Company entered into a securities purchase agreement with Armistice, pursuant to which the

Company sold 1,000,000 shares of the Company's common stock for net proceeds of approximately $3.9 million (see "Armistice Private
Placements" in Note 13 below for a description of this transaction).

Lachlan Pharmaceuticals

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In November 2017, the Company acquired TRx and its wholly-owned subsidiaries, including Zylera. The previous owners of TRx
beneficially own more than 10% of our outstanding common stock. Zylera, which is our wholly owned subsidiary, entered into the First
Amended and Restated Distribution Agreement with  Lachlan, effective December 18, 2015. Pursuant to the Lachlan Agreement, Lachlan
named Zylera as its exclusive distributor of Ulesfia in the United States and agreed to supply Ulesfia to Zylera exclusively for marketing
and sale in the United States.

Zylera is obligated to purchase a minimum of 20,000 units per year, or approximately $1.2 million worth of product, from
Lachlan, subject to certain termination rights. Zylera must pay Lachlan $58.84 per unit and handling fees that are equal to $3.66 per unit of
fully packaged Ulesfia in 2018, and escalate at a rate of 10% annually, as well as reimburse Lachlan for all product liability insurance fees
incurred by Lachlan. The Lachlan Agreement also requires that Zylera make certain cumulative net sales milestone payments and royalty
payments to Lachlan with a $3.0 million annual minimum payment unless and until there has been a “Market Change” involving a new
successful competitive product. Lachlan is obligated to pay identical amounts to an unrelated third party from which it obtained rights to
Ulesfia, with the payments ultimately flowing to Summers Laboratories, Inc. (“Summers Labs”). Because of the dispute described below,
the Company has not made any payments to Lachlan under the Lachlan Agreement subsequent to the acquisition date.

On December 10, 2016, Zylera informed Lachlan that a Market Change had occurred due to the introduction of Arbor

Pharmaceuticals' lice product, Sklice®.  On June 5, 2017, Lachlan and Zylera entered into joint legal representation along with other
unrelated third parties in negotiation and arbitration of a dispute with Summers Labs regarding the existence of a Market Change and the
concomitant obligations of the parties. The arbitration panel issued an interim ruling on October 23, 2018 that no market change had
occurred up to and including the date of the hearing. The arbitration panel issued a second interim ruling on December 26, 2018. The
second interim award rejected Summers Labs' request to accelerate future minimum royalties, however, it ruled in favor of Summers Labs
that it is owed reimbursement for all reasonable costs and expenses, including legal fees, by Shionogi, as well as interest, as stipulated in the
contract. The arbitration panel issued a final award on March 1, 2019 that dictated the final amount of reimbursable costs and interest as
contemplated in the second interim ruling. The final award has no direct bearing on the Company as the Company was not a named
defendant to the original claim by Summers Labs and a federal court denied Zylera's ability to be a counterclaimant in the matter.
Furthermore, the Company is not subject to the guarantee or interest provisions identified in the second ruling as these elements of the
contractual relationship were not passed down to the Company’s agreement with Lachlan. However, the Company has interpreted this
ruling's impact on the Lachlan agreement to mean that a market change has not occurred, and the minimum purchase obligation and
minimum royalty provisions of the contract are active and due for any prior periods as well as going forward for any future periods.

The Company has recognized a $7.8 million liability for these minimum obligations in accrued liabilities as of December 31,

2018. Under the terms of the TRx Purchase Agreement, the former TRx owners are required to indemnify the Company for 100% of all
pre-acquisition losses related this arbitration, including legal costs, and possible minimum payments in excess of $1 million. Furthermore,
the former TRx owners are required to indemnify the Company for 50% of post-acquisition Ulesfia losses, which would include losses
resulting from having to fund these minimum obligations. The Company has recorded an indemnity receivable of $4.9 million in other
receivables as of December 31, 2018, which the Company believes is fully collectible. The receivable is net of $1.9 million collection made
in the fourth quarter of 2018 from a full cash escrow release with the former TRx owners from the escrow that was established as a part of
the TRx acquisition. The post-acquisition minimum obligations net of amounts recorded within the indemnity receivable of $2.2 million
has been recorded in cost of product sales for the year ended December 31, 2018. If the Company fails to make these minimum obligations
timely then the Lachlan Agreement may be terminated by Lachlan, in which case the Company would no longer be able to sell the Ulesfia
product, but it would also not be subject to future minimum obligations. Lachlan has not requested payment for the minimum obligations.

Our Strategy

The Company is building a robust pipeline of innovative therapies in neurology, pediatric healthcare, and orphan rare diseases. We
plan to use the proceeds generated from the profits of our portfolio of pediatric products toward the development of drug candidates that
have  unique  mechanisms  of  action  and  can  change  the  lives  of  patients  with  rare  orphan  diseases  in  pediatrics  and  neurology. We
systematically identify and pursue potential development candidates, ideally those for which human proof of concept exists in the intended
indication, for either the target or the compound. We target conditions where current treatments fail to address unmet medical needs, and
where we believe we can apply clinical strategies to increase efficacy signal detection with a view to optimizing the clinical development
and regulatory pathway for our product candidates.

Our strategy for increasing shareholder value includes:

•

Advancing our pipeline of compounds through development and to regulatory
approval;

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•

•

•

Pursuing targeted, differentiated preclinical and clinical stage product
candidates;

Acquiring or licensing rights to clinically meaningful and differentiated products that are already on the market for pediatric use or
in late-stage development for pediatric indications; and

Growing sales of the existing commercial products in our portfolio, including by identifying and investing in growth opportunities
such as new treatment indications and new geographic markets.

Product Pipeline Assets

The following table summarizes key information about our product candidates and further detail regarding each product candidate

follows:

Neurology Pipeline Assets

•

CERC‑301:  Orphan  Neurological  Indication. CERC-301  is  currently  being  developed  as  an  adjunct  therapy  in  Parkinson’s
Disease patients suffering from nOH, which is a condition that is part of a larger category called orthostatic hypotension ("OH")
also  known  as  postural  hypotension. nOH  is  caused  by  dysfunction  in  the  autonomic  nervous  system  and  causes  people  to  feel
faint  when  they  stand  or  sit  up. CERC‑301 belongs to a class of compounds known as antagonists of the N‑methyl‑D‑aspartate
("NMDA")  receptor,  a  receptor  subtype  of  the  glutamate  neurotransmitter  system  that  is  responsible  for  controlling  neurologic
adaptation. We believe CERC‑301 selectively blocks the NMDA receptor subunit 2B ("NR2B") (also called GluN2B).

CERC‑301  has  been  shown  to  be  safe  and  well  tolerated  in  over  350  patients  and  healthy  volunteers  during  several  clinical
investigations. Throughout various trials, CERC-301 produced consistent and robust increases in blood pressure, which we believe
will  provide  long-term  clinical  benefit  of  reducing  the  frequency  and  severity  of  symptoms  associated  with  nOH. We  anticipate
progressing development into Phase 2 efficacy and dose ranging studies in nOH with the goal of obtaining the first chronic use label
with  symptomatic  benefit. Currently approved therapies for nOH, Nothera (droxidopa) and Midodrine, have conditional approval
(Sub-part H) and have not demonstrated and are not labeled for long-term

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•

•

clinical benefits. As such, we believe CERC-301 may be well suited to address unmet medical needs in neurologic indications.

While  listed  as  an  orphan  condition  affecting  less  than  200,000  patients  in  the  United  States,  nOH  results  from  failure  of  the
autonomic nervous system to regulate blood pressure in response to postural change, due to an inadequate release of norepinephrine.
This  leads  to  both  orthostatic  hypotension  upon  standing  and  supine  hypertension  when  lying.  nOH  is  a  hallmark  of  several
neurodegenerative diseases, including multiple systems atrophy, Parkinson’s disease, and primary autonomic failure.

CERC‑406  and  COMTi  Platform:  Adjunctive  Treatment  of  Parkinson's  Disease. CERC-406  is  a  preclinical  candidate  from
our proprietary platform of compounds that inhibit catechol-O-methyltransferase ("COMT") within the brain, which we refer to as
our  COMTi  platform.  We  believe  it  may  have  the  potential  to  be  developed  for  the  adjunct  treatment  of  Parkinson’s  Disease.
Preclinically,  CERC-406  has  demonstrated  a  greater  selectivity  for  Central  Nervous  System  COMT  as  compared  to  peripheral
COMT,  which  we  believe  may  represent  an  opportunity  to  treat  both  the  neuromuscular  and  cognitive  manifestations  of
Parkinson's Disease while minimizing the systemic toxicities associated with the currently approved COMTi’s.

COMT  is  an  enzyme  that  is  critical  for  the  inactivation  and  metabolism  of  dopamine  and  its  inhibition  in  the  brain  has  potential
applicability  in  treating  subjects  with  neuropsychiatric  conditions,  including  major  depressive  disorder  ("MDD"),  schizophrenia,
Parkinson’s Disease and pathological gambling. CERC-406 is our first preclinical candidate from the COMTi platform, specifically
designed to preferentially inhibit Central Nervous System COMT over peripheral COMT.

COMT  inhibitors  have  shown  to  be  clinically  effective  in  increasing  the  “on”  and  decreasing  the  “off”  times  of
levodopa/decarboxylase  inhibitor  therapy  in  PD  patients. Tolcapone  is  the  only  approved  COMTi  that  crosses  the  blood  brain
barrier  but  is  associated  with  serious  liver  toxicities. In  preclinical  testing,  CERC-406  had  a  lower  potential  for  peripheral  (non-
CNS) side effects, rapid absorption and bioavailability, good brain penetration and a favorable dose dependent biomarker profile.
We have also observed in rats, that CERC-406 appears to have an “off rate” on brain COMT that is slower than tolcapone, implying
it may have a superior duration of effect.

Similarly, CERC-425 is an orally active small molecule, COMT inhibitor. The Company has de-prioritized the development of
CERC-425 in order to focus on CERC-406, as described above.

CERC-611:  Adjunctive  Treatment  of  Partial-Onset  Seizures  in  Epilepsy. CERC-611  is  a  potent  and  selective  antagonist  of
transmembrane alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid ("AMPA") receptor regulatory protein (“TARP”)-γ8-
dependent AMPA  currently  in  development  as  an  adjunct  therapy  for  refractory  partial-onset  seizures.  TARPs  are  a  recently
discovered family of proteins that have been found to associate with, and modulate the activity of, AMPA receptors. TARP γ8-
dependent AMPA receptors are localized primarily in the hippocampus, a region of the brain with importance in complex partial
seizures and particularly relevant to seizure origination and/or propagation.

We believe CERC-611 is the first drug candidate to selectively target and functionally block region-specific AMPA receptors after
oral dosing, which we believe may improve the efficacy and side effect profile of CERC-611 over current anti-epileptics. Research
also suggests that selectively targeting individual TARPs may enable selective modulation of specific brain circuits without globally
affecting synaptic transmission. The clinical strategy for CERC-611 is currently being reevaluated due to a partial clinical hold.  The
exposure limits imposed by the agency currently allows for subtherapeutic dosing.  We are investigating opportunities to broaden
the exposure limits. We intend to develop CERC-611 as an adjunctive therapy for the treatment of partial-onset seizures in patients
with epilepsy.

Pediatric Rare Orphan Disease Pipeline Assets

•

CERC-800 Series (CERC-801, CERC-802, and CERC-803): Substrate Replacement Therapies for CDGs. CERC-801, CERC-
802  and  CERC-803  represent  genetically-targeted,  small  molecule,  substrate  replacement  therapies  with  established  therapeutic
utility  for  the  treatment  of  CDGs.  CDGs  are  a  rapidly  expanding  group  of  rare  Inborn  Errors  of  Metabolism  ("IEMs")  due  to
defects  in  glycosylation.  Glycosylation  is  the  process  by  which  carbohydrate  complexes  are  created,  modified  and  attached  to
proteins  and  lipids,  creating  glycoconjugates  that  are  essential  for  cell  structure  and  function  in  all  tissues  and  organs.  CDG  is
caused by a specific inherited mutation and more than 100 CDGs have been identified to date. CDGs typically present in infancy
and  can  be  associated  with  a  broad  spectrum  of  symptoms  that  include  severe,  disabling  or  life-threatening  cases.  Oral
administration of CERC-801, CERC-802 or CERC-803 can replenish critical metabolic intermediates that are reduced or absent
due to genetic mutation, overcoming single enzyme

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defects to support glycoprotein synthesis, maintenance and function. CERC-801 utilizes D-galactose as the active pharmaceutical
ingredient  to  treat  Phosphoglucomutase  1  (PGM1)  Deficiency;  CERC-802  utilizes  D-mannose  as  the  active  pharmaceutical
ingredient to treat Mannose-Phosphate Isomerase (MPI) Deficiency; and CERC-803 utilizes L-fucose as the active pharmaceutical
ingredient to treat Leukocyte Adhesion Deficiency Type II (LADII).

The FDA has granted Rare Pediatric Disease Designation and Orphan Drug Designation to CERC-801, CERC-802 and CERC-803. 
Under the FDA’s PRV program, upon the approval of an NDA for the treatment of a rare pediatric disease, the sponsor of such
application would be eligible for a PRV that can be used to obtain priority review for a subsequent new drug application or biologics
license application. The PRV may be sold or transferred an unlimited number of times. Furthermore, we plan to leverage the 505(b)
(2) NDA pathway for all three compounds to accelerate development and approval.

The below chart depicts the benefits associated with ODD and RPDD for each of the CERC-800 series compounds:

•

CERC-913: ProTide Nucleotide for Mitochondrial Disorder. CERC-913 is a genetically-targeted, small molecule substrate
replacement therapy that uses a prodrug approach to overcome a single enzyme defect to treat mitochondrial DNA mtDNA
depletion syndromes ("MDS"). A prodrug is a medication or compound that, after administration, is metabolized into a
pharmacologically active substance. The ProTide prodrug platform is a clinically-validated approach to nucleoside
monophosphate prodrugs. Some patients suffering from MDS lack a nucleoside kinase that produces nucleoside monophosphates
for mtDNA synthesis. Direct substrate replacement of nucleoside monophosphates is impractical due to instability in plasma and
low cell permeability. By masking a nucleoside monophosphate as a prodrug with improved drug-like properties, we can deliver
the substrate to the desired subcellular compartment and bypass the missing nucleoside kinase. CERC-913 is intended for pediatric
MDS patients with symptoms that manifest primarily in the liver, with 50% of patients experiencing liver failure in the first few
years of life.

Commercially Marketed Products

•

•

Poly-Vi-Flor: This  medication  is  a  combination  product  of  vitamins  and  fluoride.  It  is  used  in  infants  and  children  to  treat  or
prevent deficiency due to poor diet or low levels of fluoride in drinking water and other sources. Vitamins are important building
blocks of the body and help keep you in good health. Fluoride is used to prevent dental cavities.

Tri-Vi-Flor:  Multivitamins  provide  essential  vitamins  and  minerals  that  are  not  taken  in  to  the  body  through  diet. Fluoride
strengthens  tooth  enamel,  which  helps  prevent  dental  cavities.  In  most  major  U.S.  communities,  fluoride  is  put  into  the  water
supply. Tri-Vi-Flor  are  used  as  a  supplement  to  the  diet  of  infants  and  children  who  do  not  receive  adequate  fluoride  through
drinking water. Tri-Vi-Flor are also used to prevent tooth decay in people treated with radiation, which may cause dryness of the
mouth and increased risk of tooth decay.

• Millipred®: Prednisolone is a man-made form of a natural substance (corticosteroid hormone) made by the adrenal gland. It is
used to treat conditions such as arthritis, blood problems, immune system disorders, skin and eye conditions, breathing problems,
cancer,  and  severe  allergies.  It  decreases  your  immune  system's  response  to  various  diseases  to  reduce  symptoms  such  as  pain,
swelling and allergic-type reactions. Supplied in 5mg tablets and 10mg in oral solution.

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•

Ulesfia®: Ulesfia® Lotion is indicated for the topical treatment of head lice infestation in patients six months of age and older.
This product is not toxic to lice but kills them by depriving them of oxygen.

• Karbinal™ ER: Carbinoxamine is an antihistamine used to relieve symptoms of allergy, hay fever, and the common cold. These
symptoms  include  rash,  watery  eyes,  itchy  eyes/nose/throat/skin,  cough,  runny  nose,  and  sneezing. This  medication  works  by
blocking  a  certain  natural  substance  (histamine)  that  your  body  makes  during  an  allergic  reaction.  By  blocking  another  natural
substance made by your body (acetylcholine), it helps dry up some body fluids to relieve symptoms such as watery eyes and runny
nose.

•

•

•

AcipHex® Sprinkle™: AcipHex® Sprinkle™ or Rabeprazole is used to treat certain stomach and esophagus problems (such as
acid  reflux,  ulcers).  It  works  by  decreasing  the  amount  of  acid  your  stomach  makes.  It  relieves  symptoms  such  as  heartburn,
difficulty swallowing, and persistent cough. This medication helps heal acid damage to the stomach and esophagus, helps prevent
ulcers, and may help prevent cancer of the esophagus. Rabeprazole belongs to a class of drugs known as proton pump inhibitors
("PPIs").

Cefaclor for Oral Suspension: This medication is a second-generation cephalosporin-type antibiotic used to treat a wide variety
of bacterial infections (e.g., middle ear, skin, urine and respiratory tract infections). It works by stopping the growth of bacteria.
This antibiotic only treats bacterial infections. It will not work for viral infections (e.g., common cold, flu). Unnecessary use or
overuse of any antibiotic can lead to its decreased effectiveness.

Flexichamber™: When a child is diagnosed with asthma, doctors often prescribe a metered dose inhaler ("MDI") - commonly
referred to as an inhaler. Using an inhaler requires refined coordination and inhalation techniques that can be tricky, especially for
small children. To ensure the child receives the optimal dose, many doctors prescribe a spacer - such as Flexichamber - to be used
with an inhaler. Flexichamber was designed to overcome problems that patients commonly experience when using just an inhaler
to  administer  their  asthma  medication.  When  used  properly  and  as  prescribed  by  a  doctor,  Flexichamber  helps  deliver  asthma
medication from the inhaler to tissue deep within the lungs, reduces the amount of medication that settles onto the child’s mouth
and throat, and allows caregivers to visually monitor breathing techniques and provide additional instructions if needed.

Intellectual Property

Our success depends in part on our ability to obtain and maintain proprietary protection for the technology and know-how upon
which  our  products  are  based,  to  operate  without  infringing  the  proprietary  rights  of  others  and  to  prevent  others  from  infringing  our
proprietary rights.

We  hold  ownership,  trademark  rights  and/or  exclusivity  to  develop  and  commercialize  our  products  and  product  candidates
covered  by  patents  and  patent  applications. Our  portfolio  of  patents  includes  patents  or  patent  applications  with  claims  directed  to
compositions of matter, including compounds, pharmaceutical formulations, methods of use, methods of manufacturing the compounds, or
a combination of these claims. Depending upon the timing, duration and specifics of FDA approval of the use of a compound for a specific
indication, some of our U.S. patents may be eligible for a limited patent term extension under the Drug Price Competition and Patent Term
Restoration Act of 1984, referred to as the Hatch-Waxman Act.  Similar extensions to patent term may be available in other countries for
particular patents in Cerecor’s portfolio.

The patent portfolios for our most advanced programs are summarized below:

• CERC‑301: Orphan Neurological Indication. We possess worldwide exclusive rights to manufacture, use, and sell certain
NR2B  antagonist  compounds. The  CERC‑301  patent  portfolio  consists  of  three  patent  families. The  first  family  consists  of
patents that have issued in the United States, Germany, France, and United Kingdom. The patents in the first family include
composition  of  matter  claims  and  use  claims  that  generically  cover  CERC‑301. The  expiration  date  of  the  U.S.  patent  is
June 3, 2022, not including any potential patent term extension or market exclusivity period. The  second  family  consists  of
patents that have issued in United States, Australia, Canada, Germany, France, Switzerland, United Kingdom, and Japan.  The
patents in the second family include composition of matter and use claims of varying scope (foreign patents only), including
picture claims to CERC‑301 or a pharmaceutically acceptable salt thereof. The expiration date of the U.S. patent in the second
family is August 31, 2026, not including any patent term extension or market exclusivity period which may apply.  The third
family consists of a patent issued in the United States and patent applications in the United States, Australia, Canada, China,
Europe, India, and Japan, with claims to compositions of matter, methods of use, and methods of manufacture that cover the
crystalline form of CERC-301. The expiration date of the U.S. patent is December 18, 2035 and any patents

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issuing  from  the  pending  applications  would  expire  on  December  18,  2035  at  the  earliest,  not  including  any  potential  patent
term adjustment, patent term extension, or market exclusivity period.

• CERC‑406 and COMTi Platform:  Adjunctive Treatment of Parkinson's Disease.  We possess worldwide exclusive rights
to manufacture, use, and sell COMT inhibitor compounds. The  COMT  patent  portfolio  consists  of  two  patent  families. The
first family consists of patents that have issued in the United States, Australia, Canada, China, Japan, and patent applications
in Europe and India with claims to compositions of matter and methods of use. The expiration date of the United States patent
in the first family, exclusive of any patent term extension, is February 28, 2031.  The second family consists of patents that
have issued in the United States, Australia, China, Europe, Japan, and patent applications in Canada and India with claims to
compositions  of  matter  and  methods  of  use. The  expiration  date  of  the  U.S.  patent  in  the  second  family,  exclusive  of  any
patent term extension, is February 28, 2031.

• CERC-611: Adjunctive  Treatment  of  Partial-Onset  Seizures  in  Epilepsy. We  possess  worldwide  exclusive  rights  to
manufacture,  use,  and  sell  LY3130481,  now  known  as  CERC‑611.    The  CERC-611  patent  portfolio  consists  of  two  patent
families. The  first  family  consists  of  patents  that  have  issued  in  the  United  States,  Australia,  Canada,  China,  France,
Germany, Italy, Spain, Switzerland, United Kingdom, Japan, and a patent application in India with composition of matter and
use  claims  for  CERC-611.    The  expiration  date  of  the  United  States  patent,  exclusive  of  any  patent  term  extension,  is
November  20,  2033.    The  second  family  consists  of  patents  that  have  issued  in  the  United  States, Australia,  Canada,  and
Japan, and international patent applications in China (allowed) and India with composition of matter and use claims of varying
scope  for  additional  selective  TARP  γ8-dependent  AMPA  receptor  antagonists.    The  expiration  date  of  the  U.S.  patent,
exclusive of any patent term extension, is May 21, 2035.

• CERC-913: ProTide Nucleotide for Mitochondrial Disorder. The CERC-913 patent portfolio consists of patent applications
in the United States, Australia, Canada, China, Europe, India, and Japan with claims to compositions of matter and methods of
use. Any  patents  issuing  from  these  applications  would  expire  in  November  16,  2036  at  the  earliest,  not  including  any
potential patent term adjustment, patent term extension, or market exclusivity period.

•

Flexichamber. The  Flexichamber  patent  portfolio  consists  of  patents  that  have  issued  in  the  United  States, Australia  and
Japan,  and  patent  applications  in  the  United  States, Australia,  Canada,  China,  Europe,  and  India  with  claims  to  the  device,
methods  for  forming  the  device,  and  methods  of  use. The  expiration  date  of  the  U.S.  patent,  exclusive  of  any  patent  term
extension, is June 23, 2034.

We  are  actively  seeking  to  augment  our  portfolio  of  compounds  by  focusing  on  the  development  of  new  chemical  entities
("NCEs"), which have not previously received FDA approval. Upon approval by the FDA, NCEs are entitled to market and data exclusivity
in the United States with respect to generic drug competition for a period of five years from the date of FDA approval, even if the related
patents have expired.

Manufacturing

We do not have any manufacturing facilities or personnel. We rely on contract manufacturing organizations ("CMOs") to produce
our drug candidates in accordance with applicable provisions of the FDA’s current Good Manufacturing Practice ("GMP") regulations for
use in our clinical studies. The manufacture of pharmaceuticals is subject to extensive GMP regulations, which impose various procedural
and documentation requirements and govern all areas of record keeping, production processes and controls, personnel and quality control.

Sales and Marketing

We promote our commercially marketed products through a sales force of 42 territory managers. During the third quarter of 2018,
the  Company  initiated  an  expansion  of  the  sales  force,  which  is  expected  to  be  largely  completed  during  the  first  quarter  of  2019.
Additionally,  during  the  fourth  quarter  of  2018,  we  collaborated,  on  a  limited  basis,  with  a  third-party  sales  force  to  market  specific
products  to  health  care  professionals. In  the  future,  we  may  collaborate  with  a  third-party  sales  force  to  market  specific  products  on  a
limited  basis. Our  team  is  comprised  of  a  complete  support  staff  internally  and  we  also  partner  with  numerous  world  class  vendors  to
increase our effectiveness and efficiency.

     As pediatric specialists, our reach and frequency with key physicians and pharmacies is data driven to maximize our coverage of these
important healthcare professionals. With established commercial operations, the Company is poised to be both flexible and scalable based
on opportunities within the market.

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For our neurology pipeline assets (CERC-301, CERC-406 and CERC-611), we intend to selectively retain commercialization or
co‑commercialization  rights  in  the  United  States. We  may  complement  with  co-development  and  or  co‑promotion  agreements  with
partners.  For  those  product  candidates  for  which  we  receive  marketing  approval,  we  will  evaluate  expanding  our  sales  force  into  other
specialty markets. We may also collaborate with third parties to market the approved product candidates in the United States. We may also
seek to commercialize any of our approved products outside of the United States and may do so either through an expansion of our sales
force or through collaboration with third parties.

For our pediatric rare orphan disease pipeline assets (CERC-800 series and CERC-913), we intend to retain commercialization in
the United States. We may complement with co‑promotion agreements with partners in and outside the United States. We may also seek to
commercialize any of our approved products outside of the United States and may do so either through an expansion of our sales force or
through collaboration with third parties.

Competition—Pipeline Assets

We face, and will continue to face, intense competition from pharmaceutical and biotechnology companies, as well as numerous
academic and research institutions and governmental agencies, both in the United States and abroad. We compete, or will compete, with
existing  and  new  products  being  developed  by  our  competitors.  Some  of  these  competitors  are  pursuing  the  development  of
pharmaceuticals that target the same diseases and conditions that our research and development programs target.

Competition—Neurology Pipeline Assets

•

•

•

CERC‑301: Orphan Neurological Indication. CERC‑301 will compete with other drugs used as therapies for the treatment of
nOH.  Medication  management  of  nOH  is  added  when  patients  have  persistent  symptoms  despite  these  non-pharmacological
approaches. Fludrocortisone is a synthetic mineralocorticoid that acts to retain sodium and water. Midodrine is an alpha-adrenergic
agonist that can increase blood pressure by increasing peripheral vascular resistance. Pyridostigmine has also been used to treat
nOH. Pyridostigmine is a peripheral inhibitor of acetylcholinesterase, which can cause a mild increase in standing blood pressure
without  significantly  increasing  supine  blood  pressure.  Droxidopa  (L-threo-3-4-dihydroxyphenylserine  ("L-threo  DOPS"))  is  an
oral prodrug converted by decarboxylation to norepinephrine in both the central and the peripheral nervous systems.

CERC-406  and  COMTi  Platform: Adjunctive  Treatment  of  Parkinson's  Disease. There  are  no  approved  pharmacologic
treatments for cognitive impairment associated in the U.S. at this time. In March 2015, vortioxetine (Brintellix®), marketed in the
United  States  by  Lundbeck  Pharmaceuticals,  which  was  originally  developed  and  commercialized  for  the  treatment  of  MDD,
received  a  positive  opinion  from  the  Committee  for  Medicinal  Products  for  Human  Use  of  the  European  Medicines Agency  to
expand  the  label  to  include  information  for  cognitive  function  in  patients  with  depression. A  supplemental  application  for  the
addition of clinical data to the FDA approved product label for Brintellix was not approved by the FDA.

Our potential products for the treatment of the cognitive and motoric impairment of Parkinson’s disease may compete with existing
COMT inhibitors Comtan (entacapone), marketed by Novartis Pharmaceuticals Corp. ("Novartis") (licensed from Orion), Tasmar
(tolcapone),  marketed  by  Valeant,  and  Stalevo  (fixed  combinations  of  entacapone  and  levodopa/carbidopa),  also  marketed  by
Novartis  (licensed  from  Orion).  Comtan,  Tasmar,  and  Stalevo  are  all  generic  in  the  United  States.  Currently,  no  treatments  are
approved for cognitive impairment in Parkinson’s disease.

CERC-611: Adjunctive Treatment of Partial-Onset Seizures in Epilepsy.  The epilepsy market is crowded with current therapies
targeting  a  variety  of  mechanisms,  including  gamma-aminobutyric  acid  ("GABA")  receptor  agonism,  T-type  calcium  channel
blockers,  sodium  channel  modulators,  synaptic  vesicle  protein  SV2A  modulation,  and  inhibition  of  GABA  transaminase.  More
recently, a new class of AMPA receptor antagonists have been approved for the treatment of epilepsy.

CERC-611, if we are successful in developing it and it gains regulatory approval, would compete with a number of branded and
generic  anti-epileptic  drugs. A  few  major  pharmaceutical  companies  (GSK  (Lamictal/XR),  Pfizer  (Lyrica))  and  specialty  players
(UCB  (Vimpat,  Keppra),  Lundbeck  (Sabril)  and  Supernus  (Trokendi  XR))  dominate  the  anti-epilepsy  drug  therapy  market.  New
market  entrants  such  as  Sage  Pharmaceuticals  and  GW  Pharmaceuticals  are  targeting  difficult  to  treat  orphan  patient  populations
such  as  super-refractory  status  epilepticus  and  Dravet  Syndrome,  respectively.  To  our  knowledge,  there  are  no  other  TARP  γ-8-
dependent AMPA receptor antagonist s in development other than CERC-611.

Competition—Pediatric Rare Orphan Disease Pipeline Assets

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•

•

CERC‑800 series (CERC-801, CERC-802 and CERC-803): Substrate Replacement Therapy for CDGs. Currently there are no
FDA or EMEA approved products for the treatment of CDG using the following: D-Galactose Substrate replacement therapy for
PGM1  CDG  (CERC-801),  Mannose  Phosphate  Isomerase  ("MPI")  deficiency,  also  known  as  MPI-CDG  (CERC-802),  and  L-
Fucose  Substrate  replacement  therapy  for  the  treatment  of  Leukocyte  Adhesion  Deficiency  Type  II  (LADII),  also  known  as
SLC35C1-CDG (CERC-803).

CERC-913: ProTide  Nucleotide  for  Mitochondrial  Disorder. Currently there are no FDA or EMEA approved products for the
treatment  of  Mitochondrial  Depletion  Syndrome  MDA  using  a  ProTide  Nucleotide  therapy  for  Mitochondrial  DNA  Depletion
Syndrome ("MDS").

Competition—Commercially Marketed Products

Across  all  our  product  lines  there  is  over-the-counter  ("OTC")  branded  and  generic  competition. However,  we  believe  our
products  do  have  significant  aspects  of  clinical  and  competitive  differentiation  in  the  marketplace  that  allows  us  to  effectively  market,
compete and grow market share in the face of competition.

•

Poly-Vi-Flor  /  Tri-Vi-Flor:  Poly-Vi-Flor  /  Tri-Vi-Flor  primarily  compete  against  generic  prescription  multi-vitamin  fluoride
market  and  the  brands  of  FLORIVA  and  QFLORA.  Our  primary  point  of  differentiation  is  Metafolin  and  that  our  form  of
Metafolin is a body-ready folate to aid in cell reproduction. As well, we offer formulations that are patient friendly in terms of size
of tablet and taste of medication ensuring compliance of their daily fluoride vitamin supplementation.

• Millipred®: Millipred®  Tablets  primarily  compete  in  the  generic  prednisolone  market. We  believe  our  primary  point  of
differentiation is that we offer the lowest strength prednisolone in the market place allowing HCPs greater flexibility when dosing
a  glucocorticoid  steroid  across  a  variety  of  pediatric  indications. Additionally,  Millipred®  utilizes  the  proprietary  double  taste-
masking technology to provide a pleasant grape taste with no bitterness, which makes the product easier to administer to children.

•

Ulesfia®: Ulesfia® competes in a market place that is primarily made up of step-wise therapy utilizing OTC remedies. Once into
the prescription marketplace Sklice® is the market leader differentiated primarily by pricing and contracting. However, Ulesfia is
the leader in providing a non-neuro toxic / non-pesticide for treating headlice.

• Karbinal™  ER: Karbinal™  ER  faces  competition  from  OTC  products  such  as  non-sedating  antihistamines,  sedating
antihistamines as well as nasal steroids. Karbinal’s greatest point of differentiation is our LIQUIDRX Technology that allows for
extended  release  and  flexible  BID  dosing. This  feature  makes  Karbinal  ER  the  only  BID  first  generation  antihistamine.
Additionally,  Karbinal  has  a  significant  anticholinergic  /  drying  effect  on  the  symptoms  associated  with  seasonal,  perennial,  as
well as vasomotor allergic rhinitis.

•

•

•

AcipHex® Sprinkle™: AcipHex® Sprinkle™ primarily faces competition from the OTC Proton Pump Inhibitors, however those
products  (Nexium  OTC  and  Prilosec  OTC)  are  not  indicated  for  children  less  than  18  years  of  age. In  the  branded  space  the
primary  competition  is  from  Nexium  Packets. We  clinically  differentiate AcipHex  Sprinkle  as  the  only  PPI  that  is  proven  to
demonstrate esophageal mucosal healing as determined by endoscopy in children less than 18 years of age.

Cefaclor  for  Oral  Suspension: Cefaclor  for  Oral  Suspension  faces  significant  competition  from  the  generic  antibiotics  of
amoxicillin  as  well  as  Omnicef  /  Ceftin. We  feel  our  keep  point  of  differentiation  is  through  our  clinical  positioning  for
appropriate patients who have failed first line therapies. Cefaclor is the best first choice as a second line treatment for antibiotics
that  have  failed  patients  suffering  from  streptococcus,  urinary  tract  infections  and  otitis  media. Cefaclor  is  a  second  generation
antibiotic indicated against a broad range of pathogens with a broad range of indications.

Flexichamber™: Flexichamber™ is  a  patented  and  proprietary  design  that  allows  a  patient  with  a  necessary  spacer  that  is
conveniently  portable. There  are  numerous  competitors  in  the  market  place  with  the  main  competition  being  AreoChamber.
Flexichamber’s collapsibility / portability is unique compared to the competition.

Overall Competitive Climate and Risks

In addition, the companies described above and other competitors may have a variety of drugs in development or may be awaiting
FDA  approval  that  could  reach  the  market  and  become  established  before  we  have  a  product  to  sell.  Our  competitors  may  also  develop
alternative therapies that could further limit the market for any drugs that we may develop. Many of our

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competitors are using technologies or methods different or similar to ours to identify and validate drug targets and to discover novel small
compound drugs. Many of our competitors and their collaborators have significantly greater experience than we do in the following:

•

•

•

•

and 

validating

compounds 

identifying 
targets;
screening 
targets;
preclinical  and  clinical  trials  of  potential  pharmaceutical  products;
and
obtaining 
clearances.

regulatory

against

other 

FDA 

and 

In addition, many of our competitors and their collaborators have substantially greater advantages in the following areas:

•

•

capital
resources;
research 
resources; 
• manufacturing 

and 

development

capabilities;

•

and
sales 
marketing.

and

Smaller  companies  may  also  prove  to  be  significant  competitors,  particularly  through  proprietary  research  discoveries  and
collaborative  arrangements  with  large  pharmaceutical  and  established  biotechnology  companies.  Many  of  our  competitors  have  products
that have been approved or are in advanced development. We face competition from other companies, academic institutions, governmental
agencies  and  other  public  and  private  research  organizations  for  collaborative  arrangements  with  pharmaceutical  and  biotechnology
companies,  in  recruiting  and  retaining  highly  qualified  scientific  and  management  personnel  and  for  licenses  to  additional  technologies.
Our competitors, either alone or with their collaborators, may succeed in developing technologies or drugs that are more effective, safer,
and  more  affordable  or  more  easily  administered  than  ours  and  may  achieve  patent  protection  or  commercialize  drugs  sooner  than  us.
Developments by others may render our product candidates or our technologies obsolete. Our failure to compete effectively could have a
material adverse effect on our business.

For  additional  information  on  risks  regarding  our  competition,  refer  to  the  section  entitled  “Risk  Factors”  in  Item  1A  of  this

Annual Report Form 10-K.

Government Regulation and Product Approval

Government  authorities  in  the  United  States,  at  the  federal,  state  and  local  level,  and  in  other  countries  extensively  regulate,
among other things, the research, development, testing, manufacture, packaging, storage, recordkeeping, labeling, advertising, promotion,
distribution,  marketing,  import  and  export,  pricing,  and  government  contracting  related  to  pharmaceutical  products  such  as  those  we  are
developing.  The  processes  for  obtaining  marketing  approvals  in  the  United  States  and  in  foreign  countries,  along  with  subsequent
compliance with applicable statutes and regulations, require the expenditure of substantial time and financial resources.

United States Government Regulation

In the United States, the FDA regulates drugs under the Federal Food, Drug, and Cosmetic Act ("FDCA") and its implementing
regulations. The process of obtaining marketing approvals and the subsequent compliance with appropriate federal, state, local and foreign
statutes and regulations requires the expenditure of substantial time and financial resources. Failure to comply with the applicable United
States requirements at any time during the product development process, approval process or after approval, may subject an applicant to a
variety of administrative or judicial sanctions, or other actions, such as the FDA’s delay in review of or refusal to approve a pending NDA,
withdrawal of an approval, imposition of a clinical hold or study termination, issuance of Warning Letters or Untitled Letters, mandated
modifications  to  promotional  materials  or  issuance  of  corrective  information,  requests  for  product  recalls,  consent  decrees,  corporate
integrity agreements, deferred prosecution agreements, product seizures or detentions, refusal to allow product  import  or  export,  total  or
partial  suspension  of  or  restriction  of  or  imposition  of  other  requirements  relating  to  production  or  distribution,  injunctions,  fines,
debarment from government contracts and refusal of future orders under existing contracts, exclusion from participation in federal and state
healthcare programs, FDA debarment, restitution, disgorgement or civil or criminal penalties, including fines and imprisonment.

FDA Marketing Approval

Obtaining  FDA  marketing  approval  for  new  products  may  take  many  years  and  require  the  expenditure  of  substantial  financial
resources. In order for FDA to determine that a product is safe and effective for the proposed indication, the product must first undergo
testing in animals (preclinical studies). The data generated from preclinical studies is used to support the filing of an

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IND Application under which human studies are conducted. There are three phases of human testing generally conducted under an IND,
following GCP guidelines:

•

•

•

Phase  1  studies  evaluate  the  safety  of  the  drug,  generally  in  normal,  healthy
volunteers;
Phase  2  studies  evaluate  safety  and  efficacy,  as  well  as  explore  dosing  ranges;  these  studies  are  typically  conducted  in
patient volunteers who suffer from the particular disease condition that the drug is designed to treat; and
Phase 3 studies evaluate safety and efficacy of the product, at specific doses, in a large clinical
trial

In addition to human testing in clinical studies, the manufacturing process (Chemistry, Manufacturing and Controls ("CMC")) of
the potential product must be developed in accordance with FDA cGMP regulations. Prior to the approval of a new product, The FDA will
inspect the facilities at which the proposed drug product is manufactured, to ensure cGMP compliance.

The  safety  and  efficacy  data  generated  from  the  clinical  study  phases  described  above,  CMC  information,  animal  data  and
proposed  labeling  are  used  as  the  basis  to  support  a  NDA  submission  to  FDA.  The  preparation  of  an  NDA  requires  the  expenditure  of
substantial  funds  and  the  commitment  of  substantial  resources. Additionally,  in  most  cases,  the  submission  of  an  NDA  is  subject  to  a
substantial application user fee, to be filed at the time of submission. The FDA conducts a preliminary review of all NDAs within the first
60 days after submission, before accepting them for filing and full review.

After evaluating the NDA and all related information, including the advisory committee recommendation, if any, and inspection
reports regarding the manufacturing facilities and clinical trial sites, the FDA may issue an approval letter, or, in some cases, a complete
response letter. A complete response letter generally contains a statement of specific conditions that must be met in order to secure final
approval  of  the  NDA  and  may  require  additional  clinical  or  preclinical  testing,  or  other  information,  in  order  for  FDA  to  reconsider  the
application.  The  FDA  has  a  review  goal  of  completing  its  review  of  90%  of  resubmissions  within  two  or  six  months  after  receipt,
depending on the type of information included. Even with submission of this additional information, the FDA ultimately may decide that
the application does not satisfy the regulatory criteria for approval. If and when those conditions have been met to the FDA’s satisfaction,
the  FDA  may  issue  an  approval  letter.  An  approval  letter  authorizes  commercial  marketing  of  the  drug  with  specific  prescribing
information for specific indications.

The  development  and  approval  of  new  drugs  requires  substantial  time,  effort  and  financial  resources.  Data  obtained  from  the
development  program  are  not  always  conclusive  and  may  be  susceptible  to  varying  interpretations.  These  instances  may  delay,  limit  or
prevent regulatory approval. The FDA may not grant approval on a timely basis, or at all. We may encounter difficulties or unanticipated
costs in our efforts to secure necessary governmental approvals, which could delay or preclude us from marketing our products. The FDA
may limit the indications for use or place other conditions on any approvals that could restrict the commercial application of the products.
After approval, some types of changes to the approved product, such as manufacturing changes and additional labeling claims, are subject
to further FDA review and approval.

FDA Post‑Approval Requirements

Drugs manufactured or distributed pursuant to FDA approvals are subject to continuing regulation by the FDA, including, among
other things, requirements relating to recordkeeping, manufacturing, periodic reporting, product sampling and distribution, advertising and
promotion,  and  reporting  of  adverse  experiences  with  the  product  and  drug  shortages.  After  approval,  most  changes  to  the  approved
product, such as adding new indications or other labeling claims are subject to prior FDA review and approval. There also are continuing,
annual user fee requirements for any marketed products and new application fees for supplemental applications with clinical data. The FDA
may  also  impose  post‑approval  requirements  as  a  condition  of  approval  of  an  NDA.  For  example,  the  FDA  may  require  post‑marketing
testing,  including  Phase  4  clinical  trials  and  surveillance  to  further  assess  and  monitor  the  product’s  safety  and  effectiveness  after
commercialization.  Once  an  approval  is  granted,  the  FDA  may  withdraw  the  approval  if  compliance  with  regulatory  requirements  and
standards is not maintained or if problems occur after the product becomes available in the market.

Additionally, the FDA strictly regulates the labeling, advertising and promotion of products under an approved NDA. The FDA
and other agencies actively enforce the laws and regulations prohibiting the promotion of off‑label uses, and a company that is found to
have improperly marketed or promoted off‑label uses may be subject to significant liability, including criminal and civil penalties under the
FDCA and False Claims Act, exclusion from participation in federal healthcare programs debarment from government contracts and refusal
of future orders under existing contracts, and mandatory compliance programs under corporate integrity agreements or deferred prosecution
agreements.

Other Regulations of the Healthcare Industry

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In addition to FDA regulations for the marketing of pharmaceutical products, there are various other state and federal laws that

may restrict business practices in the biopharmaceutical industry. These include the following:

•

•

•

•

•

•

The federal Medicare and Medicaid Anti-Kickback laws, which prohibit persons from knowingly and willfully soliciting,
offering, receiving or providing remuneration, directly or indirectly, in cash or in kind, to induce either the referral of an
individual,  or  furnishing  or  arranging  for  a  good  or  service,  for  which  payment  may  be  made  under  federal  healthcare
programs such as the Medicare and Medicaid programs;
Other Medicare laws, regulations, rules, manual provisions and policies that prescribe the requirements for coverage and
payment for services performed by our customers, including the amount of such payment;
The federal False Claims Act which imposes civil and criminal liability on individuals and entities who submit, or cause
to be submitted, false or fraudulent claims for payment to the government;
The  Foreign  Corrupt  Practices  Act  ("FCPA"),  which  prohibits  certain  payments  made  to  foreign  government
officials;
State  and  foreign  law  equivalents  of  the  foregoing  and  state  laws  regarding  pharmaceutical  company  marketing
compliance, reporting and disclosure obligations; and
The  Patient  Protection  and  Affordable  Care  Act  ("ACA"),  which  among  other  things  changes  access  to  healthcare
products and services; creates new fees for the pharmaceutical and medical device industries; changes rebates and prices
for health care products and services; and requires additional reporting and disclosure.

If our operations are found to be in violation of any of these laws, regulations, rules or policies or any other law or governmental
regulation, or if interpretations of the foregoing change, we may be subject to civil and criminal penalties, damages, fines, exclusion from
the Medicare and Medicaid programs and the curtailment or restructuring of our operations.

To the extent that any of our products are sold in a foreign country, we may be subject to similar foreign laws and regulations,
which  may  include,  for  instance,  applicable  post‑marketing  requirements,  including  safety  surveillance,  anti‑fraud  and  abuse  laws,  and
implementation  of  corporate  compliance  programs  and  reporting  of  payments  or  transfers  of  value  to  healthcare  professionals. This  is
currently not applicable as none of our products are currently sold in a foreign country.

Coverage and Reimbursement

The commercial success of our product candidates and our ability to commercialize any approved product candidates successfully
will depend in part on the extent to which governmental authorities, private health insurers and other third‑party payers provide coverage
for and establish adequate reimbursement levels for our therapeutic product candidates. In the United States, the European Union and other
potentially  significant  markets  for  our  product  candidates,  government  authorities  and  third‑party  payers  are  increasingly  imposing
additional  requirements  and  restrictions  on  coverage,  attempting  to  limit  reimbursement  levels  or  regulate  the  price  of  drugs  and  other
medical products and services, particularly for new and innovative products and therapies, which often has resulted in average selling prices
lower than they would otherwise be. For example, in the United States, federal and state governments reimburse covered prescription drugs
at varying rates generally below average wholesale price. Federal programs also impose price controls through mandatory ceiling prices on
purchases by federal agencies and federally funded hospitals and clinics and mandatory rebates on retail pharmacy prescriptions paid by
Medicaid and Tricare. These restrictions and limitations influence the purchase of healthcare services and products. Legislative proposals to
reform healthcare or reduce costs under government programs may result in lower reimbursement for our product candidates or exclusion
of our product candidates from coverage. Moreover, the Medicare and Medicaid programs increasingly are used as models for how private
payers and other governmental payers develop their coverage and reimbursement policies.

In  addition,  the  increased  emphasis  on  managed  healthcare  in  the  United  States  and  on  country  and  regional  pricing  and
reimbursement controls in the European Union will put additional pressure on product pricing, reimbursement and utilization, which may
adversely  affect  our  future  product  sales  and  results  of  operations.  These  pressures  can  arise  from  rules  and  practices  of  managed  care
groups, competition within therapeutic classes, availability of generic equivalents, judicial decisions and governmental laws and regulations
related to Medicare, Medicaid and healthcare reform, coverage and reimbursement policies and pricing in general. The cost containment
measures  that  healthcare  payers  and  providers  are  instituting  and  any  healthcare  reform  implemented  in  the  future  could  significantly
reduce our revenues from the sale of any approved product candidates. We cannot provide any assurances that we will be able to obtain and
maintain third‑party coverage or adequate reimbursement for our product candidates in whole or in part.

Impact of Healthcare Reform on Coverage, Reimbursement, and Pricing

The Medicare Prescription Drug, Improvement, and Modernization Act of 2003 ("the MMA") imposed new requirements for the

distribution and pricing of prescription drugs for Medicare beneficiaries. Under Part D, Medicare beneficiaries may enroll

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in prescription drug plans offered by private entities that provide coverage of outpatient prescription, pharmacy drugs pursuant to federal
regulations.  Part  D  plans  include  both  standalone  prescription  drug  benefit  plans  and  prescription  drug  coverage  as  a  supplement  to
Medicare Advantage plans. Unlike Medicare Part A and B, Part D coverage is not standardized. In general, Part D prescription drug plan
sponsors have flexibility regarding coverage of Part D drugs, and each drug plan can develop its own drug formulary that identifies which
drugs  it  will  cover  and  at  what  tier  or  level.  However,  Part  D  prescription  drug  formularies  must  include  drugs  within  each  therapeutic
category and class of covered Part D drugs, though  not  necessarily  all  the  drugs  in  each  category  or  class,  with  certain  exceptions. Any
formulary used by a Part D prescription drug plan must be developed and reviewed by a pharmacy and therapeutic committee. Government
payment  for  some  of  the  costs  of  prescription  drugs  may  increase  demand  for  any  products  for  which  we  receive  marketing  approval.
However,  any  negotiated  prices  for  our  future  products  covered  by  a  Part  D  prescription  drug  plan  will  likely  be  discounted,  thereby
lowering  the  net  price  realized  on  our  sales  to  pharmacies.  Moreover,  while  the  MMA  applies  only  to  drug  benefits  for  Medicare
beneficiaries,  private  payers  often  follow  Medicare  coverage  policy  and  payment  limitations  in  setting  their  own  payment  rates.  Any
reduction in payment that results from Medicare Part D may result in a similar reduction in payments from non‑governmental payers.

The American Recovery and Reinvestment Act of 2009 provides funding for the federal government to compare the effectiveness
of different treatments for the same illness. A plan for the research will be developed by the Department of Health and Human Services,
the Agency for Healthcare Research and Quality and the National Institutes for Health, and periodic reports on the status of the research and
related expenditures will be made to Congress. Although the results of the comparative effectiveness studies are not intended to mandate
coverage policies for public or private payers, it is not clear what effect, if any, the research will have on the sales of any product, if any
such product or the condition that it is intended to treat is the subject of a study. It is also possible that comparative effectiveness research
demonstrating  benefits  in  a  competitor’s  product  could  adversely  affect  the  sales  of  our  product  candidates.  If  third‑party  payers  do  not
consider our product candidates to be cost‑effective compared to other available therapies, they may not cover our product candidates, once
approved,  as  a  benefit  under  their  plans  or,  if  they  do,  the  level  of  payment  may  not  be  sufficient  to  allow  us  to  sell  our  products  on  a
profitable basis.

The United States and some foreign jurisdictions are considering enacting or have enacted a number of additional legislative and
regulatory  proposals  to  change  the  healthcare  system  in  ways  that  could  affect  our  ability  to  sell  our  products  profitably. Among  policy
makers  and  payers  in  the  United  States  and  elsewhere,  there  is  significant  interest  in  promoting  changes  in  healthcare  systems  with  the
stated goals of containing healthcare costs, improving quality and expanding access. In the United States, the pharmaceutical industry has
been  a  particular  focus  of  these  efforts  and  has  been  significantly  affected  by  major  legislative  initiatives,  including,  most  recently,  the
Affordable Care Act, which became law in March 2010 and substantially changes the way healthcare is financed by both governmental and
private insurers. Among other cost containment measures, the Affordable Care Act establishes an annual, nondeductible fee on any entity
that  manufactures  or  imports  specified  branded  prescription  drugs  and  biologic  agents;  a  new  Medicare  Part  D  coverage  gap  discount
program; expansion of Medicaid benefits and a new formula that increases the rebates a manufacturer must pay under the Medicaid Drug
Rebate Program; and expansion of the 340B drug discount program that mandates discounts to certain hospitals, community centers and
other qualifying providers. In the future, there may continue to be additional proposals relating to the reform of the United States healthcare
system,  some  of  which  could  further  limit  the  prices  we  are  able  to  charge  or  the  amounts  of  reimbursement  available  for  our  product
candidates once they are approved.

The Foreign Corrupt Practices Act

The  FCPA  prohibits  any  U.S.  individual  or  business  from  paying,  offering,  or  authorizing  payment  or  offering  of  anything  of
value, directly or indirectly, to any foreign official, political  party  or  candidate  for  the  purpose  of  influencing  any  act  or  decision  of  the
foreign entity in order to assist the individual or business in obtaining or retaining business. The FCPA also obligates companies whose
securities are listed in the United States to comply with accounting provisions requiring the company to maintain books and records that
accurately and fairly reflect all transactions of the corporation, including international subsidiaries, and to devise and maintain an adequate
system of internal accounting controls for international operations. Activities that violate the FCPA, even if they occur wholly outside the
United States, can result in criminal and civil fines, imprisonment, disgorgement, oversight, and debarment from government contracts.

Exclusivity and Approval of Competing Products

Hatch‑Waxman Patent Exclusivity

In seeking approval for a drug through an NDA, applicants are required to list with the FDA each patent with claims that cover the
applicant’s product or a method of using the product. Upon approval of a drug, each of the patents listed in the application for the drug is
then published in the FDA’s Approved Drug Products with Therapeutic Equivalence Evaluations, commonly known as the Orange Book.
Drugs  listed  in  the  Orange  Book  can,  in  turn,  be  cited  by  potential  competitors  in  support  of  approval  of  an  abbreviated  new  drug
application ("ANDA") or 505(b)(2) NDA. Generally, an ANDA provides for marketing of a drug product

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that has the same active ingredients in the same strengths, dosage form and route of administration as the listed drug and has been shown to
be bioequivalent through in vitro or in vivo testing or otherwise to the listed drug. ANDA applicants are not required to conduct or submit
results  of  preclinical  or  clinical  tests  to  prove  the  safety  or  effectiveness  of  their  drug  product,  other  than  the  requirement  for
bioequivalence testing. Drugs approved in this way are commonly referred to as “generic equivalents” to the listed drug, and can often be
substituted by pharmacists under prescriptions written for the reference listed drug. 505(b)(2) NDAs generally are submitted for changes to
a previously approved drug product, such as a new dosage form or indication.

The ANDA or 505(b)(2) NDA applicant is required to provide a certification to the FDA in the product application concerning any
patents listed for the approved product in the FDA’s Orange Book, except for patents covering methods of use for which the applicant is
not seeking approval. Specifically, the applicant must certify with respect to each patent that:

•

•

•

•

has

listed 

patent 

the  required  patent  information  has  not  been
filed;
the 
expired;
the listed patent has not expired, but will expire on a particular date and approval is sought after patent expiration;
or
the  listed  patent  is  invalid,  unenforceable,  or  will  not  be  infringed  by  the  new
product.

Generally,  the ANDA  or  505(b)(2)  NDA  cannot  be  approved  until  all  listed  patents  have  expired,  except  when  the ANDA  or
505(b)(2) NDA applicant challenges a listed patent or if the listed patent is a patented method of use for which approval is not being sought.
A certification that the proposed product will not infringe the already approved product’s listed patents or that such patents are invalid or
unenforceable is called a Paragraph IV certification. If the applicant does not challenge the listed patents or does not indicate that it is not
seeking approval of a patented method of use, the ANDA or 505(b)(2) NDA application will not be approved until all the listed patents
claiming the referenced product have expired.

If  the ANDA  or  505(b)(2)  NDA  applicant  has  provided  a  Paragraph  IV  certification  to  the  FDA,  the  applicant  must  also  send
notice of the Paragraph IV certification to the NDA and patent holders once the application has been accepted for filing by the FDA. The
NDA  and  patent  holders  may  then  initiate  a  patent  infringement  lawsuit  in  response  to  the  notice  of  the  Paragraph  IV  certification.  The
filing of a patent infringement lawsuit within 45 days after the receipt of notice of the Paragraph IV certification automatically prevents the
FDA  from  approving  the ANDA  or  505(b)(2)  NDA  until  the  earlier  of  30  months,  expiration  of  the  patent,  settlement  of  the  lawsuit,  a
decision in the infringement case that is favorable to the ANDA applicant or other period determined by a court.

