Quarterlytics / Healthcare / Biotechnology / Hoth Therapeutics, Inc.

Hoth Therapeutics, Inc.

hoth · NASDAQ Healthcare
Claim this profile
Ticker hoth
Exchange NASDAQ
Sector Healthcare
Industry Biotechnology
Employees 1-10
← All annual reports
FY2022 Annual Report · Hoth Therapeutics, Inc.
Sign in to download
Loading PDF…
UNITED STATES
SECURITIES AND EXCHANGE COMMISSION
Washington, D.C. 20549

FORM 10-K

☒ ANNUAL REPORT PURSUANT TO SECTION 13 OR 15(d) OF THE SECURITIES EXCHANGE ACT OF 1934

For the fiscal year ended  December 31, 2022

☐ TRANSITION REPORT PURSUANT TO SECTION 13 OR 15(d) OF THE SECURITIES EXCHANGE ACT OF 1934

For the transition period from ______ to ______

Commission file number 001-38803

HOTH THERAPEUTICS, INC.
(Exact name of registrant as specified in charter)

Nevada
(State or other jurisdiction of 
incorporation or organization)

1 Rockefeller Plaza, Suite 1039, New York, New York
(Address of principal executive offices)

82-1553794
I.R.S. Employer 
Identification No.

10020
(Zip code)

(646) 756-2997
(Registrant’s telephone number, including area code)

Securities registered pursuant to Section 12(b) of the Act:

Title of Each Class
Common Stock, par value $0.0001 per share  

Trading Symbol(s)
HOTH

Name of Each Exchange on Which Registered
The Nasdaq Stock Market LLC

Indicate by check mark if the registrant is a well-known seasoned issuer, as defined in Rule 405 of the Securities Act. Yes  ☐ No ☒

Indicate by check mark if the registrant is not required to file reports pursuant to Section 13 or Section 15(d) of the Act. Yes  ☐ No ☒

Securities registered pursuant to Section 12(g) of the Act:  None.

Indicate by check mark whether the registrant (1) has filed all reports required to be filed by Section 13 or 15(d) of the Securities Exchange Act of 1934
during the preceding 12 months (or for such shorter period that the registrant was required to file such reports), and (2) has been subject to such filing
requirements for the past 90 days. Yes ☒ No ☐

Indicate by check mark whether the registrant has submitted electronically every Interactive Data File required to be submitted pursuant to Rule 405 of
Regulation S-T (§ 232.405 of this chapter) during the preceding 12 months (or for such shorter period that the registrant was required to submit such
files). Yes ☒ No ☐

Indicate by check mark whether the registrant is a large accelerated filer, an accelerated filer, a non-accelerated filer, a smaller reporting company, or an
emerging growth company. See definition of “large accelerated filer,” “accelerated filer,” “smaller reporting company,” and “emerging growth company” in
Rule 12b-2 of the Exchange Act.

Large accelerated filer
Non-accelerated filer

☐
☒

☐
Accelerated filer
Smaller reporting company   ☒
Emerging growth company ☒

If an emerging growth company, indicate by check mark if the registrant has elected not to use the extended transition period for complying with any new
or revised financial accounting standards provided pursuant to Section 13(a) of the Exchange Act. ☐

Indicate by check mark whether the registrant has filed a report on and attestation to its management’s assessment of the effectiveness of its internal
control over financial reporting under Section 404(b) of the Sarbanes-Oxley Act (15 U.S.C. 7262(b)) by the registered public accounting firm that prepared
or issued its audit report. ☐

If securities are registered pursuant to Section 12(b) of the Act, indicate by check mark whether the financial statements of the registrant included in the
filing reflect the correction of an error to previously issued financial statements. ☐

Indicate  by  check  mark  whether  any  of  those  error  corrections  are  restatements  that  required  a  recovery  analysis  of  incentive-based  compensation
received by any of the registrant’s executive officers during the relevant recovery period pursuant to §240.10D-1(b). ☐

Indicate by check mark whether the registrant is a shell company (as defined by Rule 12b-2 of the Exchange Act) Yes  ☐ No ☒

The aggregate market value of the voting stock and non-voting common equity held by non-affiliates of the registrant as of the last business day of the
registrant’s  most  recently  completed  second  fiscal  quarter  ended  June  30,  2022  was  $13.1  million  based  upon  the  closing  price  of  the  registrant’s
common stock of $10.48 on The Nasdaq Capital Market as of that date.

Number of shares of common stock outstanding as of March 17, 2023 was  3,302,113. 

Documents Incorporated by Reference: None.

Table of Contents

Part I
Item 1.
Item 1A.
Item 1B.
Item 2.
Item 3.
Item 4.

Business
Risk Factors
Unresolved Staff Comments
Properties
Legal Proceedings
Mine Safety Disclosures

1
1
12
38
38
38
38

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Part II
Item 5.
Item 6.
Item 7.
Item 7A.
Item 8.
Item 9.
Item 9A.
Item 9B.
Item 9C.

Part III
Item 10.
Item 11.
Item 12.
Item 13.
Item 14.

Part IV
Item 15.

Market For Registrant’s Common Equity, Related Stockholder Matters and Issuer Purchases of Equity Securities
[Reserved]
Management’s Discussion and Analysis of Financial Condition and Results of Operations
Quantitative and Qualitative Disclosures about Market Risk
Financial Statements and Supplementary Data
Changes in and Disagreements With Accountants on Accounting and Financial Disclosure
Controls and Procedures
Other Information
Disclosure Regarding Foreign Jurisdictions that Prevent Inspections

Directors, Executive Officers and Corporate Governance
Executive Compensation
Security Ownership of Certain Beneficial Owners and Management and Related Stockholder Matters
Certain Relationships and Related Transactions, and Director Independence
Principal Accountant Fees and Services

Exhibit and Financial Statement Schedules

Item 16.
Signatures

Form 10-K Summary

i

39
39
39
39
43
F-1
44
44
45
45

46
46
49
55
57
58

59

59
62
63

CAUTIONARY NOTE ON FORWARD-LOOKING STATEMENTS

This  Annual  Report  on  Form  10-K  contains  certain  forward-looking  statements  within  the  meaning  of  Section  27A  of  the  Securities  Act  of  1933,  as
amended  (the  “Securities  Act”),  and  Section  21E  of  the  Securities  Exchange  Act  of  1934,  as  amended  (the  “Exchange  Act”).  Any  statements  in  this
Annual Report on Form 10-K about our expectations, beliefs, plans, objectives, assumptions or future events or performance are not historical facts and
are forward-looking statements. These statements are often, but not always, made through the use of words or phrases such as “believe,” “will,” “expect,”
“anticipate,”  “estimate,”  “intend,”  “plan”  and  “would.”  For  example,  statements  concerning  financial  condition,  possible  or  assumed  future  results  of
operations,  growth  opportunities,  industry  ranking,  plans  and  objectives  of  management,  markets  for  our  common  stock  and  future  management  and
organizational  structure  are  all  forward-looking  statements.  Forward-looking  statements  are  not  guarantees  of  performance.  They  involve  known  and
unknown risks, uncertainties and assumptions that may cause actual results, levels of activity, performance or achievements to differ materially from any
results, levels of activity, performance or achievements expressed or implied by any forward-looking statement.

Any  forward-looking  statements  are  qualified  in  their  entirety  by  reference  to  the  risk  factors  discussed  throughout  this  Annual  Report  on  Form  10-K.
Some  of  the  risks,  uncertainties  and  assumptions  that  could  cause  actual  results  to  differ  materially  from  estimates  or  projections  contained  in  the
forward-looking statements include, but are not limited to:

●

●

●

●

●

●

●

●

●

●

●

●

our business strategies;

the timing of regulatory submissions;

our ability to obtain and maintain regulatory approval of our existing product candidates and any other product candidates we may develop, and
the labeling under any approval we may obtain;

risks relating to the timing and costs of clinical trials and the timing and costs of other expenses;

risks related to market acceptance of products;

the ultimate impact of any health epidemics on our business, our clinical trials, our research programs, healthcare systems or the global economy
as a whole;

intellectual property risks;

risks associated with our reliance on third-party organizations;

our competitive position;

our industry environment;

our anticipated financial and operating results, including anticipated sources of revenues;

assumptions regarding the size of the available market, benefits of our products, product pricing and timing of product launches;

● management’s expectation with respect to future acquisitions;

●

●

statements regarding our goals, intentions, plans and expectations, including the introduction of new products and markets; and

our cash needs and financing plans.

The foregoing list sets forth some, but not all, of the factors that could affect our ability to achieve results described in any forward-looking statements.
You should read this Annual Report on Form 10-K and the documents that we reference herein and have filed as exhibits to the Annual Report on Form
10-K, completely and with the understanding that our actual future results may be materially different from what we expect. You should assume that the

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
information appearing in this Annual Report on Form 10-K is accurate as of the date hereof. Because the risk factors referred to on page 13 of Annual
Report on Form 10-K could cause actual results or outcomes to differ materially from those expressed in any forward-looking statements made by us or
on our behalf, you should not place undue reliance on any forward-looking statements. Further, any forward-looking statement speaks only as of the date
on  which  it  is  made,  and  except  as  required  by  law,  we  undertake  no  obligation  to  update  any  forward-looking  statement  to  reflect  events  or
circumstances after the date on which the statement is made or to reflect the occurrence of unanticipated events. New factors emerge from time to time,
and it is not possible for us to predict which factors will arise. In addition, we cannot assess the impact of each factor on our business or the extent to
which  any  factor,  or  combination  of  factors,  may  cause  actual  results  to  differ  materially  from  those  contained  in  any  forward-looking  statements.  We
qualify  all  of  the  information  presented  in  this  Annual  Report  on  Form  10-K,  and  particularly  our  forward-looking  statements,  by  these  cautionary
statements.

ii

RISK FACTOR SUMMARY

Our business is subject to significant risks and uncertainties that make an investment in us speculative and risky. Below we summarize what we believe
are the principal risk factors but these risks are not the only ones we face, and you should carefully review and consider the full discussion of our risk
factors in the section titled “Risk Factors,” together with the other information in this Annual Report on Form 10-K. If any of the following risks actually
occurs (or if any of those listed elsewhere in this Annual Report on Form 10-K occur), our business, reputation, financial condition, results of operations,
revenue, and future prospects could be seriously harmed. Additional risks and uncertainties that we are unaware of, or that we currently believe are not
material, may also become important factors that adversely affect our business.

Risk Related to our Financial Position and Need for Capital

● We have generated no revenue from commercial sales and our future profitability is uncertain. If we fail to obtain the capital necessary to fund

our operations, we will be unable to continue or complete our product development.

Risk Related to Product Development, Regulatory Approval, Manufacturing and Commercialization

●

The  marketing  approval  process  is  lengthy,  time  consuming  and  inherently  unpredictable,  and  if  we  are  ultimately  unable  to  obtain  marketing
approval for the product candidates we intend to develop, our business may be substantially harmed.

● We may encounter substantial delays in completing our clinical studies which in turn will require additional costs, or we may fail to demonstrate
adequate safety and efficacy to the satisfaction of applicable regulatory authorities. If we are not able to obtain any required regulatory approvals
for our product candidates, we will not be able to commercialize our product candidates and our ability to generate revenue will be limited.

● Conducting successful clinical studies may require the enrollment of large numbers of patients, and suitable patients may be difficult to identify

and recruit.

● We rely on and intend to rely on third parties to conduct our clinical trials, to assist us with pre-clinical development and for manufacturing and
marketing of our proposed product candidates. If we are not able to secure favorable arrangements with such third parties, or such third parties
do not perform as contractually required or expected, we may not be able to obtain regulatory approval for or commercialize our products and our
business and financial condition could be harmed.

● Even  if  our  product  candidates  are  approved  by  regulatory  authorities,  if  we  or  our  suppliers  fail  to  comply  with  ongoing  U.S.  Food  and  Drug
Administration  regulations  or  if  we  experience  unanticipated  problems  with  our  products,  these  products  could  be  subject  to  restrictions  or
withdrawal from the market.

● Our revenue stream will depend upon third-party reimbursement.

● Our products will face significant competition, and if they are unable to compete successfully, our business will suffer.

●

If  we  fail  to  comply  with  healthcare  regulations,  we  could  face  substantial  enforcement  actions,  including  civil  and  criminal  penalties  and  our
business, operations and financial condition could be adversely affected.

iii

Risk Related to our Intellectual Property Rights

● Our  business  depends  upon  us  securing  and  protecting  critical  intellectual  property.  Patent  positions  in  our  industry  are  highly  uncertain  and

involve complex legal and factual questions.

● We rely upon licenses granted to us by various licensors, and if such licensors do not adequately defend such licenses, our business may be

harmed.

Risk Related to our Company

● We have expanded and may continue to expand, our business through the acquisition of rights to new drug candidates that could disrupt our

business, harm our financial condition and may also dilute current shareholders’ ownership interests in our Company.

●

If a product liability claim is successfully brought against us for uninsured liabilities, or such claim exceeds our insurance coverage, we could be
forced to pay substantial damage awards that could materially harm our business.

● Any international operations we undertake may subject us to risks inherent with operations outside of the United States.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Risks Related to our Common Stock

● Market and economic conditions may negatively impact our business, financial condition and share price.

●

Future sales and issuances of our securities could result in additional dilution of the percentage ownership of our shareholders and could cause
our share price to fall.

● We do not intend to pay cash dividends on our shares of common stock so any returns will be limited to the value of our shares.

●

If we are unable to maintain listing of our securities on The Nasdaq Capital Market or any stock exchange, our stock price could be adversely
affected and the liquidity of our stock and our ability to obtain financing could be impaired.

● Our Amended and Restated Bylaws provide that the Eighth Judicial District Court of Clark County, Nevada will be the sole and exclusive forum
for  certain  disputes  which  could  limit  shareholders’  ability  to  obtain  a  favorable  judicial  forum  for  disputes  with  us  or  our  directors,  officers,
employees or agents.

iv

PART I

Throughout this Annual Report on Form 10-K, the “Company,” “Hoth,” “we,” “us,” and “our” refers to Hoth Therapeutics, Inc., individually, or as the context
requires, collectively with its subsidiary, Hoth Therapeutics Australia Pty Ltd.

ITEM 1. BUSINESS

Overview

We  are  a  clinical-stage  biopharmaceutical  company  focused  on  developing  new  generation  therapies  for  unmet  medical  needs.  We  are  focused  on
developing (i) a topical formulation for treating side effects from drugs used for the treatment of cancer (HT-001); (ii) a treatment for mast-cell derived
cancers  and  anaphylaxis  (HT-KIT);  (iii)  a  treatment  for  traumatic  brain  injury  and  ischemic  stroke  (HT-TBI);  and  (iv)  a  treatment  and/or  prevention  for
Alzheimer’s  or  other  neuroinflammatory  diseases  (HT-ALZ).  We  also  have  assets  being  developed  for  (i)  atopic  dermatitis  (also  known  as  eczema)
(BioLexa); (ii) a treatment for asthma and allergies using inhalational administration (HT-004); and (iii) a treatment for acne as well as inflammatory bowel
diseases (HT-003). In addition, we are continuing to evaluate a novel peptide that may be used to slow the transmission of SARS-CoV-2 (HT-002). We
are  also  developing  a  diagnostic  device  via  a  mobile  device.  Furthermore,  we  have  interests  in  certain  other  assets  being  developed  by  third  parties
including  a  treatment  for  patients  with  lupus  that  is  being  developed  by  Zylö  Therapeutics,  Inc.  and  potential  product  candidates  being  developed
pursuant to our agreement with Voltron Therapeutics, Inc. for the prevention of COVID-19.

Primary Development:

HT-001

On February 1, 2020, we entered into a patent license agreement with The George Washington University (“GW”) pursuant to which GW granted us a
license to certain patent rights to, among other things, make, use, offer and sell certain licensed products throughout the world with respect to HT-001
which we intend to seek approval for use for treating dermatological side effects from epidermal growth factor receptor (“EGFR”) inhibitors, and potentially
other drugs used for the treatment of cancer. HT-001 is a topical formulation under development for the treatment of patients with rash and skin disorders
associated with initial and repeat courses of tyrosine kinase EGFR inhibitor therapy. EGFR inhibitors are used for the treatment of cancers with EGFR up-
regulation (such as non-small cell lung cancer, pancreatic cancer, breast cancer and colon cancer); however, EGFR inhibitors are often associated with
dose-limiting skin toxicities that can result in the interruption or reduction of treatment. HT-001 is targeted to treat these EGFR-induced skin disorders to
allow patients to achieve the best potential outcomes of EGFR therapy. HT-001 has achieved positive results in its initial pre-clinical studies conducted at
GW. In November 2022, we submitted an IND to the FDA with respect to HT-001 as a concomitant therapy with EGFR inhibitors, for a Phase 2a clinical
trial  in  humans.  We  have  engaged  Worldwide  Clinical  Trials  (“Worldwide”)  as  our  clinical  research  organization  to  provide  clinical  management,  data
management, biostatistical, medical monitoring, pharmacovigilance, and other related services to support the CLEER-001 Phase 2a clinical trial in the
United States. We received FDA approval to proceed with our clinical study on December 28, 2022.

We believe that the key elements for our market success with respect to HT-001 include:

●

●

●

To our knowledge, there are currently no drugs approved for the treatment of skin toxicities associated with EFGR inhibitor therapy and 49-100%
of patients develop skin toxicities during EGFR inhibitory therapy;

The main active ingredient of HT-001 is already approved in oral and IV dosage forms which supports pursuit of the 505(b)(2) regulatory pathway
to reduce development time and cost;

To our knowledge, there are no current topical formulations available using HT-001’s active ingredient so we believe that there is no direct market
competition; and

● We have the potential to pursue other indications such as chronic pruritus, atopic dermatitis and other skin toxicities that develop from anti-cancer

therapies using the HT-001 formulation.

1

HT-KIT

We have obtained from North Carolina State University (“NC State”) an exclusive, worldwide, royalty bearing license to certain intellectual property to,
among other things, discover, develop, make, have made, use and sell certain licensed products and sell, use and practice certain licensed services with

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
respect  to  cancer  and  anaphylaxis;  this  is  being  developed  as  HT-KIT.  The  HT-KIT  drug  is  designed  to  more  specifically  target  the  receptor  tyrosine
kinase KIT in mast cells, which is required for the proliferation, survival and differentiation of bone marrow-derived hematopoietic stem cells. Mutations in
the KIT pathway have been associated with several human cancers, such as gastrointestinal stromal tumors and mast cell-derived cancers (mast cell
leukemia and mast cell sarcoma). Based on the initial proof-of-concept success, we intend to initially target mast cell neoplasms for development of HT-
KIT, which is a rare, aggressive cancer with poor prognosis.

The same target, KIT, also plays a key role in mast cell-mediated anaphylaxis, a serious allergic reaction that is rapid in onset and may cause death.
Anaphylaxis typically occurs after exposure to an external allergen that results in an immediate and severe immune response. We also intend to pursue
the anaphylaxis indication for HT-KIT in parallel to cancer treatment.

On  November  15,  2021,  we  entered  into  a  sponsored  research  agreement  with  NC  State  to  focus  on  characterizing  the  HT-KIT  dose  and  dosing
frequency for treatment of aggressive mastocytosis and mast cell neoplasms using humanized tumor mouse models.

In  December  2021,  we  submitted  an  Orphan  Drug  Designation  (“ODD”)  request  to  the  U.S.  Food  and  Drug  Administration  (“FDA”)  for  HT-KIT  for  the
treatment of mastocytosis, and on March 10, 2022, we received such ODD. Drugs intended to treat orphan diseases (rare diseases that affect less than
200,000 people in the U.S.) are eligible to apply for ODD, which provides benefits such as 7-year marketing exclusivity and tax incentives to the sponsor
during development and after approval.

HT-ALZ

In February 2021, we filed a provisional patent application with the United States Patent and Trademark Office for the use of the active ingredient of HT-
001 to treat and prevent Alzheimer’s disease and other neuroinflammatory diseases, and in February 2022, we filed a  Patent Cooperation Treaty patent
application, receiving confirmation of such filing on April 4, 2022.

We intend to develop HT-ALZ for use in patients following the Section 505(b)(2) regulatory pathway of the FDA rules. Section 505(b)(2) of the Federal
Food,  Drug,  and  Cosmetic  Act  (“FDCA”)  was  enacted  to  enable  sponsors  to  seek  New  Drug  Application  (“NDA”)  approval  for  novel  repurposed  drugs
without the need for such sponsors to undertake time consuming and expensive pre-clinical safety studies and Phase 1 safety studies. Proceeding under
this regulatory pathway, we will be able to rely upon publicly available data with respect to our active ingredient in our NDA submission to the FDA for
marketing approval.

On  June  7,  2021,  we  entered  into  a  sponsored  research  agreement  with  Washington  University  in  St.  Louis  to  investigate  the  effects  of  HT-ALZ  on
behavioral  and  pathological  markers  of  Alzheimer’s  disease  and  to  determine  if  HT-ALZ  can  improve  learning  and  memory  in  an  animal  model  of
Alzheimer’s disease. Our study will also determine if behavior is improved utilizing HT-ALZ in blocking NK-1Rs. The study commenced in August 2021
and  after  positive  initial  preclinical  results,  a  chronic  dosing  study  in  mice  was  initiated.  We  expect  preclinical  results  from  the  chronic  dosing  study  in
2023.

HT-TBI

In October 2022, we filed a provisional patent application with the United States Patent and Trademark Office for the use of the active ingredient of HT-
001  to  treat  traumatic  brain  injury  and  ischemic  stroke.  We  intend  to  develop  HT-ALZ  for  use  in  patients  following  the  Section  505(b)(2)  regulatory
pathway  of  the  FDA  rules  pursuant  to  which  we  will  be  able  to  rely  upon  publicly  available  data  with  respect  to  our  active  ingredient  in
our NDA submission to the FDA for marketing approval.

2

HT-TBI injection is being developed as a ready-to-inject autoinjector for intramuscular injection to be used in both traumatic brain injuries and ischemic
stroke. The same dose and formulation can be used across both TBI and stroke indications in age two years through adult. Our focus of development is
for point-of-care use in ambulatory and emergency room settings. HT-TBI’s active ingredient targets substance P/NK-1 pathway, identified as a leading
cause of post-brain injury inflammation and edema. Preclinical data has shown an NK-1 Antagonist significantly reduces brain edema and blood brain
barrier disruption post-TBI and post-stroke.

The BioLexa Platform

We have obtained an exclusive license from the University of Cincinnati to make, use, have made, import, offer for sale, and sell products based upon or
involving  the  use  of  (i)  topical  compositions  comprising  a  zinc  chelator  and  gentamicin  and  (ii)  zinc  chelators  to  inhibit  biofilm  formation  (the  “BioLexa
Platform” or “BioLexa”). The license enables us to develop the platform for any indications in humans. The BioLexa Platform is a proprietary, patented,
drug  compound  platform  for  the  treatment  of  eczema.  It  combines  an  FDA  approved  zinc  chelator  with  one  or  more  approved  antibiotics  in  a  topical
dosage  form  to  address  unchecked  eczema  flare-ups  by  preventing  the  formation  of  infectious  biofilms  and  the  resulting  clogging  of  sweat  ducts.  We
intend to develop the BioLexa Platform for use in patients following the Section  505(b)(2)  regulatory  pathway  of  the  FDA  rules.  Proceeding  under  this
regulatory pathway, we will be able to rely upon publicly available data with respect to gentamicin and the zinc chelator in our NDA submission to the
FDA for marketing approval.

In  December  2020,  we  received  approval  from  the  Belberry  Human  Research  Ethics  Committee  in  Australia  to  conduct  our  Phase  1b  clinical  trial  of
BioLexa, and we have engaged Novotech (Australia) Pty Limited as our local clinical research organization in Australia to provide clinical management,
data management, biostatistical, medical monitoring, pharmacovigilance, and other related services to support the first in human clinical trial of BioLexa.
Phase 1b of the trial was initiated in 2021 and final dosing of patients concluded in September 2022. At this time, we do not anticipate conducting any
further trials/studies in Australia.

We believe that the key elements for our market success with respect to BioLexa include:

●

●

the proprietary formulation of two FDA-approved drugs to treat bacterial proliferation which may reduce development time and costs by giving us
the ability to rely on safety and efficacy data from the two approved drugs;

our proprietary formulation is not a topical corticosteroid, and provides a novel mechanism of action and potentially a preferred safety profile as a
market differentiator; and

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
●

the  literature  set  forth  below  reaffirms  the  critical role  that S.  aureus  plays  in  the  development  of  atopic  dermatitis  flare-ups  within  the
international medical community, supporting the targeted mechanism of action of BioLexa.

Shi et al, “MRSA Colonization is Associated with Decreased Skin Commensal Bacteria in Atopic Dermatitis,” Invest Dermatol. 2018.

Blicharz, et al, “Staphylococcus aureus: an underestimated factor in the pathogenesis of atopic dermatitis?,” Adv Dermatol Allergol 2019.

Preclinical Development

HT-003

On  July  30,  2020  (the  “Isoprene  Effective  Date”),  we  entered  into  a  Sublicense  Agreement  (the  “Isoprene  Sublicense  Agreement”)  with  Isoprene
Pharmaceuticals, Inc. (“Isoprene”) pursuant to the commercial evaluation sublicense and option agreement dated March 8, 2019 by and among us, the
University of Maryland, Baltimore and Isoprene. Pursuant to the Isoprene Sublicense Agreement, Isoprene granted us an exclusive sublicense to certain
intellectual  property  (i)  to  make,  have  made,  use,  sell,  offer  to  sell  and  import  certain  licensed  products,  (ii)  in  connection  therewith,  to  use  certain
inventions and licensed materials and (iii) to practice certain patent rights for the treatment of dermatological conditions or diseases, referred to as HT-
003.

3

Retinoids,  which  include  Vitamin  A  (retinol)  and  its  analogues  (both  synthetic  and  metabolites),  play  a  critical  role  in  cell  signaling  and  biological
processes, including regulation of immune cells and inflammation, signaling pathways that control normal skin maintenance, embryonic development and
cell  growth/differentiation/repair.  Deficiencies  in  retinoids  and  their  active  metabolites  have  been  implicated  in  a  wide  variety  of  diseases.  In  the  skin,
retinol deficiency leads to hyperkeratosis and keratinizing metaplasia that is observed in skin disorders like psoriasis and acne. Vitamin A and retinoic acid
also play a crucial role in regulating cell proliferation, differentiation, and apoptosis and therefore, altered metabolism of retinoids has been suspected as
playing  a  potential  role  in  tumorigenesis.  Accordingly,  retinoids  have  been  approved  in  the  U.S.  for  treatment  of  acne  and  psoriasis  as  well  as  other
therapeutic indications such as acute promyelocytic leukemia and cutaneous T-cell lymphoma; however, the therapeutic use of exogenous retinoids has
been limited due to negative effects associated with high systemic concentrations. A new therapeutic approach to increase intracellular retinoic acid (the
active metabolite of retinol) potentially without causing negative side effects of exogenous retinoic acid is to use inhibitors of RAMBAs, which prolong the
presence of retinoic acid. HT-003 is a novel RAMBA under investigation for topical treatment in acne and psoriasis applications.

In December 2019, we entered into a research collaboration agreement with Weill Cornell Medicine for the completion of pre-clinical studies investigating
the mechanism of action of HT-003 that was renewed in January 2021 as a result of positive preclinical results. Dr. Jonathan Zippin, M.D., Ph.D., FAAD,
Associate Professor of Dermatology at Weill Cornell Medicine and our Senior Scientific Advisor, is the principal investigator for such pre-clinical studies.

The retinoic acid metabolism blocking agents (“RAMBAs”) have the potential to be developed as a platform for multiple inflammatory-based indications.
Accordingly,  we  entered  into  a  Sublicense  Agreement  with  Isoprene  on  July  2,  2021  pursuant  to  the  option  agreement  dated  December  22,  2020  to
expand  the  therapeutic  indication  of  the  sublicensed  RAMBAs  from  Isoprene  to  include  inflammatory  bowel  diseases,  including  Crohn’s  disease  and
ulcerative  colitis.  Preclinical  proof-of-concept  studies  were  conducted  in  2021  for  the  investigation  of  RAMBAs  for  treatment  of  inflammatory  bowel
diseases, including Crohn’s disease and ulcerative colitis.

HT-004

On November 20, 2019, we entered into a license agreement with NC State pursuant to which NC State granted us an exclusive license to, among other
things, develop, make, use, offer and sell certain licensed products throughout the world with respect to HT-004 for treating allergic diseases. HT-004 is a
potential disease-modifying agent that uses exon-skipping oligonucleotide-targeted methods to reduce mast cell responses to immunoglobulin E (IgE)-
directed  antigens,  which  is  one  of  the  key  mechanisms  in  the  pathophysiology  of  asthma,  atopic  dermatitis  and  other  allergic  diseases.  HT-004  is
currently under investigation for the treatment of asthma and allergies using inhalational administration.

In  December  2019,  we  entered  a  sponsored  research  agreement  with  NC  State  for  proof  of  principle  in  targeting  allergic  inflammation  in  the  airways.
Preclinical  proof-of-concept  data  was  generated  in  October  2020  supporting  efficacy  of  HT-004  after  inhalational  delivery  in  a  mouse  model.  Critical
proof-of-concept studies in a humanized mouse model are planned to be initiated in 2022 and was completed in 2023.

We believe that the key elements for our market success with respect to HT-004 include:

●

●

To our knowledge, there are currently no disease-modifying agents for asthma or allergy diseases;

The  active  pharmaceutical  ingredient  in  HT-004  is  a  novel  molecular  class  that  we  believe  would  prevent  generic  competition  after
commercialization;

● HT-004 is being developed for inhalational administration by either inhaler or nebulizer for easy access at home by patients; and

● HT-004 is applicable for both adult and pediatric patient populations with asthma and/or allergies.

4

HT-002

On May 18, 2020, we entered into an Exclusive License Agreement with the Virginia Commonwealth University Intellectual Property Foundation (“VCU”)
pursuant to which VCU granted us an exclusive, royalty bearing license to HT-002, a novel peptide developed by researchers at VCU that may be used to
slow  the  transmission  of  SARS-CoV-2  (the  “VCU  Peptide”)  and  a  non-exclusive  royalty  bearing,  worldwide  license  with  respect  to  certain  licensed
technical information patents to make, have made, use, offer to sell, sell and import certain licensed products and perform certain licensed services. On
June 29, 2020, we entered into a Sponsored Project Agreement (“VCU SPA”) with VCU for the development of a potential COVID-19 treatment using the
VCU Peptide. The VCU SPA was amended on April 28, 2021 to extend the period of research and to add additional scope of investigation to include the

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
variants of SARS-CoV-2. Proof-of-Concept preclinical studies were completed in 2022.

Direct Detect Breath Diagnostic Device

On  August  7,  2020,  we  entered  into  a  Patent  License  Agreement  (“GW  Patent  License  Agreement”)  with  GW  pursuant  to  which  GW  granted  us  an
exclusive,  worldwide,  royalty  bearing  license  to  certain  intellectual  property  that  can  be  used  to  develop  a  device  designed  to  detect  the  presence  of
viruses. Specifically, the GW Patent License Agreement permits us to make, have made, use, import, offer for sale and sell certain licensed products in
the field of virus sensing and detection. We have engaged a company to develop a platform prototype and, once developed, we will select target analytes
for further development.

Product Development Pipeline

The following table summarizes our product development pipeline.

Other Interests

We have interests in certain other assets being developed by third parties. Specifically, in December 2021, we entered into a license agreement with Zylö
Therapeutics,  Inc.  (“Zylö”)  with  respect  to  the  development  of  HT-005.  We  had  previously  entered  into  a  sublicense  agreement  with  Zylö  pursuant  to
which we had advanced the development of HT-005 for patients with lupus. (See Note 6 to the consolidated financial statements for a discussion of our
agreement  with  Zylö).  In  addition,  in  March  2020,  we  entered  into  a  Royalty  and  Development  Agreement  (the  “Voltron  Agreement”)  with  Voltron
Therapeutics,  Inc.  (“Voltron”)  with  respect  to  the  development  of  potential  product  candidates  for  the  prevention  of  COVID-19.  (See  Note  6  to  the
consolidated financial statements for a discussion of our agreement with Voltron).

Competition

The biopharmaceutical industry utilizes rapidly advancing technologies and is characterized by intense competition. There is also a strong emphasis on
intellectual  property  and  proprietary  products.  In  the  segment  of  the  biopharmaceutical  industry,  competition  from  different  sources  including  major
biopharmaceutical  companies,  academic  institutions,  government  agencies,  and  public  and  private  research  institutions  will  continue.  Many  of  our
competitors  have  significantly  greater  financial  resources  and  expertise  in  product  candidate  development  and  may  have  progressed  further  toward
approval  and  marketing.  In  addition,  smaller  or  early-stage  companies  may  also  prove  to  be  significant  competitors,  particularly  through  collaborative
arrangements with large and established companies.

5

Manufacturing and Supply

We do not have any manufacturing capability and therefore we currently rely on and intend to continue to rely on contract manufacturing organizations to
produce our product candidates in accordance with regulatory requirements.

Commercialization

Our success depends not only on the successful development and approval of our products candidates but also on the commercialization of our potential
products. If and when our product candidates receive regulatory approval, we intend to engage third-parties such as pharmaceutical and biotechnology
companies for the commercialization of our products.

Intellectual Property Portfolio

Our  goal  is  to  obtain,  maintain  and  enforce  patent  protection  for  our  products,  formulations,  processes,  methods  and  other  proprietary  technologies,
preserve our trade secrets, and operate without infringing on the proprietary rights of other parties, both in the U.S. and in other countries. Our policy is to
actively  seek  the  broadest  intellectual  property  protection  possible  for  our  products,  proprietary  information  and  proprietary  technology  through  a
combination of contractual arrangements and patents, both in the U.S. and elsewhere in the world. In addition, we intend to actively pursue product life-
cycle management initiatives to extend our market exclusivity.

We  intend  to  cement  our  market  exclusivity  in  conjunction  with  our  formulation-development  partners  through  additional  patents  based  on  the
pharmaceutical and clinical characteristics of our product candidates in the proprietary formulation and through the introduction of line extensions such as
combination drugs and new formulations.

In addition to any granted patents, our products may be eligible for market exclusivity to run concurrently with the term of the patent for three and a half
years  in  the  U.S.  pursuant  to  the  Hatch-Waxman  Act  and  pediatric  exclusivity  guideline  and  up  to  ten  years  of  market  exclusivity  in  the  E.U.  which
includes  eight  years  of  data  exclusivity  and  two  years  of  market  exclusivity  from  the  date  we  file  an  NDA  or  the  European  equivalent  referred  to  as
Marketing Authorization Application.

We  currently  have  licenses  to  six  U.S.  patents  and  one  pending  U.S.  patent  application,  and  we  have  licenses  to  three  patents  issued  in  Europe  and

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
  
 
 
 
 
Australia and five pending patent applications in foreign jurisdictions including Europe, Brazil, Canada and Hong Kong. Hoth also holds two pending U.S.
patent applications, one European application and one pending PCT patent application.

In addition to patents, we rely on trade secrets and know-how and continuing technological innovation to develop and maintain our competitive position.
However, trade secrets and know-how can be difficult to protect. We take measures to protect and maintain the confidentiality of proprietary information in
order to protect aspects of the business that are not amenable to, or that we do not consider appropriate for, patent protection. We require employees,
consultants,  outside  scientific  partners,  sponsored  researchers  and  other  advisors  to  execute  confidentiality  agreements  with  us  on  or  prior  to  the
commencement of employment or consulting relationships with us.

Government Regulations

Governmental  authorities  in  the  U.S.  and  other  countries  extensively  regulate  the  research,  development,  testing,  manufacture,  labeling,  promotion,
advertising, distribution and marketing of pharmaceutical products, including biological products, and medical devices, such as those being developed by
us.  In  the  U.S.,  the  FDA  regulates  such  products  under  the  FDCA  and  the  Public  Health  Services  Act  and  implements  related  regulations.  Failure  to
comply  with  applicable  FDA  requirements,  both  before  and  after  approval,  may  subject  us  to  administrative  and  judicial  sanctions,  such  as  a  delay  in
approving  or  refusal  by  the  FDA  to  approve  pending  applications,  warning  letters,  product  recalls,  product  seizures,  total  or  partial  suspension  of
production or distribution, injunctions and/or criminal prosecution.

6

U.S. Food and Drug Administration Regulations

United States Drug Development

In the United States, the FDA regulates drugs (including biological products, such as vaccines), medical devices and combinations of drugs and devices,
or combination products, under the FDCA and its implementing regulations. These products are also subject to other federal, state and local statutes and
regulations. The process of obtaining regulatory approvals and the subsequent compliance with appropriate federal, state, local and foreign statutes and
regulations  requires  the  expenditure  of  substantial  time  and  financial  resources.  Failure  to  comply  with  the  applicable  U.S.  requirements  at  any  time
during  the  product  development  process,  approval  process  or  after  approval,  may  subject  an  applicant  to  administrative  or  judicial  sanctions.  These
sanctions could include, among other actions, the FDA’s refusal to approve pending applications, withdrawal of an approval, a clinical hold, untitled or
warning  letters,  requests  for  voluntary  product  recalls  or  withdrawals  from  the  market,  product  seizures,  total  or  partial  suspension  of  production  or
distribution injunctions, fines, refusals of government contracts, restitution, disgorgement, or civil or criminal penalties. Any agency or judicial enforcement
action could have a material adverse effect on us.

The process required by the FDA before a drug may be marketed in the United States generally involves the following:

●

●

●

●

●

●

●

completion of extensive pre-clinical laboratory tests, animal studies and formulation studies in accordance with applicable regulations, including
the FDA’s Good Laboratory Practice regulations;

submission to the FDA of an IND, which must become effective before human clinical trials may begin;

performance  of  adequate  and  well-controlled  human  clinical  trials  in  accordance  with  an  applicable  IND  and  other  clinical  study  related
regulations, referred to as good clinical practice (“GCP”), to establish the safety and efficacy of the proposed drug for its proposed indication;

submission to the FDA of an NDA or biologics license application (“BLA”);

satisfactory completion of an FDA pre-approval inspection of the manufacturing facility or facilities at which the product, or components thereof,
are produced to assess compliance with the FDA’s current good manufacturing practice (“cGMP”) requirements;

potential FDA audit of the clinical trial sites that generated the data in support of the NDA or BLA; and

FDA review and approval of the NDA or BLA prior to any commercial marketing or sale.

Human clinical trials are typically conducted in three sequential phases that may overlap or be combined:

● Phase 1. The product is initially introduced into a small number of healthy human subjects or patients and tested for safety, dosage tolerance,
absorption,  metabolism,  distribution  and  excretion  and,  if  possible,  to  gain  early  evidence  on  effectiveness.  In  the  case  of  some  products  for
severe or life-threatening diseases, especially when the product is suspected or known to be unavoidably toxic, the initial human testing may be
conducted in patients.

● Phase 2. Involves clinical trials in a limited patient population to identify possible adverse effects and safety risks, to preliminarily evaluate the

efficacy of the product for specific targeted diseases and to determine dosage tolerance and optimal dosage and schedule.

● Phase 3. Clinical trials are undertaken to further evaluate dosage, clinical efficacy and safety in an expanded patient population at geographically
dispersed  clinical  trial  sites.  These  clinical  trials  are  intended  to  establish  the  overall  risk/benefit  relationship  of  the  product  and  provide  an
adequate basis for product labeling.

Post-approval trials, sometimes referred to as Phase 4 clinical trials, may be conducted after initial marketing approval. These studies are used to gain
additional experience from the treatment of patients in the intended therapeutic indication. In certain instances, the FDA may mandate the performance of
Phase  4  trials.  Phase  1,  Phase  2  and  Phase  3  clinical  trials  may  not  be  completed  successfully  within  any  specified  period,  if  at  all.  The  FDA  or  the
clinical trial sponsor may suspend or terminate a clinical trial at any time on various grounds, including a finding that the research subjects or patients are
being exposed to an unacceptable health risk. Similarly, an Institutional Review Board (“IRB”), which oversees the conduct of clinical trials, can suspend
or terminate approval of a clinical trial at its institution if the clinical trial is not being conducted in accordance with the IRB’s requirements or if the product
has  been  associated  with  unexpected  serious  harm  to  patients.  Additionally,  some  clinical  trials  are  overseen  by  an  independent  group  of  qualified
experts organized by the clinical trial sponsor, known as a data safety monitoring board or committee. This group provides authorization for whether a
trial  may  move  forward  at  designated  check  points  based  on  access  to  certain  data  from  the  study.  The  clinical  trial  sponsor  may  also  suspend  or
terminate a clinical trial based on evolving business objectives and/or competitive climate.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
7

FDA Review Process

The  results  of  product  development,  pre-clinical  studies  and  clinical  trials,  along  with  descriptions  of  the  manufacturing  process,  analytical  tests
conducted  on  the  drug,  proposed  labeling  and  other  relevant  information,  are  submitted  to  the  FDA  as  part  of  an  NDA  for  a  new  drug,  or  BLA  for  a
biological product, requesting approval to market the product. The submission of an NDA or BLA is subject to the payment of a substantial user fee, and
the sponsor of an approved NDA or BLA is also subject to an annual program user fee; although a waiver of such fee may be obtained under certain
limited circumstances.

