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Ovid Therapeutics Inc.

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FY2020 Annual Report · Ovid Therapeutics Inc.
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UNITED STATES
SECURITIES AND EXCHANGE COMMISSION
Washington, D.C. 20549

FORM 10-K

(Mark One)

☒

ANNUAL REPORT PURSUANT TO SECTION 13 OR 15(d) OF THE SECURITIES EXCHANGE ACT OF 1934

☐

TRANSITION REPORT PURSUANT TO SECTION 13 OR 15(d) OF THE SECURITIES EXCHANGE ACT OF 1934

For the Fiscal Year Ended December 31, 2020

OR

For the Transition Period from                         to                        

Commission File Number: 001-38085

Ovid Therapeutics Inc.

(Exact name of Registrant as specified in its charter)

Delaware
(State or Other Jurisdiction of
Incorporation or Organization)

2834
(Primary Standard Industrial
Classification Code Number)

46-5270895
(I.R.S. Employer
Identification Number)

1460 Broadway, Suite 15021
New York, New York 10036
(646) 661-7661
(Address, Including Zip Code, and Telephone Number, Including Area Code, of Registrant’s Principal Executive Offices)
Securities registered pursuant to Section 12(b) of the Act:

Title of each class
Common Stock, par value $0.001 per share

Trading
Symbol(s)
OVID

Name of each exchange on which registered
The Nasdaq Stock Market LLC

Securities registered pursuant to Section 12(g) of the Act: None

Indicate by check mark if the registrant is a well-known seasoned issuer, as defined in Rule 405 of the Securities Act.    Yes ☐    No ☒

Indicate by check mark if the registrant is not required to file reports pursuant to Section 13 or 15(d) of the Securities Act.    Yes ☐    No ☒
Indicate by check mark whether the registrant (1) has filed all reports required to be filed by Section 13 or 15(d) of the Securities Exchange Act of 1934 during the preceding 12 months (or for

such shorter period that the registrant was required to file such reports), and (2) has been subject to the filing requirements for the past 90 days.    Yes ☒    No ☐

Indicate by check mark whether the registrant has submitted electronically every Interactive Data File required to be submitted pursuant to Rule 405 of Regulation S-T (§ 232.405 of this

chapter) during the preceding 12 months (or for such shorter period that the registrant was required to submit such files).    Yes ☒    No ☐

Indicate by check mark whether the registrant is a large accelerated filer, an accelerated filer, a non-accelerated filer, smaller reporting company or an emerging growth company. See the

definitions of “large accelerated filer,” “accelerated filer,” “smaller reporting company,” and “emerging growth company” in Rule 12b-2 of the Exchange Act.:

Large Accelerated Filer
Non-accelerated Filer
Emerging growth company

  ☐
  ☒ 
  ☒

  Accelerated Filer
  Smaller Reporting Company

  ☐
  ☒

If an emerging growth company, indicate by check mark if the registrant has elected not to use the extended transition period for complying with any new or revised financial accounting

standards provided pursuant to Section 13(a) of the Exchange Act ☒

Indicate by check mark whether the registrant has filed a report on and attestation to its management’s assessment of the effectiveness of its internal control over financial reporting under

Section 404(b) of the Sarbanes-Oxley Act (15 U.S.C. 7262(b)) by the registered public accounting firm that prepared or issued its audit report.  Yes ☐    No ☒

Indicate by check mark whether the registrant is a shell company (as defined in Rule 12b-2 of the Exchange Act.)    Yes ☐    No ☒
As of June 30, 2020, the last day of the registrant’s most recently completed second fiscal quarter, the aggregate market value of the Common Stock held by non-affiliates of the registrant was
approximately $293.7 million based on the closing price of the registrant’s common stock on June 30, 2020.  The calculation excludes shares of the registrant’s common stock held by current executive
officers, directors and stockholders that the registrant has concluded are affiliates of the registrant.  This determination of affiliate status is not a determination for other purposes.

As of March 8, 2021, there were 65,753,570 shares of common stock outstanding.

DOCUMENTS INCORPORATED BY REFERENCE

Portions of the registrant’s definitive proxy statement for its 2021 Annual Meeting of Stockholders, which the registrant intends to file pursuant to Regulation 14A with the Securities and

Exchange Commission not later than 120 days after the registrant’s fiscal year ended December 31, 2020, are incorporated by reference into Part III of this Annual Report on Form 10-K.