Hatch‑Waxman Non‑Patent Exclusivity

Market and data exclusivity provisions under the FDCA also can delay the submission or the approval of certain applications for
competing products. The FDCA provides a five‑year period of non‑patent data exclusivity within the United States to the first applicant to
gain approval of an NDA for a new chemical entity. A drug is a new chemical entity if the FDA has not previously approved any other new
drug containing the same active moiety, which is the molecule or ion responsible for the therapeutic activity of the drug substance. During
the exclusivity period, the FDA may not accept for review an ANDA or a 505(b)(2) NDA submitted by another company that contains the
previously approved active moiety. However, an ANDA or 505(b)(2) NDA may be submitted after four years if it contains a certification of
patent invalidity or non‑infringement.

The FDCA also provides three years of marketing exclusivity for an NDA, 505(b)(2) NDA, or supplement to an existing NDA or
505(b)(2)  NDA  if  new  clinical  investigations,  other  than  bioavailability  studies,  that  were  conducted  or  sponsored  by  the  applicant,  are
deemed by the FDA to be essential to the approval of the application or supplement. Three‑year exclusivity may be awarded for changes to
a  previously  approved  drug  product,  such  as  new  indications,  dosages,  strengths  or  dosage  forms  of  an  existing  drug.  This  three‑year
exclusivity covers only the conditions of use associated with the new clinical investigations and, as a general matter, does not prohibit the
FDA from approving ANDAs or 505(b)(2) NDAs for generic versions of the original, unmodified drug product. Five‑year and three‑year
exclusivity will not delay the submission or approval of a full NDA; however, an applicant submitting a full NDA would be required to
conduct  or  obtain  a  right  of  reference  to  all  of  the  preclinical  studies  and  adequate  and  well‑controlled  clinical  trials  necessary  to
demonstrate safety and effectiveness.

Pediatric Exclusivity. Pediatric exclusivity is another type of non‑patent marketing exclusivity in the United States and, if granted,
provides for the attachment of an additional six months of marketing protection to the term of any existing regulatory exclusivity, including
the non‑patent exclusivity period described above. This six‑month exclusivity may be granted if an NDA sponsor submits pediatric data
that fairly respond to a written request from the FDA for such data. The data do not need to show the product to be effective in the pediatric
population studied; rather, if the clinical trial is deemed to fairly respond to the FDA’s request, the additional protection is granted. This is
not a patent term extension, but it effectively extends the regulatory period during which the FDA cannot approve an ANDA or 505(b)(2)
application owing to regulatory exclusivity or listed patents.

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Orphan  Drug  Designation  and  Exclusivity.  The Orphan Drug Act provides incentives for the development of drugs intended to
treat rare diseases or conditions, which generally are diseases or conditions affecting less than 200,000 individuals annually in the United
States, or affecting more than 200,000 in the United States and for which there is no reasonable expectation that the cost of developing and
making the drug available in the United States will be recovered from United States sales. Additionally, sponsors must present a plausible
hypothesis for clinical superiority to obtain orphan designation if there is a drug already approved by the FDA that is intended for the same
indication and that is considered by the FDA to be the same drug as the already approved drug. Orphan drug designation entitles a party to
financial incentives such as opportunities for grant funding towards clinical study costs, tax advantages, and user‑fee waivers. In addition, if
a product receives FDA approval for the indication for which it has orphan designation, the product is generally entitled to orphan drug
exclusivity, which means the FDA may not approve any other application to market the same drug for the same indication for a period of
seven years, except in limited circumstances, such as a showing of clinical superiority over the product with orphan exclusivity.

Foreign Regulation

In  order  to  market  any  product  outside  of  the  United  States,  we  would  need  to  comply  with  numerous  and  varying  regulatory
requirements of other countries regarding drug development and commercialization. The approval process varies from country to country
and  can  involve  additional  product  testing  and  additional  administrative  review  periods.  The  time  required  to  obtain  approval  in  other
countries might differ from and be longer than that required to obtain FDA approval. Regulatory approval in one country does not ensure
regulatory approval in another, but a failure or delay in obtaining regulatory approval in one country may negatively impact the regulatory
process in others.

European Union Drug Approval Process

To  obtain  a  marketing  authorization  of  a  drug  in  the  European  Union,  we  may  submit  marketing  authorization  applications

("MAAs") either under the so‑called centralized or national authorization procedures.

Centralized procedure

The  centralized  procedure  provides  for  the  grant  of  a  single  marketing  authorization  following  a  favorable  opinion  by  the
European Medicines Agency ("EMA") that is valid in all European Union member states, as well as Iceland, Liechtenstein and Norway.
The centralized procedure is compulsory for medicines produced by specified biotechnological processes, products designated as orphan
medicinal products, and products with a new active substance indicated for the treatment of specified diseases, such as HIV/AIDS, cancer,
diabetes, neurodegenerative disorders or autoimmune diseases and other immune dysfunctions. The centralized procedure is optional for
products that represent a significant therapeutic, scientific or technical innovation, or whose authorization would be in the interest of public
health. Under the centralized procedure the maximum timeframe for the evaluation of an MAA by the EMA is 210 days, excluding clock
stops, when additional written or oral information is to be provided by the applicant in response to questions asked by the Committee of
Medicinal  Products  for  Human  Use  ("CHMP"). Accelerated  assessment  might  be  granted  by  the  CHMP  in  exceptional  cases,  when  a
medicinal  product  is  expected  to  be  of  a  major  public  health  interest,  particularly  from  the  point  of  view  of  therapeutic  innovation.  The
timeframe for the evaluation of an MAA under the accelerated assessment procedure is of 150 days, excluding stop‑clocks.

National authorization procedures

There are also two other possible routes to authorize medicinal products in several European Union countries, which are available

for investigational medicinal products that fall outside the scope of the centralized procedure:

•
Decentralized  procedure. Using the decentralized procedure, an applicant may apply for simultaneous authorization in
more than one European Union country of medicinal products that have not yet been authorized in any European Union country
and that do not fall within the mandatory scope of the centralized procedure.

•
Mutual  recognition  procedure. In  the  mutual  recognition  procedure,  a  medicine  is  first  authorized  in  one  European
Union Member State, in accordance with the national procedures of that country. Following this, further marketing authorizations
can  be  sought  from  other  European  Union  countries  in  a  procedure  whereby  the  countries  concerned  agree  to  recognize  the
validity of the original, national marketing authorization.

In the European Union, new products authorized for marketing (i.e., reference products) qualify for eight years of data exclusivity
and an additional two years of market exclusivity upon marketing authorization. The data  exclusivity  period  prevents  generic  applicants
from relying on the preclinical and clinical trial data contained in the dossier of the reference product when

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applying for a generic marketing authorization in the EU during a period of eight years from the date on which the reference product was
first authorized in the EU. The market exclusivity period prevents a successful generic applicant from commercializing its product in the
EU until ten years have elapsed from the initial authorization of the reference product in the EU. The ten‑year market exclusivity period
can be extended to a maximum of eleven years if, during the first eight years of those ten years, the marketing authorization holder obtains
an authorization for one or more new therapeutic indications which, during the scientific evaluation prior to their authorization, are held to
bring a significant clinical benefit in comparison with existing therapies.

Employees

As  of  December  31, 2018,  we  had  64  full‑time  employees,  five  of  whom  were  primarily  engaged  in  research  and  development
activities  and  47  were  engaged  in  commercialization  activities.  None  of  our  employees  is  represented  by  a  labor  union  or  covered  by  a
collective bargaining agreement. We consider our relationship with our employees to be good.

Corporate Information

We  were  incorporated  in  2011  and  commenced  operations  in  the  second  quarter  of  2011. Our  principal  executive  offices  are
located  at  540  Gaither  Road,  Suite  400,  Rockville,  Maryland  20850,  and  our  phone  number  is  (410)  522-8707. Our  website  address  is
www.cerecor.com. The information on, or that can be accessed through, our website is not part of this report.

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Item 1A. Risk Factors.

You should consider carefully the following information about t

he  risks  described  below,  together  with  the  other  information  contained  in  this  Annual  Report  on  Form  10-K  and  in  our  other  public
filings, in evaluating our business. If any of the following risks actually occurs, our business, financial condition, results of operations and
future growth prospects would likely be materially and adversely affected. In these circumstances, the market price of our warrants and
common stock would likely decline.

Risks Related to Our Business and Industry

Our success and revenue depend on two portfolios of products; if either is not successfully commercialized or if we do not acquire new
products, our revenue might not grow, which could affect our stock price.

We currently have rights to only two portfolios of commercial pharmaceutical products consisting of eight commercial assets,
those we acquired with TRx in November 2017 and Avadel’s pediatric products, which we acquired in February 2018. Our prospects over
the next three to five years are substantially dependent on the successful commercialization and growth of revenue from these products,
including their acceptance by the medical community and third-party payers as useful and cost-effective. We might be required to engage in
expensive advertising, educational programs, provide discounts or other means to market these products.

Even if our current products generate significant revenue and profits, our ability to increase revenue in the future will depend in
part  on  our  success  in  in-licensing  or  acquiring,  and  developing,  additional  pharmaceutical  products.  We  currently  intend  to  seek  to  in-
license  or  acquire  development  stage  compounds  and  commercialized  pharmaceutical  products,  focusing  on  the  pediatric  space.  These
kinds of compounds and pharmaceutical products might not be available to us on attractive terms.

Our  product  candidates  that  we  intend  to  commercialize  are  in  early  stages  of  development.  If  we  do  not  successfully  complete
preclinical testing and clinical development of our product candidates or experience significant delays in doing so, our business may be
materially harmed.

We  have  invested  a  significant  portion  of  our  efforts  and  financial  resources  in  the  identification  and  preclinical  and  clinical
development of product candidates. Our ability to increase product revenues will depend on our ability to advance our one clinical product
candidate  and  our  preclinical  product  candidates  into  clinical  development  and  successfully  complete  preclinical  testing  of  our  clinical
stage product candidates. The outcome of preclinical studies and Phase 1 clinical trials might not predict the success of future clinical trials.
Preclinical data are often susceptible to varying interpretations and analyses, and many companies that believed their product candidates
performed  satisfactorily  in  preclinical  studies  have  nonetheless  failed  in  clinical  development.  Our  inability  to  successfully  complete
development  of  our  product  candidates  could  result  in  additional  costs  to  us  relating  to  product  development  and  obtaining  marketing
approval and impair our ability to generate product revenues and commercialization and sales milestone payments and royalties on product
sales.

If clinical trials of our product candidates fail to demonstrate safety and efficacy to the satisfaction of regulatory authorities or do not
otherwise  produce  positive  results,  we  may  incur  additional  costs  or  experience  delays  in  completing,  or  ultimately  be  unable  to
complete, the development and commercialization of our product candidates.

Before  obtaining  required  approvals  from  regulatory  authorities  for  the  sale  of  future  product  candidates,  we  alone,  or  with  a
partner, must conduct extensive clinical trials to demonstrate the safety and efficacy of the product candidates in humans. Clinical testing is
expensive and difficult to design and implement, can take many years to complete and is uncertain as to outcome. A failure of one or more
clinical trials can occur at any stage of testing. The outcome of preclinical studies and early clinical trials might not predict the success of
later  clinical  trials,  and  interim  results  of  a  clinical  trial  do  not  necessarily  predict  final  results.  A  number  of  companies  in  the
pharmaceutical  and  biotechnology  industries  have  suffered  significant  setbacks  in  advanced  clinical  trials  due  to  lack  of  efficacy  or
unacceptable safety profiles, notwithstanding promising results in earlier trials. Our product candidates will require additional clinical and
preclinical  development,  management  of  clinical,  preclinical  and  manufacturing  activities,  regulatory  approval  in  multiple  jurisdictions,
obtaining manufacturing supply on our own or from a third party, expansion of our commercial organization, and substantial investment
and significant marketing efforts before we generate any revenues from sales of any of those product candidates approved for marketing.
We  do  not  know  whether  the  clinical  trials  we  or  our  partners  may  conduct  will  demonstrate  adequate  efficacy  and  safety  to  result  in
regulatory approval to market any of our product candidates in any particular jurisdiction or jurisdictions. If later stage clinical trials do not
produce favorable results, our ability to achieve regulatory approval for any of our product candidates would be adversely impacted.

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If  we  experience  delays  in  clinical  testing,  we  will  be  delayed  in  obtaining  regulatory  approvals  and  commercializing  our  product
candidates, our costs may increase and our business may be harmed.

We do not know whether any clinical trials will begin as planned, whether the design will be revised prior to or during conduct of
the  study,  completed  on  schedule  or  conducted  at  all.  Our  product  development  costs  will  increase  if  we  experience  delays  in  clinical
testing. Significant clinical trial delays also could shorten any periods during which we may have the exclusive right to commercialize our
product  candidates  or  allow  our  competitors  to  bring  products  to  market  before  we  do,  which  would  impair  our  ability  to  successfully
commercialize our product candidates and may harm our business, results of operations and prospects.

Events which may result in a delay or unsuccessful completion of clinical development include:

•

•

•

•

•

•

•

•

•

•

•

•

•

delays  in  reaching  an  agreement  with  or  failure  in  obtaining  authorization  from  the  FDA,  other  regulatory  authorities  or
institutional review boards, or IRBs, to commence or amend a clinical trial;

imposition of a clinical hold or trial termination following an inspection of our clinical trial operations or trial sites by the FDA
or other regulatory authorities, or due to concerns about trial design, or a decision by the FDA, other regulatory authorities,
IRBs or the company, or recommendation by a data safety monitoring board, to place the trial on hold or otherwise suspend or
terminate clinical trials at any time for safety issues or for any other reason;

delays in reaching agreement on acceptable terms with prospective contract research organizations ("CROs") and clinical trial
sites;

deviations  from  the  trial  protocol  by  clinical  trial  sites  and  investigators,  or  failing  to  conduct  the  trial  in  accordance  with
regulatory requirements;

failure  of  our  third  parties,  such  as  CROs,  to  satisfy  their  contractual  duties  or  meet  expected
deadlines;

failure  to  enter  into  agreements  with  third  parties  to  obtain  the  results  of  clinical
trials;

delays  in  the  importation  and  manufacture  of  clinical
supply;

delays  in  the  testing,  validation  and  delivery  of  the  clinical  supply  of  the  product  candidates  to  the  clinical
sites;

for clinical trials in selected subject populations, delays in identification and auditing of central or other laboratories and the
transfer and validation of assays or tests to be used to identify selected subjects;

delays  in  recruiting  suitable  subjects  to  participate  in  a
trial;

delays  in  having  subjects  complete  participation  in  a  trial  or  return  for  post‑treatment
follow‑up;

delays  caused  by  subjects  dropping  out  of  a  trial  due  to  side  effects  or  disease
progression;

delays  in  adding  new  investigators  and  clinical  trial
sites;

• withdrawal of clinical trial sites from our clinical trials as a result of changing standards of care or the ineligibility of a site to

participate in our clinical trials; or

•

changes  in  government  regulations  or  administrative  actions  or  lack  of  adequate  funding  to  continue  the  clinical
trials.

Any  inability  by  us  or  our  partners  to  timely  complete  clinical  development  could  result  in  additional  costs  to  us  relating  to
product  development  and  obtaining  marketing  approval  and  impair  our  ability  to  generate  product  revenues  and  commercialization  and
sales milestone payments and royalties on product sales.

If we are unable to enroll appropriate subjects in clinical trials, we will be unable to complete these trials on a timely basis or at all.

Identifying and qualifying subjects to participate in clinical trials of our product candidates is critical to our success. The timing of
our clinical trials depends on the speed at which we can recruit appropriate subjects to participate in testing our product candidates as well
as completion of required follow‑up periods. If subjects are unwilling to participate in our trials because of negative publicity from

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adverse events in the biotechnology industry or for other reasons, including competitive clinical trials for similar subject populations, the
timeline for recruiting subjects, conducting trials and obtaining marketing approval of potential products may be delayed.

Difficulty  or  delays  in  patient  recruitment  into  our  trials  could  result  in  increased  costs,  delays  in  advancing  our  product
development,  delays  in  testing  the  effectiveness  of  our  technology  or  termination  of  the  clinical  trials  altogether.  Many  factors  affect
subject enrollment, including:

•

•

•

•

•

•

•

•

•

•

•

•

•

size  and  nature  of 

the 
population;

the 

subject

the  number  and  location  of  clinical  sites  we
enroll;

the  proximity  of  subjects  to  clinical
sites;

perceived  risks  and  benefits  of  the  product  candidate  under
trial;

competition  with  other  companies  for  clinical  sites  or
subjects;

competing 
trials;

clinical

the  eligibility  and  exclusion  criteria  for  the
trial;

the  design  of  the  clinical
trial;

effectiveness  of  publicity  for  the  clinical
trials;

inability 
consents;

to  obtain  and  maintain  subject

ability to monitor subjects adequately during and after the administration of the product candidate and the ability of subjects
to comply with the clinical trial requirements;

risk  that  enrolled  subjects  will  drop  out  or  be  withdrawn  before  completion;
and

clinicians’  and  subjects’  perceptions  as  to  the  potential  advantages  of  the  drug  being  studied  in  relation  to  other  available
therapies, including any new drugs that may be approved for the indications we are investigating.

There  is  significant  competition  for  recruiting  subjects  in  clinical  trials  for  product  candidates  for  the  treatment  of  neurological
disorders  and  we  or  our  partners  may  be  unable  to  enroll  the  subjects  we  need  to  complete  clinical  trials  on  a  timely  basis  or  at  all.
Furthermore,  we  rely  on  CROs  and  clinical  trial  sites  to  ensure  the  proper  and  timely  conduct  of  our  clinical  trials,  and  while  we  have
agreements  governing  their  committed  activities,  we  have  limited  influence  over  their  actual  performance.  If  we  are  unable  to  enroll
sufficient  subjects  in  our  clinical  trials,  if  enrollment  is  slower  than  we  anticipate,  or  if  our  clinical  trials  require  more  subjects  than  we
anticipate,  our  clinical  trials  may  be  delayed  or  might  not  be  completed.  If  we  experience  delays  in  our  clinical  trials,  the  commercial
prospects of our product candidates will be harmed. In addition, any delays in completing our clinical trials will increase our costs, slow
down  our  product  candidate  development  and  approval  process  and  jeopardize  our  ability  to  commence  product  sales  and  generate
revenues. In  addition,  many  of  the  factors  that  could  cause  a  delay  in  the  commencement  or  completion  of  clinical  trials  may  also
ultimately lead to the denial of regulatory approval of our lead product candidates or our other product candidates.

We may face significant delays in our clinical studies and trials due to an inability to recruit patients for our clinical studies and trials
or to retain patients in the clinical studies and trials we may perform.

We may not be able to locate and enroll enough eligible patients to participate in these trials as required by the FDA, the EMA or
similar regulatory authorities outside the United States and the European Union. This may result in our failure to initiate or continue clinical
trials  for  our  product  candidates  or  may  cause  us  to  abandon  one  or  more  clinical  trials  altogether.  In  particular,  because  several  of  our
programs are focused on the treatment of patients with rare, orphan or ultra-orphan diseases, our ability to enroll eligible patients in these
trials may be limited or slower than we anticipate in light of the small patient populations involved and the specific age range required for
treatment eligibility in some indications. In addition, our potential competitors, including major pharmaceutical, specialty pharmaceutical
and biotechnology companies, academic institutions and governmental agencies and public and private research institutions, may seek to
develop competing therapies, which would further limit the small patient pool available for our studies.

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Completion  of  orphan  clinical  trials  may  take  considerably  more  time  than  other  trials,  sometimes  years,  depending  on  factors
such as type, complexity, novelty and intended use of a product candidate. As a result of the uncertainties described above, there can be no
assurance that we will meet timelines that we establish for any of our clinical trials.

We may in the future conduct clinical trials for certain of our product candidates at sites outside the United States, and the FDA might
not accept data from trials conducted in such locations.

We may in the future choose to conduct one or more of our clinical trials outside the United States. Although the FDA may accept
data from clinical trials conducted outside the United States, acceptance of this data is subject to certain conditions imposed by the FDA.
For example, the clinical trial must be well-designed and conducted and performed by qualified investigators in accordance with ethical
principles and current Good Clinical Practice, or GCPs. The trial population must also adequately represent the U.S. population, and the
data  must  be  applicable  to  the  U.S.  population  and  medical  practice  in  ways  that  the  FDA  deems  clinically  meaningful.  Generally,  the
patient  population  for  any  clinical  trials  conducted  outside  of  the  United  States  must  be  representative  of  the  population  for  whom  we
intend to seek approval in the United States. In addition, while these clinical trials are subject to the applicable local laws, FDA acceptance
of the data will be dependent upon its determination that the trials also complied with all applicable U.S. laws and regulations. There can be
no assurance that the FDA will accept data from trials conducted outside of the United States. If the FDA does not accept the data from any
of our clinical trials that we determine to conduct outside the United States, it would likely result in the need for additional trials, which
would be costly and time‑consuming and delay or permanently halt our development of the product candidate.

We may fail to successfully identify, in‑license, acquire, develop or commercialize potential product candidates.

The success of our business depends in part upon our ability to identify and validate new therapeutic targets and identify, develop
and  commercialize  therapeutics,  which  we  may  develop  ourselves,  in‑license  or  acquire  from  others.  Research  programs  designed  to
identify  product  candidates  require  substantial  technical,  financial  and  human  resources,  whether  or  not  any  product  candidates  are
ultimately identified. Our research efforts may initially show promise in identifying potential therapeutic targets or candidates, yet fail to
yield product candidates for clinical development for a number of reasons, including:

•

•

our  methodology,  including  our  screening  technology,  might  not  successfully  identify  medically  relevant  potential  product
candidates;

our  competitors  may  develop  alternatives  that  render  our  product  candidates
obsolete;

• we may encounter product manufacturing difficulties that limit yield or produce undesirable characteristics that increase the

cost of goods, cause delays or make the product candidates unmarketable;

•

•

•

•

•

our product candidates may cause adverse effects in subjects, even after successful initial toxicology studies, which may make
the product candidates unmarketable;

our product candidates might not be capable of being produced in commercial quantities at an acceptable cost, or at
all;

our  product  candidates  might  not  demonstrate  a  meaningful  benefit  to
subjects;

our  potential  collaboration  partners  may  change  their  development  profiles  or  plans  for  potential  product  candidates  or
abandon a therapeutic area or the development of a partnered product; and

our reliance on third party clinical trials may cause us to be denied access to clinical results that may be significant to further
clinical development.

Additionally,  we  may  focus  our  efforts  and  resources  on  potential  programs  or  product  candidates  that  ultimately  prove  to  be
unsuccessful. If any of these events occur, we may be forced to abandon our development efforts for a program or programs, which would
have a material adverse effect on our business, operating results and prospects and could potentially cause us to cease operations.

We might not be successful in our efforts to develop and commercialize our preclinical product candidates.

Our continued development of our preclinical product candidates will be dependent on receiving positive preclinical and clinical
data that, in our judgment, merits advancing such programs. Even if we are successful in continuing to build and expand our pipeline, the
potential product candidates that we identify might not be suitable for clinical development, including as a result of being shown to have
harmful side effects or other characteristics that indicate that they are unlikely to be products that will receive marketing approval

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and  achieve  market  acceptance.  Similarly,  even  if  the  FDA  approves  our  INDs,  there  is  no  guarantee  that  we  will  be  successful  in  our
efforts  to  advance  our  preclinical  product  candidates  into  clinical  trials. If  we  do  not  successfully  develop  and  commercialize  product
candidates based upon our technological approach, we will not be able to obtain product revenues in future periods, which likely would
result in significant harm to our financial position and adversely affect our stock price.

The marketing approval processes of the FDA and comparable foreign regulatory authorities are lengthy, time ‑consuming, costly and
inherently unpredictable. Our inability to obtain regulatory approval for our product candidates would substantially harm our business.

The  time  required  to  obtain  approval  to  market  new  drugs  by  the  FDA  and  comparable  foreign  regulatory  authorities  is
unpredictable  but  typically  takes  many  years  following  the  commencement  of  preclinical  studies  and  clinical  trials  and  depends  upon
numerous factors, including the discretion of the regulatory authorities. In addition, approval policies, regulations or the type and amount of
clinical data necessary to gain approval may change during the course of a product candidate’s clinical development and may vary among
jurisdictions.  We  have  not  obtained  regulatory  approval  for  any  product  candidate  and  it  is  possible  that  none  of  our  existing  product
candidates or any future product candidates will ever obtain regulatory approval. Moreover, the filing of an NDA for products that have not
been granted Orphan Drug Designation requires a payment of a significant PDUFA NDA application fee upon submission. Any subsequent
clinical data submissions to the NDA (i.e. for new indications) are also assessed an NDA application fee. The filing of an NDA for our
product candidates may be delayed due to our lack of financial resources to pay such user fee.

Our product candidates could fail to receive regulatory approval from the FDA or a comparable foreign regulatory authority for

many reasons, including:

•

•

•

•

the  FDA  or  comparable  foreign  regulatory  authorities  may  disagree  on  the  design  or  implementation  of  our  clinical  trials,
including the methodology used in our trial, our chosen endpoints, our statistical analysis, or our proposed product indication.
For instance, the FDA may find that the designs that we are utilizing in our planned clinical trial do not support an adequate
and well‑controlled study. The FDA also might not agree with the various disease scales and evaluation tools that we may use
in  our  clinical  trials  to  assess  the  efficacy  of  our  product  candidates.  Further,  the  FDA  might  not  agree  with  our  endpoints
and/or indications selected for our development programs;

the  FDA  or  comparable  foreign  regulatory  authorities  may  disagree  with  our  development  plans  for  our  product
candidates;

our failure to demonstrate to the satisfaction of the FDA or comparable regulatory authorities that a product candidate is safe
and effective for its proposed indication;

our  clinical  trials  may  fail  to  meet  the  level  of  statistical  significance  required  for
approval;

• we  may  fail  to  demonstrate  that  a  product  candidate’s  clinical  and  other  benefits  outweigh  its  safety

risks;

•

•

the FDA or comparable foreign regulatory authorities may disagree with our interpretation of data from preclinical studies or
clinical trials;

data  collected  from  clinical  trials  of  our  product  candidates  may  be  insufficient  to  support  the  submission  and  filing  of  an
NDA, other submission or to obtain marketing approval, and FDA may require additional studies to show that our product
candidates are safe or effective;

• we  may  fail  to  obtain  approval  of  the  manufacturing  processes  or  facilities  of  third‑party  manufacturers  with  whom  we

contract for clinical and commercial supplies; or

•

there  may  be  changes  in  the  approval  policies  or  regulations  that  render  our  preclinical  and  clinical  data  insufficient  for
approval.

The  FDA  or  comparable  foreign  regulatory  authority  may  require  more  information,  including  additional  preclinical  or  clinical
studies  to  support  approval,  which  may  delay  or  prevent  approval  and  our  commercialization  plans,  or  we  may  decide  to  abandon  the
development program. This lengthy approval process, as well as the unpredictability of future clinical trial results, may result in our failing
to obtain approval to market our product candidates, which would significantly harm our business, results of operations and prospects. In
addition, even if we were to obtain approval, regulatory authorities may approve any or all of our product candidates for fewer or more
limited  indications  than  we  request,  may  require  that  contraindications,  warnings  or  precautions  be  included  in  the  product  labeling,
including  a  black‑box  warning,  may  grant  approval  with  a  requirement  of  costly  post‑marketing  clinical  trials  or  other  post‑market
requirements, or may approve a product candidate with a label that does not include the labeling claims necessary or desirable for the

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successful  commercialization  of  that  product  candidate. Any  of  the  foregoing  scenarios  could  materially  harm  the  commercial  prospects
for our product candidates.

As  appropriate,  we  intend  to  seek  all  available  periods  of  regulatory  exclusivity  for  our  product  candidates.  However,  there  is  no
guarantee that we will be granted these periods of regulatory exclusivity or that we will be able to maintain these periods of exclusivity.

The FDA grants product sponsors certain periods of regulatory exclusivity, during which the agency might not approve, and in
certain instances, might not accept, certain marketing applications for competing drugs. For example, product sponsors may be eligible for
five years of exclusivity from the date of approval of a new chemical entity, seven years of exclusivity for drugs that are designated to be
orphan drugs, and/or a six‑month period of exclusivity added to any existing exclusivity period or patent life for the submission of FDA
requested pediatric data. While we intend to apply for all periods of market exclusivity that we may be eligible for, there is no guarantee
that we will receive all such periods of market exclusivity. Additionally, under certain circumstances, the FDA may revoke the period of
market exclusivity. Thus, there is no guarantee that we will be able to maintain a period of market exclusivity, even if granted. Moreover,
we have not sought to obtain orphan drug designation for any of our product candidates, which the FDA must first grant to be eligible for
orphan drug exclusivity, but may if we determine that we may be eligible. In the case of orphan designation, other benefits, such as tax
credits and exemption from user fees may be available. If we are not able to obtain or maintain orphan drug designation or any period of
market  exclusivity  to  which  we  may  be  entitled,  we  will  be  materially  harmed,  as  we  will  potentially  be  subject  to  greater  market
competition and may lose the benefits associated with programs.

Our  product  candidates  may  cause  undesirable  side  effects  or  have  other  properties  that  could  delay  or  prevent  their  marketing
approval,  limit  the  commercial  profile  of  an  approved  label,  or  result  in  significant  negative  consequences  following  any  marketing
approval.

Undesirable  side  effects  caused  by  our  product  candidates  could  cause  us  or  regulatory  authorities  to  interrupt,  delay  or  halt
clinical trials (Clinical Hold) and could result in a more restrictive label or the delay or denial of marketing approval by the FDA or other
comparable foreign regulatory authority. Results of our trials could reveal a high and unacceptable severity and prevalence of side effects or
unexpected characteristics.

Should our clinical studies of our product candidates reveal undesirable side effects, we could suspend or terminate our trials or
the  FDA  or  comparable  foreign  regulatory  authorities  as  well  as  IRBs  could  order  us  to  suspend  or  cease  clinical  trials.  The  FDA  or
comparable  regulatory  authorities  could  also  deny  approval  of  our  product  candidates  for  any  or  all  targeted  indications  or  only  for  a
limited  indication  or  patient  population  or  could  require  label  warnings,  contraindications  or  precautions,  including  black  box  warnings,
post‑market  studies,  testing  and  surveillance  programs  or  other  conditions  including  distribution  restrictions  or  other  risk  management
mechanisms under a costly risk evaluation and mitigation strategy ("REMS"). Drug‑related side effects could affect subject recruitment or
the ability of enrolled subjects to complete the trial or result in potential product liability claims. Any of these occurrences may harm our
business, financial condition and prospects significantly.

Additionally,  if  one  or  more  of  our  product  candidates  receives  marketing  approval,  and  we  or  others  (Regulatory Agencies,
Consumers, etc.) later identify undesirable side effects caused by such products, a number of potentially significant negative consequences
could result, including:

• we  may  suspend  marketing  of,  or  withdraw  or  recall,  such

product;

•

•

•

•

•

regulatory  authorities  may  withdraw  approvals  of  such
product;

regulatory  authorities  may  require  additional  warnings  on  the  label  or  other  label
modifications;

the  FDA  or  other  regulatory  bodies  may  issue  safety  alerts,  Dear  Healthcare  Provider  letters,  press  releases  or  other
communications containing warnings about such product;

the FDA may require the establishment or modification of a REMS or other restrictions on marketing and distribution, or a
comparable  foreign  regulatory  authority  may  require  the  establishment  or  modification  of  a  similar  strategy  that  may,  for
instance, require us to issue a medication guide outlining the risks of such side effects for distribution to patients or restrict
distribution of our products and impose burdensome implementation requirements on us;

regulatory  authorities  may  require  that  we  conduct  post‑marketing  studies;
and

• we  could  be  sued  and  held  liable  for  harm  caused  to  subjects  or

patients.

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Any  of  these  events  could  prevent  us  from  achieving  or  maintaining  market  acceptance  of  the  particular  product  candidate  or
otherwise  materially  harm  the  commercial  prospects  for  the  product  candidate,  if  approved,  and  could  significantly  harm  our  business,
financial condition, results of operations and prospects.

Changes in product candidate manufacturing or formulation may result in additional costs or delay.

As  product  candidates  are  developed  through  preclinical  studies  to  late‑stage  clinical  trials  towards  regulatory  approval  and
commercialization, it is common that various aspects of the development program, such as  manufacturing  methods  and  formulation,  are
altered in an effort to optimize processes and results. Such changes carry the risk that they will not achieve these intended objectives. Any
of these changes could cause our product candidates to perform differently and affect the results of planned clinical trials or other future
clinical trials conducted with the altered materials. Such changes may also require additional testing, FDA notification or FDA approval.

Similarly,  changes  in  the  location  of  manufacturing  or  addition  of  manufacturing  facilities  may  increase  our  costs  and  require
additional studies and FDA approval. This may require us to ensure that the new facility meets all applicable regulatory requirements, is
adequately validated and qualified, and to conduct additional studies of product candidates manufactured at the new location. Any of the
above could delay completion of clinical trials, require the conduct of bridging clinical trials or the repetition of one or more clinical trials,
increase clinical trial costs, delay regulatory approval of our product candidates and jeopardize our ability to commence product sales and
generate revenue.

Even if we complete the necessary clinical trials, we cannot predict when or if we will obtain marketing approval to commercialize a
product candidate or the approval may be for a narrower indication than we expect.

We cannot commercialize a product candidate until the appropriate regulatory authorities have reviewed and approved the product
candidate. Even if our product candidates demonstrate safety and efficacy in clinical trials, the regulatory agencies might not complete their
review  processes  in  a  timely  manner,  or  we  might  not  be  able  to  obtain  marketing  approval  from  the  relevant  regulatory  agencies.
Additional  delays  may  result  if  the  FDA,  an  FDA  Advisory  Committee  or  other  regulatory  authority  recommends  non‑approval  or
restrictions  on  approval.  In  addition,  we  may  experience  delays  or  rejections  based  upon  additional  government  regulation  from  future
legislation or administrative action, or changes in regulatory agency policy during the period of product development, clinical trials and the
review  process.  Regulatory  authorities  also  may  approve  a  product  candidate  for  fewer  or  more  limited  indications  than  requested,  may
impose significant limitations in the form of narrow indications, warnings, including black‑box warnings, precautions or contra‑indications
with  respect  to  conditions  of  use  or  may  grant  approval  subject  to  the  performance  of  costly  post‑marketing  clinical  trials  or  other
post‑marketing requirements, including a REMS. In addition, regulatory agencies might not approve the labeling claims that are necessary
or  desirable  for  the  successful  commercialization  of  our  product  candidates. Our  drugs,  if  approved,  may  be  required  to  carry  warnings
comparable to this and other class‑wide warnings. Any of the foregoing scenarios could materially harm the commercial prospects for our
product candidates.

Even if we were to obtain approval for our product candidates with the Rare Pediatric Disease Designation, the Rare Pediatric Disease
Priority Review Voucher Program may no longer be in effect at the time of such approval or we might not be able to capture the value of
the Rare Pediatric Disease Priority Review Voucher Program.

Rare pediatric disease designation by the FDA is granted in the case of serious or life-threatening diseases affecting fewer than
200,000 people in the United States in which the serious or life-threatening manifestations are primarily in individuals 18 years of age and
younger.  The  designation  provides  regulatory  incentives  for  companies  to  develop  and  market  therapies  that  treat  these  conditions.  The
sponsor of a drug for a rare pediatric disease may be eligible for a priority review voucher upon approval of the drug that can be used to
obtain a priority review of a subsequent marketing application. The priority review voucher may be sold or transferred an unlimited number
of  times.  Congress  has  extended  the  priority  review  voucher  program  until  September  30,  2020  with  new  drug  approvals  that  meet  the
voucher criteria grandfathered through 2022. This program has been subject to criticism, including by the FDA, and it is possible that even
if we obtain approval for some of our product candidates and qualify for such a priority review voucher, the program may no longer be in
effect at the time of approval. Also, although Priority Review Vouchers may be sold or transferred to third parties, there is no guaranty that
we will be able to realize any value if we were to sell a Priority Review Voucher.

Even if we were able to commercialize our products focused on rare orphan diseases, product sales of these products might not justify
the cost of development.

Because  of  the  small  patient  population  for  a  rare  orphan  disease,  if  pricing  is  not  approved  or  accepted  in  the  market  at  an

appropriate level for an approved therapeutic product with orphan drug designation, such drug may not generate enough revenue to offset

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costs  of  development,  manufacturing,  marketing,  and  commercialization  despite  any  benefits  received  from  the  rare  orphan  drug
designation, such as market exclusivity, assistance in clinical trial design, or a reduction in user fees or tax credits related to development
expense.  Furthermore,  our  estimates  regarding  potential  market  size  for  any  rare  indication  may  be  materially  different  from  what  we
discover to exist at the time we commence commercialization, if any, for a therapeutic product, which could result in significant changes in
our business plan and have a material adverse effect on our business, financial condition, results of operations, and prospects.

Once  commercialized,  some  of  our  products  may  face  significant  competition  from  non-prescription  competition  and  consumer
substitution, and our operating results will suffer if we fail to compete effectively.

We may be subject to non-prescription competition and consumer substitution for certain of our pipeline assets. For example, the
three preclinical therapies in our pediatric orphan rare disease pipeline, CERC-801, CERC-802 and CERC-803, are ultra-pure formulations
of D-galactose, D-mannose and L-fucose, respectively. These formulations are naturally occurring substances contained in various foods,
including dairy products and fruit. Additionally, these formulations, particularly D-mannose, are also marketed by others as non-
prescription dietary supplements. Once approved by the FDA and commercially available, we cannot be sure physicians will view the
pharmaceutical grade purity and tested safety of CERC-801, CERC-802 or CERC-803 as having a superior therapeutic profile to the
naturally occurring formulations and dietary supplements. In addition, to the extent the net price of CERC-801, CERC-802 or CERC-803,
after insurance and offered discounts, is significantly higher than the prices of commercially available formulations marketed by other
companies as dietary supplements (through that lack of coverage by insurers or otherwise), physicians and pharmacists may recommend
these commercial alternatives instead of writing or filling prescriptions for CERC-801, CERC-802 or CERC-803, or patients may elect on
their own to take commercially available supplements. Either of these outcomes may adversely impact our results of operations by limiting
how we price our product and limiting the revenue we receive from the sale of CERC-801, CERC-802 and CERC-803 due to reduced
market acceptance.

Even  if  our  product  candidates  receive  marketing  approval,  we  will  still  be  subject  to  ongoing  regulatory  obligations  and  continued
regulatory  review,  which  may  result  in  significant  additional  expense.  Additionally,  our  product  candidates,  if  approved,  could  be
subject to labeling and other restrictions and market withdrawal and we may be subject to administrative sanctions or penalties if we
fail to comply with regulatory requirements or experience unanticipated problems with our products.

Even  if  we  obtain  marketing  approval  for  a  product  candidate,  we  would  be  subject  to  ongoing  requirements  by  the  FDA  and
comparable  foreign  regulatory  authorities  governing  the  manufacture,  quality  control,  further  development,  labeling,  packaging,  storage,
distribution, safety surveillance, import, export, advertising, promotion, recordkeeping and annual reporting of safety and other post‑market
information. The FDA and comparable foreign regulatory authorities will continue to closely monitor the safety profile of any product even
after approval. If the FDA or comparable foreign regulatory authorities become aware of new safety information after approval of any of
our  product  candidates,  they  may  withdraw  approval,  require  labeling  changes  or  establishment  of  a  REMS  or  similar  strategy,  impose
significant  restrictions  on  a  product’s  indicated  uses  or  marketing,  or  impose  ongoing  requirements  for  potentially  costly  post‑approval
studies  or  post‑market  surveillance.  In  addition,  any  marketing  approvals  that  we  obtain  for  our  product  candidates  may  be  subject  to
limitations on the approved indicated uses for which the product may be marketed or to the conditions of approval or contain requirements
for  potentially  costly  post‑marketing  testing  and  other  requirements,  including  Phase  4  clinical  trials,  imposition  of  a  REMS  and
surveillance to monitor the safety and efficacy of the product candidate.

In addition, manufacturers of drug products and their facilities, including contracted facilities, are subject to periodic inspections
by  the  FDA  and  other  regulatory  authorities  for  compliance  with  current  GMP  regulations  and  standards.  If  we  or  a  regulatory  agency
discover previously unknown problems with the facility where the product is manufactured, we may be subject to reporting obligations and
a regulatory agency may impose restrictions on that product, the manufacturing facility, us, or our suppliers, including requesting recalls or
withdrawal  of  the  product  from  the  market  or  suspension  of  manufacturing.  If  we,  our  product  candidates,  our  contractors,  the
manufacturing facilities for our product candidates or others working on our behalf fail to comply with applicable regulatory requirements,
either before or after marketing approval, a regulatory agency may:

•

issue  Warning  Letters  or  Untitled
Letters;

• mandate  modifications  to  promotional  materials  or  labeling,  or  require  us  to  provide  corrective  information  to  healthcare

practitioners;

•

•

require us to enter into a consent decree, which can include imposition of various fines, reimbursements for inspection costs,
required due dates for specific actions and penalties for noncompliance;

seek  an  injunction  or  impose  civil  or  criminal  penalties  or  monetary  fines,  restitution  or  disgorgement,  as  well  as
imprisonment;

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•

•

•

•

•

•

suspend 
approval;

or  withdraw  marketing

suspend  or 
studies;

terminate  any  ongoing  clinical

refuse  to  approve  pending  applications  or  supplements  to  applications  filed  by
us;

debar  us  from  submitting  marketing  applications,  exclude  us  from  participation  in  federal  healthcare  programs,  require  a
corporate  integrity  agreement  or  deferred  prosecution  agreements,  debar  us  from  government  contracts  and  refuse  future
orders under existing contracts;

suspend  or  impose  restrictions  on  operations,  including  restrictions  on  marketing,  distribution  or  manufacturing  of  the
product, or the imposition of costly new manufacturing requirements or use of alternative suppliers; or

seize  or  detain  products,  refuse  to  permit  the  import  or  export  of  products,  or  request  that  we  initiate  a  product
recall.

The  occurrence  of  any  event  or  penalty  described  above  may  inhibit  our  ability  to  continue  our  development  programs,

commercialize our products and generate revenue.

Advertising and promotion of any product candidate that obtains approval in the United States will be heavily scrutinized by the
FDA,  the  Department  of  Justice,  the  Department  of  Health  and  Human  Services’  Office  of  Inspector  General,  state  attorneys  general,
members of Congress and the public. While the FDA does not restrict physicians from prescribing approved drugs for uses outside of the
drugs’ approved labeling, known as off‑label use, pharmaceutical manufacturers are strictly prohibited from promoting and marketing their
products  for  such  uses.  Violations,  including  promotion  of  our  products  for  off‑label  uses,  are  subject  to  enforcement  letters,  inquiries,
investigations, civil and criminal sanctions by the government, corporate integrity agreements, deferred prosecution agreements, debarment
from  government  contracts  and  refusal  of  future  orders  under  existing  contracts,  and  exclusion  from  participation  in  federal  healthcare
programs.  Additionally,  comparable  foreign  regulatory  authorities  will  heavily  scrutinize  advertising  and  promotion  of  any  product
candidate that obtains approval outside of the United States.

In the United States, engaging in the impermissible promotion of our products for off‑label uses can also subject us to false claims
litigation under federal and state statutes, which can lead to civil and criminal penalties and fines, debarment from government contracts and
refusal of future orders under existing contracts, deferred prosecution agreements, and corporate integrity agreements with governmental
authorities that materially restrict the manner in which a company promotes or distributes drug products. These false claims statutes include
the federal civil False Claims Act, which allows any individual to bring a lawsuit against a pharmaceutical company on behalf of the federal
government  alleging  submission  of  false  or  fraudulent  claims,  or  causing  to  present  such  false  or  fraudulent  claims,  for  payment  by  a
federal program such as Medicare or Medicaid. If the government decides to intervene and prevails in the lawsuit, the individual will share
in any fines or settlement funds. If the government does not intervene, the individual may proceed on his or her own. Since 2004, these
False  Claims  Act  lawsuits  against  pharmaceutical  companies  have  increased  significantly  in  volume  and  breadth,  leading  to  several
substantial civil and criminal settlements, such as settlements regarding certain sales practices promoting off‑label drug uses involving fines
that are as much as $3.0 billion. This growth in litigation has increased the risk that a pharmaceutical company will have to defend a false
claim action, pay settlement fines or restitution, agree to comply with burdensome reporting and compliance obligations, and be excluded
from Medicare, Medicaid and other federal and state healthcare programs. If we do not lawfully promote our approved products, we may
become  subject  to  such  litigation  and,  if  we  do  not  successfully  defend  against  such  actions,  those  actions  may  have  a  material  adverse
effect on our business, financial condition, results of operations and prospects.

The  FDA’s  policies  may  change,  and  additional  government  regulations  may  be  enacted  that  could  prevent,  limit  or  delay
marketing  approval,  and  the  sale  and  promotion  of  our  product  candidates.  If  we  are  slow  or  unable  to  adapt  to  changes  in  existing
requirements or the adoption of new requirements or policies, or if we are not able to maintain regulatory compliance, we may lose any
marketing  approval  that  we  may  have  obtained,  which  would  adversely  affect  our  business,  prospects  and  ability  to  achieve  or  sustain
profitability.

If we are unable to, or are delayed in obtaining, state regulatory licenses for the distribution of our products, we would not be able to
sell our product candidates in such states.

The majority of states require manufacturer and/or wholesaler licenses for the sale and distribution of drugs into that state. The
application process is complicated, time consuming, costly and requires dedicated personnel or a third party to oversee and manage. If we
are delayed in obtaining these state licenses, or denied the licenses, even with FDA approval, we would not be able to sell or ship product
into that state which would adversely affect our sales and revenues.

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If  any  of  our  product  candidates  are  ultimately  regulated  as  controlled  substances,  we,  our  contract  manufacturers,  as  well  as
distributors,  prescribers,  and  dispensers  will  be  required  to  comply  with  additional  regulatory  requirements  which  could  delay  the
marketing of our product candidates, and increase the cost and burden of manufacturing, distributing, dispensing, and prescribing our
product candidates.

Before we can commercialize our product candidates, the United States Drug Enforcement Administration, or DEA, may need to
determine  the  controlled  substance  Schedule,  taking  into  account  the  recommendation  of  the  FDA.  This  may  be  a  lengthy  process  that
could delay our marketing of a product candidate and could potentially diminish any regulatory exclusivity periods for which we may be
eligible. While we currently do not know whether any of our product candidates will be considered to be controlled substances, certain of
our product candidates may be regulated as controlled substances.

If any of our product candidates are regulated as controlled substances, depending on the controlled substance schedule in which
the  product  candidates  are  placed,  we,  our  contract  manufacturers,  and  any  distributers,  prescribers,  and  dispensers  of  the  scheduled
product candidates may be subject to significant regulatory requirements, such as registration, security, recordkeeping, reporting, storage,
distribution, importation, exportation, inventory, quota and other requirements administered by the DEA. Moreover, if any of our product
candidates  are  regulated  as  controlled  substances,  we  and  our  contract  manufacturers  would  be  subject  to  initial  and  periodic  DEA
inspection. If we or our contract manufacturers are not able to obtain or maintain any necessary DEA registrations, we might not be able to
commercialize  any  product  candidates  that  are  deemed  to  be  controlled  substances  or  we  may  need  to  find  alternative  contract
manufacturers, which would take time and cause us to incur additional costs, delaying or limit our commercialization efforts.

Because  of  their  restrictive  nature,  these  laws  and  regulations  could  limit  commercialization  of  our  product  candidates,  should
they be deemed to contain controlled substances. Failure to comply with the applicable controlled substance laws and regulations can also
result in administrative, civil or criminal enforcement. The DEA may seek civil penalties, refuse to renew necessary registrations, or initiate
administrative proceedings to revoke those registrations. In some circumstances, violations could result in criminal proceedings or consent
decrees. Individual states also independently regulate controlled substances.

Our failure to obtain regulatory approval in international jurisdictions would prevent us from marketing our product candidates outside
the United States, which would limit our market opportunities and adversely affect our business.

In  order  to  market  and  sell  our  products  in  other  jurisdictions,  we  must  obtain  separate  marketing  approvals  and  comply  with
numerous  and  varying  regulatory  requirements.  The  approval  procedure  varies  among  countries  and  can  involve  additional  testing.  The
time  required  to  obtain  approval  may  differ  substantially  from  that  required  to  obtain  FDA  approval.  The  regulatory  approval  process
outside the United States generally includes all of the risks associated with obtaining FDA approval. In addition, in many countries outside
the United States, we must secure product reimbursement approvals before regulatory authorities will approve the product for sale in that
country.  Obtaining  foreign  regulatory  approvals  and  compliance  with  foreign  regulatory  requirements  could  result  in  significant  delays,
difficulties  and  costs  for  us  and  could  delay  or  prevent  the  introduction  of  our  products  in  certain  countries.  Further,  clinical  trials
conducted  in  one  country  might  not  be  accepted  by  regulatory  authorities  in  other  countries.  If  we  fail  to  comply  with  the  regulatory
requirements  in  international  markets  and  receive  applicable  marketing  approvals,  our  target  market  will  be  reduced  and  our  ability  to
realize the full market potential of our product candidates will be harmed and our business will be adversely affected. We might not obtain
foreign regulatory approvals on a timely basis, if at all. Approval by the FDA does not ensure approval by regulatory authorities in other
countries or jurisdictions. Approval by one regulatory authority outside the United States does not ensure approval by regulatory authorities
in other countries or jurisdictions or by the FDA. Also, regulatory approval for any of our product candidates may be withdrawn. However,
the failure to obtain approval in one jurisdiction may negatively impact our ability to obtain approval in another jurisdiction. Our failure to
obtain approval of any of our product candidates by regulatory authorities in another country may significantly diminish the commercial
prospects of that product candidate and our business prospects could decline.

If  we  obtain  approval  to  commercialize  our  product  candidates  outside  of  the  United  States,  a  variety  of  risks  associated  with
international operations could materially adversely affect our business.

If any of our product candidates are approved for commercialization, we may enter into agreements with third parties to market
them on a worldwide basis or in more limited geographical regions. We expect that we will be subject to additional risks related to entering
into international business relationships, including:

•

•

different  regulatory  requirements  for  approval  of  drugs  in  foreign
countries;

challenges enforcing our contractual and intellectual property rights, especially in those foreign countries that do not respect and
protect intellectual property rights to the same extent as the United States;

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•

•

•

•

•

•

•

•

•

•

•

foreign 
regimes;

reimbursement,  pricing  and 

insurance

unexpected  changes 
requirements;

in 

tariffs, 

trade  barriers  and 

regulatory

economic  weakness,  including  inflation,  or  political  instability  in  particular  foreign  economies  and
markets;

compliance  with  tax,  employment,  immigration  and  labor  laws  for  employees  living  or  traveling
abroad;

foreign  currency  fluctuations,  which  could  result  in  increased  operating  expenses  and  reduced  revenues,  and  other  obligations
incident to doing business in another country;

foreign
taxes;

difficulties 
operations;

staffing 

and  managing 

foreign

workforce  uncertainty  in  countries  where  labor  unrest  is  more  common  than  in  the  United
States;

potential  liability  under  the  Foreign  Corrupt  Practices  Act  of  1977  or  comparable  foreign
regulations;

production shortages resulting from any events affecting raw material supply or manufacturing capabilities abroad;
and

business interruptions resulting from geopolitical actions, including war and terrorism, or natural disasters including earthquakes,
typhoons, floods and fires.

These and other risks associated with our international operations may materially adversely affect our ability to attain or maintain

profitable operations.

We face substantial competition and rapid technological change and the possibility that others may discover, develop or commercialize
products before or more successfully than us.

The  biotechnology  and  pharmaceutical  industries  are  intensely  competitive  and  subject  to  rapid  and  significant  technological
change. We face competition with respect to our current product candidates and will face competition with respect to any future product
candidates from major pharmaceutical companies, specialty pharmaceutical companies and biotechnology companies worldwide. Many of
our competitors have significantly greater financial, technical and human resources. Smaller and early‑stage companies may also prove to
be significant competitors, particularly through collaborative arrangements with large and established companies.

Our competitors may obtain marketing approval of their products more rapidly than we may or may obtain patent protection or
other  intellectual  property  rights  that  limit  our  ability  to  develop  or  commercialize  our  product  candidates.  Our  competitors  may  also
develop drugs that are more effective, more convenient, more widely used and less costly or have a better safety profile than our products
and these competitors may also be more successful than us in manufacturing and marketing their products.

Our competitors will also compete with us in recruiting and retaining qualified scientific, management and commercial personnel,
establishing clinical trial sites and subject registration for clinical trials, as well as in acquiring technologies complementary to, or necessary
for, our programs.

There  are  numerous  currently  approved  therapies  for  treating  the  pediatric  conditions  our  products  address  and,  consequently,
competition in these markets is intense. Many of these approved drugs are well established therapies or products and are widely accepted
by physicians, patients and third-party payors. Some of these drugs are branded and subject to patent protection and non-patent regulatory
exclusivity, and others are available on a generic basis.

Insurers and other third‑party payors may also encourage the use of generic products or specific branded products. We expect that
any or our product candidates, if approved, would be priced at a significant premium over competitive generic, including branded generic,
products, but, any new product that competes with an approved product must demonstrate compelling advantages in efficacy, convenience,
tolerability  and  safety  in  order  to  overcome  price  competition  and  to  be  commercially  successful.  This  may  make  it  difficult  for  us  to
differentiate  our  product  from  currently  approved  therapies,  which  may  adversely  impact  our  business  strategy.  If  we  are  not  able  to
compete effectively against our current and future competitors, our business will not grow, and our financial condition and operations will
suffer.

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Our products might not achieve adequate market acceptance among physicians, patients, third ‑party payors and others in the medical
community necessary for commercial success.

Even  if  our  product  candidates  have  or  receive  marketing  approval,  they  might  not  gain  adequate  market  acceptance  among
physicians, patients and others in the medical community. Our commercial success also depends on coverage and adequate reimbursement
of  our  product  candidates  by  third‑party  payors,  including  government  payors,  generally,  which  may  be  difficult  or  time‑consuming  to
obtain, may be limited in scope or might not be obtained in all jurisdictions in which we may seek to market our products. The degree of
market acceptance of any of our approved product candidates will depend on a number of factors, including:

•

•

•

•

•

•

•

•

•

•

•

the efficacy and safety profile of our product candidates, including relative to marketed  products  and  product  candidates  in
development by third parties;

prevalence  and  severity  of  any  side  effects  of  our  product
candidates;

relative  convenience  and  ease  of  administration  of  our  product
candidates;

effectiveness 

cost 
candidates;

of 

our 

product

the claims we may make for our product candidates based on the approved label or any restrictions placed upon our marketing
and distribution of our product candidates;

the  time  it  takes  for  our  product  candidates  to  complete  clinical  development  and  receive  marketing
approval;

how quickly and effectively we alone, or with a partner, can market, launch, and distribute any of our product candidates that
receive marketing approval;

the  ability  to  commercialize  any  of  our  product  candidates  that  receive  marketing
approval;

the  price  of  our  products,  including  in  comparison  to  branded  or  generic  competitors  and  relative  to  alternative
treatments;

potential  or  perceived  advantages  of  disadvantages  over  alternative
treatments;

the  ability  to  collaborate  with  others  in  the  development  and  commercialization  of  new
products;

• whether coverage and adequate levels of reimbursement are available under private and governmental health insurance plans,

including Medicare;

•

•

•

•

•

•

•

•

the  ability  to  establish,  maintain  and  protect  intellectual  property  rights  related  to  our  product
candidates;

the  entry  of  generic  versions  of  our  products  onto  the
market;

the  number  of  products  in  the  same  therapeutic  class  as  our  product
candidates;

the  effect  of  current  and  future  healthcare  laws  on  our  drug
candidates;

the  ability  to  secure  favorable  managed  care  formulary  positions,  including  federal  healthcare  program
formularies;

the  ability  to  manufacture  commercial  quantities  of  any  of  our  product  candidates  that  receive  marketing
approval;

acceptance of any of our product candidates that receive marketing approval by physicians and other healthcare providers;
and

potential  post-marketing  commitments  imposed  on  regulatory  authorities,  such  as  patient
registries.