The  FDA  reviews  all  NDAs  submitted  before  it  accepts  them  for  filing  and  may  request  additional  information  rather  than  accepting  an  NDA  for  filing.
Under  the  goals  and  policies  agreed  to  by  the  FDA  under  the  Prescription  Drug  User  Fee  Act  (“PDUFA”),  the  FDA’s  goal  to  complete  its  substantive
review of a standard NDA and respond to the applicant is ten months from the receipt of the NDA. The FDA does not always meet its PDUFA goal dates,
and  the  review  process  is  often  significantly  extended  by  FDA  requests  for  additional  information  or  clarification  and  may  go  through  multiple  review
cycles.

The review and evaluation of an NDA or BLA by the FDA is extensive and time consuming and may take longer than originally planned to complete, and
we may not receive a timely approval, if at all.

Before approving an NDA, the FDA will conduct a pre-approval inspection of the manufacturing facilities for the new product to determine whether they
comply with cGMPs. The FDA will not approve the product unless it determines that the manufacturing processes and facilities are in compliance with
cGMP requirements and adequate to assure consistent production of the product within required specifications. In addition, before approving an NDA, the
FDA may also audit data from clinical trials to ensure compliance with GCP requirements.

There is no assurance that the FDA will ultimately approve a product for marketing in the United States, and we may encounter significant difficulties or
costs during the review process. If a product receives marketing approval, the approval may be significantly limited to specific diseases and dosages or
the  indications  for  use  may  otherwise  be  limited,  which  could  restrict  the  commercial  value  of  the  product.  Further,  the  FDA  may  require  that  certain
contraindications, warnings or precautions be included in the product labeling or may condition the approval of the NDA or BLA on other changes to the
proposed labeling, development of adequate controls and specifications, or a commitment to conduct post-market testing or clinical trials and surveillance
to monitor the effects of approved products. For example, the FDA may require Phase 4 clinical trials to further assess drug safety and effectiveness and
may require testing and surveillance programs to monitor the safety of approved products that have been commercialized. The FDA may also place other
conditions on approvals, including the requirement for a risk evaluation and mitigation strategy (“REMS”), to assure the safe use of the drug.

Section 505(b)(2) Regulatory Approval Pathway

Section 505(b)(2) of the FDCA provides an alternate regulatory pathway for approval of a new drug by allowing the FDA to rely on data not developed by
the applicant. Specifically, Section 505(b)(2) permits the submission of an NDA where one or more of the investigations relied upon by the applicant for
approval  was  not  conducted  by  or  for  the  applicant  and  for  which  the  applicant  has  not  obtained  a  right  of  reference.  The  applicant  may  rely  upon
published literature and/or the FDA’s findings of safety and effectiveness for an approved drug already on the market. Approval or submission of a 505(b)
(2) application, like those for abbreviated new drugs (“ANDAs”), may be delayed because of patent and/or exclusivity rights that apply to the previously
approved drug.

8

A 505(b)(2) application may be submitted for a new chemical entity (“NCE”) when some part of the data necessary for approval is derived from studies
not conducted by or for the applicant and when the applicant has not obtained a right of reference.

Section  505(b)(2)  applications  also  may  be  entitled  to  marketing  exclusivity  if  supported  by  appropriate  data  and  information.  Three-year  new  data
exclusivity  may  be  granted  to  the  505(b)(2)  application  if  one  or  more  clinical  investigations  conducted  in  support  of  the  application,  other  than
bioavailability/bioequivalence studies, were essential to the approval and conducted or sponsored by the applicant. Five years of marketing exclusivity
may be granted if the application is for an NCE, and pediatric exclusivity is likewise available.

Orange Book Listing and Paragraph IV Certification

For  NDA  submissions,  including  those  under  Section  505(b)(2),  applicants  are  required  to  list  with  the  FDA  certain  patents  with  claims  that  cover  the
applicant’s  product.  Upon  approval,  each  of  the  patents  listed  in  the  application  is  published  in Approved Drug Products with Therapeutic Equivalence
Evaluations, commonly referred to as the Orange Book. Any applicant who subsequently files an ANDA or 505(b)(2) NDA that references a drug listed in
the Orange Book must certify to the FDA that (1) no patent information on the drug product that is the subject of the application has been submitted to the
FDA; (2) such patent has expired; (3) the date on which such patent expires; or (4) such patent is invalid or will not be infringed upon by the manufacture,
use or sale of the drug product for which the application is submitted. This last certification is known as a Paragraph IV Certification.

If an applicant has provided a Paragraph IV Certification to the FDA, the applicant must also send notice of the Paragraph IV Certification to the holder of
the NDA for the approved drug and the patent owner once the application has been accepted for filing by the FDA. The NDA holder or patent owner may
then initiate a patent infringement lawsuit in response to notice of the Paragraph IV Certification. The filing of a patent infringement lawsuit within 45 days
of the receipt of a Paragraph IV Certification prevents the FDA from approving the ANDA or 505(b)(2) application until the earlier of 30 months from the
date of the lawsuit, the applicant’s successful defense of the suit, or expiration of the patent.

United States Medical Device Regulation

Medical devices, including diagnostic test devices, also are subject to extensive and rigorous regulation by the FDA under the FDCA, as well as other
federal and state regulatory bodies in the United States, and laws and regulations of foreign authorities in other countries. FDA requirements specific to
medical devices are wide ranging and govern, among other things, the design, development and manufacturing, human clinical trials, preclearance or
approval, advertising and promotion, and product import and export. Unless an exemption applies, medical devices distributed in the United States must
receive either premarket clearance under Section 510(k) of the FDCA or premarket approval of a premarket application (“PMA”). During the COVID-19
public  health  emergency,  the  FDA  had  authorized  COVID-19  diagnostic  tests  under  its  Emergency  Use  Authorization  (“EUA”)  authority;  however,  on

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
January  31,  2023,  President  Biden  issued  a  Statement  of  Administration  Policy  indicating  that  the  administration  intends  for  the  COVID-19  national
emergency and public health emergency to end on May 11, 2023. When the public health emergency ends, the FDA will continue to have the authority to
issue EUAs until that authority is formally terminated by the Secretary of HHS through a separate process. Medical devices are classified into one of three
classes-Class I, Class II, or Class III-depending on the degree or risk associated with each medical device and the extent of control needed to ensure
safety  and  effectiveness.  Medical  devices  deemed  to  pose  relatively  low  risk  are  placed  in  either  Class  I  or  II.  Class  II  devices  generally  require  the
manufacturer to submit a premarket notification under Section 510(k) of the FDCA requesting permission for commercial distribution. Devices deemed by
the FDA to pose the greatest risk, such as life-sustaining, life-supporting or implantable devices are placed in Class III requiring PMA approval.

9

Reimbursement

Potential sales of any of our product candidates, if approved, will depend, at least in part, on the extent to which such products will be covered by third-
party  payors,  such  as  government  health  care  programs,  commercial  insurance  and  managed  healthcare  organizations.  These  third-party  payors  are
increasingly limiting coverage and/or reducing reimbursements for medical products and services. A third-party payor’s decision to provide coverage for a
drug product does not imply that an adequate reimbursement rate will be approved. Further, one payor’s determination to provide coverage for a drug
product does not assure that other payors will also provide coverage for the drug product. In addition, the U.S. government, state legislatures and foreign
governments  have  continued  implementing  cost-containment  programs,  including  price  controls,  restrictions  on  reimbursement  and  requirements  for
substitution of generic products. Adoption of price controls and cost-containment measures, and adoption of more restrictive policies in jurisdictions with
existing controls and measures, could further limit our future revenues and results of operations. Decreases in third-party reimbursement or a decision by
a  third-party  payor  to  not  cover  a  product  candidate,  if  approved,  or  any  future  approved  products  could  reduce  physician  usage  of  our  products,  and
have a material adverse effect on our sales, results of operations and financial condition.

In the United States, the Medicare Part D program provides a voluntary outpatient drug benefit to Medicare beneficiaries for certain products. We do not
know  whether  our  product  candidates,  if  approved,  will  be  eligible  for  coverage  under  Medicare  Part  D,  but  individual  Medicare  Part  D  plans  offer
coverage subject to various factors such as those described above. Furthermore, private payors often follow Medicare coverage policies and payment
limitations in setting their own coverage policies.

 Orphan Drug Designation

Under the Orphan Drug Act, the FDA may grant orphan designation to a drug or biologic intended to treat a rare disease or condition, which is a disease
or condition that affects fewer than 200,000 individuals in the United States, or more than 200,000 individuals in the United States for which there is no
reasonable expectation that the cost of developing and making available in the United States a drug or biologic for this type of disease or condition will be
recovered from sales in the United States for that drug or biologic. Orphan drug designation must be requested before submitting an NDA or BLA. After
the FDA grants orphan drug designation, the generic identity of the therapeutic agent and its potential orphan use are disclosed publicly by the FDA. The
orphan drug designation does not convey any advantage in, or shorten the duration of, the regulatory review or approval process.

If a product that has orphan drug designation subsequently receives the first FDA approval for the disease for which it has such designation, the product
is entitled to orphan drug exclusive approval (or exclusivity), which means that the FDA may not approve any other applications, including a full NDA or
BLA, to market the same drug for the same indication for seven years, except in limited circumstances, such as a showing of clinical superiority to the
product with orphan drug exclusivity. Orphan drug exclusivity does not prevent the FDA from approving a different drug or biologic for the same disease
or condition, or  the  same  drug  or  biologic  for  a  different  disease  or  condition.  Among  the  other  benefits  of  orphan  drug  designation  are  tax  credits  for
certain research and a waiver of the application user fee.

A  designated  orphan  drug  may  not  receive  orphan  drug  exclusivity  if  it  is  approved  for  a  use  that  is  broader  than  the  indication  for  which  it  received
orphan designation. In addition, exclusive marketing rights in the United States may be lost if the FDA later determines that the request for designation
was materially defective or if the manufacturer is unable to assure sufficient quantities of the product to meet the needs of patients with the rare disease
or condition.

Healthcare Laws and Regulations

Sales of our product candidates, if approved, or any other future product candidate will be subject to healthcare regulation and enforcement by the federal
government and the states and foreign governments in which we might conduct our business. The healthcare laws and regulations that may affect our
ability to operate include the following:

●

●

The federal Anti-Kickback Statute makes it illegal for any person or entity to knowingly and willfully, directly or indirectly, solicit, receive, offer, or
pay any remuneration that is in exchange for or to induce the referral of business, including the purchase, order, lease of any good, facility, item
or service for which payment may be made under a federal healthcare program, such as Medicare or Medicaid. The term “remuneration” has
been broadly interpreted to include anything of value.

Federal false claims and false statement laws, including the federal civil False Claims Act, prohibits, among other things, any person or entity
from  knowingly  presenting,  or  causing  to  be  presented,  for  payment  to,  or  approval  by,  federal  programs,  including  Medicare  and  Medicaid,
claims for items or services, including drugs, that are false or fraudulent.

● Health  Insurance  Portability  and  Accountability  Act  of  1996  (“HIPAA”)  created  additional  federal  criminal  statutes  that  prohibit  among  other
actions, knowingly and willfully executing, or attempting to execute, a scheme to defraud any healthcare benefit program, including private third-
party payors or making any false, fictitious or fraudulent statement in connection with the delivery of or payment for healthcare benefits, items or
services.

10

● HIPAA,  as  amended  by  the  Health  Information  Technology  for  Economic  and  Clinical  Health  Act  of  2009  and  their  implementing  regulations,
impose  obligations  on  certain  types  of  individuals  and  entities  regarding  the  electronic  exchange  of  information  in  common  healthcare
transactions, as well as standards relating to the privacy and security of individually identifiable health information.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
●

The  federal  Physician  Payments  Sunshine  Act  requires  certain  manufacturers  of  drugs,  devices,  biologics  and  medical  supplies  for  which
payment is available under Medicare, Medicaid or the Children’s Health Insurance Program, with specific exceptions, to report annually to the
Centers for Medicare & Medicaid Services information related to payments or other transfers of value made to physicians and teaching hospitals,
as well as ownership and investment interests held by physicians and their immediate family members.

Also, many states have similar laws and regulations, such as anti-kickback and false claims laws that may be broader in scope and may apply regardless
of  payor,  in  addition  to  items  and  services  reimbursed  under  Medicaid  and  other  state  programs.  Additionally,  we  may  be  subject  to  state  laws  that
require pharmaceutical companies to comply with the federal government’s and/or pharmaceutical industry’s voluntary compliance guidelines, state laws
that require drug manufacturers to report information related to payments and other transfers of value to physicians and other healthcare providers or
marketing expenditures, as well as state and foreign laws governing the privacy and security of health information, many of which differ from each other in
significant ways and often are not preempted by HIPAA.

Additionally, to the extent that our product is sold in a foreign country, we may be subject to similar foreign laws.

Employees

As  of  March  17,  2023,  we  employed  a  total  of  2  full-time  employees,  3  employee  consultants,  and  1  part-time  employee.  We  are  not  a  party  to  any
collective bargaining agreements. We believe that we maintain good relations with our employees.

Our Corporate Information and History

We were incorporated as a Nevada corporation on May 16, 2017. On  October 20, 2022, we filed a Certificate of Change with the Nevada Secretary of
State to effectuate a 1-for-25 reverse stock split of our issued and outstanding and authorized shares of common stock. The reverse stock split became
effective  on  October  26,  2022. All  share  data,  per  share  data  and  related  information  contained  in  this  Annual  Report  on  Form  10-K  has  been
retrospectively  adjusted  to  reflect  the  effect  of  the  reverse  stock  split.   On  November  2,  2022,  we  filed  a  Certificate  of  Designation  of  the  Series  B
Preferred Stock (the “Certificate of Designation”) with the Secretary of State of the State of Nevada to create a new class of Series B Preferred Stock, par
value $0.0001 per share (“Series B Preferred Stock”), designating 2,000,000 shares of our authorized preferred stock as Series B Preferred Stock. On
November 2, 2022, we also entered into a Subscription and Investment Representation Agreement with an investor pursuant to which we issued and sold
2,000,000 shares of our newly designated Series B Preferred Stock to such investor for an aggregate purchase price of $1,000. The Series B Preferred
Stock  were  not  entitled  to  receive  dividends  or  any  other  distributions.  The  Series  B  Preferred  Stock  were  entitled  to  ten  votes  per  share  and  voted
together  with  the  issued  and  outstanding  shares  of  our  common  stock  as  a  single  class  exclusively  with  respect  to  the  Authorized  Stock  Increase  (as
defined in the Certificate of Designation). The Series B Preferred Stock had no rights as to any distribution or assets of our Company upon a liquidation,
bankruptcy, reorganization, merger, acquisition, sale, dissolution or winding up of our Company. The 2,000,000 outstanding shares of Series B Preferred
Stock were redeemed for an aggregate price of $10 on December 13, 2022 in connection with the filing of the Amendment (as defined herein) with the
Secretary  of  State  of  the  State  of  Nevada.  Pursuant  to  the  Certificate  of  Designation, the  shares  of  Series  B  Preferred  Stock  redeemed  by  us  were
automatically retired and restored to the status of an authorized but unissued share of preferred stock.

On December 13, 2022, we filed a Certificate of Amendment (the “Amendment”) to our Articles of Incorporation, as amended, to increase our authorized
shares of common stock from 3,000,000 shares to 50,000,000 shares.

Our principal executive offices are located at 1 Rockefeller Plaza, Suite 1039, New York, New York 10020 and our telephone number is (646) 756-2997.

11

Available Information

Our website address is www.hoththerapeutics.com. The contents of, or information accessible through, our website are not part of this Annual Report on
Form 10-K, and our website address is included in this document as an inactive textual reference only. We make our filings with the U.S. Securities and
Exchange  Commission  (“SEC”),  including  our  Annual  Report  on  Form  10-K,  Quarterly  Reports  on  Form  10-Q,  Current  Reports  on  Form  8-K  and  all
amendments to those reports, available free of charge on our website as soon as reasonably practicable after we file such reports with, or furnish such
reports  to,  the  SEC.  The  public  may  read  and  copy  the  materials  we  file  with  the  SEC  at  the  SEC’s  Public  Reference  Room  at  100  F  Street,  NE,
Washington,  DC  20549.  The  public  may  obtain  information  on  the  operation  of  the  Public  Reference  Room  by  calling  the  SEC  at  1-800-SEC-0330.
Additionally, the SEC maintains an internet site that contains reports, proxy and information statements and other information. The address of the SEC’s
website is www.sec.gov. The information contained in the SEC’s website is not intended to be a part of this filing.

ITEM 1A. RISK FACTORS

An investment in our common stock involves a high degree of risk. You should carefully consider the following risk factors and the other information in
this Annual Report on Form 10-K before investing in our common stock. Our business and results of operations could be seriously harmed by any of the
following risks. The risks set out below are not the only risks we face. Additional risks and uncertainties not currently known to us or that we currently
deem to be immaterial also may materially adversely affect our business, financial condition and/or operating results. If any of the following events occur,
our business, financial condition and results of operations could be materially adversely affected. In such case, the value and trading price of our common
stock could decline, and you may lose all or part of your investment.

Risks Related to Our Financial Position and Need for Capital

We have generated no revenue from commercial sales to date and our future profitability is uncertain.

We were incorporated in May 2017 and have a limited operating history and our business is subject to all of the risks inherent in the establishment of a
new  business  enterprise.  Our  likelihood  of  success  must  be  considered  in  light  of  the  problems,  expenses,  difficulties,  complications  and  delays
frequently  encountered  in  connection  with  development  and  expansion  of  a  new  business  enterprise.  Since  inception,  we  have  incurred  losses  and
expect to continue to operate at a net loss for at least the next several years as we commence our research and development efforts, conduct clinical
trials and develop manufacturing, sales, marketing and distribution capabilities. Our net losses for the years ended December 31, 2022 and 2021 were
$11,371,953  and  $14,313,705,  respectively,  and  our  accumulated  deficit  as  of  December  31,  2022  and  2021  was  $45,099,116  and  $33,727,163,
respectively. There can be no assurance that the products under development by us will be approved for sale in the U.S. or elsewhere. Furthermore,
there can be no assurance that if such products are approved they will be successfully commercialized, and the extent of our future losses and the timing
of our profitability are highly uncertain. If we are unable to achieve profitability, we may be unable to continue our operations.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
12

If we fail to obtain the capital necessary to fund our operations, we will be unable to continue or complete our product development and you
will likely lose your entire investment.

We will need to continue to seek capital from time to time to continue development of our product candidates. We cannot provide any assurances that any
revenues that we may generate in the future will be sufficient to fund our ongoing operations. We believe that we will need to raise substantial additional
capital to fund our operations and the development and commercialization of our product candidates.

Our business or operations may change in a manner that may consume available funds more rapidly than anticipated and substantial additional funding
may  be  required  to  maintain  operations,  fund  expansion,  commercialize  our  product  candidates,  develop  new  or  enhanced  products,  acquire
complementary products, business or technologies or otherwise respond to competitive pressures and opportunities, such as a change in the regulatory
environment or a change in preferred treatment modalities. In addition, we may need to accelerate the growth of our sales capabilities and distribution
beyond what is currently envisioned, and this would require additional capital. However, we may not be able to secure funding on favorable terms, if at all.

If  we  cannot  raise  adequate  funds  to  satisfy  our  capital  requirements,  we  may  have  to  delay,  scale  back  or  eliminate  our  research  and  development
activities,  clinical  studies  or  operations.  We  may  also  be  required  to  obtain  funds  through  arrangements  with  collaborators,  which  arrangements  may
require us to relinquish rights to certain intellectual property, technologies or products that we otherwise would not consider relinquishing, including rights
to future product candidates or certain major geographic markets. This could result in sharing revenues which we might otherwise retain for ourselves.
Any of these actions may harm our business, financial condition and results of operations.

The  amount  of  capital  we  may  need  depends  on  many  factors,  including  the  progress,  timing  and  scope  of  our  product  development  programs;  the
progress, timing and scope of our pre-clinical studies and clinical trials; the time and cost necessary to obtain regulatory approvals; the time and cost
necessary  to  further  develop  manufacturing  processes  and  arrange  for  contract  manufacturing;  our  ability  to  enter  into  and  maintain  collaborative,
licensing  and  other  commercial  relationships;  and  our  partners’  commitment  of  time  and  resources  to  the  development  and  commercialization  of  our
products.

Even if we can raise additional funding, we may be required to do so on terms that are dilutive to you.

The capital markets have been unpredictable in the recent past for unprofitable companies such as ours. The amount of capital that a company such as
ours is able to raise often depends on variables that are beyond our control. As a result, we may not be able to secure financing on terms attractive to us,
or at all. If we are able to consummate a financing arrangement, the amount raised may not be sufficient to meet our future needs. If adequate funds are
not  available  on  acceptable  terms,  or  at  all,  our  business,  including  our  results  of  operations,  financial  condition  and  our  continued  viability  will  be
materially adversely affected.

Risks Related to Product Development, Regulatory Approval, Manufacturing and Commercialization

We  are  dependent  upon  the  clinical  success  of  our  licensed  products  and  technologies.  If  we  are  unable  to  generate  revenues  from  our
licensed products and technologies, our ability to create shareholder value may be limited.

We do not currently generate revenues from any of our product candidates, and we may not be successful in obtaining regulatory approvals to commence
our  clinical  trials.  If  we  do  not  obtain  such  approvals,  the  time  in  which  we  expect  to  commence  clinical  programs  for  our  product  candidates  will  be
extended and such extension may increase our expenses and our need for additional capital. Moreover, there is no guarantee that our clinical trials will be
successful or that we will continue clinical development in support of an approval from the regulatory agencies for any indication. We note that most drug
candidates never reach the clinical stage and even those that do commence clinical development have only a small chance of successfully completing
clinical  development  and  gaining  regulatory  approval.  Therefore,  our  business  currently  depends  entirely  on  the  successful  development,  regulatory
approval and commercialization of our product candidates, which may never occur.

13

Although we have entered into the Voltron Agreement pursuant to which we and HaloVax intend to jointly develop products to prevent COVID-
19,  no  assurance  can  be  given  as  to  when,  if  ever,  we  will  be  able  to  develop  any  products  for  such  purpose  and  if  developed  that  such
products will be successfully commercialized.

In March 2020, we entered into the Voltron Agreement pursuant to which we and HaloVax will work to jointly develop potential products candidates to
prevent COVID-19; however, no assurance can be given as to when, if ever, we will be able to develop any products for such purpose. Furthermore, we
are subject to risks including, but not limited to, the following with respect to the development of a treatment for COVID-19:

●

the EUA marketing approval processes of the FDA are lengthy, time consuming and inherently unpredictable, and we cannot guarantee that we
will ever have a marketable product

● we may encounter substantial delays in completing our clinical studies which in turn will require additional costs, or we may fail to demonstrate

adequate safety and efficacy to the satisfaction of applicable regulatory authorities;

●

●

conducting successful clinical studies may require the enrollment of large numbers of patients, and suitable patients may be difficult to identify
and recruit;

to be commercially successful, physicians must be persuaded that using our products are effective alternatives to other existing therapies and
treatments;

● we may depend on third parties for manufacturing our proposed product candidates and any conflicts with such partners could delay or prevent

the development or commercialization of such product candidates;

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
●

●

●

if third-party contract manufacturers upon whom we rely to formulate and manufacture our product candidates do not perform, fail to manufacture
according to our specifications or fail to comply with strict regulations, our clinical studies could be adversely affected and the development of our
product candidates could be delayed or terminated or we could incur significant additional expenses;

adverse events involving our products may lead the FDA to delay or deny clearance for our products or result in product recalls that could harm
our reputation, business and financial results; and

if  we  fail  to  comply  with  healthcare  regulations,  we  could  face  substantial  enforcement  actions,  including  civil  and  criminal  penalties  and  our
business, operations and financial condition could be adversely affected.

In addition to the foregoing, on January 31, 2023, President Biden issued a Statement of Administration Policy indicating that the administration intends
for the COVID-19 national emergency and public health emergency to end on May 11, 2023. EUAs are issued under a separate declaration based on a
determination of whether certain conditions are met. Therefore, when the public health emergency ends, current EUAs may remain authorized and the
FDA  will  continue  to  have  the  authority  to  issue  new  EUAs  as  long  as  those  conditions  are  met  and  until  that  authority  is  formally  terminated  by  the
Secretary of HHS through a separate process. The Company anticipates that the end of the public health emergency may reduce the likelihood of an
EUA pathway for its potential products candidates to prevent COVID-19 even if the EUA declaration remains in place and that the EUA pathway may
become unavailable within a short period after a notice of the termination of the EUA declaration is published in the Federal Register.

If our joint venture with HaloVax, LLC (“HaloVax”) is not successful or if we fail to realize the benefits we anticipate from such joint venture,
we may not be able to capitalize on the full market potential of our potential products.

In March 2020, we entered into the Voltron Agreement to form a joint venture entity named HaloVax to jointly develop potential product candidates for the
prevention  of  the  COVID-19.  Pursuant  to  the  terms  of  the  Voltron  Agreement  we  are  entitled  to  receive  sales-based  royalties  at  low  single  digit
percentages and shall contribute proceeds of the development of products to prevent COVID-19. In addition, in 2020, we purchased 6% of HaloVax’s
outstanding  membership  interests;  however,  during  the  fourth  quarter  of  2022,  we  identified  indicators  of  impairment  for  the  HaloVax  investment  as  a
result of adverse changes in HaloVax’s business operations, including liquidity concerns. As a result, we investment in HaloVax was valued at $0 and
$350,000 as of December 31, 2022 and 2021. If and to the extent we and HaloVax are unable to develop potential product candidates for the prevention
of COVID-19, we will not be entitled to any sale-based royalties and the value of our ownership interest in HaloVax could decline in which case we may
lose all or part of our investment in HaloVax.

14

While Voltron has agreed to cooperate and use commercially reasonable efforts to exchange information and resources that will lead to the development
activities and established a Joint Development Committee consisting of seven members, two of which were selected by us, to plan, review, coordinate
and  oversee  the  performance  of  the  development  activities  and  timelines  with  respect  to  development  activities,  we  have  limited  contractual  rights  to
direct  its  activities.  Moreover,  we  will  not  have  any  other  control  with  respect  to  the  operations  of  HaloVax.  Therefore,  HaloVax  will  have  a  greater
influence with respect to its commercialization efforts and other operations. In general, our joint venture with HaloVax subjects us to a number of related
risks including that:

● we may not receive sales-based royalties pursuant to the terms of the Voltron Agreement;

● we may not be successful in the development of any product candidates;

● HaloVax may not commit sufficient resources to the marketing and distribution of our products;

● HaloVax may infringe the intellectual property rights of third parties, which may expose us to litigation and other potential liability;

●

disputes may arise between us and HaloVax that result in the delay or termination of the commercialization of our products or product candidates
or that result in costly litigation or arbitration that diverts management attention and resources including, but not limited to, disputes with respect
to commercializing products upon terms mutually agreeable or beneficial to us and HaloVax;

●

any products, if developed, will be sold or licensed on terms that are beneficial to us;

● HaloVax may not provide us with timely and accurate information regarding commercialization status or results, which could adversely impact our
ability  to  manage  our  own  commercialization  efforts,  accurately  forecast  financial  results  or  provide  timely  information  to  our  shareholders
regarding our commercialization efforts; and

●

if  any  product  candidates  are  successfully  developed  that  we  will  be  able  to  commercialize  such  products  upon  terms  mutually  agreeable  or
beneficial to us and HaloVax.

If HT-005 is not commercialized by Zylö or otherwise acquired by a third party, we may not be able to capitalize on the full market potential of
our interests with respect to HT-005.

In December 2021, we licensed HT-005 back to Zylö and are entitled to receive a low single digit percent of the net proceeds attributable to the sale of
HT-005  to  a  third  party,  a  low  single  digit  percent  of  the  net  proceeds  from  the  sale  of  HT-005  in  the  United  States  and  Canada  and  their  respective
territories (collectively, the “Territory”) and a low double digit percent of any royalty Zylö receives through the sublicense to a third party based on the net
sales of HT-005 in the Territory. In connection with the license of HT-005 back to Zylö, we acquired 100,000 shares of Zylö’s Class B common stock. As
of December 31, 2022, we own 220,000 shares of Zylö’s Class B common stock. If Zylö is unable to sell or otherwise commercialize HT-005, we will not
be entitled to any proceeds or sale-based royalties and the value of our ownership interest in Zylö could decline in which case we may lose all or part of
our investment in Zylö.

The marketing approval process of the FDA is lengthy, time consuming and inherently unpredictable, and if we are ultimately unable to obtain
marketing approval for the product candidates we intend to develop, our business may be substantially harmed.

None  of  the  product  candidates  we  intend  to  develop  have  gained  marketing  authorization,  approval  or  clearance  in  the  U.S.  or  elsewhere,  and  we
cannot  guarantee  that  we  will  ever  have  marketable  products.  Our  business  is  substantially  dependent  on  our  ability  to  complete  the  development  of,
obtain  marketing  approval  for,  and  successfully  commercialize  our  product  candidates  in  a  timely  manner.  We  cannot  commercialize  our  product
candidates  in  the  United  States  or  elsewhere  without  first  obtaining  approval  from  regulatory  agencies  such  as  the  FDA  to  market  each  product

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
candidate. Our product candidates could fail to receive marketing approval for many reasons, including among others:

●

●

●

the FDA or other regulatory agencies may disagree with the design or implementation of our clinical trials;

the FDA could determine that we cannot rely on Section 505(b)(2) for any of our product candidates; and

the FDA may determine that we have identified the wrong reference listed drug or drugs or that approval of our Section 505(b)(2) application for
any of our product candidates is blocked by patent or non-patent exclusivity of the reference listed drug or drugs.

15

In  addition,  the  process  of  seeking  regulatory  clearance  or  approval  to  market  the  product  candidates  we  intend  to  develop  is  expensive  and  time
consuming and, notwithstanding the effort and expense incurred, clearance or approval is never guaranteed. If we are not successful in obtaining timely
clearance or approval of our product candidates from the FDA or other foreign regulatory agencies, we may never be able to generate significant revenue
and may be forced to cease operations. The NDA process is costly, lengthy and uncertain. Any NDA application filed by us will have to be supported by
extensive data, including, but not limited to, technical, pre-clinical, clinical, manufacturing and labeling data, to demonstrate to the FDA’s satisfaction the
safety and efficacy of the product for its intended use.

Obtaining  clearances  or  approvals  from  the  FDA  and  from  regulatory  agencies  in  other  countries  is  an  expensive  and  time-consuming  process  and  is
uncertain as to outcome. The FDA and other agencies could ask us to supplement our submissions, collect non-clinical data, conduct additional clinical
trials or engage in other time-consuming actions, or it could simply deny our applications. In addition, even if we obtain an NDA approval or pre-market
approvals  in  other  countries,  the  approval  could  be  revoked  or  other  restrictions  imposed  if  post-market  data  demonstrates  safety  issues  or  lack  of
effectiveness.  We  cannot  predict  with  certainty  how,  or  when,  the  FDA  or  other  regulatory  agencies  will  act.  If  we  are  unable  to  obtain  the  necessary
regulatory  approvals,  our  financial  condition  and  cash  flow  may  be  adversely  affected,  and  our  ability  to  grow  domestically  and  internationally  may  be
limited. Additionally, even if cleared or approved, our products may not be approved for the specific indications that are most necessary or desirable for
successful commercialization or profitability.

We  may  encounter  substantial  delays  in  completing  our  clinical  studies  which  in  turn  will  require  additional  costs,  or  we  may  fail  to
demonstrate adequate safety and efficacy to the satisfaction of applicable regulatory authorities.

It  is  impossible  to  predict  if  or  when  any  of  our  product  candidates  will  prove  safe  or  effective  in  humans  or  will  receive  regulatory  approval.  Before
obtaining marketing approval from regulatory authorities for the sale of our product candidates, we must conduct extensive clinical studies to demonstrate
the  safety  and  efficacy  of  the  product  candidates  in  humans.  Clinical  testing  is  expensive,  time-consuming  and  uncertain  as  to  outcome.  We  cannot
guarantee that any clinical studies will be conducted as planned or completed on schedule, if at all. A failure of one or more clinical studies can occur at
any stage of testing. Events that may prevent successful or timely completion of clinical development include:

●

●

●

●

●

●

●

●

●

●

●

●

●

●

delays in reaching, or failing to reach, a consensus with regulatory agencies on study design;

delays in reaching, or failing to reach, agreement on acceptable terms with a sufficient number of prospective contract research organizations
(“CROs”) and clinical study sites, the terms of which can be subject to extensive negotiation and may vary significantly among different CROs
and trial sites;

delays in obtaining required IRB or Ethics Committee (“EC”) approval at each clinical study site;

delays in recruiting a sufficient number of suitable patients to participate in our clinical studies;

imposition of a clinical hold by regulatory agencies, after an inspection of our clinical study operations or study sites;

failure by our CROs, other third parties or us to adhere to clinical study, regulatory or legal requirements;

failure to perform in accordance with the FDA’s GCP or applicable regulatory guidelines in other countries;

delays in the testing, validation, manufacturing and delivery of sufficient quantities of our product candidates to the clinical sites;

delays in having patients complete participation in a study or return for post-treatment follow-up;

clinical study sites or patients dropping out of a study;

delay or failure to address any patient safety concerns that arise during the course of a trial;

unanticipated costs or increases in costs of clinical trials of our product candidates;

occurrence of serious adverse events associated with the product candidate that are viewed to outweigh its potential benefits; or

changes in regulatory requirements and guidance that require amending or submitting new clinical protocols.

We could also encounter delays if a clinical trial is suspended or terminated by us, by the IRBs or ECs of the institutions in which such trials are being
conducted,  by  an  independent  Safety  Review  Board  for  such  trial  or  by  the  FDA,  Therapeutics  Goods  Administration  (“TGA”),  European  Medicines
Agency (“EMA”), or other regulatory authorities. Such authorities may suspend or terminate a clinical trial due to a number of factors, including failure to
conduct the clinical trial in accordance with regulatory requirements or our clinical protocols, inspection of the clinical trial operations or trial site by the
FDA,  TGA,  or  other  regulatory  authorities  resulting  in  the  imposition  of  a  clinical  hold,  unforeseen  safety  issues  or  adverse  side  effects,  failure  to
demonstrate  a  benefit  from  using  a  drug,  changes  in  governmental  regulations  or  administrative  actions  or  lack  of  adequate  funding  to  continue  the
clinical trial.

16

 
  
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Any inability to successfully complete pre-clinical and clinical development could result in additional costs to us or impair our ability to generate revenues
from  product  sales,  regulatory  and  commercialization  milestones  and  royalties.  In  addition,  if  we  make  manufacturing  or  formulation  changes  to  our
product candidates, we may need to conduct additional studies to bridge our modified product candidates to earlier versions.

Clinical study delays could also shorten any periods during which we may have the exclusive right to commercialize our product candidates or allow our
competitors to bring products to market before we do, which could impair our ability to successfully commercialize our product candidates. In addition, any
delays in completing our clinical trials will increase our costs, slow down our product candidate development and approval process and jeopardize our
ability  to  commence  product  sales  and  generate  revenues.  Any  of  these  occurrences  may  significantly  harm  our  business,  financial  condition  and
prospects. In addition, many of the factors that cause, or lead to, a delay in the commencement or completion of clinical trials may also ultimately lead to
the denial of regulatory approval of our product candidates.

The outcome of pre-clinical studies and early clinical trials may not be predictive of the success of later clinical trials, and interim results of a clinical trial
do  not  necessarily  predict  final  results.  Further,  pre-clinical  and  clinical  data  are  often  susceptible  to  various  interpretations  and  analyses,  and  many
companies that have believed their product candidates performed satisfactorily in pre-clinical studies and clinical trials have nonetheless failed to obtain
marketing  approval.  If  the  results  of  our  clinical  studies  are  inconclusive  or  if  there  are  safety  concerns  or  adverse  events  associated  with  our  other
product candidates, we may:

●

●

●

●

●

●

●

●

be delayed in obtaining marketing approval for our product candidates, if approved at all;

obtain approval for indications or patient populations that are not as broad as intended or desired;

obtain approval with labeling that includes significant use or distribution restrictions or safety warnings;

be required to change the way the product is administered;

be required to perform additional clinical studies to support approval or be subject to additional post-marketing testing requirements;

have regulatory authorities withdraw their approval of a product or impose restrictions on its distribution in the form of a modified risk evaluation
and mitigation strategy;

be sued; or

experience damage to our reputation.

Additionally,  our  product  candidates  could  potentially  cause  other  adverse  events  that  have  not  yet  been  predicted.  The  inclusion  of  ill  patients  in  our
clinical studies may result in deaths or other adverse medical events due to other therapies or medications that such patients may be using. As described
above,  any  of  these  events  could  prevent  us  from  achieving  or  maintaining  market  acceptance  of  our  product  candidates  and  impair  our  ability  to
commercialize our products.

If we are not able to obtain any required regulatory approvals for our product candidates, we will not be able to commercialize our product
candidates and our ability to generate revenue will be limited.

We  must  successfully  complete  clinical  trials  for  our  product  candidates  before  we  can  apply  for  marketing  approval.  Even  if  we  complete  our  clinical
trials, it does not assure marketing approval. Our pre-clinical trials may be unsuccessful, which would materially harm our business. Even if our initial pre-
clinical  trials  are  successful,  we  are  required  to  conduct  clinical  trials  to  establish  our  product  candidates’  safety  and  efficacy,  before  a  marketing
application  (NDA  or  BLA  or  their  foreign  equivalents)  can  be  filed  with  the  FDA,  the  EMA,  or  comparable  foreign  regulatory  authorities  for  marketing
approval of our product candidates.

Clinical  testing  is  expensive,  is  difficult  to  design  and  implement,  can  take  many  years  to  complete  and  is  uncertain  as  to  outcome.  Success  in  early
phases of pre-clinical and clinical trials does not ensure that later clinical trials will be successful, and interim results of a clinical trial do not necessarily
predict  final  results.  A  failure  of  one  or  more  of  our  clinical  trials  can  occur  at  any  stage  of  testing.  We  may  experience  numerous  unforeseen  events
during,  or  as  a  result  of,  the  clinical  trial  process  that  could  delay  or  prevent  our  ability  to  receive  regulatory  approval  or  commercialize  our  product
candidates.  The  research,  testing,  manufacturing,  labeling,  packaging,  storage,  approval,  sale,  marketing,  advertising  and  promotion,  pricing,  export,
import  and  distribution  of  drug  products  are  subject  to  extensive  regulation  by  the  FDA,  EMA,  and  other  regulatory  authorities  in  the  United  States,
European  Union,  and  other  countries,  where  regulations  differ  from  country  to  country.  We  are  not  permitted  to  market  our  product  candidates  as
prescription pharmaceutical products in the United States until we receive approval of an NDA from the FDA, or in any foreign countries until we receive
the requisite approval from such countries. In the United States, the FDA generally requires the completion of clinical trials of each drug to establish its
safety  and  efficacy  and  extensive  pharmaceutical  development  to  ensure  its  quality  before  an  NDA  is  approved.  Regulatory  authorities  in  other
jurisdictions impose similar requirements. Of the large number of drugs in development, only a small percentage result in the submission of an NDA to
the FDA or other regulatory authorities and even fewer are eventually approved for commercialization. We have not submitted an NDA to the FDA or
comparable  applications  to  other  regulatory  authorities.  If  our  development  efforts  for  our  product  candidates,  including  regulatory  approval,  are  not
successful  for  their  planned  indications,  or  if  adequate  demand  for  our  product  candidates  is  not  generated,  our  business  will  be  materially  adversely
affected.