 
 
 
 
 
 
 
 
 
 
   
   
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
SPECIAL NOTE REGARDING FORWARD-LOOKING STATEMENTS

TABLE OF CONTENTS

Item 1.
Item 1A.
Item 1B.
Item 2.
Item 3.
Item 4.

Item 5.
Item 6.

Item 7.
Item 7A.
Item 8.
Item 9.
Item 9A.
Item 9B.

Item 10.
Item 11.
Item 12.
Item 13.
Item 14.

Item 15.
Item 16.

  Business
  Risk Factors
  Unresolved Staff Comments
  Properties
  Legal Proceedings
  Mine Safety Disclosures

PART I

PART II

  Market for Registrant’s Common Equity, Related Stockholder Matters and Issuers Purchases of Equity Securities
  Selected Financial Data

  Management’s Discussion and Analysis of Financial Condition and Results of Operations
  Quantitative and Qualitative Disclosures about Market Risk
  Financial Statements and Supplementary Data
  Changes in and Disagreements with Accountants on Accounting and Financial Disclosure
  Controls and Procedures
  Other Information

  Directors, Executive Officers and Corporate Governance
  Executive Compensation
  Security Ownership of Certain Beneficial Owners and Management and Related Stockholder Matters
  Certain Relationships and Related Transactions, and Director Independence
  Principal Accountant Fees and Services

PART III

  Exhibits and Financial Statement Schedules
  Form 10-K Summary

PART IV

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 SPECIAL NOTE REGARDING FORWARD-LOOKING STATEMENTS

This Annual Report on Form 10-K contains forward-looking statements within the meaning of Section 27A of the Securities Act of 1933, as amended, or the
Securities Act, and Section 21E of the Securities Exchange Act of 1934, as amended, or the Exchange Act. All statements other than statements of historical fact are
“forward-looking  statements”  for  purposes  of  this  Annual  Report  on  Form  10-K.  In  some  cases,  you  can  identify  forward-looking  statements  by  terminology  such  as
“aim,”  “anticipate,”  “assume,”  “believe,”  “contemplate,”  continue,”  “could,”  “design,”  “due,”  “estimate,”  “expect,”  “goal,”  “intend,”  “may,”  “objective,”  “plan,”
“positioned,” “potential,” “predict,” “project,” “should,” “target,” “will,” “would” or the negative or plural of those terms, and similar expressions.

Forward-looking statements include, but are not limited to, statements about:

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statements  regarding  the  impact  of  the  COVID-19  pandemic  and  its  effects  on  our  operations,  access  to  capital,  research  and  development  and
clinical trials and potential disruption in the operations and business of third-party manufacturers, contract research organizations, or CROs, other
service providers, and collaborators with whom we conduct business;

our estimates regarding expenses, future revenue, capital requirements and needs for additional financing;

our ability to identify additional novel compounds with significant commercial potential to acquire or in-license; 

our ability to successfully acquire or in-license additional drug candidates on reasonable terms;

our ability to obtain regulatory approval of our current and future drug candidates;

our expectations regarding the potential market size and the rate and degree of market acceptance of such drug candidates;

our ability to fund our working capital requirements;

the implementation of our business model and strategic plans for our business and drug candidates;

developments or disputes concerning our intellectual property or other proprietary rights;

our ability to maintain and establish collaborations or obtain additional funding;

our expectations regarding government and third-party payor coverage and reimbursement;

our ability to compete in the markets we serve;

the impact of government laws and regulations;

developments relating to our competitors and our industry; and

the factors that may impact our financial results.

Factors that may cause actual results to differ materially from current expectations include, among other things, those set forth in Part I, Item 1A, “Risk Factors,”
herein and for the reasons described elsewhere in this Annual Report on Form 10-K. Any forward-looking statement in this Annual Report on Form 10-K reflects our
current view with respect to future events and is subject to these and other risks, uncertainties and assumptions relating to our operations, results of operations, industry
and  future  growth.  Given  these  uncertainties,  you  should  not  rely  on  these  forward-looking  statements  as  predictions  of  future  events.  Although  we  believe  that  the
expectations reflected in the forward-looking statements are reasonable, we cannot guarantee future results, levels of activity, performance or achievements. Except as
required by law, we assume no obligation to update or revise these forward-looking statements for any reason, even if new information becomes available in the future.

This Annual Report on Form 10-K also contains estimates, projections and other information concerning our industry, our business and the markets for certain
drugs and consumer products, including data regarding the estimated size of those markets, their projected growth rates and the incidence of certain medical conditions.
Information that is based on estimates, forecasts, projections or similar methodologies is inherently subject to uncertainties and actual events or circumstances may differ
materially from events and circumstances reflected in this information. Unless otherwise expressly stated, we obtained these industry, business, market and other data
from reports, research surveys, studies and similar data prepared by third parties, industry, medical and general publications, government data and similar sources and we
have not independently verified the data from third party sources. In some cases, we do not expressly refer to the sources from which these data are derived.