    
If  any  product  candidate  is  approved  but  does  not  achieve  an  adequate  level  of  acceptance  by  physicians,  hospitals,  third‑party
payors  and  patients,  we  might  not  generate  or  derive  sufficient  revenue  from  that  product  candidate  and  might  not  become  or  remain
profitable.

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Even if we commercialize any of our product candidates, these products may become subject to unfavorable third‑party coverage and
reimbursement policies, healthcare reform initiatives, or pricing regulations, any of which could negatively impact our business.

Our  ability  to  commercialize  any  products  successfully  will  depend  in  part  on  the  extent  to  which  coverage  and  adequate
reimbursement for these products will be available from government authorities (such as Medicare and Medicaid), private health insurers,
health maintenance organizations and other entities. These third‑party payors determine which medications they will cover and establish
reimbursement  levels,  and  increasingly  attempt  to  control  costs  by  limiting  coverage  and  the  amount  of  reimbursement  for  particular
medications. Several third‑party payors are requiring that drug companies provide them with predetermined discounts from list prices, are
using preferred drug lists to leverage greater discounts in competitive classes and are challenging the prices charged for drugs. In addition,
federal programs impose penalties on drug manufacturers in the form of mandatory additional rebates and/or discounts if commercial prices
increase at a rate greater than the Consumer Price Index‑Urban, and these rebates and/or discounts, which can be substantial, may impact
our  ability  to  raise  commercial  prices.  We  cannot  be  sure  that  coverage  and  reimbursement  will  be  available  for  any  product  that  we
commercialize and, if coverage is available, what the level of reimbursement will be. Coverage and reimbursement may impact the demand
for,  or  the  price  of,  any  product  candidate  for  which  we  obtain  marketing  approval.  If  coverage  and  reimbursement  are  not  available  or
available only to limited levels, we might not successfully commercialize any product candidate for which we obtain marketing approval.

There may be significant delays in obtaining coverage and reimbursement for newly approved drugs, and coverage may be more
limited than the purposes for which the drug is approved by the FDA or comparable foreign regulatory authorities. Moreover, eligibility for
coverage and reimbursement does not imply that a drug will be paid for in all cases or at a rate that covers our costs, including research,
development, manufacture, sale and distribution. Interim reimbursement levels for new drugs, if applicable, may also not be sufficient to
cover our costs and may only be temporary. Reimbursement rates for a drug may vary according to the clinical setting in which it is used
and  may  be  based  on  reimbursement  levels  already  set  for  lower  cost  drugs  and  may  be  incorporated  into  existing  payments  for  other
services.  Prices  paid  for  a  drug  also  vary  depending  on  the  class  of  trade.  Prices  charged  to  government  customers  are  subject  to  price
controls and private institutions obtain discounts through group purchasing organizations. Net prices for drugs may be further reduced by
mandatory discounts or rebates required by government healthcare programs and demanded by private payors, and by any future relaxation
of  laws  that  presently  restrict  imports  of  drugs  from  countries  where  they  may  be  sold  at  lower  prices  than  in  the  United  States.  Our
inability  to  promptly  obtain  coverage  and  profitable  reimbursement  rates  from  both  government‑funded  and  private  payors  for  any
approved  products  that  we  develop  could  have  a  material  adverse  effect  on  our  operating  results,  our  ability  to  raise  capital  needed  to
commercialize products and our overall financial condition.

Moreover,  the  regulations  that  govern  marketing  approvals,  pricing,  coverage  and  reimbursement  for  new  drug  products  vary
widely  from  country  to  country.  Current  and  future  legislation  may  significantly  change  the  approval  requirements  in  ways  that  could
involve additional costs and cause delays in obtaining approvals. Some countries require approval of the sale price of a drug before it can
be marketed. In many countries, the pricing review period begins after marketing or product licensing approval is granted. In some foreign
markets, prescription pharmaceutical pricing remains subject to continuing governmental control even after initial approval is granted. As a
result,  we  might  obtain  marketing  approval  for  a  product  in  a  particular  country,  but  then  be  subject  to  price  regulations  that  delay  our
commercial launch of the product, possibly for lengthy time periods, which could negatively impact the revenues we generate from the sale
of  the  product  in  that  particular  country. Adverse  pricing  limitations  may  hinder  our  ability  to  recoup  our  investment  in  one  or  more
product candidates even if our product candidates obtain marketing approval.

We may expend our limited resources to pursue a particular product candidate or indication and fail to capitalize on product candidates
or indications that may be more profitable or for which there is a greater likelihood of success.

 Because we have limited financial and managerial resources, we may forego or delay pursuit of opportunities with other product
candidates or for other indications that later prove to have greater commercial potential. Our resource allocation decisions may cause us to
fail  to  capitalize  on  viable  commercial  products  or  profitable  market  opportunities.  Our  spending  on  current  and  future  research  and
development  programs  and  product  candidates  for  specific  indications  might  not  yield  any  commercially  viable  products.  If  we  do  not
accurately evaluate the commercial potential or target market for a particular product candidate, we may relinquish valuable rights to that
product candidate through collaboration, licensing or other royalty arrangements in cases in which it would have been more advantageous
for us to retain sole development and commercialization rights to such product candidate.

Recently enacted and future legislation may increase the difficulty and cost for us to obtain marketing approval of and commercialize
our product candidates and affect the prices we may obtain.

In the United States and some foreign jurisdictions, there have been a number of legislative and regulatory changes and proposed

changes regarding the healthcare system that could, among other things, prevent or delay marketing approval of our product

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candidates, restrict or regulate post-approval activities and affect our ability to profitably sell any product candidates for which we obtain
marketing approval.

For example, in March 2010, the Patient Protection and Affordable Care Act, as amended by the Health Care and Education

Reconciliation Act, collectively the Affordable Care Act, was enacted to broaden access to health insurance, reduce or constrain the growth
of healthcare spending, enhance remedies against fraud and abuse, add new transparency requirements for health care and health insurance
industries, impose new taxes and fees on the health industry and impose additional health policy reforms. The law has continued the
downward pressure on pharmaceutical pricing, especially under the Medicare program, and increased the industry’s regulatory burdens and
operating costs. Among the provisions of the Affordable Care Act of importance to our potential drug candidates are the following:

•

•

•

•

•

•

•

•

•

•

•

an  annual,  nondeductible  fee  payable  by  any  entity  that  manufactures  or  imports  specified  branded  prescription  drugs  and
biologic agents;

revised  the  definition  of  “average  manufacturer  price,”  or AMP,  for  reporting  purposes,  which  can  increase  the  amount  of
Medicaid drug rebates manufacturers are required to pay to states, and created a separate AMP for certain categories of drugs
provided in non‑retail outpatient settings;

an  increase  in  the  statutory  minimum  rebates  a  manufacturer  must  pay  under  the  Medicaid  Drug  Rebate
Program;

a  new  methodology  by  which  rebates  owed  by  manufacturers  under  the  Medicaid  Drug  Rebate  Program  are  calculated  for
drugs that are inhaled, infused, instilled, implanted or injected;

a  new  Medicare  Part  D  coverage  gap  discount  program,  in  which  manufacturers  must  agree  to  offer  50%  (and  70%
commencing January 1, 2019) point-of-sale discounts off negotiated prices of applicable brand drugs to eligible beneficiaries
under their coverage gap period, as a condition for the manufacturer’s outpatient drugs to be covered under Medicare Part D;

extension  of  manufacturers’  Medicaid  rebate  liability  to  individuals  enrolled  in  Medicaid  managed  care
organizations;

expansion  of  eligibility  criteria  for  Medicaid  programs  in  certain
states;

expansion  of  the  entities  eligible  for  discounts  under  the  Public  Health  Service  pharmaceutical  pricing
program;

a  new  requirement  to  annually  report  drug  samples  that  manufacturers  and  distributors  provide  to
physicians;

a  new  Patient-Centered  Outcomes  Research  Institute  to  oversee,  identify  priorities  in,  and  conduct  comparative  clinical
effectiveness research, along with funding for such research; and

enacted  substantial  new  provisions  affecting  compliance  which  may  affect  our  business  practices  with  healthcare
practitioners.

We cannot predict the full impact of the Affordable Care Act on pharmaceutical companies, as many of the reforms require the

promulgation of detailed regulations implementing the statutory provisions, some of which has not yet fully occurred. For example, in
January 2016, the Centers for Medicare and Medicaid Services issued a final rule regarding the Medicaid Drug Rebate Program, effective
April 1, 2016, that, among other things, revises the manner in which the “average manufacturer price” is to be calculated by manufacturers
participating in the program and implements certain amendments to the Medicaid rebate statute created under the Affordable Care Act.
Further, there have been judicial and Congressional challenges to certain aspects of the Affordable Care Act, and we expect there will be
additional challenges and amendments to the Affordable Care Act in the future. Since January 2017, the President of the United States has
signed two Executive Orders and other directives designed to delay the implementation of any certain provisions of the Affordable Care
Act or otherwise circumvent some of the requirements for health insurance mandated by the Affordable Care Act. The Tax Cuts and Jobs
Act of 2017 includes a provision repealing, effective January 1, 2019, the tax-based shared responsibility payment imposed by the
Affordable Care Act on certain individuals who fail to maintain qualifying health coverage for all or part of a year that is commonly
referred to as the “individual mandate.” Congress will likely consider other legislation to replace elements of the Affordable Care Act. The
Affordable Care Act is likely to continue the downward pressure on pharmaceutical pricing and may also increase our regulatory burdens
and operating costs. We continue to evaluate the effect that the Affordable Care Act and its possible repeal and replacement has on our
business.

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Other legislative changes have been proposed and adopted since the Affordable Care Act was enacted. For example, in August

2011, President Obama signed into law the Budget Control Act of 2011, which, among other things, created the Joint Select Committee on
Deficit Reduction to recommend to Congress proposals in spending reductions. The Joint Select Committee did not achieve a targeted
deficit reduction of at least $1.2 trillion for the years 2013 through 2021, triggering the legislation’s automatic reduction to several
government programs. This included further reductions to Medicare payments to providers of 2% per fiscal year, which went into effect in
April 2013 and, due to subsequent legislative amendments to the statute, will stay in effect through 2025 unless additional Congressional
action is taken. Additionally, in January 2013, the American Taxpayer Relief Act of 2012 was signed into law, which, among other things,
reduced Medicare payments to several providers and increased the statute of limitations period in which the government may recover
overpayments to providers from three to five years.

Further, there have been several recent U.S. Congressional inquiries and proposed federal and state legislation designed to, among

other things, bring more transparency to drug pricing, review the relationship between pricing and manufacturer patient programs, reduce
the out-of-pocket cost of prescription drugs and reform government program reimbursement methodologies for drugs. Such scrutiny has
resulted in several recent Congressional inquiries and proposed and enacted federal and state legislation designed to, among other things,
bring more transparency to pharmaceutical product pricing, review the relationship between pricing and manufacturer patient programs,
and reform government program reimbursement methodologies for products. At the federal level, the current administration’s budget
proposal for fiscal year 2019 contains further drug price control measures that could be enacted during the 2019 budget process or in other
future legislation, including, for example, measures to permit Medicare Part D plans to negotiate the price of certain drugs under Medicare
Part B, to allow some states to negotiate drug prices under Medicaid, and to eliminate cost sharing for generic drugs for low-income
patients. Additionally, on May 11, 2018, the President of the United States laid out his administration’s “Blueprint to Lower Drug Prices
and Reduce Out-of-Pocket Costs” to reduce the cost of prescription drugs while preserving innovation and cures. The Department of Health
and Human Services, or HHS, has already started the process of soliciting feedback on some of these measures and, at the same time, is
immediately implementing others under its existing authority. Although some of these and other proposals will require authorization
through additional legislation to become effective, Congress and the U.S. presidential administration have each indicated that they will
continue to seek new legislative and/or administrative measures to control drug costs. At the state level, legislatures have become
increasingly aggressive in passing legislation and implementing regulations designed to control pharmaceutical and biological product
pricing, including price or patient reimbursement constraints, discounts, restrictions on certain product access and marketing cost disclosure
and transparency measures, and, in some cases, designed to encourage importation from other countries and bulk purchasing.

Moreover, the Drug Supply Chain Security Act, which was enacted in 2012 as part of the Food and Drug Administration Safety

and Innovation Act, imposes new obligations on manufacturers of pharmaceutical products related to product tracking and tracing.
Legislative and regulatory proposals have been made to expand post-approval requirements and restrict sales and promotional activities for
pharmaceutical products. We are not sure whether additional legislative changes will be enacted, whether the current regulations, guidance
or interpretations will be changed, or what the impact of such changes on our business, if any, may be. In addition, increased scrutiny by
the U.S. Congress of the FDA’s approval process may significantly delay or prevent marketing approval, as well as subject us to more
stringent product labeling and post-marketing testing and other requirements.

We expect that additional state and federal healthcare reform measures will be adopted in the future, any of which could limit the

amounts that federal and state governments will pay for healthcare products and services, which could result in reduced demand for our
product candidates or additional pricing pressures.

Product liability lawsuits against us could cause us to incur substantial liabilities and to limit commercialization of any products that we
may develop.

We face an inherent risk of product liability exposure related to the testing of our product candidates in human clinical trials and
related to the commercial sale of our products. Product liability claims may be brought against us by subjects enrolled in our clinical trials,
patients, healthcare providers or others using, administering or selling our products. For example, we may be sued if any product we sell
allegedly causes injury or is found to be otherwise unsuitable during product testing, manufacturing, marketing or sale. Any such product
liability claims may include allegations of defects in manufacturing, defects in design, a failure to warn of dangers inherent in the product,
negligence,  strict  liability  and  a  breach  of  warranties.  Claims  could  also  be  asserted  under  state  consumer  protection  acts.  If  we  cannot
successfully defend ourselves against claims that our product candidates or products that we may develop caused injuries, we could incur
substantial liabilities. Regardless of merit or eventual outcome, liability claims may result in:

•

•

decreased  demand  for  any  product  candidates  or  products  that  we  may
develop;

termination  of  clinical 
programs;

trial  sites  or  entire 

trial

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•

injury  to  our  reputation  and  significant  negative  media
attention;

• withdrawal 
participants;

of 

clinical 

trial

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significant  costs 
litigation;

to  defend 

the 

related

substantial  monetary  awards 
patients;

to 

trial  subjects  or

loss 
revenue;

of

product 
restrictions;

recalls,  withdrawals  or 

labeling,  marketing  or  promotional

diversion  of  management  and  scientific  resources  from  our  business
operations;

the  inability  to  commercialize  any  products  that  we  may  develop;
and

a  decline 
price.

in  our  stock

We currently hold product and clinical trial liability insurance coverage, but it might not adequately cover all liabilities that we
incur. We might not be able to maintain clinical trial insurance coverage at a reasonable cost or in an amount adequate to satisfy any liability
that  may  arise.  We  also  maintain  insurance  coverage  for  our  commercially  available  products,  which  might  not  adequately  cover  all
liabilities that we may incur. We might not be able to maintain insurance coverage for our approved products at a reasonable cost or in an
amount adequate to satisfy any liability that may arise. Large judgments have been awarded in class action lawsuits based on drugs that had
unanticipated  side  effects. A  product  liability  claim  or  series  of  claims  brought  against  us,  whether  or  not  successful,  but  particularly  if
judgments exceed our insurance coverage, could decrease our cash and adversely affect our reputation and business.

Our relationships with commercial and government customers, healthcare providers, and third ‑party payors and others are subject to
applicable anti‑kickback, fraud and abuse, transparency and other healthcare related laws, regulations and requirements, which could
expose us to criminal sanctions, civil penalties, exclusion from participation in federal healthcare programs, contractual damages and
consequences, reputational harm, administrative burdens and diminished profits and future earnings.

Pharmaceutical companies participating in federal and/or state healthcare programs such as Medicare and Medicaid are subject to a
multitude of federal and state laws and regulations which are intended to address and prevent “fraud and abuse”. These laws also apply to
the  physicians  and  third‑party  payors  who  play  a  primary  role  in  the  recommendation  and  prescription  of  our  commercially-available
products.  Our  arrangements  with  providers,  payors,  and  patients  may  expose  us  to  broadly-applicable  fraud  and  abuse  laws.  These  laws
may constrain the business or financial arrangements and relationships through which we market, sell, and distribute our products. There
are also laws, regulations, and requirements applicable to the award and performance of federal grants and contracts.

Actions resulting in violations of these laws regulations, and requirements may result in civil and criminal liability, damages and
restitution,  as  well  as  exclusion  from  participation  in  federal  healthcare  programs,  corporate  integrity  agreements,  deferred  prosecution
agreements, debarment from government contracts and grants and refusal of future orders under existing contracts or contractual damages,
and other consequences. Restrictions under applicable federal and state healthcare related laws and regulations, include the following:

•

•

the  federal Anti‑Kickback  Statute  prohibits  persons  from,  among  other  things,  knowingly  and  willfully  soliciting,  offering,
receiving or providing remuneration, directly or indirectly, overtly or covertly, in cash or in kind, to induce or reward, or in
return for, the referral of an individual for the furnishing or arranging for the furnishing, or the purchase, lease or order, or
arranging  for  or  recommending  purchase,  lease  or  order,  of  any  good  or  service  for  which  payment  may  be  made  under  a
federal healthcare program such as Medicare or Medicaid;

the civil federal False Claims Act imposes civil penalties, including through civil whistleblower or qui tam actions, against
individuals or entities for knowingly presenting, or causing to be presented, to the federal government, claims for payment that
are false or fraudulent; knowingly making, using or causing to be made or used, a false record or statement to get a false or
fraudulent claim paid or approved by the government; conspiring to defraud the government by getting a false or fraudulent
claim  paid  or  approved  by  the  government;  or  knowingly  making,  using  or  causing  to  be  made  or  used  a  false  record  or
statement to avoid, decrease or conceal an obligation to pay money to the federal government. Civil False Claims Act liability
may be imposed for Medicare or Medicaid overpayments, for example, overpayments caused by understated rebate amounts,
that  are  not  refunded  within  60  days  of  discovering  the  overpayment,  even  if  the  overpayment  was  not  cause  by  a  false  or
fraudulent act;

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•

•

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the  criminal  federal  False  Claims Act  imposes  criminal  fines  or  imprisonment  against  individuals  or  entities  who  willfully
make or present a claim to the government knowing such claim to be false, fictitious or fraudulent;

the Veterans Health Care Act requires manufacturers of covered drugs to offer them for sale on the Federal Supply Schedule,
which requires compliance with applicable federal procurement laws and regulations and subjects us to contractual remedies
as well as administrative, civil and criminal sanctions;

the  federal  Health  Insurance  Portability  and  Accountability  Act  and  its  related  regulations,  collectively  HIPAA,  impose
criminal  liability  for,  among  other  actions,  knowingly  and  willfully  executing  a  scheme  to  defraud  any  healthcare  benefit
program, knowingly and willfully embezzling or stealing from a health care benefit program, willfully obstructing a criminal
investigation of a health care offense, or knowingly and willfully making false statements relating to healthcare matters;

• HIPAA,  as  amended  by  the  Health  Information  Technology  for  Economic  and  Clinical  Health  Act  of  2009  and  its
implementing regulations, also imposes obligations on certain covered entity health care providers, health plans, and health
care clearinghouses as well as their business associates that perform certain services involving individually identifiable health
information,  including  mandatory  contractual  terms,  with  respect  to  safeguarding  the  privacy,  security  and  transmission  of
individually identifiable health information, as well as directly applicable privacy and security standards and requirements

•

•

•

•

the civil monetary penalties statute imposes penalties against any person or entity who, among other things, is determined to
have presented or caused to be presented a claim to a federal health program that the person knows or should know is for an
item or service that was not provided as claimed or is false or fraudulent;

the federal Physician Sunshine Act, created under Section 6002 of the Affordable Care Act and its implementing regulations,
requires  manufacturers  of  drugs,  devices,  biologics  and  medical  supplies  for  which  payment  is  available  under  Medicare,
Medicaid or the Children’s Health Insurance Program (with certain exceptions) to report annually to the Centers for Medicare
and Medicaid Services, or CMS, information related to payments or other “transfers of value” made to physicians (defined to
include  doctors,  dentists,  optometrists,  podiatrists  and  chiropractors)  and  teaching  hospitals,  and  requires  applicable
manufacturers and applicable group purchasing organizations to report annually to CMS ownership and investment interests
held by physicians (as defined above) and their immediate family members;

the FCPA prohibits any U.S. individual or business from paying, offering, or authorizing payment or offering of anything of
value,  directly  or  indirectly,  to  any  foreign  official,  political  party  or  candidate  for  the  purpose  of  influencing  any  act  or
decision of the foreign entity in order to assist the individual or business in obtaining or retaining business. The FCPA also
obligates  companies  whose  securities  are  listed  in  the  United  States  to  comply  with  accounting  provisions  requiring  the
company  to  maintain  books  and  records  that  accurately  and  fairly  reflect  all  transactions  of  the  corporation,  including
international  subsidiaries,  and  to  devise  and  maintain  an  adequate  system  of  internal  accounting  controls  for  international
operations; and

analogous or similar state, federal, and foreign laws, regulations, and requirements such as state anti‑kickback and false claims
laws, which may apply to sales or marketing arrangements and claims involving healthcare items or services reimbursed by
non‑governmental third‑party payors, including private insurers; state and foreign laws that require pharmaceutical companies
to  comply  with  the  pharmaceutical  industry’s  voluntary  compliance  guidelines  and  the  applicable  compliance  guidance
promulgated  by  the  federal  government  or  otherwise  restrict  payments  that  may  be  made  to  healthcare  providers;  state  and
foreign  laws  that  require  drug  manufacturers  to  report  information  related  to  payments  and  other  transfers  of  value  to
physicians  and  other  healthcare  providers  or  marketing  expenditures;  laws,  regulations,  and  requirements  applicable  to  the
award and performance of federal contracts and grants and state, federal and foreign laws that govern the privacy and security
of health and other information in certain circumstances, many of which differ from each other in significant ways and often
are not preempted by HIPAA, thus complicating compliance efforts.

Efforts  to  ensure  that  our  business  arrangements  with  third  parties  will  comply  with  applicable  healthcare  laws  and  regulations
involve substantial costs. For example, we must ensure that all applicable price concessions are included in prices calculated and reported to
federal  agencies.  Because  of  the  breadth  of  these  laws  and  the  narrowness  of  the  statutory  exceptions  and  safe  harbors  available,  it  is
possible that governmental authorities will conclude that our business practices do not comply with current or future statutes, regulations,
or  case  law  interpreting  applicable  fraud  and  abuse  or  other  healthcare  laws  and  regulations.  In  addition,  recent  health  care  reform
legislation has strengthened these laws. For example, recent case law from the U.S. Supreme Court interpreted the federal False Claims Act
to include liability for implied false certifications, in certain instances. If our operations are found to be in violation of any of these

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laws  or  any  other  governmental  regulations  or  requirements  that  may  apply  to  us,  we  may  be  subject  to  significant  civil,  criminal  and
administrative  penalties,  damages,  fines,  imprisonment,  restitution  exclusion  from  government  funded  healthcare  programs,  such  as
Medicare and Medicaid, corporate integrity agreements, deferred prosecution agreements, debarment from government contracts and grants
and  refusal  of  future  orders  under  existing  contracts,  contractual  damages,  the  curtailment  or  restructuring  of  our  operations  and  other
consequences. If any of the physicians or other healthcare providers or entities with whom we expect to do business are found not to be in
compliance with applicable laws, that person or entity may be subject to criminal, civil or administrative sanctions, including exclusions
from government funded healthcare programs. Moreover, availability of any federal grant funds which we may receive or for which we
may apply is subject to federal appropriations law. Grant funding may also be withdrawn or denied for other reasons.

We may be subject to numerous and varying privacy and security laws, and our failure to comply could result in penalties and

reputational damage.

We maintain a large quantity of sensitive information, including confidential business information and information associated with
clinical  trials.  If  our  security  measures  are  breached  or  fail  and/or  are  bypassed  because  of  third-party  action,  inadvertent  disclosures
through  technological  or  human  error  (including  employee  error),  malfeasance,  hacking,  ransomware,  social  engineering  (including
phishing schemes), computer viruses, malware, or otherwise, unauthorized acquisition of or access to sensitive information may occur. As
a result, our reputation could be damaged, our business might suffer, information might be lost, and we could face damages for breach of
contract, penalties for violation of applicable laws or regulations, costly litigation or government investigations, and significant costs for
remediation  and  remediation  efforts  to  prevent  future  occurrences.  The  harm  associated  with  these  negative  results  is  likely  to  be
exacerbated if the affected information is personally identifiable.

We  may  be  subject  to  laws  and  regulations  governing  the  privacy  and  security  of  personal  information,  including  regulations
pertaining to health information. The legislative and regulatory landscape for privacy and data security continues to evolve, and there has
been an increasing focus on privacy and data security issues that may affect our business. In the U.S., there are numerous federal and state
privacy and data security laws and regulations that govern the collection, use, disclosure, and protection of personal information, including
federal  and  state  health  information  privacy  laws,  federal  and  state  security  breach  notification  laws,  and  federal  and  state  consumer
protection laws. Each of these laws is subject to varying interpretations by courts and government agencies, creating complex compliance
issues  for  us.  If  we  fail  to  comply  with  applicable  laws  and  regulations,  we  could  be  subject  to  penalties  or  sanctions.  For  example,
violations of the Health Insurance Portability and Accountability Act (“HIPAA”) may result in civil fines of up to $57,051 per violation and
a maximum civil penalty of $1,711,533in a calendar year for violations of the same requirement, as well as criminal penalties. Recently,
the  U.S.  Department  of  Health  and  Human  Services  Office  for  Civil  Rights,  which  enforces  HIPAA,  appears  to  have  increased  its
enforcement activities. Additionally, state attorneys general may bring civil actions seeking either injunctions or damages in response to
violations of HIPAA that threaten the privacy of state residents. Privacy and data security has become an area of emphasis for some state
legislatures.  For  example,  California  recently  enacted  and  amended  the  California  Consumer  Protection  Act  (“CCPA”),  which  could
present  implementation  challenges  and  risk  of  enforcement.  There  may  be  additional  amendments  to  the  CCPA,  and  regulations
promulgated pursuant to the CCPA may alter how the law applies; therefore, the extent to and manner in which the CCPA would apply to
our operations is unclear. In addition to the risk associated with enforcement, compliance with these evolving laws, rules, and regulations
regarding the privacy, security and protection of personal information could result in higher compliance and technology costs for us and
present challenges for our business model.

There  are  numerous  federal  and  state  laws  that  generally  require  notice  to  affected  individuals,  regulators,  and  sometimes  the
media  or  credit  reporting  agencies  in  the  event  of  a  data  breach  impacting  personal  information.  For  example,  at  the  federal  level,  the
HIPAA  Breach  Notification  Rule  mandates  notification  of  breaches  affecting  protected  health  information  to  affected  individuals  and
regulators  under  conditions  set  forth  in  the  Rule.  Covered  Entities  must  report  breaches  of  unsecured  protected  health  information  to
affected individuals without unreasonable delay, but not to exceed 60 days of discovery of the breach by a Covered Entity or its agents.
Notification must also be made to Department of Health and Human Services and, in certain circumstances involving large breaches, to the
media.  Business  Associates  must  report  breaches  of  unsecured  protected  health  information  to  Covered  Entities  within  60  days  of
discovery of the breach by the Business Associate or its agents. All states, the District of Columbia, Guam, Puerto Rico, and the Virgin
Islands have enacted data breach notification laws. These laws may impose notification obligations in addition to, or inconsistent with, the
HIPAA Breach Notification Rule when a data breach implicates protected health information. In that event that we fail to detect or timely
report  a  data  breach  we  may  be  subject  to  significant  penalties  under  federal  and  state  law.  In  the  event  that  we  report  a  data  breach  as
required by federal or state law, federal or state regulators may initiate an investigation into, and/or litigation related to, our privacy or data
security practices. Private plaintiffs may also initiate costly class-action litigation following a data breach.

Numerous other countries have, or are developing, laws governing the collection, use, and transmission of personal information.
These  laws  often  impose  significant  compliance  obligations.  For  example,  since  May  25,  2018,  the  General  Data  Protection  Regulation
(“GDPR”),  has  imposed  more  stringent  obligations  and  restrictions  on  the  ability  to  collect,  analyze,  and  transfer  personal  information,
including health data from clinical trials and substantial fines for breaches of the data protection rules in the European Economic Area.

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To the extent that our activities are or become subject to the GDPR, we may need to devote significant effort and resources to complying
with those legal regimes. Any failure to comply with the rules arising from the GDPR could lead to government enforcement actions and
significant  penalties  against  us  and  adversely  impact  our  operating  results.  Under  GDPR,  for  example,  fines  of  $20.0  million  or  4%  of
global turnover may be imposed for violations.

If we fail to attract and keep management and other key personnel, as well as our board members, we may be unable to develop our
product candidates or otherwise implement our business plan.

We might not be able to attract or retain qualified management and other key personnel in the future due to the intense competition
for qualified personnel among biotechnology, pharmaceutical and other businesses. Our industry has experienced a high rate of turnover of
management  personnel  in  recent  years. As  such,  we  could  have  difficulty  attracting  experienced  personnel  to  our  company  and  may  be
required to expend significant financial resources in our employee recruitment and retention efforts. Many of the other biotechnology and
pharmaceutical companies with whom we compete for qualified personnel have greater financial and other resources, different risk profiles
and  longer  histories  in  the  industry  than  we  do.  They  also  may  provide  more  diverse  opportunities  and  better  chances  for  career
advancement. Some of these characteristics may be more appealing to high quality candidates than that which we have to offer. If we are
not able to attract and retain the necessary personnel to accomplish our business objectives, we may experience constraints that will impede
significantly our ability to implement our business strategy and achieve our business objectives.

In addition, we have scientific and clinical advisors who assist us in formulating our development and clinical strategies. These
advisors are not our employees and may have commitments to, or consulting or advisory contracts with, other entities that may limit their
availability to us. In addition, our advisors may have arrangements with other companies to assist those companies in developing products
or technologies that may compete with ours.

If our employees, independent contractors, principal investigators, CROs, manufacturers, consultants or vendors commit fraud or other
misconduct,  including  noncompliance  with  regulatory  standards  and  requirements  and  insider  trading,  our  business  may  experience
serious adverse consequences.

We are exposed to the risk that our employees, independent contractors, principal investigators, CROs, manufacturers, consultants
and  vendors  may  engage  in  fraudulent  or  other  illegal  activity.  Misconduct  by  these  parties  could  include  intentional,  reckless  and/or
negligent  conduct  or  disclosure  of  unauthorized  activities  to  us  that  violates:  (1)  FDA  regulations,  including  those  laws  requiring  the
reporting of true, complete and accurate information to the FDA, (2) manufacturing standards, (3) federal and state healthcare fraud and
abuse laws and regulations or (4) laws that require the true, complete and accurate reporting of financial information or data. Specifically,
sales,  marketing  and  business  arrangements  in  the  healthcare  industry  are  subject  to  extensive  laws  and  regulations  intended  to  prevent
fraud,  kickbacks,  self‑dealing  and  other  abusive  practices.  These  laws  and  regulations  may  restrict  or  prohibit  a  wide  range  of  pricing,
discounting, marketing and promotion, sales commission, customer incentive programs and other business arrangements. The improper use
of information obtained in the course of clinical trials could also result in significant legal sanctions and serious harm to our reputation. In
addition, federal procurement laws and regulations impose substantial penalties for misconduct in connection with government contracts
and require contractors to maintain a code of business conduct and ethics. We have adopted a Code of Business Conduct and Ethics, but it
is not always possible to identify and deter misconduct by our employees and other third parties, and the precautions we take to detect and
prevent  this  activity  might  not  be  effective  in  controlling  unknown  or  unmanaged  risks  or  losses  or  in  protecting  us  from  governmental
investigations or other actions or lawsuits stemming from a failure to be in compliance with such laws or regulations. If any such actions are
instituted against us, and we are not successful in defending ourselves or asserting our rights, those actions could have a significant impact
on our business, including regulatory enforcement action, the imposition of significant criminal and civil fines, penalties, or other sanctions,
including  imprisonment,  exclusion  from  participation  in  federal  healthcare  programs,  and  deferred  prosecution  and  corporate  integrity
agreements.

In addition, during the course of our operations, our directors, executives and employees may have access to material, nonpublic
information  regarding  our  business,  our  results  of  operations  or  potential  transactions  we  are  considering.  We  have  adopted  an  Insider
Trading and Window Period Policy, but despite the adoption of such policy, we might not be able to prevent a director, an executive or an
employee  from  trading  in  our  common  stock  on  the  basis  of,  or  while  having  access  to,  material,  nonpublic  information.  If  a  director,
executive or employee was to be investigated, or an action was to be brought against a director, executive or employee for insider trading, it
could have a negative impact on our reputation and our stock price. Such a claim, with or without merit, could also result in substantial
expenditures of time and money, and divert attention of our management team from other tasks important to the success of our business.

We may fail to realize all of the anticipated benefits of recent acquisitions or those benefits may take longer to realize than expected,
and  our  future  results  of  will  suffer  if  we  do  not  effectively  manage  our  expanded  operations  following  the  completion  of  the
acquisitions.

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In  November  2017  we  acquired  TRx  Pharmaceuticals,  LLC  and  its  franchise  of  commercial  medications,  in  February  2018  we
acquired  pediatric  products  from Avadel  U.S.  Holdings,  Inc.,  and  in  September  2018  we  acquired  Ichorion’s  in-process  research  and
development  for  three  preclinical  therapies  for  inherited  metabolic  disorder.  Our  ability  to  realize  the  anticipated  benefits  of  these
acquisitions  will  depend,  to  a  large  extent,  on  our  ability  to  integrate  the  acquisitions  into  our  business,  which  might  be  particularly
challenging  because  these  are  our  first  commercial  operations. As  a  result,  our  management  team  will  devote  a  significant  amount  of
attention and resources into integrating these acquisitions into our business practices and operations. This integration process may disrupt
our current business.

Our  future  success  depends,  in  part,  upon  our  ability  to  integrate  and  manage  these  new  product  lines,  pipeline  assets,  and  any
future acquisitions, which poses substantial challenges for management, including challenges related to the management and monitoring of
new operations and associated increased costs and complexity. If we are unsuccessful in integrating and managing our new product lines,
pipeline assets, and any future acquisitions, our operations and financial condition could be adversely affected, and we might not be able to
take advantage of business development opportunities anticipated when making the acquisitions.

We may encounter difficulties in managing our growth and expanding our operations successfully.

As  we  seek  to  advance  our  product  candidates  through  clinical  trials,  we  will  need  to  expand  our  development,  regulatory,
manufacturing,  administrative,  marketing  and  sales  capabilities  or  contract  with  third  parties  to  provide  these  capabilities  for  us. As  our
operations expand, we expect that we will need to manage additional relationships with various strategic partners, suppliers and other third
parties. Future growth will impose significant added responsibilities on members of management. Our future financial performance and our
ability to commercialize our product candidates and to compete effectively will depend, in part, on our ability to manage any future growth
effectively.  To  that  end,  we  must  be  able  to  manage  our  development  efforts  and  clinical  trials  effectively  and  hire,  train  and  integrate
additional management, administrative and sales and marketing personnel. The hiring, training and integration of new employees may be
more difficult, costly and/or time‑consuming for us because we have fewer resources than a larger organization. We might not be able to
accomplish these tasks, and our failure to accomplish any of them could prevent us from successfully growing our company.

If, in the future, we are unable to grow  our  own  sales,  or  establish  marketing  and  distribution  capabilities  or  enter  into  licensing  or
collaboration agreements for these purposes, we might not be successful in commercializing our product candidates.

We currently have a relatively small number of employees and did not have a sales or marketing infrastructure until we acquired
TRx. We do not have any significant sales, marketing or distribution experience as a company. To develop and expand our internal sales,
distribution and marketing capabilities, we will have to invest significant amounts of financial and management resources, some of which
will be committed prior to any confirmation that any new product candidates will be approved. For product candidates for which we decide
to perform sales, marketing and distribution functions ourselves, we could face a number of additional risks, including:

•

•

•

•

•

•

•

our  inability  to  recruit  and  retain  adequate  numbers  of  effective  sales  and  marketing
personnel;

inability  of  marketing  personnel 
materials;

to  develop  effective  marketing

the  inability  of  sales  personnel  to  obtain  access  to  physicians  or  educate  adequate  numbers  of  physicians  on  the  clinical
benefits of our products to achieve market acceptance;

the lack of complementary products to be offered by sales personnel, which may put us at a competitive disadvantage relative
to companies with more extensive product lines;

the  costs  associated  with  training  sales  personnel  on  legal  compliance  matters  and  monitoring  their
actions;

liability  for  sales  personnel  failing  to  comply  with  the  applicable  legal  requirements;
and

unforeseen  costs  and  expenses  associated  with  creating  an  independent  sales  and  marketing
organization.

Where and when appropriate, we may elect to utilize contract sales forces or strategic partners to assist in the commercialization of
our  product  candidates.  If  we  enter  into  arrangements  with  third  parties  to  perform  sales,  marketing  and  distribution  services  for  our
products,  the  resulting  revenues  or  the  profitability  from  these  revenues  to  us  are  likely  to  be  lower  than  if  we  had  sold,  marketed  and
distributed our products ourselves. In addition, we might not be successful in entering into arrangements with third parties to sell, market
and distribute our product candidates or may be unable to do so on terms that are favorable to us. We likely will have little control over
such third parties, and any of these third parties may fail to devote the necessary resources and attention to sell, market and distribute our

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products effectively. Such third parties may also not comply with the applicable regulatory requirements, which could potentially expose us
to regulatory and legal enforcement actions.

Risks Related to Our Dependence on Third Parties

We might not succeed in establishing and maintaining development collaborations, which could adversely affect our ability to develop
and commercialize product candidates.

A  part  of  our  strategy  is  to  enter  into  product  development  collaborations  in  the  future,  including  collaborations  with  major
biotechnology  or  pharmaceutical  companies  for  the  development  or  commercialization  of  our  current  and  future  product  candidates. We
also face significant competition in seeking appropriate development partners and the negotiation process is time‑consuming and complex.
We might not succeed in our efforts to establish development collaborations or other alternative arrangements for any of our existing or
future  product  candidates  and  programs  because  our  research  and  development  pipeline  may  be  insufficient,  our  product  candidates  and
programs may be deemed to be at too early a stage of development for collaborative effort and/or third parties might not view our product
candidates and programs as having the requisite potential to demonstrate safety and efficacy.

Furthermore, any collaborations that we enter into might not be successful. The success  of  our  development  collaborations  will
depend heavily on the efforts and activities of our collaborators. Furthermore, any collaborations that we enter into might not be successful.
The success of our development collaborations will depend heavily on the efforts and activities of our collaborators. Our relationship with
any future collaborations may pose several risks, including the following:

•

•

•

•

•

collaborators have significant discretion in determining the amount and timing of the efforts and resources that they will apply
to these collaborations;

collaborators may not perform their obligations as
expected;

the nonclinical studies and clinical trials conducted as part of these collaborations may not be
successful;

collaborators may not pursue development and commercialization of any product candidates that achieve regulatory approval
or may elect not to continue or renew development or commercialization programs based on nonclinical study or clinical trial
results, changes in the collaborators’ strategic focus or available funding or external factors, such as an acquisition, that divert
resources or create competing priorities;

collaborators may delay nonclinical studies and clinical trials, provide insufficient funding for nonclinical studies and clinical
trials, stop a nonclinical study or clinical trial or abandon a product candidate, repeat or conduct new nonclinical studies or
clinical trials or require a new formulation of a product candidate for nonclinical studies or clinical trials;

• we may not have access to, or may be restricted from disclosing, certain information regarding product candidates being

developed or commercialized under a collaboration and, consequently, may have limited ability to inform our stockholders
about the status of such product candidates;

•

•

•

•

collaborators could independently develop, or develop with third parties, products that compete directly or indirectly with our
product candidates if the collaborators believe that competitive products are more likely to be successfully developed or can
be commercialized under terms that are more economically attractive than ours;

product candidates developed in collaboration with us may be viewed by our collaborators as competitive with their own
product candidates or products, which may cause collaborators to cease to devote resources to the commercialization of our
product candidates;

a collaborator with marketing and distribution rights to one or more of our product candidates that achieve regulatory approval
may not commit sufficient resources to the marketing and distribution of any such product candidate;

disagreements with collaborators, including disagreements over proprietary rights, contract interpretation or the preferred
course of development of any product candidates, may cause delays or termination of the research, development or
commercialization of such product candidates, may lead to additional responsibilities for us with respect to such product
candidates or may result in litigation or arbitration, any of which would be time consuming and expensive;

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•

•

•

•

•

collaborators may not properly maintain or defend our intellectual property rights or may use our proprietary information in
such a way as to invite litigation that could jeopardize or invalidate our intellectual property or proprietary information or
expose us to potential litigation;

disputes may arise with respect to the ownership or inventorship of intellectual property developed pursuant to our
collaborations;

collaborators may infringe the intellectual property rights of third parties, which may expose us to litigation and potential
liability;

the terms of our collaboration agreement may restrict us from entering into certain relationships with other third parties,
thereby limiting our options; and

collaborations may be terminated for the convenience of the collaborator and, if terminated, we could be required to raise
additional capital to pursue further development or commercialization of the applicable product candidates.

Even  if  we  are  successful  in  our  efforts  to  establish  development  collaborations,  the  terms  that  we  agree  upon  might  not  be
favorable  to  us  and  we  might  not  be  able  to  maintain  such  development  collaborations  if,  for  example,  development  or  approval  of  a
product  candidate  is  delayed  or  sales  of  an  approved  product  candidate  are  disappointing.  Any  delay  in  entering  into  development
collaboration agreements related to our product candidates could delay the development and commercialization of our product candidates
and  reduce  their  competitiveness  if  they  reach  the  market. Additionally,  collaborations  with  pharmaceutical  or  biotechnology  companies
and other third parties often are terminated or allowed to expire by the other party. Any such termination or expiration would adversely
affect us financially and could harm our business reputation.

If we fail to establish and maintain additional development collaborations related to our product candidates:

•

•

the  development  of  certain  of  our  current  or  future  product  candidates  may  be  terminated  or
delayed;

our  cash  expenditures  related  to  development  of  certain  of  our  current  or  future  product  candidates  would  increase
significantly and we may need to seek additional financing, which might not be available on favorable terms, or at all;

• we may be required to hire additional employees or otherwise develop expertise, such as sales and marketing expertise, for

which we have not budgeted;

• we  will  bear  all  of  the  risk  related  to  the  development  of  any  such  product

candidates;

• we may have to expend unexpected efforts and funds if we are unable to obtain the results of third-party clinical trials;

and

•

the  competitiveness  of  any  product  candidate  that  is  commercialized  could  be
reduced.

We rely on third parties to conduct, supervise and monitor our clinical trials. The failure of these third parties to successfully carry out
their  contractual  duties  or  meet  expected  deadlines  could  substantially  harm  our  business  because  we  might  not  obtain  marketing
approval for or commercialize our product candidates in a timely manner or at all.

We rely upon third‑party CROs to monitor and manage data for our clinical programs. We rely on these parties for execution of
our clinical trials and, while we have agreements governing their activities, we have limited influence over their actual performance and
control  only  certain  aspects  of  their  activities.  Nevertheless,  we  are  responsible  for  ensuring  that  each  of  our  studies  is  conducted  in
accordance with the applicable protocol, legal, regulatory and scientific standards, and our reliance on the CROs does not relieve us of our
regulatory responsibilities. We, our clinical trial sites, and our CROs are required to comply with GCP requirements, which are regulations
and guidelines enforced by the FDA, the Competent Authorities of the Member States of the European Economic Area and comparable
foreign  regulatory  authorities  for  all  of  our  products  in  clinical  development.  Regulatory  authorities  enforce  these  GCP  requirements
through  periodic  inspections  of  trial  sponsors,  principal  investigators  and  trial  sites.  If  we,  any  of  our  CROs  or  clinical  trial  sites  fail  to
comply  with  applicable  GCP  requirements,  the  clinical  data  generated  in  our  clinical  trials  may  be  deemed  unreliable  and  the  FDA  or
comparable foreign regulatory authorities may require us to perform additional clinical trials before approving our marketing applications,
if at all. In addition, we are required to report certain financial interests of our third‑party investigators if these relationships exceed certain
financial  thresholds  or  meet  other  criteria.  The  FDA  or  comparable  foreign  regulatory  authorities  may  question  the  integrity  of  the  data
from those clinical trials conducted by principal investigators who previously served or currently serve as scientific advisors or consultants
to us from time to time and receive cash compensation in connection with such services or otherwise receive compensation

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from us that could be deemed to impact study outcome, proprietary interests in a product candidate, certain company equity interests, or
significant payments of other sorts. We cannot assure you that upon inspection by a given regulatory authority, such regulatory authority
will determine that any of our clinical trials complies with GCP requirements. In addition, we must conduct our clinical trials with product
produced under applicable GMP requirements. Failure to comply with these regulations may require us to repeat preclinical and clinical
trials, which would delay the marketing approval process.

Our CROs and clinical trial sites are not our employees, and, except for remedies available to us under our agreements with such
CROs and clinical trial sites, we cannot control whether or not they devote sufficient time and resources to our ongoing clinical, nonclinical
and  preclinical  programs.  These  CROs  and  clinical  trial  sites  may  also  have  relationships  with  other  commercial  entities,  including  our
competitors,  for  whom  they  may  also  be  conducting  clinical  trials  or  other  drug  development  activities  that  could  harm  our  competitive
position. If CROs or clinical trial sites do not successfully carry out their contractual duties or obligations or meet expected deadlines, or if
the  quality  or  accuracy  of  the  clinical  data  they  obtain  is  compromised  due  to  the  failure  to  adhere  to  our  clinical  protocols,  regulatory
requirements or for other reasons, our clinical trials may be extended, delayed or terminated and we might not be able to obtain marketing
approval for or successfully commercialize our product candidates or we may be subject to regulatory enforcement actions. As a result, our
results of operations and the commercial prospects for our product candidates would be harmed, our costs could increase and our ability to
generate revenues could be delayed. To the extent we are unable to successfully identify and manage the performance of third‑party service
providers in the future, our business may be adversely affected.

Switching  or  adding  CROs  involves  substantial  cost  and  requires  extensive  management  time  and  focus.  In  addition,  there  is  a
natural transition period when a new CRO commences work. As a result, delays occur, which can materially impact our ability to meet our
desired clinical development timelines. Though we carefully manage our relationships with our CROs, there can be no assurance that we
will not encounter similar challenges or delays in the future or that these delays or challenges will not have a material adverse impact on
our business, prospects, financial condition and results of operations.

We use third parties to manufacture all of our product candidates. This may increase the risk that we will not have sufficient quantities
of  our  product  candidates  to  conduct  our  clinical  trials  or  such  quantities  at  an  acceptable  cost,  which  could  result  in  the  delay,
prevention, or impairment of clinical development and commercialization of our product candidates.

We  do  not  own  or  operate,  and  have  no  plans  to  establish,  any  manufacturing  facilities  for  our  product  candidates.  We  have
limited personnel with experience in drug manufacturing and we lack the resources and the capabilities to manufacture any of our product
candidates on a clinical or commercial scale.

We currently outsource all manufacturing of our product candidates to third parties typically without any guarantee that there will
be sufficient supplies to fulfill our requirements or that we may obtain such supplies on acceptable terms. Any delays in obtaining adequate
supplies with respect to our product candidates may delay the development or commercialization of our other product candidates.

In addition, we do not currently have any agreements with third‑party manufacturers for the long‑term commercial supply of our
product candidates. We may be unable to enter agreements for commercial supply with third‑party manufacturers, or may be unable to do
so on acceptable terms. Even if we enter into these agreements, the various manufacturers of each product candidate will likely be single
source suppliers to us for a significant period of time.

The facilities used by our contract manufacturers to manufacture our product candidates must be approved by the FDA pursuant to
inspections that will be conducted after we submit our NDA to the FDA. While we are ultimately responsible for the manufacture of our
product candidates, other than through our contractual arrangements, we do not control the manufacturing process of, and are completely
dependent  on,  our  contract  manufacturing  partners  for  compliance  with  the  regulatory  requirements,  known  as  GMP  requirements,  for
manufacture  of  both  active  drug  substances  and  finished  drug  products  for  clinical  supply  and  eventually  for  commercial  supply,  if  we
receive regulatory approval. If our contract manufacturers cannot successfully manufacture material that conforms to our specifications and
the  strict  regulatory  requirements  of  the  FDA  or  other  regulatory  authorities,  we  will  not  be  able  to  secure  and/or  maintain  regulatory
approval  for  their  manufacturing  facilities.  Failure  of  our  contract  manufacturers  to  comply  with  the  applicable  regulatory  requirements
may also subject us to regulatory enforcement actions. In addition, other than through our contractual agreements, we have no control over
the ability of our contract manufacturers to maintain adequate quality control, quality assurance and qualified personnel. If the FDA or a
comparable foreign regulatory authority does not approve these facilities for the manufacture of our product candidates or if it withdraws
any such approval in the future, we may need to find alternative manufacturing facilities, which would significantly impact our ability to
develop, obtain marketing approval for or market our product candidates, if approved.

Reliance  on  third‑party  manufacturers  subjects  us  to  risks  that  would  not  affect  us  if  we  manufactured  the  product  candidates

ourselves, including:

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•

•

•

•

•

•

•

•

  reliance  on  the  third  parties  for  regulatory  compliance  and  quality
assurance;

the  possible  breach  of  the  manufacturing  agreements  by  the  third  parties  because  of  factors  beyond  our
control;

the  possible  misappropriation  of  our  proprietary  information,  including  trade  secrets  and  know-
how;

the possibility of termination or nonrenewal of the agreements by the third parties because of our breach of the manufacturing
agreement or based on their own business priorities;

the  disruption  and  costs  associated  with  changing  suppliers,  including  additional  regulatory
filings.

to 
failure 
obligations;

satisfy 

their  contractual  duties  or

inability 
consistently;

to  meet  our  product  specifications  and  quality  requirements

delay  or  inability  to  procure  or  expand  sufficient  manufacturing
capacity;

• manufacturing and/or product quality issues related to manufacturing development and scale-

up;

•

•

•

•

•

•

•

•

•

•

•

•

costs and validation of new equipment and facilities required for scale-
up;

failure  to  comply  with  applicable  laws,  regulations,  and  standards,  including  cGMP  and  similar  foreign
standards;
deficient 
keeping;

improper 

record-

or 

contractual  restrictions  on  our  ability 
manufacturers;

to  engage  additional  or  alternative

inability  to  negotiate  manufacturing  agreements  with  third  parties  under  commercially  reasonable
terms;

termination or nonrenewal of manufacturing agreements with third parties in a manner or at a time that is costly or damaging
to us;

reliance on a limited number of sources, and in some cases, single sources for product components, such that if we are unable
to secure a sufficient supply of these product components, we will be unable to manufacture and sell our product candidates or
any future product candidate in a timely fashion, in sufficient quantities or under acceptable terms;

lack  of  qualified  backup  suppliers  for  those  components  that  are  currently  purchased  from  a  sole  or  single  source
supplier;

lack  of  access  or  licenses  to  proprietary  manufacturing  methods  used  by  third-party  manufacturers  to  make  our  product
candidates;

operations  of  our  third-party  manufacturers  or  suppliers  could  be  disrupted  by  conditions  unrelated  to  our  business  or
operations, including the bankruptcy of the manufacturer or supplier or regulatory sanctions related to the manufacture of our
or other company’s products;

carrier  disruptions  or  increased  costs  that  are  beyond  our  control;
and

failure  to  deliver  our  products  under  specified  storage  conditions  and  in  a  timely
manner.

Our product candidates may compete with other products and product candidates for access to manufacturing facilities. There are
a limited number of manufacturers that operate under GMP regulations and that are both capable of manufacturing for us and willing to do
so. If our existing third‑party manufacturers, or the third parties that we engage in the future to manufacture a product for commercial sale
or  for  our  clinical  trials,  should  cease  to  continue  to  do  so  for  any  reason,  we  likely  would  experience  delays  in  obtaining  sufficient
quantities  of  our  product  candidates  for  us  to  meet  commercial  demand  or  to  advance  our  clinical  trials  while  we  identify  and  qualify
replacement suppliers. If for any reason we are unable to obtain adequate supplies of our product candidates or the drug substances used to

manufacture them, it will be more difficult for us to develop our product candidates and compete effectively.

Our suppliers are subject to regulatory requirements, covering manufacturing, testing, quality control, manufacturing, and record

keeping relating to our product candidates, and subject to ongoing inspections by the regulatory agencies. Failure by any of our suppliers

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to comply with applicable regulations may result in long delays and interruptions to our manufacturing capacity while we seek to secure
another  supplier  that  meets  all  regulatory  requirements,  as  well  as  market  disruption  related  to  any  necessary  recalls  or  other  corrective
actions.

Risks Related to Intellectual Property

If  we  are  unable  to  obtain  or  maintain  intellectual  property  rights,  or  if  the  scope  of  patent  protection  is  not  sufficiently  broad,
competitors could develop and commercialize products similar or identical to ours, and we might not be able to compete effectively in
our market.

Our  success  depends  in  significant  part  on  our  and  our  licensors’,  licensees’  or  collaborators’  ability  to  establish,  maintain  and
protect patents and other intellectual property rights and operate without infringing the intellectual property rights of others. We have filed
numerous patent applications both in the United States and in foreign jurisdictions to obtain patent rights to inventions we have discovered.
We have also licensed from third parties' rights to patent portfolios.

The  patent  prosecution  process  is  expensive  and  time‑consuming,  and  we  and  our  current  or  future  licensors,  licensees  or
collaborators might not be able to prepare, file and prosecute all necessary or desirable patent applications at a reasonable cost or in a timely
manner. It is also possible that we or our licensors, licensees or collaborators will fail to identify patentable aspects of inventions made in
the  course  of  development  and  commercialization  activities  before  it  is  too  late  to  obtain  patent  protection  on  them.  Moreover,  in  some
circumstances,  we  might  not  have  the  right  to  control  the  preparation,  filing  and  prosecution  of  patent  applications,  or  to  maintain  the
patents,  covering  technology  that  we  license  from  or  license  to  third  parties  and  are  reliant  on  our  licensors,  licensees  or  collaborators.
Therefore,  these  patents  and  applications  might  not  be  prosecuted  and  enforced  in  a  manner  consistent  with  the  best  interests  of  our
business. If our current or future licensors, licensees or collaborators fail to establish, maintain or protect such patents and other intellectual
property rights, such rights may be reduced or eliminated. If our licensors, licensees or collaborators are not fully cooperative or disagree
with us as to the prosecution, maintenance or enforcement of any patent rights, such patent rights could be compromised.