17

Our success depends on the receipt of regulatory approval and the issuance of such regulatory approvals is uncertain and subject to a number of

risks, including the following:

●

●

the results of nonclinical or toxicology studies may not support the filing of an IND or foreign equivalent for our product candidates;

the FDA, EMA, or comparable foreign regulatory authorities or IRBs or ECs may disagree with the design or implementation of our clinical trials;

● we may not be able to provide acceptable evidence of our product candidates’ safety and efficacy;

●

the results of our clinical trials may not be satisfactory or may not meet the level of statistical or clinical significance required by the FDA, EMA, or
other regulatory agencies for marketing approval;

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
●

●

●

●

●

●

●

●

the dosing of our product candidates in a particular clinical trial may not be at an optimal level;

patients in our clinical trials may suffer adverse effects for reasons that may or may not be related to our product candidates;

the data collected from clinical trials may not be sufficient to support the submission of an NDA, BLA or other marketing application or to obtain
regulatory approval in the United States or elsewhere;

the requirement for additional studies;

the  FDA,  EMA,  or  comparable  foreign  regulatory  authorities  may  fail  to  approve  the  manufacturing  processes  or  facilities  of  third-party
manufacturers with which we contract for clinical and commercial supplies;

the  approval  policies  or  regulations  of  the  FDA,  EMA,  or  comparable  foreign  regulatory  authorities  may  significantly  change  in  a  manner
rendering our clinical data insufficient for approval;

the  FDA,  EMA,  or  comparable  foreign  regulatory  authorities  may  disagree  on  the  design  or  implementation  of  our  clinical  trials,  including  the
methodology used in our studies, our chosen endpoints, our statistical analysis, or our proposed product indication;

our failure to demonstrate to the satisfaction of the FDA, EMA, or comparable regulatory authorities that a product candidate is safe and effective
for its proposed indication;

● we may fail to demonstrate that a product candidate’s clinical and other benefits outweigh its safety risks;

●

●

●

immunogenicity might affect a product candidate’s efficacy and/or safety;

the FDA, EMA, or comparable foreign regulatory authorities may disagree with our interpretation of data from nonclinical studies or clinical trials;

data collected from clinical trials of our product candidates may be insufficient to support the submission and filing of a marketing application or to
obtain marketing approval. For example, the FDA may require additional studies to show that our product candidates are safe or effective;

● we  may  fail  to  obtain  approval  of  the  manufacturing  processes  or  facilities  of  third-party  manufacturers  with  whom  we  contract  for  clinical  and

commercial supplies;

●

●

there may be changes in the approval policies or regulations that render our nonclinical and clinical data insufficient for approval; or

the FDA, EMA or comparable foreign regulatory authority may require more information, including additional nonclinical or clinical data to support
approval, which may delay or prevent approval and our commercialization plans, or we may decide to abandon the development program.

Failure to obtain regulatory approval for our product candidates for the foregoing, or any other reasons, will prevent us from commercializing our product
candidates, and our ability to generate revenue will be materially impaired. We cannot guarantee that regulators will agree with our assessment of the
results of the clinical trials we intend to conduct in the future or that such trials will be successful. The FDA, EMA and other regulators have substantial
discretion in the approval process and may refuse to accept any application or may decide that our data is insufficient for approval and require additional
clinical trials, or pre-clinical or other studies. In addition, varying interpretations of the data obtained from pre-clinical and clinical testing could delay, limit
or prevent regulatory approval of our product candidates.

We have only limited experience in filing the applications necessary to gain regulatory approvals and expect to rely on consultants and third party CROs
with expertise in this area to assist us in this process. Securing regulatory approvals to market a product requires the submission of pre-clinical, clinical,
and/or pharmacokinetic data, information about product manufacturing processes and inspection of facilities, proposed product labeling and supporting
information  to  the  appropriate  regulatory  authorities  for  each  therapeutic  indication  to  establish  a  product  candidate’s  safety  and  efficacy  for  each
indication. Our product candidates may prove to have undesirable or unintended side effects, toxicities or other characteristics that may preclude us from
obtaining regulatory approval or prevent or limit commercial use with respect to one or all intended indications.

18

The process of obtaining regulatory approvals is expensive, often takes many years, if approval is obtained at all, and can vary substantially based upon,
among other things, the type, complexity and novelty of the product candidates involved, the jurisdiction in which regulatory approval is sought and the
substantial discretion of the regulatory authorities. Changes in regulatory approval policies during the development period, changes in or the enactment of
additional statutes or regulations, or changes in regulatory review for a submitted product application may cause delays in the approval or rejection of an
application. Regulatory approval obtained in one jurisdiction does not necessarily mean that a product candidate will receive regulatory approval in all
jurisdictions in which we may seek approval, but the failure to obtain approval in one jurisdiction may negatively impact our ability to seek approval in a
different jurisdiction. Failure to obtain regulatory marketing approval for our product candidates in any indication will prevent us from commercializing our
product candidates, and our ability to generate revenue will be materially impaired.

If we are unable to submit an application for product candidate approval under Section 505(b)(2) of the FDCA or if we are required to generate
additional data related to the safety and efficacy of a product candidate in order to obtain approval under Section 505(b)(2), we may be unable
to meet our anticipated development and commercialization timelines.

We may seek marketing authorization in the United States under Section 505(b)(2) of the FDCA which permits use of a marketing application, referred to
as a 505(b)(2) application, where at least some of the information required for approval comes from studies not conducted by or for the applicant and for
which the applicant has not obtained a right of reference or use. The FDA interprets this to mean that an applicant may rely for approval on such data as
that found in published literature or the FDA’s finding of safety or effectiveness, or both, of a previously approved drug product owned by a third party.
There is no assurance that the FDA would find third-party data relied upon by us in a 505(b)(2) application sufficient or adequate to support approval and
may require us to generate additional data to support the safety and efficacy of a product candidate. Consequently, we may need to conduct substantial
new research and development activities beyond those we currently plan to conduct. Such additional new research and development activities would be
costly and time consuming and there is no assurance that such data generated from such additional activities would be sufficient to obtain approval.

If the data to be relied upon in a 505(b)(2) application is related to drug products previously approved by the FDA and covered by patents that are listed in

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
the FDA’s Orange Book, we would be required to submit with our 505(b)(2) application a Paragraph IV Certification in which we must certify that we do
not infringe the listed patents or that such patents are invalid or unenforceable, and provide notice to the patent owner or the holder of the approved NDA.
The  patent  owner  or  NDA  holder  would  have  45  days  from  receipt  of  the  notification  of  our  Paragraph  IV  Certification  to  initiate  a  patent  infringement
action against us. If an infringement action is initiated, the approval of our NDA would be subject to a stay of up to 30 months or more while we defend
against  such  a  suit.  Approval  of  our  product  candidates  under  Section  505(b)(2)  may  therefore  be  delayed  until  patent  exclusivity  expires  or  until  we
successfully challenge the applicability of those patents to our product candidates. Alternatively, we may elect to generate sufficient clinical data so that
we  would  no  longer  need  to  rely  on  third-party  data,  which  would  be  costly  and  time  consuming  and  there  would  be  no  assurance  that  such  data
generated from such additional activities would be sufficient to obtain approval.

We may not be able to obtain shortened review of our applications, and the FDA may not agree that a product candidate qualifies for marketing approval.
If  we  are  required  to  generate  additional  data  to  support  approval,  we  may  be  unable  to  meet  anticipated  or  reasonable  development  and
commercialization  timelines,  may  be  unable  to  generate  the  additional  data  at  a  reasonable  cost,  or  at  all,  and  may  be  unable  to  obtain  marketing
approval. If the FDA changes its interpretation of Section 505(b)(2) allowing reliance on data in a previously approved drug application owned by a third
party,  or  there  is  a  change  in  the  law  affecting  Section  505(b)(2),  this  could  delay  or  even  prevent  the  FDA  from  approving  any  Section  505(b)(2)
application that we submit.

We may not be able to obtain or maintain ODD or exclusivity for our product candidates.

Regulatory authorities in some jurisdictions, including the United States, may designate drugs for relatively small patient populations as “orphan drugs.”
Under the Orphan Drug Act, the FDA may designate a drug candidate as an orphan drug if it is intended to treat a rare disease or condition, which is
generally defined as a patient population of fewer than 200,000 individuals in the United States, or if the disease or condition affects more than 200,000
individuals  in  the  United  States  and  there  is  no  reasonable  expectation  that  the  cost  of  developing  and  making  a  drug  product  available  in  the  United
States for the type of disease or condition will be recovered from sales of the product.

ODD  entitles  a  party  to  financial  incentives,  such  as  opportunities  for  grant  funding  towards  clinical  trial  costs,  tax  advantages  and  user-fee  waivers.
Additionally,  if  a  product  that  has  orphan  designation  subsequently  receives  the  first  FDA  approval  for  the  disease  or  condition  for  which  it  has  such
designation, the product is entitled to orphan drug exclusivity. This means that the FDA may not approve any other applications to market the same drug
or biological product for the same indication for seven years, except in certain circumstances, including proving clinical superiority (i.e., another product is
safer, more effective or makes a major contribution to patient care) to the product with orphan exclusivity. Competitors, however, may receive approval of
different products for the indication for which the orphan product has exclusivity, or obtain approval for the same product but for a different indication than
that for which the orphan product has exclusivity. In addition, exclusive marketing rights in the United States may be limited if we seek approval for an
indication  broader  than  the  orphan-designated  indication  or  may  be  lost  if  the  FDA  later  determines  that  the  request  for  designation  was  materially
defective.

19

Modifications to our products may require new drug or device approvals.

Once a particular product receives FDA approval or clearance, expanded uses or uses in new indications of our products may require additional human
clinical  trials  and  new  regulatory  approvals  or  clearances,  including  additional  IND  and  NDA/BLA  submissions  or  premarket  approvals  before  we  can
begin clinical development, and/or prior to marketing and sales. If the FDA requires new clearances or approvals for a particular use or indication, we
may be required to conduct additional clinical studies, which would require additional expenditures and harm our operating results. If the products are
already  being  promoted  for  these  new  indications,  we  may  also  be  subject  to  significant  enforcement  actions.  Conducting  clinical  trials  and  obtaining
clearances and approvals can be a time-consuming process, and delays in obtaining required future clearances or approvals could adversely affect our
ability to introduce new or enhanced products in a timely manner, which in turn would harm our future growth.

Conducting  successful  clinical  studies  may  require  the  enrollment  of  large  numbers  of  patients,  and  suitable  patients  may  be  difficult  to
identify and recruit.

Patient  enrollment  in  clinical  trials  and  completion  of  patient  participation  and  follow-up  depends  on  many  factors,  including  the  size  of  the  patient
population;  the  nature  of  the  trial  protocol;  the  attractiveness  of,  or  the  discomforts  and  risks  associated  with,  the  treatments  received  by  enrolled
subjects; the availability of appropriate clinical trial investigators; support staff; proximity of patients to clinical sites; ability to comply with the eligibility and
exclusion criteria for participation in the clinical trial; and patient compliance. For example, patients may be discouraged from enrolling in our clinical trials
if  the  trial  protocol  requires  them  to  undergo  extensive  post-treatment  procedures  or  follow-up  to  assess  the  safety  and  effectiveness  of  our  product
candidates  or  if  they  determine  that  the  treatments  received  under  the  trial  protocols  are  not  attractive  or  involve  unacceptable  risks  or  discomforts.
Patients may also not participate in our clinical trials if they choose to participate in contemporaneous clinical trials of competitive products.

Additional  delays  to  the  completion  of  clinical  studies  may  result  from  modifications  being  made  to  the  protocol  during  the  clinical  trial,  if
such modifications are warranted and/or required by the occurrences in the given trial.

Each modification to the protocol during a clinical trial has to be submitted to the FDA. This could result in the delay or halt of a clinical trial while the
modification  is  evaluated.  In  addition,  depending  on  the  quantity  and  nature  of  the  changes  made,  the  FDA  could  take  the  position  that  the  data
generated by the clinical trial is not poolable because the same protocol was not used throughout the trial. This might require the enrollment of additional
subjects, which could result in the extension of the clinical trial and the FDA delaying clearance or approval of a product. Any such delay could have a
material adverse effect on our business and results of operations.

There can be no assurance that the data generated from our clinical trials using modified protocols will be acceptable to FDA.

There can be no assurance that the data generated using modified protocols will be acceptable to the FDA or that if future modifications during the trial
are  necessary,  that  any  such  modifications  will  be  acceptable  to  the  FDA.  If  the  FDA  believes  that  its  prior  approval  is  required  for  a  particular
modification, it can delay or halt a clinical trial while it evaluates additional information regarding the change.

Serious injury or death resulting from a failure of one of our drug candidates during clinical trials could also result in the FDA delaying our clinical trials or
denying  or  delaying  clearance  or  approval  of  a  product  candidate.  Even  though  an  adverse  event  may  not  be  the  result  of  the  failure  of  our  drug
candidate, the FDA or an IRB could delay or halt a clinical trial for an indefinite period of time while an adverse event is reviewed, and likely would do so
in the event of multiple such events.

Any  delay  or  termination  of  our  current  or  future  clinical  trials  as  a  result  of  the  risks  summarized  above,  including  delays  in  obtaining  or  maintaining

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
required approvals from IRBs, delays in patient enrollment, the failure of patients to continue to participate in a clinical trial, and delays or termination of
clinical  trials  as  a  result  of  protocol  modifications  or  adverse  events  during  the  trials,  may  cause  an  increase  in  costs  and  delays  in  the  filing  of  any
product  submissions  with  the  FDA,  delay  the  approval  and  commercialization  of  our  products  or  result  in  the  failure  of  the  clinical  trial,  which  could
adversely affect our business, operating results and prospects.

We rely on third parties to conduct our clinical trials and to assist us with pre-clinical development. If these third parties do not perform as
contractually required or expected, we may not be able to obtain regulatory approval for or commercialize our products.

We do not have the ability to independently conduct our pre-clinical and clinical trials for our product candidates, and we must rely on third parties, such
as  CROs,  medical  institutions,  clinical  investigators  and  contract  laboratories  to  conduct  such  trials.  If  these  third  parties  do  not  successfully  carry  out
their contractual duties or regulatory obligations, meet expected deadlines or need to be replaced, or if the quality or accuracy of the data they obtain is
compromised due to the failure to adhere to our clinical protocols or regulatory requirements or for other reasons, our pre-clinical development activities or
clinical  trials  may  be  extended,  delayed,  suspended  or  terminated,  and  we  may  not  be  able  to  obtain  regulatory  approval  for,  or  successfully
commercialize, our products on a timely basis, if at all. Furthermore, our third-party clinical trial investigators may be delayed in conducting our clinical
trials for reasons outside of their control. The occurrence of any of the foregoing may adversely affect our business, operating results and prospects.

20

The  future  results  of  our  current  or  future  clinical  trials  may  not  support  our  product  candidate  claims  or  may  result  in  the  discovery  of
unexpected adverse side effects.

Even  if  our  clinical  trials  are  completed  as  planned,  we  cannot  be  certain  that  their  results  will  support  our  drug  candidate  claims  or  that  the  FDA  or
foreign regulatory agencies will agree with our conclusions regarding them. Success in pre-clinical studies and early clinical trials does not ensure that
later clinical trials will be successful, and we cannot be sure that the later trials will replicate the results of prior trials and pre-clinical studies. The clinical
trial  process  may  fail  to  demonstrate  that  our  drug  candidates  are  safe  and  effective  for  the  proposed  indicated  uses.  If  the  FDA  or  other  regulatory
agencies  conclude  that  the  clinical  trials  for  any  of  our  product  candidates  has  failed  to  demonstrate  safety  and  effectiveness,  we  would  not  receive
clearance from the FDA or other regulatory agencies to market that product in the United States or internationally for the indications sought.

In addition, such an outcome could cause us to abandon the product candidate and might delay development of other product candidates. Any delay or
termination  of  our  clinical  trials  will  delay  the  filing  of  any  product  submissions  with  the  FDA  and,  ultimately,  our  ability  to  commercialize  our  product
candidates and generate revenues. It is also possible that patients enrolled in clinical trials will experience adverse side effects that are not currently part
of the product candidate’s profile. In addition, our clinical trials may involve a relatively small patient population. Because of the small sample size, our
results may not be indicative of future results.

Even if our product candidates are approved by regulatory authorities, if we or our suppliers fail to comply with ongoing FDA regulations or if
we experience unanticipated problems with our products, these products could be subject to restrictions or withdrawal from the market.

The manufacturing processes, reporting requirements, post-approval clinical data and promotional activities for any product candidate for which we obtain
regulatory approval will be subject to continued regulatory review, oversight and periodic inspections by the FDA. In particular, we and our suppliers are
required  to  comply  with  FDA’s  Quality  System  Regulations  and  International  Standards  Organization  (“ISO”)  regulations  for  the  manufacture  of  our
products  and  other  regulations  which  cover  the  methods  and  documentation  of  the  design,  testing,  production,  control,  quality  assurance,  labeling,
packaging,  storage  and  shipping  of  any  product  for  which  we  obtain  clearance  or  approval.  Regulatory  bodies,  such  as  the  FDA,  enforce  these
regulations through periodic inspections. The failure by us or one of our suppliers to comply with applicable statutes and regulations administered by the
FDA and other regulatory bodies, or the failure to timely and adequately respond to any adverse inspectional observations or product safety issues, could
result in, among other things, enforcement actions by the FDA.

If  any  of  these  actions  were  to  occur  it  would  harm  our  reputation  and  cause  our  product  sales  and  profitability  to  suffer  and  may  prevent  us  from
generating  revenue.  Furthermore,  our  key  component  suppliers  may  not  currently  be  or  may  not  continue  to  be  in  compliance  with  all  applicable
regulatory requirements which could result in our failure to produce our products on a timely basis and in the required quantities, if at all.

Even if regulatory clearance or approval of a product is granted, such clearance or approval may be subject to limitations on the intended uses for which
the  product  may  be  marketed  and  reduce  the  potential  to  successfully  commercialize  the  product  and  generate  revenue  from  the  product.  If  the  FDA
determines that the product promotional materials, labeling, training or other marketing or educational activities constitute promotion of an unapproved
use,  it  could  request  that  we  or  our  commercialization  partners  cease  or  modify  our  training  or  promotional  materials  or  subject  us  to  regulatory
enforcement actions. It is also possible that other federal, state or foreign enforcement authorities might take action if they consider such training or other
promotional materials to constitute promotion of an unapproved use, which could result in significant fines or penalties under other statutory authorities,
such as laws prohibiting false claims for reimbursement.

In addition, we may be required to conduct costly post-market testing and surveillance to monitor the safety or effectiveness of our products, and we must
comply with adverse event and pharmacovigilance reporting requirements, including the reporting of adverse events which occur in connection with, and
whether  or  not  directly  related  to,  our  products.  Later  discovery  of  previously  unknown  problems  with  our  products,  including  unanticipated  adverse
events or adverse events of unanticipated severity or frequency, manufacturing problems, or failure to comply with regulatory requirements, may result in
changes  to  labeling,  restrictions  on  such  products  or  manufacturing  processes,  withdrawal  of  the  products  from  the  market,  voluntary  or  mandatory
recalls, a requirement to recall, replace or refund the cost of any product we manufacture or distribute, fines, suspension of regulatory approvals, product
seizures, injunctions or the imposition of civil or criminal penalties which would adversely affect our business, operating results and prospects.

21

Our revenue stream will depend upon third-party reimbursement.

The commercial success of our products in both domestic and international markets will be substantially dependent on whether third-party coverage and
reimbursement  is  available  for  patients  that  use  our  products.  However,  the  availability  of  insurance  coverage  and  reimbursement  for  newly  approved
therapies is uncertain, and therefore, third-party coverage may be particularly difficult to obtain even if our products are approved by the FDA as safe and
efficacious. Patients using existing approved therapies are generally reimbursed all or part of the product cost by Medicare or other third-party payors.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Medicare,  Medicaid,  health  maintenance  organizations  and  other  third-party  payors  are  increasingly  attempting  to  contain  healthcare  costs  by  limiting
both  coverage  and  the  level  of  reimbursement  of  new  drugs,  and,  as  a  result,  they  may  not  cover  or  provide  adequate  payment  for  these  products.
Submission of applications for reimbursement approval generally does not occur prior to the filing of an NDA for that product and may not be granted for
as long as many months after NDA approval. In order to obtain reimbursement arrangements for these products, we or our commercialization partners
may have to agree to a net sales price lower than the net sales price we might charge in other sales channels. The continuing efforts of government and
third-party payors to contain or reduce the costs of healthcare may limit our revenue. Initial dependence on the commercial success of our products may
make our revenues particularly susceptible to any cost containment or reduction efforts.

Current  and  future  legislation  may  increase  the  difficulty  and  cost  for  us  to  obtain  marketing  approval  of  and  commercialize  our  product
candidates and affect the prices we may obtain for such product candidates.

In the United States and some foreign jurisdictions, there have been a number of legislative and regulatory changes and proposed changes regarding the
healthcare system that could prevent or delay marketing approval for our product candidates, restrict or regulate post-approval activities and affect our
ability to profitably sell our product candidates. Legislative and regulatory proposals have been made to expand post-approval requirements and restrict
sales and promotional activities for pharmaceutical products. We do not know whether additional legislative changes will be enacted, or whether the FDA
regulations, guidance or interpretations will be changed, or what the impact of such changes on the marketing approvals of our product candidates, if any,
may be. In addition, increased scrutiny by the U.S. Congress of the FDA’s approval process may significantly delay or prevent marketing approval, as
well as subject us to more stringent product labeling and post-marketing testing and other requirements.

In the United States, the Medicare Modernization Act (“MMA”) changed the way Medicare covers and pays for pharmaceutical products. The legislation
expanded Medicare coverage for drug purchases by the elderly and introduced a new reimbursement methodology based on average sales prices for
drugs. In addition, this legislation authorized Medicare Part D prescription drug plans to use formularies where they can limit the number of drugs that will
be covered in any therapeutic class. As a result of this legislation and the expansion of federal coverage of drug products, we expect that there will be
additional pressure to contain and reduce costs. These cost reduction initiatives and other provisions of this legislation could decrease the coverage and
price  that  we  receive  for  our  product  candidates  and  could  seriously  harm  our  business.  While  the  MMA  applies  only  to  drug  benefits  for  Medicare
beneficiaries, private payors often follow Medicare coverage policy and payment limitations in setting their own reimbursement rates, and any reduction in
reimbursement that results from the MMA may result in a similar reduction in payments from private payors.

The Patient Protection and Affordable Care Act, as amended by the Health Care and Education Affordability Reconciliation Act of 2010 (collectively, the
“Health Care Reform Law”) is a sweeping law intended to broaden access to health insurance, reduce or constrain the growth of healthcare spending,
enhance remedies against fraud and abuse, add new transparency requirements for healthcare and health insurance industries, impose new taxes and
fees  on  the  health  industry  and  impose  additional  health  policy  reforms.  The  Health  Care  Reform  Law  revised  the  definition  of  “average  manufacturer
price” for reporting purposes, which could increase the amount of Medicaid drug rebates to states. Further, the law imposed a significant annual fee on
companies that manufacture or import branded prescription drug products.

The Health Care Reform Law remains subject to legislative efforts to repeal, modify or delay the implementation of the law. However, if the Health Care
Reform  Law  is  repealed  or  modified,  or  if  implementation  of  certain  aspects  of  the  Health  Care  Reform  Law  are  delayed,  such  repeal,  modification  or
delay may materially adversely impact our business, strategies, prospects, operating results or financial condition. We are unable to predict the full impact
of any repeal, modification or delay in the implementation of the Health Care Reform Law on us at this time. Due to the substantial regulatory changes
that will need to be implemented by the Centers for Medicare & Medicaid Services and others, and the numerous processes required to implement these
reforms, we cannot predict which healthcare initiatives will be implemented at the federal or state level, the timing of any such reforms, or the effect such
reforms or any other future legislation or regulation will have on our business.

In addition, other legislative changes have been proposed and adopted in the United States since the Health Care Reform Law was enacted. We expect
that additional federal healthcare reform measures will be adopted in the future, any of which could limit the amounts that federal and state governments
will pay for healthcare products and services, and in turn could significantly reduce the projected value of certain development projects and reduce or
eliminate our profitability.

22

We are dependent on third parties for manufacturing and marketing of our proposed product candidates. If we are not able to secure favorable
arrangements with such third parties, our business and financial condition could be harmed.

We will not manufacture any of our proposed product candidates for commercial sale nor do we have the resources necessary to do so. In addition, we
currently do not have the capability to market our drug products ourselves. In addition to our internal sales force efforts, we have contracted with and
intend  to  continue  to  contract  with  specialized  manufacturing  companies  to  manufacture  our  proposed  product  candidates  and  partner  with  larger
pharmaceutical companies for commercialization of our products. In connection with our efforts to commercialize our proposed product candidates, we
will seek to secure favorable arrangements with third parties to distribute, promote, market and sell our proposed product candidates. If our internal sales
force  is  unable  to  successfully  distribute,  market  and  promote  our  product  candidates  and  we  are  not  able  to  secure  favorable  commercial  terms  or
arrangements  with  third  parties  for  the  distribution,  marketing,  promotion  and  sales  of  our  proposed  product  candidates,  we  may  have  to  retain
promotional and marketing rights and seek to develop the commercial resources necessary to promote or co-promote or co-market certain or all of our
proposed drug candidates to the appropriate channels of distribution in order to reach the specific medical market that we are targeting. We may not be
able to enter into any partnering arrangements on this or any other basis. If we are not able to secure favorable partnering arrangements or are unable to
develop the appropriate resources necessary for the commercialization of our proposed product candidates, our business and financial condition could
be harmed. In addition, we will have to hire additional employees or consultants, since our current employees have limited experience in these areas.
Sufficient employees with relevant skills may not be available to us. Any increase in the number of our employees would increase our expense level and
could have an adverse effect on our financial position.

In  addition,  we,  or  our  potential  commercial  partners,  may  not  successfully  introduce  our  proposed  product  candidates  or  such  candidates  may  not
achieve acceptance by patients, health care providers and insurance companies. Further, it is possible that we may not be able to secure arrangements
to  manufacture,  market,  distribute,  promote  and  sell  our  proposed  product  candidates  at  favorable  commercial  terms  that  would  permit  us  to  make  a
profit. To the extent that corporate partners conduct clinical trials, we may not be able to control the design and conduct of these clinical trials.

We may have conflicts with our partners that could delay or prevent the development or commercialization of our product candidates.

We may have conflicts with our partners, such as conflicts concerning the interpretation of pre-clinical or clinical data, the achievement of milestones, the
interpretation of contractual obligations, payments for services, development obligations or the ownership of intellectual property developed during our
collaboration. If any conflicts arise with any of our partners, such partner may act in a manner that is averse to our best interests. Any such disagreement

 
 
 
 
 
 
 
 
 
 
 
 
 
could result in one or more of the following, each of which could delay or prevent the development or commercialization of our product candidates, and in
turn prevent us from generating revenues: unwillingness on the part of a partner to pay us milestone payments or royalties we believe are due to us under
a  collaboration;  uncertainty  regarding  ownership  of  intellectual  property  rights  arising  from  our  collaborative  activities,  which  could  prevent  us  from
entering into additional collaborations; unwillingness by the partner to cooperate in the development or manufacture of the product, including providing us
with  product  data  or  materials;  unwillingness  on  the  part  of  a  partner  to  keep  us  informed  regarding  the  progress  of  its  development  and
commercialization activities or to permit public disclosure of the results of those activities; initiating of litigation or alternative dispute resolution options by
either party to resolve the dispute; or attempts by either party to terminate the agreement.

23

Even if we receive regulatory approval for any of our product candidates, we may not be able to successfully commercialize the product and
the revenue that we generate from its sales, if any, may be limited.

If approved for marketing, the commercial success of our product candidates will depend upon each product’s acceptance by the medical community,
including physicians, patients and health care payors. The degree of market acceptance for any of our product candidates will depend on a number of
factors, including:

●

●

●

●

●

●

●

●

●

●

●

●

demonstration of clinical safety and efficacy;

relative convenience, dosing burden and ease of administration;

the prevalence and severity of any adverse effects;

the willingness of physicians to prescribe our product candidates, and the target patient population to try new therapies;

efficacy of our product candidates compared to competing products;

the  introduction  of  any  new  products  that  may  in  the  future  become  available  targeting  indications  for  which  our  product  candidates  may  be
approved;

new procedures or therapies that may reduce the incidences of any of the indications in which our product candidates may show utility;

pricing and cost-effectiveness;

the inclusion or omission of our product candidates in applicable therapeutic and vaccine guidelines;

the effectiveness of our own or any future collaborators’ sales and marketing strategies;

limitations or warnings contained in approved labeling from regulatory authorities;

our  ability  to  obtain  and  maintain  sufficient  third-party  coverage  or  reimbursement  from  government  health  care  programs,  including  Medicare
and  Medicaid,  private  health  insurers  and  other  third-party  payors  or  to  receive  the  necessary  pricing  approvals  from  government  bodies
regulating the pricing and usage of therapeutics; and

●

the willingness of patients to pay out-of-pocket in the absence of third-party coverage or reimbursement or government pricing approvals.

If any of our product candidates are approved, but do not achieve an adequate level of acceptance by physicians, health care payors, and patients, we
may not generate sufficient revenue and we may not be able to achieve or sustain profitability. Our efforts to educate the medical community and third-
party payors on the benefits of our product candidates may require significant resources and may never be successful.

In addition, even if we obtain regulatory approvals, the timing or scope of any approvals may prohibit or reduce our ability to commercialize our product
candidates  successfully.  For  example,  if  the  approval  process  takes  too  long,  we  may  miss  market  opportunities  thereby  giving  other  companies  the
ability to develop competing products or establish market dominance. Any regulatory approval we ultimately obtain may be limited or subject to restrictions
or post-approval commitments that render our product candidates not commercially viable. For example, regulatory authorities may approve any of our
product  candidates  for  fewer  or  more  limited  indications  than  we  request,  may  grant  approval  contingent  on  the  performance  of  costly  post-marketing
clinical  trials,  or  may  approve  any  of  our  product  candidates  with  a  label  that  does  not  include  the  labeling  claims  necessary  or  desirable  for  the
successful  commercialization  for  that  indication.  Further,  the  FDA  or  comparable  foreign  regulatory  authorities  may  place  conditions  on  approvals  or
require risk management plans or a REMS to assure the safe use of the drug. If the FDA concludes a REMS is needed, the sponsor of the NDA must
submit  a  proposed  REMS.  The  FDA  will  not  approve  the  NDA  without  an  approved  REMS,  if  required.  A  REMS  could  include  medication  guides,
physician  communication  plans,  or  elements  to  assure  safe  use,  such  as  restricted  distribution  methods,  patient  registries  and  other  risk  minimization
tools.  The  FDA  may  also  require  a  REMS  for  an  approved  product  when  new  safety  information  emerges.  Any  of  these  limitations  on  approval  or
marketing could restrict the commercial promotion, distribution, prescription or dispensing of our product candidates. Moreover, product approvals may
be  withdrawn  for  non-compliance  with  regulatory  standards  or  if  problems  occur  following  the  initial  marketing  of  the  product.  Any  of  the  foregoing
scenarios could materially harm the commercial success of our product candidates.

24

Our products will face significant competition, and if they are unable to compete successfully, our business will suffer.

Our  product  candidates  face,  and  will  continue  to  face,  intense  competition  from  large  pharmaceutical  companies,  as  well  as  academic  and  research
institutions. We compete in an industry that is characterized by: (i) rapid technological change, (ii) evolving industry standards, (iii) emerging competition
and  (iv)  new  product  introductions.  Our  competitors  have  and  may  develop  products  and  technologies  that  will  compete  with  our  products  and
technologies. Because several competing companies and institutions have greater financial resources than us, they may be able to: (i) provide broader
services and product lines, (ii) make greater investments in research and development and (iii) carry on larger research and development initiatives. Our

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
competitors  also  have  greater  development  capabilities  than  we  do  and  have  substantially  greater  experience  in  undertaking  pre-clinical  and  clinical
testing of products, obtaining regulatory approvals, and manufacturing and marketing pharmaceutical products. They also have greater name recognition
and better access to customers than us.

Adverse events involving our products may lead the FDA or other regulatory agencies to delay or deny clearance for our products or result in
product recalls that could harm our reputation, business and financial results.

Once a product receives clearance or approval, the agency has the authority to require the recall of commercialized products in the event of adverse side
effects, material deficiencies or defects in design or manufacture. With respect to the FDA, the authority to require a recall must be based on an FDA
finding that there is a reasonable probability that the product would cause serious injury or death. Manufacturers may, under their own initiative, recall a
product if any material deficiency in a product is found. A government-mandated or voluntary recall by us or one of our distributors could occur as a result
of  adverse  side  effects,  impurities  or  other  product  contamination,  manufacturing  errors,  design  or  labeling  defects  or  other  deficiencies  and  issues.
Recalls  of  any  of  our  products  would  divert  managerial  and  financial  resources  and  have  an  adverse  effect  on  our  financial  condition  and  results  of
operations.  In  addition,  the  FDA  requires  that  certain  classifications  of  recalls  be  reported  to  FDA  within  ten  working  days  after  the  recall  is  initiated.
Companies are required to maintain certain records of recalls, even if they are not reportable to the FDA. We may initiate voluntary recalls involving our
products in the  future  that  we  determine  do  not  require  notification  of  the  FDA.  If  the  FDA  disagrees  with  our  determinations,  they  could  require  us  to
report those actions as recalls. A future recall announcement could harm our reputation with customers and negatively affect our sales. In addition, the
FDA could take enforcement action for failing to report the recalls when they were conducted.

If we fail to comply with healthcare regulations, we could face substantial enforcement actions, including civil and criminal penalties and our
business, operations and financial condition could be adversely affected.

Sales of our product candidates, if approved, or any other future product candidate will be subject to healthcare regulation and enforcement by the federal
government and the states and foreign governments in which we might conduct our business. The healthcare laws and regulations that may affect our
ability to operate include the following:

●

●

the federal Anti-Kickback Statute makes it illegal for any person or entity to knowingly and willfully, directly or indirectly, solicit, receive, offer, or
pay any remuneration that is in exchange for or to induce the referral of business, including the purchase, order, lease of any good, facility, item
or service for which payment may be made under a federal healthcare program, such as Medicare or Medicaid. The term “remuneration” has
been broadly interpreted to include anything of value;

the Omnibus Budget Reconciliation Act of 1993 (42 U.S.C. § 1395nn) (the “Stark Law”) prohibit referrals by a physician of “designated health
services” which are payable, in whole or in part, by Medicare or Medicaid, to an entity in which the physician or the physician’s immediate family
member has an investment interest or other financial relationship, subject to several exceptions. The Stark Law also prohibits billing for services
rendered pursuant to a prohibited referral. Several states have enacted laws similar to the Stark Law. These state laws may cover all (not just
Medicare and Medicaid) patients. Many federal healthcare reform proposals in the past few years have attempted to expand the Stark Law to
cover all patients as well. We consider the Stark Law in planning our products, marketing and other activities, and believe that our operations are
in  compliance  with  the  Stark  Law.  If  we  violate  the  Stark  Law,  our  financial  results  and  operations  could  be  adversely  affected.  Penalties  for
violations  include  denial  of  payment  for  the  services,  significant  civil  monetary  penalties,  and  exclusion  from  the  Medicare  and  Medicaid
programs; 

●

federal  false  claims  and  false  statement  laws,  including  the  federal  civil  False  Claims  Act  and  the  Civil  Monetary  Penalties  Law  (“CMPL”),
prohibits, among other things, any person or entity from knowingly presenting, or causing to be presented, for payment to, or approval by, federal
programs, including Medicare and Medicaid, claims for items or services, including drugs, that are false or fraudulent;

● HIPAA, created additional federal criminal statutes that prohibit among other actions, knowingly and willfully executing, or attempting to execute,
a scheme to defraud any healthcare benefit program, including private third-party payors or making any false, fictitious or fraudulent statement in
connection with the delivery of or payment for healthcare benefits, items or services;

● HIPAA,  as  amended  by  the  Health  Information  Technology  for  Economic  and  Clinical  Health  Act  of  2009  and  their  implementing  regulations,
impose  obligations  on  certain  types  of  individuals  and  entities  regarding  the  electronic  exchange  of  information  in  common  healthcare
transactions, as well as standards relating to the privacy and security of individually identifiable health information;

●

●

the  FDCA  which  among  other  things,  strictly  regulates  drug  and  biologics  manufacturing,  sales,  distribution,  prohibits  the  adulteration  or
misbranding of drugs and biologics prohibits manufacturers from marketing drug products for off-label use and regulates the distribution of drug
samples; and

the  federal  Physician  Payments  Sunshine  Act  requires  certain  manufacturers  of  drugs,  devices,  biologics  and  medical  supplies  for  which
payment is available under Medicare, Medicaid or the Children’s Health Insurance Program, with specific exceptions, to report annually to the
Centers for Medicare & Medicaid Services information related to payments or other transfers of value made to physicians and teaching hospitals,
as well as ownership and investment interests held by physicians and their immediate family members.

25

Also, many states have similar laws and regulations, such as Stark Law, anti-kickback and false claims laws that may be broader in scope and may apply
regardless of payor, in addition to items and services reimbursed under Medicaid and other state programs. Additionally, we may be subject to state laws
that require pharmaceutical companies to comply with the federal government’s and/or pharmaceutical industry’s voluntary compliance guidelines, state
laws that require drug manufacturers to report information related to payments and other transfers of value to physicians and other healthcare providers
or  marketing  expenditures,  as  well  as  state  and  foreign  laws  governing  the  privacy  and  security  of  health  information,  many  of  which  differ  from  each
other in significant ways and often are not preempted by HIPAA.

The laws and regulations applicable to our business are complex, changing and often subject to varying interpretations. As a result, we may not be able to
adhere to all applicable laws and regulations. Any violation or alleged violation of any of these laws or regulations by us could have a material adverse
effect on our business, financial condition, cash flows and results of operations. We may be a party to various lawsuits, demands, claims, qui tam suits,
government investigations and audits, of which any could result in, among other things, substantial financial penalties or awards against us, reputational
harm,  termination  of  relationships  or  contracts  related  to  our  business,  mandated  refunds,  substantial  payments  made  by  us,  required  changes  to  our
business practices, exclusion from future participation in Medicare and other healthcare programs, seizure of product and possible criminal penalties.

  
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
If  we  are  found  in  violation  of  applicable  laws  or  regulations,  we  could  suffer  severe  consequences  that  would  have  a  material  adverse  effect  on  our
business, results of operations, financial condition, cash flows, reputation and stock price, including:

●

●

●

suspension or termination of our participation in federal healthcare programs;

criminal  or  civil  liability,  fines,  damages  or  monetary  penalties  for  violations  of  healthcare  fraud  and  abuse  laws,  including  the  federal  False
Claims Act, CMPL, and Anti-Kickback Statute;

enforcement actions by governmental agencies or claims for monetary damages by patients under federal or state patient privacy laws, including
HIPAA;

●

repayment of amounts received in violation of law or applicable payment program requirements, and related monetary penalties;

● mandated changes to our practices or procedures that materially increase operating expenses;

●

●

●

imposition of corporate integrity agreements that could subject us to ongoing audits and reporting requirements as well as increased scrutiny of
our business practices;

termination of various relationships or contracts related to our business; and

harm to our reputation which could negatively affect our business relationships, decrease our ability to attract or retain patients and physicians,
decrease access to new business opportunities and impact our ability to obtain financing, among other things.

Responding to lawsuits and other proceedings as well as defending ourselves in such matters will continue to require management’s attention and cause
us to incur significant legal expense. It is also possible that criminal proceedings may be initiated against us or individuals in our business in connection
with investigations by the federal government.

Furthermore, to the extent that our product is sold in a foreign country, we may be subject to similar foreign laws.

If a third-party contract manufacturing organization (“CMO”) upon whom we rely to formulate and manufacture our product candidates does
not perform, fails to manufacture according to our specifications or fails to comply with strict regulations, our pre-clinical studies or clinical
trials  could  be  adversely  affected,  and  the  development  of  our  product  candidates  could  be  delayed  or  terminated  or  we  could  incur
significant additional expenses.