The  patent  position  of  biotechnology  and  pharmaceutical  companies  generally  is  highly  uncertain,  involves  complex  legal  and
factual questions and has in recent years been the subject of much litigation. As a result, the issuance, scope, validity, enforceability and
commercial value of our and our current or future licensors’, licensees’ or collaborators’ patent rights are highly uncertain. Our and our
licensors’,  licensees’  or  collaborators’  pending  and  future  patent  applications  might  not  result  in  patents  being  issued  which  protect  our
technology  or  products,  in  whole  or  in  part,  or  which  effectively  prevent  others  from  commercializing  competitive  technologies  and
products. The patent examination process may require us or our licensors, licensees or collaborators to narrow the scope of the claims of
our or our licensors’, licensees’ or collaborators’ pending and future patent applications, which may limit the scope of patent protection that
may be obtained. Our and our licensors’, licensees’ or collaborators’ patent applications cannot be enforced against third parties practicing
the technology claimed in such applications unless and until a patent issues from such applications, and then only to the extent the issued
claims cover the technology.

Furthermore,  given  the  amount  of  time  required  for  the  development,  testing  and  regulatory  review  of  new  product  candidates,
patents  protecting  such  candidates  might  expire  before  or  shortly  after  such  candidates  are  commercialized. As  a  result,  our  owned  and
licensed patent portfolio might not provide us with sufficient rights to exclude others from commercializing products similar or identical to
ours.  We  expect  to  seek  extensions  of  patent  terms  where  these  are  available  in  any  countries  where  we  are  prosecuting  patents.  This
includes  in  the  United  States  under  the  Drug  Price  Competition  and  Patent  Term  Restoration Act  of  1984,  which  permits  a  patent  term
extension  of  up  to  five  years  beyond  the  expiration  of  the  patent.  However,  the  applicable  authorities,  including  the  FDA  in  the  United
States,  and  any  equivalent  regulatory  authority  in  other  countries,  might  not  agree  with  our  assessment  of  whether  such  extensions  are
available,  and  may  refuse  to  grant  extensions  to  our  patents,  or  may  grant  more  limited  extensions  than  we  request.  If  this  occurs,  our
competitors may take advantage of our investment in development and clinical trials by referencing our clinical and preclinical data and
launch their product earlier than might otherwise be the case.

If  we  breach  the  license  agreements  related  to  our  product  candidates,  we  could  lose  the  ability  to  develop  and  commercialize  our
product candidates.

Our  commercial  success  depends  upon  our  ability,  and  the  ability  of  our  licensors  and  collaborators,  to  develop,  manufacture,
market  and  sell  our  product  candidates  and  use  our  and  our  licensors’  or  collaborators’  proprietary  technologies  without  infringing  the
proprietary rights of third parties. If we fail to comply with our obligations in the agreements under which we license intellectual property
rights from third parties or otherwise experience disruptions to our business relationships with our licensors, we could lose the ability to
continue  the  development  and  commercialization  of  our  product  candidates  or  face  other  penalties  under  these  agreements.  We  have
entered into exclusive license agreements with Merck & Co., Inc. and its affiliates ("Merck") pursuant to which Merck has granted us rights
to the compounds used in CERC-301 and the COMTi platform, including CERC‑406. We have also entered into an exclusive

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license,  development  and  commercialization  agreement  with  Eli  Lilly  and  Company  ("Lilly")  pursuant  to  which  we  received  exclusive
global  rights  to  develop  and  commercialize  CERC-611.  If  we  fail  to  comply  with  the  obligations  under  these  agreements,  including
payment terms, Merck and Lilly may have the right to terminate any of these agreements, in which event we might not be able to develop,
market  or  sell  the  relevant  product  candidate.  Such  an  occurrence  could  materially  adversely  affect  the  value  of  the  product  candidate
being  developed  under  any  such  agreement.  Termination  of  these  agreements  or  reduction  or  elimination  of  our  rights  under  these
agreements may result in our having to negotiate new or reinstated agreements, which might not be available to us on equally favorable
terms, or at all, or cause us to lose our rights under these agreements, including our rights to intellectual property or technology important to
our development programs. Any of these occurrences may harm our business, financial condition and prospects significantly.

Obtaining and maintaining our patent protection depends on compliance with various procedural, document submission, fee payment
and  other  requirements  imposed  by  governmental  patent  agencies,  and  our  patent  protection  could  be  reduced  or  eliminated  for
non‑compliance with these requirements.

Periodic maintenance and annuity fees on any issued patent are due to be paid to the United States Patent and Trademark Office,
or  USPTO,  and  foreign  patent  agencies  in  several  stages  over  the  lifetime  of  the  patent.  The  USPTO  and  various  foreign  governmental
patent agencies require compliance with a number of procedural, documentary, fee payment and other similar provisions during the patent
application process. While an inadvertent lapse can in many cases be cured by payment of a late fee or by other means in accordance with
the  applicable  rules,  there  are  situations  in  which  noncompliance  can  result  in  abandonment  or  lapse  of  the  patent  or  patent  application,
resulting in partial or complete loss of patent rights in the relevant jurisdiction. Non‑compliance events that could result in abandonment or
lapse of a patent or patent application include failure to respond to official actions within prescribed time limits, non‑payment of fees and
failure  to  properly  legalize  and  submit  formal  documents.  If  we  or  our  licensors  or  collaborators  fail  to  maintain  the  patents  and  patent
applications  covering  our  product  candidates,  our  competitors  might  be  able  to  enter  the  market,  which  would  have  a  material  adverse
effect on our business.

Third  parties  may  initiate  legal  proceedings  against  us  alleging  that  we  infringe  their  intellectual  property  rights,  or  we  may  initiate
legal proceedings against third parties to challenge the validity or scope of intellectual property rights controlled by third parties, the
outcome of which would be uncertain and could have a material adverse effect on the success of our business.

Third  parties  may  initiate  legal  proceedings  against  us  or  our  licensors  or  collaborators  alleging  that  we  or  our  licensors  or
collaborators infringe their intellectual property rights or we or our licensors or collaborators may initiate legal proceedings against third
parties to challenge the validity or scope of intellectual property rights controlled by third parties, including in oppositions, interferences,
reexaminations,  inter  partes  reviews  or  derivation  proceedings  before  the  United  States  or  other  jurisdictions.  These  proceedings  can  be
expensive and time‑consuming and many of our or our licensors’ or collaborators’ adversaries in these proceedings may have the ability to
dedicate substantially greater resources to prosecuting these legal actions than we or our licensors or collaborators can.

An unfavorable outcome could require us or our licensors or collaborators to cease using the related technology or developing or
commercializing our product candidates, or to attempt to license rights to it from the prevailing party. Our business could be harmed if the
prevailing party does not offer us or our licensors or collaborators a license on commercially reasonable terms or at all. Even if we or our
licensors  or  collaborators  obtain  a  license,  it  may  be  non‑exclusive,  thereby  giving  our  competitors  access  to  the  same  technologies
licensed to us or our licensors or collaborators. In addition, we could be found liable for monetary damages, including treble damages and
attorneys’ fees, if we are found to have willfully infringed a patent. A finding of infringement could prevent us from commercializing our
product candidates or force us to cease some of our business operations, which could materially harm our business.

We  may  become  involved  in  lawsuits  to  protect  or  enforce  our  intellectual  property,  which  could  be  expensive,  time‑consuming  and
unsuccessful and have a material adverse effect on the success of our business.

Third  parties  may  infringe  on  our  or  our  licensors’  or  collaborators’  patents  or  misappropriate  or  otherwise  violate  our  or  our
licensors’ or collaborators’ intellectual property rights. In the future, we or our licensors or collaborators may initiate legal proceedings to
enforce or defend our or our licensors’ or collaborators’ intellectual property rights, to protect our or our licensors’ or collaborators’ trade
secrets  or  to  determine  the  validity  or  scope  of  intellectual  property  rights  we  own  or  control.  Also,  third  parties  may  initiate  legal
proceedings against us or our licensors or collaborators to challenge the validity or scope of intellectual property rights we own or control.
The proceedings can be expensive and time‑consuming and many of our or our licensors’ or collaborators’ adversaries in these proceedings
may have the ability to dedicate substantially greater resources to prosecuting these legal actions than we or our licensors or collaborators
can. Accordingly, despite our or our licensors’ or collaborators’ efforts, we or our licensors or collaborators might not prevent third parties
from infringing upon or misappropriating intellectual property rights we own or control, particularly in countries where the laws might not
protect  those  rights  as  fully  as  in  the  United  States.  Litigation  could  result  in  substantial  costs  and  diversion  of  management  resources,
which could harm our business and financial results. In addition, in an infringement proceeding, a court may decide that a patent owned by
or licensed to us is invalid or unenforceable, or may refuse to stop the other party from using the technology at issue on the grounds

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that our or our licensors’ or collaborators’ patents do not cover the technology in question. An adverse result in any litigation proceeding
could  put  one  or  more  of  our  or  our  licensors’  or  collaborators’  patents  at  risk  of  being  invalidated,  held  unenforceable  or  interpreted
narrowly.

Third  party  preissuance  submission  of  prior  art  to  the  USPTO,  or  opposition,  derivation,  reexamination,  inter  partes  review  or
interference proceedings, or other preissuance or post‑grant proceedings in the United States or other jurisdictions provoked by third parties
or  brought  by  us  or  our  licensors  or  collaborators  may  be  necessary  to  determine  the  priority  of  inventions  with  respect  to  our  or  our
licensors’  or  collaborators’  patents  or  patent  applications. An  unfavorable  outcome  could  require  us  or  our  licensors  or  collaborators  to
cease  using  the  related  technology  and  commercializing  our  product  candidates,  or  to  attempt  to  license  rights  to  it  from  the  prevailing
party. Our business could be harmed if the prevailing party does not offer us or our licensors or collaborators a license on commercially
reasonable  terms  or  at  all.  Even  if  we  or  our  licensors  or  collaborators  obtain  a  license,  it  may  be  non‑exclusive,  thereby  giving  our
competitors  access  to  the  same  technologies  licensed  to  us  or  our  licensors  or  collaborators.  In  addition,  if  the  breadth  or  strength  of
protection  provided  by  our  or  our  licensors’  or  collaborators’  patents  and  patent  applications  is  threatened,  it  could  dissuade  companies
from collaborating with us to license, develop or commercialize current or future product candidates. Even if we successfully defend such
litigation or proceeding, we may incur substantial costs and it may distract our management and other employees. We could be found liable
for monetary damages, including treble damages and attorneys’ fees if we are found to have willfully infringed a patent.

Furthermore, because of the substantial amount of discovery required in connection with intellectual property litigation, there is a
risk that some of our confidential information could be compromised by disclosure during this type of litigation. There could also be public
announcements of the results of hearings, motions or other interim proceedings or developments. If securities analysts or investors perceive
these results to be negative, it could have a material adverse effect on the price of our warrants or shares of our common stock.

We  may  be  subject  to  claims  by  third  parties  asserting  that  our  employees  or  we  have  misappropriated  their  intellectual  property,  or
claiming ownership of what we regard as our own intellectual property.

Many of our employees, including our senior management, were previously employed at universities or at other biotechnology or
pharmaceutical  companies,  including  our  competitors  or  potential  competitors.  Some  of  these  employees  executed  proprietary  rights,
non‑disclosure  and  non‑competition  agreements  in  connection  with  such  previous  employment.  We  may  be  subject  to  claims  that  we  or
these  employees  have  used  or  disclosed  confidential  information  or  intellectual  property,  including  trade  secrets  or  other  proprietary
information, of any such employee’s former employer. In addition, we may be subject to claims that former employees, collaborators, or
other third parties have an ownership interest in our patents or other intellectual property. While it is our policy to require our employees
and contractors who may be involved in the development of intellectual property to execute agreements assigning such intellectual property
to us, we may be unsuccessful in executing such an agreement to each party who in fact develops intellectual property that we regard as our
own.  We  could  be  subject  to  ownership  disputes  arising,  for  example,  from  conflicting  obligations  of  consultants  or  others  who  are
involved in developing our product candidates. Litigation may be necessary to defend against these claims.

If we fail in prosecuting or defending any such claims, in addition to paying monetary damages, we may lose valuable intellectual
property  rights  or  personnel  or  sustain  damages.  Such  intellectual  property  rights  could  be  awarded  to  a  third  party,  and  we  could  be
required to obtain a license from such third party to commercialize our technology or products. Such a license might not be available on
commercially  reasonable  terms  or  at  all.  Even  if  we  successfully  prosecute  or  defend  against  such  claims,  litigation  could  result  in
substantial costs and distract management.

Our inability to protect our confidential information and trade secrets would harm our business and competitive position.

In  addition  to  seeking  patents  for  some  of  our  technology  and  products,  we  also  rely  on  trade  secrets,  including  unpatented
know‑how,  technology  and  other  proprietary  information,  to  maintain  our  competitive  position.  Though  we  seek  to  protect  these  trade
secrets,  in  part,  by  entering  into  non‑disclosure  and  confidentiality  agreements  with  parties  who  have  access  to  them,  such  as  our
employees, corporate collaborators, outside scientific collaborators, contract manufacturers, consultants, advisors and other third parties, as
well as by entering into confidentiality and invention or patent assignment agreements with our employees and consultants, any of these
parties may breach the agreements and disclose our proprietary information, including our trade secrets, and we might not be able to obtain
adequate  remedies  for  such  breaches.  Enforcing  a  claim  that  a  party  illegally  disclosed  or  misappropriated  a  trade  secret  is  difficult,
expensive and time‑consuming, and the outcome is unpredictable. In addition, some courts both within and outside the United States may
be less willing or unwilling to protect trade secrets. If a competitor lawfully obtained or independently developed any of our trade secrets,
we would have no right to prevent such competitor from using that technology or information to compete with us, which could harm our
competitive position.

Changes in patent law could diminish the value of patents in general, thereby impairing our ability to protect our product candidates.

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As is the case with other biotechnology and pharmaceutical companies, our success is heavily dependent on intellectual property,
particularly  patents.  Obtaining  and  enforcing  patents  in  the  biopharmaceutical  industry  involve  technological  and  legal  complexity,  and
obtaining and enforcing biopharmaceutical patents is costly, time‑consuming, and inherently uncertain. The Supreme Court has ruled on
several  patent  cases  in  recent  years,  either  narrowing  the  scope  of  patent  protection  available  in  certain  circumstances  or  weakening  the
rights  of  patent  owners  in  certain  situations.  In  addition  to  increasing  uncertainty  with  regard  to  our  and  our  licensors’  or  collaborators’
ability to obtain patents in the future, this combination of events has created uncertainty with respect to the value of patents, once obtained.
Depending  on  decisions  by  Congress,  the  federal  courts,  and  the  USPTO  the  laws  and  regulations  governing  patents  could  change  in
unpredictable ways that would weaken our and our licensors’ or collaborators’ ability to obtain new patents or to enforce existing patents
and patents we and our licensors or collaborators may obtain in the future. Recent patent reform legislation could increase the uncertainties
and costs surrounding the prosecution of our and our licensors’ or collaborators’ patent applications and the enforcement or defense of our
or our licensors’ or collaborators’ issued patents. On September 16, 2011, the Leahy‑Smith America Invents Act, or the Leahy‑Smith Act,
was signed into law. The Leahy‑Smith Act includes a number of significant changes to United States patent law. These include provisions
that affect the way patent applications are prosecuted and may also affect patent litigation. The USPTO recently developed new regulations
and procedures to govern administration of the Leahy‑Smith Act, and many of the substantive changes to patent law associated with the
Leahy‑Smith Act, and in particular, the first to file provisions, only became effective on March 16, 2013. Accordingly, it is not clear what,
if  any,  impact  the  Leahy‑Smith Act  will  have  on  the  operation  of  our  business.  However,  the  Leahy‑Smith Act  and  its  implementation
could increase the uncertainties and costs surrounding the prosecution of our or our licensors’ or collaborators’ patent applications and the
enforcement or defense of our or our licensors’ or collaborators’ issued patents, all of which could have a material adverse effect on our
business and financial condition.

We might not be able to protect our intellectual property rights throughout the world.

Filing,  prosecuting,  enforcing  and  defending  patents  on  product  candidates  in  all  countries  throughout  the  world  would  be
prohibitively expensive, and our or our licensors’ or collaborators’ intellectual property rights in some countries outside the United States
can be less extensive than those in the United States. In addition, the laws of some foreign countries do not protect intellectual property
rights to the same extent as federal and state laws in the United States. Consequently, we and our licensors or collaborators might not be
able to prevent third parties from practicing our and our licensors’ or collaborators’ inventions in all countries outside the United States, or
from  selling  or  importing  products  made  using  our  and  our  licensors’  or  collaborators’  inventions  in  and  into  the  United  States  or  other
jurisdictions. Competitors may use our and our licensors’ or collaborators’ technologies in jurisdictions where we have not obtained patent
protection to develop their own products and further, may export otherwise infringing products to territories where we and our licensors or
collaborators have patent protection, but enforcement is not as strong as that in the United States. These products may compete with our
product  candidates  and  our  and  our  licensors’  or  collaborators’  patents  or  other  intellectual  property  rights  might  not  be  effective  or
sufficient to prevent them from competing.

Many  companies  have  encountered  significant  problems  in  protecting  and  defending  intellectual  property  rights  in  foreign
jurisdictions. The legal systems of certain countries, particularly certain developing countries, do not favor the enforcement of patents and
other  intellectual  property  protection,  particularly  those  relating  to  biopharmaceuticals,  which  could  make  it  difficult  for  us  and  our
licensors or collaborators to stop the infringement of our and our licensors’ or collaborators’ patents or marketing of competing products in
violation  of  our  and  our  licensors’  or  collaborators’  proprietary  rights  generally.  Proceedings  to  enforce  our  and  our  licensors’  or
collaborators’ patent rights in foreign jurisdictions could result in substantial costs and divert our and our licensors’ or collaborators’ efforts
and attention from other aspects of our business, could put our and our licensors’ or collaborators’ patents at risk of being invalidated or
interpreted narrowly and our and our licensors’ or collaborators’ patent applications at risk of not issuing and could provoke third parties to
assert claims against us or our licensors or collaborators. We or our licensors or collaborators might not prevail in any lawsuits that we or
our licensors or collaborators initiate and the damages or other remedies awarded, if any, might not be commercially meaningful.

The  requirements  for  patentability  may  differ  in  certain  countries,  particularly  developing  countries.  For  example,  unlike  other
countries, China has a heightened requirement for patentability, and specifically requires a detailed description of medical uses of a claimed
drug. In India, unlike the United States, there is no link between regulatory approval of a drug and its patent status. Furthermore, generic or
biosimilar  drug  manufacturers  or  other  competitors  may  challenge  the  scope,  validity  or  enforceability  of  our  or  our  licensors’  or
collaborators’  patents,  requiring  us  or  our  licensors  or  collaborators  to  engage  in  complex,  lengthy  and  costly  litigation  or  other
proceedings. Generic or biosimilar drug manufacturers may develop, seek approval for, and launch biosimilar versions of our products. In
addition to India, certain countries in Europe and developing countries, including China, have compulsory licensing laws under which a
patent owner may be compelled to grant licenses to third parties. In those countries, we and our licensors or collaborators may have limited
remedies if patents are infringed or if we or our licensors or collaborators are compelled to grant a license to a third party, which could
materially diminish the value of those patents. This could limit our potential revenue opportunities. Accordingly, our and our licensors’ or
collaborators’  efforts  to  enforce  intellectual  property  rights  around  the  world  may  be  inadequate  to  obtain  a  significant  commercial
advantage from the intellectual property that we own or license.

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Risks Related to Our Financial Position and Capital Needs

We  might  require  additional  capital  to  continue  to  fund  our  operations  and  to  finance  the  further  advancement  of  our  product
candidates, which might not be available to us on acceptable terms, or at all. Failure to obtain any necessary capital will force us to
delay, limit or terminate our product development efforts or cease our operations.

At December 31, 2018, we had $10.6 million in cash and cash equivalents and $26.2 million in current liabilities. Accordingly, we
might  not  currently  have  sufficient  funds  to  finance  our  continuing  operations  beyond  the  short  term  or  to  further  advance  any  of  our
product candidates.

As a research and development company until our November 2017 acquisition of TRx, our operations have consumed substantial
amounts of cash since inception. Research and development remain an important part of our business, and our new commercial operations
might  not  be  profitable  or  generate  enough  funds  to  support  our  operations.  Identifying  potential  product  candidates  and  conducting
preclinical testing and clinical trials is a time‑consuming, expensive and uncertain process that takes years to complete, and we expect our
research  and  development  expenses  to  increase  substantially  in  connection  with  our  ongoing  activities,  particularly  as  we  advance  our
product candidates into clinical trials or obtain and advance additional product candidates. Circumstances may cause us to consume capital
more rapidly than we currently anticipate. We may need to raise additional funds or otherwise obtain funding through collaborations if we
choose to initiate additional clinical trials for product candidates.

Additionally,  as  part  of  the Avadel  acquisition,  we  assumed  financial  obligations  to  Deerfield  CSF,  LLC,  which  include  a  $15
million loan due in January 2021. Depending on the Company’s cash position in January 2021, we may need to raise additional capital to
repay the loan obligation.

Additional fundraising efforts may divert our management from our day‑to‑day activities, which may adversely affect our ability
to develop and commercialize our product candidates. In addition, we cannot guarantee that future financing will be available in sufficient
amounts or on terms acceptable to us, if at all. If we do not raise additional capital when required or on acceptable terms, we may need to:

•

•

•

significantly delay, scale back or discontinue the development or commercialization of one or more of our product candidates
or cease operations altogether;

seek strategic alliances for research and development programs at an earlier stage than we would otherwise desire or on terms
less favorable than might otherwise be available; or

relinquish,  or  license  on  unfavorable  terms,  our  rights  to  technologies  or  any  future  product  candidates  that  we  otherwise
would seek to develop or commercialize ourselves.

Our future funding requirements, both short and long term, will depend on many factors, including:

•

•

•

•

•

the  integration  and  profitability  of  our  recently  acquired  commercial  businesses  (TRx  in  November  2017  and  Avadel’s
pediatric business in February 2018);

the  initiation,  progress,  timing,  costs  and  results  of  preclinical  and  clinical  studies  for  our  product  candidates  and  future
product candidates we may develop;

the outcome, timing and cost of seeking and obtaining regulatory approvals from the FDA and comparable foreign regulatory
authorities,  including  the  potential  for  such  authorities  to  require  that  we  perform  more  studies  than  we  currently  expect  to
perform;

the cost to establish, maintain, expand and defend the scope of our intellectual property portfolio, including the amount and
timing of any payments we may be required to make, or that we may receive, in connection with licensing, preparing, filing,
prosecuting, defending and enforcing any patents or other intellectual property rights;

effect  of 

the 
developments;

competing 

technological 

and  market

• market 

acceptance  of 

any 

approved  product

candidates;

•

the  costs  of  acquiring,  licensing  or  investing  in  additional  businesses,  products,  product  candidates  and
technologies;

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•

•

the cost and timing of selecting, auditing and potentially validating a manufacturing site for commercial‑scale manufacturing;
and

the  cost  of  expanding  our  sales,  marketing  and  distribution  capabilities  to  accommodate  any  of  our  product  candidates  for
which we receive marketing approval and that we determine to commercialize ourselves or in collaboration with our partners.

Failure to comply with the financial covenants under the debt agreement assumed during the acquisition of Avadel’s pediatric products
could allow Deerfield CSF to call for immediate repayment of the outstanding borrowings.

As part of the Avadel acquisition, we assumed financial obligations to Deerfield CSF, LLC, which include a $15 million loan due
in  January  2021  (“Deerfield  Obligation”),  fixed  quarterly  payments  of  $262,500  through  January  2020  and  contingent  consideration  of
$12,500,000  paid  quarterly  as  15%  of  acquired  Avadel  pediatric  product  sales.  The  Deerfield  Obligation  is  governed  an  agreement
containing certain covenants. There can be no assurance that we will be in compliance with all of these covenants in the future and that
Deerfield  will  not  immediately  call  for  repayment  of  the  outstanding  borrowings  in  the  event  we  are  not  in  compliance  with  any  of  the
covenants.

We have incurred significant net losses in most periods since our inception and we might continue to incur net losses in the future.

Until our acquisition of TRx in November 2017, we were a clinical‑stage biotechnology company with a limited operating history.
Investment in biopharmaceutical product development is highly speculative because it entails substantial upfront capital expenditures and
significant risk that any potential product candidate will fail to demonstrate an adequate effect or acceptable safety profile, gain marketing
approval and become commercially viable. Historically, we financed our operations primarily through private placements of our common
and convertible preferred stock and convertible debt. We incurred net loss of $40.1 million for the year ended December 31, 2018. As of
December  31,  2018,  we  had  an  accumulated  deficit  of $98.2 million. Substantially  all  of  our  operating  losses  have  resulted  from  costs
incurred  in  connection  with  our  research  and  development  program  and  from  general  and  administrative  costs  associated  with  our
operations.

Even though we now have approved products and commercial operations, we might continue to incur losses in the future. Even if
we  do  generate  product  sales,  we  might  never  achieve  or  sustain  profitability  on  an  annual  basis.  We  may  also  encounter  unforeseen
expenses, difficulties, complications, delays and other unknown factors that may adversely affect our business. Our future profitability will
depend, in part, on the rate of future growth of our expenses and our ability to generate significant revenues. Our prior losses and expected
future losses have had and will continue to have an adverse effect on our stockholders’ equity and working capital.

Our ability to use our net operating loss carryforwards and certain other tax attributes may be limited.

The Company had a significant amount of gross net operating losses ("NOLs") for federal and state purposes that will begin to

expire in 2031.

Unused  losses  for  the  current  tax  year  and  prior  tax  years  will  carry  forward  to  offset  future  taxable  income,  if  any,  until  such
unused losses expire. Unused losses generated after December 31, 2017, under new tax legislation signed into law on December 22, 2017,
known  as  the  Tax  Cuts  and  Jobs Act  of  2017,  or  the  Tax Act,  will  not  expire  and  may  be  carried  forward  indefinitely  but  will  be  only
deductible to the extent of 80% of current year taxable income in any given year. In addition, both our current and our future unused losses
may be subject to limitation under Sections 382 and 383 of the Internal Revenue Code of 1986, as amended (the "IRC"). Sections 382 and
383 of the IRC subject the future utilization of NOLs and certain other tax attributes, such as research and experimental tax credits, to an
annual limitation in the event of certain ownership changes, as defined (in general, an “ownership change” is defined as a greater than 50%
change (by value) in equity ownership over a three-year period).

U.S. federal income tax reform could adversely affect our business and financial condition.

The Tax Act significantly revised the IRC. The revised federal income tax law, among other things, contains significant changes
to corporate taxation, including reduction of the corporate tax rate from a top marginal rate of 35% to a flat rate of 21%, limitation of the
tax deduction for interest expense to 30% of adjusted earnings (except for certain small businesses), limitation of the deduction for NOLs to
80% of current year taxable income and elimination of NOL carrybacks, one time taxation of offshore earnings at reduced rates regardless
of whether they are repatriated, elimination of U.S. tax on foreign earnings (subject to certain important exceptions), immediate deductions
for certain new investments instead of deductions for depreciation expense over time, and modifying or repealing many business
deductions and credits (including reduction of tax credits under the Orphan Drug Act). Notwithstanding the reduction in the corporate
income tax rate, the overall impact of the new federal tax law is uncertain and our

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business and financial condition could be adversely affected. In addition, it is uncertain if and to what extent various states will conform to
the newly enacted federal tax law.

In connection with the reporting of our financial condition and results of operations, we are required to make estimates and judgments
which involve uncertainties, and any significant differences between our estimates and actual results could have an adverse impact on
our financial position, results of operations and cash flows.

Our discussion and analysis of our financial condition and results of operations are based on our financial statements, which have
been  prepared  in  accordance  with  generally  accepted  accounting  principles  in  the  United  States,  or  GAAP.  The  preparation  of  these
financial  statements  requires  us  to  make  estimates  and  judgments  that  affect  the  reported  amounts  of  assets,  liabilities,  expenses  and
revenues  and  related  disclosure  of  contingent  assets  and  liabilities.  For  example,  we  estimate  returns,  wholesaler  fees,  prompt  payment
discounts, chargebacks and government rebates. We also estimate clinical trial costs incurred using subject data and information from our
CROs. If we underestimate or overestimate these expenses, adjustments to expenses may be necessary in future periods. Any significant
differences  between  our  actual  results  and  our  estimates  and  assumptions  could  negatively  impact  our  financial  position,  results  of
operations and cash flows.

Our limited commercial operating history may make it difficult for you to evaluate the success of our business to date and to assess our
future viability.

We commenced commercial operations upon our acquisition of TRx in November 2017. Prior to that, our operations consisted of
organizing and staffing our company, business planning, raising capital and developing our product candidates and platform. We have not
yet demonstrated our ability to successfully develop any product candidate, obtain marketing approvals, manufacture a commercial scale
product  or  arrange  for  a  third  party  to  do  so  on  our  behalf,  or  conduct  sales  and  marketing  activities  necessary  for  successful  product
commercialization. Consequently, any predictions you make about our future success or viability might not be as accurate as they could be
if we had a longer commercial operating history.

In  addition,  as  an  early-stage  business,  we  may  encounter  unforeseen  expenses,  difficulties,  complications,  delays  and  other
known and unknown factors. Our transition from a company with a research and development focus to a company capable of supporting
commercial activities might not be successful.

Our operating results fluctuate from quarter to quarter and year-to-year, making future operating results difficult to predict.

Our quarterly and annual operating results historically have fluctuated and are likely to continue to fluctuate depending on several
factors, many of which are beyond our control. Accordingly, our quarterly and annual results are difficult to predict prior to the end of the
quarter or year, and we may be unable to confirm or adjust expectations with respect to our operating results for a particular period until
that period has closed. Any failure to meet our quarterly or annual revenue or earnings targets could adversely impact the market price of
our  securities.  Therefore,  you  should  not  rely  upon  the  results  of  any  quarterly  or  annual  periods  as  indications  of  future  operating
performance.

We engage in in‑licensing, acquisitions or other strategic transactions that could impact our liquidity, increase our expenses and divert
a significant amount of our management’s time.

Since  inception,  we  have  acquired  or  in‑licensed  each  of  our  product  candidates,  including  pediatric  products from Avadel  and
TRx, and most recently product candidates we acquired Ichorion. As a part of the Ichorion acquisition, we issued approximately  5,798,735
shares of our common stock, and payment of certain development milestones of up to an additional $15,000,000, payable either in shares of
our common stock or in cash. As part of the Avadel acquisition, we assumed financial obligations to Deerfield CSF, LLC, which include a
$15 million loan due in January 2021 and royalty payments of 15% of net sales through February 2026. As a part of the TRx acquisition,
we  issued  7,534,884  shares  of  our  common  stock  to  the  sellers  and  the  potential  to  pay  Lachlan  Pharmaceuticals  up  to  $4.0  million  in
milestone  payments. From  time  to  time  we  may  consider  additional  in‑licensing  of  products  and  other  strategic  transactions,  such  as
acquisitions of companies, asset purchases and out‑licensing of product candidates or technologies. Additional potential transactions that
we  may  consider  include  a  variety  of  different  business  arrangements,  including  strategic  partnerships,  collaborations,  joint  ventures,
business  combinations  and  investments. Any  such  transaction  may  require  us  to  incur  non‑recurring  or  other  charges,  may  increase  our
near  and  long‑term  expenditures  and  may  pose  significant  integration  challenges  or  disrupt  our  management  or  business,  which  could
adversely affect our operations and financial results. For example, these transactions may entail numerous operational and financial risks,
including:

•

exposure 
liabilities;

to 

unknown

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•

•

•

•

•

•

•

•

disruption of our business and diversion of our management’s time and attention in order to develop acquired products, product
candidates or technologies;

incurrence  of  substantial  debt  or  dilutive  issuances  of  equity  securities  to  pay  for  acquisitions  or  to  fund  the
operations;

higher  than  expected  acquisition  and  integration
costs;

write‑downs  of  assets  or  goodwill  or 
charges;

impairment

increased 
expenses;

amortization

difficulty  and  cost  in  combining  the  operations  and  personnel  of  any  acquired  businesses  with  our  operations  and
personnel;

impairment of relationships with key suppliers or other counterparties of any acquired businesses due to changes in management
and ownership; and

inability 
businesses.

to  retain  key  employees  of  any  acquired

Risks Related to our Stock

If we are not able to comply with the applicable continued listing requirements or standards of The NASDAQ Capital Market, NASDAQ
could delist our common stock.

Our common stock is currently listed on the NASDAQ Capital Market ("NASDAQ"). In order to maintain that listing, we must
satisfy  minimum  financial  and  other  continued  listing  requirements  and  standards,  including  those  regarding  director  independence  and
independent  committee  requirements,  minimum  stockholders’  equity,  minimum  share  price,  and  certain  corporate  governance
requirements. There can be no assurances that we will be able to comply with the applicable listing standards.

In the event that our common stock is delisted  from  NASDAQ  and  is  not  eligible  for  quotation  or  listing  on  another  market  or
exchange,  trading  of  our  common  stock  could  be  conducted  only  in  the  over-the-counter  market  or  on  an  electronic  bulletin  board
established  for  unlisted  securities  such  as  the  Pink  Sheets  or  the  OTC  Bulletin  Board.  In  such  event,  it  could  become  more  difficult  to
dispose  of,  or  obtain  accurate  price  quotations  for,  our  common  stock,  and  there  would  likely  also  be  a  reduction  in  our  coverage  by
securities analysts and the news media, which could cause the price of our common stock to decline further. Also, it may be difficult for us
to raise additional capital if we are not listed on a major exchange.

Such a de-listing would also likely have a negative effect on the price of our common stock and would impair your ability to sell or

purchase our common stock when you wish to do so. In the event of a de-listing, we may take actions to restore our compliance with
NASDAQ’s listing requirements, but we can provide no assurance that any such action taken by us would allow our common stock to
become listed again, stabilize the market price or improve the liquidity of our common stock, prevent our common stock from dropping
below the NASDAQ minimum bid price requirement or prevent future non-compliance with NASDAQ’s listing requirements.

An active trading market for our securities might not be sustained.

Although  our  common  shares  are  listed  on  the  NASDAQ  we  cannot  assure  you  that  an  active  trading  market  for  our  common
shares will continue to develop or be sustained, particularly because one investor, Armistice Capital, now holds a significant amount of our
outstanding stock. If an active market for our common shares is not sustained it may impair your ability to sell your warrants or shares of
our common stock at the time you wish to sell them or at a price that you consider reasonable, you may not be able to sell your shares
quickly  or  at  the  market  price. An  inactive  market  may  also  impair  our  ability  to  raise  capital  to  continue  to  fund  operations  by  selling
common shares and may impair our ability enter into strategic collaborations or acquire companies or products by using our by using our
common shares as consideration.

The market price of our stock is volatile, and you could lose all or part of your investment.

The  market  price  of  our  shares  of  our  common  stock  has  been  highly  volatile  and  subject  to  wide  fluctuations  in  response  to
various factors, some of which we cannot control. From our initial public offering in October 2015 through December 31, 2018, the per
share trading price of our common stock has been as high as $6.65 and as low as $0.34. As a result of this volatility, you might not be able
to sell your shares of our common stock at a favorable price. In addition to the factors discussed in this “Risk Factors” section and

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elsewhere in this Annual Report on Form 10-K, these factors that could negatively affect or result in fluctuations in the market price of
shares of our common stock include:

•

•

•

•

•

•

•

•

•

•

•

•

•

•

•

•

•

•

•

if

or

of 

products 

competitive 

to  commercialize  our  product  candidates, 

our  ability  to  generate  significant  product  revenues,  cash  flows  and  a
profit;
the  development  status  of  our  product  candidates,  and  when  any  of  our  product  candidates  receive  marketing
approval;
our decision to initiate a clinical trial, not to initiate a clinical trial or to terminate an existing clinical
trial;
our  failure 
approved;
success 
the 
technologies;
regulatory  actions  with  respect  to  our  products  or  our  competitors’
products;
actual  or  anticipated  changes  in  our  growth  rate  relative  to  our
competitors;
announcements by us or our competitors of significant acquisitions, strategic collaborations, joint ventures, collaborations or
capital commitments;
results  of  preclinical  studies  and  clinical  trials  of  our  product  candidates  or  those  of  our
competitors;
regulatory  or  legal  developments  in  the  United  States  and  other
countries;
developments  or  disputes  concerning  patent  applications,  issued  patents  or  other  proprietary
rights;
the 
personnel;
the  level  of  expenses  related  to  any  of  our  product  candidates  or  clinical  development
programs;
the  results  of  our  efforts  to  discover,  develop,  in‑license  or  acquire  additional  product  candidates  or
products;
actual  or  anticipated  changes  in  estimates  as  to  financial  results,  development  timelines  or  recommendations  by  securities
analysts;
the  performance  of  third  parties  on  whom  we  rely  to  manufacture  our  products  and  product  candidates,  supply API  and
conduct our clinical trials, including their ability to comply with regulatory requirements;
variations in our financial results or those of companies that are perceived to be similar to
us;
variations  in  the  level  of  expenses  related  to  our  product  candidates  or  preclinical  and  clinical  development  programs,
including relating to the timing of invoices from, and other billing practices of, our CROs and clinical trial sites;
fluctuations in the valuation of companies perceived by investors to be comparable to
us;

recruitment  or  departure  of  key

• warrant  or  share  price  and  volume  fluctuations  attributable  to  inconsistent  trading  volume  levels  of  our  warrants  or

•

•

•

•

shares;
announcement  or  expectation  of  additional  financing
efforts;
sales  of  our  warrants  or  shares  of  our  common  stock  by  us,  our  insiders  or  our  other  security
holders;
changes 
systems;
changes  in  operating  performance  and  stock  market  valuations  of  other  pharmaceutical
companies;

the  structure  of  healthcare  payment

in 

• market  conditions  in  the  pharmaceutical  and  biotechnology

•

•

•

•

•

•

•

•

sectors;
our execution of collaborative, co‑promotion, licensing or other arrangements, and the timing of payments we may make or
receive under these arrangements;
additional  state  and  federal  healthcare  reform  measures  that  could  put  downward  pricing  pressure  on  our
products;
the  public’s  response  to  press  releases  or  other  public  announcements  by  us  or  third  parties,  including  our  filings  with  the
SEC and announcements relating to litigation or other disputes, strategic transactions or intellectual property impacting us or
our business;
announcement 
litigation;
fluctuations in quarterly operating results, as well as differences between our actual financial and operating results and those
expected by investors;
the  financial  projections  we  may  provide  to  the  public,  any  changes  in  these  projections  or  our  failure  to  meet  these
projections;
changes in financial estimates by any securities analysts who follow our warrants or shares of common stock, our failure to
meet these estimates or failure of those analysts to initiate or maintain coverage of our warrants or shares of common stock;
ratings  downgrades  by  any  securities  analysts  who  follow  our  warrants  or  shares  of  common
stock;

related 

to

•

•

•

•

•

the  development  and  sustainability  of  an  active  trading  market  for  our  shares  of  common
stock;
future  sales  of  our  shares  of  common  stock  by  our  officers,  directors  and  significant
stockholders;
other  events  or  factors,  including  those  resulting  from  war,  incidents  of  terrorism,  natural  disasters  or  responses  to  these
events;
changes  in  accounting  principles;
and
general 
conditions.

and  market

economic, 

industry 

In addition, the stock market in general, and the market for biotechnology companies in particular, have experienced extreme price
and volume fluctuations that have often been unrelated or disproportionate to the operating performance of these companies. Broad market
and industry factors may negatively affect the market price of shares of common stock, regardless of our actual operating performance. The
realization of any of the above risks or any of a broad range of other risks, including those described in this “Risk Factors” section, could
have a material adverse impact on the market price of our shares of common stock. When the market price of a

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stock is volatile, security holders often institute class action litigation against the company that issued the stock. If we become involved in
this type of litigation, regardless of the outcome, we could incur substantial legal costs and our management's attention could be diverted
from the operation of our business, which could have a material adverse effect on our business, financial condition, results of operations
and cash flows.

Future  sales  and  issuances  of  shares  of  our  common  stock  or  rights  to  purchase  common  stock,  including  pursuant  to  our  equity
incentive plans, could result in additional dilution of the percentage ownership of our stockholders and could cause our stock price to
fall.

We expect that additional capital may be needed in the future to continue our planned operations, including conducting clinical
trials, commercialization efforts, expanded research and development activities and costs associated with operating a public company. To
raise  capital,  we  may  sell  common  stock,  convertible  securities  or  other  equity  securities  in  one  or  more  transactions  at  prices  and  in  a
manner  we  determine  from  time  to  time.  If  we  sell  common  stock,  convertible  securities  or  other  equity  securities  in  more  than  one
transaction,  investors  may  be  materially  diluted  by  subsequent  sales.  Such  sales  may  also  result  in  material  dilution  to  our  existing
stockholders, and new investors could gain rights, preferences and privileges senior to our existing stockholders.

We are authorized to grant equity awards, including stock grants and stock options, to our employees, directors and consultants. As
of December 31, 2018, there were 602,657 shares available for future issuance under the 2016 Equity Incentive Plan ("the 2016 Amended
Plan"). During the term of the 2016 Amended Plan, the share reserve will automatically increase on the first trading day in January of each
calendar year, by an amount equal to 4% of the total number of outstanding shares of common stock of the Company on the last trading
day in December of the prior calendar year. On January 1, 2019, on the terms of the 2016 Amended Plan an additional 1,632,167 shares
were made available for issuance for a total of 2,234,824 shares available for issuance. In  addition, as of December 31, 2018, there were
783,983 shares available for future issuance under the 2016 Employee Stock Purchase Plan (the "ESPP"). On January 1 of each calendar
year, the aggregate number of shares that may be issued under the ESPP shall automatically increase by a number equal to the lesser of (i)
1%  of  the  total  number  of  shares  of  the  Company’s  capital  stock  outstanding  on  December  31  of  the  preceding  calendar  year,  and  (ii)
500,000  shares  of  the  Company’s  common  stock,  or  (iii)  a  number  of  shares  of  the  Company’s  common  stock  as  determined  by  the
Company’s board of directors or compensation committee.  Future issuances, as well as the possibility of future issuances, under our 2016
Plan or 2016 ESPP or other equity incentive plans could cause the market price of our common stock to decrease.

Armistice Capital has significant influence over our company, and its interests may be different from or conflict with those of our other
stockholders.

Armistice Capital beneficially own approximately 60% of our outstanding common stock. As a consequence, Armistice Capital
continues to be able to exert a significant degree of influence over our management, affairs, and matters requiring stockholder approval,
including  the  election  of  directors,  a  merger,  consolidation  or  sale  of  all  or  substantially  all  of  our  assets,  and  any  other  significant
transaction. The interests of Armistice Capital might not always coincide with our interests or the interests of our other stockholders. For
instance, this concentration of ownership may have the effect of delaying or preventing a change in control of us otherwise favored by our
other stockholders and could depress our stock price.

Armistice  Capital  makes  investments  in  companies  and  may,  from  time  to  time,  acquire  and  hold  interests  in  businesses  that
compete  directly  or  indirectly  with  us. Armistice  Capital  may  also  pursue,  for  its  own  account,  acquisition  opportunities  that  may  be
complementary to our business, and as a result, those acquisition opportunities might not be available to us. The interests of the Armistice
Capital may supersede ours, causing Armistice Capital or their affiliates to compete against us or to pursue opportunities instead of us, for
which we have no recourse. Such actions on the part of Armistice Capital and inaction on our part could have a material adverse effect on
our business, financial condition, results of operations and cash flows.

Armistice  Capital  controls  a  seat  on  our  board  of  directors.  Since  Armistice  Capital  could  invest  in  entities  that  directly  or
indirectly  compete  with  us,  when  conflicts  arise  between  the  interests  of Armistice  Capital  and  the  interests  of  our  stockholders,  this
director might not be disinterested.

Sales of a significant number of shares of our common stock in the public markets, or the perception that such sales could occur, could
depress the market price of our common stock.

Sales of a substantial number of shares of our common stock in the public markets could depress the market price of our common
stock  and  impair  our  ability  to  raise  capital  through  the  sale  of  additional  equity  securities. As  additional  shares  of  our  common  stock
become available for resale in the public market pursuant to this offering, and otherwise, the supply of our common stock will increase,
which could decrease its price. In addition, some or all of the shares of common stock may be offered from time to time in the open

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market pursuant to Rule 144, and these sales may have a depressive effect on the market for our shares of common stock. Therefore, we
cannot predict the effect that future sales of our common stock would have on the market price of our common stock.

We have never paid cash dividends on our capital stock, and we do not anticipate paying any cash dividends in the foreseeable future.

The continued operation and expansion of our business will require substantial funding. We currently intend to retain all of our
future earnings, if any, to finance the growth and development of our business. Accordingly, we do not anticipate that we will pay any cash
dividends  on  shares  of  our  common  stock  for  the  foreseeable  future.  Consequently,  currently  stockholders  must  rely  on  sales  of  their
common  stock  after  price  appreciation,  which  may  never  occur,  as  the  only  way  to  realize  any  future  gains  on  their  investment. Any
determination to pay dividends in the future will be at the discretion of our board of directors and will depend upon results of operations,
financial condition, contractual restrictions, restrictions imposed by applicable law and other factors our board of directors deems relevant.

We are an “emerging growth company” as defined in the Jumpstart Our Business Startups Act of 2012 ("JOBS Act") and will be able
to avail ourselves of reduced disclosure requirements applicable to emerging growth companies, which could make our securities less
attractive to investors and adversely affect the market price of our securities.

For  so  long  as  we  remain  an  “emerging  growth  company”  as  defined  in  the  JOBS  Act,  we  may  take  advantage  of  certain

exemptions from various requirements applicable to public companies that are not “emerging growth companies” including:

•

•

•

•

the provisions of Section 404(b) of the Sarbanes‑Oxley Act of 2002, or Sarbanes‑Oxley Act, requiring that our independent
registered  public  accounting  firm  provide  an  attestation  report  on  the  effectiveness  of  our  internal  control  over  financial
reporting;

the “say on pay” provisions (requiring a non‑binding shareholder vote to approve compensation of certain executive officers)
and  the  “say  on  golden  parachute”  provisions  (requiring  a  non‑binding  shareholder  vote  to  approve  golden  parachute
arrangements for certain executive officers in connection with mergers and certain other business combinations) of the Dodd-
Frank Act  and  some  of  the  disclosure  requirements  of  the  Dodd-Frank Act  relating  to  compensation  of  our  chief  executive
officer.

the  requirement  to  provide  detailed  compensation  discussion  and  analysis  in  proxy  statements  and  reports  filed  under  the
Securities  Exchange  Act  of  1934,  as  amended,  or  the  Exchange  Act,  and  instead  provide  a  reduced  level  of  disclosure
concerning executive compensation; and

any  rules  that  the  Public  Company Accounting  Oversight  Board  may  adopt  requiring  mandatory  audit  firm  rotation  or  a
supplement to the auditor’s report on the financial statements.

We  may  take  advantage  of  these  exemptions  until  we  are  no  longer  an  “emerging  growth  company.”  We  would  cease  to  be  an
“emerging  growth  company”  upon  the  earliest  of:  (i)  the  first  fiscal  year  following  the  fifth  anniversary  of  our  initial  public  offering;
(ii)  the  first  fiscal  year  after  our  annual  gross  revenues  are  $1.07  billion  or  more;  (iii)  the  date  on  which  we  have,  during  the  previous
three‑year period, issued more than $1.07 billion in non‑convertible debt securities; or (iv) as of the end of any fiscal year in which the
market value of our common stock held by non‑affiliates exceeded $700 million as of the end of the second quarter of that fiscal year.

We  have  determined  to  take  advantage  of  some,  but  not  all,  of  the  reduced  regulatory  and  reporting  requirements  that  will  be
available to us so long as we qualify as an “emerging growth company.” For example, we have irrevocably elected not to take advantage of
the extension of time to comply with new or revised financial accounting standards available under Section 102(b) of the JOBS Act. Our
independent  registered  public  accounting  firm  will  not  be  required  to  provide  an  attestation  report  on  the  effectiveness  of  our  internal
control  over  financial  reporting  so  long  as  we  qualify  as  an  “emerging  growth  company,”  which  may  increase  the  risk  that  material
weaknesses or significant deficiencies in our internal control over financial reporting go undetected. Likewise, so long as we qualify as an
“emerging growth company,” we may elect not to provide you with certain information, including certain financial information and certain
information regarding compensation of our executive officers, that we would otherwise have been required to provide in filings we make
with  the  SEC  which  may  make  it  more  difficult  for  investors  and  securities  analysts  to  evaluate  our  company.  Even  after  we  no  longer
qualify as an emerging growth company, we may still qualify as a “smaller reporting company,” which would allow us to take advantage of
many  of  the  same  exemptions  from  disclosure  requirements,  including  not  being  required  to  comply  with  the  auditor  attestation
requirements  of  Section  404(b)  of  the  Sarbanes‑Oxley Act  and  reduced  disclosure  obligations  regarding  executive  compensation  in  our
periodic reports and proxy statements. We cannot predict if investors will find our securities less attractive because we may rely on these
exemptions. If some investors find our securities less attractive as a result, there may be a less active trading market for our securities, and
the securities prices may be more volatile and may decline.

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We may be subject to future litigation against us, including securities litigation, which could be costly and time-consuming to defend.

The market price of our securities may be volatile, and in the past, companies that have experienced volatility in the market price
of  their  securities  have  been  subject  to  securities  class  action  litigation.  We  may  be  the  target  of  this  type  of  litigation  in  the  future.
Securities litigation against us could result in substantial costs and divert our management’s attention from other business concerns, which
could seriously harm our business. Any adverse determination in litigation could also subject us to significant liabilities.

We may also become subject, from time to time, to legal proceedings and claims that arise in the ordinary course of business such
as claims brought by our clients in connection with commercial disputes, or employment claims made by our current or former associates.
Litigation might result in substantial costs and may divert management’s attention and resources, which might seriously harm our business,
overall financial condition, and operating results. Insurance might not cover such claims, might not provide sufficient payments to cover all
the costs to resolve one or more such claims, and might not continue to be available on terms acceptable to us. A claim brought against us
that is uninsured or underinsured could result in unanticipated costs, thereby reducing our operating results and leading analysts or potential
investors to reduce their expectations of our performance, which could reduce the trading price of our stock.

If  securities  or  industry  analysts  do  not  publish  research  or  publish  inaccurate  or  unfavorable  research  about  our  business,  our
securities prices and trading volume could decline.

The trading market for our securities will depend in part on the research and reports that securities or industry analysts publish
about us or our business. We currently have limited, and might not sustain, research coverage by securities and industry analysts. If we do
not sustain coverage of our company, the trading price for securities would be negatively impacted.  If the securities and industry analysts
are unable to predict accurately the demand and net  of  sales  our  products,  that  could  result  in  our  reported  revenues  and  earnings  being
lower than the so-called “market consensus” of our projected revenues, which could negatively affect our stock price. Additionally, if the
securities and industry analysts are unable to predict accurately the cost of advancing our pipeline, that could result in our reported costs
being different than expectations, which could negatively affect our stock price. If we do obtain securities or industry analyst coverage and
if one or more of the analysts who covers us downgrades our securities or publishes inaccurate or unfavorable research about our business,
our securities prices would likely decline. If one or more of these analysts ceases coverage of us or fails to publish reports on us regularly,
demand for our securities could decrease, which could cause our securities prices and trading volume to decline.

The  requirements  of  being  a  public  company  may  strain  our  resources  and  divert  management’s  attention,  and  our  minimal  public
company operating experience may impact our business and stock price.

As a public company, we incur significant legal, accounting and other expenses, and these expenses may increase even more after
we are no longer an “emerging growth company.” We are subject to the reporting requirements of the Exchange Act, the Sarbanes‑Oxley
Act, the Dodd‑Frank Wall Street Reform and Protection Act, as well as rules adopted, and to be adopted, by the SEC, NASDAQ and other
applicable  securities  rules  and  regulations  imposed  on  public  companies,  including  the  establishment  and  maintenance  of  effective
disclosure and financial controls and corporate governance practices. Our management and other personnel will need to devote a substantial
amount  of  time  to  these  compliance  initiatives.  Moreover,  we  expect  these  rules  and  regulations  to  substantially  increase  our  legal  and
financial compliance costs and to make some activities more time‑consuming and costly. The increased costs will increase our net loss. For
example, we expect these rules and regulations to make it more difficult and more expensive for us to obtain director and officer liability
insurance and we may be required to incur substantial costs to maintain sufficient coverage. The impact of these requirements could also
make it more difficult for us to attract and retain qualified persons to serve on our board of directors, our board committees or as executive
officers.

Because these rules and regulations are often subject to varying interpretations, it is difficult to accurately estimate or predict the
amount or timing of these additional costs. Further, the lack of specificity of many of the rules and regulations may result in an application
in  practice  that  may  evolve  over  time  as  new  guidance  is  provided  by  regulatory  and  governing  bodies.  This  could  result  in  continuing
uncertainty regarding compliance matters and higher costs necessitated by ongoing revisions to disclosure and governance practices.

Our disclosure controls and procedures might not prevent or detect all errors or acts of fraud.

We  are  subject  to  the  periodic  reporting  requirements  of  the  Exchange  Act,  Sarbanes‑Oxley  Act  and  NASDAQ  rules  and
regulations.  The  Sarbanes‑Oxley Act  requires,  among  other  things,  that  we  maintain  effective  disclosure  controls  and  procedures  and
internal control over financial reporting. We designed our disclosure controls and procedures to reasonably assure that information we must
disclose in reports we file or submit under the Exchange Act is accumulated and communicated to management, and recorded, processed,
summarized and reported within the time periods specified in the rules and forms of the SEC. We believe that any disclosure controls and
procedures or internal controls and procedures, no matter how well‑conceived and operated, can provide only reasonable,

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not absolute, assurance that the objectives of the control system are met. We cannot assure, in the future, a material weakness or significant
deficiency will not exist or otherwise be discovered. If that were to happen, it could harm our operating results and cause stockholders to
lose confidence in our reported financial information. Any such loss of confidence would have a negative effect on the trading price of our
securities.

These inherent limitations include the realities that judgments in decision‑making can be faulty, and that breakdowns can occur
because of simple error or mistake. Additionally, controls can be circumvented by the individual acts of some persons, by collusion of two
or  more  people  or  by  an  unauthorized  override  of  the  controls. Accordingly,  because  of  the  inherent  limitations  in  our  control  system,
misstatements due to error or fraud may occur and not be detected.

Our  amended  and  restated  certificate  of  incorporation  provides  that  the  Court  of  Chancery  of  the  State  of  Delaware  is  the  sole  and
exclusive forum for certain litigation that may be initiated by our stockholders, which could limit our stockholders’ ability to obtain a
favorable judicial forum for disputes with us or our directors, officers or employees.