We do not own or operate any manufacturing facilities. We rely on and intend to continue to rely on CMOs to formulate and manufacture our pre-clinical
and clinical materials. Our reliance on a CMO exposes us to a number of risks, any of which could delay or prevent the completion of our pre-clinical
studies or clinical trials, or the regulatory approval or commercialization of our product candidates, result in higher costs, or deprive us of potential product
revenues. Some of these risks include:

●

●

●

●

●

●

our CMO failing to develop an acceptable formulation to support later-stage clinical trials for, or the commercialization of, our product candidates;

our  CMO  failing  to  manufacture  our  product  candidate  according  to  our  specifications,  the  FDA’s  cGMP  requirements,  or  otherwise
manufacturing material that we or the FDA may deem to be unsuitable in our clinical trials;

our CMO being unable to increase the scale of, increase the capacity for, or reformulate the form of our product candidates. We may experience
a shortage in supply, or the cost to manufacture our products may increase to the point where it may adversely affect the cost of our product
candidates. We cannot assure you that our CMO will be able to manufacture our product candidates at a suitable scale, or we will be able to find
alternative manufacturers acceptable to us that can do so;

our CMO placing a priority on the manufacture of their own products, or other customers’ products;

our CMO failing to perform as agreed upon or not remain in business; and

our CMOs’ plants being closed as a result of regulatory sanctions, natural disasters, health epidemics or otherwise.

26

Manufacturers  of  pharmaceutical  products  are  subject  to  ongoing  periodic  inspections  by  the  FDA,  the  U.S.  Drug  Enforcement  Administration  and
corresponding  state  and  foreign  agencies  to  ensure  strict  compliance  with  FDA  mandated  cGMPs,  other  government  regulations  and  corresponding
foreign  standards.  While  we  are  obligated  to  audit  their  performance,  we  do  not  have  control  over  our  CMO’s  compliance  with  these  regulations  and
standards. Failure by any of our CMOs, or us, to comply with applicable regulations could result in sanctions being imposed on us or the CMOs. These
sanctions may include fines, injunctions, civil penalties, failure of the government to grant pre-market approval of drugs, delays, suspension or withdrawal
of  approvals,  seizures  or  recalls  of  product,  operating  restrictions  and  criminal  prosecutions,  any  of  which  could  significantly  and  adversely  affect  our
business.

In  the  event  that  we  need  to  change  our  CMOs,  our  pre-clinical  studies,  clinical  trials  or  the  commercialization  of  our  product  candidates
could be delayed, adversely affected or terminated, or such a change may result in significantly higher costs.

Various  steps  in  the  manufacture  of  our  product  candidates  may  need  to  be  sole-sourced.  In  accordance  with  cGMP,  changing  manufacturers  may
require the re-validation of manufacturing processes and procedures, and may require further pre-clinical studies or clinical trials to show comparability
between the materials produced by different manufacturers. Changing our current or future CMOs may be difficult for us and could be costly, which could
result  in  our  inability  to  manufacture  our  product  candidates  for  an  extended  period  of  time  and  therefore  a  delay  in  the  development  of  our  product
candidates. Further, in order to maintain our development time lines in the event of a change in our CMOs, we may incur significantly higher costs to
manufacture our product candidates.

Healthcare Reform in the United States.

In  the  United  States,  there  have  been,  and  continue  to  be,  a  number  of  legislative  and  regulatory  changes  and  proposed  changes  to  the  healthcare

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
system  that  could  affect  the  future  results  of  pharmaceutical  manufactures’  operations.  In  particular,  there  have  been  and  continue  to  be  a  number  of
initiatives at the federal and state levels that seek to reduce healthcare costs. On the federal level, the Affordable Care Act (“ACA”) was enacted in March
2010, and included measures to significantly change the way healthcare is financed by both governmental and private insurers. Among the provisions of
the ACA that have been of greatest importance to the pharmaceutical and biotechnology industry are the following:

●

●

●

●

●

●

●

●

●

●

an  annual,  nondeductible  fee  on  any  entity  that  manufactures  or  imports  certain  branded  prescription  drugs  and  biologic  agents,  apportioned
among these entities according to their market share in certain government healthcare programs;

implementation of the federal physician payment transparency requirements, sometimes referred to as the “Physician Payments Sunshine Act”;

a licensure framework for follow-on biologic products;

creation  of  Patient-Centered  Outcomes  Research  Institute  to  oversee,  identify  priorities  in,  and  conduct  comparative  clinical  effectiveness
research, along with funding for such research;

establishment  of  a  Center  for  Medicare  Innovation  at  the  Centers  for  Medicare  &  Medicaid  Services  to  test  innovative  payment  and  service
delivery models to lower Medicare and Medicaid spending, potentially including prescription drug spending;

an  increase  in  the  statutory  minimum  rebates  a  manufacturer  must  pay  under  the  Medicaid  Drug  Rebate  Program,  to  23.1%  and  13%  of  the
average manufacturer price for most branded and generic drugs, respectively and capped the total rebate amount for innovator drugs at 100% of
the Average Manufacturer Price;

adoption  of  methodology  by  which  rebates  owed  by  manufacturers  under  the  Medicaid  Drug  Rebate  Program  are  calculated  for  certain  drugs
and biologics, including our product candidates, that are inhaled, infused, instilled, implanted or injected;

extension  of  manufacturers’  Medicaid  rebate  liability  to  covered  drugs  dispensed  to  individuals  who  are  enrolled  in  Medicaid  managed  care
organizations;

expansion of eligibility criteria for Medicaid programs by, among other things, allowing states to offer Medicaid coverage to additional individuals
and by adding new mandatory eligibility categories for individuals with income at or below 133% of the federal poverty level, thereby potentially
increasing manufacturers’ Medicaid rebate liability;

creation  of  a  Medicare  Part  D  coverage  gap  discount  program,  in  which  manufacturers  must  agree  to  offer  50%  point-of-sale  discounts  off
negotiated  prices  of  applicable  brand  drugs  to  eligible  beneficiaries  during  their  coverage  gap  period,  as  a  condition  for  the  manufacturer’s
outpatient drugs to be covered under Medicare Part D; and

●

expansion of the entities eligible for discounts under the Public Health program.

27

Although there have been legal and political challenges to certain aspects of the ACA, the Biden Administration has affirmed support for the law and,
entered its own executive orders to enforce and strengthen it. Because of the volatility surrounding the implementation and enforcement of the ACA since
its passage, and at this time, the full effect that the ACA would have on a pharmaceutical manufacturer remains unclear. This uncertainty is heightened
by  President  Biden’s  January  28,  2021  Executive  Order  on  Strengthening  Medicaid  and  the  Affordable  Care  Act  which  indicates  that  the  Biden
Administration may significantly modify the ACA and further reform the ACA and other federal programs in manner that may impact our operations. The
Biden Administration has indicated that a goal of its administration is to expand and support Medicaid and the ACA and to make high-quality healthcare
accessible and affordable. The potential increase in patients covered by government funded insurance may impact our pricing. Further, it is possible that
the Biden Administration may further increase scrutiny of drug pricing. Indeed, the Biden Administration has been vocal that lowering prescription drug
prices is a priority for the Biden Administration.

In addition, we cannot predict the likelihood, nature or extent of government regulation that may arise from future legislation or administrative or executive
action, either in the United States or abroad. We expect that additional state and federal health care reform measures will be adopted in the future, any of
which could limit the amounts that federal and state governments will pay for health care products and services.

Further, there is uncertainty surrounding the applicability of the biosimilars provisions under the ACA. The FDA has issued several guidance documents,
but no implementing regulations, on biosimilars. A number of biosimilar applications have been approved over the past few years. The regulations that
are  ultimately  promulgated  and  their  implementation  are  likely  to  have  considerable  impact  on  the  way  pharmaceutical  manufacturers  conduct  their
business and may require changes to current strategies. A biosimilar is a biological  product  that  is  highly  similar  to  an  approved  drug  notwithstanding
minor differences in clinically inactive components, and for which there are no clinically meaningful differences between the biological product and the
approved drug in terms of the safety, purity, and potency of the product.

Individual  states  have  become  increasingly  aggressive  in  passing  legislation  and  implementing  regulations  designed  to  control  pharmaceutical  and
biological  product  pricing,  including  price  or  patient  reimbursement  constraints,  discounts,  restrictions  on  certain  product  access,  and  marketing  cost
disclosure  and  transparency  measures,  and  to  encourage  importation  from  other  countries  and  bulk  purchasing.  Legally  mandated  price  controls  on
payment  amounts  by  third-party  payors  or  other  restrictions  could  harm  a  pharmaceutical  manufacturer’s  business,  results  of  operations,  financial
condition and prospects. In addition, regional healthcare authorities and individual hospitals are increasingly using bidding procedures to determine what
pharmaceutical  products  and  which  suppliers  will  be  included  in  their  prescription  drug  and  other  healthcare  programs.  This  could  reduce  ultimate
demand  for  certain  products  or  put  pressure  product  pricing,  which  could  negatively  affect  a  pharmaceutical  manufacturer’s  business,  results  of
operations, financial condition and prospects.

In  addition,  given  recent  federal  and  state  government  initiatives  directed  at  lowering  the  total  cost  of  healthcare,  Congress  and  state  legislatures  will
likely continue to focus on healthcare reform, the cost of prescription drugs and biologics and the reform of the Medicare and Medicaid programs. While
no  one  cannot  predict  the  full  outcome  of  any  such  legislation,  it  may  result  in  decreased  reimbursement  for  drugs  and  biologics,  which  may  further
exacerbate  industry-wide  pressure  to  reduce  prescription  drug  prices.  This  could  harm  a  pharmaceutical  manufacturer’s  ability  to  generate  revenue.
Increases in importation or re-importation of pharmaceutical products from foreign countries into the United States could put competitive pressure on a
pharmaceutical manufacturer’s ability to profitably price products, which, in turn, could adversely affect business, results of operations, financial condition
and prospects. A pharmaceutical manufacturer might elect not to seek approval for or market products in foreign jurisdictions in order to minimize the risk
of  re-importation,  which  could  also  reduce  the  revenue  generated  from  product  sales.  It  is  also  possible  that  other  legislative  proposals  having  similar

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
effects will be adopted.

Furthermore, regulatory authorities’ assessment of the data and results required to demonstrate safety and efficacy can change over time and can be
affected by many factors, such as the emergence of new information, including on other products, changing policies and agency funding, staffing and
leadership.  We  cannot  be  sure  whether  future  changes  to  the  regulatory  environment  will  be  favorable  or  unfavorable  to  our  business  prospects.  For
example, average review times at the FDA for marketing approval applications can be affected by a variety of factors, including budget and funding levels
and statutory, regulatory and policy changes.

28

Security  threats  to  our  information  technology  infrastructure  and/or  our  physical  buildings  could  expose  us  to  liability  and  damage  our
reputation and business.

It is essential to our business strategy that our technology and network infrastructure and our physical buildings remain secure and are perceived by our
customers and corporate partners to be secure. Despite security measures, however, any network infrastructure may be vulnerable to cyber-attacks by
hackers and other security threats. We may face cyber-attacks that attempt to penetrate our network security, sabotage or otherwise disable our research,
products and services, misappropriate our or our customers’ and partners’ proprietary information, which may include personally identifiable information,
or  cause  interruptions  of  our  internal  systems  and  services.  Despite  security  measures,  we  also  cannot  guarantee  security  of  our  physical  buildings.
Physical building penetration or any cyber-attacks could negatively affect our reputation, damage our network infrastructure and our ability to deploy our
products and services, harm our relationship with customers and partners that are affected, and expose us to financial liability.

Additionally, there are a number of state, federal and international laws protecting the privacy and security of health information and personal data. For
example,  HIPAA  imposes  limitations  on  the  use  and  disclosure  of  an  individual’s  healthcare  information  by  healthcare  providers,  healthcare
clearinghouses, and health insurance plans, or, collectively, covered entities, and also grants individuals rights with respect to their health information.
HIPAA  also  imposes  compliance  obligations  and  corresponding  penalties  for  non-compliance  on  individuals  and  entities  that  provide  services  to
healthcare  providers  and  other  covered  entities.  As  part  of  the  American  Recovery  and  Reinvestment  Act  of  2009  (“ARRA”)  the  privacy  and  security
provisions  of  HIPAA  were  amended.  ARRA  also  made  significant  increases  in  the  penalties  for  improper  use  or  disclosure  of  an  individual’s  health
information under HIPAA and extended enforcement authority to state attorneys general. As amended by ARRA and subsequently by the final omnibus
rule  adopted  in  2013,  HIPAA  also  imposes  notification  requirements  on  covered  entities  in  the  event  that  certain  health  information  has  been
inappropriately  accessed  or  disclosed,  notification  requirements  to  individuals,  federal  regulators,  and  in  some  cases,  notification  to  local  and  national
media.  Notification  is  not  required  under  HIPAA  if  the  health  information  that  is  improperly  used  or  disclosed  is  deemed  secured  in  accordance  with
encryption or other standards developed by the U.S. Department of Health and Human Services. Most states have laws requiring notification of affected
individuals and/or state regulators in the event of a breach of personal information, which is a broader class of information than the health information
protected  by  HIPAA.  Many  state  laws  impose  significant  data  security  requirements,  such  as  encryption  or  mandatory  contractual  terms,  to  ensure
ongoing  protection  of  personal  information.  Activities  outside  of  the  U.S.  implicate  local  and  national  data  protection  standards,  impose  additional
compliance requirements and generate additional risks of enforcement for non-compliance. We may be required to expend significant capital and other
resources to ensure ongoing compliance with applicable privacy and data security laws, to protect against security breaches and hackers or to alleviate
problems caused by such breaches.

Risks Related to Our Intellectual Property Rights

We rely upon licenses granted to us by various licensors, and if such licensors do not adequately defend such licenses, our business may be
harmed.

We  have  entered  into  and  may,  in  the  future,  enter  into  license  and  sublicense  agreements  with  respect  to  our  product  candidates.  We  have  limited
control  over  the  activities  of  our  licensors,  and  we  rely  upon  our  licensors  to  protect  their  intellectual  property,  including  the  patents  covered  by  our
licenses.  We  cannot  be  certain  that  activities  conducted  by  our  licensors  have  been  or  will  be  conducted  in  compliance  with  applicable  laws  and
regulations. Furthermore, we have no or limited control or input over whether, and in what manner, our licensors may enforce or defend the patents that
we  license  against  a  third-party.  Our  licensors  may  defend  the  patents  we  license  less  vigorously  than  if  we  had  enforced  or  defended  the  patents
ourselves.  Furthermore,  our  licensors  may  not  necessarily  seek  enforcement  in  scenarios  in  which  we  would  feel  that  enforcement  was  in  our  best
interests. For example, our licensors may not enforce the patents against a competitor of ours who is not a direct competitor of such licensor. If our in-
licensed intellectual property is found to be invalid or unenforceable, then our licensors may not be able to enforce the patents against a competitor of
ours. Moreover, if we fail to meet our obligations under our license agreements, the licensor may terminate the license agreement. Furthermore, if we fail
to meet our obligations under our sublicense agreements or our sublicensor fails to meet its obligations to the licensor, such licensor may terminate the
license agreement thereby terminating our sublicense agreement.

Our business depends upon us securing and protecting critical intellectual property.

To the extent we develop intellectual property, our commercial success will depend in part on obtaining and maintaining patent, trade secret, copyright
and trademark protection of our technologies in the United States and other jurisdictions as well as successfully enforcing and defending such intellectual
property rights against third-party challenges. We will only be able to protect our intellectual property from unauthorized use by third parties to the extent
that valid and enforceable intellectual property protection, such as patents or trade secrets, cover them. In particular, we place considerable emphasis on
obtaining patent and trade secret protection for significant new technologies, products and processes. Furthermore, the degree of future protection of our
proprietary rights is uncertain because legal means afford only limited protection and may not adequately protect our rights or permit us to gain or keep
our  competitive  advantage.  Moreover,  the  degree  of  future  protection  of  our  proprietary  rights  is  uncertain  for  products  that  are  currently  in  the  early
stages  of  development  because  we  cannot  predict  which  of  these  products  will  ultimately  reach  the  commercial  market  or  whether  the  commercial
versions of these products will incorporate proprietary technologies.

29

Patent positions in our industry are highly uncertain and involve complex legal and factual questions.

Patent positions in our industry are highly uncertain and involve complex legal and factual questions. Accordingly, we cannot predict the breadth of claims
that  may  be  allowed  or  enforced  in  our  patents  or  in  third-party  patents.  For  example,  we  or  our  licensors  might  not  have  been  the  first  to  make  the

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
inventions covered by our pending patent applications and issued patents, as applicable; we or our licensors might not have been the first to file patent
applications for these inventions; others may independently develop similar or alternative technologies or duplicate any of our technologies; it is possible
that none of our pending patent applications or the pending patent applications of our licensors will result in issued patents; our issued patents and issued
patents of our licensors may not provide a basis for commercially viable technologies, or may not provide us with any competitive advantages, or may be
challenged and invalidated by third parties; and, we may not develop additional proprietary technologies that are patentable. As a result, our owned and
licensed patents may not be valid, and we may not be able to obtain and enforce patents and to maintain trade secret protection for the full commercial
extent of our technology. The extent to which we are unable to do so could materially harm our business.

We and/or our licensors have applied for and will continue to apply for patents for certain products. Such applications may not result in the issuance of
any patents, and any patents now held or that may be issued may not provide us with adequate protection from competition. Furthermore, it is possible
that patents issued or licensed to us may be challenged successfully. In that event, if we have a preferred competitive position because of such patents,
any preferred position held by us would be lost. If we are unable to secure or to continue to maintain a preferred position, we could become subject to
competition from the sale of generic products. Failure to receive, inability to protect, or expiration of our patents for medical use, manufacture, conjugation
and labeling of any of our product candidates may adversely affect our business and operations.

Patents issued or licensed to us may be infringed by the products or processes of others. The cost of enforcing our patent rights against infringers, if such
enforcement is required, could be significant, and we do not currently have the financial resources to fund such litigation. Further, such litigation can go
on  for  years  and  the  time  demands  could  interfere  with  our  normal  operations.  There  has  been  substantial  litigation  and  other  proceedings  regarding
patent and other intellectual property rights in the pharmaceutical industry. We may become a party to patent litigation and other proceedings. The cost to
us of any patent litigation, even if resolved in our favor, could be substantial. Some of our competitors may be able to sustain the costs of such litigation
more effectively than we can because of their substantially greater financial resources. Litigation may also absorb significant management time.

Unpatented trade secrets, improvements, confidential know-how and continuing technological innovation are important to our scientific and commercial
success. Although we attempt to and will continue to attempt to protect our proprietary information through reliance on trade secret laws and the use of
confidentiality agreements with our corporate partners, collaborators, employees and consultants and other appropriate means, these measures may not
effectively prevent disclosure of our proprietary information, and, in any event, others may develop independently, or obtain access to, the same or similar
information.

If  we  are  found  to  be  infringing  on  patents  or  trade  secrets  owned  by  others,  we  may  be  forced  to  cease  or  alter  our  product  development
efforts, obtain a license to continue the development or sale of our products, and/or pay damages.

Our  manufacturing  processes  and  potential  products  may  violate  proprietary  rights  of  patents  that  have  been  or  may  be  granted  to  competitors,
universities or others, or the trade secrets of those persons and entities. As the pharmaceutical industry expands and more patents are issued, the risk
increases that our processes and potential products may give rise to claims that they infringe the patents or trade secrets of others. These other persons
could  bring  legal  actions  against  us  claiming  damages  and  seeking  to  enjoin  clinical  testing,  manufacturing  and  marketing  of  the  affected  product  or
process.  If  any  of  these  actions  are  successful,  in  addition  to  any  potential  liability  for  damages,  we  could  be  required  to  obtain  a  license  in  order  to
continue to conduct clinical tests, manufacture or market the affected product or use the affected process. Required licenses may not be available on
acceptable  terms,  if  at  all,  and  the  results  of  litigation  are  uncertain.  If  we  become  involved  in  litigation  or  other  proceedings,  it  could  consume  a
substantial portion of our financial resources and the efforts of our personnel.

Our ability to protect and enforce any patents we may obtain does not guaranty that we will secure the right to commercialize such patents.

A patent is a limited monopoly right conferred upon an inventor, and his successors in title, in return for the making and disclosing of a new and non-
obvious  invention.  This  monopoly  is  of  limited  duration  but,  while  in  force,  allows  the  patent  holder  to  prevent  others  from  making  and/or  using  his
invention. While a patent gives the holder this right to exclude others, it is not a license to commercialize the invention, where other permissions may be
required  for  permissible  commercialization  to  occur.  For  example,  a  drug  cannot  be  marketed  without  the  appropriate  authorization  from  the  FDA,
regardless of the existence of a patent covering the product. Further, the invention, even if patented itself, cannot be commercialized if it infringes the
valid patent rights of another party.

30

We rely on confidentiality agreements to protect our trade secrets. If these agreements are breached by our employees or other parties, our
trade secrets may become known to our competitors.

We  rely  on  trade  secrets  which  we  seek  to  protect  through  confidentiality  agreements  with  our  employees  and  other  parties.  If  these  agreements  are
breached, our competitors may obtain and use our trade secrets to gain a competitive advantage over us. We may not have any remedies against our
competitors and any remedies that may be available to us may not be adequate to protect our business or compensate us for the damaging disclosure. In
addition, we may have to expend resources to protect our interests from possible infringement by others.

Risks Related to the Company

We have expanded and may continue to expand, our business through the acquisition of rights to new drug candidates that could disrupt our
business, harm our financial condition and may also dilute current shareholders’ ownership interests in our Company.

Our business strategy includes expanding our products and capabilities, and we may seek acquisitions of additional drug candidates or technologies to do
so. Acquisitions involve numerous risks, including substantial cash expenditures; potentially dilutive issuance of equity securities; incurrence of debt and
contingent liabilities, some of which may be difficult or impossible to identify at the time of acquisition; difficulties in assimilating the acquired technologies
or  the  operations  of  the  acquired  companies;  diverting  our  management’s  attention  away  from  other  business  concerns;  risks  of  entering  markets  in
which we have limited or no direct experience; and the potential loss of our key employees or key employees of the acquired companies.

We  cannot  assure  you  that  any  acquisition  will  result  in  short-term  or  long-term  benefits  to  us.  We  may  misjudge  the  value  or  worth  of  an  acquired
product,  company  or  business.  In  addition,  our  future  success  would  depend  in  part  on  our  ability  to  manage  the  rapid  growth  associated  with
acquisitions. We cannot assure you that we will be able to make the combination of our business with that of acquired products, businesses or companies
work  or  be  successful.  Furthermore,  the  development  or  expansion  of  our  business  or  any  acquired  products,  business  or  companies  may  require  a
substantial capital investment by us. We may not have these necessary funds or they might not be available to us on acceptable terms or at all. We may
also  seek  to  raise  funds  by  selling  shares  of  our  preferred  or  common  stock,  which  could  dilute  each  current  shareholder’s  ownership  interest  in  the
Company.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Any international operations we undertake may subject us to risks inherent with operations outside of the United States.

We may seek to obtain market clearance for in foreign markets that we deem to generate significant opportunities. However, even with the cooperation of
a commercialization partner, conducting drug development in foreign countries involves inherent risks, including, but not limited to: difficulties in staffing,
funding and managing foreign operations; unexpected changes in regulatory requirements; export restrictions; tariffs and other trade barriers; difficulties
in  protecting,  acquiring,  enforcing  and  litigating  intellectual  property  rights;  fluctuations  in  currency  exchange  rates;  and  potentially  adverse  tax
consequences.  If  we  were  to  experience  any  of  the  difficulties  listed  above,  or  any  other  difficulties,  our  international  development  activities  and  our
overall financial condition may suffer and cause us to reduce or discontinue our international development and registration efforts.

We may not be successful in hiring and retaining key employees, including executive officers.

Our future operations and successes depend in large part upon the strength of our management team. We rely heavily on the continued service of each
member of our management team. Accordingly, if any member of our management team were to terminate their employment with us, such departure may
have  a  material  adverse  effect  on  our  business.  In  addition,  our  future  success  depends  on  our  ability  to  identify,  attract,  hire  or  engage,  retain  and
motivate other well-qualified financial, managerial, technical, clinical and regulatory personnel. There can be no assurance that these professionals will be
available  in  the  market,  or  that  we  will  be  able  to  retain  existing  professionals  or  to  meet  or  to  continue  to  meet  their  compensation  requirements.
Furthermore,  the  cost  base  in  relation  to  such  compensation,  which  may  include  equity  compensation,  may  increase  significantly,  which  could  have  a
material  adverse  effect  on  us.  Failure  to  establish  and  maintain  an  effective  management  team  and  work  force  could  adversely  affect  our  ability  to
operate, grow and manage our business.

Managing our growth as we expand operations may strain our resources.

We expect to grow rapidly in order to support additional, larger, and potentially international, pivotal clinical trials of our drug candidates, which will place
a  significant  strain  on  our  financial,  managerial  and  operational  resources.  In  order  to  achieve  and  manage  growth  effectively,  we  must  continue  to
improve and expand our operational and financial management capabilities. Moreover, we will need to increase staffing and to train, motivate and manage
our employees. All of these activities will increase our expenses and may require us to raise additional capital sooner than expected. Failure to manage
growth effectively could harm our business, financial condition or results of operations.

31

If a product liability claim is successfully brought against us for uninsured liabilities, or such claim exceeds our insurance coverage, we could
be forced to pay substantial damage awards that could materially harm our business.

The  use  of  any  of  our  existing  or  future  product  candidates  in  clinical  trials  and  the  sale  of  any  approved  pharmaceutical  products  may  expose  us  to
significant product liability claims. We currently do not have product liability insurance coverage but we intend to obtain such insurance. Such insurance
coverage may not protect us against any or all of the product liability claims that may be brought against us in the future. We may not be able to acquire
or  maintain  adequate  product  liability  insurance  coverage  at  a  commercially  reasonable  cost  or  in  sufficient  amounts  or  scope  to  protect  us  against
potential losses. In the event a product liability claim is brought against us, we may be required to pay legal and other expenses to defend the claim, as
well as uncovered damage awards resulting from a claim brought successfully against us. In the event our product candidate is approved for sale by the
FDA or other regulatory agency and commercialized, we may need to substantially increase the amount of our product liability coverage. Defending any
product  liability  claim  or  claims  could  require  us  to  expend  significant  financial  and  managerial  resources,  which  could  have  an  adverse  effect  on  our
business.

Our business may be adversely affected by health epidemics such as the coronavirus pandemic.

The outbreak of the novel Coronavirus (“COVID-19”) evolved into a global pandemic and spread to many regions of the world. The extent to which the
coronavirus  impacts  our  business  and  operating  results  may  continue  to  depend  on  future  developments  that  are  uncertain  and  cannot  be  accurately
predicted, including new information that may emerge concerning the coronavirus, including variants, and the actions to contain the coronavirus or treat
its impact, among others.

For  example,  staffing  issues  related  to  a  health  epidemic  such  as  COVID-19  may  disrupt  our  business  operations  ,including  our  clinical  trials.  Site
initiation,  participant  recruitment  and  enrollment,  participant  dosing,  distribution  of  clinical  trial  materials,  study  monitoring  and  data  analysis  may  be
paused  or  delayed  due  to  changes  in  hospital  or  university  policies,  federal,  state  or  local  regulations,  prioritization  of  hospital  resources  toward  other
efforts,  or  other  staffing  issues  related  to  any  such  health  epidemic.  Also,  some  participants  and  clinical  investigators  may  not  be  able  to  comply  with
clinical trial protocols. For example, quarantines or other travel limitations (whether voluntary or required) stemming from a health epidemic may impede
participant  movement,  affect  sponsor  access  to  study  sites,  or  interrupt  healthcare  services,  and  we  may  be  unable  to  conduct  our  clinical  trials.  In
addition,  if  any  third  parties  in  the  supply  chain  for  materials  used  in  the  production  of  our  product  candidates  are  adversely  impacted  by  a  health
epidemic  such  as  COVID-19,  our  supply  chain  may  be  disrupted,  limiting  our  ability  to  manufacture  our  product  candidates  for  our  clinical  trials  and
research and development operations. Furthermore, we may be at a risk of delaying, defaulting and/or not performing under existing agreements, which
may increase our costs. These cost increases may not be fully recoverable or adequately covered by insurance. Infections and deaths related to a health
epidemic  may  also  disrupt  the  United  States’  healthcare  and  healthcare  regulatory  systems  which  could  divert  healthcare  resources  away  from,  or
materially delay FDA review and/or approval of our product candidates.

The spread of the coronavirus, which caused a broad impact globally, may have a material economic effect on our business. While the potential economic
impact brought by the pandemic may be difficult to assess or predict, it has already caused, and is likely to result in further, significant disruption of global
financial markets, which may reduce our ability to access capital either at all or on favorable terms. In addition, a recession, depression or other sustained
adverse market event resulting from COVID-19 could materially and adversely affect our business and the value of our common stock.

The ultimate impact of the current pandemic, or any other health epidemic, is highly uncertain and subject to change. We do not yet know the full extent
of potential delays or impacts on our business, our clinical trials, our research programs, healthcare systems or the global economy as a whole. However,
these effects could have a material impact on our operations.

32

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
  
Risks Related to Our Common Stock

The price of our common stock may fluctuate substantially.

You should consider an investment in our common stock to be risky, and you should invest in our common stock only if you can withstand a significant
loss and wide fluctuations in the market value of your investment. Some factors that may cause the market price of our common stock to fluctuate, in
addition to the other risks mentioned in this “Risk Factors” section and elsewhere in this Annual Report on Form 10-K, are:

●

●

●

●

●

●

●

●

●

●

●

●

●

●

●

●

●

●

●

●

●

●

●

●

sale of our common stock by our shareholders, executives, and directors;

volatility and limitations in trading volumes of our shares of common stock;

our ability to obtain financings to conduct and complete research and development activities including, but not limited to, our clinical trials, and
other business activities;

the timing and success of introductions of new products by us or our competitors or any other change in the competitive dynamics of our industry,
including consolidation among competitors;

our ability to attract new customers;

our ability to secure resources and the necessary personnel to conduct clinical trials on our desired schedule;

commencement, enrollment or results of our clinical trials for our product candidates;

changes in the development status of our product candidates;

any delays or adverse developments or perceived adverse developments with respect to a regulatory agency’s review of our planned pre-clinical
and clinical trials;

any delay in our submission for studies or product approvals or adverse regulatory decisions, including failure to receive regulatory approval for
our product candidates;

unanticipated safety concerns related to the use of our product candidates;

changes in our capital structure or dividend policy, future issuances of securities and sales of large blocks of common stock by our shareholders;

our cash position;

announcements and events surrounding financing efforts, including debt and equity securities;

our inability to enter into new markets or develop new products;

reputational issues;

announcements  of  acquisitions,  partnerships,  collaborations,  joint  ventures,  new  products,  capital  commitments,  or  other  events  by  us  or  our
competitors;

changes in general economic, political and market conditions in or any of the regions in which we conduct our business;

changes in industry conditions or perceptions;

analyst research reports, recommendation and changes in recommendations, price targets, and withdrawals of coverage;

departures and additions of key personnel;

disputes and litigations related to intellectual properties, proprietary rights, and contractual obligations;

changes in applicable laws, rules, regulations, or accounting practices and other dynamics; and

other events or factors, many of which may be out of our control, including, but not limited to, pandemics such as COVID-19, war, or other acts of
God.

In  addition,  if  the  market  for  stocks  in  our  industry  or  industries  related  to  our  industry,  or  the  stock  market  in  general,  experiences  a  loss  of  investor
confidence, the trading price of our common stock could decline for reasons unrelated to our business, financial condition and results of operations. If any
of the foregoing occurs, it could cause our stock price to fall and may expose us to lawsuits that, even if unsuccessful, could be costly to defend and a
distraction to management.

33

We may acquire other companies or technologies, which could divert our management’s attention, result in dilution to our shareholders and
otherwise disrupt our operations and adversely affect our operating results.

We may in the future seek to acquire or invest in businesses, applications and services or technologies that we believe could complement or expand our
services,  enhance  our  technical  capabilities  or  otherwise  offer  growth  opportunities.  The  pursuit  of  potential  acquisitions  may  divert  the  attention  of
management  and  cause  us  to  incur  various  expenses  in  identifying,  investigating  and  pursuing  suitable  acquisitions,  whether  or  not  they  are
consummated.

In  addition,  we  do  not  have  any  experience  in  acquiring  other  businesses.  If  we  acquire  additional  businesses,  we  may  not  be  able  to  integrate  the

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
acquired personnel, operations and technologies successfully, or effectively manage the combined business following the acquisition. We also may not
achieve the anticipated benefits from the acquired business due to a number of factors, including:

●

●

●

●

●

●

●

●

●

●

inability to integrate or benefit from acquired technologies or services in a profitable manner;

unanticipated costs or liabilities associated with the acquisition;

difficulty integrating the accounting systems, operations and personnel of the acquired business;

difficulties and additional expenses associated with supporting legacy products and hosting infrastructure of the acquired business;

difficulty converting the customers of the acquired business onto our platform and contract terms, including disparities in the revenue, licensing,
support or professional services model of the acquired company;

diversion of management’s attention from other business concerns;

adverse effects to our existing business relationships with business partners and customers as a result of the acquisition;

the potential loss of key employees;

use of resources that are needed in other parts of our business; and

use of substantial portions of our available cash to consummate the acquisition.

In addition, a significant portion of the purchase price of companies we acquire may be allocated to acquired goodwill and other intangible assets, which
must be assessed for impairment at least annually. In the future, if our acquisitions do not yield expected returns, we may be required to take charges to
our operating results based on this impairment assessment process, which could adversely affect our results of operations. Acquisitions could also result
in dilutive issuances of equity securities or the incurrence of debt, which could adversely affect our operating results. In addition, if an acquired business
fails to meet our expectations, our operating results, business and financial position may suffer.

Unstable market and economic conditions and adverse developments with respect to financial institutions and associated liquidity risk may
have serious adverse consequences on our business, financial condition and stock price.

The  global  credit  and  financial  markets  have  recently  experienced  extreme  volatility  and  disruptions,  including  severely  diminished  liquidity  and  credit
availability, declines in consumer confidence, declines in economic growth, inflationary pressure and interest rate changes, increases in unemployment
rates and uncertainty about economic stability. The financial markets and the global economy may also be adversely affected by the current or anticipated
impact  of  military  conflict,  including  the  conflict  between  Russia  and  Ukraine,  terrorism  or  other  geopolitical  events.  Sanctions  imposed  by  the  United
States and other countries in response to such conflicts, including the one in Ukraine, may also adversely impact the financial markets and the global
economy, and any economic countermeasures by the affected countries or others could exacerbate market and economic instability. More recently, the
closures  of  Silicon  Valley  Bank  and  Signature  Bank  and  their  placement  into  receivership  with  the  Federal  Deposit  Insurance  Corporation  (“FDIC”)
created bank-specific and broader financial institution liquidity risk and concerns. Although the Department of the Treasury, the Federal Reserve, and the
FDIC jointly released a statement that depositors at SVB and Signature Bank would have access to their funds, even those in excess of the standard
FDIC insurance limits, under a systemic risk exception, future adverse developments with respect to specific financial institutions or the broader financial
services  industry  may  lead  to  market-wide  liquidity  shortages,  impair  the  ability  of  companies  to  access  near-term  working  capital  needs,  and  create
additional market and economic uncertainty. We have significant cash balances at financial institutions which, throughout the year, regularly exceed the
federally insured limit of $250,000. Any loss incurred or a lack of access to such funds could have a significant adverse impact on our financial condition,
results of operations, and cash flows.

34

There can be no assurance that future credit and financial market instability and a deterioration in confidence in economic conditions will not occur. Our
general  business  strategy  may  be  adversely  affected  by  any  such  economic  downturn,  liquidity  shortages,  volatile  business  environment  or  continued
unpredictable  and  unstable  market  conditions.  If  the  equity  and  credit  markets  deteriorate,  or  if  adverse  developments  are  experienced  by  financial
institutions,  it  may  cause  short-term  liquidity  risk  and  also  make  any  necessary  debt  or  equity  financing  more  difficult,  more  costly  and  more  dilutive.
Failure  to  secure  any  necessary  financing  in  a  timely  manner  and  on  favorable  terms  could  have  a  material  adverse  effect  on  our  growth  strategy,
financial performance and stock price and could require us to delay or abandon clinical development plans. In addition, there is a risk that one or more of
our financial institutions, manufacturers and other third parties with whom we engage may be adversely affected by the foregoing risks, which may have
a material adverse effect on our business.

Future  sales  and  issuances  of  our  securities  could  result  in  additional  dilution  of  the  percentage  ownership  of  our  shareholders  and  could
cause our share price to fall.

We  expect  that  significant  additional  capital  will  be  needed  in  the  future  to  continue  our  planned  operations,  including  research  and  development,
increased  marketing,  hiring  new  personnel,  commercializing  our  products,  and  continuing  activities  as  an  operating  public  company.  To  the  extent  we
raise  additional  capital  by  issuing  equity  securities,  our  shareholders  may  experience  substantial  dilution.  We  may  sell  common  stock,  convertible
securities  or  other  equity  securities  in  one  or  more  transactions  at  prices  and  in  a  manner  we  determine  from  time  to  time.  If  we  sell  common  stock,
convertible securities or other equity securities in more than one transaction, investors may be materially diluted by subsequent sales. Such sales may
also result in material dilution to our existing shareholders, and new investors could gain rights superior to our existing shareholders.

We do not intend to pay cash dividends on our shares of common stock so any returns will be limited to the value of our shares.

We have never paid or declared any cash dividends on our common stock, and we do not anticipate paying any cash dividends on our common stock in
the  foreseeable  future.  We  currently  anticipate  that  we  will  retain  future  earnings  for  the  development,  operation  and  expansion  of  our  business.  Any
future determination to pay dividends will be at the discretion of our board of directors and will depend upon a number of factors, including our results of
operations,  financial  condition,  future  prospects,  contractual  restrictions,  restrictions  imposed  by  applicable  law  and  other  factors  that  our  board  of
directors deems relevant. Therefore, any return to shareholders will be limited to the increase, if any, of our share price.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
We are an “emerging growth company” and will be able to avail ourselves of reduced disclosure requirements applicable to emerging growth
companies, which could make our common stock less attractive to investors.

We  are  an  “emerging  growth  company,”  as  defined  in  the  Jumpstart  Our  Business  Startups  Act  of  2012  (the  “JOBS  Act”),  and  we  intend  to  take
advantage  of  certain  exemptions  from  various  reporting  requirements  that  are  applicable  to  other  public  companies  that  are  not  “emerging  growth
companies”  including  not  being  required  to  comply  with  the  auditor  attestation  requirements  of  Section  404(b)  of  the  Sarbanes-Oxley  Act  of  2002,  as
amended  (“Sarbanes-Oxley”),  reduced  disclosure  obligations  regarding  executive  compensation  in  our  periodic  reports  and  proxy  statements,  and
exemptions from the requirements of holding a nonbinding advisory vote on executive compensation and shareholder approval of any golden parachute
payments not previously approved. In addition, pursuant to Section 107 of the JOBS Act, as an “emerging growth company” we intend to take advantage
of the extended transition period provided in Section 7(a)(2)(B) of the Securities Act, for complying with new or revised accounting standards. In other
words,  an  “emerging  growth  company”  can  delay  the  adoption  of  certain  accounting  standards  until  those  standards  would  otherwise  apply  to  private
companies. We cannot predict if investors will find our common stock less attractive because we may rely on these exemptions. If some investors find
our common stock less attractive as a result, there may be a less active trading market for our common stock and our stock price may be more volatile.
We  may  take  advantage  of  these  reporting  exemptions  until  we  are  no  longer  an  “emerging  growth  company.”  We  will  remain  an  “emerging  growth
company” until the earliest of (i) the last day of the fiscal year in which we have total annual gross revenues of $1.235 billion or more; (ii) the last day of
our  fiscal  year  following  the  fifth  anniversary  of  the  date  of  our  initial  public  offering;  (iii)  the  date  on  which  we  have  issued  more  than  $1.0  billion  in
nonconvertible debt during the previous three years; or (iv) the date on which we are deemed to be a large accelerated filer under the rules of the SEC.

We may be at risk of securities class action litigation.

We may be at risk of securities class action litigation. In the past, biotechnology and pharmaceutical companies have experienced significant stock price
volatility,  particularly  when  associated  with  binary  events  such  as  clinical  trials  and  product  approvals.  If  we  face  such  litigation,  it  could  result  in
substantial costs and a diversion of management’s attention and resources, which could harm our business and results in a decline in the market price of
our common stock.

35

We are currently listed on The Nasdaq Capital Market. If we are unable to maintain listing of our securities on Nasdaq or any stock exchange,
our stock price could be adversely affected and the liquidity of our stock and our ability to obtain financing could be impaired and it may be
more difficult for our shareholders to sell their securities.

Although our common stock is currently listed on The Nasdaq Capital Market, we may not be able to continue to meet the exchange’s minimum listing
requirements or those of any other national exchange. The Listing Rules of Nasdaq require listing issuers to comply with certain standards in order to
remain  listed  on  its  exchange.  If,  for  any  reason,  we  should  fail  to  maintain  compliance  with  these  listing  standards  and  Nasdaq  should  delist  our
securities  from  trading  on  its  exchange  and  we  are  unable  to  obtain  listing  on  another  national  securities  exchange,  a  reduction  in  some  or  all  of  the
following may occur, each of which could have a material adverse effect on our shareholders:

●

●

●

●

●

●

●

the liquidity of our common stock;

the market price of our common stock;

our ability to obtain financing for the continuation of our operations;

the number of investors that will consider investing in our common stock;

the number of market makers in our common stock;

the availability of information concerning the trading prices and volume of our common stock; and

the number of broker-dealers willing to execute trades in shares of our common stock.

Our Articles of Incorporation, as amended (“Articles of Incorporation”), our Amended and Restated Bylaws, and Nevada law may have anti-
takeover effects that could discourage, delay or prevent a change in control, which may cause our stock price to decline.

Our Articles of Incorporation, Amended and Restated Bylaws, and Nevada law could make it more difficult for a third party to acquire us, even if closing
such a transaction would be beneficial to our shareholders. We are authorized to issue up to 10,000,000 shares of preferred stock, none of which are
outstanding  as  of  March  17,  2023.  This  preferred  stock  may  be  issued  in  one  or  more  series,  the  terms  of  which  may  be  determined  at  the  time  of
issuance by our board of directors without further action by shareholders. The terms of any series of preferred stock may include voting rights (including
the right to vote as a series on particular matters), preferences as to dividend, liquidation, conversion and redemption rights and sinking fund provisions.
As of March 17, 2023, 5,000,000 shares of our preferred stock have been designated as Series A Preferred Stock of which 3,102,480 shares of Series A
Preferred  Stock  were  previously  issued  and  converted  into  common  stock  at  the  time  of  our  initial  public  offering  and  1,897,520  shares  of  Series  A
Preferred Stock remain authorized. The issuance of any preferred stock could materially adversely affect the rights of the holders of our common stock,
and therefore, reduce the value of our common stock. In particular, specific rights granted to future holders of preferred stock could be used to restrict our
ability to merge with, or sell our assets to, a third party and thereby preserve control by the present management.

Provisions  of  our  Articles  of  Incorporation,  our  Amended  and  Restated  Bylaws  and  Nevada  law  also  could  have  the  effect  of  discouraging  potential
acquisition proposals or making a tender offer or delaying or preventing a change in control, including changes a shareholder might consider favorable.
Such  provisions  may  also  prevent  or  frustrate  attempts  by  our  shareholders  to  replace  or  remove  our  management.  In  particular,  the  Articles  of
Incorporation, our Amended and Restated Bylaws and Nevada law, as applicable, among other things:

●

●

●

provide the board of directors with the ability to alter the Amended and Restated Bylaws without shareholder approval;

place limitations on the removal of directors;

establish advance notice requirements for nominations for election to the board of directors or for proposing matters that can be acted upon at
shareholder meetings; and

●

provide that vacancies on the board of directors may be filled by a majority of directors in office, although less than a quorum.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
36

Our  Amended  and  Restated  Bylaws  provide  that  the  Eighth  Judicial  District  Court  of  Clark  County,  Nevada  will  be  the  sole  and  exclusive
forum  for  certain  disputes  which  could  limit  shareholders’  ability  to  obtain  a  favorable  judicial  forum  for  disputes  with  us  or  its  directors,
officers, employees or agents.

Our Amended and Restated Bylaws provide that unless we consent in writing to the selection of an alternative forum, the Eighth Judicial District Court of
Clark County, Nevada shall be the sole and exclusive forum for state law claims with respect to: (i) any derivative action or proceeding brought in the
name or right of us or on our behalf, (ii) any action asserting a claim for breach of any fiduciary duty owed by any director, officer, employee or agent to us
or our shareholders, (iii) any action arising or asserting a claim arising pursuant to any provision of Nevada Revised Statutes Chapters 78 or 92A or any
provision of our Articles of Incorporation or Amended and Restated Bylaws or (iv) any action asserting a claim governed by the internal affairs doctrine,
including,  without  limitation,  any  action  to  interpret,  apply,  enforce  or  determine  the  validity  of  our  Articles  of  Incorporation  or  Amended  and  Restated
Bylaws. This exclusive forum provision would not apply to suits brought to enforce any liability or duty created by the Securities Act or the Exchange Act
or any other  claim  for  which  the  federal  courts  have  exclusive  jurisdiction.  To  the  extent  that  any  such  claims  may  be  based  upon  federal  law  claims,
Section 27 of the Exchange Act creates exclusive federal jurisdiction over all suits brought to enforce any duty or liability created by the Exchange Act or
the rules and regulations thereunder. Furthermore, Section 22 of the Securities Act creates concurrent jurisdiction for federal and state courts over all
suits brought to enforce any duty or liability created by the Securities Act or the rules and regulations thereunder.

This  choice  of  forum  provision  may  limit  a  shareholder’s  ability  to  bring  a  claim  in  a  judicial  forum  that  it  finds  favorable  for  disputes  with  us  or  our
directors, officers, other employees or agents and may result in increased costs to our shareholders, which may discourage such lawsuits against us and
our  directors,  officers,  other  employees  and  agents.  Alternatively,  if  a  court  were  to  find  the  choice  of  forum  provision  contained  in  our  Amended  and
Restated  Bylaws  to  be  inapplicable  or  unenforceable  in  an  action,  we  may  incur  additional  costs  associated  with  resolving  such  action  in  other
jurisdictions, which could have a material adverse effect on our business, results of operations, and financial condition.

General Risk Factors

If securities or industry analysts do not publish research or reports, or publish unfavorable research or reports about our business, our stock
price and trading volume may decline.

The trading market for our common stock will rely in part on the research and reports that industry or financial analysts publish about us, our business, our
markets and our competitors. We do not control these analysts. If securities analysts do not cover our common stock, the lack of research coverage may
adversely affect the market price of our common stock. Furthermore, if one or more of the analysts who do cover us  downgrade  our  stock  or  if  those
analysts  issue  other  unfavorable  commentary  about  us  or  our  business,  our  stock  price  would  likely  decline.  If  one  or  more  of  these  analysts  cease
coverage of us or fails to regularly publish reports on us, we could lose visibility in the market and interest in our stock could decrease, which in turn could
cause  our  stock  price  or  trading  volume  to  decline  and  may  also  impair  our  ability  to  expand  our  business  with  existing  customers  and  attract  new
customers.

Financial reporting obligations of being a public company in the United States are expensive and time-consuming, and our management will
be required to devote substantial time to compliance matters.

As a publicly traded company we incur significant legal, accounting and other expenses. The obligations of being a public company in the United States
require significant expenditures and places significant demands on our management and other personnel, including costs resulting from public company
reporting obligations under the Exchange Act and the rules and regulations regarding corporate governance practices, including those under Sarbanes-
Oxley, the Dodd-Frank Wall Street Reform and Consumer Protection Act, and the listing requirements of The Nasdaq Capital Market. These rules require
the establishment and maintenance of effective disclosure and financial controls and procedures, internal control over financial reporting and changes in
corporate governance practices, among many other complex rules that are often difficult to implement, monitor and maintain compliance with. Moreover,
despite recent reforms made possible by the JOBS Act, the reporting requirements, rules, and regulations will make some activities more time-consuming
and costly, particularly after we are no longer an “emerging growth company.” Our management and other personnel will need to devote a substantial
amount of time to ensure that we comply with all of these requirements and to keep pace with new regulations, otherwise we may fall out of compliance
and risk becoming subject to litigation or being delisted, among other potential problems.

Failure to maintain effective internal controls could cause our investors to lose confidence in us and adversely affect the market price of our
common stock. If our internal controls are not effective, we may not be able to accurately report our financial results or prevent fraud.

Section 404 of Sarbanes-Oxley requires annual management assessments of the effectiveness of our internal controls over financial reporting.  Effective
internal  control  over  financial  reporting  is  necessary  for  us  to  provide  reliable  financial  reports  in  a  timely  manner.  In  connection  with  the  audit  of  our
financial statements for the year ended December 31, 2022, our independent registered public accounting firm identified a material weakness. A material
weakness  is  a  significant  deficiency,  or  a  combination  of  significant  deficiencies,  in  internal  controls  over  financial  reporting  such  that  it  is  reasonably
possible  that  a  material  misstatement  of  the  annual  or  interim  financial  statements  will  not  be  prevented  or  detected  on  a  timely  basis.  The  material
weakness that has been identified by our independent registered public accounting firm relates to the lack of sufficient resources necessary to provide
adequate segregation of duties related to the preparation and review of financial information used in financial reporting and review of controls over the
financial reporting process, including cutoff related to accruals and prepaids. While we intend to take steps to remediate the material weakness in our
internal control over financial reporting by updating and expanding our accounts payable tracking and booking, we may not be successful in remediating
such weakness in a timely manner, if at all, which may undermine our ability to provide accurate, timely and reliable reports on our financial and operating
results. Furthermore, if we remediate our current material weakness but identify new material weaknesses in our internal control over financial reporting
in the future, investors may lose confidence in the accuracy and completeness of our financial reports and the market price of our common stock may be
negatively affected. As a result of such failures, we could also become subject to investigations by Nasdaq, the SEC, or other regulatory authorities, and
become  subject  to  litigation  from  investors  and  shareholders,  which  could  harm  our  reputation,  financial  condition  or  divert  financial  and  management
resources from our business.

37

ITEM 1B. UNRESOLVED STAFF COMMENTS

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Not applicable.

ITEM 2. PROPERTIES

Our  executive  office  is  located  at  1  Rockefeller  Plaza,  Suite  1039,  New  York,  NY  10020.  We  currently  lease  such  office  for  approximately  $2,500  per
month pursuant to a lease which terminates on January 1, 2025. We lease an additional office located at 33 West 60th Street, Floors 2, 11-12, New York,
NY 10023 pursuant  to  a  lease  which  expires  on  March  21,  2023.  We  believe  that  our  existing  facilities  are  suitable  and  adequate  to  meet  our  current
needs. We intend to add new facilities or expand existing facilities as we add employees, and we believe that suitable additional or substitute space will
be available as needed to accommodate any such expansion of our operations.

ITEM 3. LEGAL PROCEEDINGS

From time to time, we may become involved in various lawsuits and legal proceedings, which arise in the ordinary course of business. Litigation is subject
to inherent uncertainties, and an adverse result in these or other matters may arise from time to time that may harm our business. We are currently not
aware  of  any  such  legal  proceedings  or  claims  that  will  have,  individually  or  in  the  aggregate,  a  material  adverse  effect  on  our  business,  financial
condition or operating results.

ITEM 4. MINE SAFETY DISCLOSURES

Not applicable.

38

PART II

ITEM  5.  MARKET  FOR  REGISTRANT’S  COMMON  EQUITY,  RELATED  STOCKHOLDER  MATTERS  AND  ISSUER  PURCHASES  OF  EQUITY
SECURITIES

Market Information

On February 15, 2019, our common stock began trading on The Nasdaq Capital Market under the symbol “HOTH.” Prior to that time, there was no public
market for our common stock.

Shareholders

As of March 17, 2023, there were 98 shareholders of record of our common stock. The actual number of holders of our common stock is greater than this
number of record holders, and includes shareholders who are beneficial owners, but whose shares are held in street name by brokers or held by other
nominees. This number of holders of record also does not include shareholders whose shares may be held in trust by other entities.

Dividend Policy

We have never paid or declared any cash dividends on our common stock, and we do not anticipate paying any cash dividends on our common stock in
the foreseeable future. We intend to retain all available funds and any future earnings to fund the development, operation and expansion of our business.
Any future determination to pay dividends will be at the discretion of our board of directors and will depend upon a number of factors, including our results
of  operations,  financial  condition,  future  prospects,  contractual  restrictions,  restrictions  imposed  by  applicable  law  and  other  factors  that  our  board  of
directors deems relevant.

Recent Sales of Unregistered Securities

During the period from October 1, 2022 to December 31, 2022, the Company issued an aggregate of 1,729 shares of the Company’s common stock,
which shares were subject to a vesting schedule, to members of the Company’s board of directors for services.

The foregoing issuances were exempt from registration under Section 4(a)(2) of the Securities Act.

ITEM 6. [RESERVED]

ITEM 7. MANAGEMENT’S DISCUSSION AND ANALYSIS OF FINANCIAL CONDITIONS AND RESULTS OF OPERATIONS

You  should  read  the  following  discussion  and  analysis  of  our  financial  condition  and  results  of  operations  together  with  and  our  consolidated  financial
statements  and  the  related  notes  appearing  elsewhere  in  this  Annual  Report  on  Form  10-K.  In  addition  to  historical  information,  this  discussion  and
analysis  contains  forward-looking  statements  that  involve  risks,  uncertainties  and  assumptions.  Our  actual  results  may  differ  materially  from  those
discussed below. Factors that could cause or contribute to such differences include, but are not limited to, those identified below, and those discussed in
the section titled “Risk Factors” included elsewhere in this Annual Report on Form 10-K. All amounts in this report are in U.S. dollars, unless otherwise
noted.

Overview

We  are  a  clinical-stage  biopharmaceutical  company  focused  on  developing  new  generation  therapies  for  unmet  medical  needs.  We  are  focused  on
developing (i) a topical formulation for treating side effects from drugs used for the treatment of cancer (HT-001); (ii) a treatment for mast-cell derived
cancers  and  anaphylaxis  (HT-KIT);  (iii)  a  treatment  for  traumatic  brain  injury  and  ischemic  stroke  (HT-TBI);  and  (iv)  a  treatment  and/or  prevention  for
Alzheimer’s  or  other  neuroinflammatory  diseases  (HT-ALZ).  We  also  have  assets  being  developed  for  (i)  atopic  dermatitis  (also  known  as  eczema)
(BioLexa); (ii) a treatment for asthma and allergies using inhalational administration (HT-004); and (iii) a treatment for acne as well as inflammatory bowel
diseases (HT-003). In addition, we are continuing to evaluate a novel peptide that may be used to slow the transmission of SARS-CoV-2 (HT-002). We
are  also  developing  a  diagnostic  device  via  a  mobile  device.  Furthermore,  we  have  interests  in  certain  other  assets  being  developed  by  third  parties
including a treatment for patients with lupus that is being developed by Zylö and potential product candidates being developed pursuant to our agreement
with Voltron for the prevention of COVID-19.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
39

Results of Operations

Comparison of Our Results of Operations for the Years Ended December 31, 2022 and 2021

Operating Costs and Expenses

Research and Development Expenses

For  the  year  ended  December  31,  2022,  research  and  development  expenses  were  approximately  $4.9  million,  of  which  approximately  $87,000  was
related to licenses acquired and approximately $4.8 million was related to other research and development expenses. Specifically, during the year ended
December  31,  2022,  our  research  and  development  costs  consisted  primarily  of  the  following  costs  for  each  of  our  key  research  and  development
projects: (i) BioLexa, approximately $1 million related to clinical trial costs; (ii) HT-001, approximately $2.9 million related to manufacturing, preclinical and
clinical activities; (iii) HT-TBI, approximately $0.4 million related to manufacturing and preclinical activities; (iv) HT-003, approximately $41,000 related to
preclinical  studies;  (v)  HT-004,  approximately  $0.1  million  related  to  sponsored  research;  (vi)  HT-006,  approximately  $51,000  related  to  sponsored
research  (on  July  12,  2022,  our  non-exclusive  commercial  evaluation  license  agreement  with  the  United  States  Army  Medical  Research  and
Development Command terminated and we are no longer pursuing HT-006); (vii) GW breath based diagnostic device, approximately $76,000 related to
research and development with respect to the design of device; (viii) HT-KIT, approximately $0.2 million related to manufacturing and preclinical activities;
and  (ix)  HT-ALZ,  approximately  $0.2  million  in  sponsored  research.  In  addition  to  the  foregoing,  we  also  incurred  fees  of  approximately  $0.3  million
payable to members of our scientific advisory board for services. 

For the year ended December 31, 2021, research and development expenses were approximately $7.5 million, of which approximately $0.2 million was
related to licenses acquired and approximately $7.4 million was related to other research and development expenses. Specifically, during the year ended
December  31,  2021,  our  research  and  development  costs  consisted  primarily  of  the  following  costs  for  each  of  our  key  research  and  development
projects: (i) BioLexa, approximately $1.7 million related to clinical trial costs; (ii) HT-001, approximately $4.1 million related to manufacturing, preclinical
and  clinical  activities;  (iii)  HT-002,  approximately  $56,000  related  to  sponsored  research;  (iv)  HT-003,  approximately  $0.4  million  related  to  preclinical
studies; (v) HT-004, approximately $17,000 related to sponsored research; (vi) HT-006, approximately $51,000 related to sponsored research; (vii) GW
breath based diagnostic device, approximately $0.3 million related to research and development with respect to the design of device; and (viii) HT-KIT,
approximately $0.4 million related to research and development manufacturing. In addition to the foregoing, we also incurred fees of approximately $0.2
million payable to members of our scientific advisory board for services.

We  expect  our  research  and  development  activities  to  increase  as  we  develop  our  existing  product  candidates  and  potentially  acquire  new  product
candidates, reflecting increasing costs associated with the following:

●

●

●

●

●

employee-related expenses, which include salaries and benefits, and rent expenses;

fees related to in-licensed products and technology;

expenses incurred under agreements with CROs, investigative sites and consultants that conduct our clinical trials and a substantial portion of
our pre-clinical activities;

the cost of acquiring and manufacturing clinical trial materials; and

costs associated with non-clinical activities and regulatory approvals.

Compensation, Professional Fees, Rent and Other (“General and Administrative Expenses”)

For  the  year  ended  December  31,  2022,  General  and  Administrative  Expenses  were  approximately  $6.1  million,  which  primarily  consisted  of
approximately $2.6 million related to payroll expenses and stock-based compensation, approximately $2.5 million for professional fees and approximately
$1.0 million for other expenses.

For  the  year  ended  December  31,  2021,  General  and  Administrative  Expenses  were  approximately  $6.6  million,  which  primarily  consisted  of
approximately $3.0 million related to payroll expenses and stock-based compensation, approximately $2.7 million for professional fees and approximately
$0.8 million for other expenses.

We anticipate that our General and Administrative expenses will increase in future periods, reflecting continued and increasing costs associated with:

●

●

●

●

support of our research and development activities;

stock compensation granted to key employees and non-employees;

support of business development activities; and

increased professional fees and other costs associated with the regulatory requirements.

40

Other Income (Expenses)

For the year ended December 31, 2022, other expenses was approximately $0.3 million, which primarily resulted from $0.4 million losses on marketable
securities and $0.4 million change in fair value of investments in joint ventures, partially offset by $0.5 million of other income related to a research and
development tax credit pursuant to Australian regulations.

For the year ended December 31, 2021, other expenses were approximately $0.2 million, which consisted of the realized gain or loss, unrealized gain or

 
 
 
 
 
 
 
  
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
loss, and dividend income related to marketable securities.

Liquidity and Capital Resources 

To date we have funded our operations primarily through the sale of equity and debt securities. As of December 31, 2022, we had approximately $6.4
million  in  cash,  marketable  securities  of  approximately  $0.2  million,  working  capital  of  approximately  $5.3  million  and  an  accumulated  deficit  of
approximately $45.0 million. Net cash used in operating activities was $9.3 million and $12.1 million for the years ended December 31, 2022 and 2021,
respectively. We incurred losses of approximately $11.4 million and $14.3 million for the years ended December 31, 2022 and 2021, respectively. We
have incurred substantial operating losses since inception and expect to continue to incur significant operating losses for the foreseeable future as we
continue our pre-clinical and clinical development of our product candidates. We have not yet commercialized any products and have never generated
any revenue from product sales. We believe that our existing cash as of December 31, 2022 will enable us to fund our operating expenses and capital
expenditure requirements for at least 12 months from the date that our audited financial statements are available to be issued.

We have entered into certain license, sublicense, sponsored research and option agreements with third parties. Pursuant to such agreements, we may
be required to make certain: (i) license maintenance fee payments; (ii) out-of-pocket expense payments, including, but not limited to, payments related to
intellectual  property  and  research  related  expenses;  (iii)  development  and  commercialization  expense  payments;  (iv)  annual  and  quarterly  minimum
payments; (v) diligence expense payments; and (vi) revenue interest payments. In addition, subject to the achievement of certain development and/or
commercialization events, we may also be required to make certain: (i) minimum royalty payments, ranging from middle to high five figures, (ii) sales-
based royalties and running royalties, ranging from low single digits to low double digits; and (iii) milestone payments, of up to approximately $15.6 million
(if all milestones in all of our current agreements are achieved).

Additional funding will be necessary to fund our future clinical and pre-clinical activities. We may obtain additional financing through sales of our equity
and  debt  securities  or  entering  into  strategic  partnership  arrangements,  or  a  combination  of  the  foregoing.  There  are  no  assurances  that  we  will  be
successful in obtaining an adequate level of financing as and when needed to finance our operations on terms acceptable to us or at all, particularly in
light of the economic downturn. If we are unable to secure adequate additional funding as and when needed, we may have to significantly delay, scale
back  or  discontinue  the  development  and  commercialization  of  one  or  more  of  our  product  candidates.  In  addition,  the  magnitude  and  duration  of  the
COVID-19 pandemic and its impact on our liquidity and future funding requirements is uncertain as of the filing date of this Annually Report on Form 10-K.

Cash Flows from Operating Activities

For the year ended December 31, 2022, net cash used in operating activities was approximately $9.3 million, which primarily resulted from a net loss of
approximately  $11.3  million  and  $0.1  million  unrealized  gain  on  marketable  securities,  partially  offset  by  approximately  $0.6  million  in  stock-based
compensation,  $0.6  million  realized  loss  on  marketable  securities,  $0.4  million  change  in  fair  value  of  investments  in  joint  ventures  and  changes  in
operating assets and liabilities of approximately $0.4 million.

For the year ended December 31, 2021, net cash used in operating activities was approximately $12.1 million, which primarily resulted from a net loss of
approximately  $14.3  million,  and  was  partially  offset  by  changes  in  operating  assets  and  liabilities  of  approximately  $0.5  million,  unrealized  loss  on
marketable securities of approximately $0.2 million, and approximately $1.3 million stock-based compensation.

41

Cash Flows from Investing Activities

For the year ended December 31, 2022, net cash provided by investing activities was approximately $1.2 million which was primarily related to the sale of
marketable securities.

For the year ended December 31, 2021, net cash used in investing activities was approximately $0.2 million, which was primarily related to the sale of
marketable securities of approximately $2.5 million, and was partially offset by the purchase of marketable securities of approximately $2.6 million.

Cash Flows from Financing Activities

For  the  year  ended  December  31,  2022,  net  cash  provided  by  financing  activities  was  approximately  $6.0  million,  which  primarily  resulted  from  net
proceeds from the issuance of common stock.

For  the  year  ended  December  31,  2021,  net  cash  provided  by  financing  activities  was  approximately  $18.2  million.  Which  primarily  resulted  from
approximately $17.8 million in net proceeds from the issuance of common stock, common stock warrants and pre-funded warrants, and $0.4 million in
proceeds from the exercise of warrants.

Our ultimate success is dependent on our ability to obtain additional financing and generate sufficient cash flow to meet our obligations on a timely basis.
We  will  require  significant  amounts  of  capital  to  sustain  operations,  and  we  will  need  to  make  the  investments  we  need  to  execute  our  longer-term
business  plan  to  support  new  technologies  and  help  advance  innovation.  Absent  generation  of  sufficient  revenue  from  the  execution  of  our  long-term
business plan, we will need to obtain debt or equity financing, especially if we experience downturns in our business that are more severe or longer than
anticipated, or if we experience significant increases in expense levels resulting from being a publicly traded company or from operations. Such additional
debt or equity financing may not be available to us on favorable terms, if at all.

We plan to pursue our plans with respect to the research and development of our pre-clinical products which will require resources beyond those that we
currently have, ultimately requiring additional capital from third party sources. We currently do not expect to generate any revenue.

Critical Accounting Policies and Significant Judgments and Estimates

Our management’s discussion and analysis of our financial condition and results of operations is based on our consolidated financial statements, which
have  been  prepared  in  accordance  with  U.S.  generally  accepted  accounting  principles  (“GAAP”).  The  preparation  of  these  consolidated  financial
statements requires us to make estimates, judgments and assumptions that affect the reported amounts of assets and liabilities, disclosure of contingent
assets and liabilities as of the date of the balance sheet and the reported amounts of expenses during the reporting period. In accordance with GAAP, we
evaluate  our  estimates  and  judgments  on  an  ongoing  basis.  The  most  significant  estimates  relate  to  the  valuation  of  stock  options  and  the  valuation
allowance  of  deferred  tax  assets  resulting  from  net  operating  losses.  We  base  our  estimates  and  assumptions  on  current  facts,  our  limited  historical
experience and various other factors that we believe are reasonable under the circumstances, the results of which form the basis for making judgments
about the carrying value of assets and liabilities that are not readily apparent from other sources. Actual results may differ from these estimates under

  
 
 
 
  
 
 
 
 
 
 
 
  
 
 
 
 
 
 
different assumptions or conditions.

We define our critical accounting policies as those accounting principles that require us to make subjective estimates and judgments about matters that
are uncertain and are likely to have a material impact on our financial condition and results of operations, as well as the specific manner in which we
apply  those  principles.  While  our  significant  accounting  policies  are  more  fully  described  in  Note  2  to  our  consolidated  financial  statements  appearing
elsewhere  in  Annual  Report  on  Form  10-K,  we  believe  the  following  are  the  critical  accounting  policies  used  in  the  preparation  of  our  consolidated
financial statements that require significant estimates and judgments:

Stock-based compensation

We expense stock-based compensation to employees and non-employees over the requisite service period based on the estimated grant-date fair value
of  the  awards.  Stock-based  awards  with  graded-vesting  schedules  are  recognized  on  a  straight-line  basis  over  the  requisite  service  period  for  each
separately vesting portion of the award. We record the expense for stock-based compensation awards subject to performance-based milestone vesting
over  the  remaining  service  period  when  management  determines  that  achievement  of  the  milestone  is  probable.  Management  evaluates  when  the
achievement of a performance-based milestone is probable based on the expected satisfaction of the performance conditions at each reporting date. All
stock-based compensation costs are recorded in general and administrative or research and development costs in the statements of operations based
upon the underlying employees’ or non-employees’ roles.

42

Income taxes

Income taxes are recorded in accordance with Accounting Standards Codification (“ASC”) 740, Income Taxes (“ASC 740”) which provides for deferred
taxes using an asset and liability approach. We recognize deferred tax assets and liabilities for the expected future tax consequences of events that have
been included in our consolidated financial statements or tax returns. Deferred tax assets and liabilities are determined based on the difference between
our  financial  statement  and  tax  bases  of  assets  and  liabilities  using  enacted  tax  rates  in  effect  for  the  year  in  which  the  differences  are  expected  to
reverse. Valuation allowances are provided, if based upon the weight of available evidence, it is more likely than not that some or all of the deferred tax
assets will not be realized.

We account for uncertain tax positions in accordance with the provisions of ASC 740. When uncertain tax positions exist, we recognize the tax benefit of
tax positions to the extent that the benefit would more likely than not be realized assuming examination by the taxing authority. The determination as to
whether the tax benefit will more likely than not be realized is based upon the technical merits of the tax position as well as consideration of the available
facts and circumstances.

Significant Accounting Policies

See Note 2 to the consolidated financial statements for a discussion of recent accounting policies.

JOBS Act

On  April  5,  2012,  the  JOBS  Act  was  enacted.  Section  107  of  the  JOBS  Act  provides  that  an  “emerging  growth  company”  can  take  advantage  of  the
extended transition period provided in Section 7(a)(2)(B) of the Securities Act, for complying with new or revised accounting standards. In other words, an
“emerging growth company” can delay the adoption of certain accounting standards until those standards would otherwise apply to private companies.

We have chosen to take advantage of the extended transition periods available to emerging growth companies under the JOBS Act for complying with
new or revised accounting standards until those standards would otherwise apply to private companies provided under the JOBS Act. As a result, our
consolidated financial statements may not be comparable to those of companies that comply with public company effective dates for complying with new
or revised accounting standards.

Subject to certain conditions set forth in the JOBS Act, as an “emerging growth company,” we intend to rely on certain of these exemptions, including,
without  limitation,  (i)  providing  an  auditor’s  attestation  report  on  our  system  of  internal  controls  over  financial  reporting  pursuant  to  Section  404(b)  of
Sarbanes-Oxley and (ii) complying with any requirement that may be adopted by the Public Company Accounting Oversight Board regarding mandatory
audit  firm  rotation  or  a  supplement  to  the  auditor’s  report  providing  additional  information  about  the  audit  and  the  financial  statements,  known  as  the
auditor discussion and analysis. We will remain an “emerging growth company” until the earliest of (i) the last day of the fiscal year in which we have total
annual gross revenues of $1.235 billion or more; (ii) the last day of our fiscal year following the fifth anniversary of the date of our initial public offering; (iii)
the date on which we have issued more than $1 billion in nonconvertible debt during the previous three years; or (iv) the date on which we are deemed to
be a large accelerated filer under the rules of the SEC.

ITEM 7A. QUANTITATIVE AND QUALITATIVE DISCLOSURES ABOUT MARKET RISK.

As a smaller reporting company, we are not required to provide the information required by this item.

43

ITEM 8. FINANCIAL STATEMENTS AND SUPPLEMENTARY DATA

Hoth Therapeutics, Inc.
Consolidated Financial Statements

TABLE OF CONTENTS

Consolidated Financial Statements 

Page  No.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Report of Independent Registered Public Accounting Firm (PCAOB ID: 100)

Consolidated Balance Sheets as of December 31, 2022 and 2021

Consolidated Statements of Operations and Comprehensive Loss for the years ended December 31, 2022 and 2021

Consolidated Statements of Changes in Stockholders’ Equity for the years ended December 31, 2022 and 2021

Consolidated Statements of Cash Flows for the years ended December 31, 2022 and 2021

Notes to Consolidated Financial Statements

F-2

F-3

F-4

F-5

F-6

F-7

F-1

Report of Independent Registered Public Accounting Firm  

To the Stockholders and the Board of Directors of
Hoth Therapeutics, Inc.

Opinion on the Consolidated Financial Statements

We have audited the accompanying consolidated balance sheets of Hoth Therapeutics, Inc. (the “Company”) as of December 31, 2022 and 2021, the
related consolidated statements of operations and comprehensive loss, changes in stockholders’ equity and cash flows, for each of the two years in the
period  ended  December  31,  2022,  and  the  related  notes  (collectively  referred  to  as  the  “consolidated  financial  statements”).  In  our  opinion,  the
consolidated financial statements present fairly, in all material respects, the consolidated financial position of the Company as of December 31, 2022 and
2021, and the consolidated results of its operations and its cash flows for each of the two years in the period ended December 31, 2022, in conformity
with accounting principles generally accepted in the United States of America.

Basis for Opinion

These  consolidated  financial  statements  are  the  responsibility  of  the  Company’s  management.  Our  responsibility  is  to  express  an  opinion  on  the
Company’s  consolidated  financial  statements  based  on  our  audits.  We  are  a  public  accounting  firm  registered  with  the  Public  Company  Accounting
Oversight  Board  (United  States)  (“PCAOB”)  and  are  required  to  be  independent  with  respect  to  the  Company  in  accordance  with  the  U.S.  federal
securities laws and the applicable rules and regulations of the Securities and Exchange Commission and the PCAOB.

We  conducted  our  audits  in  accordance  with  the  standards  of  the  PCAOB.  Those  standards  require  that  we  plan  and  perform  the  audits  to  obtain
reasonable  assurance  about  whether  the  consolidated  financial  statements  are  free  of  material  misstatement,  whether  due  to  error  or  fraud.  The
Company is not required to have, nor were we engaged to perform, an audit of its internal control over financial reporting. As part of our audits we are
required to obtain an understanding of internal control over financial reporting but not for the purpose of expressing an opinion on the effectiveness of the
Company’s internal control over financial reporting. Accordingly, we express no such opinion.

Our audits included performing procedures to assess the risks of material misstatement of the consolidated financial statements, whether due to error or
fraud, and performing procedures that respond to those risks. Such procedures included examining, on a test basis, evidence regarding the amounts and
disclosures in the consolidated financial statements. Our audits also included evaluating the accounting principles used and significant estimates made by
management,  as  well  as  evaluating  the  overall  presentation  of  the  consolidated  financial  statements.  We  believe  that  our  audits  provide  a  reasonable
basis for our opinion.

/S/ WithumSmith+Brown, PC

We have served as the Company’s auditor since 2018.

New York, New York
March 31, 2023
PCAOB ID No. 100

ASSETS
Current assets

Cash
Marketable equity securities, at fair value
Prepaid expenses
Note receivable - current
Total current assets

Investment in joint ventures at fair value

F-2

Hoth Therapeutics, Inc.
Consolidated Balance Sheets

  December 31,     December 31,  

2022

2021

  $

6,428,611    $
209,320     
88,450     
-     
6,726,381     

8,538,270 
1,892,837 
93,972 
50,000 
10,575,079 

33,000     

410,000 

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
 
   
     
 
   
     
 
   
   
   
   
 
   
      
  
   
Total assets

LIABILITIES AND STOCKHOLDERS’ EQUITY
Current liabilities

Accounts payable
Accrued expenses
Accrued license fee - current portion

Total current liabilities

Accrued license fee - less current portion
Total liabilities

Commitments and contingencies

  $

6,759,381    $

10,985,079 

  $

694,989    $
667,742     
25,000     
1,387,731     

360,964 
426,823 
80,000 
867,787 

250,000     
1,637,731     

235,000 
1,102,787 

Stockholders’ equity
Preferred stock, $0.0001 par value,  10,000,000 shares authorized; 2,000,000 and -0- shares issued and outstanding

at December 31, 2022 and 2021, respectively

Series A Convertible Preferred Stock, $ 0.0001 par value,  5,000,000 shares designated; -0- shares issued and

outstanding at December 31, 2022 and 2021

Series B Preferred Stock, $ 0.0001 par value,  2,000,000 shares designated; -0- shares issued and outstanding at

December 31, 2022 and 2021

Common stock, $0.0001 par value,  50,000,000 shares authorized; 1,302,113 and 959,009 shares issued and

outstanding at December 31, 2022 and 2021, respectively

Additional paid-in capital
Accumulated deficit
Accumulated other comprehensive income
Total stockholders’ equity
Total liabilities and stockholders’ equity

-     

-     

-     

- 

- 

- 

130     
50,198,630     
(45,099,116)    
22,006     
5,121,650     
6,759,381    $

96 
43,591,773 
(33,727,163)
17,586 
9,882,292 
10,985,079 

  $

The accompanying notes are an integral part of these consolidated financial statements.

F-3

Hoth Therapeutics, Inc.
Consolidated Statements of Operations and Comprehensive Loss

Operating costs and expenses
Research and development
Research and development - licenses acquired (including stock-based compensation)
Compensation and related expenses (including stock-based compensation)
Professional fees (including stock-based compensation)
Rent
Other general and administrative expenses

Total operating expenses

Loss from operations

Other (expenses) income

Losses on marketable securities
Change in fair value of investments in joint ventures
Interest income
Other income (expenses), net

Total other expenses

Net loss
Other comprehensive income

Foreign currency translation adjustment

Total comprehensive loss

Deemed dividend to Series B Preferred Stock being redeemed
Net Loss Attributable to Common Stockholders

Net loss per share applicable to common stockholders - basic and diluted

Weighted average number of common shares outstanding, basic and diluted

For the Years Ended
December 31,

2022

2021

  $

4,844,578    $
86,586     
2,588,595     
2,494,132     
66,834     
984,829     
11,065,554     
(11,065,554)    

7,354,708 
174,782 
3,036,034 
2,703,837 
46,871 
785,208 
14,101,440 
(14,101,440)

(386,909)    
(377,000)    
6,370     
451,140     
(306,399)    

(152,682)
- 
- 
(59,583)
(212,265)

  $ (11,371,953)   $ (14,313,705)

4,420     

32,937 
  $ (11,367,533)   $ (14,280,768)
- 
990     
  $ (11,370,963)   $ (14,280,768)

  $

(9.50)   $
1,197,521     

(16.02)
893,226 

The accompanying notes are an integral part of these consolidated financial statements.

F-4

 
   
      
  
   
      
  
   
      
  
   
   
   
 
   
      
  
   
   
 
   
      
  
   
      
  
 
   
      
  
   
      
  
   
   
   
   
   
   
   
   
 
 
 
 
 
 
 
 
 
 
   
 
   
     
 
   
   
   
   
   
   
   
 
   
      
  
   
      
  
   
   
   
   
   
 
   
      
  
   
      
  
   
   
 
   
      
  
   
 
 
 
Hoth Therapeutics, Inc.
Consolidated Statements of Changes in Stockholders’ Equity

Series B
Preferred Stock

Common Stock

Shares     Amount     Shares     Amount    

Additional
Paid-in
Capital

    Accumulated   
Deficit

Accumulated
Other
Comprehensive   
Income

-     

273,079     

27      13,407,605     

-     

-     

13,407,632 

Balance at December 31, 2020

-    $

-     

537,558    $

54    $ 24,074,348    $ (19,413,458)   $

(15,351)   $

Issuance of common stock, common stock
warrants and prefunded warrants (net of
offering costs of $1,591,600)

Issuance of common stock and warrants (net of

offering costs of $572,500)

Warrant exercise
Stock-based compensation
Cumulative translation adjustment
Net loss

Balance at December 31, 2021
Stock-based compensation
Issuance of common stock (net of offering costs of

$1,014,896)

Issuance of Series B preferred stock
Redemption of Series B preferred stock
Fractional shares adjusted for reverse split
Cumulative translation adjustment
Net loss

Balance at December 31, 2022

-     

-     
-     
-     
-     
-     
-     
-     

-     
-     
-     
-     
-     
-     
-     

99,010     
45,069     
4,293     
-     
-     
959,009     
1,801     

10      4,427,491     
5     
359,508     
-      1,322,821     
-     
-     
-     
-     
96      43,591,773     
620,798     

-     

-     
-     
-     
-     
(14,313,705)    
(33,727,163)    
-     

-     
    2,000,000     
    (2,000,000)    
-     
-     
-     
-    $

329,412     
-     
-     
1,000     
-     
(1,000)    
11,891     
-     
-     
-     
-     
-     
-      1,302,113    $

-     
33      5,985,070     
-     
-     
-     
990     
-     
(1)    
-     
-     
(11,371,953)    
-     
130    $ 50,198,630    $ (45,099,116)   $

-     
-     
1     
-     
-     

Total
Stockholders’  
Equity
4,645,593 

-     
-     
-     
32,937     
-     
17,586     
-     

4,427,501 
359,513 
1,322,821 
32,937 
(14,313,705)
9,882,292 
620,798 

-     
-     
-     
-     
4,420     
-     
22,006    $

5,985,103 
1,000 
(10)
- 
4,420 
(11,371,953)
5,121,650 

The accompanying notes are an integral part of these consolidated financial statements.