Our amended and restated certificate of incorporation provides that the Court of Chancery of the State of Delaware is the sole and
exclusive forum for (i) any derivative action or proceeding brought on behalf of the company; (ii) any action asserting a claim of breach of
a fiduciary duty owed by any director, officer or other employee of the company to the company or the company’s stockholders; (iii) any
action asserting a claim against the company arising pursuant to any provision of the Delaware General Corporation Law, our amended and
restated certificate of incorporation or our second amended and restated bylaws; or (iv) any action asserting a claim against the company
governed  by  the  internal  affairs  doctrine.   Any  person  or  entity  purchasing  or  otherwise  acquiring  any  interest  in  our  securities  shall  be
deemed  to  have  notice  of  and  to  have  consented  to  the  provisions  of  our  amended  and  restated  certificate  of  incorporation  described
above.  The  choice  of  forum  provision  may  limit  a  stockholder’s  ability  to  bring  a  claim  in  a  judicial  forum  that  it  finds  favorable  for
disputes with us or our directors, officers or other employees, which may discourage such lawsuits against us and our directors, officers and
other employees. Alternatively, if a court were to find the choice of forum provision contained in our amended and restated certificate of
incorporation to be inapplicable or unenforceable in an action, we may incur additional costs associated with resolving such action in other
jurisdictions, which could adversely affect our business, financial condition and results of operations.

Some provisions of our charter documents and Delaware law may have anti‑takeover effects that could discourage an acquisition of us
by others, even if an acquisition would benefit our stockholders and may prevent attempts by our stockholders to replace or remove our
current management.

Provisions in our amended and restated certificate of incorporation and second amended and restated bylaws, as well as provisions
of Delaware law, could make it more difficult for a third party to acquire us or increase the cost of acquiring us, even if doing so would
benefit our stockholders, or remove our current management. These provisions include:

•

•

•

•

•

authorizing the issuance of “blank check” preferred stock, the terms of which we may establish and shares of which we may
issue without stockholder approval;

prohibiting  cumulative  voting  in  the  election  of  directors,  which  would  otherwise  allow  for  less  than  a  majority  of
stockholders to elect director candidates;

prohibiting  stockholder  action  by  written  consent,  thereby  requiring  all  stockholder  actions  to  be  taken  at  a  meeting  of  our
stockholders;

eliminating  the  ability  of  stockholders  to  call  a  special  meeting  of  stockholders;
and

establishing advance notice requirements for nominations for election to the board of directors or for proposing matters that
can be acted upon at stockholder meetings.

These  provisions  may  frustrate  or  prevent  any  attempts  by  our  stockholders  to  replace  or  remove  our  current  management  by
making it more difficult for stockholders to replace members of our board of directors, who are responsible for appointing the members of
our management. Because we are incorporated in Delaware, we are governed by the provisions of Section 203 of the Delaware General
Corporation Law (the "DGCL") which may discourage, delay or prevent someone from acquiring us or merging with us whether or not it is
desired by or beneficial to our stockholders. Under the DGCL, a corporation might not, in general, engage in a business combination with
any  holder  of  15%  or  more  of  its  capital  stock  unless  the  holder  has  held  the  stock  for  three  years  or,  among  other  things,  the  board  of
directors  has  approved  the  transaction. Any  provision  of  our  amended  and  restated  certificate  of  incorporation  or  second  amended  and
restated bylaws or Delaware law that has the effect of delaying or deterring a change of control could limit the opportunity for our

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stockholders to receive a premium for their shares of our common stock, and could also affect the price that some investors are willing to
pay for our securities.

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Item 1B. Unresolved Staff Comments.

None. 

Item 2. Properties.

Our headquarters are located in Rockville, Maryland, where we occupy approximately 5,000 square feet of administrative office
space. The term of the headquarters' lease expires January 31, 2030. We have the ability to expand this office space based on our growth
and employee headcount.

Item 3. Legal Proceedings.

Lachlan Pharmaceuticals

In  November  2017,  the  Company  acquired  TRx  and  its  wholly-owned  subsidiaries,  including  Zylera. The  previous  owners  of  TRx
beneficially own more than 10% of our outstanding common stock. Zylera, which is our wholly owned subsidiary, entered into the First
Amended and Restated Distribution Agreement with  Lachlan, effective December 18, 2015. Pursuant to the Lachlan Agreement, Lachlan
named Zylera as its exclusive distributor of Ulesfia in the United States and agreed to supply Ulesfia to Zylera exclusively for marketing
and sale in the United States.

Zylera is obligated to purchase a minimum of 20,000 units per year, or approximately $1.2 million worth of product, from
Lachlan, subject to certain termination rights. Zylera must pay Lachlan $58.84 per unit and handling fees that are equal to $3.66 per unit of
fully packaged Ulesfia in 2018, and escalate at a rate of 10% annually, as well as reimburse Lachlan for all product liability insurance fees
incurred by Lachlan. The Lachlan Agreement also requires that Zylera make certain cumulative net sales milestone payments and royalty
payments to Lachlan with a $3 million annual minimum payment unless and until there has been a “Market Change” involving a new
successful competitive product. Lachlan is obligated to pay identical amounts to an unrelated third party from which it obtained rights to
Ulesfia, with the payments ultimately flowing to Summers Laboratories, Inc. (“Summers Labs”). Because of the dispute described below,
the Company has not made any payments to Lachlan under the Lachlan Agreement subsequent to the acquisition date.

On December 10, 2016, Zylera informed Lachlan that a Market Change had occurred due to the introduction of Arbor

Pharmaceuticals' lice product, Sklice®.  On June 5, 2017, Lachlan and Zylera entered into joint legal representation along with other
unrelated third parties in negotiation and arbitration of a dispute with Summers Labs regarding the existence of a Market Change and the
concomitant obligations of the parties. The arbitration panel issued an interim ruling on October 23, 2018 that no market change had
occurred up to and including the date of the hearing. The arbitration panel issued a second interim ruling on December 26, 2018. The
second interim award rejected Summers Labs' request to accelerate future minimum royalties, however, it ruled in favor of Summers Labs
that it is owed reimbursement for all reasonable costs and expenses, including legal fees, by Shionogi, as well as interest, as stipulated in the
contract. The arbitration panel issued a final award on March 1, 2019 that dictated the final amount of reimbursable costs and interest as
contemplated in the second interim ruling. The final award has no direct bearing on the Company as the Company was not a named
defendant to the original claim by Summers Labs and a federal court denied Zylera's ability to be a counterclaimant in the matter.
Furthermore, the Company is not subject to the guarantee or interest provisions identified in the second ruling as these elements of the
contractual relationship were not passed down to the Company’s agreement with Lachlan. However, the Company has interpreted this
ruling's impact on the Lachlan agreement to mean that a market change has not occurred, and the minimum purchase obligation and
minimum royalty provisions of the contract are active and due for any prior periods as well as going forward for any future periods.

The Company has recognized a $7.8 million liability for these minimum obligations in accrued liabilities as of December 31,

2018. Under the terms of the TRx Purchase Agreement, the former TRx owners are required to indemnify the Company for 100% of all
pre-acquisition losses related this arbitration, including legal costs, and possible minimum payments in excess of $1 million. Furthermore,
the former TRx owners are required to indemnify the Company for 50% of post-acquisition Ulesfia losses, which would include losses
resulting from having to fund these minimum obligations. The Company has recorded an indemnity receivable of $4.9 million in other
receivables as of December 31, 2018, which the Company believes is fully collectible. The receivable is net of $1.9 million collection made
in the fourth quarter of 2018 from a full cash escrow release with the former TRx owners from the escrow that was established as a part of
the TRx acquisition. The post-acquisition minimum obligations net of amounts recorded within the indemnity receivable of $2.2 million
has been recorded in cost of product sales for the year ended December 31, 2018. If the Company fails to make these minimum obligations
timely then the Lachlan Agreement may be terminated by Lachlan, in which case the Company would no longer be able to sell the Ulesfia
product, but it would also not be subject to future minimum obligations. Lachlan has not requested payment for the minimum obligations.

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Item 4. Mine Safety Disclosures.

Not applicable.

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PART II

 Item 5. Market for Registrant’s Common Equity, Related Stockholder Matters and Issuer Purchases of Equity Securities.

Market Information

Our  common  stock  is  listed  and  publicly  traded  on  the  NASDAQ  Capital  Market  under  the  symbol  “CERC.”  Our  Class  A

warrants (“CERCW”) expired in October 2018 and our Class B warrants ("CERCZ") expired in April 2017.

Holders

As of March 11, 2019, there were approximately 56 holders of record of our common stock. This number does not include

beneficial owners whose shares are held by nominees in street name.

Dividends

We have never declared or paid cash dividends on our capital stock. We intend to retain all of our available funds and future

earnings, if any, to finance the growth and development of our business. We do not intend to pay cash dividends to our stockholders in the
foreseeable future. Any future determination related to our dividend policy will be made at the discretion of our board of directors and will
depend upon, among other factors, our results of operations, financial condition, capital requirements, contractual restrictions, business
prospects and other factors our board of directors may deem relevant.

Recent Sales of Unregistered Securities

Except for sales of unregistered securities that have been previously reported by the Company in either its quarterly reports on

Form 10-Q or current reports on Form 8-K, there were no sales of unregistered securities of the Company during the period covered by this
report.

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Item 6. Selected Financial Data.

As a smaller reporting company, we are not required to provide the information required by this Item.

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Item 7. Management’s Discussion and Analysis of Financial Condition and Results of Operations.

The following discussion and analysis of our financial condition and results of operations should be read in conjunction with our
consolidated  financial  statements  and  related  notes  included  elsewhere  in  this  Annual  Report  on  Form  10-K.  Some  of  the  information
contained in this discussion and analysis or set forth elsewhere in this Annual Report on Form 10-K, including information with respect to
our plans and strategy for our business, includes forward-looking statements that involve risks and uncertainties. You should review the
“Risk Factors” section in this Annual Report on Form 10-K for a discussion of important factors that could cause actual results to differ
materially from the results described in or implied by the forward-looking statements contained in the following discussion and analysis.

Results of Operations

Comparison of the Years Ended December 31, 2018 and 2017

The following table summarizes our revenue for the years ended December 31, 2018 and 2017

Product revenue, net
Sales force revenue
License and other revenue
Grant revenue

Product revenue, net    

Year Ended

December 31,

2018

2017

(in thousands)

  $

  $

17,871   $
456  
—  
—  
18,327   $

1,910
278
25,000
625
27,813

Product revenue, net was $17.9 million for the year ended December 31, 2018, compared to $1.9 million for the year ended

December 31, 2017. The net product revenue for the year ended December 31, 2018 represents a full year of revenues from the sale of
products acquired in the acquisition of TRx on November 17, 2017 and nearly a full year of sales of products acquired from the acquisition
of Avadel's pediatric products on February 16, 2018. The net product revenue for the year ended December 31, 2017 represents revenues
from the sale of our pediatric products following the acquisition of TRx on November 17, 2017.

Sales force revenue

As part of the acquisition of TRx in November 2017, the Company acquired a sales and marketing agreement with Pharmaceutical
Associates, Inc. ("PAI") in which the Company received a monthly marketing fee to promote, market and sell certain products on behalf of
PAI. The Company was also entitled to a share of PAI's profits. Sales force revenue was $0.5 million for the year ended December 31,
2018 as compared to $0.3 million for the year ended December 31, 2017. The increase was due to 1.5 months of revenue in 2017 as
compared to four months of revenue in 2018. The PAI contract was canceled during the second quarter of 2018.

License and other revenue

There was no license and other revenue for the year ended December 31, 2018, compared to $25.0 million for the year ended

December 31, 2017. In the third quarter of 2017, the Company sold CERC-501 to Janssen in exchange for initial gross proceeds of $25.0
million. Under this agreement, we are also eligible for a potential future $20.0 million regulatory milestone payment. The terms of the
agreement provide that Janssen will assume ongoing clinical trials and be responsible for any new development and commercialization of
CERC-501.

Grant revenue

There was no grant revenue for the year ended December 31, 2018, compared to  $0.6 million  for  the  year  ended December 31,
2017. The grant revenues for the year ended December 31, 2017 related to CERC-501 and were dependent upon the timing and progress of
the underlying studies and development activities. The grant revenue and study costs related to these grants were discontinued with the sale
of CERC-501 to Janssen in August 2017.

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Cost of product sales

Cost  of  product  sales  was $7.5 million  for  the  year  ended  December  31,  2018,  compared  to $0.6  million  for  the  year  ended
December 31, 2017. Cost of product sales related to sales of products from our pediatric products that we recently acquired. The increase of
$6.9 million in cost of product sales in the current year is due to the Company having a full year of sales of products acquired from the TRx
acquisition in 2017 and nearly a full year of sales of products acquired from the acquisition of Avadel's pediatric products on  February 16,
2018, while in the previous year the Company had approximately one month of sales since TRx was acquired on November 17, 2017.

Research and Development Expenses

The following table summarizes our research and development expenses for the years ended December 31, 2018 and 2017:

Preclinical expenses
Clinical expenses
CMC expenses
Internal expenses not allocated to programs:

Salaries, benefits and related costs
Stock-based compensation expense
Other

Year Ended

December 31,

2018

2017

(in thousands)

  $

  $

1,886   $
1,693  
389  

1,223  
101  
495  
5,787   $

1,162
607
677

1,476
152
299
4,373

Research  and  development  expenses  were $5.8  million  for  the  year  ended  December  31, 2018,  an  increase  of $1.4  million
compared to the same period in 2017. Preclinical expenses increased by $0.7 million primarily due to toxicology studies performed during
2018 in support of clinical development. Clinical expenses increased by $1.1 million compared to the same period in 2017 primarily due to
activities  related  to  the  CERC-301  clinical  study  in  nOH  and  activities  related  to  CERC-801,  CERC-802,  and  CERC-803,  which  were
acquired as part of the Ichorion acquisition in September 2018. Chemistry, Manufacturing, and Controls ("CMC") expenses decreased  $0.3
million  for  the  year  ended  December  31,  2018  compared  to  the  same  period  in  2017  due  to  higher  prior  year  spending  on  clinical  trial
material stability and drug product to support clinical development.

Acquired In-Process Research and Development Expenses

The following table summarizes our acquired in-process research and development ("IPR&D") expenses for years ended

December 31, 2018 and 2017:

Year Ended

December 31,

2018

2017

(in thousands)

Acquired in-process research and development

  $

18,724   $

—

As part of the asset acquisition of Ichorion, the Company acquired  $18.7 million of IPR&D expenses for three preclinical

therapies for inherited metabolic disorders known as CDGs (CERC-801, CERC-802 and CERC-803). The fair value of the IPR&D was
immediately recognized as acquired in-process research and development expense as the IPR&D asset has no other alternate use due to the
stage of development. There was no acquired in-process research and development expense for the year ended December 31, 2017.

General and Administrative Expenses

The following table summarizes our general and administrative expenses for the years ended December 31, 2018 and 2017: 

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Salaries, benefits and related costs
Legal, consulting and other professional expenses
Stock-based compensation expense
Other

Year Ended

December 31,

2018

2017

(in thousands)

  $

  $

3,607   $
4,426  
2,136  
508  
10,677   $

2,433
3,944
1,001
564
7,942

General  and  administrative  expenses  were $10.7  million  for  the  year  ended  December  31,  2018,  an  increase  of $2.7  million
compared  to  the  period  in  2017. Salaries,  benefits  and  related  costs  increased  by $1.2 million  for  the  year  ended  December  31,  2018
compared to the same period of 2017 due to an increase in salary related costs. Legal, consulting and other professional expenses increased
by $0.5 million compared to the same period of 2017 primarily as a result of the legal, compliance and integration costs associated with our
acquisitions. Stock-based  compensation  expense  increased  by $1.1 million  over  the  same  period  comparison  primarily  as  a  result  of  the
acceleration of the vesting of stock options of a senior executive who was separated in the period and the subsequent recognition of the
additional expense, in addition to stock compensation expense related to awards granted to new senior executives.

Sales and Marketing Expenses

The following table summarizes our sales and marketing expenses for the years ended December 31, 2018 and 2017: 

Salaries, benefits and related costs
Consulting and other professional expenses
Stock-based compensation expense
Advertising and marketing expense
Other

Year Ended

December 31,

2018

2017

(in thousands)

  $

  $

5,571   $
1,458  
194  
1,161  
138  
8,522   $

303
140
4
71
52
570

The Company began to incur sales and marketing expenses after the TRx acquisition on November 17, 2017. Sales and marketing
expenses  were $8.5 million  for  the  year  ended  December  31,  2018  as  compared  to $0.6 million  for  the  year  ended  December  31,  2017.
Salaries, benefits and related costs increased as a result of increasing sales and sales support personnel needed to maintain and grow our
commercial sales activities in connection with the acquired TRx and Avadel's pediatric products.  Logistics, insurance and other commercial
operations expenses were incurred in order to support commercial operations. Advertising and marketing expenses were incurred to support
the portfolio of pediatric drug products for sale. During the third quarter of 2018, the Company initiated an expansion of the sales force
which is expected to be largely completed by the end of the first quarter of 2019.

Amortization expense

The following table summarizes our amortization expense for the years ended December 31, 2018 and 2017:

Amortization of intangible assets

  $

4,532   $

404

Amortization  expense  was $4.5 million  for  the  year  ended  December  31,  2018  as  compared  to $0.4 million  for  the  year  ended
December 31, 2017. The amortization expense relates to the acquisition of intangible assets as part of the acquisitions of TRx in November

62

Year Ended

December 31,

2018

2017

(in thousands)

 
 
 
 
 
 
 
 
   
   
 
 
 
 
 
 
 
  
 
 
 
 
 
 
 
 
 
   
   
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
   
 
 
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2017 and Avadel's pediatric products in February 2018.  The increase of amortization expense of $4.1 million for the year ended December
31, 2018 as compared to 2017 is driven by a full year of amortization for the intangible assets acquired as part of the TRx acquisition and
amortization from February 16, 2018 through December 31, 2018 for the intangible assets acquired as part of Avadel's pediatric products in
2018. In 2017, the amortization relates only to the intangible assets acquired as part of the TRx acquisition for the period between the TRx
acquisition date on November 17, 2017 and December 31, 2017.

Impairment of Intangible Assets

The Company recorded impairment of intangible asset expense of $1.9 million for the year ended December 31, 2018 due to the
impairment  of  the  PAI  sales  and  marketing  agreement  intangible  asset  upon  termination  of  the  corresponding  agreement.  No  expense
related to impairment of intangible assets was recognized for the year ended December 31, 2017.

Change in fair value of contingent consideration

The Company recognized a loss on the change in fair value of contingent consideration of  $58,366 for the year ended December
31,  2018  as  compared  to  $0  for  the  same  period  in  2017.  The contingent consideration is related to the potential for future payment of
consideration  that  is  contingent  upon  the  achievement  of  operation  and  commercial  milestones  and  royalty  payments  on  future  product
sales  as  part  of  the  Company's  acquisitions  of  Avadel's  pediatric  products  and  TRx.  The  fair  value  of  contingent  consideration  was
determined  at  the  acquisition  date  (see  Note  5  for  more  information). Subsequent  to  the  acquisition  date,  at  each  reporting  period,  the
contingent  consideration  liability  is  remeasured  at  the  current  fair  value  with  changes  recorded  to  its  own  standalone  line  in  operating
expenses in the consolidated statement of operations.

Other expense, net

The following table summarizes our other expense, net for the years ended December 31, 2018 and 2017:

Change in fair value of warrant liability and unit purchase option liability
Other income, net
Interest expense, net

Year Ended

December 31,

2018

2017

  $

  $

(in thousands)

25   $
14  
(812)  
(773)   $

(30)
—
(24)
(54)

Other  expense,  net  was $0.8 million for the year ended December 31, 2018 as compared to $0.1 million for the same period in
2017. Interest expense increased $0.8 million for the year ended December 31, 2018 as compared to the same period in 2017. The interest
expense  recognized  in  the  year  ended  December  31,  2018  relates  to  interest  for  the  Deerfield  obligation  assumed  as  part  of  the Avadel
Pediatric Products Acquisition, which took place in the first quarter of 2018.  Interest expense was minimal for the year ended December
31, 2017 due to the reduction in the principal balance of the secured term loan facility which was paid off in August 2017.

Income tax (benefit) expense

The income tax benefit was $33,910 for the year ended December 31, 2018. The provision for income taxes for the year ended
December 31, 2018 is composed of an adjustment benefit from the return to provision true up of a prior year tax liability, offset by state
income tax of one subsidiary, and deferred income tax expense, all of which were not significant. The provision for income taxes was $2.0
million for the year ended December 31, 2017 due to the net income generated from the sale of CERC-501 to Janssen during the third
quarter of 2017. The annual effective tax rate was 0.09% and 14.21% for the years ended December 31, 2018 and 2017, respectively.

Non-GAAP Financial Metrics

In addition to disclosing financial results that are determined in accordance with U.S. Generally Accepted Accounting Standards

("GAAP"), the Company also uses the following non-GAAP financial metrics to understand and evaluate our operating performance:

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EBITDA, which the Company defines as GAAP net income adjusted for (i) taxes, (ii) interest expense, (iii) interest income, (iv)

amortization of intangible assets, (v) depreciation, and (vi) inventory step-up adjustment recognized in earnings.

Adjusted EBITDA, which the Company defines as EBITDA as defined above further adjusted for (i) stock-based compensation

expense, (ii) change in fair value of contingent consideration, (iii) change in fair value of warrant liability and unit purchase option
liability, (iv) restructuring costs, (v) acquisition and integration-related expenses, (vi) impairment of intangible assets, (vii) arbitration costs
related to the Lachlan transaction, which is further described in Item 1 Note 7, (viii) acquired IPR&D, which is further described in Item 1
Note 4, and (ix) sale or out-licensing of Company assets.

The Company updated our definition of Adjusted EBITDA during the third quarter of 2018 to further adjust for acquired IPR&D

and sale or out-licensing of Company assets. These updates did not impact previous presentation of prior periods.

The Company believes that providing this additional information is useful to the reader to better assess and understand our
operating performance, primarily because management typically monitors the business adjusted for these items in addition to GAAP
results. These non-GAAP financial metrics should be considered supplemental to and not a substitute for financial information prepared in
accordance with GAAP. Our definition of these non-GAAP metrics may differ from similarly titled metrics used by others. The Company
views these non-GAAP financial metrics as a means to facilitate our financial and operational decision-making, including evaluation of our
historical operating results and comparison to competitors’ operating results. These non-GAAP financial metrics reflect an additional way
of viewing aspects of our operations that, when viewed with GAAP results may provide a more complete understanding of factors and
trends affecting our business. The determination of the amounts that are adjusted from these non-GAAP financial metrics is a matter of
management judgment and depends upon, among other factors, the nature of the underlying expense or income amounts. Because non-
GAAP financial metrics adjust for the effect of items that will increase or decrease our reported results of operations, we strongly
encourage investors to review our consolidated financial statements and periodic reports in their entirety.

The following tables present reconciliations of these non-GAAP financial metrics to the most directly comparable GAAP

financial measure for the years ended December 31, 2018 and 2017:

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GAAP Net (loss) income
Non-GAAP Adjustments:
Income tax expense
Interest expense, net
Amortization of intangible assets
Depreciation
Inventory step-up adjustment recorded in earnings
EBITDA
Non-GAAP Adjustments:
Stock-based compensation
Change in fair value of contingent consideration
Change in fair value of warrant liability and unit purchase option liability
Restructuring costs
Acquisition and integration related expenses
Impairment of intangible assets
Lachlan legal arbitration costs
Acquired in-process research and development
Sale or out-licensing of Company assets
     Total Non-GAAP Adjustments
Adjusted EBITDA

Liquidity, Capital Resources and Expenditure Requirements

Year Ended December 31,

2018

2017

  $

(40,053)   $

11,870

(34)  
812  
4,532  
23  
301  
(34,419)   $

2,431  
58  
(25)  
533  
985  
1,862  
(178)  
18,724  
—  
24,390  
(10,029)   $

1,967
24
404
22
138
14,425

1,157
—
30
1,125
247
—
178
—
(25,000)
(22,263)
(7,838)

  $

  $

The  Company  applies  a  disciplined  decision-making  methodology  as  it  evaluates  the  optimal  allocation  of  the  Company's
resources between investing in the Company's current commercial product line, the Company's development portfolio and acquisitions or
in-licensing of new assets in order to meet its cash flow needs. For the year ended December 31, 2018, the Company generated a net loss of
$40.1 million and negative cash flow from operations of $3.1 million. As of December 31, 2018, the Company had an accumulated deficit
of $98.2 million and a balance of $10.6 million in cash and cash equivalents. During the third quarter of 2018, the Company entered into a
securities purchase agreement with Armistice, pursuant to which the Company sold 1,000,000 shares of the Company's common stock that
generated net proceeds of approximately $3.9 million (see "Armistice Private Placements" in Note 13 for a description of this transaction).
During  the  fourth  quarter  of  2018,  Armistice  exercised  warrants  for  convertible  preferred  stock  that  generated  net  proceeds  of
approximately  $5.7  million  (see  "December  2018  Armistice  Private  Placement"  in  Note  13  for  a  description  of  this  transaction).
Additionally,  during  the  first  quarter  of  2019,  the  Company  closed  on  an  underwritten  public  offering  of  common  stock  for 1,818,182
shares of common stock of the Company, at a price to the public of $5.50 per share ("public price"). Armistice participated in the offering
by purchasing 363,637 shares of common stock of the Company from the underwriter at the public price. The net proceeds to the Company
from the offering was approximately $9.0 million.

The Company plans to use cash and the anticipated positive net cash flows from the Company's existing product sales to offset

costs related to its pediatric rare disease preclinical programs, neurology clinical programs, business development, costs associated with its
organizational infrastructure and debt principal and interest payments. The Company expects to continue to incur significant expenses and
operating losses for the immediate future as it continues to invest in its pipeline assets. Our ability to achieve and maintain profitability in
the future is dependent on, among other things, the development, regulatory approval and commercialization of our new product candidates
and achieving a level of revenues from our existing product sales adequate to support our cost structure, which includes significant
investment in our pipeline assets.

The Company believes it will require additional financing to continue to execute its clinical development strategy and/or fund

future operations. The Company plans to meet its capital requirements through operating cash flows from product sales and some
combination of equity or debt financings, collaborations, out-licensing arrangements, strategic alliances, federal and private grants,

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marketing, distribution or licensing arrangements or the sale of current or future assets. If the Company is not able to secure adequate
additional funding, the Company may be forced to make reductions in spending, extend payment terms with suppliers, liquidate assets
where possible or suspend or curtail planned programs. If the Company raises additional funds through collaborations, strategic alliances or
licensing arrangements with third parties, the Company may have to relinquish valuable rights to our technologies, future revenue streams,
research programs or product candidates.

Our plan to aggressively develop our pipeline, including our recently acquired pediatric rare disease preclinical programs, will
require substantial cash inflows in excess of what the Company expects our current commercial operations to generate.  The Company
expects that our existing cash and cash equivalents, together with anticipated revenue, will enable us to fund our operating expenses, capital
expenditure requirements, and other non-operating cash payments such as fixed quarterly payments on our outstanding debt balances
through at least March 2020.

Uses of Liquidity
Ichorion Asset Acquisition

On September 24, 2018, the Company entered into a merger agreement in which we acquired Ichorion Therapeutics, Inc. The

consideration for the Ichorion acquisition at closing consisted of 5.8 million shares of the Company’s Common Stock, par value $0.001 per
share, as adjusted for estimated working capital.  The shares are subject to a lockup date of December 31, 2019. Consideration for the
Merger included certain development milestones worth up to an additional $15 million, payable either in shares of Company common stock
or in cash, at the election of the Company. There will be future cash outflow for research and development costs associated with the
development of the assets acquired as part of the Ichorion acquisition (CERC-801, CERC-802, CERC-803 and CERC-913).

Avadel Pediatric Products Acquisition

On  February  16,  2018,  the  Company  entered  into  an  asset  purchase  agreement  with  Avadel  US  Holdings,  Inc.,  Avadel
Pharmaceuticals (USA), Inc., Avadel Pediatrics, Inc., Avadel Therapeutics, LLC and Avadel Pharmaceuticals PLC (collectively “Avadel”)
to purchase and acquire all rights in Avadel’s pediatric products.  The Company made a nominal cash payment for the acquired assets and
assumed  certain  of  Avadel’s  financial  obligations  to  Deerfield  CSF,  LLC,  ("Deerfield")  which  include  a  $15  million  loan  due  in
January 2021 and certain royalty obligations through February 2026.

TRx Pharmaceuticals, LLC Acquisition

On  November  17,  2017,  Cerecor  and  TRx  Pharmaceuticals,  LLC  ("TRx")  entered  into  a  purchase  agreement  in  which  the
Company acquired TRx, including subsidiary Zylera Pharmaceuticals, LLC and its franchise of pediatric medications. The consideration
for the acquisition consists of $18.9 million in cash, subject to working capital adjustments, as well as approximately 7.5 million shares of
our common stock having a market value of $8.5 million and certain contingent consideration with a fair value of $1.4 million.

Deerfield Debt Obligation

In relation to the Company's acquisition of Avadel's pediatric products on February 16, 2018, the Company assumed an obligation
that Avadel had to Deerfield, (the "Deerfield Obligation"). Beginning in July 2018 through October 2020, the Company will pay a quarterly
payment of $262,500 to Deerfield. In January 2021, a balloon payment of $15,250,000 is due. The Deerfield Obligation was $15.4 million
as of December 31, 2018, of which $1.1 million is recorded as a current liability.

The  Deerfield  Obligation  contains  certain  covenants,  explained  below,  in  which  the  Company  is  in  compliance  with  as  of
December  31,  2018. The  Company  cannot  waive,  breach,  terminate  or  materially  amend  any  of  the  acquired Avadel  pediatric  products'
commercial,  supply,  and  distribution  agreements  which  include  the  Karbinal  Agreement,  the  AcipHex  Agreement,  and  the  Cefaclor
Agreement (See Note 11 for a full description of each of these agreements) until the Deerfield Obligation is paid in full. Further, until the
obligation  is  paid  in  full,  each  year  the  Company  must  complete  no  fewer  than  60,000  P1  product  details  and  no  fewer  than  50,000  P2
product details. A product detail is a meeting between a sales person and a health care professional where the sales person presents on the
Company's  products. A P1 is either the first presentation made or is the longest presentation during a meeting, while a P2 is the second
longest presentation made during a meeting. The restrictive nature of the Deerfield Obligation may impact the Company's ability to obtain
additional financings.

Cash Flows

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The following table summarizes our cash flows for the years ended December 31, 2018 and 2017: 

Net cash provided by (used in):
Operating activities
Investing activities
Financing activities
Net increase (decrease) in cash and cash equivalents

Net cash (used in) provided by operating activities

Year Ended

December 31,

2018

2017

(in thousands)

  $

  $

(3,128)   $
865  
10,404  
8,141   $

12,579
(18,912)
3,737
(2,596)

Net cash used in operating activities was $3.1 million for the year ended December 31, 2018 and consisted primarily of a net loss
of $40.1 million, offset by non-cash acquired in-process research and development of $18.7 million, depreciation and amortization of $4.6
million,  non-cash  stock-based  compensation  expense  of $2.4  million,  impairment  of  intangible  assets  of $1.9  million  and  changes  in
working  capital,  primarily,  an  increase  in  accrued  expenses  of  $7.8  million,  largely  related  to  the  Lachlan  minimum  obligations  as
discussed in Note 11 and an decrease in escrowed cash receivable of $3.8 million.

     Net cash provided by operating activities was $12.6 million for the year ended December 31, 2017 and consisted primarily of net
income of $11.9 million, adjusted for non-cash stock-based compensation expense of $1.2 million, depreciation and amortization of $0.4
million and changes in deferred tax liabilities of $0.8 million, and changes in working capital, primarily, a change in income tax payable
of $2.3 million and accrued expenses and other current liabilities of $2.0 million, offset by a change in escrowed cash receivable of $3.8
million.

Net cash provided by (used in) investing activities

Net cash provided by investing activities was $0.9 million for the year ended December 31, 2018 and consisted of $1.4 million of
cash acquired from the acquisition of Ichorion partially offset by purchase of property, plant and equipment of $0.6 million, which includes
leasehold improvement costs incurred as part of our lease for the Company's new corporate headquarters.

Net  cash  used  in  investing  activities  was $18.9 million  for  the  year  ended  December  31,  2017  and  consisted  primarily  of  the

upfront cash payment for the acquisition of TRx of $18.9 million.

Net cash provided by financing activities

Net cash provided by financing activities was $10.4 million for the year ended December 31, 2018, which consisted primarily of
proceeds of $5.7 million from the warrant exercise of non-voting preferred stock by Armistice Capital in December 2018, net proceeds of
$3.9 million from a private placement of equity securities to Armistice Capital in August 2018, and $1.1 million of proceeds from option
and warrant exercises throughout the year. The increase was partially offset by $0.3 million payment of contingent consideration related to
the Avadel acquisition.

Net cash provided by financing activities was $3.7 million for the year ended December 31, 2017, which consisted primarily of
net proceeds from the Armistice Capital transaction of  $4.6 million, proceeds from the sale of common stock to Maxim and Aspire Capital
of $1.4 million, offset by principal payments on our term loan of $2.4 million.

Critical Accounting Estimates and Assumptions

In preparing the financial statements, the Company makes estimates and assumptions that have an impact on assets, liabilities,
revenue and expenses reported. These estimates can also affect supplemental information disclosed by us, including information about
contingencies, risk and financial condition. The Company believes, given current facts and circumstances, our estimates and assumptions
are reasonable, adhere to GAAP and are consistently applied. Inherent in the nature of an estimate or assumption is the fact that actual
results may differ from estimates, and estimates may vary as new facts and circumstances arise.

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While  our  significant  accounting  policies  are  more  fully  described  in  Note  2  to  the  audited  consolidated  financial  statements
appearing at the end of this Annual Report on Form 10-K, we believe the following accounting policies are critical to the understanding of
our financial condition and results.

Product Revenue, Net

The Company generates substantially all of our revenue from sales of prescription pharmaceutical products to our customers and
have  identified  a  single  product  delivery  performance  obligation,  which  is  the  provision  of  prescription  pharmaceutical  products  to  our
customers  based  upon  master  service  agreements  in  place  with  wholesaler  distributors,  purchase  orders  from  retail  pharmacies  or  other
direct customers and a contractual arrangement with a specialty pharmacy. The performance obligation is satisfied at a point in time, when
control of the product has been transferred to the customer, either at the time the product has been received by the customer or to a lesser
extent  when  the  product  is  shipped.  The  Company  determines  the  transaction  price  based  on  fixed  consideration  in  its  contractual
agreements and the transaction price is allocated entirely to the performance obligation to provide pharmaceutical products. In determining
the  transaction  price,  a  significant  financing  component  does  not  exist  because  the  timing  from  when  the  Company  delivers  product  to
when the customers pay for the product is less than one year and the customers do not pay for product in advance of the transfer of the
product.

Revenues from sales of products are recorded net of any variable consideration for estimated allowances for returns, chargebacks,
distributor  fees,  prompt  payment  discounts,  government  rebates  and  other  common  gross-to-net  revenue  adjustments.  The  identified
variable  consideration  is  recorded  as  a  reduction  of  revenue  at  the  time  revenues  from  product  sales  are  recognized.  The  Company
recognizes revenue only to the extent that it is probable that a significant revenue reversal will not occur in a future period.

Provisions for returns and government rebates are included within current liabilities in the consolidated balance sheet. Provisions
for  prompt  payment  discounts  and  distributor  fees,  are  included  as  a  reduction  to  accounts  receivable.  Calculating  these  items  involves
estimates and judgments based on sales or invoice data, contractual terms, historical utilization rates, new information regarding changes in
these programs’ regulations and guidelines that would impact the amount of the actual rebates, our expectations regarding future utilization
rates  for  these  programs,  and  channel  inventory  data.  These  estimates  may  differ  from  actual  consideration  amount  received  and  the
Company will re-assess these estimates and judgments each reporting period to adjust accordingly.

Returns and Allowances

Consistent  with  industry  practice,  the  Company  maintains  a  return  policy  that  allows  customers  to  return  product  within  a
specified period both prior to and, in certain cases, subsequent to the product's expiration date. Our return policy generally allows customers
to receive credit for expired products within six months prior to expiration and within one year after expiration. The provision for returns
and  allowances  consists  of  estimates  for  future  product  returns  and  pricing  adjustments.  The  primary  factors  considered  in  estimating
potential product returns include:

•

•

•

•

•

the shelf life or expiration date of each
product;
historical levels of expired product
returns;
external data with respect to inventory levels in the wholesale distribution
channel;
external data with respect to prescription demand for our products;
and
the estimated returns liability to be processed by year of sale based on analysis of lot information related to actual historical
returns.

The Company's estimate for returns and allowances may be impacted by a number of factors, but the principal factor relates to the

level of inventory in the distribution channel.

Rebates

The Company is also subject to rebates on sales made under governmental pricing programs. For example, Medicaid rebates are
amounts  owed  based  upon  contractual  agreements  or  legal  requirements  with  public  sector  (Medicaid)  benefit  providers  after  the  final
dispensing of the product by a pharmacy to a benefit plan participant. Medicaid reserves are based on expected payments, which are driven
by patient usage, contract performance and field inventory that will be subject to a Medicaid rebate. Medicaid rebates are typically billed up
to 180 days after the product is shipped, however can be as much as 270 days after the quarter in which the product is dispensed to the
Medicaid participant. In addition to the estimates mentioned above, our calculation also requires other estimates, such as estimates of sales
mix, to determine which sales are subject to rebates and the amount of such rebates. Periodically, the Company adjusts the Medicaid rebate
provision  based  on  actual  claims  paid.  Due  to  the  delay  in  billing,  adjustments  to  actual  claims  paid  may  incorporate  revisions  of  this
provision  for  several  periods.  Because  Medicaid  pricing  programs  involve  particularly  difficult  interpretations  of  complex  statutes  and
regulatory guidance, our estimates could differ from actual experience.

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In  determining  estimates  for  these  rebates,  the  Company  considers  the  terms  of  the  contracts,  relevant  statutes,  historical

relationships of rebates to revenues, past payment experience, estimated inventory levels and estimated future trends.

Accounting Policy Elections Related to Adoption of New Revenue Recognition Standard

The Company elected the following practical expedients in applying Topic 606 to its identified revenue streams:

•

Portfolio approach - contracts within each revenue stream have similar characteristics and the Company believes this approach
would not differ materially than if applying Topic 606 to each individual contract.

• Modified retrospective approach - the Company applied Topic 606 only to contracts with customers which were not

•

•

•

completed at the date of initial application, January 1, 2018.
Significant financing component - the Company does not adjust the promised amount of consideration for the effects of a
significant financing component as the Company expects, at contract inception, that the period between when the Company
transfers a promised good or service to a customer and when the customer pays for that good or service will be one year or
less.
Shipping and handling activities - the Company considers any shipping and handling costs that are incurred after the customer
has obtained control of the product as a cost to fulfill a promise and will account for them as an expense.
Contract costs - the Company recognizes the incremental costs of obtaining a contract as an expense when incurred if the
amortization period of the asset that the Company otherwise would have recognized is one year or less.

The  Company  does  not  incur  costs  to  obtain  a  contract  or  costs  to  fulfill  a  contract  that  would  result  in  the  capitalization  of
contract costs. Specifically, internal sales commissions are costs to fulfill a contract and are expensed in the same period that revenue is
recognized,  which  is  typically  within  the  same  quarterly  reporting  period. Contract  costs  are  expensed  or  amortized  in  “Operating
expenses” on the accompanying Consolidated Statements of Operations.

The Company has not made significant changes to the judgments made in applying ASU 2014-09,  Revenue from Contracts with

Customers (Topic 606) ("ASU 2014-09") for the year ended December 31, 2018.

Cost of Product Sales

Cost  of  product  sales  is  comprised  of  (i)  costs  to  acquire  products  sold  to  customers,  (ii)  royalty,  license  payments  and  other
agreements granting the Company rights to sell related products, (iii) distribution costs incurred in the sale of products; (iv) the value of
any write-offs of obsolete or damaged inventory that cannot be sold, (v) minimum sale obligations, and (vi) minimum purchase obligations.
The Company acquired the rights to sell certain of its commercial products through license and assignment agreements with the original
developers  or  other  parties  with  interests  in  these  products.  These  agreements  obligate  the  Company  to  make  payments  under  varying
payment structures based on its net revenue from related products.

Stock-Based Compensation

The  Company  applies  the  provisions  of  ASC  718,  Compensation—Stock  Compensation  (“ASC  718”),  which  requires  the
measurement and recognition of compensation expense for all stock‑based awards made to employees, including employee stock options,
in the statements of operations.

For stock options issued to employees and members of the board of directors for their services, the Company estimates the grant
date fair value of each option using the Black‑Scholes option pricing model. The use of the Black‑Scholes option pricing model requires
management to make assumptions with respect to the expected term of the option, the expected volatility of the common stock consistent
with  the  expected  life  of  the  option,  risk‑free  interest  rates  and  expected  dividend  yields  of  the  common  stock.  For  awards  subject  to
service‑based  vesting  conditions,  including  those  with  a  graded  vesting  schedule,  the  Company  recognizes  stock‑based  compensation
expense equal to the grant date fair value of stock options on a straight‑line basis over the requisite service period, which is generally the
vesting term. Forfeitures are recorded as they are incurred as opposed to being estimated at the time of grant and revised.

For stock option grants with market-based conditions, compensation expense is recognized ratably over the attribution period. The
Company  estimates  the  fair  value  of  the  market-based  stock  option  grants  using  a  Monte-Carlo  simulation.  The  Company  generally
estimates fair value using assumptions, including the risk-free interest rate, the expected volatility of a peer group of similar companies, the
expected  term  of  the  awards  and  the  expected  dividend  yield.  The  expected  term  for  market-based  stock  option  awards  is  based  on  the
expected  term  calculated  using  a  Monte-Carlo  simulation.  These  estimates  involve  inherent  uncertainties  and  the  application  of
management’s judgment. If factors change and different assumptions are used, our stock-based compensation expense could be materially
different in the future.

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The assumptions we used to determine the fair value of stock options granted to employees and members of the board of directors

are as follows:

Service-based options
Risk-free interest rate
Expected term of options (in years)
Expected stock price volatility
Expected annual dividend yield
Market-based options
Risk-free interest rate
Expected term of options (in years)
Expected stock price volatility
Expected annual dividend yield

Year Ended December 31,

2018
2.51%   —  
5.0
  —  
55%   —  
0%   —  

3.01%  
6.25

65%  
0%  

2017
1.85%   —  
5.0
  —  
55%   —  
0%   —  

2.38%  
6.25
100%  
0%  

2.84%
2.8
60%
0%

The estimates involved in the valuations include inherent uncertainties and the application of our judgment. As a result, if factors
change and we use significantly different assumptions or estimates when valuing our stock options, our stock‑based compensation expense
could be materially different. We recognize compensation expense for only the portion of awards that are expected to vest.

Estimated Fair Value and Change in Fair Value of Contingent Consideration

The  Company's  business  acquisitions  of  Avadel's  pediatric  products  and  TRx  involve  the  potential  for  future  payment  of
consideration  that  is  contingent  upon  the  achievement  of  operation  and  commercial  milestones  and  royalty  payments  on  future  product
sales. The fair value of contingent consideration was determined at the acquisition date utilizing unobservable inputs such as the estimated
amount and timing of projected cash flows, the probability of success (achievement of the contingent event) and the risk-adjusted discount
rate used to present value the probability-weighted cash flows. Subsequent to the acquisition date, at each reporting period, the contingent
consideration liability is remeasured at the current fair value with changes recorded to its own standalone line in operating expenses in the
consolidated statement of operations.

As  part  of  the  acquisition  of Avadel's  pediatric  products,  in  connection  with  the  Deerfield  debt  obligation  the  Company  also
assumed a 15% annual royalty on net sales of the acquired Avadel pediatric products through February 2026.  The fair value of the future
royalty  is  the  expected  future  value  of  the  contingent  payments  discounted  to  a  present  value. The  estimated  fair  value  of  the  royalty
payments as of December 31, 2018 was $7.8 million. The significant assumptions used in estimating the fair value of the royalty payment
as of December 31, 2018 include (i) the expected net sales of the acquired Avadel pediatric products that are subject to the 15% royalty
based on the Company's net sales forecast, and (ii) the risk-adjusted discount rate of 8.1%, which is comprised of the risk-free interest rate
of 2.6% and a counterparty risk of 5.5%.

The  consideration  for  the  TRx  acquisition  includes  certain  potential  contingent  payments. First,  pursuant  to  the  TRx  purchase
agreement, the Company is required to pay $3.0 million to the Sellers upon the gross profit related to TRx products achieving or exceeding
a gross profit of $12.6 million in 2018. The Company did not achieve this contingent event in 2018 and therefore no value was assigned to
the  contingent  payout  for  the  year  ended  December  31,  2018. Additionally,  the  Company  will  pay $2.0 million  upon  the  transfer  of  the
Ulesfia  NDA  to  the  Company  ("NDA  Transfer  Milestone").  Finally,  the  Company  will  pay $2.0 million  upon  FDA  approval  of  a  new
dosage of Ulesfia ("FDA Approval Milestone").  The main inputs utilized to determine the fair value of each milestone is the probability of
the milestone's success, the expected time to successfully reach the milestone, and the risk-adjusted discount rate. The estimated fair value
of the NDA Transfer Milestone as of December 31, 2018 was $0.9 million. The significant assumptions used in estimating the fair value of
the NDA Transfer Milestone as of December 31, 2018 include (i) probability of milestone success of 45.0%, (ii) expected time to milestone
of 0.5 years, and (iii) risk-adjusted discount rate of 7.9%, which is comprised of the risk free rate of 2.4% and a counterparty risk of 5.5%.
The estimated fair value of the FDA Approval Milestone as of December 31, 2018 was  $0.4 million. The significant assumptions used in
estimating the fair value of the FDA Approval Milestone as of December 31, 2018 include (i) probability of milestone success at  22.5%,
(ii) expected time to milestone of 1.5 years, and (iii) risk-adjusted discount rate of 8.0%, which is comprised of the risk free rate of 2.5%
and a counterparty risk of 5.5%.

Income Taxes

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The Company accounts for income taxes under the asset and liability method in accordance with ASC 740, Income Taxes (“ASC
740”).  Deferred  tax  assets  and  liabilities  are  recognized  for  the  future  tax  consequences  attributable  to  differences  between  the  financial
statement carrying amounts of existing assets and liabilities and their respective tax bases using enacted tax rates in effect for the year in
which the differences are expected to affect taxable income. Deferred tax assets primarily include net operating loss ("NOL") and tax credit
carryforwards, accrued expenses not currently deductible and the cumulative temporary differences related to certain research and patent
costs. Certain tax attributes, including NOLs and research and development credit carryforwards, may be subject to an annual limitation
under Sections 382 and 383 of the Internal Revenue Code (the "IRC"). The portion of any deferred tax asset for which it is more likely than
not that a tax benefit will not be realized must then be offset by recording a valuation allowance. The Company recognizes the tax benefit
from  an  uncertain  tax  position  only  if  it  is  more  likely  than  not  to  be  sustained  upon  examination  based  on  the  technical  merits  of  the
position.  The  amount  for  which  an  exposure  exists  is  measured  as  the  largest  amount  of  benefit  determined  on  a  cumulative  probability
basis that the Company believes is more likely than not to be realized upon ultimate settlement of the position. The Company’s policy is to
record interest and penalties on uncertain tax positions as income tax expense. As of December 31, 2018, the Company did not believe any
material uncertain tax positions were present.

On  December  22,  2017,  the  “Tax  Cuts  and  Jobs Act”  ("TCJA"  or  "the Act")  was  enacted,  that  significantly  reforms  the  IRC.
Among its numerous changes to the IRC, the Act reduces U.S. federal corporate tax rate from 35% to 21%.  The analysis of the tax effects
of the Act was completed in 2018 and there were no material adjustments in 2018.

Inventory Valuation

Inventories are recorded at the lower of cost or net realizable value, with cost determined on a first-in, first-out basis. Cost is

determined based on actual cost. An allowance is established when management determines that certain inventories may not be saleable. If
inventory costs exceed expected market value due to obsolescence or quantities in excess of expected demand, we record reserves for the
difference between the cost and the market value. These reserves are recorded based upon various factors for our products, including the
level of product manufactured by the Company, the level of product in the distribution channel, current and projected product demand, the
expected shelf life of the product and firm inventory purchase commitments, demand, the expected shelf life of the product and firm
inventory purchase commitments.

Acquisitions

For acquisitions that meet the definition of a business under ASC 805, the Company records the acquisition using the acquisition

method of accounting. All of the assets acquired, liabilities assumed, contractual contingencies, and contingent consideration, when
applicable, are recorded at fair value at the acquisition date. Any excess of the purchase price over the fair value of the net assets acquired
is recorded as goodwill.  The application of the acquisition method of accounting requires management to make significant estimates and
assumptions in the determination of the fair value of assets acquired and liabilities assumed in order to properly allocate purchase price
consideration. For acquisitions that do not meet the definition of a business under ASC 805, the Company accounts for the transaction as an
asset acquisition.

Segment Information

Operating segments are identified as components of an enterprise about which separate discrete financial information is available
for  evaluation  by  the  chief  operating  decision  maker,  or  decision‑making  group,  in  making  decisions  on  how  to  allocate  resources  and
assess performance. The Company’s chief operating decision maker is the Company's Chief Executive Officer ("CEO").  The CEO views
the Company’s operations and manages the business as one operating segment. All long‑lived assets of the Company reside in the United
States.

Goodwill

Goodwill relates to the amount that arose in connection with the acquisitions of TRx and Avadel's pediatric products. Goodwill
represents the excess of the purchase price over the fair value of the net assets acquired when accounted for using the acquisition method
of accounting for business combinations. Goodwill is not amortized but is evaluated for impairment on an annual basis or more frequently
if an event occurs or circumstances change that would more-likely-than-not reduce the fair value of the Company's reporting unit below its
carrying amount. The Company consists of one reporting unit.

Intangible Assets

Intangible assets with definite useful lives are amortized over their estimated useful lives and reviewed for impairment if certain

events or changes in circumstances indicate that the carrying amount of an asset may not be recoverable. Intangible assets subject to

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amortization are reviewed for impairment whenever events or changes in circumstances indicate that the carrying amount of an intangible
asset might not be recoverable. Impairment losses are measured and recognized to the extent the carrying value of such assets exceeds their
fair value.

Off‑Balance Sheet Arrangements

The Company does not have any off‑balance sheet arrangements, as defined by applicable SEC rules and regulations.

Recently Adopted Accounting Pronouncements

For a discussion of new accounting standards please see Note 2 of Notes to Consolidated Financial Statements contained in this

Annual Report on Form 10-K.

JOBS Act

The JOBS Act contains provisions that, among other things, reduce reporting requirements for an “emerging growth company.”
As an emerging growth company, we have elected to not take advantage of the extended transition period afforded by the JOBS Act for the
implementation  of  new  or  revised  accounting  standards  and,  as  a  result,  will  comply  with  new  or  revised  accounting  standards  on  the
relevant dates on which adoption of such standards is required for non‑emerging growth companies.

Internal Control Over Financial Reporting

Assessing our staffing and training procedures to improve our internal control over financial reporting is an ongoing process. We
are not currently required to comply with all of Section 404 of the Sarbanes‑Oxley Act of 2002, or the Sarbanes‑Oxley Act.  For the year
ended  December  31,  2018,  management  is  required  to  make  an  assessment  of  the  effectiveness  of  our  internal  control  over  financial
reporting as required by Section 404(a) of the Sarbanes-Oxley Act, as further described in Item 9A of this Annual Report on Form 10-K.
The Dodd-Frank Wall Street Reform and Consumer Protection Act exempts non-accelerated filers from compliance with Section 404(b) of
the  Sarbanes-Oxley Act,  which  relates  to  the  independent  auditor's  attestation  on  the  effectiveness  of  the  issuer's  internal  control  over
financial reporting. As such, our independent registered public accounting firm has not been engaged to express, nor have they expressed,
an opinion on the effectiveness of our internal control over financial reporting as of December 31, 2018.

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Item 7A. Quantitative and Qualitative Disclosures About Market Risk.

Interest Rate Risk

As a smaller reporting company, we are not required to provide the information required by this Item.

Item 8. Financial Statements and Supplementary Data.

The consolidated financial statements required to be filed pursuant to this Item 8 are appended to this report. An index of those

consolidated financial statements is found in Item 15 of Part IV of this Annual Report on Form 10-K.

Item 9. Changes in and Disagreements with Accountants on Accounting and Financial Disclosure.

None.

Item 9A. Controls and Procedures.

Evaluation of Disclosure Controls and Procedures    

Under  the  supervision  and  with  the  participation  of  our  management,  including  our  principal  executive  officer  and  principal
financial officer, we conducted an evaluation of the effectiveness of the design and operation of our disclosure controls and procedures, as
defined in Rules 13a-15(e) and 15d-15(e) under the Exchange Act, as of the end of the period covered by this report.

In designing and evaluating our disclosure controls and procedures, management recognizes that any disclosure controls and

procedures, no matter how well designed and operated, can provide only reasonable assurance of achieving the desired control objectives.
In addition, the design of disclosure controls and procedures must reflect the fact that there are resource constraints and that management is
required to apply its judgment in evaluating the benefits of possible controls and procedures relative to their costs.

Based on their evaluation, our principal executive officer and principal financial officer concluded that as of December 31, 2018,
our disclosure controls and procedures are designed to, and are effective to, provide assurance at a reasonable level that the information we
are required to disclose in reports that we file or submit under the Exchange Act is recorded, processed, summarized and reported within
the time periods specified in SEC rules and forms, and that such information is accumulated and communicated to our management,
including our principal executive officer and principal financial officer, as appropriate, to allow timely decisions regarding required
disclosures as of December 31, 2018.

Management's Annual Report on Internal Control Over Financial Reporting

Our  management,  including  our  principal  executive  officer  and  principal  financial  officer,  is  responsible  for  establishing  and
maintaining  adequate  internal  control  over  financial  reporting  (as  defined  in  Rules  13a-15(f)  and  15d-15(f)  under  the  Exchange Act).
Internal control over financial reporting is a process designed to provide reasonable assurance regarding the reliability of financial reporting
and the preparation of financial statements for external purposes in accordance with GAAP. Our internal control over financial reporting
includes those policies and procedures that: (i) pertain to the maintenance of records that, in reasonable detail, accurately and fairly reflect
the  transactions  and  dispositions  of  our  assets;  (ii)  provide  reasonable  assurance  that  transactions  are  recorded  as  necessary  to  permit
preparation of financial statements in accordance with GAAP, and that our receipts and expenditures are being made only in accordance
with  authorizations  of  our  management  and  directors;  and  (iii)  provide  reasonable  assurance  regarding  prevention  or  timely  detection  of
unauthorized acquisition, use, or disposition of our assets that could have a material effect on the financial statements.

Under the supervision and with the participation of our management, including our Chief Executive Officer and Chief Financial
Officer, we conducted an evaluation of the effectiveness of our internal control over financial reporting as of December 31, 2018, based on
the Internal Control-Integrated Framework (2013) issued by the Committee of Sponsoring Organizations of the Treadway Commission
("COSO") (2013 Framework). Based on this evaluation under the 2013 Framework, our principal executive officer and principal financial
officer have concluded that our internal control over financial reporting was effective at a reasonable level of assurance as of December 31,
2018.

Changes in Internal Control Over Financial Reporting

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There were no changes in our internal control over financial reporting identified in  management’s  evaluation  pursuant  to  Rules
13a-15(d)  or  15d-15(d)  of  the  Exchange Act  during  the  most  recent  fiscal  quarter  that  materially  affected,  or  are  reasonably  likely  to
materially affect, our internal control over financial reporting.

Attestation Report of Registered Public Accounting Firm

This Annual Report on Form 10-K does not include an attestation report of our independent registered public accounting firm due to

an exemption established by the JOBS Act for emerging growth companies.