F-5

Hoth Therapeutics, Inc.
Consolidated Statements of Cash Flows

Cash flows from operating activities
Net loss
Adjustments to reconcile net loss to net cash used in operating activities:

Research and development – licenses acquired
Change in fair value of investments in joint ventures
Stock-based compensation
Realized loss on marketable equity securities
Unrealized (gain) loss on marketable equity securities
Loss on foreign currency exchange
Changes in operating assets and liabilities:

Prepaid expenses
Accounts payable and accrued expenses

Net cash used in operating activities

Cash flows from investing activities

Purchase of research and development licenses
Purchase of marketable equity securities
Sale of marketable equity securities

Net cash provided by (used in) investing activities

Cash flows from financing activities

Proceeds from issuance common stock, common stock warrants and prefunded warrants, net of offering cost
Proceeds from issuance common stock and warrants, net of offering cost
Proceeds from issuance common stock, net of offering cost
Proceeds from issuance of Series B Preferred Stock
Redemption of Series B Preferred Stock
Proceeds from exercise of warrants
Proceeds from repayment of note receivable and interest received

Net cash provided by financing activities

Effect of exchange rate changes on cash and cash equivalents

Net change in cash
Cash, beginning of period

Cash, end of period

Non-cash investing and financing activities
Fractional shares adjusted for reverse split

For the Years Ended
December 31,

2022

2021

  $ (11,371,953)   $ (14,313,705)

34,000     
377,000     
620,798     
567,692     
(119,870)    
-     

92,470 
- 
1,322,821 
41,808 
176,974 
59,583 

3,847     
590,632     
(9,297,854)    

(5,420)
535,340 
(12,090,129)

(74,000)    
-     
1,235,695     
1,161,695     

(116,970)
(2,556,135)
2,507,750 
(165,355)

-     
-     
5,985,103     
1,000     
(10)    
-     
50,000     
6,036,093     

13,407,632 
4,427,501 
- 
- 
- 
359,513 
- 
18,194,646 

(9,593)    

(30,562)

(2,100,066)    
8,538,270     

5,939,162 
2,629,670 

  $

6,428,611    $

8,538,270 

  $

1    $

- 

 
 
 
 
   
   
 
 
   
   
   
 
   
   
   
   
   
   
   
   
   
   
   
   
   
   
 
 
 
 
 
 
 
 
 
 
   
 
   
     
 
   
      
  
   
   
   
   
   
   
   
      
  
   
   
   
 
   
      
  
   
      
  
   
   
   
   
 
   
      
  
   
      
  
   
   
   
   
   
   
   
   
 
   
      
  
   
 
   
      
  
   
   
 
   
      
  
 
   
      
  
   
      
  
 
   
      
  
The accompanying notes are an integral part of these consolidated financial statements.

F-6

Hoth Therapeutics, Inc.
Notes to Consolidated Financial Statements

Note 1-Organization and description of business operations

Hoth Therapeutics, Inc. (together with its wholly-owned subsidiary, Hoth Therapeutics Australia Pty Ltd, the “Company”) was incorporated under the laws
of the State of Nevada on May 16, 2017. The Company is a clinical-stage biopharmaceutical company focused on developing new generation therapies
for unmet medical needs. The Company is focused on developing (i) a topical formulation for treating side effects from drugs used for the treatment of
cancer (HT-001); (ii) a treatment for mast-cell derived cancers and anaphylaxis (HT-KIT); (iii) a treatment for traumatic brain injury and ischemic stroke
(HT-TBI); and (iv) a treatment and/or prevention for Alzheimer’s or other neuroinflammatory diseases (HT-ALZ). We also have assets being developed for
(i)  atopic  dermatitis  (also  known  as  eczema)  (BioLexa);  (ii)  a  treatment  for  asthma  and  allergies  using  inhalational  administration  (HT-004);  and  (iii)  a
treatment for acne as well as inflammatory bowel diseases (HT-003). In addition, we are continuing to evaluate a novel peptide that may be used to slow
the transmission of SARS-CoV-2. In addition, the Company is developing a diagnostic device via a mobile device. The Company also has interests in
certain other assets being developed by third parties (see Note 6 for a discussion of the Company’s agreement with Zylö Therapeutics, Inc. and Voltron
Therapeutics, Inc.).

Liquidity and capital resources

Accounting  Standards  Update  (“ASU”)  No.  2014-15,  Presentation  of  Financial  Statements  -  Going  Concern ,  requires  management  to  evaluate  the
Company’s ability to continue as a going concern one year beyond the filing date of the given financial statements. This evaluation requires management
to perform two steps. First, management must evaluate whether there are conditions and events that raise substantial doubt about the entity’s ability to
continue as a going concern. Second, if management concludes that substantial doubt is raised, management is required to consider whether it has plans
in place to alleviate that doubt. Disclosures in the notes to the consolidated financial statements are required if management concludes that substantial
doubt exists or that its plans alleviate the substantial doubt that was raised.

The Company has funded its operations from proceeds from the sale of equity and debt securities. The Company will require significant additional capital
to make the investments it needs to execute its longer-term business plan. The Company’s ability to successfully raise sufficient funds through the sale of
debt or equity securities when needed is subject to many risks and uncertainties and, even if it were successful, future equity issuances may result in
dilution to its existing shareholders and future debt securities may contain covenants that limit the Company’s operations or ability to enter into certain
transactions.

The  Company  believes  its  current  cash  is  sufficient  to  fund  operations  for  at  least  the  next  12  months  from  the  issuance  date  of  these  financial
statements. However, the Company will need to raise additional funding, through strategic relationships, public or private equity or debt financings, grants
or  other  arrangements,  to  develop  and  seek  regulatory  approvals  for  the  Company’s  current  and  future  product  candidates.  If  such  funding  is  not
available,  or  not  available  on  terms  acceptable  to  the  Company,  the  Company’s  current  development  plan  and  plans  for  expansion  of  its  general  and
administrative infrastructure may be curtailed.

On December 29, 2022, the Company entered into a securities purchase agreement with an accredited investor pursuant to which it agreed to sell an
aggregate of (i) 140,000 shares of common stock, (ii) warrants (the “December Pre-Funded Warrants”) to purchase up to  1,860,000 shares of common
stock and (iii) warrants (the “December Common Stock Warrants”) to purchase up to 2,500,000 shares of common stock at a purchase price of $ 5.00 per
share and accompanying warrant (less $0.001 for each December Pre-Funded Warrant and accompanying warrant) in a private placement for aggregate
gross proceeds of approximately $10 million, exclusive of placement agent commission and fees and other offering expenses. The closing of the offering
occurred on January 3, 2023. Each December Common Stock Warrant is exercisable for a period of five and one-half years from the issuance date at an
exercise price of $5.00 per share, subject to adjustment, and may, under certain circumstances, be exercised on a cashless basis. Each December Pre-
Funded  Warrant  is  exercisable  until  exercised  in  full  at  an  exercise  price  of  $0.001  per  share  and  may  be  exercised  on  a  cashless  basis.  In  addition,
pursuant to the terms of the offering, the Company issued H.C. Wainwright & Co., LLC warrants (“December Wainwright Warrants”) to purchase up to
100,000 shares of the Company’s common stock.  The December Wainwright Warrants are exercisable for a period of five and one-half years from the
issuance date at an exercise price of $6.25 per share, subject to adjustment, and may, under certain circumstances, be exercised on a cashless basis.

F-7

Reverse Stock Split

On  October  20,  2022,  the  Company  filed  a  Certificate  of  Change  (the  “Certificate  of  Change”)  with  the  Secretary  of  State  of  the  State  of  Nevada  to
effectuate a 1-for-25 reverse stock split (the “Reverse Stock Split”) of the Company’s issued and outstanding and authorized shares of common stock.
The Reverse Stock Split became effective on October 26, 2022. Shareholders who otherwise would have been entitled to receive fractional shares of
common  stock  had  their  holdings  rounded  up  to  the  next  whole  share.  All  references  to  common  stock,  convertible  preferred  stock  conversion  ratio,
warrants to purchase common stock, options to purchase common stock, restricted stock units, restricted stock awards, share data, per share data and
related information contained in the consolidated financial statements have been retrospectively adjusted to reflect the effect of the Reverse Stock Split
for all periods presented.

Note 2-Significant accounting policies

Basis of presentation and principles of consolidation

The Company’s consolidated financial statements have been prepared in conformity with accounting principles generally accepted in the United States of
America (“GAAP”).

The accompanying consolidated financial statements include the accounts of the Company’s wholly-owned subsidiary, Hoth Therapeutics Australia Pty

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Ltd, which was incorporated under the laws of the State of Victoria in Australia on June 5, 2019. All significant intercompany balances and transactions
have been eliminated in consolidation. 

Emerging growth company

As  an  emerging  growth  company,  the  Company  may  take  advantage  of  certain  exemptions  from  various  reporting  requirements  that  are  applicable  to
other public companies that are not emerging growth companies including, but not limited  to,  not  being  required  to  comply  with  the  auditor  attestation
requirements of Section 404 of the Sarbanes-Oxley Act of 2002, as amended, reduced disclosure obligations regarding executive compensation in its
periodic  reports  and  proxy  statements,  and  exemptions  from  the  requirements  of  holding  a  nonbinding  advisory  vote  on  executive  compensation  and
shareholder approval of any golden parachute payments not previously approved.

Further, Section 102(b)(1) of the Jumpstart Our Business Startups Act of 2012 (“JOBS Act”) exempts emerging growth companies from being required to
comply with new or revised financial accounting standards until private companies (that is, those that have not had a Securities Act of 1933, as amended,
registration  statement  declared  effective  or  do  not  have  a  class  of  securities  registered  under  the  Securities  Exchange  Act  of  1934,  as  amended)  are
required to comply with the new or revised financial accounting standards. The JOBS Act provides that an emerging growth company can elect to opt out
of  the  extended  transition  period  and  comply  with  the  requirements  that  apply  to  non-emerging  growth  companies  but  any  such  election  to  opt  out  is
irrevocable. The Company has elected not to opt out of such extended transition period which means that when a standard is issued or revised and it has
different application dates for public or private companies, the Company, as an emerging growth company, can adopt the new or revised standard at the
time  private  companies  adopt  the  new  or  revised  standard.  This  may  make  comparison  of  the  Company’s  financial  statement  with  another  public
company  that  is  neither  an  emerging  growth  company  nor  an  emerging  growth  company  that  has  opted  out  of  using  the  extended  transition  period
difficult or impossible because of the potential differences in accounting standards used.

F-8

Use of estimates

The preparation of consolidated financial statements in conformity with GAAP requires management to make estimates and assumptions that affect the
reported amounts of assets and liabilities and disclosure of contingent assets and liabilities at the date of the consolidated financial statements and the
reported amounts of expenses during the reporting periods. The most significant estimates in the Company’s consolidated financial statements relate to
stock-based compensation and the valuation allowance of deferred tax assets resulting from net operating losses. These estimates and assumptions are
based on current facts, historical experience and various other factors believed to be reasonable under the circumstances, the results of which form the
basis  for  making  judgments  about  the  carrying  values  of  assets  and  liabilities  and  the  recording  of  expenses  that  are  not  readily  apparent  from  other
sources. Actual results may differ materially and adversely from these estimates. To the extent there are material differences between the estimates and
actual results, the Company’s future results of operations will be affected.

Cash and cash equivalents

The Company considers all highly liquid investments purchased with original maturities of 90 days or less at acquisition to be cash equivalents. There
were no cash equivalents as of December 31, 2022 and 2021.

Marketable securities

Marketable securities are classified as trading and are carried at fair value. The Company’s marketable securities consist of a mutual fund which is valued
at a quoted market price.

Concentrations of credit risk and off-balance sheet risk

The Company has significant cash balances at financial institutions which, throughout the year, regularly exceed the federally insured limit of $ 250,000.
Any loss incurred or a lack of access to such funds could have a significant adverse impact on the Company’s financial condition, results of operations,
and cash flows. 

Fair Value of Financial Instruments

Financial Accounting Standards Board (“FASB”) Accounting Standards Codification (“ASC”) 820,  Fair Value Measurements ,  provides  guidance  on  the
development and disclosure of fair value measurements. Under this accounting guidance, fair value is defined as an exit price, representing the amount
that would be received to sell an asset or paid to transfer a liability in an orderly transaction between market participants at the measurement date. As
such, fair value is a market-based measurement that should be determined based on assumptions that market participants would use in pricing an asset
or a liability.

The  fair  value  of  the  Company’s  assets  and  liabilities,  which  would  qualify  as  financial  instruments  under  ASC  Topic  820,  approximates  the  carrying
amounts represented in the Company’s balance sheet, primarily due to their short-term nature.

The accounting guidance classifies fair value measurements in one of the following three categories for disclosure purposes:

Level 1: Quoted prices in active markets for identical assets or liabilities.

Level 2: Inputs other than Level 1 prices for similar assets or liabilities that are directly or indirectly observable in the marketplace.

Level 3: Unobservable  inputs  which are  supported  by  little  or  no  market  activity  and  values  determined  using  pricing  models,  discounted  cash  flow
methodologies, or similar techniques, as well as instruments for which the determination of fair value requires significant judgment or estimation.

F-9

In some circumstances, the inputs used to measure fair value might be categorized within different levels of the fair value hierarchy. In those instances,

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
the  fair  value  measurement  is  categorized  in  its  entirety  in  the  fair  value  hierarchy  based  on  the  lowest  level  input  that  is  significant  to  the  fair  value
measurement.

Fair value option - Note receivable

The guidance in ASC 825,  Financial Instruments, provides a fair value option election that allows entities to make an irrevocable election of fair value as
the initial and subsequent measurement attribute for certain eligible financial assets and liabilities. Unrealized gains and losses on items for which the fair
value option has been elected are reported in earnings. The decision to elect the fair value option is determined on an instrument-by-instrument basis
and must be applied to an entire instrument and is irrevocable once elected. Assets and liabilities measured at fair value pursuant to this guidance are
required to be reported separately in the Company’s consolidated balance sheets from those instruments using another accounting method.

Investment in joint ventures

Ownership  interests  in  entities  for  which  the  Company  has  significant  influence  that  are  not  consolidated  are  accounted  for  as  equity  method
investments. SEC Staff Announcement: “Accounting for Limited Partnership Investments” (codified in ASC 323-30-S99-1) guidance requires the use of
the  equity  method  unless  the  investor’s  interest  “is  so  minor  that  the  limited  partner  may  have  virtually  no  influence  over  partnership  operating  and
financial  policies.”  The  SEC  staff’s  position  is  that  investments  in  limited  partnerships  of  greater  than 3%  to  5%  are  considered  more  than  minor  and,
therefore, should be accounted for using the equity method or fair value option. Investments accounted for using the equity method may be reported on
a lag up to three months if financial statements of the investee are not available in sufficient time for the investor to apply the equity method as of the
current  reporting  date.  The  determination  of  whether  an  investee’s  results  are  recorded  on  a  lag  is  made  on  an  investment-by-investment  basis.  This
investment in joint ventures is further described in Note 6 of these consolidated financial statements.

Research and development costs

Research  and  development  costs,  including  acquired  in-process  research  and  development  expenses  for  which  there  is  no  alternative  future  use,  are
expensed as incurred. Advance payments for goods and services that will be used in future research and development activities are expensed when the
activity has been performed or when the goods have been received rather than when the payment is made.

Stock-based compensation

The  Company  accounts  for  share-based  payment  awards  exchanged  for  services  at  the  estimated  grant  date  fair  value  of  the  award.  Stock  options
issued under the Company’s long-term incentive plans are granted with an exercise price equal to no less than the market price of the Company’s stock
at the date of grant and expire up to ten years from the date of grant. These options generally vest over a one to five year period . The Company accounts
for forfeited awards as they occur.

The Company estimates the fair value of stock option grants using the Black-Scholes option pricing model and the assumptions used in calculating the
fair  value  of  stock-based  awards  represent  management’s  best  estimates  and  involve  inherent  uncertainties  and  the  application  of  management’s
judgment.

Expected Term - The expected term of options represents the period that the Company’s stock-based awards are expected to be outstanding

based on the simplified method, which is the half-life from vesting to the end of its contractual term.

Expected Volatility - The Company computes stock price volatility over expected terms based on its historical common stock trading prices.

Risk-Free Interest Rate  - The Company bases the risk-free interest rate on the implied yield available on U.S. Treasury zero-coupon issues with

an equivalent remaining term.

Expected  Dividend -  The  Company  has  never  declared  or  paid  any  cash  dividends  on  its  common  shares  and  does  not  plan  to  pay  cash

dividends in the foreseeable future, and, therefore, uses an expected dividend yield of zero in its valuation models.

F-10

Income taxes

Income  taxes  are  recorded  in  accordance  with  ASC  740,  Income Taxes   (“ASC  740”),  which  provides  for  deferred  taxes  using  an  asset  and  liability
approach. The Company recognizes deferred tax assets and liabilities for the expected future tax consequences of events that have been included in the
consolidated  financial  statements  or  tax  returns.  Deferred  tax  assets  and  liabilities  are  determined  based  on  the  difference  between  the  financial
statement and tax bases of assets and liabilities using enacted tax rates in effect for the year in which the differences are expected to reverse. Valuation
allowances are provided, if based upon the weight of available evidence, it is more likely than not that some or all of the deferred tax assets will not be
realized.

The  Company  accounts  for  uncertain  tax  positions  in  accordance  with  the  provisions  of  ASC  740.  When  uncertain  tax  positions  exist,  the  Company
recognizes  the  tax  benefit  of  tax  positions  to  the  extent  that  the  benefit  would  more  likely  than  not  be  realized  assuming  examination  by  the  taxing
authority. The determination as to whether the tax benefit will more likely than not be realized is based upon the technical merits of the tax position as well
as consideration of the available facts and circumstances.

Net loss per share

Net loss per share is computed by dividing net loss by the weighted average number of common stock outstanding during the period. Since the Company
had a net loss in the periods presented, basic and diluted net loss per common share are the same. The following were excluded from the computation of
diluted shares outstanding due to the losses for each period presented, as they would have had an anti-dilutive impact on the Company’s net loss:

Potentially dilutive securities
Warrants
Options
Non-vested restricted stock awards

As of December 31,
2022

2021

402,840     
104,651     
3,384     

402,840 
52,851 
100 

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
 
   
   
   
Total

Recent accounting pronouncements

510,875     

455,791 

Currently, management does not believe that any recently issued, but not yet effective accounting pronouncements, if currently adopted, would have a
material impact on the Company’s consolidated financial statements.

Note 3-License agreements

The following summarizes the Company’s research and development expenses for licenses acquired during the years ended December 31, 2022 and
2021:

The George Washington University
Isoprene Pharmaceuticals, Inc.
North Carolina State University
Virginia Commonwealth University
Chelexa Biosciences, Inc. and the University of Cincinnati
Adjustment

F-11

For the Years Ended
December 31,

2022

2021

66,586    $
-     
27,500     
-     
7,500     
(15,000)    
86,586    $

99,782 
15,000 
30,000 
30,000 
- 
- 
174,782 

  $

  $

The George Washington University

During the year ended December 31, 2022, the Company recorded an expense of approximately $ 53,000 for related to warrants granted to The George
Washington  University  (“GW”)  pursuant  to  the  patent  license  agreement  with  GW  dated  February  1,  2020  (“GW  Patent  License  Agreement”)  and  the
patent  license  agreement  with  GW  dated  August  7,  2020  (“Second  GW  Patent  License  Agreement”).  The  Company  also  recorded  $14,000  the  year
ended December 31, 2022 for a license maintenance fee.

During  the  year  ended  December  31,  2021,  the  Company  recorded  an  expense  of  approximately  $ 0.1  million  for  related  to  warrants  granted  to  GW
pursuant to the GW Patent License Agreement and the Second GW Patent License Agreement.

Isoprene Pharmaceuticals, Inc.

During  the  years  ended  December  31,  2022  and  2021,  the  Company  paid  $ 0  and  $15,000,  respectively,  for  the  license  fee  associated  with  the
sublicense agreement by and between the Company and Isoprene Pharmaceuticals, Inc. dated July 30, 2020.

North Carolina State University

During the year ended December 31, 2022, the Company paid approximately $ 28,000 for the license fee associated with the license agreement by and
between the Company and North Carolina State University dated February 25, 2021.

During the year ended December 31, 2021, the Company paid $ 30,000 for the license fee.

Virginia Commonwealth University

During the year ended December 31, 2022 and 2021, the Company paid $ 0 and $30,000, respectively, for annual maintenance fees associated with the
exclusive license agreement between the Company and Virginia Commonwealth University Intellectual Property Foundation.

As of December 31, 2022, the Company accrued $ 150,000 for five years of annual minimum payments and $ 125,000 for annual maintenance fees.

As of December 31, 2021, the Company accrued $ 285,000 for five years of annual minimum payments and $ 30,000 for annual maintenance fees.

Chelexa Biosciences, Inc. and the University of Cincinnati

During the year ended December 31, 2022, the Company paid $ 2,500 for the annual license maintenance fee and $ 5,000 for the yearly minimum annual
royalty fee associated with the Assignment and Assumption Agreement by and between the Company and Chelexa Biosciences dated May 14, 2020.

Note 4-Note Receivable

Pursuant to the sublicense agreement dated July 30, 2020 by and between the Company and Isoprene Pharmaceuticals, Inc. (“Isoprene”), the Company
made an investment of $50,000 in Isoprene in the form of a convertible promissory note (the “Isoprene Note”) on September 10, 2020. The Isoprene Note
was due to mature on September 10, 2022 and accrued interest at a rate equal to the lower of: (i) the highest lawful rate permitted under applicable law
and (ii) 6% per annum. The Isoprene Note could not be prepaid without the prior written consent of the Company; provided, however, that if the Isoprene
Note had not been converted in connection with a Qualified Financing (as defined herein) or a Change of Control (as defined in the Isoprene Note) by the
two year anniversary of the date of the issuance of the Isoprene Note, Isoprene could elect, in its sole discretion, to repay the Isoprene Note and any
accrued interest thereon. In the event a Qualified Financing occurred before the Isoprene Note was repaid in full on the maturity date or the conversion of
such note pursuant to a Change of Control, the Isoprene Note could be converted into such number of convertible preferred stock issued in the Qualified
Financing equal to the balance of such note divided by the Capped Conversion Price. “Qualified Financing” means the first sale of Isoprene’s convertible
preferred stock in a private financing that results in gross proceeds of at least $5 million. “Capped Conversion Price” means the lesser of (i) the per share
or  unit  price  in  the  Qualified  Financing  and  (ii)  an  amount  determined  by  dividing  (A)  $15  million  by  (B)  the  fully  diluted  capitalization  of  Isoprene
immediately prior to the conversion of the Isoprene Note. In the event a Change of Control occurred before the Isoprene Note was repaid in full on the
maturity  date  or  the  conversion  of  such  note  pursuant  to  a  Qualified  Financing,  the  Isoprene  Note  could  be  converted  into  such  number  of  shares  of

   
 
 
 
 
 
 
 
 
 
 
   
 
   
   
   
   
   
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Isoprene’s common stock equal to the quotient obtained by dividing (i) the balance of the Isoprene Note by (ii) two times the fair market value of a share
of Isoprene common stock as set for in the acquisition agreement pertaining to such Change of Control. As of the maturity date of the Isoprene Note,
neither a Qualified Financing nor a Change of Control had occurred, and the Isoprene Note of $50,000 and accrued interest of approximately $ 6,000 was
paid off on October 21, 2022.

F-12

Note 5-Investments in Marketable Equity Securities

The realized gain or loss, unrealized gain or loss, and dividend income related to marketable equity securities for the years ended December 31, 2022
and 2021, which are recorded as a component of other income (expenses) on the consolidated statements of operations and comprehensive loss, are as
follows:

Unrealized gain (loss)
Realized loss
Dividend income

For the Years Ended
December 31,

2022

2021

  $

  $

119,870    $
(567,692)    
60,913     
(386,909)   $

(176,974)
(41,808)
66,100 
(152,682)

Note 6-Fair Value of Financial Assets and Liabilities

The following tables present the Company’s assets and liabilities that are measured at fair value at December 31, 2022 and 2021:

Assets

Marketable securities - mutual funds
Investment in joint ventures
Note receivable - current

Assets

Marketable securities - mutual funds
Investment in joint ventures
Note receivable - current

Level 3 Measurement

Fair value measured at December 31, 2022

Total at

December 31,    

2022

Quoted
prices in
active
markets
(Level 1)

Significant
other
observable
inputs
(Level 2)

Significant
unobservable
inputs
(Level 3)

  $
  $
  $

209,320    $
33,000    $
-    $

209,320    $
-    $
-    $

     -    $
-    $
-    $

- 
33,000 
- 

Fair value measured at December 31, 2021

Total at 

December 31,    

2021

Quoted
prices 
in active 
markets
(Level 1)

Significant
other
observable
inputs
(Level 2)

Significant
unobservable 
inputs
(Level 3)

  $
  $
  $

1,892,837    $
410,000    $
50,000    $

1,892,837    $
-    $
-    $

      -    $
-    $
-    $

- 
410,000 
50,000 

The following table sets forth a summary of the changes in the fair value of the Company’s Level 3 financial assets that are measured at fair value on a
recurring basis:

Investment in joint ventures at fair value at December 31, 2020
Investment in joint ventures at fair value at December 31, 2021

Change in fair value of investments in joint ventures

Investment in joint ventures at fair value at December 31, 2022

  $

  $

410,000 
410,000 
(377,000)
33,000 

F-13

Investment in joint ventures

The  Company  has  elected  to  measure  the  investment  in  joint  ventures  using  the  fair  value  option  at  each  reporting  date.  Under  the  fair  value  option,
bifurcation  of  an  embedded  derivative  is  not  necessary,  and  all  related  gains  and  losses  on  the  host  contract  and  derivative  due  to  change  in  the  fair
value will be reflected in interest income and other income (expense), net in the consolidated statements of operations and comprehensive loss.

The value at which the Company’s investment in joint ventures is carried on its books is adjusted to estimated fair value at the end of each quarter, taking
into account general economic and stock market conditions and those characteristics specific to the underlying investments.

Investment in HaloVax

On  March  23,  2020,  the  Company  entered  into  a  Development  and  Royalty  Agreement  (the  “Development  and  Royalty  Agreement”)  with  Voltron
Therapeutics,  Inc.  (“Voltron”)  to  form  a  joint  venture  entity  named  HaloVax,  LLC  (“HaloVax”)  to  jointly  develop  potential  product  candidates  for  the

 
 
 
 
 
 
 
 
 
 
   
 
   
   
 
 
 
 
 
 
 
 
 
   
   
 
 
 
   
   
   
 
   
     
     
     
 
 
 
 
 
 
 
   
   
 
 
 
   
   
   
 
   
     
     
     
 
 
 
 
   
   
 
 
 
 
 
 
 
prevention  of  COVID-19  based  upon  certain  technology  that  had  been  exclusively  licensed  by  Voltron  from  The  General  Hospital  Corporation  (d/b/a
Massachusetts  General  Hospital).  Pursuant  to  the  Development  and  Royalty  Agreement,  the  Company  is  entitled  to  receive  sales-based  royalties.  In
addition, pursuant to the terms of the Development and Royalty Agreement, on March 23, 2020, the Company and HaloVax entered into a Membership
Interest Purchase Agreement pursuant to which the Company purchased 5% of HaloVax’s outstanding membership interests for $ 250,000 on March 27,
2020 (the “Initial Closing Date”) and had the option to purchase up to an additional 25% of HaloVax’s membership interests (for $ 3,000,000 (inclusive of
the $250,000)), which option expired 30 days after the Initial Closing Date. On May 28, 2020, the Company entered into a Membership Interest Purchase
Agreement to purchase 1% of HaloVax’s outstanding membership interest for a purchase price of $ 100,000.

During  the  fourth  quarter  of  2022,  the  Company  identified  indicators  of  impairment  for  the  HaloVax  investment  as  a  result  of  adverse  changes  in
HaloVax’s business operations, including liquidity concerns. As a result, the Company recorded an impairment charge of approximately $0.4 million in the
fourth quarter of 2022. The investment in HaloVax was valued at $0 and $350,000 as of December 31, 2022 and 2021.

Investment in Zylö

In  connection  with  the  Company’s  March  2020  underwritten  public  offering  of  shares  of  its  common  stock,  on  May  4,  2020,  the  Company  purchased
120,000 shares of Zylö’s Class B common stock for $ 60,000. No change in fair value occurred during the nine months ended September 30, 2022. On
December  8,  2021,  the  Company  entered  into  a  third  amendment  (the  “Zylö  Amendment”)  to  the  Exclusive  Sublicense  Agreement  with  Zylö  originally
dated August 19, 2019, pursuant to which the Company licensed its novel cannabinoid therapeutic, HT-005 for lupus patients, back to Zylö. Pursuant to
the Zylö Amendment, on December 6, 2021, Zylö issued the Company 100,000 shares of its Class B common stock. In addition, pursuant to the Zylö
Amendment, within 90 days following a sale by Zylö of all of its assets and rights related to HT-005 to a third-party (a “Sale”), Zylö shall pay the Company
a  low  single  digit  percent  of  the  net  proceeds  received  by  it  attributable  to  HT-005  in  the  United  States  and  Canada  and  their  respective  territories
(collectively,  the  “Territory”)  for  the  purposes  of  therapeutic  uses  related  to  lupus  in  humans  (the  “Field”).  After  the  Sale,  any  and  all  rights  of  the
Company  pursuant  to  the  Exclusive  Sublicense  Agreement,  including  all  amendments  thereto,  shall  terminate.  Furthermore,  pursuant  to  the  Zylö
Amendment,  following  the  date  of  the  first  commercial  sale  of  HT-005  in  the  Territory,  in  the  Field,  Zylö  shall  pay  the  Company  (i)  a  low  single  digit
percent of the Net Sales (as defined in the Exclusive Sublicense Agreement) of HT-005 in the event HT-005 is sold in the Territory and (ii) a low double
digit percent of any royalty that Zylö receives through the sublicense to a third-party based on Net Sales of HT-005 in the Territory which payments shall
continue  in  each  country  in  the  Territory  until  expiration  of  the  last-to-expire  Valid  Claim  (as  defined  in  the  Exclusive  Sublicense  Agreement).  Zylö
conducted  a  409A  valuation  of  their  Class  B  common  stock  and  valued  its  share  price  at  $0.15  per  share.  This  value  was  ratified  by  Zylö’s  board  of
directors in December 2022. Therefore, the Company recorded approximate $27,000 in unrealized loss on this investment during the second quarter of
2022. The investment in Zylö was valued at $33,000 and $60,000 as of December 31, 2022 and 2021, respectively.

F-14

Note 7-Stockholders’ Equity

Preferred Stock

The Company is authorized to issue up to  10,000,000 shares of preferred stock. This preferred stock may be issued in one or more series, and shall have
such designations, preferences and relative, participating, optional or other special rights and qualifications, limitations or restrictions thereof as shall be
determined at the time of issuance by the Company’s board of directors without further action by the Company’s shareholders. As of December 31, 2022,
5,000,000  shares  of  the  Company’s  preferred  stock  has  been  designated  as  Series  A  Convertible  Preferred  Stock  and  2,000,000  shares  of  the
Company’s preferred stock has been designated as Series B Preferred Stock.

Series A Convertible Preferred Stock

The shares of Series A Convertible Preferred Stock are not mandatorily redeemable and do not embody an unconditional obligation to settle in a variable
number of equity shares. As such, the shares of Series A Convertible Preferred Stock are classified as permanent equity on the consolidated balance
sheets.  The  holders’  contingent  redemption  right  in  the  event  of  certain  deemed  liquidation  events  does  not  preclude  permanent  equity  classification.
Further, the shares of Series A Convertible Preferred Stock are considered an equity-like host for purposes of assessing embedded derivative features for
potential bifurcation. The embedded conversion feature is considered to be clearly and closely related to the associated convertible preferred stock host
instrument and therefore was not bifurcated from the equity host.

Series B Preferred Stock

On November 2, 2022, the Company filed a Certificate of Designation of the Series B Preferred Stock (the “Certificate of Designation”) with the Secretary
of State of the State of Nevada to create a new class of Series B Preferred Stock, par value $0.0001 per share (the “Series B Preferred Stock”). The
Certificate of Designation designated 2,000,000 shares of authorized preferred stock as Series B Preferred Stock. The Series B Preferred Stock were not
entitled  to  receive  dividends  or  any  other  distributions.  The  Series  B  Preferred  Stock  were  entitled  to  ten  votes  per  share  and  voted  together  with  the
Company’s  issued  and  outstanding  shares  of  common  stock  as  a  single  class  exclusively  with  respect  to  the  Authorized  Stock  Increase  (as  defined
herein).  The  Series  B  Preferred  Stock  had  no  rights  as  to  any  distribution  or  assets  of  the  Company  upon  a  liquidation,  bankruptcy,  reorganization,
merger,  acquisition,  sale,  dissolution  or  winding  up  of  the  Company.  The  outstanding  shares  of  Series  B  Preferred  Stock  were  redeemed  in  whole  an
aggregate price of $10automatically and effective immediately after the effectiveness of the Authorized Stock Increase.

On  November  2,  2022,  the  Company  entered  into  a  Subscription  and  Investment  Representation  Agreement  with  an  investor  pursuant  to  which  the
Company  issued  and  sold 2,000,000  shares  of  its  newly  designated  Series  B  Preferred  Stock  to  such  purchaser  for  an  aggregate  purchase  price  of
$1,000.

On December 12, 2022, the Company’s shareholders approved the an increase to the number of authorized shares of the Company’s common stock
from 3,000,000 to 50,000,000 shares (the “Authorized Stock Increase”). On December 13, 2022, upon filing a Certificate of Amendment to its Articles of
Incorporation,  as  amended,  to  increase  its  authorized  shares  of  common  stock,  the  Series  B  Preferred  Stock  was  automatically  redeemed  for  an
aggregate of $10.

Common Shares

On December 12, 2022, shareholders of the Company approved an increase to the number of authorized shares of the Company’s common stock from
3,000,000  shares  to  50,000,000 shares, and on December 13, 2022, the Company filed a Certificate of Amendment to its Articles of Incorporation, as
amended, to effectuate such increase.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
F-15

Securities Purchase Agreements

On  January  5,  2021,  the  Company  entered  into  a  securities  purchase  agreement  with  certain  accredited  investors  pursuant  to  which  the  Company
offered and sold to the investors an aggregate of 99,010 shares of its common stock and warrants to purchase up to  49,505 shares of common stock in a
private placement for aggregate net proceeds to the Company of $4.6 million, after deducting estimated offering expenses payable by the Company. The
combined purchase price for each share of common stock and accompanying warrant to purchase one half of a share of common stock was $50.50. The
closing of the offering occurred on January 7, 2021. Each warrant is exercisable for a period of five years from the issuance date at an exercise price of
$56.25  per  share,  subject  to  adjustment,  and  may  be  exercised  on  a  cashless  basis.  In  addition,  pursuant  to  the  terms  of  the  offering,  the  Company
issued The Benchmark Company, LLC (“Benchmark”) warrants to purchase up to  7,426 shares of the Company’s common stock. Benchmark’s warrants
are exercisable for a period of five years from the closing date of the offering at an exercise price of $ 56.25 per share, subject to adjustment, and may be
exercised on a cashless basis.

On  March  8,  2021,  the  Company  entered  into  a  securities  purchase  agreement  with  certain  institutional  and  accredited  investors  pursuant  to  which  it
offered and sold to the investors 273,079 shares of common stock, pre-funded warrants (the “March Pre-Funded Warrants”) to purchase up to  30,719
shares of common stock and warrants (the “March Common Stock Warrants”) to purchase up to 303,798 shares of common stock in a private placement
for  aggregate  net  proceeds  to  the  Company  of  $13.5  million,  after  deducting  estimated  offering  expenses  payable  by  the  Company.  The  combined
purchase price for each share of common stock and accompanying warrant was $49.375. The closing of the offering occurred on March 10, 2021. Each
March  Common  Stock  Warrant  is  exercisable  for  a  period  of three years  from  the  issuance  date  at  an  exercise  price  of  $ 46.50  per  share,  subject  to
adjustment,  and  may  be  exercised  on  a  cashless  basis.  Each  March  Pre-Funded  Warrant  is  exercisable  until  exercised  in  full  at  an  exercise  price  of
$0.025 per share and may be exercised on a cashless basis. In addition, pursuant to the terms of the offering, the Company issued H.C. Wainwright &
Co., LLC warrants (“March Wainwright Warrants”) to purchase up to 15,190 shares of the Company’s common stock. The March Wainwright Warrants
are exercisable for a period of three years from the issuance date at an exercise price of $61.72 per share, subject to adjustment, and may be exercised
on a cashless basis.

On December 29, 2022, the Company entered into a securities purchase agreement with an accredited investor pursuant to which it agreed to sell an
aggregate  of  (i) 140,000 shares of common stock, (ii) December Pre-Funded Warrants to purchase up to  1,860,000 shares of common stock and (iii)
December Common Stock Warrants to purchase up to 2,500,000 shares of common stock at a purchase price of $ 5.00 per share and accompanying
warrant  (less  $0.001  for  each  December  Pre-Funded  Warrant  and  accompanying  warrant)  in  a  private  placement  for  aggregate  gross  proceeds  of
approximately  $10  million,  exclusive  of  placement  agent  commission  and  fees  and  other  offering  expenses.  The  closing  of  the  offering  occurred  on
January  3,  2023. Each December Common Stock Warrant is exercisable for a period of five and one-half years from the issuance date at an exercise
price of $5.00 per share, subject to adjustment, and may, under certain circumstances, be exercised on a cashless basis.
 Each December Pre-Funded
Warrant is exercisable until exercised in full at an exercise price of $0.001 per share and may be exercised on a cashless basis. In addition, pursuant to
the terms of the offering, the Company issued H.C. Wainwright & Co., LLC the December Wainwright Warrants to purchase up to 100,000 shares of the
Company’s  common  stock. The  December  Wainwright  Warrants  are  exercisable  for  a  period  of  five  and  one-half  years  from  the  issuance  date  at  an
exercise price of $6.25 per share, subject to adjustment, and may, under certain circumstances, be exercised on a cashless basis.

Public Offering of Securities

On April 14, 2022, the Company closed an underwritten public offering of  329,412 shares of the Company’s common stock at a price to the public of
$21.25 per share (the “Offering Price”). Pursuant to the terms of an underwriting agreement dated April 11, 2022 between the Company and EF Hutton,
division of Benchmark Investments, LLC, as representative of the several underwriters (the “Underwriters”), the Company granted the Underwriters a 45-
day option to purchase up to an additional 49,412 shares of the Company’s common stock to cover over-allotments, if any, at the Offering Price less the
underwriting discounts and commissions. The net proceeds to the Company from the sale of the shares, after deducting the underwriting discounts and
commissions and other estimated offering expenses payable by the Company, were $6.0 million. The Underwriters did not exercise their over-allotment
option.

F-16

2018 Equity Incentive Plan

The compensation committee of the board of directors increased the number of shares reserved pursuant to the Company’s 2018 Equity Incentive Plan
(“2018 Plan”) by 26,878 shares effective as of January 1, 2021, such that as of January 1, 2021, the Company had an aggregate of  66,878 shares of
common stock reserved for issuance pursuant to the 2018 Plan. On June 24, 2021, at the annual meeting of shareholders, shareholders of the Company
approved an amendment to the  2018  Plan  to  further  increase  the  number  of  shares  reserved  for  issuance  thereunder  from 66,878  shares  to  146,878
shares. On February 2, 2022, the compensation committee of the board of directors further increased the number of shares reserved for issuance under
the 2018 Plan from 146,878 shares to  156,878 shares. On January 11, 2023, the compensation committee of the board of directors further increased the
number of shares reserved for issuance under the 2018 Plan from 156,878 shares to  166,878 shares.

2022 Equity Incentive Plan

On March 24, 2022, the Company’s board of directors adopted the Hoth Therapeutics, Inc. 2022 Omnibus Equity Incentive Plan (the “2022 Plan”) initially
reserving 96,000 shares of the Company’s common stock for issuance thereunder. The 2022 Plan became effective on June 23, 2022 upon approval of
the 2022 Plan by the Company’s shareholders at the Company’s annual meeting of shareholders.

Restricted Stock Awards

A summary of the Company’s restricted stock awards granted under the equity incentive plans during the years ended December 31, 2022 and 2021 is
as follows:

Number of
Restricted
Stock
Awards

Weighted
Average
Grant Day
Fair Value  

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
Nonvested at December 31, 2020

Granted
Vested

Nonvested at December 31, 2021

Granted
Vested

Nonvested at December 31, 2022

385    $

4,000     
(4,285)    
100    $
5,075     
(1,791)    
3,384    $

46.61 

31.00 
30.89 
75.00 
3.16 
7.17 
3.16 

As of December 31, 2022, there is approximately $ 10,000 of unrecognized stock-based compensation expense related to restricted stock awards. The
weighted average remaining contractual terms of unvested restricted stock awards is approximately 1.45 years at December 31, 2022.