Item 9B. Other Information.

None.

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PART III

Item 10. Directors, Executive Officers and Corporate Governance.

Pursuant to Paragraph G(3) of the General Instructions to the Annual Report on Form 10-K, the information required by Part III

(Items 10, 11, 12, 13 and 14) is being incorporated by reference herein from our definitive proxy statement (or an amendment to our
Annual Report on Form 10-K) to be filed with the SEC within 120 days after the end of the fiscal year ended December 31, 2018 in
connection with our 2019 Annual Meeting of Stockholders.

Item 11. Executive Compensation.

See Item 10.

Item 12. Security Ownership of Certain Beneficial Owners and Management and Related Stockholder Matters.

See Item 10.

Item 13. Certain Relationships and Related Transactions, and Director Independence.

See Item 10.

Item 14. Principal Accounting Fees and Services.

See Item 10.

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 Item 15. Exhibits; Financial Statement Schedules.

(a) Documents filed as part of this
report.

PART IV

1.

The following consolidated financial statements of Cerecor Inc. and Report of Ernst & Young, LLP, Independent Registered
Public Accounting Firm, are included in this report:

Report of Independent Registered Public Accounting Firm 
Consolidated Balance Sheets as of December 31, 2018 and 2017
Consolidated Statements of Operations for the years ended December 31, 2018 and 2017
Consolidated Statements of Changes in Stockholders’ Equity for the period from January 1, 2017 to
December 31, 2018
Consolidated Statements of Cash Flows for the years ended December 31, 2018 and 2017
Notes to Financial Statements 

F-2
F-3
F-4

F-5
F-6
F-8

2.

3.

List of financial statement schedules. All schedules are omitted because they are not applicable or the required information is
shown in the financial statements described above.

List of Exhibits required by Item 601 of Regulation S-K. See part (b)
below.

(b) Exhibits.

The following is a list of exhibits filed as part of this Annual Report on Form 10-K. Where so indicated by footnote, exhibits that
were previously filed are incorporated by reference. For exhibits incorporated by reference, the location of the exhibit in the previous filing
is indicated.

Exhibit
Number

Description of Exhibit

2.1*

Asset Purchase Agreement, dated as of August 14, 2017, between Cerecor, Inc. and Janssen Pharmaceuticals, Inc.
(incorporated by reference to Exhibit 2.1 to the Current Report on Form 8-K filed on August 14, 2017).

2.2*

2.3*

2.4*#

Equity Interest Purchase Agreement, dated as of November 17, 2017, by and among Cerecor, Inc., TRx
Pharmaceuticals, LLC, Fremantle Corporation, LRS International LLC, the selling members of TRx
Pharmaceuticals, LLC, and solely for limited purposes stated therein, Randal O. Jones and Robert C. Moscato, Jr.
(incorporated by reference to Exhibit 2.1 to the Current Report on Form 8-K filed on November 17, 2017).

Agreement and Plan of Merger and Reorganization, dated as of November 17, 2017, by and among Cerecor, Inc.,
ZPC Merger Corp., a direct wholly owned subsidiary of Cerecor, Inc., Zylera Pharma Corp., Zylera
Pharmaceuticals, LLC, Fremantle Corporation and LRS International LLC (incorporated by reference to Exhibit
2.2 to the Current Report on Form 8-K filed on November 17, 2017).

Asset Purchase Agreement, dated February 12, 2018, by and between Cerecor Inc., Avadel US Holdings, Inc.,
Avadel Pharmaceuticals (USA), Inc., Avadel Pediatrics, Inc., FSC Therapeutics, LLC and Avadel
Pharmaceuticals PLC (incorporated by reference to Exhibit 2.1 to the Quarterly Report on Form 10-Q on May 11,
2018).

2.5*

Agreement and Plan of Merger, dated as of September 24, 2018, among Cerecor, Inc., ITX Merger Sub, Inc.,
Second ITX Merger Sub, LLC, Ichorion Therapeutics, Inc. and David Maizenberg, as holders’ representative
(incorporated by reference to Exhibit 2.1 to the Current Report on Form 8-K filed on September 26, 2018).

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3.1

Amended and Restated Certificate of Incorporation of Cerecor Inc. (incorporated by reference to Exhibit 3.1.2 to
the Current Report on Form 8-K filed on May 17, 2018).

3.1.1

Form of Certificate of Designation of Preferences, Rights and Limitations of Series A Convertible Preferred Stock
of Cerecor Inc. (incorporated by reference to Exhibit 3.1 to the Current Report on Form 8-K filed on April 28,
2017).

3.1.2

Form of Certificate of Series B Non-Voting Convertible Preferred Stock of Cerecor Inc. (incorporated by
reference to Exhibit 3.1 to the Current Report on Form 8-K filed on December 27, 2018).

3.2

4.1

4.2

4.3

4.4

4.5

4.6

4.7

4.8

4.9

4.1

4.11

4.12

Cerecor Inc. Second Amended and Restated Bylaws (incorporated by reference to Exhibit 3.2.1 to the Current
Report on Form 8-K filed on May 17, 2018).

Second Amended and Restated Investors' Rights Agreement, dated as of July 11, 2014 (incorporated by reference
to Exhibit 4.1 to the Registration Statement on Form S-1 filed on June 12, 2015).

Form of Warrant to Purchase Shares of Common Stock issued in connection with the sale of Series A Convertible
Preferred Stock (incorporated by reference to Exhibit 4.2 to the Registration Statement on Form S-1 filed on June
12, 2015).

Form of Warrant to Purchase Shares of Common Stock issued in connection with the sale of Series A-1
Convertible Preferred Stock, as amended by the Amendment to Common Stock Warrants, dated as of July 11,
2014 (incorporated by reference to Exhibit 4.3 to the Registration Statement on Form S-1 filed on June 12, 2015).

Form of Warrant to Purchase Shares of Common Stock, issued to CIFCO International Group and its affiliate
(incorporated by reference to Exhibit 4.5 to the Registration Statement on Form S-1 filed on June 12, 2015).

Form of Warrant to Purchase Shares of Common Stock issued in connection with the issuance of convertible
promissory notes from April 2014 through June 2014 (incorporated by reference to Exhibit 4.6 to the Registration
Statement on Form S-1 filed on June 12, 2015).

Warrant Agreement, dated as of August 19, 2014, issued to Hercules Technology Growth Capital, Inc.
(incorporated by reference to Exhibit 4.7 to the Registration Statement on Form S-1 filed on June 12, 2015).

Form of Unit Purchase Option (incorporated by reference to Annex IV of Exhibit 1.1 to the Registration
Statement on Form S-1 filed on June 12, 2015).

Form of Class A Warrant Agreement (incorporated by reference to Exhibit 4.9 to the Registration Statement on
Form S-1 filed on October 13, 2015).

Specimen Class A Warrant Certificate (incorporated by reference to Exhibit 4.10 to the Registration Statement on
Form S-1 filed on October 13, 2015).

Form of Class B Warrant Agreement (incorporated by reference to Exhibit 4.11 to the Registration Statement on
Form S-1 filed on October 13, 2015).

Specimen Class B Warrant Certificate (incorporated by reference to Exhibit 4.12 to the Registration Statement on
Form S-1 filed on October 13, 2015).

Specimen Unit Certificate (incorporated by reference to Exhibit 4.13 to the Registration Statement on Form S-1
filed on October 13, 2015).

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4.13

4.14

4.15

Registration Rights Agreement, dated as of September 8, 2016, by and between Aspire Capital Fund, LLC and
Cerecor Inc. (incorporated by reference to Exhibit 4.1 to the Current Report on Form 8-K filed on September 12,
2016).

Form of Warrant to Purchase Common Stock of Cerecor Inc. issued to Armistice Capital Master Fund Ltd.
(incorporated by reference to Exhibit 4.1 to the Current Report on Form 8-K filed on April 28, 2017).

Form of Warrant to Purchase Shares of Series B Non-Voting Convertible Preferred Stock of Cerecor Inc. issued
to Armistice Capital Master Fund Ltd. (incorporated by reference to Exhibit 4.1 to the Current Report on Form 8-
K filed on December 27, 2018).

4.16

Form of Warrant to Purchase Common Stock of Cerecor Inc. issued to Armistice Capital Master Fund Ltd.
(incorporated by reference to Exhibit 4.2 to the Current Report on Form 8-K filed on December 27, 2018).

10.1 #

10.2 #

10.3 #

Exclusive Patent and Know-How License Agreement, effective as of March 19, 2013, by and between Essex
Chemie AG and Cerecor Inc. (incorporated by reference to Exhibit 10.1 to the Registration Statement on Form S-
1 filed on June 12, 2015).

Exclusive Patent and Know-How License Agreement, effective as of March 19, 2013, by and between Essex
Chemie AG and Cerecor Inc. (incorporated by reference to Exhibit 10.2 to the Registration Statement on Form S-
1 filed on June 12, 2015).

Exclusive Patent and Know-How License Agreement, effective as of February 18, 2015, by and between Eli Lilly
and Company and Cerecor Inc. (incorporated by reference to Exhibit 10.3 to the Registration Statement on Form
S-1 filed on June 12, 2015).

10.4 +

Separation and Release Agreement, dated July 13, 2018, by and between Cerecor Inc. and Mariam Morris
(incorporated by reference to Exhibit 10.2 to the Current Report on Form 8-K filed on July 16, 2018).

10.5 +

Form of Director Indemnification Agreement (incorporated by reference to Exhibit 10.12 to the Registration
Statement on Form S-1 filed on September 8, 2015).

10.6

10.7

List of current directors with a Director Indemnification Agreement in the form provided as Exhibit 10.6
(incorporated by reference to Exhibit 10.13 to the Registration Statement on Form S-1 filed on September 8,
2015).

Loan and Security Agreement, dated as of August 19, 2014, by and between Cerecor Inc. and Hercules
Technology Growth Capital, Inc. (incorporated by reference to Exhibit 10.15 to the Registration Statement on
Form S-1 filed on June 12, 2015).

10.8

Non-Employee Director Compensation Policy, amended January 10, 2016 (incorporated by reference to Exhibit
10.17 to the Annual Report on Form 10-K filed on March 23, 2016).

10.9 +

Cerecor Inc. 2016 Employee Stock Purchase Plan (incorporated by reference to Exhibit 10.2 to the Current
Report on Form 8-K filed on May 20, 2016).

10.10#

License Agreement, dated as of September 8, 2016, by and between Cerecor Inc. and Eli Lilly and Company
(incorporated by reference to Exhibit 10.1 to the Quarterly Report on Form 10-Q filed on November 8, 2016).

78

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
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10.11

Addendum to Exclusive License Agreement, dated as of October 13, 2016, by and between Cerecor Inc. and Eli
Lilly and Company (incorporated by reference to Exhibit 10.1.1 to the Quarterly Report on Form 10-Q filed on
November 8, 2016).

10.12#

Securities Purchase Agreement, dated as of April 27, 2017, by and between Cerecor, Inc. and Armistice Capital
Master Fund Ltd. (incorporated by reference to Exhibit 10.1 to the Current Report on Form 8-K filed on April
28, 2017).

10.13

Registration Rights Agreement, dated as of April 27, 2017, by and between Cerecor, Inc. and Armistice Capital
Master Fund Ltd. (incorporated by reference to Exhibit 10.2 to the Current Report on Form 8-K filed on April
28, 2017).

10.14.1+

Employment Agreement by and between Cerecor Inc. and Robert C. Moscato, Jr., effective November 20, 2017
(incorporated by reference to Exhibit 10.25 to the Annual Report on Form 10-K on April 2, 2018).

10.14.2+

Separation and Release Agreement, dated April 23, 2018, by and between Cerecor, Inc. and Robert Moscato
(incorporated by reference to Exhibit 10.2 to the Current Report on Form 8-K filed on April 27, 2018).

10.15+

Employment Agreement, dated March 27, 2018, by and between Cerecor Inc. and Peter Greenleaf (incorporated
by reference to Exhibit 10.1 to the Current Report on Form 8-K filed on April 2, 2018).

10.16#

License and Development Agreement, dated February 16, 2018, by and between Cerecor Inc. and Flamel Ireland
Limited (incorporated by reference to Exhibit 10.2 to the Quarterly Report on Form 10-Q on May 11, 2018).

10.17+

Employment Agreement, dated January 22, 2018, by and between Cerecor Inc. and Matthew Phillips
(incorporated by reference to Exhibit 10.1 to the Current Report on Form 8-K filed on April 10, 2018).

10.18+

Employment Agreement, dated April 19, 2018, by and between Cerecor Inc. and James A. Harrell, Jr.
(incorporated by reference to Exhibit 10.1 to the Current Report on Form 8-K filed on April 27, 2018).

10.19+

Cerecor Inc. Amended and Restated 2016 Equity Incentive Plan (incorporated by reference to Exhibit 10.1 to the
Current Report on Form 8-K filed on May 17, 2018).

10.20+

Employment Agreement, dated July 12, 2018, by and between Cerecor Inc. and Joseph M. Miller (incorporated
by reference to Exhibit 10.1 to the Current Report on Form 8-K filed on July 16, 2018).

10.21+

Employment Agreement, dated July 16, 2018, by and between Cerecor Inc. and Pericles Calias (incorporated by
reference to Exhibit 10.3 to the Current Report on Form 8-K filed on July 16, 2018).

10.22

Securities Purchase Agreement, dated as of August 17, 2018, by and among Cerecor Inc. and each of the
investors (incorporated by reference to Exhibit 10.1 to the Current Report on Form 8-K filed on August 20,
2018).

10.23

Registration Rights Agreement, dated as of August 20, 2018, between Cerecor Inc. and each of the several
purchasers (incorporated by reference to Exhibit 10.2 to the Current Report on Form 8-K filed on August 20,
2018).

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
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Table of Contents

10.24

Lease dated September 14, 2018 by and between FP 540 Gaither, LLC and Cerecor Inc. (incorporated by
reference to Exhibit 10.1 to the Current Report on Form 8-K filed on September 18, 2018).

10.25

Securities Purchase Agreement, dated as of December 27, 2018, by and among Cerecor, Inc. and Armistice
Capital Master Fund Ltd. (incorporated by reference to Exhibit 10.1 to the Current Report on Form 8-K filed on
December 27, 2018).

10.26

Registration Rights Agreement, dated as of December 27, 2018, between Cerecor, Inc. and Armistice Capital
Master Fund Ltd. (incorporated by reference to Exhibit 10.2 to the Current Report on Form 8-K filed on
December 27, 2018).

21.1  

List of Subsidiaries of the Registrant.

23.1   Consent of Ernst & Young LLP, independent registered public accounting firm.

31.1   Certification of Principal Executive Officer pursuant to Section 302 of the Sarbanes-Oxley Act of 2002.

31.2   Certification of Principal Financial Officer pursuant to Section 302 of the Sarbanes-Oxley Act of 2002.

32.1 **

Certification of Chief Executive Officer and Chief Financial Officer pursuant to Section 906 of the Sarbanes-
Oxley Act of 2002.

101.INS   XBRL Instance Document.

101.SCH   XBRL Taxonomy Extension Schema Document.

101.CAL   XBRL Taxonomy Extension Calculation Linkbase Document.

101.DEF   XBRL Taxonomy Extension Definition Linkbase Document.

101.LAB   XBRL Taxonomy Extension Label Linkbase Document.

101.PRE   XBRL Taxonomy Extension Presentation Linkbase Document.

* The schedules to these agreements have been omitted pursuant to Item 601(b)(2) of Regulation S-K. The Company agrees to furnish a
copy of any schedule omitted from the agreements to the SEC upon request.

# Confidential treatment requested under 17 C.F.R. §§ 200.80(b)(4) and 230.406. The confidential portions of this exhibit have been
omitted and are marked accordingly. The confidential portions have been filed separately with the Securities and Exchange Commission.

+ Management contract or compensatory agreement.

80

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
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** This certification is being furnished solely to accompany this 10-K pursuant to 18 U.S.C. Section 1350, and are not being filed for
purposes of Section 18 of the Securities Exchange Act of 1934, as amended, and are not to be incorporated by reference into any filing of
the registrant, whether made before or after the date hereof, regardless of any general incorporation language in such filing.

Item 16. 10-K Summary.

None.

81

Table of Contents

Pursuant to the requirements of Section 13 or 15(d) of the Securities and Exchange Act of 1934, the registrant has duly caused this

report to be signed on its behalf by the undersigned thereunto duly authorized.

SIGNATURES

Cerecor Inc.

/s/    Peter Greenleaf
Peter Greenleaf
Chief Executive Officer

Date: March 18, 2019

Pursuant  to  the  requirements  of  the  Securities  and  Exchange Act  of  1934,  this  report  has  been  signed  below  by  the  following

persons on behalf of the registrant and in the capacities and on the dates indicated.

Signature

Title

/s/ Peter Greenleaf
Peter Greenleaf

  Chief Executive Officer and Director
  (Principal Executive Officer)

/s/    Joseph M. Miller
Joseph M. Miller

  Chief Financial Officer
  (Principal Financial and Accounting Officer)

Date

March 18, 2019

March 18, 2019

/s/    Uli Hacksell
Uli Hacksell

/s/    Isaac Blech
Isaac Blech

/s/    Steven J. Boyd
Steven J. Boyd

/s/    Phil Gutry
Phil Gutry

/s/    Simon C. Pedder
Simon C. Pedder

/s/    Magnus Persson

Magnus Persson

  Chairman of the Board

March 18, 2019

  Director

  Director

  Director

  Director

  Director

82

March 18, 2019

March 18, 2019

March 18, 2019

March 18, 2019

March 18, 2019

 
 
 
 
 
 
 
  
  
 
   
 
 
 
   
 
   
 
 
 
 
 
 
   
   
 
   
   
 
   
 
 
 
   
 
 
 
   
 
 
 
   
 
 
 
   
 
 
 
   
 
 
 
   
   
 
   
 
 
 
   
   
 
   
 
 
 
   
   
Table of Contents

CERECOR INC.
INDEX TO CONSOLIDATED FINANCIAL STATEMENTS

Report of Independent Registered Public Accounting Firm 
Consolidated Balance Sheets as of December 31, 2018 and 2017
Consolidated Statements of Operations for the years ended December 31, 2018 and 2017
Consolidated Statements of Changes in Stockholders’ Equity for the period from January 1, 2017 to
December 31, 2018
Consolidated Statements of Cash Flows for the years ended December 31, 2018 and 2017
Notes to Financial Statements 

F-2
F-3
F-4

F-5
F-6
F-8

F-1

Table of Contents

Report of Independent Registered Public Accounting Firm

To the Stockholders and the Board of Directors of Cerecor Inc.

Opinion on the Financial Statements

We have audited the accompanying consolidated balance sheets of Cerecor Inc. and subsidiaries (the Company) as of December 31, 2018
and 2017, the related consolidated statements of operations, changes in stockholders’ equity and cash flows for each of the two years in the
period ended December 31, 2018, and the related notes (collectively referred to as the “consolidated financial statements”). In our opinion,
the consolidated financial statements present fairly, in all material respects, the financial position of the Company at December 31, 2018
and  2017,  and  the  results  of  its  operations  and  its  cash  flows  for  each  of  the  two  years  in  the  period  ended  December  31,  2018,  in
conformity with U.S. generally accepted accounting principles.

Basis for Opinion

These financial statements are the responsibility of the Company's management. Our responsibility is to express an opinion on the financial
statements based on our audits. We are a public accounting firm registered with the Public Company Accounting Oversight Board (United
States) (PCAOB) and are required to be independent with respect to the Company in accordance with the U.S. federal securities laws and
the applicable rules and regulations of the Securities and Exchange Commission and the PCAOB.

We conducted our audits in accordance with the standards of the PCAOB. Those standards require that we plan and perform the audit to
obtain reasonable assurance about whether the financial statements are free of material misstatement, whether due to error or fraud. The
Company is not required to have, nor were we engaged to perform, an audit of its internal control over financial reporting. As part of our
audits  we  are  required  to  obtain  an  understanding  of  internal  control  over  financial  reporting  but  not  for  the  purpose  of  expressing  an
opinion on the effectiveness of the Company's internal control over financial reporting. Accordingly, we express no such opinion.

Our audits included performing procedures to assess the risks of material misstatement of the financial statements, whether due to error or
fraud, and performing procedures that respond to those risks. Such procedures included examining, on a test basis, evidence regarding the
amounts  and  disclosures  in  the  financial  statements.  Our  audits  also  included  evaluating  the  accounting  principles  used  and  significant
estimates  made  by  management,  as  well  as  evaluating  the  overall  presentation  of  the  financial  statements.  We  believe  that  our  audits
provide a reasonable basis for our opinion.

/s/ Ernst & Young LLP
We have served as the Company’s auditor since 2013.
Baltimore, Maryland
March 18, 2019

F-2

Table of Contents

CERECOR INC. and SUBSIDIARIES

Consolidated Balance Sheets

Assets
Current assets:

Cash and cash equivalents
Accounts receivable, net
Other receivables
Escrowed cash receivable
Inventory, net
Prepaid expenses and other current assets
Restricted cash, current portion

Total current assets
Property and equipment, net
Intangibles assets, net
Goodwill
Restricted cash, net of current portion

Total assets
Liabilities and stockholders’ equity
Current liabilities:

Accounts payable
Accrued expenses and other current liabilities
Income taxes payable
Long-term debt, current portion
Contingent consideration, current portion

Total current liabilities
Long term debt, net of current portion
Contingent consideration, net of current portion
Deferred tax liability, net
License obligations
Other long-term liabilities
Total liabilities

Stockholders’ equity:

Common Stock—$0.001 par value; 200,000,000 shares authorized at December 31, 2018 and
2017; 40,804,189 and 31,266,989 shares issued and outstanding at December 31, 2018 and
2017, respectively

Preferred Stock—$0.001 par value; 5,000,000 shares authorized at December 31, 2018 and
2017; 2,857,143 and zero shares issued and outstanding at December 31, 2018 and 2017,
respectively

Additional paid-in capital
Contingently issuable shares
Accumulated deficit
Total stockholders’ equity
Total liabilities and stockholders’ equity

  $

  $

  $

December 31,

2018

2017

10,646,301   $
3,157,555  
5,469,011  
—  
1,110,780  
1,529,516  
18,730  
21,931,893  
586,512  
31,239,468  
16,411,123  
81,725  
70,250,721   $

1,446,141   $
19,731,373  
2,032,258  
1,050,000  
1,956,807  
26,216,579  
14,327,882  
7,093,757  
69,238  
1,250,000  
385,517  
49,342,973  

2,472,187
2,935,025
427,241
3,752,390
382,153
703,225
1,959
10,674,180
44,612
17,664,480
14,292,282
131,353
42,806,907

1,298,980
7,531,122
2,259,148
—
—
11,089,250
—
2,576,633
7,144
1,250,000
24,272
14,947,299

40,804  

31,268

2,857  
119,082,157  
—  
(98,218,070)  
20,907,748  
70,250,721   $

—
83,338,136
2,655,464
(58,165,260)
27,859,608
42,806,907

  $

See accompanying notes to the consolidated financial statements.

F-3

 
 
 
 
 
 
 
      
      
   
   
 
 
 
 
 
 
 
 
 
 
 
   
   
   
   
 
 
 
 
 
 
 
 
 
 
 
   
   
 
 
 
 
 
 
 
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CERECOR INC. and SUBSIDIARIES

Consolidated Statements of Operations

Revenues

Product revenue, net
Sales force revenue
License and other revenue
Grant revenue

Total revenues, net

Operating expenses:

Cost of product sales
Research and development
Acquired in-process research and development
General and administrative
Sales and marketing
Amortization expense
Impairment of intangible assets
Change in fair value of contingent consideration

Total operating expenses

(Loss) income from operations
Other (expense) income:

Change in fair value of warrant liability and unit purchase option liability
Other income, net
Interest expense, net
Total other expense, net
Net (loss) income before taxes
Income tax (benefit) expense

Net (loss) income after taxes
Net (loss) income
Net (loss) income attributable to common shareholders

Net (loss) income per share of common stock, basic

Net (loss) income per share of common stock, diluted
Weighted-average shares of common stock outstanding, basic

Weighted-average shares of common stock outstanding, diluted

Year Ended December 31,

2018

2017

  $

17,870,745   $
456,056  
—  
—  
18,326,801  

1,910,403
278,165
25,000,000
624,569
27,813,137

7,478,262  
5,786,635  
18,723,952  
10,676,881  
8,522,461  
4,532,448  
1,861,562  
58,366  
57,640,567  
(39,313,766)  

25,010  
13,657  
(811,621)  
(772,954)  
(40,086,720)  
(33,910)  
(40,052,810)   $
(40,052,810)   $
(41,710,193)   $
(1.20)   $
(1.20)   $

34,773,613  
34,773,613  

635,648
4,372,578
—
7,941,584
569,825
403,520
—
—
13,923,155
13,889,982

(29,624)
—
(24,016)
(53,640)
13,836,342
1,966,519
11,869,823

11,869,823
7,772,084

0.42

0.42
18,410,005
18,754,799

  $
  $
  $
  $
  $

See accompanying notes to the consolidated financial statements.

F-4

 
 
 
 
 
 
 
   
   
 
 
 
 
 
   
   
   
   
 
 
 
 
 
 
 
 
 
 
   
   
 
 
 
 
 
 
 
 
 
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Balance, December 31, 2016
Issuance of common stock from
sale of shares under common
stock purchase agreement, net of
offering costs
Issuance of preferred and
common stock to Armistice
Capital, net of offering costs
Issuance of shares in acquisition
of TRx
Contingently issuable stock in
acquisition of TRx
Shares purchased through
employee stock purchase plan
Stock-based compensation
Conversion of Armistice Capital
preferred to common stock
Net income

Balance, December 31, 2017
Issuance of contingently
issuable shares in acquisition of
TRx
Issuance of shares pursuant to
common stock private
placement, net of offering costs
Issuance of shares in acquisition
of Ichorion assets

Issuance of Series B convertible
preferred stock upon warrant
exercise, net of offering costs
Exercise of stock options and
warrants
Shares purchased through
employee stock purchase plan
Stock-based compensation
Net loss

CERECOR INC. and SUBSIDIARIES

Consolidated Statements of Changes in Stockholders’ Equity

Stockholders’ Equity
  Additional

Total

Common stock

Preferred Stock

paid‑in

Shares
9,434,141   $

  Amount   Shares

  Amount  

9,434  

—   $

capital
—   $ 70,232,651   $

Contingently
issuable stock   Accumulated stockholders’
deficit
—   $(70,035,083)   $

Amount

207,002

equity

1,502,593

4,561,658

5,858,955

2,655,464

46,861
1,157,252

2,301,598  

2,302  

—  

—  

1,500,291    

2,345,714  

2,346  

—  

4  

4,559,308    

5,184,920  

5,185  

—    

5,853,770    

—  

60,616  
—  

—  

61  
—  

11,940,000  
—  

11,940  
—  
31,266,989   $ 31,268  

—  

—  
—  

—  
—  
—   $

—  

—  
—  

—  

2,655,464    

46,800    
1,157,252    

(11,936 )  
(4)  
—  
—    
—   $ 83,338,136  

—  

—
11,869,823   11,869,823
2,655,464   $(58,165,260)   $ 27,859,608

—  

2,349,968  

2,350    

2,653,114  

(2,655,464 )    

—

1,000,000  

1,000    

3,856,106    

5,774,464  

5,774    

19,965,780    

  2,857,143  

2,857  

5,682,181    

370,361  

370    

1,083,583    

42,407  

—  

42    

72,194    
2,431,063    
—  
$ 40,804   2,857,143   $ 2,857   $119,082,157  

—  

—  

—  

3,857,106

  19,971,554

5,685,038

1,083,953

72,236
2,431,063
—  
(40,052,810)   (40,052,810)
—   $(98,218,070)   $ 20,907,748

See accompanying notes to the consolidated financial statements.

F-5

Balance, December 31, 2018

40,804,189

 
 
 
 
   
   
 
 
 
 
 
 
 
 
 
 
 
   
 
   
 
 
   
 
 
   
 
   
 
 
   
 
 
   
 
   
 
   
 
   
 
   
   
 
   
 
   
 
   
 
   
 
 
   
   
   
 
   
 
 
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CERECOR INC. and SUBSIDIARIES

Consolidated Statements of Cash Flows

Operating activities
Net (loss) income
Adjustments to reconcile net (loss) income (used in) provided by to net cash (used in) provided by
operating activities:

Depreciation and amortization
Impairment of intangible assets
Stock-based compensation
Acquired in-process research and development, including transaction costs
Deferred taxes
Amortization of inventory fair value adjustment associated with acquisition of TRx and Avadel
Pediatric Product
Non-cash interest expense
Change in fair value of contingent consideration liability
Change in fair value of warrant liability and unit purchase option liability
Changes in assets and liabilities:

Accounts receivable, net
Other receivables
Inventory, net
Prepaid expenses and other assets

Escrowed cash receivable
Accounts payable
Income taxes payable
Accrued expenses and other liabilities
Other long term liabilities

Net cash (used in) provided by operating activities
Investing activities
Acquisition of TRx, net of cash acquired
Acquisition of Avadel Pediatric Products
Net cash acquired from acquisition of Ichorion Therapeutics, Inc.
Purchase of property and equipment
Net cash provided by (used in) investing activities
Financing activities
Proceeds from exercise of stock options and warrants
Proceeds from issuance of Series B convertible preferred stock upon warrant exercise, net
Proceeds from sale of shares pursuant to common stock private placement, net
Proceeds from sales of common stock purchased through employee stock purchase plan
Proceeds from sale of shares under common stock purchase agreement
Payment of contingent consideration
Principal payments on term debt
Payment of fractional shares upon conversion of preferred stock to common stock
Payment of offering costs
Net cash provided by financing activities
Increase (decrease) in cash and cash equivalents
Cash and cash equivalents at beginning of period

F-6

Year Ended December 31,

2018

2017

  $

(40,052,810)   $

11,869,823

4,554,963  
1,861,562  
2,431,063  
18,723,952  
(16,745 )  

300,573  
302,882  
58,366  
(25,010 )

(222,530)  
(2,277,255 )  
(311,199)  

(241,641)  
3,752,390  
82,451  
(226,890)  
7,792,259  
385,517  
(3,128,102 )  

—  
(1)  
1,429,877  
(564,415)  
865,461  

1,083,953  
5,685,038  
3,857,106  
72,236  
—  
(294,435)  
—  
—  
—  
10,403,898  
8,141,257  
2,605,499  

425,476
—
1,157,252
—
(832,629)

137,900
20,364
—
29,624

(247,195)
(427,241)
(24,276 )

(177,691)
(3,752,390 )
96,065
2,259,148
2,044,548
—
12,578,778

(18,888,932)
—
—
(23,325 )
(18,912,257)

—
—
4,649,996
46,861
1,693,498
—
(2,374,031 )
4
(279,247)
3,737,081
(2,596,398 )
5,201,897

 
 
 
 
 
 
      
      
   
   
 
 
 
 
 
 
 
 
 
   
   
 
 
 
 
 
 
 
 
 
 
   
   
 
 
 
 
 
   
   
 
 
 
 
 
 
 
 
 
 
 
 
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Cash and cash equivalents at end of period
Supplemental disclosures of cash flow information
Cash paid for interest

Cash paid for taxes

Supplemental disclosures of non-cash investing and financing activities
Debt assumed in Avadel Pediatric Products acquisition

Issuance of common stock in TRx acquisition

Contingently issuable shares in TRx acquisition

  $

  $
  $

  $
  $
  $

10,746,756   $

2,605,499

525,000   $
354,000   $

72,526

540,000

(15,075,000)   $
—   $
—   $

—

5,858,955

2,655,464

The following table provides a reconciliation of cash, cash equivalents and restricted cash reported within the consolidated balance

sheets that sum to the total of the same such amounts shown in the consolidated statements of cash flows:

Cash and cash equivalents
Restricted cash, current
Restricted cash, non-current

Total cash, cash equivalents and restricted cash

December 31,

2018

2017

  $

  $

10,646,301   $
18,730  
81,725  
10,746,756   $

2,472,187
1,959
131,353
2,605,499

See accompanying notes to the consolidated financial statements.

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1. Business

CERECOR INC. and SUBSIDIARIES

Notes to Consolidated Financial Statements

As of and for the Years Ended December 31, 2018 and 2017

Cerecor  Inc.  (the  "Company"  or  “Cerecor”)  is  a  fully  integrated  biopharmaceutical  company  with  commercial  operations  and
research  and  development  capabilities. The  Company  is  building  a  robust  pipeline  of  innovative  therapies  in  pediatric  healthcare,
neurology, and orphan rare diseases. The Company's neurology pipeline is led by CERC-301, which is currently in a Phase I safety study
for  Neurogenic  Orthostatic  Hypotension  ("nOH"). The  Company  is  also  developing two  other  neurological  clinical  and  preclinical  stage
compounds. The  Company's  pediatric  orphan  rare  disease  pipeline  is  led  by  CERC-801,  CERC-802  and  CERC-803. All three  of  these
compounds are preclinical therapies for inherited metabolic disorders known as Congenital Disorders of Glycosylation ("CDGs") by means
of  substrate  replacement  therapy. The  U.S.  Food  and  Drug  Administration  ("FDA")  has  granted  Rare  Pediatric  Disease  designation
("RPDD")  and  Orphan  Drug  Designation  ("ODD")  to  all three  compounds. Under  the  FDA’s  Rare  Pediatric  Disease  Priority  Review
Voucher ("PRV") program, upon the approval of a new drug application ("NDA") for the treatment of a rare pediatric disease, the sponsor
of  such  application  would  be  eligible  for  a  PRV  that  can  be  used  to  obtain  priority  review  for  a  subsequent  new  drug  application  or
biologics  license  application. The  PRV  may  be  sold  or  transferred  an  unlimited  number  of  times.  The  Company  plans  to  leverage  the
505(b)(2)  NDA  pathway  for  all three  compounds  to  accelerate  development  and  approval. The  Company  is  also  in  the  process  of
developing one other preclinical pediatric orphan rare disease compound, CERC-913.

The  Company  also  has  a  diverse  portfolio  of  marketed  products. Our  marketed  products  are  led  by  our  prescribed  dietary
supplements and prescribed drugs. Our prescribed dietary supplements include Poly-Vi-Flor and Tri-Vi-Flor which are prescription vitamin
and fluoride supplements used in infants and children to treat or prevent deficiency of essential vitamins and fluoride. The Company also
markets  a  number  of  prescription  drugs  that  treat  a  range  of  pediatric  diseases,  disorders  and  conditions. Cerecor's  prescription  drugs
include  Millipred®,  Ulesfia®,  Karbinal™  ER, AcipHex®  Sprinkle™  and  Cefaclor  for  Oral  Suspension.  Finally,  the  Company  has  one
marketed medical device, Flexichamber™.

Cerecor was incorporated in 2011, commenced operations in the second quarter of 2011 and completed an initial public offering in
October  2015. In August  2017,  the  Company  sold  its  worldwide  rights  to  CERC-501  to  Janssen  Pharmaceuticals,  Inc.  (“Janssen”)  in
exchange  for  initial  gross  proceeds  of $25  million,  of  which $3.75  million  was  deposited  into  a twelve-month  escrow  to  secure
indemnification obligations to Janssen. The Company collected the full amount of the escrow in August of 2018. Additionally, there is a
potential future $20 million regulatory milestone payment to the Company. The terms of the agreement provide that Janssen will assume
ongoing clinical trials and be responsible for any new development and commercialization of CERC-501.

On November 17, 2017, the Company acquired TRx Pharmaceuticals, LLC (“TRx”) and its wholly-owned subsidiaries (see "TRx

Acquisition" in Note 4 below for a description of the transaction).

On February 16, 2018, Cerecor acquired all rights to Avadel Pharmaceuticals PLC’s (“Avadel”) marketed pediatric products (the
“Acquired Products”) for the assumption of certain of Avadel's financial obligations (see "Avadel Pediatric Products Acquisition" in Note 4
below for a description of the transaction).

On September 25, 2018, the Company acquired Ichorion Therapeutics, Inc., a privately-held biopharmaceutical company focused
on developing treatments and increasing awareness of inherited metabolic disorders known as CDGs (see "Ichorion Asset Acquisition" in
Note 4 below for a description of the transaction).

Liquidity

The Company applies a disciplined decision-making methodology as it evaluates the optimal allocation of the Company's
resources between investing in the Company's current commercial product line, the Company's development portfolio and acquisitions or
in-licensing of new assets in order to meet its cash flow needs. For the year ended December 31, 2018, Cerecor generated a net loss of
$40.1 million and negative cash flow from operations of $3.1 million. As of December 31, 2018, Cerecor had an accumulated deficit of
$98.2 million and a balance of $10.6 million in cash and cash equivalents. During the third quarter of 2018, the Company entered into a
securities purchase agreement with Armistice Capital Master Fund Ltd. ("Armistice"), pursuant to which the Company sold 1,000,000
shares of the Company's common stock that generated net proceeds of approximately $3.9 million (see "Armistice Private Placements" in
Note 13 below for a description of the transaction). During the fourth quarter of 2018, Armistice exercised warrants for convertible
preferred stock that generated net proceeds of approximately $5.7 million (see "December 2018 Armistice

F-8

 
 
 
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Private Placement" in Note 13 below for a description of the transaction). Additionally, during the first quarter of 2019, the Company
closed on an underwritten public offering of common stock for 1,818,182 shares of common stock of the Company, at a price to the public
of $5.50 per share ("public price"). Armistice participated in the offering by purchasing 363,637 shares of common stock of the Company
from the underwriter at the public price. The net proceeds of the offering was approximately $9.0 million.

The Company plans to use cash and the anticipated positive net cash flows from the Company's existing product sales to offset

costs related to its pediatric rare disease programs, neurology clinical programs, business development, costs associated with its
organizational infrastructure and debt principal and interest payments. Cerecor expects to continue to incur significant expenses and
operating losses for the immediate future as it continues to invest in the Company's pipeline assets. Our ability to achieve and maintain
profitability in the future is dependent on, among other things, the development, regulatory approval and commercialization of our new
product candidates and achieving a level of revenues from our existing product sales adequate to support our cost structure, which includes
significant investment in our pipeline assets.

The Company believes it will require additional financing to continue to execute its clinical development strategy and/or fund

future operations. The Company plans to meet its capital requirements through operating cash flows from product sales and some
combination of equity or debt financings, collaborations, out-licensing arrangements, strategic alliances, federal and private grants,
marketing, distribution or licensing arrangements or the sale of current or future assets. If the Company is not able to secure adequate
additional funding, the Company may be forced to make reductions in spending, extend payment terms with suppliers, liquidate assets
where possible or suspend or curtail planned programs. If the Company raises additional funds through collaborations, strategic alliances or
licensing arrangements with third parties, the Company may have to relinquish valuable rights to our technologies, future revenue streams,
research programs or product candidates.

Our plan to aggressively develop our pipeline, including our recently acquired pediatric rare disease preclinical programs, will
require substantial cash inflows in excess of what the Company expects our current commercial operations to generate.  The Company
expects that our existing cash and cash equivalents, together with anticipated revenue, will enable us to fund our operating expenses, capital
expenditure requirements, and other non-operating cash payments such as fixed quarterly payments on our outstanding debt balances
through at least March 2020.

2. Significant Accounting Policies

Basis of Presentation

The accompanying consolidated financial statements have been prepared in accordance with U.S. generally accepted accounting
principles  (“GAAP”). Any  reference  in  these  notes  to  applicable  guidance  is  meant  to  refer  to  the  authoritative  GAAP  as  found  in  the
Accounting  Standards  Codification  (“ASC”)  and Accounting  Standards  Updates  (“ASU”)  of  the  Financial Accounting  Standards  Board
(the “FASB”).

Reclassification

During  2018,  the  Company  concluded  that  going  forward  it  would  net  amounts  due  to  distributors  against  open  receivable
balances. The Company has reclassified $0.3 million from accrued expenses and other current liabilities to accounts receivable, net in the
December 31, 2017 balance sheet to conform with current period presentation.

During 2018, the Company concluded that going forward it would include amortization expense within its own standalone line in
operating  expenses  in  the  Company's  consolidated  statements  of  operations. The  Company  has  reclassified $0.4 million  from  sales  and
marketing expenses in the December 31, 2017 statements of operations to conform with current period presentation.

Principles of Consolidation

The consolidated financial statements include the accounts of Cerecor Inc. and its wholly-owned subsidiaries after elimination of

all intercompany balances and transactions.

Use of Estimates

The  preparation  of  consolidated  financial  statements  in  conformity  with  GAAP  requires  management  to  make  estimates  and
assumptions  that  affect  the  reported  amounts  of  assets,  liabilities,  revenues,  expenses,  and  related  disclosures.  On  an  ongoing  basis,
management evaluates its estimates, including estimates related to but not limited to, revenue recognition, cost of product sales, stock-based
compensation,  fair  value  measurements  (including  those  relating  to  contingent  consideration),  cash  flows  used  in  management's  going
concern assessment, income taxes, goodwill and other intangible assets, and clinical trial accruals. The Company bases its estimates

F-9

 
 
 
 
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on historical experience and other market‑specific or other relevant assumptions that it believes to be reasonable under the circumstances.
Actual results may differ from those estimates or assumptions.

Cash and Cash Equivalents

The Company considers all highly liquid investments with an original maturity of three months or less when purchased to be cash
equivalents. The carrying amounts reported in the balance sheets for cash and cash equivalents are valued at cost, which approximates their
fair value.

Escrowed Cash Receivable

On August  14,  2017,  the  Company  sold  all  of  its  rights  to  CERC-501  to  Janssen  in  exchange  for  initial  gross  proceeds  of $25
million,  of  which $3.75 million  was  deposited  into  a twelve-month  escrow  to  secure  certain  indemnification  obligations  to  Janssen.  The
Company collected the full escrow amount in August 2018.

Restricted Cash

Restricted cash consists of the 2016 Employee Stock Purchase Plan (the "Plan") deposits and credit card deposits. In exchange for
receiving business credit card services from Silicon Valley Bank, the Company deposited $50,000 as collateral with Silicon Valley Bank.
These  deposits  are  recorded  as  restricted  cash,  net  of  current  portion  on  the  balance  sheet  at  December  31,  2018. Additionally,  deposits
made by employees for future stock purchases as part of the Plan is recorded as restricted cash. As part of the Plan, eligible employees can
purchase common stock through accumulated payroll deductions at such times as are established by the Plan administrator.

The Company adopted ASU No. 2016-18, Restricted Cash ("ASU 2016-18") effective January 1, 2018 and now includes
restricted cash balances within the cash, cash equivalents and restricted cash balance on the statement of cash flows. All prior periods were
retrospectively adjusted to conform to the current period presentation.

Accounts Receivable, net

Accounts receivable, net is comprised of amounts due from customers in the ordinary course of business. Management considers

all accounts receivable to be fully collectible at December 31, 2018, and accordingly, no allowance for doubtful accounts has been
recorded. Bad debt expense is charged to operations as amounts are determined to be uncollectible. Accounts receivable are written off
when deemed uncollectible and recoveries of receivables previously written off are recorded when received.

Accounts receivable are considered to be past due if any portion of the receivable balance is outstanding for more than the
payment terms negotiated with the customer. The Company generally negotiates payment terms of 30 days. The Company offers wholesale
distributors a prompt payment discount, which is typically 2% as an incentive to remit payment within this timeframe. Accounts receivable
are stated net of the estimated prompt pay discount.

Concentration of Credit Risk

Financial instruments that potentially subject the Company to concentrations of credit risk are primarily cash and cash equivalents.
The  Company  maintains  a  portion  of  its  cash  and  cash  equivalent  balances  in  the  form  of  a  money  market  account  with  a  financial
institution that management believes to be creditworthy. The Company has no financial instruments with off‑balance sheet risk of loss.

Inventory

Inventory consists primarily of finished goods stated at the lower of cost or net realizable value, with cost determined on a first-in,
first-out  basis.  The  Company  reviews  the  composition  of inventory  at  each  reporting  period  in  order  to  identify  obsolete,  slow-moving,
quantities in excess of expected demand, or otherwise non-saleable items. If non-saleable items are observed and there are no alternate uses
for the inventory, the Company will record a write-down to net realizable value in the period that the decline in value is first recognized.
These  valuation  adjustments  are  recorded  based  upon  various  factors  for  the  Company’s  products,  including  the  level  of   product
manufactured by the Company, the level of product in the distribution channel, current and projected product demand, the expected shelf
life of the product and firm inventory purchase commitments.

Property and Equipment

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Table of Contents

Property and equipment consists of computers, office equipment, furniture, and leasehold improvements and is recorded at cost.
Maintenance and repairs that do not improve or extend the lives of the respective assets are expensed to operations as incurred. Property
and  equipment  are  depreciated  on  a  straight‑line  basis  over  their  estimated  useful  lives.  The  Company  uses  a  life  of four  years  for
computers and software, and five years for equipment and furniture. For leasehold improvements, deprecation of the asset will begin at the
date it is placed in service and the depreciable life of the leasehold improvement is the shorter of the lease term or the improvement's useful
life. The  Company  uses  a  life  of ten years for  leasehold  improvements. Upon  retirement  or  sale,  the  cost  of  the  disposed  asset  and  the
related accumulated depreciation are removed from the accounts and any resulting gain or loss is recognized.

Acquisitions

For acquisitions that meet the definition of a business under ASC 805, the Company records the acquisition using the acquisition

method of accounting. All of the assets acquired, liabilities assumed, contractual contingencies, and contingent consideration, when
applicable, are recorded at fair value at the acquisition date. Any excess of the purchase price over the fair value of the net assets acquired
is recorded as goodwill.  The application of the acquisition method of accounting requires management to make significant estimates and
assumptions in the determination of the fair value of assets acquired and liabilities assumed in order to properly allocate purchase price
consideration. For acquisitions that do not meet the definition of a business under ASC 805, the Company accounts for the transaction as an
asset acquisition.

Segment Information

Operating segments are identified as components of an enterprise about which separate discrete financial information is available
for  evaluation  by  the  chief  operating  decision  maker,  or  decision‑making  group,  in  making  decisions  on  how  to  allocate  resources  and
assess  performance.  The  Company’s  chief  operating  decision  maker  is  the  Company's  Chief  Executive  Officer.  The  CEO  views  the
Company’s  operations  and  manages  the  business  as  one  operating  segment. All  long‑lived  assets  of  the  Company  reside  in  the  United
States.

Goodwill

Goodwill relates to the amount that arose in connection with the acquisitions of TRx and Avadel's pediatric products. Goodwill
represents the excess of the purchase price over the fair value of the net assets acquired when accounted for using the acquisition method
of accounting for business combinations. Goodwill is not amortized but is evaluated for impairment on an annual basis or more frequently
if an event occurs or circumstances change that would more-likely-than-not reduce the fair value of the Company's reporting unit below its
carrying amount. The Company consists of one reporting unit.

Intangible Assets

Intangible assets with definite useful lives are amortized over their estimated useful lives and reviewed for impairment if certain
events  or  changes  in  circumstances  indicate  that  the  carrying  amount  of  an  asset  may  not  be  recoverable.  Intangible  assets  subject  to
amortization are reviewed for impairment whenever events or changes in circumstances indicate that the carrying amount of an intangible
asset might not be recoverable. Impairment losses are measured and recognized to the extent the carrying value of such assets exceeds their
fair value.

Product Revenues, net

The Company generates substantially all of its revenue from sales of prescription pharmaceutical products to its customers and has
identified a single product delivery performance obligation, which is the provision of prescription pharmaceutical products to its customers
based  upon  master  service  agreements  in  place  with  wholesaler  distributors,  purchase  orders  from  retail  pharmacies  or  other  direct
customers and a contractual arrangement with a specialty pharmacy. The performance obligation is satisfied at a point in time, when control
of the product has been transferred to the customer, either at the time the product has been received by the customer or to a lesser extent
when the product is shipped. The Company determines the transaction price based on fixed consideration in its contractual agreements and
the transaction price is allocated entirely to the performance obligation to provide pharmaceutical products. In determining the transaction
price, a significant financing component does not exist because the timing from when the Company delivers product to when the customers
pay for the product is less than one year and the customers do not pay for product in advance of the transfer of the product.

Revenues from sales of products are recorded net of any variable consideration for estimated allowances for returns, chargebacks,

distributor fees, prompt payment discounts, government rebates, and other common gross-to-net revenue adjustments. The identified

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Table of Contents

variable  consideration  is  recorded  as  a  reduction  of  revenue  at  the  time  revenues  from  product  sales  are  recognized. The  Company
recognizes revenue only to the extent that it is probable that a significant revenue reversal will not occur in a future period.

Provisions for returns and government rebates are included within current liabilities in the consolidated balance sheet. Provisions
for  prompt  payment  discounts  and  distributor  fees  are  included  as  a  reduction  to  accounts  receivable.  Calculating  these  items  involves
estimates and judgments based on sales or invoice data, contractual terms, historical utilization rates, new information regarding changes in
these programs’ regulations and guidelines that would impact the amount of the actual rebates, our expectations regarding future utilization
rates  for  these  programs,  and  channel  inventory  data. These  estimates  may  differ  from  actual  consideration  amount  received  and  the
Company will re-assess these estimates and judgments each reporting period to adjust accordingly.

The following table presents net revenues disaggregated by type:

Prescribed dietary supplements
Prescription drugs
Sales force revenue
License and other revenue
Grant revenue

Total revenues, net

Concentration with Customer

Year Ended December 31,

2018

  $

7,678,003   $
10,192,742  
456,056  
—  
—  
  $ 18,326,801  

2017
1,092,271
818,132
278,165
25,000,000
624,569
$27,813,137

As is typical in the pharmaceutical industry, the Company sells its prescription pharmaceutical products (which include prescribed
dietary  supplements  and  prescription  drugs)  in  the  United  States  primarily  through  wholesale  distributors  and  a  specialty  contracted
pharmacy. Wholesale distributors account for substantially all of the Company’s net product revenues and trade receivables. In addition,
the  Company  earns  revenue  from  sales  of  its  prescription  pharmaceutical  products  directly  to  retail  pharmacies.      For  the  year  ended
December  31,  2018,  the  Company’s  three  largest  customers  accounted  for  approximately 30%,  30%,  and 25%,  respectively,  of  the
Company's  total  net  product  revenues  from  sale  of  prescription  pharmaceutical  products. For  the  year  ended  December  31,  2017,  the
Company’s  three  largest  customers  accounted  for  approximately  40%, 25%  and 22%,  respectively,  of  the  Company’s  total  net  product
revenues from sale of prescription pharmaceutical products.

Returns and Allowances

Consistent  with  industry  practice,  the  Company  maintains  a  return  policy  that  allows  customers  to  return  product  within  a
specified  period  both  prior  to  and,  in  certain  cases,  subsequent  to  the  product's  expiration  date.  The  Company’s  return  policy  generally
allows  customers  to  receive  credit  for  expired  products  within  six  months  prior  to  expiration  and  within  one  year  after  expiration.  The
provision  for  returns  and  allowances  consists  of  estimates  for  future  product  returns  and  pricing  adjustments.  The  primary  factors
considered in estimating potential product returns include:

the shelf life or expiration date of each product;
historical levels of expired product returns;
external data with respect to inventory levels in the wholesale distribution channel;
external data with respect to prescription demand for the Company’s products; and
the estimated returns liability to be processed by year of sale based on analysis of lot information related to actual

•
•
•
•
•
historical returns.

The Company’s estimate for returns and allowances may be impacted by a number of factors, but the principal factor relates to the level of
inventory in the distribution channel.

Rebates

The  Company  is  subject  to  rebates  on  sales  made  under  governmental  pricing  programs. For  example,  Medicaid  rebates  are
amounts  owed  based  upon  contractual  agreements  or  legal  requirements  with  public  sector  (Medicaid)  benefit  providers  after  the  final
dispensing of the product by a pharmacy to a benefit plan participant. Medicaid reserves are based on expected payments, which are

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driven by patient usage, contract performance and field inventory that will be subject to a Medicaid rebate. Medicaid rebates are typically
billed up to 180 days after the product is shipped, however can be as much as 270 days after the quarter in which the product is dispensed to
the  Medicaid  participant. In addition to the estimates mentioned above, the Company’s calculation also requires other estimates, such as
estimates of sales mix, to determine which sales are subject to rebates and the amount of such rebates. Periodically, the Company adjusts
the Medicaid rebate provision based on actual claims paid. Due to the delay in billing, adjustments to actual claims paid may incorporate
revisions of this provision for several periods. Because Medicaid pricing programs involve particularly difficult interpretations of complex
statutes and regulatory guidance, our estimates could differ from actual experience.

In  determining  estimates  for  these  rebates,  the  Company  considers  the  terms  of  the  contracts,  relevant  statutes,  historical

relationships of rebates to revenues, past payment experience, estimated inventory levels and estimated future trends.

Sales Force Revenue

Pursuant to a marketing agreement with Pharmaceutical Associates, Inc. (“PAI”), the Company received a monthly marketing fee

to promote, market and sell certain products on behalf of PAI. The Company was also entitled to a share of PAI's profits under the
agreement. Marketing fees and profit-sharing was recognized as sale force revenue when all the performance obligations have been
satisfied and to the extent that it was probable that a significant revenue reversal would not occur in a future period. The marketing
agreement with PAI was terminated in April 2018.

License and Other Revenue

The  Company  recognizes  revenues  from  collaboration,  license  or  other  research  or  sale  arrangements  when  or  as  performance
obligations  are  satisfied. For  milestone  payments,  the  Company  assesses,  at  contract  inception,  whether  the  milestones  are  considered
probable of being achieved. If it is probable that a significant revenue reversal will occur, the Company will not record revenue until the
uncertainty  has  been  resolved. Milestone  payments  that  are  contingent  upon  regulatory  approval  are  not  considered  probable  until  the
approvals are obtained as it is outside of the control of the Company.  If it is probable that significant revenue reversal will not occur, the
Company  will  estimate  the  milestone  payments  using  the  most  likely  amount  method. The  Company  will  re-assess  the  milestones  each
reporting period to determine the probability of achievement.

Grant Revenue

Grant revenues are derived from government grants that support the Company’s efforts on specific research projects. The

Company determined that the government agencies providing grants to the Company are not our customers. The Company recognizes
grant revenue when there is reasonable assurance of compliance with the conditions of the grant and reasonable assurance that the grant
revenue will be received.

Accounting Policy Elections Related to Adoption of New Revenue Recognition Standard

The Company elected the following practical expedients in applying Topic 606 to its identified revenue streams:

•

Portfolio approach - contracts within each revenue stream have similar characteristics and the Company believes this approach
would not differ materially than if applying Topic 606 to each individual contract.

• Modified retrospective approach - the Company applied Topic 606 only to contracts with customers that were not completed

•

•

•

at the date of initial application, January 1, 2018.
Significant financing component - the Company does not adjust the promised amount of consideration for the effects of a
significant financing component as the Company expects, at contract inception, that the period between when the Company
transfers a promised good or service to a customer and when the customer pays for that good or service will be one year or
less.
Shipping and handling activities - the Company considers any shipping and handling costs that are incurred after the customer
has obtained control of the product as a cost to fulfill a promise and will account for them as an expense.
Contract costs - the Company recognizes the incremental costs of obtaining a contract as an expense when incurred if the
amortization period of the asset that the Company otherwise would have recognized is one year or less.