Stock Options

During  the  year  ended  December  31,  2022,  pursuant  to  and  subject  to  the  available  number  of  shares  reserved  under  the  2018  Plan,  the  Company
issued an aggregate of 51,800 options to the Company’s directors. The aggregate grant date fair value of these options was approximately $ 0.6 million.

During  the  year  ended  December  31,  2021,  pursuant  to  and  subject  to  the  available  number  of  shares  reserved  under  the  2018  Plan,  the  Company
issued an aggregate of 25,280 options to the Company’s directors. The aggregate grant date fair value of these options was approximately $ 1.1 million.

F-17

The fair value of options granted in 2022 and 2021 was estimated using the following assumptions:

Exercise price
Term (years)
Expected stock price volatility
Risk-free rate of interest

For the Years Ended
December 31,

2022

2021

  $

  $

14.75 
10.0 
96.10%   
2.10%   

52.75 
10.0 
119.20%
0.42%

A summary of option activity under the Company’s stock option plan for the years ended December 31, 2022 and 2021 is presented below:

Outstanding as of December 31, 2020

Employee options issued

Outstanding as of December 31, 2021

Employee options issued

Outstanding as of December 31, 2022
Options vested and exercisable as of December 31, 2022

Number of
Shares

Weighted
Average
Exercise
Price

Total
Intrinsic
Value

27,571    $
25,280     
52,851    $
51,800     
104,651    $
104,651    $

112.94    $
52.75     
84.15    $
14.75     
49.80    $
49.80    $

Weighted
Average
Remaining
Contractual
Life
(in years)

-     
-     
-     
-     
-     
-     

8.8 
9.3 
8.6 
9.2 
8.3 
8.3 

All stock compensation associated with the amortization of employee stock option expense was recorded as a component of compensation and related
expense in the consolidated statements of operations and comprehensive loss. All stock compensation associated with the amortization of nonemployee
stock option expense was recorded as a component of professional fees in the consolidated statements of operations and comprehensive loss.

Estimated future stock-based compensation expense relating to unvested stock options is approximately $ 0.

Stock Based Compensation

Stock-based compensation expense for the years ended December 31, 2022 and 2021 was as follows:

Employee stock option awards
Employee restricted stock awards
Non-employee restricted stock awards
Non-employee stock warrant awards

For the Years Ended
December 31,

2022

560,376    $
7,836     
-     
52,586     
620,798    $

2021
1,092,428 
6,611 
124,000 
99,782 
1,322,821 

  $

  $

Employee and director related stock-based compensation was included in compensation and related expenses, and non-employee related stock-based
compensation  was  included  in  professional  fees  and  research  and  development  related  with  licenses  acquisition  in  the  consolidated  statements  of
operations and comprehensive loss.

F-18

   
   
   
   
   
   
   
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
   
   
   
 
 
 
 
   
   
   
 
   
   
   
   
   
   
 
 
 
 
 
 
 
 
 
 
   
 
   
   
   
 
 
 
 
 
Warrants

A summary of warrant activity for the years ended December 31, 2022 and 2021 is presented below:

Outstanding as of December 31, 2020

Issued
Expired
Exercised

Outstanding as of December 31, 2021
Outstanding as of December 31, 2022
Warrants exercisable as of December 31, 2022

Number of
Warrants

Weighted
Average
Exercise
Price

Total
Intrinsic
Value

49,417    $
406,643     
(8,151)    
(45,069)    
402,840    $
402,840    $
401,312    $

76.85    $
44.92     
200.00     
7.98     
49.83    $
49.83    $
49.73    $

696,334     
-     
-     
-     
-     
-     
-     

Weighted
Average
Remaining
Contractual
Life
(in years)

3.4 
2.3 
- 
- 
2.3 
1.4 
1.5 

The Company has determined that the warrants should be accounted as a component of stockholders’ equity.

Note 8-Commitments and contingencies

The Company leases office space for approximately $ 4,500 a month. Rent expense for the years ended December 31, 2022 and 2021 was approximately
$67,000 and $47,000, respectively. The Company is not a party to a lease that is in excess of 12 months.

Litigation

The Company is not currently a party to any material legal proceedings and is not aware of any pending or threatened claims. From time to time, the
Company may be subject to various legal proceedings and claims that arise in the ordinary course of its business activities.

Note 9-Income taxes

The table below presents the components of the provision for taxes:

The Company's provision is primarily driven by the full valuation allowance in 2022 and 2021.

Current
U.S. Federal
U.S. State
U.S. Foreign

Total current provision

Deferred
U.S. Federal
U.S. State
U.S. Foreign

Total deferred benefit
Change in valuation allowance
Total provision for income taxes

  $

As of December 31,
2022

2021

-    $

-     

-     
-     
-     
-     

- 
- 

- 
- 
- 
- 
- 

  $

-     
      -    $

    - 

F-19

At  December  31,  2022  and  2021,  the  tax  effects  of  the  temporary  differences  and  carryforwards  that  give  rise  to  deferred  tax  assets  consist  of  the
following:

Net operating loss carryforwards
Research and development credits
Capitalized research costs
Equity based compensation
Licenses acquired
Depreciation
Accruals and other temporary differences

Gross deferred tax assets

Depreciation
Accruals and other temporary differences

Less valuation allowance
Net deferred taxes

As of December 31,
2022

2021

  $

  $

10,378,471    $
-     
1,211,477     
670,035     
338,239     
-     
215,152     
12,813,374     
-     
-     
(12,813,374)    
  $

-

6,752,718 
444,866 
- 
590,050 
341,171 
72 
155,816 
8,284,693 
- 
- 
(8,284,693)
- 

A reconciliation of the statutory income tax rates and the Company’s effective tax rate for the years ended December 31, 2022 and 2021 is as follows:

 
 
 
 
   
   
   
 
   
   
   
   
   
   
   
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
 
 
 
   
 
 
   
      
   
  
   
      
  
   
   
   
   
   
      
   
  
 
 
 
 
 
 
 
 
 
   
 
 
 
 
   
 
 
   
   
   
   
   
   
   
   
   
   
 
 
Tax provision at statutory rate
State taxes, net of federal benefit
Impact of non-U.S. earnings
Permanent items
Credits
Equity compensation
Rate changes
Foreign rate differential
RTP and other
Other
Increase/(decrease) in valuation reserve
Total

Years Ended
December 31,

2022

2021

21.0%    
9.5%    
0.0%    
(0.9)%   
0.0%    
(0.1)%   
0.0%    
0.0%    
10.0%    
0.0%    
(39.6)%   
0.0%    

21.0%
8.2%
0.0%
(1.8)%
6.7%
(2.4)%
2.4%
0.0%
0.0%
(0.3)%
(30.0)%
3.80%

The Company has determined, based upon available evidence, that it is more likely than not that the net deferred tax assets will not be realized and,
accordingly, has provided a full valuation allowance against its net deferred tax assets.

As of December 31, 2022, the Company has net operating loss carryforwards of approximately $ 32.9 million and $ 65.8 million available to reduce future
taxable income, if any, for Federal and state income tax purposes, respectively. Approximately $ 1.5 million of Federal net operating losses can be carried
forward  to  future  tax  years  and  expire  in  2037.  The  Federal  net  operating  loss  generated  during  the  years  ended  after  December  31,  2017  of
approximately $31.4  million  can  be  carried  forward  indefinitely;  however,  the  deduction  for  net  operating  losses  incurred  in  tax  years  beginning  after
January  1,  2018  is  limited  to 80%  of  annual  taxable  income.  In  addition,  the  Company  had  approximately  $ 0.3  million  of  net  operating  losses  at  its
subsidiary located in Australia, as of December 31, 2022.

As required by the 2017 Tax Cuts and Jobs Act and effective in 2022, the deferred tax asset as of December 31, 2022 included $ 1.2 million related to the
mandatory capitalization of research and development expenses.

F-20

As of December 31, 2022, the Company does not have any research and development credits available to reduce future income taxes for Federal and
state income tax purposes. The Federal credits expire if not utilized by 2042.

The utilization of the Company’s net operating loss carryforwards and research tax credit carryovers could be subject to annual limitations under Section
382 and 383 of the Internal Revenue Code of 1986, as amended (the “Code”), and similar state tax provisions, due to ownership change limitations that
may have occurred previously or that could occur in the future. These ownership changes limit the amount of net operating loss carryforwards and other
deferred tax assets that can be utilized to offset future taxable income and tax, respectively. In general, an ownership change, as defined by Section 382
and 383 of the Code, results from transactions increasing ownership of certain stockholders or public groups in the stock of the corporation by more than
50 percent points over a three-year period. The Company has not conducted an analysis of an ownership change under Section 382 of the Code. To the
extent that a study is completed and an ownership change is deemed to occur, the Company’s net operating losses and tax credits could be limited.

At December 31, 2022 and 2021, the Company did not have any significant uncertain tax positions. The Company will recognize interest and penalties
related to uncertain tax positions, as applicable, in income tax expense. As of December 31, 2022 and 2021, the Company had no accrued interest or
penalties related to uncertain tax positions and no amounts have been recognized in the Company’s statements of operations. The Company does not
anticipate a material change to unrecognized tax benefits in the next twelve months.

All of the Company’s tax years will remain open for examination by the Federal and state tax authorities from the date of utilization of the net operating
loss.

Note 10-Subsequent Events

The Company has evaluated subsequent events and transactions that occurred up to the date the consolidated financial statements were issued. Based
upon this review, except for as noted below, the Company did not identify any subsequent events that would have required adjustment or disclosure in
the consolidated financial statements.

On December 29, 2022, the Company entered into a securities purchase agreement with certain institutional and accredited investors pursuant to which
it agreed to sell an aggregate of (i) 140,000 shares of common stock, (ii) December Pre-Funded Warrants to purchase up to 1,860,000 shares of common
stock  and  (iii)  December  Common  Stock  Warrants  to  purchase  up  to  2,500,000  shares  of  common  stock  at  a  purchase  price  of  $5.00  per  share  and
accompanying  warrant  (less  $0.001  for  each  December  Pre-Funded  Warrant  and  accompanying  warrant)  in  a  private  placement  for  aggregate  gross
proceeds  of  approximately  $10  million,  exclusive  of  placement  agent  commission  and  fees  and  other  offering  expenses.  The  closing  of  the  Offering
occurred on January 3, 2023. Each December Common Stock Warrant is exercisable for a period of five and one-half years from the issuance date at an
exercise price of $5.00 per share, subject to adjustment, and may be exercised on a cashless basis. Each December Pre-Funded Warrant is exercisable
until exercised in full at an exercise price of $0.001 per share and may be exercised on a cashless basis. In addition, pursuant to the terms of the offering,
the  Company  issued  H.C.  Wainwright  &  Co.,  LLC  the  December  Wainwright  Warrants  to  purchase  up  to  100,000  shares  of  the  Company’s  common
stock. The December Wainwright Warrants are exercisable for a period of five and one-half years from the issuance date at an exercise price of $6.25
per share, subject to adjustment, and may be exercised on a cashless basis.

On January 11, 2023, the compensation committee of the board of directors increased the number of shares reserved for issuance under the 2018 Plan
from 156,878 shares to  166,878 shares.

F-21

 
 
 
 
 
 
 
 
   
   
   
   
   
   
   
   
   
   
   
   
 
 
 
 
 
 
 
 
 
   
 
 
 
 
 
 
ITEM 9. CHANGES IN AND DISAGREEMENTS WITH ACCOUNTANTS AND FINANCIAL DISCLOSURE

None.

ITEM 9A. CONTROLS AND PROCEDURES

Evaluation of Disclosure Controls

Our principal executive officer and principal financial officer, after evaluating the effectiveness of the Company’s “disclosure controls and procedures” (as
defined in Exchange Act Rule 13a-15(e) and 15d-15(e)) as of December 31, 2022, the end of the period covered by this Annual Report on Form 10-K,
have concluded that our disclosure controls and procedures were effective such that the information required to be disclosed by us in reports filed under
the  Exchange  Act  is  (i)  recorded,  processed,  summarized  and  reported  within  the  time  periods  specified  in  the  SEC’s  rules  and  forms  and  (ii)
accumulated and communicated to our management, including our principal executive officer and principal financial officer, as appropriate to allow timely
decisions  regarding  disclosure.  In  designing  and  evaluating  the  disclosure  controls  and  procedures,  management  recognizes  that  any  controls  and
procedures, no matter how well designed and operated, cannot provide absolute assurance that the objectives of the controls system are met, and no
evaluation of controls can provide absolute assurance that all control issues and instances of fraud, if any, within a company have been detected.

Management’s Report on Internal Control Over Financial Reporting

Our management is responsible for establishing and maintaining adequate internal control over financial reporting as such term is defined in Exchange
Act Rule 13a-15(f). Internal control over financial reporting is a process designed under the supervision and with the participation of our management,
including our principal executive officer and principal financial officer, to provide reasonable assurance regarding the reliability of financial reporting and
the  preparation  of  consolidated  financial  statements  for  external  purposes  in  accordance  with  GAAP.  All  internal  control  systems,  no  matter  how  well
designed,  have  inherent  limitations.  Therefore,  even  those  systems  determined  to  be  effective  can  provide  only  reasonable  assurance  with  respect  to
financial statement preparation and presentation.

As  of  December  31,  2022,  under  the  supervision  and  with  the  participation  of  our  management,  including  our  principal  executive  officer  and  principal
financial officer, we conducted an evaluation of the effectiveness of our internal control over financial reporting based on the Committee of Sponsoring
Organizations  of  the  Treadway  Commission  in  Internal  Control-Integrated  Framework  -  2013.  Based  on  this  assessment,  our  management  concluded
that,  as  of  December  31,  2022,  our  internal  control  over  financial  reporting  was  not  effective  because  it  identified  a  material  weakness.  A  material
weakness is a significant deficiency or a combination of significant deficiencies in internal control over financial reporting such that there is a reasonable
possibility that a material misstatement of the annual or interim financial statements will not be prevented or detected on a timely basis.

Specifically,  our  management  concluded  that  we  lacked  sufficient  resources  necessary  to  provide  adequate  segregation  of  duties  related  to  the
preparation and review of our financial information used in financial reporting and review of controls over the financial reporting process, including cutoff
related to accruals and prepaids.

We expect to be materially dependent upon third parties to provide us with accounting consulting services for the foreseeable future which we believe
mitigates the impact of the material weaknesses discussed above. In light of the material weakness, we performed additional analysis and other post-
closing procedures to ensure the reliability of financial reporting and that our financial statements were prepared in accordance with GAAP. Accordingly,
we  believe  that  the  financial  statements  included  in  this  report  fairly  present,  in  all  material  respects,  our  financial  condition,  results  of  operations  and
cash flows for the periods presented.

Our management, including our principal executive officer and principal financial officer, does not expect that our disclosure controls and procedures or
our internal controls will prevent all error and all fraud. A control system, no matter how well conceived and operated, can provide only reasonable, not
absolute, assurance that the objectives of the control system are met. Further, the design of a control system must reflect the fact that there are resource
constraints, and the benefits of controls must be considered relative to their costs. Due to the inherent limitations in all control systems, no evaluation of
controls can provide absolute assurance that all control issues and instances of fraud, if any, within our company have been detected.

Remediation Plans

In order to address the material weakness related to accruals and prepaids, we have implemented a new closing process for each quarter and year end
to properly account for and book expenses as required.

Attestation Report of our Registered Public Accounting Firm

This Annual Report on Form 10-K does not include an attestation report of our registered public accounting firm regarding internal control over financial
reporting. Management’s report was not subject to attestation by the Company’s independent registered public accounting firm pursuant to the exemption
provided to issuers that are not “large accelerated filers” nor “accelerated filers” under the Dodd-Frank Wall Street Reform and Consumer Protection Act.

Changes in Internal Control Over Financial Reporting

There have been no changes in our internal control over financial reporting that occurred during our last fiscal quarter that have materially affected, or are
reasonably likely to materially affect, our internal control over financial reporting.

44

ITEM 9B. OTHER INFORMATION

Robb Knie Employment Agreement

On March 28, 2023, we entered into an employment agreement (the “2023 Knie Employment Agreement”) with Robb Knie, pursuant to which Mr. Knie
continues to serve as our Chief Executive Officer. The term of the 2023 Knie Employment Agreement will continue for a period of three years from the
date of execution and automatically renews for successive one year periods at the end of each term until either party delivers written notice of their intent
not  to  review  at  least  six  months  prior  to  the  expiration  of  the  then  effective  term.  Mr.  Knie’s  base  salary  is  $450,000  per  year.  Mr.  Knie  is  eligible  to
receive an annual bonus of up to $350,000 per year at the discretion of the compensation committee of the Company, based upon the achievement of
Company and individual performance targets established by the compensation committee. Under the 2023 Knie Employment Agreement, Mr. Knie is also
entitled to receive equity-based compensation awards. In addition, the 2023 Knie Employment Agreement contains standard non-competition and non-

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
solicitation provisions. Mr. Knie is also eligible to receive additional equity-based compensation awards as the Company may grant from time to time. The
2023 Knie Employment Agreement further provides for standard expense reimbursement, vacation time and other standard executive benefits.

Pursuant  to  the  2023  Knie  Employment  Agreement,  in  the  event  Mr.  Knie’s  employment  is  terminated  without  Cause  (as  defined  in  the  2023  Knie
Employment Agreement), due to a non-renewal by the Company, he voluntarily resigns, or if he resigns for Good Reason (as defined in the 2023 Knie
Employment Agreement), Mr. Knie is entitled to (i) a cash payment equal to the sum of (x) 24 months of his base salary at the then current rate (or 36
months if such termination occurs within 12 months of a Change in Control (as defined in the 2023 Knie Employment Agreement)) and (y) annual bonus
in effect on his last day of employment; (ii) continuation of health benefits for a period of 24 months (or 36 months if such termination occurs within 12
months of a Change in Control); (iii) a lump sum payment equal to the amount of any annual bonus earned with respect to a prior fiscal year, but unpaid
as of the date of termination; (iv) a lump sum payment equal to the amount of annual bonus that was accrued through the date of termination for the year
in which employment ends; and (v) subject to Mr. Knie’s compliance with his restrictive covenants, the outstanding and unvested portion of any equity
award will accelerate and immediately vest on the date of Mr. Knie’s termination.

In the event that Mr. Knie’s employment is terminated due to his death or disability, he will be entitled to receive (i) a lump sum payment equal to the
amount of any annual bonus earned with respect to a prior fiscal year, but unpaid as of the date of termination; (ii) a lump sum payment equal to the
amount of annual bonus that was accrued for the year in which employment ends; and (iii) the treatment of any equity awards in accordance with their
respective equity award agreements.

In the event that Mr. Knie’s employment is terminated due to his non-renewal or resignation without Good Reason, he will be entitled to receive a lump
sum payment equal to the amount of any annual bonus earned with respect to a prior fiscal year, but unpaid as of the date of termination.

The foregoing description of the material terms of the  2023 Knie Employment Agreement  does not purport to be complete and is qualified in its entirety by
reference to the full text of the 2023 Knie Employment Agreement , a copy of which is filed as Exhibit 10.36 to this Annual Report on Form 10-K and is
incorporated herein by reference.

ITEM 9C. DISCLOSURE REGARDING FOREIGN JURISDICTIONS THAT PREVENT INSPECTIONS.

Not applicable.

45

PART III

ITEM 10. DIRECTORS, EXECUTIVE OFFICERS AND CORPORATE GOVERNANCE

The following table sets forth the name, age and positions of our executive officers and directors as of March 17, 2023.

NAME
Robb Knie
David Briones
Wayne Linsley 
David B. Sarnoff
Graig Springer
Jeff Pavell

AGE   POSITION

54
46
66
55
43
56

  President, Chief Executive Officer and Director
  Chief Financial Officer
  Director
  Director
  Director
  Director

The business background and certain other information about our directors and executive officers is set forth below.

Robb Knie

Robb Knie has served as President and Chief Executive Officer and as a director of the Company since May 2017 and served as our principal financial
and accounting officer from June 2018 until March 2019. Since October 2020, Mr. Knie has served as the Chief Executive Officer, Chief Financial Officer
and  chairman  of  the  board  of  directors  of  FoxWayne  Enterprises  Acquisition  Corp.  (“FoxWayne”),  a  special  purpose  acquisition  corporation.  Mr.  Knie
served  as  the  President  of  Lifeline  Industries  Inc.  since  its  inception  in  1995.  From  2002  to  2010  he  was  a  Semiconductor  Analyst  for  PAW  Partners.
From 1993 until 1995, Mr. Knie served as Northeast Regional Manager of American Express Financial Advisors. Mr. Knie has served as a board member
for Nasdaq-listed companies. He has been featured on Bloomberg, The Wall Street Journal and Forbes Magazine as an Independent Equity Analyst. Mr.
Knie  has  over  20  years  of  equity  markets  experience.  Mr.  Knie  has  been  a  member  of  the  American  Chemical  Society,  Institute  of  Electrical  and
Electronics  Engineers,  as  well  as  The  National  Alliance  for  Youth  Sports.  We  believe  that  Mr.  Knie  is  qualified  to  serve  as  a  director  because  of  his
business and leadership experience and experience as a board member of public companies in the healthcare industry.

David Briones

David Briones has served as Chief Financial Officer of the Company since March 2019 and has over 24 years of public accounting and executive level
experience.  He  consults  with  various  public  companies  in  financial  reporting,  internal  control  development  and  evaluation,  budgeting  and  forecasting.
Since September 2021, Mr. Briones has served as Chief Financial Officer, Treasurer and Secretary and a member of the board of directors of Larkspur
Healthcare Acquisition Corp. (Nasdaq: LSPR), a special purpose acquisition corporation. Since October 2010, he has served as the managing member
and founder of Brio Financial Group, LLC, a full-service financial consulting firm that brings experienced finance and accounting expertise to both public
and  private  companies.  Since  2010,  Mr.  Briones  has  served  over  75  companies  as  well  as  numerous  banks,  hedge  funds,  venture  capital  funds  and
private equity firms. In addition, from May 2018 until its dissolution in April 2021, Mr. Briones served as Executive Chair of Zovis Pharmaceuticals, and
from August 2013 to January 2020, Mr. Briones served as Chief Financial Officer of Petro River Oil Corp. (“PTRC”), an independent energy company
focused  on  the  exploration  and  development  of  conventional  oil  and  gas  assets.  Mr.  Briones  also  served  as  interim  Chief  Financial  Officer  of  AdiTx
Therapeutics,  Inc.  (Nasdaq:  ADTX),  a  pre-clinical  stage,  life  sciences  company  with  a  mission  to  prolong  life  and  enhance  life  quality  of  transplanted
patients from January 2018 to July 2020 (until the company’s initial public offering). From October 2017 to May 2018, Mr. Briones served as the Chief
Financial  Officer  of  Bitzumi,  Inc.,  a  Bitcoin  exchange  and  marketplace.  Prior  to  founding  Brio  Financial  Group,  LLC,  Mr.  Briones  was  an  auditor  with
Bartolomei Pucciarelli, LLC in Lawrenceville, New Jersey and PricewaterhouseCoopers LLP in New York, New York. Since May 2020, Mr. Briones has
served  as  a  member  of  the  board  of  directors  of  Unique  Logistics  International  Inc  (OTC  Pink:  UNQL).  Mr.  Briones  received  a  bachelors  of  science
degree in accounting from Fairfield University.

Wayne Linsley

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
  
Wayne  D.  Linsley  has  served  as  a  director  of  the  Company  since  April  2020.  Mr.  Linsley  has  been  in  business  management  for  over  40  years.  He
possesses a wide and varied skillset including sales and sales management, finance (for both public and private companies), accounting, audit support
and financial reporting. He has a bachelor’s in business administration from Siena College in Loudonville, NY. From 2009 to September 2021 he worked
for a financial reporting firm that works with publicly traded companies. He has extensive knowledge of financial statements, MD&A, SEC Filings (10-K,
10-Q,  8-K,  etc.)  Edgar,  etc.  He  often  negotiated  on  behalf  of  clients  in  such  areas  as  audit  fees,  transfer  agents,  Edgar  companies,  etc.  He  currently
serves as an independent director for DatChat Inc. (Nasdaq: DATS), serving the chair of its audit committee, compensation committee and nominating
and  corporate  governance  committee,  and  Silo  Pharma,  Inc.  (OTCQB:  SILO).  We  believe  Mr.  Linsley  is  qualified  to  serve  as  a  member  of  the  board
because his business management experience.

46

David B. Sarnoff

David  Sarnoff  has  served  as  a  director  of  the  Company  since  August  2018.  Since  May  2015,  Mr.  Sarnoff  has  served  as  the  founder  and  Principal  of
Sarnoff  Group,  LLC,  and  since  January  2019,  he  has  served  as  the  Director  of  Strategic  Partnerships  and  Executive  Leadership  Coach  at  Loeb
Leadership. In addition, since December 2021, Mr. Sarnoff has served as Adjunct Faculty at iCoach Global (formally known as iCoach New York) with
respect  to  a  professional  coaching  program  affiliated  with  the  Zicklin  School  of  Business  at  Baruch  College.  From  October  2003  until  May  2015,  Mr.
Sarnoff  served  as  the  co-founder  and  Principal  of  Morandi,  Taub  &  Sarnoff  LLC,  an  executive  search  firm,  and  from  July  1998  until  October  2003  he
served as a Legal Recruiter for Schneider Legal Search, Inc. From August 1994 until July 1998, Mr. Sarnoff served as a litigation associate attorney at
Wachtel Missry LLP (formerly known as Gold & Wachtel LLP). Since July 2018, Mr. Sarnoff has served as a member of the advisory committee of the
New Jersey Association of School Resource Officers. From January 2015 until January 2018, Mr. Sarnoff served as board President of Fort Lee Board of
Education and served as a board member from January 2013 through January 2019. In September of 2020, Mr. Sarnoff was appointed to a three year
term on the Diversity, Equity & Inclusion Committee of the New York City Bar Association, and in September 2022, he was appointed as Co-Chair of that
committee. Mr. Sarnoff received his Juris Doctor from Rutgers University School of Law and his bachelor of arts from Hofstra University. Mr. Sarnoff is
admitted to the New York and New Jersey (retired status) state bars. We believe that Mr. Sarnoff is qualified to serve as a director because of his legal
experience as well as his extensive experience in executive leadership and business development.

Graig Springer

Graig Springer has served as a director of the Company since February 2020. Since April 2021, Mr. Springer has served as Vice President for Brookfield
Oaktree Wealth Solutions LLC (“Brookfield”) in their Legal and Regulatory Department, and from August 2020 to April 2021, he served as a consultant to
Brookfield  Public  Securities  Group  LLC.  From  May  2019  to  August  2019,  Mr.  Springer  assisted  with  product  development  and  governance  at  Invesco
U.S.,  an  investment  management  company,  and  from  December  2013  to  May  2019,  he  served  in  various  capacities  at  OppenheimerFunds,  Inc.,  an
investment management company acquired by Invesco U.S., including distribution compliance and product development. In addition, Mr. Springer served
on the Sub-Adviser Oversight Committee at OppenheimerFunds, Inc. Mr. Springer received his bachelor of arts from Columbia University and his Juris
Doctor from Fordham University School of Law. Mr. Springer also holds a Series 7 and a Series 24 license. We believe that Mr. Springer is qualified to
serve as a director because of his fifteen years of experience within the financial services industry overseeing and advising firms’ compliance with federal
rules and regulations.

Jeff Pavell

Jeff  Pavell  has  served  as  a  director  of  the  Company  since  December  2022.  Since  January  2017,  Dr.  Pavell  has  served  as  Chief  of  Rehabilitation
Medicine  at  Englewood  Health,  and  since  November  2021,  he  has  been  on  the  teaching  staff  at  New  York-Presbyterian.  In  addition,  since  December
2020 he has been on the teaching staff at Hackensack Meridian School of Medicine at Seton Hall. Furthermore, since 2010, Dr. Pavell has served as a
partner at Patient Care Associates, an outpatient surgical center, and since 2002, he has served as a Partner at the Physical Medicine and Rehabilitation
Center, a private medical practice serving patients with spine, sports and occupational injuries. Dr. Pavell is a Board Certified physician specializing in the
field of physical medicine and rehabilitation. Dr. Pavell is also certified in pain medicine and specializes in the most advanced non-operative treatments
for  spine,  sports  and  interventional  pain  medicines.  Dr.  Pavell  received  his  bachelor  of  arts  from  Johns  Hopkins  University  and  his  D.O.  degree  with
honors from the New York College of Osteopathic Medicine. Since January 2021, Dr. Pavell has served as a member of the board of directors as well as
chairman of the audit committee and a member of the compensation committee of FoxWayne, a special purpose acquisition corporation. Furthermore,
since  September  2022,  Dr.  Pavell  has  served  as  a  director  of  Silo  Pharma,  Inc.  (Nasdaq:  SILO)  (“Silo”)  as  well  as  a  member  of  the  audit  committee,
compensation committee and chair of the nominating and corporate governance committee of Silo. We believe that Dr. Pavell is qualified to serve as a
director  due  to  his  extensive  experience  practicing  in  the  healthcare  industry  as  well  as  his  prior  experience  serving  as  a  director  for  other  public
companies.

Family Relationships

There are no family relationships among any of our executive officers or directors.

Arrangements between Officers and Directors

Except as set forth herein, to our knowledge, there is no arrangement or understanding between any of our officers or directors and any other person
pursuant to which the officer or director was selected to serve as an officer or director.

Involvement in Certain Legal Proceedings

We are not aware of any of our directors or officers being involved in any legal proceedings in the past ten years relating to any matters in bankruptcy,
insolvency,  criminal  proceedings  (other  than  traffic  and  other  minor  offenses),  or  being  subject  to  any  of  the  items  set  forth  under  Item  401(f)  of
Regulation S-K.

47

Committees of Our Board of Directors

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Our board of directors directs the management of our business and affairs, as provided by Nevada law, and conducts its business through meetings of
the  board  of  directors  and  its  standing  committees.  We  have  a  standing  audit  committee,  compensation  committee  and  nominating  and  corporate
governance  committee.  In  addition,  from  time  to  time,  special  committees  may  be  established  under  the  direction  of  the  board  of  directors  when
necessary to address specific issues.

Our board of directors has determined that all of the members of the audit committee, the compensation committee and the nominating and corporate
governance committee are independent as defined under the applicable rules of The Nasdaq Capital Market, including, in the case of all of the members
of our audit committee, the independence requirements contemplated by Rule 10A-3 under the Exchange Act. In making such determination, the board of
directors considered the relationships that each director has with our Company and all other facts and circumstances that the board of directors deemed
relevant in determining director independence, including the beneficial ownership of our capital stock by each director.

Audit Committee

Our audit committee is responsible for, among other things:

●

●

●

●

●

●

●

●

approving and retaining the independent registered public accounting firm to conduct the annual audit of our consolidated financial statements;

reviewing the proposed scope and results of the audit;

reviewing and pre-approval of audit and non-audit fees and services;

reviewing accounting and financial controls with the independent registered public accounting firm and our financial and accounting staff;

reviewing and approving transactions between us and our directors, officers and affiliates;

establishing procedures for complaints received by us regarding accounting matters;

overseeing internal audit functions, if any; and

preparing  the  report  of  the  audit  committee  that  the  rules  of  the  Securities  and  Exchange  Commission  require  to  be  included  in  our  annual
meeting proxy statement.

Our  audit  committee  consists  of  Wayne  Linsley,  David  Sarnoff  and  Graig  Springer,  with  Wayne  Linsley  serving  as  chair.  Each  member  of  our  audit
committee meets the financial literacy requirements of the Nasdaq rules. In addition, our board of directors has determined that Wayne Linsley qualifies
as an “audit committee financial expert,” as such term is defined in Item 407(d)(5) of Regulation S-K.

Our board of directors adopted a written charter for the audit committee which is available on our website at www.hoththerapeutics.com .

Compensation Committee

Our compensation committee is responsible for, among other things:

●

●

●

●

reviewing  and  recommending  the  compensation  arrangements  for  management,  including  the  compensation  for  our  president  and  chief
executive officer;

establishing and reviewing general compensation policies with the objective to attract and retain superior talent, to reward individual performance
and to achieve our financial goals;

administering our stock incentive plans; and

preparing  the  report  of  the  compensation  committee  that  the  rules  of  the  Securities  and  Exchange  Commission  require  to  be  included  in  our
annual meeting proxy statement.

On December 7, 2022, David Sarnoff resigned as a member of our compensation committee. Our audit committee currently consists of Wayne Linsley,
Graig Springer and Jeff Pavell, with Wayne Linsley serving as chair.

Our board of directors adopted a written charter for the compensation committee which is available on our website at www.hoththerapeutics.com.

48

Nominating and Governance Committee

Our nominating and governance committee is responsible for, among other things:

●

●

●

identifying and nominating members of the board of directors;

developing and recommending to the board of directors a set of corporate governance principles applicable to our Company; and

overseeing the evaluation of our board of directors.

Our nominating and corporate governance committee consists of Wayne Linsley, Graig Springer and David Sarnoff, with Graig Springer serving as chair.

Our  board  of  directors  adopted  a  written  charter  for  the  nominating  and  corporate  governance  committee  which  is  available  on  our  website  at
www.hoththerapeutics.com.

Scientific Advisory Board

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
  
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
In July 2017, the board of directors formed a Scientific Advisory Board (formerly known as the Technology Advisory Board). As of March 17, 2023, the
members  of  such  board  are  as  follows:  (i)  Dr.  Mario  Lacouture,  Dr.  William  Weglicki,  Dr.  Mark  Heaney  and  Dr.  Adam  Friedman  as  Medical  Doctor
members and (ii) Dr. Andrew Herr, Dr. Glenn Cruse, Dr. Vincent Njar, Dr. Carla Yuede, Dr. John Cirrito, Dr. Stefanie Johns and Sergio Traversa as Non-
Medical Doctor members.

Code of Business Code and Ethics Conduct

We adopted a written code of business conduct and ethics that applies to our directors, officers and employees, including our principal executive officer,
principal financial officer, principal accounting officer or controller, or persons performing similar functions. A copy of the code is posted on our website at
www.hoththerapeutics.com.  Disclosure  regarding  any  amendments  to,  or  waivers  from,  provisions  of  the  code  of  conduct  and  ethics  that  apply  to  our
the  “Investors-Corporate  Governance”  section  of  our  website  at
directors,  principal  executive  and  financial  officers  will  be  posted  on 
www.hoththerapeutics.com  or  will  be  included  in  a  Current  Report  on  Form  8-K,  which  we  will  file  within  four  business  days  following  the  date  of  the
amendment or waiver.

Changes in Nominating Procedures

None.

ITEM 11. EXECUTIVE COMPENSATION

Summary Compensation Table 

The  following  table  sets  forth  the  compensation  paid  or  accrued  during  the  fiscal  year  ended  December  31,  2022  and  2021  to  our  principal  executive
officer and an additional officer (collectively, the “named executive officers”):

● Robb Knie, Chief Executive Officer and President; and

● Stefanie Johns, former Chief Scientific Officer.

49

Salary
($)

Bonus
($)(1)

  Year    
  2022       450,000      300,000     

Stock
Awards
($)

Option
Awards
($)(2)
-      216,361     

Non-Equity
Incentive Plan
Compensation
($)

Nonqualified
deferred
compensation
earnings ($)

All Other
Compensation
($)(3)

Total
($)

Name and Principal
Position
Robb Knie
Chief Executive
Officer and
President
Stefanie Johns
Former Chief

  2021       400,000      200,000     
20,000     
  2022       382,443     

-      388,919     
-      108,181     

Scientific Officer

  2021       253,333     

10,000     

-      216,066     

-     

-     
-     

-     

-     

94,009      1,060,370 

-     
-     

-     

86,261      1,075,180 
695,886 

185,263     

46,894     

526,293 

(1) Represents payments of discretionary bonuses for performance during the applicable years as determined by the board, and as further described

below Bonus Arrangements.

(2) Represents the  aggregate  grant  date  fair  value  of  options  granted  for  the  fiscal  year  ended  December 31,  2022  and  December  31,  2021  as
determined in accordance with FASB ASC Topic 718, rather  than the amount paid to or realized by Robb Knie and Stefanie Johns. See Note 7,
“Stockholders’ Equity” in the notes to the Company’s consolidated financial statements for the fiscal year ended December 31, 2022 and December
31,  2021  included  in  this  Annual  Report on  Form  10-K  for  more  information  regarding  the  Company’s  accounting  for  share-based compensation
plans.

(3) All other compensation represents the employer matching contributions to each Robb Knie’s and Stefanie Johns’ 401(k) accounts and the amounts
received for their executive health or supplemental health insurance premiums. Mr. Knie received (i) an employer 401(k) contribution in the amount
$18,000  and  $15,917  for  fiscal  years  2022  and  2021,  respectively,  and  (ii)  payments  for  executive  health  or  supplemental  medical  insurance
premiums  in  the  amounts  of $76,009  and  $70,344  for  fiscal  years  2022  and  2021,  respectively.  Ms.  Johns  received  (A)  an  employer  401(k)
contribution in the amount $18,300 and $6,475 for fiscal years 2022 and 2021, respectively, and (B) payments for executive health or supplemental
medical insurance premiums in the amounts of $34,463 and $40,419 for fiscal years 2022 and 2021, respectively. For 2022, all other compensation
for Ms. Johns includes the following in connection with payments received under the Stefanie Johns Separation Agreement and General Release,
dated December 9, 2022, pursuant to which Ms. Johns was entitled to the following payments for the fiscal year ended on December 31, 2022:

Name
Stefanie Jones

Employment Agreements

Robb Knie Employment Agreement

  $

50

Separation
Payment

132,500    $

Total of All
Other
Compensation 
132,500 

On  February  20,  2019  (the  “Knie  Effective  Date”),  the  Company  entered  into  an  amended  and  restated  employment  agreement  with  Robb  Knie,  as
amended  on  June  25,  2021  (as  amended,  the  “Employment  Agreement”),  pursuant  to  which  Robb  Knie  serves  as  Chief  Executive  Officer  of  the

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
   
   
   
   
   
   
 
  
 
 
 
 
 
 
   
 
 
 
 
 
Company.  The  term  of  the  Employment  Agreement  will  continue  for  a  period  of  one  year  from  the  Knie  Effective  Date  and  automatically  renews  for
successive one year periods at the end of each term until either party delivers written notice of their intent not to review at least six months prior to the
expiration of the then effective term. Pursuant to the Employment Agreement, Mr. Knie (i) shall receive an annual base salary of $450,000 (effective as of
July 1, 2021) and (ii) shall be entitled to receive an annual bonus of $350,000 (effective as July 1, 2021), which annual bonus may be increased by the
compensation committee of the Company in its sole discretion, upon the achievement of additional criteria established by the compensation committee
from time to time. In addition, Mr. Knie is also entitled to participate in any and all Benefit Plans (as defined in the Employment Agreement), from time to
time, in effect for senior executives, along with vacation, sick and holiday pay in accordance with the Company’s policies established and in effect from
time to time.

The Employment Agreement may be terminated upon (i) Mr. Knie’s death, (ii) Mr. Knie’s Total Disability (as defined in the Employment Agreement), (iii)
expiration of the term if either party has provided a timely non-renewal notice, (iv) at Mr. Knie’s option (A) upon 90 days prior written notice; provided,
however, Mr. Knie may terminate the Employment Agreement by providing written notice at any time within 40 days of the consummation of a Change in
Control  Transaction  (as  defined  in  the  Employment  Agreement)  or  (B)  for  Good  Reason  (as  defined  in  the  Employment  Agreement);  or  (v)  at  the
Company’s option (A) for Cause (as defined in the Employment Agreement) or (B) upon 90 days prior written notice without Cause (as defined in the
Employment Agreement).