The  Company  does  not  incur  costs  to  obtain  a  contract  or  costs  to  fulfill  a  contract  that  would  result  in  the  capitalization  of
contract costs. Specifically, internal sales commissions are costs to fulfill a contract and are expensed in the same period that revenue is
recognized,  which  is  typically  within  the  same  quarterly  reporting  period. Contract  costs  are  expensed  or  amortized  in  “Operating
expenses” on the accompanying Consolidated Statements of Operations.

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The Company has not made significant changes to the judgments made in applying ASU 2014-09,  Revenue from Contracts with

Customers (Topic 606) for the year ended December 31, 2018.

Cost of Product Sales

Cost  of  product  sales  is  comprised  of  (i)  costs  to  acquire  products  sold  to  customers,  (ii)  royalty,  license  payments  and  other
agreements granting the Company rights to sell related products, (iii) distribution costs incurred in the sale of products; (iv) the value of
any write-offs of obsolete or damaged inventory that cannot be sold, (v) minimum sale obligations and (vi) minimum purchase obligations.
The Company acquired the rights to sell certain of its commercial products through license and assignment agreements with the original
developers  or  other  parties  with  interests  in  these  products.  These  agreements  obligate  the  Company  to  make  payments  under  varying
payment structures based on its net revenue from related products.

Shipping, Handling, and Freight

The Company includes the cost of shipping, handling, and freight associated with product sales as part of cost of product sales.

Research and Development Costs

Research and development costs are expensed as incurred. These costs include, but are not limited to, employee‑related expenses,
including  salaries,  benefits  and  stock‑based  compensation  of  research  and  development  personnel;  expenses  incurred  under  agreements
with  contract  research  organizations  and  investigative  sites  that  conduct  clinical  trials  and  preclinical  studies;  the  cost  of  acquiring,
developing and manufacturing clinical trial materials; other supplies; facilities, depreciation and other expenses, such as direct and allocated
expenses  for  rent,  utilities  and  insurance;  and  costs  associated  with  preclinical  activities  and  regulatory  operations,  pharmacovigilance,
quality and travel.

Costs  for  certain  development  activities,  such  as  clinical  trials,  are  recognized  based  on  an  evaluation  of  the  progress  to
completion of specific tasks using data such as patient enrollment, clinical site activations, or information provided to the Company by its
vendors, such as clinical research organizations, with respect to their actual costs incurred. Payments for these activities are based on the
terms of the individual arrangements, which may differ from the pattern of costs incurred, and are reflected in the financial statements as
prepaid or accrued research and development expense, as the case may be.

Clinical Trial Expense Accruals

As  part  of  the  process  of  preparing  its  financial  statements,  the  Company  is  required  to  estimate  its  expenses  resulting  from  its
obligations under contracts with vendors, clinical research organizations and consultants and under clinical site agreements in connection
with conducting clinical trials. The financial terms of these contracts are subject to negotiations, which vary from contract to contract and
may  result  in  payment  flows  that  do  not  match  the  periods  over  which  materials  or  services  are  provided  under  such  contracts.  The
Company’s objective is to reflect the appropriate trial expenses in its financial statements by matching those expenses with the period in
which services are performed and efforts are expended. The Company accounts for these expenses according to the progress of the trial as
measured by subject progression and the timing of various aspects of the trial. The Company determines accrual estimates by taking into
account  discussion  with  applicable  personnel  and  outside  service  providers  as  to  the  progress  or  state  of  consummation  of  trials,  or  the
services completed. During the course of a clinical trial, the Company adjusts its clinical expense recognition if actual results differ from its
estimates.  The  Company  makes  estimates  of  its  accrued  expenses  as  of  each  balance  sheet  date  based  on  the  facts  and  circumstances
known to it at that time. The Company’s clinical trial accruals are dependent upon the timely and accurate reporting of contract research
organizations and other third‑party vendors. Although the Company does not expect its estimates to be materially different from amounts
actually  incurred,  its  understanding  of  the  status  and  timing  of  services  performed  relative  to  the  actual  status  and  timing  of  services
performed might vary and might result in it reporting amounts that are too high or too low for any particular period.

Acquired In-Process Research and Development Expenses

Acquired in-process research and development ("IPR&D") expense includes the initial costs of IPR&D projects, acquired directly

in a transaction other than a business combination, that do not have an alternative future use.

Amortization Expense

Amortization  expense  includes  the  amortization  of  the  Company's  acquired  intangible  assets. There  is  no  amortization  expense
included in cost of product sales or sales and marketing expense as all amortization expense is included within its own standalone line in
operating expenses in the Company's consolidated statements of operations.

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Estimated Fair Value and Change in Fair Value of Contingent Consideration

The  Company's  business  acquisitions  of  Avadel's  pediatric  products  and  TRx  involve  the  potential  for  future  payment  of
consideration  that  is  contingent  upon  the  achievement  of  operation  and  commercial  milestones  and  royalty  payments  on  future  product
sales. The fair value of contingent consideration was determined at the acquisition date utilizing unobservable inputs such as the estimated
amount and timing of projected cash flows, the probability of success (achievement of the contingent event) and the risk-adjusted discount
rate used to present value the probability-weighted cash flows. Subsequent to the acquisition date, at each reporting period, the contingent
consideration liability is remeasured at the current fair value with changes recorded in the consolidated statement of operations.

There is no change in fair value of contingent consideration included in cost of product sales or research and development costs as
the  change  in  fair  value  of  contingent  consideration  is  included  within  its  own  standalone  line  in  operating  expenses  in  the  Company's
consolidated statements of operations.

Stock‑Based Compensation

The  Company  applies  the  provisions  of  ASC  718,  Compensation—Stock  Compensation  (“ASC  718”),  which  requires  the
measurement and recognition of compensation expense for all stock‑based awards made to employees, including employee stock options,
in the statements of operations.

For stock options issued to employees and members of the board of directors for their services, the Company estimates the grant
date fair value of each option using the Black‑Scholes option pricing model. The use of the Black‑Scholes option pricing model requires
management to make assumptions with respect to the expected term of the option, the expected volatility of the common stock consistent
with  the  expected  life  of  the  option,  risk‑free  interest  rates  and  expected  dividend  yields  of  the  common  stock.  For  awards  subject  to
service‑based  vesting  conditions,  including  those  with  a  graded  vesting  schedule,  the  Company  recognizes  stock‑based  compensation
expense equal to the grant date fair value of stock options on a straight‑line basis over the requisite service period, which is generally the
vesting term. Forfeitures are recorded as they are incurred as opposed to being estimated at the time of grant and revised.

For stock option grants with market-based conditions, compensation expense is recognized ratably over the attribution period. The
Company  estimates  the  fair  value  of  the  market-based  stock  option  grants  using  a  Monte-Carlo  simulation.  The  Company  generally
estimates fair value using assumptions, including the risk-free interest rate, the expected volatility of a peer group of similar companies, the
expected  term  of  the  awards  and  the  expected  dividend  yield.  The  expected  term  for  market-based  stock  option  awards  is  based  on  the
expected  term  calculated  using  a  Monte-Carlo  simulation.  These  estimates  involve  inherent  uncertainties  and  the  application  of
management’s judgment. If factors change and different assumptions are used, our stock-based compensation expense could be materially
different in the future.

Income Taxes

The Company accounts for income taxes under the asset and liability method in accordance with ASC 740, Income Taxes (“ASC
740”).  Deferred  tax  assets  and  liabilities  are  recognized  for  the  future  tax  consequences  attributable  to  differences  between  the  financial
statement carrying amounts of existing assets and liabilities and their respective tax bases using enacted tax rates in effect for the year in
which the differences are expected to affect taxable income. Deferred tax assets primarily include net operating loss ("NOL") and tax credit
carryforwards, accrued expenses not currently deductible and the cumulative temporary differences related to certain research and patent
costs. Certain tax attributes, including NOLs and research and development credit carryforwards, may be subject to an annual limitation
under Sections 382 and 383 of the Internal Revenue Code (the "IRC"). See Note 15 for further information. The portion of any deferred tax
asset for which it is more likely than not that a tax benefit will not be realized must then be offset by recording a valuation allowance. The
Company recognizes the tax benefit from an uncertain tax position only if it is more likely than not to be sustained upon examination based
on the technical merits of the position. The amount for which an exposure exists is measured as the largest amount of benefit determined on
a cumulative probability basis that the Company believes is more likely than not to be realized upon ultimate settlement of the position. The
Company’s  policy  is  to  record  interest  and  penalties  on  uncertain  tax  positions  as  income  tax  expense. As  of  December  31,  2018,  the
Company did not believe any material uncertain tax positions were present.

On December 22, 2017, the “Tax Cuts and Jobs Act” ("TCJA" or "the Act") was enacted, that significantly reforms the IRC. The
TCJA,  among  other  things,  includes  changes  to  U.S.  federal  tax  rates,  imposes  significant  additional  limitations  on  the  deductibility  of
interest and NOL carryforwards, allows for the expensing of capital expenditures, and puts into effect the migration from a “worldwide”
system of taxation to a territorial system. See Note 15 below for further discussion related to the tax impact to the Company.

Recently Adopted Accounting Pronouncements

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Adoption of ASC 606

In May 2014, the FASB issued ASU 2014-09,  Revenue from Contracts with Customers (Topic 606) ("ASU 2014-09"). Topic 606,
along  with  amendments  issued  in  2015,  2016  and  2017,  supersedes  the  revenue  recognition  requirements  in  Topic  605, Revenue
Recognition, including most industry-specific revenue recognition guidance throughout the Industry Topics of the Accounting Standards
Codification. ASU  2014-09  provides  a  comprehensive  new  revenue  recognition  model  that  requires  a  company  to  recognize  revenue  to
depict the transfer of goods or services to a customer in an amount that reflects the consideration it expects to receive in exchange for those
goods or services. On January 1, 2018, the Company adopted the new revenue recognition standard for all contracts not completed as of
the  adoption  date  using  the  modified  retrospective  method.  The  implementation  of  the  new  revenue  recognition  standard  did  not  have  a
material quantitative impact on the Company’s consolidated financial statements as the timing of revenue recognition for product sales did
not  significantly  change.  In  addition,  the  Company  did  not  have  a  material  cumulative  effect  adjustment  to  accumulated  deficit  upon
adoption of the new revenue recognition standard on January 1, 2018. The information presented for the periods prior to January 1, 2018
has not been restated and is reported under Topic 605.

The  Company  recognizes  revenue  when  its  performance  obligations  with  its  customers  have  been  satisfied. At  contract  inception,  the
Company  determines  if  a  contract  is  within  the  scope  of  Topic  606  and  then  evaluates  the  contract  using  the  following  five  steps:  (1)
identify  the  contract  with  the  customer;  (2)  identify  the  performance  obligations;  (3)  determine  the  transaction  price;  (4)  allocate  the
transaction price to the performance obligations; and (5) recognize revenue when (or as) the entity satisfies a performance obligation.

Other Adopted Accounting Pronouncements

In January 2017, the FASB issued ASU No. 2017-01,  Business Combinations (Topic 805): Clarifying the Definition of a Business
("ASU  2017-01").  The  standard  provides  guidance  to  assist  entities  with  evaluating  whether  transactions  should  be  accounted  for  as
acquisitions  (or  disposals)  of  assets  or  businesses.  If  substantially  all  of  the  fair  value  of  the  gross  assets  acquired  (or  disposed  of)  is
concentrated in a single asset or a group of similar assets, the assets acquired (or disposed of) are not considered a business. ASU 2017-01
is  effective  for  fiscal  periods  beginning  after  December  15,  2017  (including  interim  periods  within  those  periods)  with  early  adoption
permitted. The Company adopted this standard on January 1, 2018.

In  January  2017,  the  FASB  issued ASU  No.  2017-04  “ Intangibles-Goodwill  and  Other  (Topic  350) :  Simplifying  the  Test  for
Goodwill Impairment”  ("ASU  2017-04"). ASU  2017-04  eliminates  step  two  of  the  goodwill  impairment  test  and  specifies  that  goodwill
impairment  should  be  measured  by  comparing  the  fair  value  of  a  reporting  unit  with  its  carrying  amount. ASU  2017-04  is  effective  for
annual or interim goodwill impairment tests performed in fiscal years beginning after December 15, 2019 and early adoption is permitted.
The Company early adopted this standard on January 1, 2018. The standard was applied prospectively and the adoption of this standard did
not have an impact on the Company's financial statements.

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In  May  2017,  the  FASB  issued  ASU  No.  2017-09,  Compensation-Stock  Compensation  (Topic  718)  -  Scope  of  Modification
Accounting  (“ASU  2017-09”)  to  clarify  when  to  account  for  a  change  to  the  terms  or  conditions  of  a  stock-based  payment  award  as  a
modification.  Under  the  new  guidance,  modification  accounting  is  required  only  if  the  fair  value,  the  vesting  conditions,  or  the
classification  of  the  award  (as  equity  or  liability)  changes  as  a  result  of  the  change  in  terms  or  conditions.  The  guidance  is  effective
prospectively  for  all  companies  for  annual  periods  and  interim  periods  within  those  annual  periods,  beginning  on  or  after  December  15,
2017. The adoption of this standard on January 1, 2018 did not have a significant impact on the Company’s financial statements.

In November 2016, the FASB issued ASU No. 2016-18,  Restricted Cash ("ASU 2016-18"). The guidance is intended to address
the diversity that currently exists in the classification and presentation of changes in restricted cash on the statement of cash flows. The new
standard requires that entities show the changes in the total of cash and cash equivalents, restricted cash and restricted cash equivalents on
the  statement  of  cash  flows  and  no  longer  present  transfers  between  cash  and  cash  equivalents,  restricted  cash  and  restricted  cash
equivalents on the statement of cash flows. The new standard is effective for fiscal years beginning after December 15, 2017, including
interim  periods  within  those  fiscal  years.  The  Company  adopted  this  standard  on  January  1,  2018. Upon  adoption  of ASU  2016-18,  the
Company applied the retrospective transition method for each period presented and included $0.1 million of restricted cash in the beginning
period cash, cash equivalents and restricted cash balance as of January 1, 2017.

In October 2016, the FA SB issued ASU No. 2016-16, “ Income  Taxes  (Topic  740),  Intra-Entity  Transfers  of  Assets  Other  Than
Inventory”  ("ASU  2016-16"),  which  requires  companies  to recognize the income tax consequences  of  an  intra-entity  transfer  of  an  asset
other  than  inventory  when  the  transfer  occurs.  ASU  2016-16  is  effective  for  annual  reporting  periods,  and  interim  periods  therein,
beginning after December 15, 2017. The adoption of this standard on January 1, 2018 did not have a significant impact on the Company’s
financial statements.

In August 2016, the FASB issued ASU No. 2016-15  Statement of Cash Flows, Classification of Certain Cash Receipts and Cash
Payments  ("ASU  2016-15"),  which  reduces  existing  diversity  in  the  classification  of  certain  cash  receipts  and  cash  payments  on  the
statements of cash flows. ASU 2016-15 is effective for fiscal years beginning after December 15, 2017, and for interim periods within those
fiscal years. The adoption of this standard on January 1, 2018 did not have a significant impact on the Company’s financial statements.

Recent Accounting Pronouncements

In  February  2016,  the  FASB  issued ASU  No.  2016-02,  Leases  (Topic  842)  ("ASU  2016-02").  This  guidance  revises  existing
practice related to accounting for leases under ASC No. 840, Leases (“ASC 840”) for both lessees and lessors. The new guidance in ASU
2016-02 requires lessees to recognize a right-of-use asset and a lease liability for nearly all leases (other than leases that meet the definition
of a short-term lease). The lease liability will be equal to the present value of lease payments and the right-of-use asset will be based on the
lease liability, subject to adjustment such as for initial direct costs. For income statement purposes, the new standard retains a dual model
similar to ASC 840, requiring leases to be classified as either operating leases or capital leases. For lessees, operating leases will result in
straight-line  expense  (similar  to  current  accounting  by  lessees  for  operating  leases  under ASC  840)  while  capital  leases  will  result  in  a
front-loaded expense pattern (similar to current accounting by lessees for capital leases under ASC 840). The new standard is effective for
the  Company  beginning  January  1,  2019. In  July  2018,  the  FASB  issued  both  codification  improvements,  which  clarify  how  to  apply
certain  aspects  of  the  standard,  and  an  update  to  the  transition  methods  allowable.  Companies  can  either  adopt  the  new  standard  at  the
earliest period presented using a modified retrospective approach or continue to apply the guidance under the current lease standard in the
comparative  periods  presented.  Companies  that  elect  this  option  would  record  a  cumulative-effect  adjustment  to  the  opening  balance  of
retained  earnings  on  the  date  of  adoption,  if  necessary.  The  Company  expects  to  apply  the  new  guidance  at  the  effective  date,  without
adjusting the comparative periods. The Company anticipates that ASU 2016-02 will have an impact to the consolidated balance sheet, as
the  Company  will  record  an  asset  and  a  liability  in  connection  with  the  leased  office  space. The  Company  will  elect  the  package  of
practical expedients permitted under the transition guidance within the new standard, which among other things, allows the Company to
carryforward the historical lease classification. The Company is not electing the hindsight practical expedient.

The Company has performed a preliminary assessment on the impact to the consolidated balance sheet and preliminarily expects
that  we  will  record  a  right-of-use  liability  and  corresponding  of  approximately $1 million  and  a  corresponding  right-of-use  asset  (with
certain adjustments for the accrued rent and unamortized lease incentive balance at January 1, 2019) related to the leased office space. This
expectation is subject to change as management refines the inputs utilized in the calculation. The Company does not expect an impact to the
statement of operations or liquidity. The Company is in the process of identifying its other lease agreements that will be impacted by the
new standard to arrive at the overall impact to the consolidated financial statements, however anticipates the overall balance sheet impact
to be less than 5% of the total liabilities balance as of December 31, 2018.

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3. Net (Loss) Income Per Share of Common Stock, Basic and Diluted

The Company computes earnings per share ("EPS") using the two-class method. The two-class method of computing EPS is an
earnings  allocation  formula  that  determines  EPS  for  common  stock  and  any  participating  securities  according  to  dividends  declared  and
participation  rights  in  undistributed  earnings. Under  the  two-class  method,  EPS  for  the  common  stock,  preferred  stock  and  participating
warrants  are  computed  by  dividing  the  sum  of  distributed  earnings  to  common  shareholders  and  undistributed  earnings  allocated  to
common shareholders by the weighted average number of shares of common stock and participating warrants outstanding for the period. In
applying the two-class method, undistributed earnings are allocated to common stock, preferred stock and participating warrants based on
the weighted average shares outstanding during the period. In periods of net loss, losses are allocated to the participating security only if
the security has not only the right to participate in earnings, but also a contractual obligation to share in the Company's losses.

Diluted net (loss) income per share includes the potential dilutive effect of common stock equivalents as if such securities were
converted or exercised during the period, when the effect is dilutive. Common stock equivalents include: (i) outstanding stock options and
restricted  stock  awards  which  are  included  under  the  "treasury  stock  method"  when  dilutive,  (ii)  common  stock  to  be  issued  upon  the
assumed conversion of the Company's unit purchase option shares, which are included under the "if-converted method" when dilutive; (iii)
prior  to  issuance,  the  contingently  issuable  shares  in  the  TRx  acquisition  if  contingencies  would  have  been  satisfied  if  the  end  of  the
contingency period were as of the balance sheet date under the "if converted method" when dilutive; and (iv) common stock to be issued
upon the exercise of outstanding warrants which are included under the "treasury stock method" when dilutive. Because the impact of these
items  is  generally  anti-dilutive  during  periods  of  net  loss,  there  is  no  difference  between  basic  and  diluted  loss  per  common  share  for
periods  with  net  losses.  In  addition,  as  stated  above,  net  losses  are  not  allocated  to  the  participating  securities  unless  the  participating
security has a contractual obligation to share in both earnings and losses of the Company.

The following table sets forth the computation of basic and diluted net loss per share of common stock for the years ended

December 31, 2018 and 2017, which includes both classes of participating securities: 

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Net (loss) income per share, basic and diluted calculation:
Basic (loss) income per share
Net (loss) income
Deemed distribution to shareholder
Undistributable (loss) earnings allocable to common shares
Undistributable (loss) earnings allocable to participating warrants

Weighted average shares, basic

Common stock
Participating warrants

Basic (loss) income per share:

Common stock
Participating warrants

Diluted (loss) income per share:
Net (loss) income attributable to common shares
Net (loss) income reallocated
Undistributed (loss) earnings allocable to common shares

Weighted average number of shares attributable to common shareholders - basic
Effect of dilutive securities:

Stock options
Contingently issuable shares
Potentially dilutive shares

Weighted average number of shares - diluted

Year ended December 31,

2018

2017

  $

  $
  $

(40,052,810)   $
1,657,383  
(41,710,193)   $
—   $

11,869,823
—
7,772,084
4,097,739

34,773,613  
—  
34,773,613  

18,410,005
9,706,458
28,116,463

  $
  $

(1.20)   $
—   $

0.42
0.42

  $

(41,710,193)   $

—  

  $

(41,710,193)   $

7,772,084
49,642
7,821,726

34,773,613  

18,410,005

—  
—  
—  
34,773,613  

61,510
283,284
344,794
18,754,799

Diluted (loss) income per share

  $

(1.20)   $

0.42

On December 27, 2018, the Company entered into a series of transactions as part of a private placement with Armistice in order to
generate cash to continue to develop our pipeline assets and for general corporate purposes. The transactions are considered one transaction
for  accounting  purposes. As  part  of  the  transaction,  the  Company  exchanged  common  stock  warrants  issued  as  a  part  of  the Armistice
private placement in 2017 for the purchase up to 14,285,714 shares of the Company’s common stock at an exercise price of $0.40 per share
(the "original warrants") for like-kind warrants to purchase up to 2,857,143 shares of the Company's newly designated Series B Convertible
Preferred Stock (the "Series B Convertible Preferred Stock" or "convertible preferred stock") with an exercise price of $2.00 per share (the
"exchanged  warrants"). The convertible preferred stock has the same rights and preferences as common stock other than it is non-voting
and  converts  to  shares  of  common  stock  on  a  1  for 5  ratio. Armistice  immediately  exercised  the  exchanged  warrants  and  acquired  an
aggregate  of 2,857,143  shares  of  the  Series  B  Convertible  Preferred  Stock  to  generate  net  proceeds  of  approximately  $5.7 million.  The
convertible preferred stock is considered a separate class of stock for EPS purposes, however basic and diluted EPS is not provided for the
preferred stock for the year ended December 31, 2018 because the shares were only outstanding for five days for the year. Therefore, EPS
for the preferred stock is immaterial for the year ended December 31, 2018, however will be disclosed going forward.

In order to provide Armistice an incentive to exercise the exchanged warrants, the Company also entered into a securities purchase
agreement with Armistice pursuant to which the Company issued warrants for  4,000,000 shares of common stock of the Company with a
term  of 5.5  years  and  an  exercise  price  of $12.50  per  share  (the  "incentive  warrants"). For  accounting  purposes  the  fair  value  of  the
incentive  warrants  was  considered  a  deemed  distribution  to  Armistice  of $1.7  million.  The  deemed  distribution  is  calculated  as  the
difference  between  the  fair  value  of  the  incentive  warrants  on  the  date  of  the  transaction  of $2.2 million  and  the  value  that Armistice
forwent  by  exchanging  the  original  warrants  of $0.5 million. The  fair  value  of  the  incentive  warrant  is  estimated  using  a  Black-Scholes
option-pricing model. The significant assumptions used in the model for valuing the incentive warrant on December 27, 2018 include:

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(i) volatility of 55%, (ii) risk-free interest rate of 2.62%, (iii) unit strike price of $12.50, (iv) fair value of underlying equity of $3.02, and
(v) expected life of 5.5 years.

The  net  loss  of $40.1 million for the year ended December 31, 2018 is increased by the deemed distribution of $1.7 million  to
arrive at the net loss attributable to common shareholders of $41.7 million. While the incentive warrants do have the rights to participate in
undistributed  earnings,  the  incentive  warrants  issued  do  not  share  in  net  losses  of  the  Company. As  such,  the  incentive  warrants  are
excluded from the weighted average shares and warrants outstanding during periods of net loss. For the 2017 EPS calculation, the shares of
unexercised original warrants issued in the Armistice private placement transaction in 2017 are considered participating securities because
these warrants contain a non-forfeitable right to dividends irrespective of whether the warrants are ultimately exercised.

The following outstanding securities at December 31, 2018 and 2017 have been excluded from the computation of diluted

weighted shares outstanding, as they could have been anti-dilutive: 

Stock options
Warrants on common stock
Restricted Stock Awards
Underwriters' unit purchase option

4. Acquisition

Ichorion Asset Acquisition

December 31,

2018
4,246,597  
4,024,708  
445,000  
40,000  

2017
2,812,006
4,661,145
—
40,000

On September 24, 2018, the Company entered into, and subsequently consummated the transactions contemplated by, an

agreement and plan of merger by and among the Company and Ichorion Therapeutics, Inc., a Delaware corporation (the “Ichorion Asset
Acquisition”), with Ichorion surviving as a wholly owned subsidiary of the Company.  The consideration for the Ichorion Asset
Acquisition consisted of approximately 5.8 million shares of the Company’s common stock, par value $0.001 per share, as adjusted for
Estimated Working Capital as defined in the Merger Agreement.  The shares are subject to a lockup date through December 31, 2019,
which restricts the resale of the common stock issued as part of the acquisition until the lockup period is complete. Consideration for the
Ichorion Asset Acquisition includes certain development milestones worth up to an additional $15 million, payable either in shares of the
Company's common stock or in cash, at the election of the Company.

The fair value of the common stock shares transferred at closing was approximately  $20 million using the Company's stock price

close on September 24, 2018 and offset by an estimated discount for lack of marketability calculated using guideline public company
volatility for comparable companies. The assets acquired consisted primarily of $18.7 million of IPR&D, $1.6 million of cash and $0.2
million assembled workforce. The Company recorded this transaction as an asset purchase as opposed to a business combination as
management concluded that substantially all of the value received was related to one group of similar identifiable assets which was the
IPR&D for the three preclinical therapies for inherited metabolic disorders known as CDGs (CERC-801, CERC-802 and CERC-803). The
Company has considered these assets similar due to similarities in the risks for development, compound type, stage of development,
regulatory pathway, patient population and economics of commercialization.  The fair value of the IPR&D was immediately recognized as
Acquired In-Process Research and Development expense as the IPR&D asset has no other alternate use due to the stage of development.
The acquired IPR&D expense was not tax deductible for the year ended December 31, 2018.  The $0.2 million of transaction costs
incurred were recorded to acquire IPR&D expense. The assembled workforce asset recorded to intangible assets will be amortized over an
estimated useful life of two years.

The contingent consideration is related to  three future development milestones and if met the Company may be required to pay out

an additional $15 million. The first milestone is contingent on the first product being approved for marketing by the FDA on or prior to
December 31, 2021. If this milestone is met, the Company is required to make a milestone payment of $6 million, payable either in shares
of the Company's common stock or in cash, at the election of the Company. The second milestone is contingent on the second product
being approved for marketing by the FDA on or prior to December 31, 2021. If this milestone is met, the Company is required to make a
milestone payment of $5 million, payable in either shares of the Company's common stock or cash, at the election of the Company. The
third milestone is contingent on a protide molecule being approved by the FDA on or prior to December 31, 2023. If this milestone is met,
the Company is required to make a milestone payment of $4 million, payable in either shares of the Company's common stock or cash, at
the election of the Company.

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The contingent consideration related to the development milestones will be recognized if and when such milestones are probable

and can be reasonably estimated. As of December 31, 2018, no contingent consideration related to the development milestone has been
recognized. The Company will continue to monitor the development milestones at each reporting period.

Acquisitions of Businesses

Avadel Pediatric Products Acquisition    

On February 16, 2018, the Company entered into an Asset Purchase Agreement (the “Purchase Agreement”) with Avadel US

Holdings, Inc., Avadel Pharmaceuticals (USA), Inc., Avadel Pediatrics, Inc., Avadel Therapeutics, LLC and Avadel Pharmaceuticals PLC
(collectively, the “Sellers”) to purchase and acquire all rights to the Sellers’ pediatric products. Total consideration transferred to the Sellers
consisted of a cash payment of one dollar. In addition, the Company assumed existing seller debt due in January 2021 with a fair value
of $15.1 million and contingent consideration relating to royalty obligations through February 2026 with a fair value at acquisition date of
approximately $7.9 million. As a result of the Avadel pediatric products acquisition, the Company has currently recorded goodwill of  $3.8
million, which is deductible over 15 years for income tax purposes.

The transaction was accounted for as a business combination under the acquisition method of accounting. Accordingly, the
tangible and identifiable intangible assets acquired and liabilities assumed were recorded at fair value as of the date of acquisition, with the
remaining purchase price recorded as goodwill. The goodwill recognized is attributable primarily to strategic opportunities related to an
expanded commercial footprint and diversified pediatric product portfolio that is expected to provide revenue and cost synergies.
Transaction costs of $0.1 million were included as general and administrative expense in the consolidated statements of operations for
the year ended December 31, 2018.

During the second quarter of 2018, the Company identified and recorded measurement period adjustments to the preliminary
purchase price allocation. These adjustments are reflected in the tables below. The measurement period adjustments were the result of
additional analysis performed and information identified during the second quarter of 2018 based on facts and circumstances that existed as
of the purchase date. There were no additional measurement adjustments recorded in 2018.

The following table summarizes the preliminary fair values of the assets acquired and liabilities assumed at the date of acquisition

and as adjusted for measurement period adjustments identified during the second quarter:    

Inventory
Prepaid assets
Intangible assets
Accrued expenses
Fair value of debt assumed
Fair value of contingent consideration
Total net liabilities assumed
Consideration exchanged
     Goodwill

At February 16,
2018 (preliminary)

Measurement Period
Adjustments

At February 16,
2018 (as adjusted)

  $

2,549,000 $

—
16,453,000
—

(15,272,303 )
(7,875,165 )
(4,145,468 )
241,000
4,386,468 $

  $

(1,831,000) $
570,000
1,838,000
(362,000 )
197,303
(44,835 )
367,468
(240,999 )
(608,467) $

718,000
570,000
18,291,000
(362,000)
(15,075,000)
(7,920,000)
(3,778,000)
1
3,778,001

Based on valuation estimates utilizing the estimated sales price of inventory less sales and marketing costs and an allowance for
profit, a step-up in the value of inventory of $0.3 million was recorded in the opening balance sheet, of which approximately $0.1 million
was charged to cost of goods sold during the post-acquisition period, February 16, 2018 through December 31, 2018.

The  purchase  price  allocation  related  to  the  acquisition  of  Avadel's  pediatric  products  has  been  finalized.  The  fair  values  of
intangible assets, including marketing rights, licenses and developed technology, were determined using variations of the income approach.
Varying discount rates were also applied to the projected net cash flows. The Company believes the assumptions are representative of those
a market participant would use in estimating fair value. The preliminary fair value of intangible assets both as of the date of acquisition and
as adjusted by measurement period adjustments identified during the second quarter includes the following:

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At February 16,
2018 (preliminary)

Measurement
Period
Adjustments

At February 16,
2018 (as
adjusted)

Acquired Product Marketing Rights - Karbinal
Acquired Product Marketing Rights - AcipHex
Acquired Product Marketing Rights - Cefaclor
Acquired Developed Technology - Flexichamber
Acquired IPR&D - LiquiTime formulations
     Total

  $

  $

6,221,000 $
2,520,000
6,291,000
1,131,000
290,000
16,453,000 $

(21,000) $
283,000
1,320,000
546,000
(290,000)
1,838,000 $

6,200,000
2,803,000
7,611,000
1,677,000
—

18,291,000  

Useful Life

10 years
10 years
7 years
10 years
Indefinite

TRx Acquisition    

On November 17, 2017, the Company entered into, and consummated the transactions contemplated by, an equity interest

purchase agreement (the “TRx Purchase Agreement”) by and among the Company, TRx, Fremantle Corporation and LRS International
LLC, the selling members of TRx (collectively, the “TRx Sellers”), which provided for the purchase of all of the equity and ownership
interests of TRx by the Company (the "TRx Acquisition"). The consideration for the TRx acquisition consists of $18.9 million in cash, as
adjusted for estimated working capital, estimated cash on hand, estimated indebtedness and estimated transaction expenses, as well as
7,534,884 shares of the Company’s common stock having an aggregate value on the closing date of  $8.5 million (the "Equity
Consideration") and certain potential contingent payments. Upon closing, the Company issued 5,184,920 shares of its common stock to the
TRx Sellers.  Pursuant to the TRx Purchase Agreement, the issuance of the remaining 2,349,968 shares were subject to the Company's
stockholder approval. In May 2018, stockholder approval was obtained and the remaining shares were issued to the TRx Sellers. The
contingent shares were initially recorded to contingently issuable shares, which is recorded within stockholder's equity and were reclassed
to common stock and additional paid in capital upon issuance, on the consolidating balance sheet date. As a result of the TRx Acquisition,
the Company has currently recorded goodwill of $12.6 million, of which $8.7 million was deductible for income taxes.

During the third quarter of 2018, the Company identified and recorded measurement period adjustments to our preliminary
purchase price allocation that was disclosed in prior periods. These adjustments are reflected in the tables below. If the measurement period
adjustments were reflected in the consolidated statement of operations for the year ended December 31, 2017 its impact would have been
immaterial. The measurement period adjustments were the result of an arbitration ruling discussed in further detail in Note 11, the facts and
circumstances of which existed as of the acquisition date.

The following table summarizes the preliminary acquisition-date fair value of the consideration transferred at the date of

acquisition both as disclosed in prior periods prior to the third quarter of 2018 and as adjusted for measurement period adjustments
identified during the third quarter of 2018:

Cash
Common stock (including contingently issuable
shares)
Contingent payments

Total consideration transferred

  $

At November 17,
2017 (preliminary)

Measurement Period
Adjustments

At November 17,
2017 (as adjusted)

  $

18,900,000 $

— $

18,900,000

8,514,419
2,576,633
29,991,052

—

(1,210,000 )
(1,210,000 )

8,514,419
1,366,633
28,781,052

The TRx Acquisition was accounted for as a business combination under the acquisition method of accounting. Accordingly, the
tangible and identifiable intangible assets acquired, and liabilities assumed, were recorded at fair value as of the date of acquisition, with
the remaining purchase price recorded as goodwill. The goodwill recognized is attributable primarily to strategic opportunities related to
leveraging TRx’s research and development, intellectual property, and processes.

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The following table summarizes the preliminary fair values of the assets acquired and liabilities assumed at the date of acquisition

both as disclosed in prior periods prior to the third quarter of 2018 and as adjusted for measurement period adjustments identified during the
third quarter of 2018:

Fair value of assets acquired:
Cash and cash equivalents
Accounts receivable, net
Inventory
Prepaid expenses and other current assets
Other receivables
Identifiable Intangible Assets:
Acquired product marketing rights - Metafolin
PAI sales and marketing agreement
Acquired product marketing rights - Millipred
Acquired product marketing rights - Ulesfia
Total assets acquired

Fair value of liabilities assumed:
Accounts payable
Accrued expenses and other current liabilities
Deferred tax liability

Total liabilities assumed
Total identifiable net assets
Fair value of consideration transferred
Goodwill

At November 17,
2017 (preliminary)

Measurement Period
Adjustments

At November 17,
2017 (as adjusted)

  $

11,068 $

2,872,545
495,777
134,281
—

10,465,000
2,334,000
4,714,000
555,000
21,581,671

192,706
4,850,422
839,773
5,882,901

15,698,770
29,991,052
14,292,282 $

  $

— $
—
—
—
2,764,515

1,522,000
219,000
342,000
(555,000 )
4,292,515

—
3,764,515
78,840
3,843,355

449,160
(1,210,000 )
(1,659,160) $

11,068
2,872,545
495,777
134,281
2,764,515
—
11,987,000
2,553,000
5,056,000
—
25,874,186

192,706
8,614,937
918,613
9,726,256

16,147,930
28,781,052
12,633,122

Based on valuation estimates utilizing the estimated selling price of inventory less sales and marketing costs and an allowance for
profit, a step-up in the value of inventory of $0.2 million was recorded in the opening balance sheet, of which approximately $0.2 million
was charged to cost of product sales during the year ended December 31, 2018.

The purchase price allocation related to the TRx Acquisition has been finalized. The fair values of intangible assets, including
marketing rights, licenses and developed technology, were determined using variations of the income approach, specifically the multi-
period excess earnings method. Varying discount rates were also applied to the projected net cash flows. The Company believes the
assumptions are representative of those a market participant would use in estimating fair value. The final fair value of intangible assets both
as disclosed in prior periods and as adjusted by measurement period adjustments identified during the third quarter of 2018 includes the
following:

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At November 17,
2017 (preliminary)

Measurement
Period
Adjustments

At November 17,
2017 (as
adjusted)

Acquired product marketing rights - Metafolin
PAI sales and marketing agreement
Acquired product marketing rights - Millipred
Acquired product marketing rights - Ulesfia

     Total

  $

  $

10,465,000 $
2,334,000
4,714,000
555,000
18,068,000 $

1,522,000 $
219,000
342,000
(555,000)
1,528,000 $

11,987,000
2,553,000
5,056,000

—  
19,596,000  

Useful Life

15 years
2 years
4 years

The  Company  received  written  notice  to  terminate  the  PAI  sales  and  marketing  agreement  in  the  second  quarter  of  2018.  As  a
result, the Company reassessed the fair value of the PAI sales and marketing agreement on that date (a level III non-recurring fair value
measurement)  and  concluded  due  to  the  absence  of  future  cash  flows  beyond  the  date  of  termination  that  the  fair  value  was $0.  An
impairment  charge  was  recognized  in  the  year  ended  December  31,  2018  in  the  amount  of $1.9 million,  representing  the  remaining  net
book value of the PAI sales and marketing agreement intangible asset.

Pro Forma Impact of Business Combinations

The following supplemental unaudited pro forma information presents Cerecor’s financial results as if the acquisitions of Avadel

Pediatric Products, which was completed on February 16, 2018, and of TRx, which was completed on November 17, 2017, had each
occurred on January 1, 2017:

Year Ended December 31,

2018
Pro forma

2017
Pro forma

Total revenues, net
Net loss

Basic and diluted net (loss) income
per share

$
$

$

20,031,801 $
(40,919,015) $

51,288,212
5,963,853

(1.18) $

0.21

The above unaudited pro forma information was determined based on the historical GAAP results of Cerecor, Avadel's pediatric
products  and  TRx. The  unaudited  pro  forma  consolidated  results  are  provided  for  informational  purposes  only  and  are  not  necessarily
indicative  of  what  Cerecor’s  consolidated  results  of  operations  would  have  been  had  the  acquisitions  of Avadel's  pediatric  products  and
TRx been completed on the dates indicated or what the consolidated results of operations will be in the future.

5. Fair Value Measurements

ASC No. 820, Fair Value Measurements and Disclosures  (“ASC 820”), defines fair value as the price that would be received to
sell  an  asset,  or  paid  to  transfer  a  liability,  in  the  principal  or  most  advantageous  market  in  an  orderly  transaction  between  market
participants on the measurement date. The fair value standard also establishes a three‑level hierarchy, which requires an entity to maximize
the use of observable inputs and minimize the use of unobservable inputs when measuring fair value. The valuation hierarchy is based upon
the transparency of inputs to the valuation of an asset or liability on the measurement date. The three levels are defined as follows:

• Level  1—inputs  to  the  valuation  methodology  are  quoted  prices  (unadjusted)  for  an  identical  asset  or  liability  in  an  active

market.

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• Level  2—inputs  to  the  valuation  methodology  include  quoted  prices  for  a  similar  asset  or  liability  in  an  active  market  or
model‑derived valuations in which all significant inputs are observable for substantially the full term of the asset or liability. 

• Level  3—inputs  to  the  valuation  methodology  are  unobservable  and  significant  to  the  fair  value  measurement  of  the  asset  or

liability.

The  following  table  presents,  for  each  of  the  fair  value  hierarchy  levels  required  under ASC  820,  the  Company’s  assets  and

liabilities that are measured at fair value on a recurring basis: 

Assets
Investments in money market funds*
Liabilities
Contingent consideration
Warrant liability**
Unit purchase option liability**

Assets
Investments in money market funds*
Liabilities
Contingent consideration
Warrant liability**
Unit purchase option liability**

December 31, 2018

Fair Value Measurements Using

  Quoted prices in
  active markets for  
identical assets

(Level 1)

Significant other

Significant

observable

inputs

(Level 2)

unobservable

inputs

(Level 3)

  $

  $
  $
  $

7,324,932   $

—   $
—   $
—   $

—   $

—   $
—   $
—   $

—

9,050,564
2,950
7,216

December 31, 2017

Fair Value Measurements Using

  Quoted prices in
  active markets for  
identical assets

(Level 1)

Significant other

Significant

observable

inputs

(Level 2)

unobservable

inputs

(Level 3)

  $

  $
  $
  $

471,183   $

—   $
—   $
—   $

—   $

—   $
—   $
—   $

—

2,576,633
8,185
26,991

*Investments in money market funds are reflected in cash and cash equivalents on the accompanying Balance Sheets.
**Warrant liability and unit purchase option liability are reflected in accrued expenses and other current liabilities on the accompanying
consolidated balance sheets.

At  December  31, 2018  and 2017,  the  Company’s  financial  instruments  included  cash  and  cash  equivalents,  restricted  cash,
accounts receivable, accounts payable, accrued expenses and other current liabilities, short term and long-term debt, warrant liability, the
underwriters' unit purchase option liability and contingent consideration. The carrying amounts reported in the accompanying consolidated
financial  statements  for  cash  and  cash  equivalents,  restricted  cash,  accounts  receivable,  accounts  payable,  accrued  expenses  and  other
current liabilities approximate their respective fair values because of the short-term nature of these accounts. The estimated fair value of
the Company’s long-term debt of $14.9 million as of December 31, 2018 was based on current interest rates for similar types of borrowings
and is in Level 2 of the fair value hierarchy.

Level 3 Valuation

The tables presented below are a summary of changes in the fair value of the Company’s Level 3 valuations for the warrant

liability, unit purchase option liability and contingent consideration for the years ended December 31, 2018 and 2017:

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Balance at December 31, 2017
Issuance of contingent consideration
Payment of contingent consideration
Purchase price allocation measurement period
adjustment of contingent consideration
Change in fair value
Balance at December 31, 2018

Balance at December 31, 2016
Issuance of contingent consideration
Change in fair value
Balance at December 31, 2017

  $

  $

  $

  $

Warrant

liability

  Unit purchase

Contingent

option liability  

consideration

8,185   $
—  
—  

—  
(5,235)  
2,950   $

26,991   $

—  
—  

2,576,633   $
7,920,000  
(294,435)  

Total
2,611,809
7,920,000
(294,435)

—  
(19,775)  

7,216   $

(1,210,000)  
58,366  
9,050,564   $

(1,210,000)
33,356
9,060,730

Warrant

liability

  Unit purchase
option liability

Contingent

consideration

5,501   $
—  
2,684  
8,185   $

51   $
—  
26,940  
26,991   $

—   $

2,576,633  
—  

2,576,633   $

Total

5,552
2,576,633
29,624
2,611,809

In 2014, the Company issued warrants to purchase 625,208 shares of convertible preferred stock. Upon the closing of our initial
public offering ("IPO") in October 2015 these warrants became warrants to purchase 22,328 shares of common stock, in accordance with
their terms. The warrants expire in October 2020. The warrants represent a freestanding financial instrument that is indexed to an
obligation, which the Company refers to as the warrant liability. The warrant liability is marked-to-market each reporting period with the
change in fair value recorded to other income, net in the accompanying statements of operations until the warrants are exercised, expire or
other facts and circumstances lead the warrant liability to be reclassified to stockholders’ equity. The fair value of the warrant liability is
estimated using a Black-Scholes option-pricing model. The significant assumptions used in preparing the option pricing model for valuing
the warrant liability as of December 31, 2018, include (i) volatility of 50%, (ii) risk-free interest rate of 2.51%, (iii) strike price of $8.40,
(iv) fair value of common stock of $3.23, and (v) expected life of 1.8 years.

The underwriters’ unit purchase option (the “UPO”) was issued to the underwriters of the Company's IPO in 2015 and provides
the  underwriters  the  option  to  purchase  up  to  a  total  of 40,000 units. The units underlying  the  UPO  will  be,  immediately  upon  exercise,
separated into shares of common stock, underwriters’ Class A warrants and underwriters’ Class B warrants (such warrants together referred
to  as  the  Underwriters’  Warrants).  The  Underwriters’  Warrants  are  warrants  to  purchase  shares  of  common  stock.  The  Class  B  warrants
expired in April 2017 and the Class A warrants expired in October 2018, while the UPO expires in October 2020. The Company classifies
the UPO as a liability as it is a freestanding marked-to-market derivative instrument that is precluded from being classified in stockholders’
equity. The  UPO  liability  is  marked-to-market  each  reporting  period  with  the  change  in  fair  value  recorded  to  other  income,  net  in  the
accompanying statements of operations until the UPO is exercised, expires or other facts and circumstances lead the UPO to be reclassified
to  stockholders’  equity.  The  fair  value  of  the  UPO  liability  is  estimated  using  a  Black-Scholes  option-pricing  model.  The  significant
assumptions used in preparing the simulation model for valuing the UPO as of December 31, 2018, include (i) volatility of 50%, (ii) risk-
free interest rate of 2.51%, (iii) unit strike price of $7.47, (iv) fair value of underlying equity of $3.23, and (v) expected life of 1.8 years.

The Company's business acquisitions of Avadel's pediatric products and TRx (see Note 4) involve the potential for future payment
of consideration that is contingent upon the achievement of operation and commercial milestones and royalty payments on future product
sales. The fair value of contingent consideration was determined at the acquisition date utilizing unobservable inputs such as the estimated
amount and timing of projected cash flows, the probability of success (achievement of the contingent event) and the risk-adjusted discount
rate used to present value the probability-weighted cash flows. Subsequent to the acquisition date, at each reporting period, the contingent
consideration liabilities are remeasured at the current fair value with changes recorded in the consolidated statement of operations.

As part of the acquisition of Avadel's pediatric products, the Company will pay a  15% annual royalty on net sales of the acquired
Avadel pediatric products through February 2026 up to an aggregate amount of  $12.5 million. The fair value of the future royalty is the
expected  future  value  of  the  contingent  payments  discounted  to  a  present  value. The  estimated  fair  value  of  the  royalty  payments  as  of
December 31, 2018 was $7.8 million. The significant assumptions used in estimating the fair value of the royalty payment as of December
31,  2018  include  (i)  the  expected  net  sales  of  the  acquired Avadel  pediatric  products  that  are  subject  to  the  15%  royalty  based  on  the
Company's net sales forecast, and (ii) the risk-adjusted discount rate of 8.1%, which is comprised of the risk-free interest rate of 2.6% and a
counterparty risk of 5.5%. The liability is reduced by periodic payments.

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The  consideration  for  the  TRx  acquisition  includes  certain  potential  contingent  payments. First,  pursuant  to  the  TRx  Purchase
Agreement, the Company is required to pay $3.0 million to the Sellers upon the gross profit related to TRx products achieving or exceeding
a gross profit of $12.6 million in 2018. The Company did not achieve this contingent event in 2018 and therefore no value was assigned to
the  contingent  payout  for  the  year  ended  December  31,  2018. Additionally,  the  Company  will  pay $2.0 million  upon  the  transfer  of  the
Ulesfia  NDA  to  the  Company  ("NDA  Transfer  Milestone").  Finally,  the  Company  will  pay $2.0 million  upon  FDA  approval  of  a  new
dosage of Ulesfia ("FDA Approval Milestone").  The main inputs utilized to determine the fair value of each milestone is the probability of
the milestone's success, the expected time to successfully reach the milestone, and the risk-adjusted discount rate. The estimated fair value
of the NDA Transfer Milestone as of December 31, 2018 was $0.9 million and the significant assumptions used in estimating the fair value
include (i) probability of milestone success of 45.0%, (ii) expected time to milestone of 0.5 years, and (iii) risk-adjusted discount rate of
7.9%,  which  is  comprised  of  the  risk-free  rate  of 2.4%  and  a  counterparty  risk  of 5.5%. The  estimated  fair  value  of  the  FDA Approval
Milestone as of December 31, 2018 was $0.4 million. The significant assumptions used in estimating the fair value of the FDA Approval
Milestone as of December 31, 2018 include (i) probability of milestone success at 22.5%, (ii) expected time to milestone of 1.5 years, and
(iii) risk-adjusted discount rate of 8.0%, which is comprised of the risk-free rate of 2.5% and a counterparty risk of 5.5%.

No other changes in valuation techniques or inputs occurred during the years ended December 31, 2018 and 2017. No transfers of
assets between Level 1 and Level 2 of the fair value measurement hierarchy occurred during the years ended December 31, 2018 and 2017.

6. Inventory

Inventory consists of finished goods stated at the lower of cost or net realizable value with cost determined on a first-in, first-out

basis. The Company reviews the composition of inventory at each reporting period in order to identify obsolete, slow-moving, quantities in
excess of expected demand, or otherwise non-saleable items. 

Inventory consisted of the following as of December 31, 2018 and 2017:

Raw materials
Finished goods
Inventory reserve

Inventory, net

December 31,

2018

  $

11,392   $

1,427,935  
(328,547)  
1,110,780   $

  $

2017

—
560,499
(178,346)
382,153

During the years ended December 31, 2018 and 2017, the Company recorded a related charge to cost of goods sold for obsolete

inventory of $150,201 and $178,346, respectively.

7. Property and Equipment

Property and equipment as of December 31, 2018 and 2017 consisted of the following:

Furniture and equipment
Computers and software
Leasehold improvements
Total property and equipment
Less accumulated depreciation

Property and equipment, net

December 31,

2018
133,229   $
122,065  
463,381  
718,675  
(132,163)  
586,512   $

2017

58,126
96,133
—
154,259
(109,647)
44,612

  $

  $

Depreciation expense was $22,515 and $21,956 for the years ended December 31, 2018 and December 31, 2017, respectively.

8. Goodwill

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The changes in the carrying amount of goodwill for the years ended December 31, 2018 and 2017 were as follows:

Balance at December 31, 2016

Goodwill from acquisition of TRx Pharmaceuticals

Balance at December 31, 2017

Goodwill from acquisition of Avadel's pediatric products
Goodwill purchase price allocation measurement period adjustment from
acquisition of TRx Pharmaceuticals

Balance at December 31, 2018

$

$

$

—  
14,292,282  
14,292,282  
3,778,001  

(1,659,160)  
16,411,123  

There were no accumulated impairment losses to goodwill at December 31, 2018 or December 31, 2017.

9. Intangible Assets

The changes in intangible assets for the years ended December 31, 2018 and 2017 were as follows:

Balance at December 31, 2016

Additions
Amortization

Balance at December 31, 2017

Additions
Purchase price allocation measurement period adjustments
Amortization
Impairment

Balance at December 31, 2018

$

$

$

—  
18,068,000  
(403,520)  
17,664,480  
18,441,000  
1,527,998  
(4,532,448)  
(1,861,562)  
31,239,468  

The following is a summary of intangible assets held by the Company at December 31, 2018 and December 31, 2017,

respectively:

December 31, 2018

Gross Carrying
Amount

Accumulated
Amortization

     Impairment Loss  

Net Carrying
Amount

Acquired Product Marketing Rights
Sales and Marketing Agreement
Acquired Developed Technology
Acquired Assembled Workforce
Total Intangible Assets

  $

  $

33,656,998   $
2,553,000  
1,677,000  
150,000  
38,036,998   $

(4,080,767)   $
(691,438)  
(145,013)  
(18,750)  
(4,935,968)   $

—   $

(1,861,562)  
—  
—  

(1,861,562)   $

29,576,231  
—  
1,531,987  
131,250  
31,239,468  

December 31, 2017

Gross Carrying
Amount

Accumulated
Amortization

Impairment Loss

Net Carrying
Amount

Acquired Product Marketing Rights
Sales and Marketing Agreement
Total Intangible Assets

  $

  $

15,734,000   $
2,334,000  
18,068,000   $

(257,645)   $
(145,875)  
(403,520)   $

—   $
—  
—   $

15,476,355  
2,188,125  
17,664,480  

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Weighted-
Average
Remaining
Life

(in years)
9.45
—
9.25
1.75
9.41

Weighted-
Average
Remaining
Life

(in years)
11.20
1.90
10.05

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
 
 
 
 
 
 
 
   
   
 
    
    
 
 
 
 
 
 
 
 
 
 
   
 
 
 
 
 
 
 
   
   
 
    
    
    
 
 
 
 
 
 
 
Table of Contents

The  Company  received  written  notice  to  terminate  the  PAI  sales  and  marketing  agreement  in  the  second  quarter  of  2018. As  a
result the Company reassessed the fair value of the PAI sales and marketing agreement on that date (a level III non-recurring fair value
measurement)  and  concluded  due  to  the  absence  of  future  cash  flows  beyond  the  date  of  termination  that  the  fair  value  was $0.   An
impairment  charge  was  recognized  in  the  year  ended  December  31,  2018  in  the  amount  of $1.9  million,  representing  the  remaining  net
book value of the PAI sales and marketing agreement intangible asset on the date of assessment.

Amortization of intangibles for the next five years and thereafter is expected to be as follows:

For the Years Ending December 31,

2019
2020
2021
2022
2023
Thereafter
Total future amortization expense

Estimated

Amortization
Expense

  $

  $

4,315,318
4,296,568
4,082,334
2,976,322
2,976,322
12,592,604
31,239,468

10. Accrued Expenses and Other Current Liabilities

Accrued expenses and other current liabilities as of December 31, 2018 and 2017 consisted of the following:

Sales returns
Medicaid rebates
Minimum sales commitments, royalties payable, and purchase obligations
Compensation and benefits
Research and development expenses
General and administrative
Sales and marketing
Other
Total accrued expenses and other current liabilities

11. Agreements

Lilly CERC-611 License

December 31,

2018
3,972,510   $
2,237,269  
9,662,901  
1,953,065  
278,132  
1,112,378  
235,721  
279,397  
19,731,373   $

  $

  $

2017
3,478,349
350,681
743,010
1,401,514
299,480
1,001,454
—
256,634
7,531,122

On September 22, 2016, the Company entered into an exclusive license agreement with Eli Lilly and Company (“Lilly”) pursuant
to which the Company received exclusive, global rights to develop and commercialize CERC-611, previously referred to as LY3130481, a
potent  and  selective  Transmembrane  AMPA  Receptor  Regulatory  Proteins  (“TARP”)  ã-8-dependent  á-amino-3-hydroxy-5-methyl-4-
isoxazolepropionic acid (“AMPA”) receptor antagonist. The terms of the license agreement provide for an upfront payment of $2.0 million,
of which $750,000 was due within 30 days of the effective date of the license agreement, and the remaining balance of  $1.25 million is due
after the first subject is dosed with CERC-611 in a multiple ascending dose study and is recorded as license obligations on the balance sheet
at December 31, 2018. Additional payments may be due upon achievement of development and commercialization milestones, including
the first commercial sale. Upon commercialization, the Company is obligated to pay Lilly milestone payments and a royalty on net sales.

Merck CERC-301 License

In 2013, the Company entered into an exclusive license agreement with Merck & Co., Inc. (“Merck”) pursuant to which Merck

granted the Company rights relating to certain small molecule compounds. In consideration of the license, the Company paid an initial

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payment  of $750,000, and upon achievement of acceptance by the United States Food and Drug Administration, or FDA, of Merck pre-
clinical data and FDA approval of a Phase 3 clinical trial the Company will pay an additional  $750,000. Additional payments may be due
upon achievement of development and regulatory milestones, including the first commercial sale. Upon commercialization, the Company is
obligated to pay Merck milestone payments and royalties on net sales.

Merck CERC-406

In  2013,  the  Company  entered  into  a  separate  exclusive  license  agreement  with  Merck  pursuant  to  which  Merck  granted  the
Company certain rights in small molecule compounds which are known to inhibit the activity of COMT. In consideration of the license, the
Company  made  a $200,000  upfront  payment  to  Merck.  Additional  payments  may  be  due  upon  the  achievement  of  development  and
regulatory milestones. Upon commercialization of a COMT product, the Company is required to pay Merck royalties on net sales.

Poly-Vi-Flor and Tri-Vi-Flor Related Contracts

Supply and License Agreement, effective December 1, 2014, by and between TRx and Merck & Co. (“Merck”)

On December 1, 2014 TRx entered into a Supply and License Agreement with Merck. The initial term of the agreement expires on
December 31, 2020, and the agreement will automatically continue for subsequent one-year terms thereafter until terminated in accordance
with  its  terms.  Pursuant  to  the  agreement,  Merck  agrees  to  supply  a  specific  compound  called  Metafolin®  to  TRx  for  use  in  dietary
supplements within a defined market, and TRx agrees to purchase 100% of its Metafolin requirements from Merck. Under the agreement,
TRx has an exclusive license under a number of U.S. and international patents, as well as related trade secrets, know-how and trademark
rights, to make and sell TRx products positioned in the pediatric market (i.e., targeted for children 0-3 years of age) in the U.S. Under the
agreement,  TRx  also  has  a  non-exclusive  license  under  the  same  intellectual  property  rights  to  make  and  sell  TRx  dietary  supplement
products within the U.S. outside of certain specified fields, including products containing Metafolin in combination with folic acid or any
other folate, products positioned for type II diabetes, pharmaceutical drugs, and medical, fortified, and special dietary foods. TRx must pay
Merck a royalty of two-percent (2%) of net sales from TRx products in the pediatric field that contain Metafolin. The royalty payment does
not apply to net sales of TRx products marketed as pre-or postnatal vitamins. The royalty payment will continue to apply throughout the
initial term and any automatic renewal periods. The minimum annual  order  quantity  for  the  compound  is 1kg.  Payments  of  royalties  are
made by TRx within 45 days following the end of each calendar quarter.

Settlement and License Agreement, dated February 28, 2011, by and between TRx and Mead Johnson and Company LLC, as amended

TRx  entered  into  a  Settlement  and  License Agreement  with  Mead  Johnson  and  Company  LLC,  and  the  parties  subsequently
entered  into  an  amendment  to  such  agreement  on  October  6,  2011.  Pursuant  to  the  agreement,  Mead  Johnson  granted  TRx  an  exclusive
license to the “Poly-Vi-Flor” and “Tri-Vi-Flor” trademarks and agreed not to oppose TRx’s seeking the marks Poly-Vi-Flor and Tri-Vi-Flor
in the United States and in any other countries where Mead Johnson does not have an active registration for such marks. As consideration
for such licenses, TRx agreed to pay a royalty to Mead Johnson in the amount  of 10% of net revenues received by TRx with respect to
products sold under the Poly-Vi-Flor and Tri-Vi-Flor trademarks during the term of the agreement. The term of the agreement  is indefinite
and will continue unless terminated pursuant to the provisions of the agreement. Payments are made by TRx in arrears on a quarterly basis
within 45 days after the end of a given calendar quarter.

Redemption Agreement with Additional Poly-Vi-Flor Royalty Obligation

TRx  and  the  Selling  Members  entered  into  an  Agreement  to  Redeem  Membership  Interest  on  May  31,  2011  with  a  former
Member, Presmar Associates, Inc. Pursuant to the agreement, TRx and the Selling Members agreed to pay to Presmar Associates a royalty
payment of 5% of gross sales for Poly-Vi-Flor branded or authorized generic product and, upon the sale of the Poly-Vi-Flor trademark to a
third party, to pay to Presmar Associates 5% of the cash proceeds from such sale transaction. Any future sale of the Poly-Vi-Flor trademark
to  a  third  party  would  require  that 5%  of  the  sale  proceeds  be  paid  to  Presmar Associates.  Payments  are  made  by  TRx  in  arrears  on  a
quarterly basis within 45 days after the end of a given calendar quarter.

Millipred Related Contracts

License and Supply Agreement between TRx and Watson Laboratories, Inc.

TRx entered into a License and Supply Agreement with Watson Laboratories, Inc. on May 19, 2008, and the parties subsequently
entered into amendments of the agreement on July 19, 2013 and April 1, 2016. Pursuant to the most recent amendment, the term of the
agreement  was  extended  for  an  additional five-year  period  expiring  on April  1,  2021.  However,  TRx  has  the  option  to  terminate  the
agreement  following  the  first  commercial  sale  of  a  generic  product  which  occurred  in  April  of  2017.  If  neither  party  terminates  the
agreement prior to April 1, 2021, then the agreement will automatically renew for successive  one-year  periods. The  amended  agreement
provides that the company make license payments of $75,000 in February and August of each year through April 2021.

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Ulesfia Related Contracts

First Amended and Restated Exclusive Ulesfia Distribution Agreement, dated December 18, 2015, by and between Zylera and Lachlan
Pharmaceuticals (“Lachlan”)

In November 2017, the Company acquired TRx and its wholly-owned subsidiaries, including Zylera. The previous owners of TRx
beneficially  own  more  than 10%  of  our  outstanding  common  stock. Zylera, which is our wholly owned subsidiary, entered into the First
Amended and Restated Distribution Agreement with  Lachlan, effective December 18, 2015. Pursuant to the Lachlan Agreement, Lachlan
named Zylera as its exclusive distributor of Ulesfia in the United States and agreed to supply Ulesfia to Zylera exclusively for marketing
and sale in the United States.

Zylera is obligated to purchase a minimum of 20,000 units per year, or approximately $1.2 million worth of product, from
Lachlan, subject to certain termination rights. Zylera must pay Lachlan $58.84 per unit and handling fees that are equal to $3.66 per unit of
fully packaged Ulesfia in 2018, and escalate at a rate of 10% annually, as well as reimburse Lachlan for all product liability insurance fees
incurred by Lachlan. The Lachlan Agreement also requires that Zylera make certain cumulative net sales milestone payments and royalty
payments to Lachlan with a $3 million annual minimum payment unless and until there has been a “Market Change” involving a new
successful competitive product. Lachlan is obligated to pay identical amounts to an unrelated third party from which it obtained rights to
Ulesfia, with the payments ultimately flowing to Summers Laboratories, Inc. (“Summers Labs”). Because of the dispute described below,
the Company has not made any payments to Lachlan under the Lachlan Agreement subsequent to the acquisition date.

On December 10, 2016, Zylera informed Lachlan that a Market Change had occurred due to the introduction of Arbor

Pharmaceuticals' lice product, Sklice®.  On June 5, 2017, Lachlan and Zylera entered into joint legal representation along with other
unrelated third parties in negotiation and arbitration of a dispute with Summers Labs regarding the existence of a Market Change and the
concomitant obligations of the parties. The arbitration panel issued an interim ruling on October 23, 2018 that no market change had
occurred up to and including the date of the hearing. The arbitration panel issued a second interim ruling on December 26, 2018. The
second interim award rejected Summers Labs' request to accelerate future minimum royalties, however, it ruled in favor of Summers Labs
that it is owed reimbursement for all reasonable costs and expenses, including legal fees, by Shionogi, as well as interest, as stipulated in the
contract. The arbitration panel issued a final award on March 1, 2019 that dictated the final amount of reimbursable costs and interest as
contemplated in the second interim ruling. The final award has no direct bearing on the Company as the Company was not a named
defendant to the original claim by Summers Labs and a federal court denied Zylera's ability to be a counterclaimant in the matter.
Furthermore, the Company is not subject to the guarantee or interest provisions identified in the second ruling as these elements of the
contractual relationship were not passed down to the Company’s agreement with Lachlan. However, the Company has interpreted this
ruling's impact on the Lachlan agreement to mean that a market change has not occurred, and the minimum purchase obligation and
minimum royalty provisions of the contract are active and due for any prior periods as well as going forward for any future periods.

The Company has recognized a $7.8 million liability for these minimum obligations in accrued liabilities as of December 31,

2018. Under the terms of the TRx Purchase Agreement, the former TRx owners are required to indemnify the Company for 100% of all
pre-acquisition losses related this arbitration, including legal costs, and possible minimum payments in excess of $1 million. Furthermore,
the former TRx owners are required to indemnify the Company for 50% of post-acquisition Ulesfia losses, which would include losses
resulting from having to fund these minimum obligations. The Company has recorded an indemnity receivable of $4.9 million in other
receivables as of December 31, 2018, which the Company believes is fully collectible. The receivable is net of $1.9 million collection made
in the fourth quarter of 2018 from a full cash escrow release with the former TRx owners from the escrow that was established as a part of
the TRx acquisition. The post-acquisition minimum obligations net of amounts recorded within the indemnity receivable of $2.2 million
has been recorded in cost of product sales for the year ended December 31, 2018. If the Company fails to make these minimum obligations
timely then the Lachlan Agreement may be terminated by Lachlan, in which case the Company would no longer be able to sell the Ulesfia
product, but it would also not be subject to future minimum obligations. Lachlan has not requested payment for the minimum obligations.

Commercial, Supply, and Distribution Agreements

Acquired Product Marketing Rights - Karbinal

On February 16, 2018, in connection with the acquisition of Avadel's pediatric products, the Company entered into a supply and

distribution agreement with TRIS Pharma (the "Karbinal Agreement"), under which the Company is granted the exclusive right to
distribute and sell the product in the United States. The initial term of the Karbinal Agreement is 20 years. The Company will pay

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TRIS a royalty equal to 23.5% of net sales. Avadel has agreed to offset the 23.5% royalty payable by 8.5%, for a net royalty equal to 15%,
in fiscal year 2018 and 2019 for net sales of Karbinal. The make-whole payment is capped at $750,000 each year. The Karbinal Agreement
also contains minimum unit sales commitments, which is based on a commercial year that spans from August 1 through July 31, of 70,000
units through 2033. The Company is required to pay TRIS a royalty make whole payment of $30 for each unit under the 70,000 units
annual minimum sales commitment through 2033. The annual payment is due in August of each year. The Karbinal Agreement also has
multiple commercial milestone obligations that aggregate up to $3.0 million based on cumulative net sales, the first of which is triggered
at $40.0 million.

Acquired Product Marketing Rights - AcipHex

On February 16, 2018, in connection with the acquisition of Avadel's pediatric products, the Company assumed the License and

Assignment Agreement for AcipHex (“AcipHex Agreement”) between Eisai, Inc. and FSC Therapeutics, LLC dated June 2014 and the
Supply Agreement between Eisai, Inc. and FSC Laboratories, Inc. dated June 2014. Per the AcipHex Agreement, the Company is granted
the exclusive license to exploit the products in the territory (U.S.) and an exclusive license to use Eisai trademarks to sell the products. Eisai
will manufacture and supply the requirements for supply of the products. The term of the AcipHex Agreement is perpetual unless
terminated per the agreement. Eisai will receive (a) a royalty with respect to the sales of AcipHex equal to 15.0% of Net Sales. The royalties
are payable until the first commercial sale of an unauthorized generic product in the territory or the date that is five years from the effective
date of the agreement. A maximum $8.0 million of sales-based milestone payments is possible should AcipHex accumulated net sales
exceed $50.0 million in any twelve-month period

Acquired Product Marketing Rights- Cefaclor

On February 16, 2018, in connection with the acquisition of Avadel's pediatric products, the Company assumed the License,

Supply and Distribution Agreement for Cefaclor between Yung Shin Pharm. Ind, Co., Ltd. and FSC Therapeutics, LLC dated March 2015
(“Cefaclor Agreement”). The initial term of the Cefaclor Agreement runs through December 31, 2024 and will automatically renew for
additional, successive twelve-month periods unless terminated by either party. Yung Shin will receive a royalty equal to 15.0% of Net Sales
of Cefaclor. A maximum $6.5 million of sales-based milestone payments is possible should Cefaclor accumulated net sales exceed $40.0
million in any twelve-month period.

12. Deerfield Debt Obligation

In relation to the Company's acquisition of Avadel's pediatric products on February 16, 2018, the Company assumed an obligation
that Avadel had to Deerfield (the "Deerfield Obligation").  Beginning in July 2018 through October 2020, the Company will pay a quarterly
payment  of $262,500  to  Deerfield.  In  January  2021,  a  balloon  payment  of $15,250,000  is  due.  On  the  acquisition  date,  the  Company
determined the fair value of these payments to be $15,075,000 using a market participant's estimated cost of debt. Management performed a
credit risk analysis that determined the Company's credit rating to be B to BB plus the yield on a ten-year treasury security. The difference
between the gross value and fair value of these payments will be recorded as interest expense in the Company's consolidated statements of
operations  through  January  2021  using  the  effective  interest  method. Interest  expense  for  the  year  ended  December  31,  2018  was $0.8
million and is included in interest expense, net on the accompanying statements of operations. The amounts due within the next year are
included in current portion of long-term debt on the Company's consolidated balance sheets. The amounts due in greater than one year are
included  in  long-term  debt,  net  of  current  portion,  on  the  Company's  consolidated  balance  sheets. The  Deerfield  Obligation  was $15.4
million  as  of  December  31,  2018,  of  which $1.1  million  is  recorded  as  a  current  liability. The  Deerfield  Obligation  contains  certain
covenants in which the Company is in compliance with as of December 31, 2018.

13. Capital Structure

According to the Company's amended and restated certificate of incorporation, the Company is authorized to issue two classes of
stock, common stock and preferred stock. At December 31, 2018, the total number of shares of capital stock the Company was authorized
to issue was 205,000,000 of which 200,000,000 was common stock and 5,000,000 was preferred stock. All shares of common and preferred
stock have a par value of $0.001 per share.

On April 27, 2017, the Company further amended its certificate of incorporation in connection with the closing of the Armistice
Private  Placement  (as  defined  below)  with  the  filing  of  a  Certificate  of  Designation  of  Preferences,  Rights  and  Limitations  of  Series A
Convertible  Preferred  Stock  (“Series  A  Preferred  Stock”)  of  Cerecor  Inc.  (the  “Certificate  of  Designation  of  the  Series  A  Preferred
Stock”). The Certificate of Designation of the Series A Preferred Stock authorized the issuance of  4,179 shares of Series A Preferred Stock
to Armistice with a stated value of $1,000 per share, convertible into 11,940,000 shares of the Company’s common stock at a conversion
price of $0.35 per share and was approved by its shareholders on June 30, 2017. On July 6, 2017, Armistice converted all of its outstanding
shares of Series A Preferred Stock into common stock.

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On  December  26,  2018,  the  Company  filed  a  Certificate  of  Designation  of  Preferences  of  Series  B  Non-Voting  Convertible
Preferred Stock ("Series B Convertible Preferred Stock" or "convertible preferred stock") of Cerecor Inc. (the “Certificate of Designation of
the  Series  B  Preferred  Stock”)  classifying  and  designating  the  rights,  preferences  and  privileges  of  the  Series  B  Convertible  Preferred
Stock. The  Certificate  of  Designation  of  the  Series  B  Convertible  Preferred  Stock  authorized  the  issuance  of 2,857,143  shares  of
convertible preferred stock to Armistice with a par value of  $0.001 per share. The Series B Convertible Preferred Stock converts to shares
of common stock on a 1 for 5 ratio and holds no voting rights.

Convertible Preferred Stock

December 2018 Armistice Private Placement

On December 27, 2018, the Company entered into a series of transactions as part of a private placement with Armistice in order to
generate cash to continue to develop our pipeline assets and for general corporate purposes. The transactions are considered one transaction
for accounting purposes. As part of the transaction, the Company exchanged common stock warrants issued on April 27, 2017 to Armistice
for the purchase up to 14,285,714 shares of the Company’s common stock at an exercise price of $0.40 per share (the "original warrants")
for like-kind warrants to purchase up to 2,857,143 shares of the Company's newly designated Series B Convertible Preferred Stock with an
exercise  price  of $2.00  per  share  (the  "exchanged  warrants"). Armistice immediately  exercised  the  exchanged  warrants  and  acquired  an
aggregate of 2,857,143 shares of the convertible preferred stock. Net proceeds of the transaction were approximately $5.7 million.

In order to provide Armistice an incentive to exercise the exchanged warrants, the Company also entered into a securities purchase
agreement with Armistice pursuant to which the Company issued warrants for  4,000,000 shares of common stock of the Company with a
term  of 5.5 years  and  an  exercise  price  of $12.50  per  share  (the  "incentive  warrants"). For  accounting  purposes  this  was  considered  a
deemed  distribution  to Armistice  of $1.7 million. The  deemed  distribution  is  calculated  as  the  difference  between  the  fair  value  of  the
incentive warrants on the date of the transaction of $2.2 million and the value that Armistice forwent by exchanging the original warrants of
$0.5 million. The fair value of the incentive warrant is estimated using a Black-Scholes option-pricing model. The significant assumptions
used in the model for valuing the incentive warrant on December 27, 2018 include (i) volatility of 55%, (ii) risk free interest rate of 2.62%,
(iii) unit strike price of $12.50, (iv) fair value of underlying equity of $3.02, and (v) expected life of 5.5 years.

Voting

Holders of the Company's convertible preferred stock are not entitled to vote.

Dividends

The holders of convertible preferred stock are entitled to receive dividends, if any, as may be declared from time to time by the

board of directors out of legally available funds.

Liquidation

In the event of the Company’s liquidation, dissolution or winding up, holders of the Company’s convertible preferred stock will be
entitled to share ratably in the net assets legally available for distribution to stockholders after the payment of all debts and other liabilities.

Rights and Preferences

Each share of convertible preferred stock converts to shares of common stock on a 1 for 5 ratio. There are no other preemptive or

subscription rights and there are no redemption or sinking fund provisions applicable to the Company’s common stock.

Common Stock

Common Stock Offering

On March 8, 2019, the Company closed on an underwritten public offering of common stock for 1,818,182 shares of common
stock of the Company, at a price to the public of $5.50 per share. Armistice participated in the offering by purchasing 363,637 shares of
common stock of the Company from the underwriter at the public price. The net proceeds to the Company from the offering was
approximately $9.0 million.

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Armistice Private Placements

As  discussed  in  detail  above  (see  "December  2018  Armistice  Private  Placement"  ),  on  December  27,  2018  the  Company
exchanged previously outstanding warrants for like-kind warrants for 2,857,143 shares of the Company's convertible preferred stock with
an exercise price of $2.00 per share which Armistice immediately exercised thus acquiring 2,857,143 shares of convertible preferred stock
for net proceeds of $5.7 million. The convertible preferred stock converts to common stock on a 1 to 5  ratio  (or  to 14,285,714 shares of
common stock in total). Additionally, on December 27, 2018, in order to provide Armistice an incentive to exercise the exchanged warrants,
the Company entered into a securities purchase agreement with Armistice pursuant to which the Company issued warrants for 4,000,000
shares of common stock of the Company with a term of 5.5 years and an exercise price of $12.50 per share (the "incentive warrants"). See
"December 2018 Armistice Private Placement" above for more details.

On August 17, 2018, the Company entered into a securities purchase agreement with Armistice, pursuant to which the Company
sold 1,000,000 shares of the Company’s common stock, $0.001 par value per share for a purchase price of $3.91 per share, which was the
closing price of shares of the Common Stock on August 16, 2018. Net proceeds of this securities purchase agreement were approximately
$3.9 million.

On  April  27,  2017,  the  Company  entered  into  a  securities  purchase  agreement  with  Armistice,  pursuant  to  which  Armistice
purchased $5.0 million of the Company’s securities, consisting of  2,345,714 shares of the Company’s common stock at a purchase price of
$0.35 per share and 4,179 shares of Series A Preferred Stock at a price of  $1,000  per  share.  The  Company  received $4.65 million in net
proceeds  from  the Armistice  Private  Placement.  The  number  of  shares  of  common  stock  that  were  purchased  in  the  private  placement
constituted approximately 19.99% of the Company’s outstanding shares of common stock immediately prior to the closing of the Armistice
Private Placement. Armistice also received warrants to purchase up to 14,285,714 shares of the Company’s common stock at an exercise
price  of $0.40  per  share.  Under  the  terms  of  the  securities  purchase  agreement,  the  Series A  Preferred  Stock  were  not  convertible  into
common  stock,  and  the  warrants  were  not  exercisable  until  the  Company  received  approval  of  the  private  placement  by  the  Company’s
shareholders as required by the rules and regulations of the NASDAQ Capital Market. The Company received shareholder approval for this
transaction  on  June  30,  2017,  at  which  time  the  warrants  became  exercisable  and  the  Series A  Preferred  Stock  became  convertible  into
common stock.

As  multiple  instruments  were  issued  in  a  single  transaction,  the  Company  initially  allocated  the  issuance  proceeds  among  the
preferred stock, common stock and warrants using the relative allocation method. As the warrants were determined to be indexed to the
Company’s  stock,  and  would  only  be  settled  in  common  shares,  entirely  in  the  control  of  the  Company,  the  warrant  instrument  was
accounted for as an equity instrument. Fair value of the warrants was initially determined upon issuance using the Black-Scholes Model
(level 3 fair value measurement). Armistice converted all of the Series A Preferred Stock into  11,940,000 shares of common stock on July
6, 2017.

Ichorion Asset Acquisition

On September 25, 2018, under the terms of the Ichorion Asset Acquisition noted above in Note 4, the Company issued  5.8 million

common stock shares upon closing.

Contingently Issuable Shares

Under the terms of TRx acquisition noted above in Note 4, the Company was required to issue common stock having an aggregate
value as calculated in the TRx Purchase Agreement on the Closing Date of  $8.1 million (the “Equity Consideration”).  Upon closing, the
Company issued 5,184,920 shares of its common stock.  Pursuant to the TRx Purchase Agreement, the issuance of the remaining  2,349,968
shares  as  a  part  of  the  Equity  Consideration  was  subject  to  stockholder  approval  at  the  Company's  2018 Annual  Stockholder's  Meeting.
This approval was obtained in May 2018 and the remaining shares were issued to the TRx Sellers.

Voting

Common stock is entitled to one vote for each share held of record on all matters submitted to a vote of the stockholders, including
the election of directors, and does not have cumulative voting rights. Accordingly, the holders of a majority of the shares of common stock
entitled to vote in any election of directors can elect all of the directors standing for election.

Dividends

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The holders of common stock are entitled to receive dividends, if any, as may be declared from time to time by the board of

directors out of legally available funds.

Liquidation

In the event of the Company’s liquidation, dissolution or winding up, holders of the Company’s common stock will be entitled to

share ratably in the net assets legally available for distribution to stockholders after the payment of all debts and other liabilities.

Rights and Preferences

Holders of the Company’s common stock have no preemptive, conversion or subscription rights, and there are no redemption or

sinking fund provisions applicable to the Company’s common stock.

Common Stock Warrants

At December 31, 2018, the following common stock warrants were outstanding: 

Number of shares

underlying warrants
22,328*
2,380*
4,000,000
4,024,708

Exercise price

Expiration

per share

date

  $
  $
  $

8.40   October 2020
8.68  
12.50  

May 2022
June 2024

*Accounted for as a liability instrument (see Note 5)

14. Stock-Based Compensation

2016 Equity Incentive Plan

On April 5, 2016, the Company’s Board of Directors adopted the 2016 Equity Incentive Plan (the “2016 Plan”) as the successor to
the 2015 Omnibus Plan (the “2015 Plan”). The 2016 Plan was approved by the Company’s stockholders and became effective on May 18,
2016 (the “2016 Plan Effective Date”).

As of the 2016 Plan Effective Date, no additional grants will be made under the 2015 Plan or the 2011 Stock Incentive Plan (the
“2011 Plan”), which was previously succeeded by the 2015 Plan effective October 13, 2015. Outstanding grants under the 2015 Plan and
2011 Plan will continue according to their terms as in effect under the applicable plan.

Upon the 2016 Plan Effective Date, the 2016 Plan reserved and authorized up to 600,000 additional shares of common stock for
issuance,  as  well  as 464,476  unallocated  shares  remaining  available  for  grant  of  new  awards  under  the  2015  Plan. An Amended  and
Restated  2016  Equity  Incentive  Plan  (the  "2016 Amended  Plan")  was  approved  by  the  Company's  stockholders  in  May  2018,  which
increased  the  share  reserve  by  an  additional 1.4  million  shares. During  the  term  of  the  2016  Amended  Plan,  the  share  reserve  will
automatically  increase  on  the  first  trading  day  in  January  of  each  calendar  year,  by  an  amount  equal  to 4%  of  the  total  number  of
outstanding shares of common stock of the Company on the last trading day in December of the prior calendar year. As of December 31,
2018, there were 602,657 shares available for future issuance under the 2016 Plan. On January 1, 2019, on the terms of the 2016 Amended
Plan an additional 1,632,167 shares were made available for issuance for a total of 2,234,824 shares available for issuance.

Option grants to employees and directors expire after ten years. Employee options typically vest over four  years. Options granted
to  directors  typically  vest  over three  years. Directors  may  elect  to  receive  stock  options  in  lieu  of  board  compensation  which  vest
immediately. For  stock  options  granted  to  employees  and  non-employee  directors,  the  estimated  grant  date  fair  market  value  of  the
Company’s  stock-based  awards  is  amortized  ratably  over  the  individuals’  service  periods,  which  is  the  period  in  which  the  awards  vest.
Stock-based  compensation  expense  includes  expense  related  to  stock  options,  restricted  stock  awards  and  ESPP  shares. The  amount  of
stock-based compensation expense recognized for the years ending December 31, 2018 and 2017 was as follows:

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Research and development
General and administrative
Sales and marketing
Total stock-based compensation

Year Ended December 31,

2018

101,000   $

2,135,710  
194,353  
2,431,063   $

2017

156,047
1,001,205
—
1,157,252

  $

  $

During the third quarter of 2018, the Company modified stock options of a senior executive who was separated in the period. This
modification  resulted  in  the  recognition  of  approximately $322,000  of  compensation  expense,  which  is  included  in  general  and
administrative expenses for the year ended December 31, 2018 in the accompanying statement of operations.

Stock options with service-based vesting conditions

The  Company  has  granted  awards  that  contain  service-based  vesting  conditions. The  compensation  cost  for  these  options  is
recognized  on  a  straight-line  basis  over  the  vesting  periods. A  summary  of  option  activity  with  service-based  vesting  conditions  for  the
year ended December 31, 2018 is as follows:

Balance at December 31, 2017

Granted
Exercised
Forfeited

Balance at December 31, 2018
Exercisable at December 31, 2018

Options Outstanding

  Number of shares

Weighted average
exercise price

Grant date fair
value of options  

2,823,489   $
1,639,860   $
(243,115)    
(473,637)   $
3,746,597   $
1,997,468   $

3.93  
3.85   $

2.77   $
4.16  
4.71  

3,737,728  

1,109,083  

Weighted
average
remaining
contractual term
(in years)

7.29

7.79
6.62

The aggregate intrinsic value of stock options is calculated as the difference between the exercise price of the stock options and

the fair value of the Company’s common stock for those stock options that had exercise prices lower than the fair value of the Company’s
common stock. As of December 31, 2018, the aggregate intrinsic value of options outstanding and options currently exercisable was $1.5
million and $1.0 million, respectively. The total intrinsic value of options exercised during the year ended December 31, 2018 was $0.5
million. The total grant date fair value of shares which vested during the years ended December 31, 2018 and 2017 was $1.2 million and
$2.9 million, respectively. The per‑share weighted‑average grant date fair value of the options granted during 2018 and 2017 was estimated
at $2.28 and $0.66, respectively. There were 641,286 options that vested during the year ended December 31, 2018 with a weighted average
grant date fair value of $1.87 per share. At December 31, 2018, there was $3,062,257 of total unrecognized compensation cost related to
nonvested service-based vesting conditions awards. This unrecognized compensation cost is expected to be recognized over a weighted-
average period of 3.1 years.

Stock options with market-based vesting conditions

During  2018  the  Company  granted  awards  that  contain  market-based  vesting  conditions. A  summary  of  option  activity  with

market-based vesting conditions for the year ended December 31, 2018 is as follows:

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Balance at December 31, 2017

Granted

Balance at December 31, 2018
Exercisable at December 31, 2018

Options Outstanding

Weighted
average
remaining
contractual term
(in years)

Aggregate
intrinsic value (1)

Weighted average
exercise price

4.24    
4.24  

9.24   $

—

  Number of shares  
—    
500,000   $
500,000   $
—    

(1) The aggregate intrinsic value in the above table represents the total pre-tax amount that a participant would receive if the option had
been exercised on the last day of the respective fiscal period. Options with a market value less than its exercise value are not included in the
intrinsic value amount.

The weighted-average grant-date fair value of stock options with market-based vesting conditions granted during 2018 was $2.52
per share or $1,260,000. At December 31, 2018, there was $917,568 of total unrecognized compensation cost related to nonvested market-
based vesting conditions awards. This compensation cost is expected to be recognized over a weighted-average period of 2.05 years.

Stock-based compensation assumptions

The  following  table  shows  the  assumptions  used  to  compute  stock-based  compensation  expense  for  stock  options  granted  to
employees and members of the board of directors under the Black-Scholes valuation model, and the assumptions used to compute stock-
based compensation expense for market-based stock option grants under a Monte Carlo simulation:

Service-based options
Risk-free interest rate
Expected term of options (in years)
Expected stock price volatility
Expected annual dividend yield
Market-based options
Risk-free interest rate
Expected term of options (in years)
Expected stock price volatility
Expected annual dividend yield

Year Ended December 31,

2018

2017

  2.51%   —   3.01%   1.85%   —   2.38%  

6.25

  —  

5.0
55%   —   100%  
0%  
0%   —  

  —  
5.0
55%   —  
0%   —  

6.25
65%  
0%  

2.84%
2.8
60%
0%

The valuation assumptions were determined as follows:

• Risk‑free interest rate:  The Company bases the risk‑free interest rate on the interest rate payable on U.S. Treasury securities in

effect at the time of grant for a period that is commensurate with the assumed expected option term.

• Expected term of options:  Due to lack of sufficient historical data, the Company estimates the expected life of its stock options
with service-based vesting granted to employees and members of the board of directors as the arithmetic average of the vesting
term and the original contractual term of the option for service-based options. The expected life of stock options with market-
based vesting is derived from a Monte Carlo simulation which is the valuation technique used to value such awards.

• Expected stock price volatility:  The Company estimated the expected volatility based on actual historical volatility of the stock
price  of  other  publicly‑traded  biotechnology  companies  engaged  in  lines  of  business  that  are  the  same  or  similar  to  the
Company’s.  The  Company  calculated  the  historical  volatility  of  the  selected  companies  by  using  daily  closing  prices  over  a
period of the expected term of the associated award. The companies were selected based on their enterprise value, risk profiles,
position within the industry, and with historical share price information sufficient to meet the expected term of the associated
award. A decrease in the selected volatility would decrease the fair value of the underlying instrument.

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• Expected annual dividend yield:  The Company estimated the expected dividend yield based on consideration of its historical
dividend  experience  and  future  dividend  expectations.  The  Company  has  not  historically  declared  or  paid  dividends  to
stockholders. Moreover, it does not intend to pay dividends in the future, but instead expects to retain any earnings to invest in
the continued growth of the business. Accordingly, the Company assumed and expected dividend yield of 0.0%.

Restricted Stock Award

During 2018, the Company granted restricted stock awards ("RSA") to certain employees. The Company measures the fair value
of the restricted awards using the stock price at the date of the grant. The restricted shares vest annually over a four year period beginning
on the first anniversary of the award. A summary of RSA grants activity for the year ended December 31, 2018 is as follows:

Non-vested RSAs at December 31, 2017

Granted

Non-vested RSAs at December 31, 2018

Non-vested RSAs Outstanding

  Number of shares

Weighted average
grant date fair
value

—    
445,000   $
445,000    

4.27  

The stock compensation expense on this award for the year ended December 31, 2018 was  $346,514. At December 31, 2018, there
was $1,551,986 of total unrecognized compensation cost related to the RSA grants. This compensation cost is expected to be recognized
over a weighted-average period of 3.3 years.

Employee Stock Purchase Plan

On April 5, 2016, the Company’s board of directors approved the 2016 Employee Stock Purchase Plan (the “ESPP”). The ESPP

was approved by the Company’s stockholders and became effective on May 18, 2016 (the “ESPP Effective Date”).

Under  the  ESPP,  eligible  employees  can  purchase  common  stock  through  accumulated  payroll  deductions  at  such  times  as  are
established by the administrator. The ESPP is administered by the compensation committee of the Company’s board of directors. Under the
ESPP, eligible employees may purchase stock at  85% of the lower of the fair market value of a share of the Company’s common stock (i)
on the first day of an offering period or (ii) on the purchase date. Eligible employees may contribute up to 15% of their earnings during the
offering period. The Company’s board of directors may establish a maximum number of shares of the Company’s common stock that may
be purchased by any participant, or all participants in the aggregate, during each offering or offering period. Under the ESPP, a participant
may not accrue rights to purchase more than $25,000 of the fair market value of the Company’s common stock for each calendar year in
which such right is outstanding.

Upon the ESPP Effective Date, the Company reserved and authorized up to  500,000 shares of common stock for issuance under
the  ESPP.  On  January  1  of  each  calendar  year,  the  aggregate  number  of  shares  that  may  be  issued  under  the  ESPP  shall  automatically
increase by a number equal to the lesser of (i) 1% of the total number of shares of the Company’s capital stock outstanding on December 31
of  the  preceding  calendar  year,  and  (ii) 500,000  shares  of  the  Company’s  common  stock,  or  (iii)  a  number  of  shares  of  the  Company’s
common stock as determined by the Company’s board of directors or compensation committee. As of December 31, 2018, 783,983 shares
remained available for issuance.

In accordance with the guidance in ASC 718-50, the ability to purchase shares of the Company’s common stock at the lower of the
offering date price or the purchase date price represents an option and, therefore, the ESPP is a compensatory plan under this guidance.
Accordingly,  stock-based  compensation  expense  is  determined  based  on  the  option’s  grant-date  fair  value  and  is  recognized  over  the
requisite  service  period  of  the  option.  The  Company  used  the  Black-Scholes  valuation  model  and  recognized  stock-based  compensation
expense of $49,863 and $76,305 for the years ended December 31, 2018 and December 31, 2017, respectively, which are included in the
table above with stock-based compensation from stock options.

15. Income Taxes

The Company accounts for income taxes in accordance with ASC 740 (Topic 740, Income Taxes).  ASC Topic 740 is an asset and
liability approach that requires the recognition of deferred tax assets and liabilities for the expected tax consequences or events that have
been recognized in the financial statements or tax returns. ASC Topic 740 also clarifies the accounting for uncertainty in income

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taxes  recognized  in  the  financial  statement. The  interpretation  prescribes  a  recognition  threshold  and  measurement  attribute  for  the
financial statement recognition and measurement of a tax position taken, or expected to be taken, in a tax return. There were no significant
matters determined to be unrecognized tax benefits taken or expected to be taken in a tax return that have been recorded in our financial
statement  for  the  calendar  year  2018. Tax  years  beginning  in  2015  are  generally  subject  to  examination  by  taxing  authorities,  although
NOLs from all years are subject to examinations and adjustments for at least three years following the year in which the attributes are used.

ASC Topic 740 provides guidance on the recognition of interest and penalties related to income taxes. There were $0.2 million of
interest  and  penalties  related  to  unrecognized  tax  benefits  for  income  taxes  that  have  been  accrued  or  recognized  as  of  and  for  the  year
ended  December  31,  2018. It  is  the  Company's  policy  to  treat  interest  and  penalties,  to  the  extent  they  arise,  as  a  component  of  income
taxes.

The income tax provision consisted of the following for the years ending December 31, 2018 and 2017:

Current:
   Federal
   State
Total Current:

Deferred:
   Federal
   State
Total Deferred

Net income tax (benefit) expense

December 31,

2018

2017

(53,281)   $
36,116  
(17,165)  

2,309,285
489,863
2,799,148

(52,235)  
35,490  
(16,745)  
(33,910)   $

(789,274)
(43,355)
(832,629)
1,966,519

  $

  $

The net deferred tax liabilities consisted of the following for the years ending December 31, 2018 and 2017:

Deferred tax assets:

Net operating losses
Accrued compensation
Deferred rent
Tax credits
Stock-based compensation
Installment sale
Other reserves
Basis difference in tangible and intangible assets, net

Total deferred tax assets
Deferred tax liabilities:
Prepaid expenses
Installment sales

Total deferred tax liabilities
Deferred tax asset, net
Less valuation allowance
Net deferred taxes

December 31,

2018

2017

  $

4,421,423   $
465,430  
15,373  
252,095  
1,922,736  
508,291  
262,260  
2,968,764  
10,816,372  

(160,474)  
—  
(160,474)  
10,655,898  
(10,725,136)  

  $

(69,238)   $

716,819
271,437
4,051
—
1,291,230
—
72,881
2,019,272
4,375,690

—
(358,844)
(358,844)
4,016,846
(4,023,990)
(7,144)

As of December 31, 2018, the Company has roughly $16,426,000 of gross NOLs for federal and state tax purposes of which

approximately $3,580,000 will begin to expire in 2031, while the remaining amount of  $12,846,000 will carryforward indefinitely.

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The income tax benefit for the years ended December 31, 2018 and 2017 differed from the amounts computed by applying the

U.S. federal income tax rate as follows:

Federal statutory rate
Permanent Adjustments
Built-in-loss
State taxes
Research and development credit
Change in statutory rate due to Tax Cuts and Job Act
NOL adjustment per § 382
Non-deductible IPR&D expense
Other
Change in valuation allowance

Effective income tax rate

December 31,

2018

2017

21.00 %  
(0.37)%  
(0.33)%  
4.43 %  
0.61 %  
— %  
— %  
(9.84)%  
(0.04)%  
(15.37)%  
0.09 %  

34.00 %
0.17 %
1.52 %
27.91 %
(1.04)%
15.82 %
126.82 %
— %
0.04 %
(191.03)%
14.21 %

The valuation allowance recorded by the Company as of December 31, 2018 and December 31, 2017 resulted from the
uncertainties of the future utilization of deferred tax assets relating from NOL carry forwards for federal and state income tax purposes.
Realization of the NOL carry forwards is contingent on future taxable earnings. The deferred tax asset was reviewed for expected
utilization using a “more likely than not” approach by assessing the available positive and negative evidence surrounding its recoverability.
Accordingly, a partial valuation allowance continues to be recorded against the Company’s deferred tax asset as of December 31, 2018 and
December 31, 2017, as it was determined based upon past and projected future losses that it was “more likely than not” that the Company’s
deferred tax assets would not be realized. As of December 31, 2018 and December 31, 2017, the Company has a net deferred tax liability
due to having an indefinite life asset, referred to as a “naked credit.” The naked credit can be offset up to 80% by NOLs generated after
January 1, 2018, the remaining 20% remains as a liability. In future years, if the deferred tax assets are determined by management to be
“more likely than not” to be realized, the recognized tax benefits relating to the reversal of the valuation allowance as of December 31,
2018 and December 31, 2017 will be recorded. The Company will continue to assess and evaluate strategies that will enable the deferred
tax asset, or portion thereof, to be utilized, and will reduce the valuation allowance appropriately as such time when it is determined that
the “more likely than not” criteria is satisfied.

The Company's current and future unused losses may be subject to limitation under Sections 382 and 383 of the IRC. Sections 382

and 383 of the IRC subject the future utilization of NOLs and certain other tax attributes, such as research and experimental tax credits, to
an annual limitation in the event of certain ownership changes, as defined (in general, an “ownership change” is defined as a greater than
50% change (by value) in equity ownership over a three-year period).

On December 22, 2017, H.R. 1 (also, known as the Tax Cuts and Jobs Act (the “Act”)) was signed into law. Among its numerous

changes to the IRC, the Act reduces U.S. federal corporate tax rate from 35% to 21%. In addition, the SEC staff issued Staff Accounting
Bulletin No. 118, Income Tax Accounting Implications of the Tax Act ("SAB 118") which allowed the Company to record provisional
amounts during a measurement period not to extend beyond one year from the enactment date. Since the Tax Act was passed late in the
fourth quarter of 2017, ongoing guidance and accounting interpretation was expected over the past year, and significant data and analysis
was required to finalize amounts recorded pursuant to the Tax Act, the Company considered the accounting for the deferred tax
remeasurements and other items to be incomplete at December 31, 2017 due to the forthcoming guidance and its ongoing analysis of final
year-end data and tax positions. The Company has completed its analysis within the measurement period in accordance with SAB 118 and
there were no material additional adjustments necessary.

16. Commitments and Contingencies

Litigation

The Company is party in various contractual disputes, litigation, and potential claims arising in the ordinary course of business.

The Company does not believe that the resolution of these matters will have a material adverse effect on our financial position or results of
operations except as otherwise disclosed in this document. See Note 11 for further discussion of the Lachlan legal arbitration.

Purchase obligations

F-40

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
    
Table of Contents

The Company has unconditional purchase obligations as a result of recent acquisitions that include agreements to purchase goods

that are enforceable and legally binding and that specify all significant terms including: fixed or minimum quantities to be purchased;
fixed, minimum or variable price provisions; and the approximate timing of the transaction. Purchase obligations exclude agreements that
are cancelable at any time without penalty. The unconditional purchase obligations outstanding as of December 31, 2018 include the
following:

Lachlan Pharmaceuticals Minimum Purchase and Minimum Royalties Obligations

As discussed in Note 4, in November 2017, the Company acquired TRx and its wholly-owned subsidiaries, including Zylera. The

previous owners of TRx beneficially own more than 10% of our outstanding common stock. Zylera, which is now our wholly owned
subsidiary, entered into an agreement with Lachlan Pharmaceuticals, an Irish company controlled by the previous owners of TRx
(“Lachlan”), effective December 18, 2015. Pursuant to the Lachlan Agreement, Lachlan named Zylera as its exclusive distributor of Ulesfia
in the United States and agreed to supply Ulesfia to Zylera exclusively for marketing and sale in the United States.

The Lachlan agreement requires Zylera to purchase a minimum of  20,000 units per year, or approximately $1.2 million worth of

product, from Lachlan, unless and until there has been a “Market Change” involving a new successful competitive product. Zylera must pay
Lachlan $58.84 per unit and handling fees that are equal to $3.66 per unit of fully packaged Ulesfia in 2018 and escalate at a rate of 10%
annually. The Lachlan Agreement also requires that Zylera make certain cumulative net sales milestone payments and royalty payments to
Lachlan with a $3.0 million annual minimum payment unless and until there has been a “Market Change” involving a new successful
competitive product. The Company expects a successful competitive product will enter the market in early 2021 and therefore the future
minimum purchase obligations and royalty payments are expected through 2020.

As of December 31, 2018, future minimum purchase obligations and future minimum royalty payments to Lachlan are as follows:

2019*

2020*

2021

2022

Total*

Minimum Purchase Obligations
Minimum Royalties
     Total

1,257,326
3,000,000
4,257,326

1,265,378
3,000,000
4,265,378

—
—
—

—
—
—

$2,522,704
6,000,000
$8,522,704

*Per the TRx Purchase Agreement, the previous owners of TRx are required to indemnify the Company for 50% of post-acquisition Ulesfia
losses, which include the future minimum purchase obligations and future minimum royalties disclosed above. Thus, the Company's future
net payouts related to the Ulesfia product will be significantly reduced as a result of the indemnification.

Karbinal Royalty Make Whole Provision

As discussed in Note 4, on February 16, 2018, in connection with the acquisition of Avadel's pediatric products, the Company

entered into a supply and distribution agreement with TRIS Pharma (the "Karbinal Agreement"). As part of this agreement, the Company
has an annual minimum sales commitment, which is based on a commercial year that spans from August 1 through July 31, of 70,000 units
through 2033. The Company is required to pay TRIS a royalty make whole payment of $30 for each unit under the 70,000 units annual
minimum sales commitment through 2033. The annual payment is due in August of each year.

The Company paid $0.9 million to TRIS in August 2018 related to the make whole payment for the commercial year ended July
31, 2018. For the year ended December 31, 2018, the Company has accrued $0.7 million in accrued expenses and other current liabilities
related to the Karbinal royalty make whole for the commercial year ending July 31, 2019. The post-acquisition make whole provision
of $1.3 million has been recorded in cost of product sales for the year ended December 31, 2018. The future royalty make whole payments
is unknown as the amount owed to TRIS is dependent on the number of units sold.

Office Lease

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Table of Contents

During the third quarter of 2018, the Company entered into a lease for the Company's new corporate headquarters in Rockville,
Maryland. The  Company  obtained  access  to  the  building  in  September  2018  to  perform  leasehold  improvements,  which  resulted  in  the
lease  commencement  date  for  accounting  purposes. The Company occupied the building in January 2019. The  landlord  provided  a  lease
incentive related for leasehold improvements in the amount of $381,900, which the Company may requisition the landlord for payment on
a  monthly  basis  for  the  work  incurred-to-date. As  of  December  31,  2018,  the  Company  incurred  leasehold  improvements  for  the  full
amount  of  the  incentive  which  the  Company  has  recognized  within  other  receivables. The  Company  recognized  a  corresponding  lease
incentive obligation within other long-term liabilities. The lease incentive obligation is reduced and recognized in income as a reduction to
straight-line rental expense.

The  annual  base  rent  for  the  office  space  is  $161,671,  subject  to  annual 2.5%  increases  over  the  term  of  the  lease. The  lease
provides for a rent abatement for a period of 12 months following the Company's date of occupancy. The lease has an initial term of 10
years from the date the Company makes its first annual fixed rent payment which is expected to occur in January 2020. The Company has
the option to extend the lease two times, each for a period of five years, and may terminate the lease as of the sixth anniversary of the first
annual fixed rent payment, upon the payment of a termination fee. As of the lease commencement date, it is not reasonably certain that the
Company will exercise the renewal periods or early terminate the lease and therefore the end date of the lease for accounting purposes is
January 31, 2030.

The  Company  analyzed  the  lease  agreement  and  determined  the  lease  classification  is  operating. The  Company  recognizes
operating lease rent expense on a straight-line basis over the expected term of each lease. The Company recognized rent expense for this
property of $41,749 in general and administrative expense on the statement of operations for the year ended December 31, 2018.

As of December 31, 2018, minimum operating lease obligations for the new office space are as follows:

2019
2020
2021
2022
2023
Thereafter

Total

  Minimum Lease Payments
  $

—
155,815
169,510
173,748
178,092
1,183,290
1,860,455

  $

F-42

 
   
 
 
 
 
 
 
Exhibit 21.1

Entity Name
Ichorion Therapeutics, LLC
TRx Pharmaceuticals, LLC
Zylera Pharmaceuticals, LLC
Zylera Pharma Corp.

List of Subsidiaries of Cerecor Inc.

Jurisdiction
Delaware
North Carolina
North Carolina
North Carolina

Exhibit 23.1

Consent of Independent Registered Public Accounting Firm

We consent to the incorporation by reference in the following Registration Statements:

(1) Registration Statement (Form S-1 No. 333-204905) as filed on June 12, 2015, and amended on September 8, 2015, September

22, 2015, October 1, 2015, and October 13, 2015,

(2) Registration Statement (Form S-8 No. 333-207949) pertaining to the 2015 Omnibus Incentive Compensation Plan,

(3) Registration Statement (Form S-8 No. 333-211490) pertaining to the 2016 Equity Incentive Plan,

(4) Registration Statement (Form S-8 No. 333-211491) pertaining to the 2016 Employee Stock Purchase Plan,

(5) Registration Statement (Form S-1 No. 333-213676) as filed on September 16, 2016,

(6) Registration Statement (Form S-3 No. 333-214507) as filed on November 8, 2016, and amended on December 1, 2016,

(7) Registration Statement (Form S-3 No. 333-218252) as filed on May 26, 2017,

(8) Registration Statement (Form S-8 No. 333-226767) pertaining to the Amended and Restated 2016 Equity Incentive Plan,

(9) Registration Statement (Form S-3 No. 333-227227) as filed on September 7, 2018, and amended on October 2, 2018, and

(10) Registration Statement (Form S-3 No. 333-229283) as filed on January 17, 2019;

of our report dated March 18, 2019, with respect to the consolidated financial statements of Cerecor Inc. included in this Annual
Report (Form 10-K) of Cerecor Inc. for the year ended December 31, 2018.

/s/ Ernst & Young LLP
Baltimore, Maryland
March 18, 2019

    
 
 
Exhibit 31.1

CERTIFICATION
PURSUANT TO SECTION 302 OF THE SARBANES-OXLEY ACT OF 2002

I, Peter Greenleaf, certify that:

1.

I have reviewed this Annual Report on Form 10-K of
Cerecor Inc.;

2. Based on my knowledge, this report does not contain any untrue statement of a material fact or omit to state a material fact necessary to
make the statements made, in light of the circumstances under which such statements were made, not misleading with respect to the
period covered by this report;

3. Based on my knowledge, the financial statements, and other financial information included in this report, fairly present in all material

respects the financial condition, results of operations and cash flows of the registrant as of, and for, the periods presented in this report;

4. The registrant’s other certifying officer and I are responsible for establishing and maintaining disclosure controls and procedures (as

defined in Exchange Act Rules 13a-15(e) and 15d-15(e)) and internal control over financial reporting (as defined in Exchange Act
Rules 13a-15(f) and 15d-15(f)) for the registrant and have:

a) Designed such disclosure controls and procedures, or caused such disclosure controls and procedures to be designed under our
supervision, to ensure that material information relating to the registrant, including its consolidated subsidiaries, is made
known to us by others within those entities, particularly during the period in which this report is being prepared;

b) Designed such internal control over financial reporting, or caused such internal control over financial reporting to be designed
under our supervision, to provide reasonable assurance regarding the reliability of financial reporting and the preparation of
financial statements for external purposes in accordance with generally accepted accounting principles;

c) Evaluated the effectiveness of the registrant’s disclosure controls and procedures and presented in this report our conclusions
about the effectiveness of the disclosure controls and procedures, as of the end of the period covered by this report based on
such evaluation; and

d) Disclosed in this report any change in the registrant’s internal control over financial reporting that occurred during the

registrant’s most recent fiscal quarter (the registrant’s fourth fiscal quarter in the case of an annual report) that has materially
affected, or is reasonably likely to materially affect, the registrant’s internal control over financial reporting; and

5. The registrant’s other certifying officer and I have disclosed, based on our most recent evaluation of internal control over financial
reporting, to the registrant’s auditors and the audit committee of the registrant’s board of directors (or persons performing the
equivalent functions):

a) All significant deficiencies and material weaknesses in the design or operation of internal control over financial reporting

which are reasonably likely to adversely affect the registrant’s ability to record, process, summarize and report financial
information; and

b) Any fraud, whether or not material, that involves management or other employees who have a significant role in the

registrant’s internal control over financial reporting.

Date: March 18, 2019

/s/ Peter Greenleaf
Peter Greenleaf
Chief Executive Officer
(Registrant’s Principal Executive Officer)

 
 
 
 
 
CERTIFICATION
PURSUANT TO SECTION 302 OF THE SARBANES-OXLEY ACT OF 2002

Exhibit 31.2

I, Joseph M. Miller, certify that:

1.

I have reviewed this Annual Report on Form 10-K of
Cerecor Inc.;

2. Based on my knowledge, this report does not contain any untrue statement of a material fact or omit to state a material fact necessary to
make the statements made, in light of the circumstances under which such statements were made, not misleading with respect to the
period covered by this report;

3. Based on my knowledge, the financial statements, and other financial information included in this report, fairly present in all material

respects the financial condition, results of operations and cash flows of the registrant as of, and for, the periods presented in this report;

4. The registrant’s other certifying officer and I are responsible for establishing and maintaining disclosure controls and procedures (as

defined in Exchange Act Rules 13a-15(e) and 15d-15(e)) and internal control over financial reporting (as defined in Exchange Act
Rules 13a-15(f) and 15d-15(f)) for the registrant and have:

a) Designed such disclosure controls and procedures, or caused such disclosure controls and procedures to be designed under our
supervision, to ensure that material information relating to the registrant, including its consolidated subsidiaries, is made
known to us by others within those entities, particularly during the period in which this report is being prepared;

b) Designed such internal control over financial reporting, or caused such internal control over financial reporting to be designed
under our supervision, to provide reasonable assurance regarding the reliability of financial reporting and the preparation of
financial statements for external purposes in accordance with generally accepted accounting principles;

c) Evaluated the effectiveness of the registrant’s disclosure controls and procedures and presented in this report our conclusions
about the effectiveness of the disclosure controls and procedures, as of the end of the period covered by this report based on
such evaluation; and

d) Disclosed in this report any change in the registrant’s internal control over financial reporting that occurred during the

registrant’s most recent fiscal quarter (the registrant’s fourth fiscal quarter in the case of an annual report) that has materially
affected, or is reasonably likely to materially affect, the registrant’s internal control over financial reporting; and

5. The registrant’s other certifying officer and I have disclosed, based on our most recent evaluation of internal control over financial
reporting, to the registrant’s auditors and the audit committee of the registrant’s board of directors (or persons performing the
equivalent functions):

a) All significant deficiencies and material weaknesses in the design or operation of internal control over financial reporting

which are reasonably likely to adversely affect the registrant’s ability to record, process, summarize and report financial
information; and

b) Any fraud, whether or not material, that involves management or other employees who have a significant role in the

registrant’s internal control over financial reporting.

Date: March 18, 2019

/s/ Joseph M. Miller
Joseph M. Miller
Chief Financial Officer
(Registrant’s Principal Financial and Accounting Officer)

 
 
 
 
CERTIFICATION
PURSUANT TO
18 U.S.C. SECTION 1350,
AS ADOPTED PURSUANT TO
SECTION 906 OF THE SARBANES-OXLEY ACT OF 2002

Exhibit 32.1

In connection with the Annual Report of Cerecor Inc. (the “Registrant”) on Form 10-K for the year ended December 31, 2018 as

filed with the Securities and Exchange Commission on the date hereof (the “Report”), I, Peter Greenleaf, Chief Executive Officer
(principal executive officer) of the Registrant, and I, Joseph M. Miller, Chief Financial Officer (principal financial and accounting officer)
of the Registrant, each hereby certify, pursuant to 18 U.S.C. Section 1350, as adopted pursuant to Section 906 of the Sarbanes-Oxley Act of
2002, that, to my knowledge:

1. The Report fully complies with the requirements of Section 13(a) or 15(d) of the Securities Exchange Act of 1934, as amended;

and

2. The information contained in the Report fairly presents, in all material respects, the financial condition at the end of the period covered

by the Report and the results of operations of the Registrant for the periods covered by the Report.

Date: March 18, 2019

Date: March 18, 2019

By:
Name:

Title:

/s/ Peter Greenleaf
Peter Greenleaf

Chief Executive Officer
(Registrant’s Principal Executive Officer)

/s/ Joseph M. Miller

By:
Name:   Joseph M. Miller

Title:

Chief Financial Officer
(Registrant’s Principal Financial and Accounting Officer)

The foregoing certifications are not deemed filed with the Securities and Exchange Commission for purposes of section 18 of the Securities
Exchange Act of 1934, as amended (Exchange Act), and are not to be incorporated by reference into any filing of Cerecor Inc. under the
Securities Act of 1933, as amended, or the Exchange Act, whether made before or after the date hereof, regardless of any general
incorporation language in such filing.