Upon the termination of Mr. Knie’s employment for any reason, whether by Mr. Knie or by the Company, Mr. Knie shall be paid (i) accrued but unpaid
compensation and vacation pay through the date of termination, (ii) any other benefits accrued to him under any Benefit Plans outstanding at the date of
termination and (iii) the reimbursement of expenses incurred on or prior to such date (collectively, the “Severance Package”). In addition to the Severance
Package, upon Mr. Knie’s termination for death or Total Disability, Mr. Knie or his estate or beneficiaries, as applicable, shall receive (i) 24 months base
salary  at  the  then  current  rate,  (ii)  if  Mr.  Knie  elects  continuation  coverage  for  group  health  coverage  pursuant  to  COBRA  Rights  (as  defined  in  the
Employment Agreement), then for a period of 24 months following Mr. Knie’s termination he will be obligated to pay only the portion of the full COBRA
Rights cost of the coverage equal to an active employee’s share of premiums (if any) for coverage for the respective plan year and (iii) payment on a pro-
rated basis of any annual bonus or other payments earned in connection with any bonus plan to which the Mr. Knie was a participant as of the date of
death or Total Disability. Upon Mr. Knie’s termination for Good Reason, without Cause or Mr. Knie’s termination upon 90 days prior written notice to the
Company or notice to the Company within 40 days of the consummation of a Change in Control Transaction, in addition to the Severance Package, Mr.
Knie shall receive (i) 24 months base salary at the then current rate, (ii) if Mr. Knie elects continuation coverage for group health coverage pursuant to
COBRA Rights, then for a period of 24 months following Mr. Knie’s termination he will be obligated to pay only the portion of the full COBRA Rights cost
of the coverage equal to an active employee’s share of premiums (if any) for coverage for the respective plan year, (iii) payment on a pro-rated basis of
any  annual  bonus  or  other  payments  earned  in  connection  with  any  bonus  plan  to  which  the  Mr.  Knie  was  a  participant  as  of  the  date  of  termination;
provided, however, that the pro-rated annual bonus payable pursuant to the Employment Agreement shall be no less than $200,000 and (iv) any equity
grants to Mr. Knie shall immediately vest upon termination of Mr. Knie’s employment by him for Good Reason or by the Company at its option upon 90
days  prior  written  notice  to  Mr.  Knie,  without  Cause.  The  Employment  Agreement  also  contains  covenants  prohibiting  Mr.  Knie  from  disclosing
confidential information with respect to the Company.

On March 28, 2023, the Company entered into the 2023 Knie Employment Agreement which is fully described in “Item 9B. Other Information.” The 2023
Knie  Employment  Agreement  generally  provides  for  the  same  material  terms  described  above,  except  the  material  changes  are  as  follows:  (i)  in  the
event  Mr.  Knie’s  employment  is  terminated  without  Cause,  due  to  a  non-renewal  by  the  Company,  he  voluntarily  resigns,  or  if  he  resigns  for  Good
Reason, Mr. Knie is entitled to (A) a cash payment equal to the sum of (x) 24 months of his base salary at the then current rate (or 36 months if such
termination  occurs  within  12  months  of  a  Change  in  Control)  and  (y)  annual  bonus  in  effect  on  his  last  day  of  employment;  (B)  continuation  of  health
benefits for a period of 24 months (or 36 months if such termination occurs within 12 months of a Change in Control); (C) a lump sum payment equal to
the amount of any annual bonus earned with respect to a prior fiscal year, but unpaid as of the date of termination; (D) a lump sum payment equal to the
amount  of  annual  bonus  that  was  accrued  through  the  date  of  termination  for  the  year  in  which  employment  ends;  and  (E)  subject  to  Mr.  Knie’s
compliance with his restrictive covenants, the outstanding and unvested portion of any equity award will accelerate and immediately vest on the date of
Mr. Knie’s termination; (ii) in the event that Mr. Knie’s employment is terminated due to his death or disability, he will be entitled to receive (A) a lump sum
payment equal to the amount of any annual bonus earned with respect to a prior fiscal year, but unpaid as of the date of termination; (B) a lump sum
payment equal to the amount of annual bonus that was accrued for the year in which employment ends; and (C) the treatment of any equity awards in
accordance  with  their  respective  equity  award  agreements;  and  (iii)  in  the  event  that  Mr.  Knie’s  employment  is  terminated  due  to  his  non-renewal  or
resignation without Good Reason he will be entitled to receive a lump sum payment equal to the amount of any annual bonus earned with respect to a
prior fiscal year, but unpaid as of the date of termination. See “Item 9B. Other Information” for additional details.

51

Stephanie Johns Employment Agreement

On  August  28,  2020,  the  Company  entered  into  an  employment  agreement  with  Dr.  Johns,  as  amended  on  January  29,  2021,  June  25,  2021  and
November 10, 2022 (as amended, the “Johns Employment Agreement”), pursuant to which Dr. Johns served as Chief Scientific Officer of the Company
effective  as  of  September  8,  2020  (the  “Effective  Date”).  Pursuant  to  the  third  amendment  to  the  Johns  Employment  Agreement  dated  November  10,
2022 (the “Third Amendment”), the term of the Johns Employment Agreement was to continue for a period of no more than six months from the date of
the Third Amendment; provided, however, the Company or Dr. Johns had the right to terminate Dr. Johns’ employment prior to the expiration of such six
month period for any reason upon 10 days prior notice. Pursuant to the terms of the Johns Employment Agreement, Dr. Johns was to receive an annual
base salary of $265,000 (effective as of July 1, 2021) and was eligible to participate in Benefit Plans (as defined in the Johns Employment Agreement)
from time to time, in effect for senior employees; however, pursuant to the Third Amendment,  Dr. Johns would no longer be eligible to receive any annual
bonus or equity awards. Furthermore, pursuant to the Third Amendment,  upon separation of Dr. Johns’ employment from the Company for any reason,
the Company would be required to provide Dr. Johns with all accrued but unpaid compensation earned through her final day of employment, all accrued
but  unused  vacation  and  reimbursement  of  all  documented,  unreimbursed  expenses  incurred  prior  to  her  separation.  Moreover,  upon  Dr.  Johns’
execution of a release of claims after her final day of employment, as set forth in the Third Amendment, the Company was required to provide Dr. Johns
with certain benefits as set forth therein.

On December 9, 2022 (the “Johns Separation Date”), the employment of Stefanie Johns as Chief Scientific Officer of the Company ceased. On the Johns
Separation Date, the Company entered into a Separation Agreement and General Release (the “Johns Separation Agreement”) with Dr. Johns pursuant
to  which  Dr.  Johns  shall  (i)  receive  six  months  of  base  salary,  subject  to  applicable  withholdings  and  deductions  and  (ii)  be  entitled  to  continue  any
benefits  (the  “Benefits”)  under  Company  sponsored  health  and  medical  plans  for  a  period  of  six  months  from  the  Johns  Separation  Date;  provided,
however, in the event that Dr. Johns obtains benefits that are equivalent to or greater than the Benefits provided by the Company through an alternative
source  prior  to  the  end  of  such  six  month  period,  the  Company’s  obligation  to  provide  the  Benefits  shall  cease.  Furthermore,  pursuant  to  the  Johns
Separation Agreement, Dr. Johns agreed to release and discharge the Released Parties (as defined in the Johns Separation Agreement) from any and
all  charges,  complaints,  claims,  liabilities,  obligations,  promises,  agreements,  damages,  actions,  causes  of  action,  whether  accrued  or  to  be  accrued,
suits, rights, demands, costs, losses, debts and expenses of any nature whatsoever, whether in law or in equity, whether known or unknown and under

 
 
 
 
 
 
 
 
any legal theory whatsoever, against the Released Parties through the Johns Separation Date.

52

Equity Grant Practices

2018 Equity Incentive Plan

On May 4, 2018, the Company’s board of directors adopted the Hoth Therapeutics, Inc. 2018 Omnibus Equity Incentive Plan (the “2018 Plan”). The 2018
Plan  became  effective  on  May  4,  2018  upon  approval  of  the  2018  Plan  by  the  Company’s  shareholders  at  the  Company’s  annual  meeting  of
shareholders. Pursuant to the 2018 Plan, the Company can grant stock options, stock appreciation rights, restricted stock, restricted stock units, deferred
stock  units,  annual  or  long-term  performance  awards  or  other  stock-based  awards.  As  of  December  31,  2022,  the  outstanding  option  awards  total
104,651, as described in the table “Option Awards” below.

2022 Equity Incentive Plan

On March 24, 2022, the Company’s board of directors adopted the Hoth Therapeutics, Inc. 2022 Omnibus Equity Incentive Plan (the “2022 Plan”) initially
reserving 96,000 shares of the Company’s common stock for issuance thereunder. The 2022 Plan became effective on June 23, 2022 upon approval of
the 2022 Plan by the Company’s shareholders at the Company’s annual meeting of shareholders. Pursuant to the 2022, the Company can grant stock
options, stock appreciation rights, restricted stock, restricted stock units, deferred stock units, annual or long-term performance awards or other stock-
based awards.

Bonus Arrangements

Pursuant to the terms of the executive employment agreements described above, the Company, through the board, has the discretion to determine the
amounts of the annual incentive bonus payments which executives may receive Based on the review of the Company’s performance for calendar year
2022, the board, in its sole discretion, determined to pay the bonuses to the named executive officers listed in the summary compensation table above.

401(k) Plan

The Company maintains a defined contribution employee retirement plan, or 401(k) plan, for its employees. The 401(k) plan is intended to qualify as a
tax-qualified plan under Section 401(k) of the Code so that contributions to the 401(k) plan, and income earned on such contributions, are not taxable to
participants until withdrawn or distributed from the 401(k) plan. The Company will match a participant's contribution 100% up to 6% of their compensation,
subject to statutory limits.

Perquisites

Perquisites are not a material component of compensation. In general, named executive officers do not receive reimbursements for meals, airlines, and
travel costs, other than those costs allowed for all employees. During 2022, no named executive officers received an allowance from the Company or any
of the above or a reimbursement for any expense incurred for non-business purposes.

53

Outstanding Equity Awards at December 31, 2022

The following table provides information regarding option awards held by each of our named executive officers that were outstanding as of December 31,
2022. There were no stock awards or other equity awards outstanding as of December 31, 2022.

Name
Robb Knie

Stefanie Johns

Number of
Securities 
Underlying
Unexercised
Options (#)
Exercisable  

Option Awards

Number of
Securities
Underlying
Unexercised
Options (#)
Unexercisable   

Option
Exercise
Price ($)

Option
Expiration
Date

10,000(1)
3,201(2)
9,000(3)
20,000(4)

5,000(5)(7)     
10,000(6)(7)     

-    $
-    $
-    $
-    $
-    $
       -    $

131.50    12/24/2029  
7/21/2030  
1/29/2031  
3/16/2032  
1/29/2031  
3/16/2032  

76.25   
52.75   
14.75   
52.75   
14.75   

(1) Stock options granted to Robb Knie vested in full immediately upon grant.

(2) Stock options granted to Robb Knie vested in full immediately upon grant.

(3) Stock options granted to Robb Knie vested in full immediately upon grant.

(4) Stock options granted to Robb Knie vested in full immediately upon grant.

(5) Stock options granted to Stefanie Johns vested in full immediately upon grant.

(6) Stock options granted to Stefanie Johns vested in full immediately upon grant.

(7) On December 9, 2022, the employment of Stefanie Johns as Chief Scientific Officer of the Company ceased. As a result, on March 9, 2023, the

options which were vested but unexercised expired pursuant to the terms of the option agreements.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
   
 
   
     
 
   
     
 
   
     
 
   
     
   
 
   
 
 
 
 
 
 
 
Non-Employee Director Compensation

The  following  table  presents  the  total  compensation  for  each  person  who  served  as  a  non-employee  member  of  our  board  of  directors  and  received
compensation for such service during the fiscal year ended December 31, 2022. Other than as set forth in the table and described more fully below, we
did not pay any compensation, make any equity awards or non-equity awards to, or pay any other compensation to any of the non-employee members of
our board of directors in 2022.

Fees earned
or paid in
cash ($)

Stock
Awards ($)

Option
Awards
($)(3)(4)

Non-Equity
Incentive Plan
Compensation
($)

Nonqualified
deferred
compensation
earnings
($)

All Other
Compensation
($)

Total
($)

2,582     
42,033     
48,033     
42,033     
3,397     

-     
-     
-     
-     
           -     

21,636     
17,309     
17,309     
17,309     
-     

-     
-     
-     
-     
            -     

-     
-     
-     
-     
      -     

-     
-     
-     
-     
        -     

24,218 
59,342 
65,342 
59,342 
3,397 

Name
Vadim Mats (1)
David Sarnoff
Graig Springer
Wayne Linsley
Jeff Pavell (2)

(1) Vadim Mats resigned from the Company’s board of directors effective as of January 31, 2022.

(2)

Jeff Pavell was appointed as a member of the Company’s board of directors on December 7, 2022.

(3) Amounts reported represent the aggregate grant date fair value for option awards granted in each respective year in accordance with FASB ASC
Topic 718, excluding the effect of forfeitures. See Note 7, “Stockholders’ Equity ” in the notes to the Company’s consolidated financial statements
for the fiscal year ended 2022 included in this Annual Report on Form 10-K for the year ended 2022 for more information regarding the Company’s
accounting for share-based compensation plans.

(4) On  March  16,  2022,  Vadim  Mats  was  granted  ten-year options  to  purchase  up  to  2,000  shares  of  the  Company’s  common  stock  at  an  exercise

price of $14.75, which options vested in full upon grant.

On March 16, 2022, David Sarnoff was granted ten-year options to purchase up to 1,600 shares of the Company’s common stock at an exercise
price of $14.75, which options vested in full upon grant.

On March 16, 2022, Graig Springer was granted ten-year options to purchase up to 1,600 shares of the Company’s at an exercise price of $14.75,
which options vested in full upon grant.

On March 16, 2022, Wayne Linsley was granted ten-year options to purchase up to 1,600 shares of the Company’s common stock, at an exercise
price of $14.75, which options vested in full upon grant.

54

Non-Employee Director Compensation Policy

Our  directors  receive  $50,000  cash  compensation  per  year  for  their  service  on  the  board  of  directors,  as  well  as  reimbursement  for  out-of-pocket
expenses with respect to such directors’ attendance at meetings of the board of directors of the Company.

Committee chairs receive an additional one-time $6,000 cash compensation upon appointment for their added services in such roles.

ITEM 12. SECURITY OWNERSHIP OF CERTAIN BENEFICIAL OWNERS AND MANAGEMENT AND RELATED STOCKHOLDER MATTERS

The following table sets forth certain information regarding beneficial ownership of shares of our common stock as of March 17, 2023 by (i) each person
known to beneficially own more than 5% of our outstanding common stock, (ii) each of our directors, (iii) each of our named executive officers and (iv) all
of  our  directors  and  named  executive  officers  as  a  group.  Except  as  otherwise  indicated,  the  persons  named  in  the  table  below  have  sole  voting  and
investment power with respect to all shares beneficially owned, subject to community property laws, where applicable.

Beneficial Owner(1)
Directors and Named Executive Officers:
Robb Knie
Wayne Linsley
David Sarnoff
Graig Springer
Jeff Pavell
All Named Executive Officers and Directors as a Group (5 persons)
5% or Greater Shareholders:
Armistice Capital, LLC (8)

510 Madison Avenue, 7th Floor
New York, New York 10022

*

Represents beneficial ownership of less than 1%.

Shares of 
Common
Stock 
Beneficially
Owned

75,331(3)
3,654(4)
5,920(5)
24,567(6)
1,691(7)

111,163 

  Percentage(2)

2.25%
* 
* 
* 
* 
3.29%

144,518(9)

9.99%

(1)

The address of each person is c/o Hoth Therapeutics, Inc., 1 Rockefeller Plaza, Suite 1039, New York, New York 10020 unless otherwise indicated
herein.

 
 
 
 
   
   
   
   
   
   
 
   
   
   
   
   
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
  
 
  
   
   
   
   
   
   
   
   
   
   
   
   
   
  
   
  
   
   
 
 
(2)

The  calculation  in  this  column  is  based  upon  3,302,113  shares  of  common  stock  outstanding  on  March  17,  2023.  Beneficial  ownership  is
determined  in  accordance  with  the  rules  of  the  SEC  and  generally  includes  voting  or  investment  power  with  respect  to  the  subject  securities.
Shares of common stock that are currently exercisable or convertible within 60 days of March 17, 2023 are deemed to be beneficially owned by the
person holding such securities for the purpose of computing the percentage beneficial ownership of such person, but are not treated as outstanding
for the purpose of computing the percentage beneficial ownership of any other person.

(3)

Includes options to purchase up to 42,200 shares of the Company’s common stock.

(4)

Includes options to purchase up to 3,520 shares of the Company’s common stock.

(5)

Includes options to purchase up to 4,920 shares of the Company’s common stock.

55

(6)

Includes  (i)  134  shares  of  the  Company’s  common  stock  held  by  Graig  Springer,  (ii)  options  to  purchase  up  to  3,520  shares  of  the  Company’s
common  stock  held  by  Graig  Springer,  (iii)  1,113  shares  of  the  Company’s  common  stock  held  by  Mr.  Springer’s  spouse  and  (iv)  options  to
purchase  up  to  19,800  shares  of  the  Company’s  common  stock  held  by  Mr.  Springer’s  spouse.  Mr.  Springer’s  spouse  is  an  employee  of  the
Company.

(7)

Excludes 3,384 shares of the Company’s common stock that are subject to vesting.

(8) As set forth in the Schedule 13G filed by Armistice Capital, LLC with the SEC on February 14, 2023 (the “Armistice SC 13G”), Armistice Capital,
LLC (“Armistice Capital”) is the investment manager of Armistice Capital Master Fund Ltd. (the “Master Fund”), the direct holder of the securities,
and  pursuant  to  an  Investment  Management  Agreement,  Armistice  Capital  exercises  voting  and  investment  power  over  the  securities  of  the
Company held by the Master Fund and thus may be deemed to beneficially own the securities of the Company held by the Master Fund. Mr. Boyd,
as the managing member of Armistice Capital, may be deemed to beneficially own the securities of the Company held by the Master Fund. The
Master Fund specifically disclaims beneficial ownership of the securities of the Company directly held by it by virtue of its inability to vote or dispose
of such securities as a result of its Investment Management Agreement with Armistice Capital.

(9)

Beneficial ownership has been determined pursuant to the Armistice SC 13G.

Securities Authorized for Issuance Under Equity Compensation Plans

The following table summarizes information about our equity compensation plans as of December 31, 2022.

Number of
securities to
be issued
upon
exercise of
outstanding
options,
warrants and
rights (a)

Weighted
average
exercise price
of outstanding
options,
warrants and
rights

Number of
securities
remaining
available for
future
issuance
under equity
compensation
plans
(excluding
securities
reflected in
column (a))

120,434    $
-     
120,434     

49.80     
-     

132,444 
- 
132,444 

Plan Category
Equity compensation plans approved by security holders
Equity compensation plans not approved by security holders
Total

56

ITEM 13. CERTAIN RELATIONSHIPS AND RELATED TRANSACTIONS, AND DIRECTOR INDEPENDENCE

The following includes a summary of transactions during our fiscal years ended December 31, 2022 and December 31, 2021 to which we have been a
party, including transactions in which the amount involved in the transaction exceeds the lesser of $120,000 or 1% of the average of our total assets at
year-end for the last two completed fiscal years, and in which any of our directors, executive officers or, to our knowledge, beneficial owners of more than
5% of our capital stock or any member of the immediate family of any of the foregoing persons had or will have a direct or indirect material interest, other
than  equity  and  other  compensation,  termination,  change  in  control  and  other  arrangements,  which  are  described  elsewhere  in  this  Annual  Report  on
Form  10-K.  We  are  not  otherwise  a  party  to  a  current  related  party  transaction,  and  no  transaction  is  currently  proposed,  in  which  the  amount  of  the
transaction exceeds the lesser of $120,000 or 1% of the average of our total assets at year-end for the last two completed fiscal years and in which a
related person had or will have a direct or indirect material interest.

On December 29, 2022, we entered into a securities purchase agreement with  Armistice Capital Master Fund Ltd. (“ Armistice”) pursuant to which we
agreed to sell an aggregate of (i) 140,000 shares (the “Shares”) of common stock, (ii) pre-funded warrants to purchase up to 1,860,000 shares (the “Pre-
Funded Warrant Shares”) of common stock and (iii) warrants to purchase up to 2,500,000 shares (the “Warrant Shares” and together with the Shares and
the Pre-Funded Warrant Shares, the “Registrable Securities”) of common stock at a purchase price of $5.00 per share and accompanying warrant (less
$0.001  for  each  pre-funded  warrant  and  accompanying  warrant)  in  a  private  placement  for  aggregate  gross  proceeds  of  approximately  $10  million,
exclusive of placement agent commission and fees and other offering expenses. The closing of the offering occurred on January 3, 2023. Each common
stock warrant is exercisable for a period of five and one-half years from the issuance date at an exercise price of $5.00 per share, subject to adjustment,

 
 
 
 
 
 
 
 
 
 
  
 
 
 
   
   
 
   
   
   
      
 
 
 
 
 
and may, under certain circumstances, be exercised on a cashless basis. Each pre-funded warrant is exercisable until exercised in full at an exercise
price of $0.001 per share and may be exercised on a cashless basis. In connection with the offering, we also entered into a registration rights agreement
(the “Registration Rights Agreement”) with Armistice pursuant to which we filed a Registration Statement on Form S-3 covering the Registrable Securities
on January 13, 2023, which registration statement was declared effective by the SEC on January 25, 2023.

Related Person Transaction Policy

We have adopted a formal policy regarding approval of transactions with related parties. For purposes of our policy only, a related person transaction is a
transaction, arrangement or relationship, or any series of similar transactions, arrangements or relationships, in which we and any related person are,
were or will be participants in which the amount involved exceeds the lesser of $120,000 or 1% of our total assets at the end of our last completed fiscal
year. Transactions involving compensation for services provided to us as an employee or director are not covered by this policy. A related person is any
executive officer, director or beneficial owner of more than 5% of any class of our voting securities, including any of their immediate family members and
any entity owned or controlled by such persons.

Under the policy, if a transaction has been identified as a related person transaction, including any transaction that was not a related person transaction
when originally consummated or any transaction that was not initially identified as a related person transaction prior to consummation, our management
must  present  information  regarding  the  related  person  transaction  to  our  audit  committee,  or,  if  audit  committee  approval  would  be  inappropriate,  to
another independent body of our board of directors, for review, consideration and approval or ratification. The presentation must include a description of,
among  other  things,  the  material  facts,  the  interests,  direct  and  indirect,  of  the  related  persons,  the  benefits  to  us  of  the  transaction  and  whether  the
transaction  is  on  terms  that  are  comparable  to  the  terms  available  to  or  from,  as  the  case  may  be,  an  unrelated  third  party  or  to  or  from  employees
generally.  Under  the  policy,  we  will  collect  information  that  we  deem  reasonably  necessary  from  each  director,  executive  officer  and,  to  the  extent
feasible, significant shareholder to enable us to identify any existing or potential related-person transactions and to effectuate the terms of the policy. In
addition, under our code of business conduct and ethics, our employees and directors will have an affirmative responsibility to disclose any transaction or
relationship  that  reasonably  could  be  expected  to  give  rise  to  a  conflict  of  interest.  In  considering  related  person  transactions,  our  audit  committee,  or
other independent body of our board of directors, will take into account the relevant available facts and circumstances including, but not limited to:

●

●

●

●

the risks, costs and benefits to us;

the impact on a director’s independence in the event that the related person is a director, immediate family member of a director or an entity with
which a director is affiliated;

the availability of other sources for comparable services or products; and

the terms available to or from, as the case may be, unrelated third parties or to or from employees generally.

57

The policy requires that, in determining whether to approve, ratify or reject a related person transaction, our audit committee, or other independent body
of our board of directors, must consider, in light of known circumstances, whether the transaction is in, or is not inconsistent with, our best interests and
those  of  our  shareholders,  as  our  audit  committee,  or  other  independent  body  of  our  board  of  directors,  determines  in  the  good  faith  exercise  of  its
discretion.

Director Independence

Our board of directors determined that a majority of the board during the year ended December 31, 2022 consisted of members who were “independent”
as that term is defined under Nasdaq Listing Rule 5605(a)(2). The Board considered Wayne Linsley, David Sarnoff, Graig Springer and Jeff Pavell to be
“independent.”

ITEM 14. PRINCIPAL ACCOUNTANT FEES AND SERVICES

The following table sets forth the aggregate fees billed by WithumSmith+Brown, PC as described below:

Audit Fees
Audit Related Fees
Tax Fees
All Other Fees

Total

2022

2021

149,791    $
-     
6,650     
-     
156,441    $

98,365 
- 
3,605 
- 
101,970 

  $

  $

Audit Fees: Audit fees consist of fees billed for professional services performed by WithumSmith+Brown, PC for the audit of our annual consolidated
financial  statements,  the  review  of  interim  consolidated  financial  statements,  and  related  services  that  are  normally  provided  in  connection  with
registration  statements.  There  were  $149,791  and  $98,365  of  such  fees  incurred  by  the  Company  in  the  fiscal  years  ended  December  31,  2022  and
2021, respectively.

Audit-Related Fees: Audit related fees may consist of fees billed by an independent registered public accounting firm for assurance and related services
that are reasonably related to the performance of the audit or review of our consolidated financial statements. There were no such fees incurred by the
Company in the fiscal years ended December 31, 2022 and 2021.

Tax Fees: Tax fees may consist of fees for professional services, including tax compliance performed by WithumSmith+Brown, PC. There were $6,650
and $3,605 of such fees incurred by the Company in the fiscal years ended December 31, 2022 and 2021, respectively.

All Other Fees:  There were no such fees incurred by the Company in the fiscal years ended December 31, 2022 and 2021.

Pre-Approval Policies and Procedures

In accordance with Sarbanes-Oxley, our audit committee charter requires the audit committee to pre-approve all audit and permitted non-audit services
provided  by  our  independent  registered  public  accounting  firm,  including  the  review  and  approval  in  advance  of  our  independent  registered  public

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
  
 
 
 
 
 
 
   
 
   
   
   
 
 
 
 
 
 
accounting firm’s annual engagement letter and the proposed fees contained therein. The audit committee has the ability to delegate the authority to pre-
approve non-audit services to one or more designated members of the audit committee. If such authority is delegated, such delegated members of the
audit committee must report to the full audit committee at the next audit committee meeting all items pre-approved by such delegated members. In the
fiscal years ended December 31, 2022 and 2021 all of the services performed by our independent registered public accounting firm were pre-approved by
the audit committee.

58

PART IV

ITEM 15. EXHIBIT AND FINANCIAL STATEMENT SCHEDULES

(a) The following documents are filed as part of this report:

(1) Financial Statements:

Report of Independent Registered Public Accounting Firm (PCAOB ID: 100)
Consolidated Balance Sheets as of December 31, 2022 and 2021
Consolidated Statements of Operations and Comprehensive Loss for the years ended December 31, 2022 and 2021
Consolidated Statements of Changes in Stockholders’ Equity for the years ended December 31, 2022 and 2021
Consolidated Statements of Cash Flows for the years ended December 31, 2022 and 2021
Notes to Consolidated Financial Statements

The consolidated financial statements required by this Item are included beginning at page F-1.

(1) Financial Statement Schedules:

F-2
F-3
F-4
F-5
F-6
F-7

All  financial  statement  schedules  have  been  omitted  because  they  are  not  applicable,  not  required  or  the  information  required  is  shown  in  the
consolidated financial statements or the notes thereto.

59

EXHIBIT INDEX

Exhibit

  Articles of Incorporation (Incorporated by reference to Exhibit 3.1 to the Company’s Form S-1/A filed on December 14, 2018)

  Amendment  to  Articles  of  Incorporation  (Incorporated  by  reference  to  Exhibit  3.2  to  the  Company’s  Form  S-1/A  filed  on  December  14,

2018)

  Certificate of Designations, Preferences and Rights of the Series A Convertible Preferred Stock (Incorporated by reference to Exhibit 3.3

to the Company’s Form S-1/A filed on December 14, 2018)

  Amendment to Articles of Incorporation (Incorporated by reference to Exhibit 3.1 to the Company’s Form 8-K filed on February 20, 2019)

  Amended and Restated Bylaws (Incorporated by reference to Exhibit 3.2 to the Company’s Form 8-K filed on February 20, 2019)

  Amendment to the Amended and Restated Bylaws of Hoth Therapeutics, Inc. (Incorporated by reference to Exhibit 3.1 to the Company’s

Form 8-K filed on August 22, 2022)

  Certificate of Change dated October 20, 2022  (Incorporated by reference to Exhibit 3.1 to the Company’s Form 8-K filed on October 24,

2022)

  Certificate  of  Designation  dated  November  2,  2022  (Incorporated  by  reference  to  Exhibit  3.1  to  the  Company’s  Form  8-K  filed  on

November 3, 2022)

  Certificate of Amendment (Incorporated by reference to Exhibit 3.1 to the Company’s Form 8-K filed on December 13, 2022)

  Specimen Stock Certificate evidencing the shares of common stock (Incorporated by reference to Exhibit 4.1 to the Company’s Form S-

1/A filed on December 14, 2018)

  Form of Underwriter Warrant (Incorporated by reference to Exhibit 4.2 to the Company’s Form S-1/A filed on January 11, 2019)

  Form of Warrant (Incorporated by reference to Exhibit 4.1 to the Company’s Form 8-K filed on March 25, 2020)

  Form of Warrant (Incorporated by reference to Exhibit 4.1 to the Company’s Form 8-K filed on May 22, 2020)

(b) Exhibits

Exhibit
Number
3.1

3.2

3.3

3.4

3.5

3.6

3.7

3.8

3.9

4.1

4.2

4.3

4.4

4.5*

  Description of the Registrant’s Securities

10.1+

  Amended and Restated Employment Agreement between Hoth Therapeutics, Inc. and Robb Knie (Incorporated by reference to Exhibit

10.1 to the Company’s Form 8-K filed on February 20, 2019)

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
10.2

  Office Service Agreement with Regus dated June 26, 2017 (Incorporated by reference to Exhibit 10.7 to the Company’s Form S-1/A filed

on December 14, 2018)

10.3

  Form of Warrant (Incorporated by reference to Exhibit 10.8 to the Company’s Form S-1/A filed on December 14, 2018)

10.4+

  2018 Equity Incentive Plan (Incorporated by reference to Exhibit 10.1 to the Company’s Form S-8 filed on February 4, 2022)

10.5*

10.6

  Renewal Agreement with Regus dated July 22, 2022

  Form of Registration Rights Agreement (Incorporated by reference to Exhibit 10.14 to the Company’s Form S-1/A filed on December 14,

2018)

10.7+

  Employment Agreement between Hoth Therapeutics, Inc. and David Briones (Incorporated by reference to Exhibit 10.1 to the Company’s

Form 8-K filed on March 7, 2019)

60

10.8

10.9

10.10

10.11

  Form of Warrant (Incorporated by reference to Exhibit 10.3 to the Company’s Form 8-K filed on August 21, 2019)

  Form of Registration Rights Agreement (Incorporated by reference to Exhibit 10.4 to the Company’s Form 8-K filed on August 21, 2019)

  Form of Placement Agent Warrant (Incorporated by reference to Exhibit 10.5 to the Company’s Form 8-K filed on August 21, 2019)

  License  Agreement  with  North  Carolina  State  University  dated  November  20,  2019  (Incorporated  by  reference  to  Exhibit  10.22  to  the

Company’s Form 10-K filed on March 2, 2020)

10.12

  Development and Royalty Agreement by and between the Company and Voltron Therapeutics, Inc. dated March 23, 2020 (Incorporated

by reference to Exhibit 10.1 to the Company’s Form 8-K filed on March 23, 2020)

10.13#

  Exclusive License Agreement between the Company and Virginia Commonwealth University Intellectual Property Foundation dated May

18, 2020 (Incorporated by reference to Exhibit 10.1 to the Company’s Form 8-K filed on May 19, 2020)

10.14#

  Sublicense Agreement by and between the Company and Isoprene Pharmaceutics, Inc. dated July 30, 2020 (Incorporated by reference to

Exhibit 10.1 to the Company’s Form 8-K filed on August 5, 2020)

10.15

  License Agreement by and between the University of Cincinnati and Chelexa BioSciences, Inc. dated February 27, 2013 assigned to the

Company on May 14, 2020 (Incorporated by reference to Exhibit 10.3 to the Company’s Form 10-Q filed on August 13, 2020)

10.16

10.17

  First Amendment to Exclusive License Agreement by and between the University of Cincinnati and Chelexa BioSciences, Inc. dated April
17,  2013  assigned  to  the  Company  on  May  14,  2020  (Incorporated  by  reference  to  Exhibit  10.4  to  the  Company’s  Form  10-Q  filed  on
August 13, 2020)

  Second Amendment to Exclusive License Agreement by and between the University of Cincinnati and Chelexa BioSciences, Inc. dated
February 27, 2013 assigned to the Company on May 14, 2020 (Incorporated by reference to Exhibit 10.5 to the Company’s Form 10-Q
filed on August 13, 2020)

10.18

  Assignment and Assumption Agreement by and between the Company and Chelexa BioSciences, Inc. dated May 14, 2020 (Incorporated

by reference to Exhibit 10.6 to the Company’s Form 10-Q filed on August 13, 2020)

10.19

  Royalty  Agreement  by  and  between  the  Company  and  Chelexa  BioSciences,  Inc.  dated  May  14,  2020  (Incorporated  by  reference  to

Exhibit 10.7 to the Company’s Form 10-Q filed on August 13, 2020)

10.20

  Novation  Agreement  by  and  among  the  Company,  Chelexa  BioSciences,  Inc.  and  the  University  of  Cincinnati  dated  May  14,  2020

(Incorporated by reference to Exhibit 10.8 to the Company’s Form 10-Q filed on August 13, 2020)

10.21

  Patent License Agreement by and between the Company and the George Washington University dated August 7, 2020 (Incorporated by

reference to Exhibit 10.9 to the Company’s Form 10-Q filed on August 13, 2020)

10.22+

  Employment Agreement by and between the Company and Stefanie Johns dated August 28, 2020 (Incorporated by reference to Exhibit

10.1 to the Company’s Form 8-K filed on August 31, 2020)

10.23

10.24

10.25

  Form of Warrant (Incorporated by reference to Exhibit 10.2 to the Company’s Form 8-K filed on January 8, 2021)

  Form of Registration Rights Agreement (Incorporated by reference to Exhibit 10.3 to the Company’s Form 8-K filed on January 8, 2021)

  Form of Placement Agent Warrant (Incorporated by reference to Exhibit 10.4 to the Company’s Form 8-K filed on January 8, 2021)

61

10.26+

  First  Amendment  to  the  Employment  Agreement  between  Hoth  Therapeutics,  Inc.  and  Stefanie  Johns  (Incorporated  by  reference  to

Exhibit 10.1 to the Company’s Form 8-K filed on January 29, 2021)

10.27

  Form of Common Stock Warrants (Incorporated by reference to Exhibit 10.2 to the Company’s Form 8-K filed on March 9, 2021)

 
   
 
   
 
   
 
   
 
   
 
   
 
 
 
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
 
 
 
   
 
 
 
 
   
10.28

10.29

10.30

  Form of Pre-Funded Warrants (Incorporated by reference to Exhibit 10.3 to the Company’s Form 8-K filed on March 9, 2021)

  Form of Registration Rights Agreement (Incorporated by reference to Exhibit 10.4 to the Company’s Form 8-K filed on March 9, 2021)

  Form of Placement Agent Warrants (Incorporated by reference to Exhibit 10.5 to the Company’s Form 8-K filed on March 9, 2021)

10.31+

  First  Amendment  to  the  Amended  and  Restated  Employment  Agreement  between  the  Company  and  Robb  Knie  dated  June  25,  2021

(Incorporated by reference to Exhibit 10.1 to the Company’s Form 8-K filed on June 30, 2021)

10.32+

  Second  Amendment  to  the  Employment  Agreement  between  the  Company  and  Stefanie  Johns  dated  June  25,  2021  (Incorporated  by

reference to Exhibit 10.2 to the Company’s Form 8-K filed on June 30, 2021)

10.33+

  Hoth Therapeutics, Inc. 2022 Omnibus Equity Incentive Plan (Incorporated by reference to Appendix A to the Company’s Definitive Proxy

Statement on Schedule 14A filed with the SEC on April 27, 2022)

10.34+

  Third Amendment to Employment Agreement by and between the Company and Stefanie Johns dated November 10, 2022 (Incorporated

by reference to Exhibit 10.1 of the Company’s Form 10-Q filed on November 10, 2022)

10.35+

  Separation Agreement and General Release by and between the Company and Stefanie Johns dated December 9, 2022 (Incorporated by

reference to Exhibit 10.1 to the Company’s Form 8-K filed on December 13, 2022)

10.36*+

  Employment Agreement by and between the Company and Robb Knie dated as of March 28, 2023

21.1*

23.1*

24.1*

31.1*

  Subsidiaries of the registrant

  Consent of WithumSmith+Brown, PC 

  Power of Attorney (included on the signature page hereto)

  Certification of the Chief Executive Officer pursuant to Rule 13a-14(a) of the Exchange Act, as adopted pursuant to Section 302 of the

Sarbanes-Oxley Act of 2002

31.2*

  Certification  of  the  Chief  Financial  Officer  pursuant  to  Rule  13a-14(a)  of  the  Exchange  Act,  as  adopted  pursuant  to  Section  302  of  the

Sarbanes-Oxley Act of 2002

32.1*

  Certification  of  the  Chief  Executive  Officer  and  Chief  Financial  Officer  pursuant  to  Rule  13a-14(b)  of  the  Exchange  Act  and  18  U.S.C.

Section 1350, as adopted pursuant to Section 906 of the Sarbanes-Oxley Act of 2002

101.INS*

  Inline XBRL Instance Document

101.SCH*

  Inline XBRL Taxonomy Extension Schema Document

101.CAL*

  Inline XBRL Taxonomy Extension Calculation Linkbase Document

101.DEF*

  Inline XBRL Taxonomy Extension Definition Linkbase Document

101.LAB*

  Inline XBRL Taxonomy Extension Label Linkbase Document

101.PRE*

  Inline XBRL Taxonomy Extension Presentation Linkbase Document

104*

  Cover Page Interactive Data File - the cover page of the Registrant’s Annual Report on Form 10-K for the year ended December 31, 2022

is formatted in Inline XBRL

Filed herewith.
Indicates a management contract or any compensatory plan, contract or arrangement.

*
+
# Pursuant to Item 601(b)(10) of Regulation S-K, certain confidential portions of this exhibit were omitted by means of marking such portions with an

asterisk because it is both not material and is the type of information that the Company treats as private or confidential.

ITEM 16. FORM 10-K SUMMARY

Not applicable.

62

SIGNATURES

Pursuant to the requirements of Section 13 and 15(d) of the Securities Exchange Act of 1934, the registrant has duly caused this Annual Report

on Form 10-K to be signed on its behalf by the undersigned, thereunto duly authorized on this 31st day of March, 2023.

HOTH THERAPEUTICS, INC.

/s/ Robb Knie
Robb Knie
Chief Executive Officer
(Principal Executive Officer)

 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
   
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
/s/ David Briones

David Briones
Chief Financial Officer
(Principal Financial and Accounting Officer)

POWER OF ATTORNEY

KNOW ALL PERSONS BY THESE PRESENTS, that each person whose signature appears below hereby constitutes and appoints Robb Knie
as his or her attorney-in-fact, with full power of substitution and resubstitution, for him or her in any and all capacities, to sign any and all amendments to
this  Annual  Report  on  Form  10-K,  and  to  file  the  same,  with  exhibits  thereto  and  other  documents  in  connection  therewith,  with  the  Securities  and
Exchange  Commission,  granting  unto  said  attorney-in-fact  full  power  and  authority  to  do  and  perform  each  and  every  act  and  thing  requisite  and
necessary to be done in connection therewith as fully to all intents and purposes as he might or could do in person, hereby ratifying and confirming all that
said attorney-in-fact, or his substitute or substitutes, may lawfully do or cause to be done by virtue hereof.

Pursuant to the requirements of the Securities Act of 1934, this Annual Report on Form 10-K has been signed below by the following persons on

behalf of the registrant and in the capacities and on the dates indicated.

Signature

/s/ Robb Knie
Robb Knie

/s/ David Briones
David Briones

/s/ Wayne Linsley
Wayne Linsley

/s/ David B. Sarnoff
David B. Sarnoff

/s/ Graig Springer
Graig Springer

/s/ Jeff Pavell
Jeff Pavell

Title

  Chief Executive Officer, President and Director
  (Principal Executive Officer)

  Chief Financial Officer
  (Principal Financial and Accounting Officer)

  Director

  Director

  Director

  Director

63

Date 

March 31, 2023

March 31, 2023

March 31, 2023

March 31, 2023

March 31, 2023

March 31, 2023