In this Annual Report on Form 10-K, unless otherwise stated or as the context otherwise requires, references to “Ovid,” “the Company,” “we,” “us,” “our” and
similar references refer to Ovid Therapeutics Inc. and its wholly owned subsidiaries. This Annual Report on Form 10-K also contains references to our trademarks and to
trademarks belonging to other entities. Solely for convenience, trademarks and trade names referred to, including logos, artwork and other visual displays, may appear
without the ® or TM symbols, but such references are not intended to indicate, in any way, that their respective owners will not assert, to the fullest extent under

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applicable law, their rights thereto. We do not intend our use or display of other companies’ trade names or trademarks to imply a relationship with, or endorsement or
sponsorship of us by, any other companies.

Our business is subject to numerous risks and uncertainties, including those discussed at length in the section titled “Risk Factors.” These risks include, among others, the following:

We have incurred significant operating losses since inception and expect to continue to incur substantial operating losses for the foreseeable future.

SUMMARY OF SELECTED RISKS ASSOCIATED WITH OUR BUSINESS

We  have  never  generated  any  revenue  from  drug  sales.  Our  operating  history  may  make  it  difficult  to  evaluate  the  success  of  our  business  to  date  and  to  assess  our  future
viability.

We will require additional capital to finance our operations, which may not be available on acceptable terms, if at all. Failure to obtain this necessary capital when needed may
force us to delay, limit or terminate certain of our drug development efforts or other operations.

Our  future  success  is  dependent  on  the  successful  clinical  development,  regulatory  approval  and  commercialization  of  our  current  and  future  drug  candidates.  If  we,  or  our
licensees, are not able to obtain required regulatory approvals, we will not be able to commercialize our drug candidates, and our ability to generate revenue will be adversely
affected.

Because the results of preclinical studies or earlier clinical trials are not necessarily predictive of future results, our drug candidates may not have favorable results in planned or
future preclinical studies or clinical trials, or may not receive regulatory approval.

Interim topline and preliminary results from our clinical trials that we announce or publish from time to time may change as more patient data become available and are subject
to audit and verification procedures, which could result in material changes in the final data.

We may encounter substantial delays in our clinical trials or we may fail to demonstrate safety and efficacy to the satisfaction of applicable regulatory authorities.

Angelman syndrome has no treatments approved by the U.S. Food and Drug Administration, and the primary clinical endpoint, CGI-I-AS, has not previously been used as a
sole primary endpoint in a pivotal clinical trial.

If  we  are  not  successful  in  discovering,  developing  and  commercializing  additional  drug  candidates,  our  ability  to  expand  our  business  and  achieve  our  strategic  objectives
would be impaired.

Our drug candidates may cause undesirable side effects or have other properties that could delay or prevent their regulatory approval, limit the commercial potential or result in
significant negative consequences following any potential marketing approval.

Even if our current or future drug candidates receive marketing approval, they may fail to achieve market acceptance by physicians, patients, third-party payors or others in the
medical community necessary for commercial success.

If we are unable to establish sales and marketing capabilities, or enter into agreements with third parties to market and sell our current or any future drug candidates, we may be
unable to generate any revenue from drug sales.

We are heavily dependent on our relationship with Takeda Pharmaceutical Company Limited (“Takeda”) for the development and commercialization of OV935. Any disruption
in our relationship with Takeda could lead to delays in, or the termination of, the development of OV935, which would materially harm our business.

We are dependent on our relationship with Angelini Pharma Rare Diseases AG (“Angelini”) for the development and commercialization of OV101 in the European Economic
Area as well as Switzerland, the United Kingdom, Russia and Turkey. Any disruption in our relationship with Angelini could lead to delays in the development and achievement
of regulatory approval in these countries, which would materially harm our business.

We may be required to make significant payments in connection with our licenses of OV101 from H. Lundbeck A/S and OV935 from Takeda.

Our relationships with customers, physicians, and third-party payors may be subject, directly or indirectly, to federal and state healthcare fraud and abuse laws, false claims
laws, health information privacy and security laws, and other healthcare laws and regulations. If we are unable to comply, or have not fully complied, with such laws, we could
face substantial penalties.

Coverage and adequate reimbursement may not be available for our current or any future drug candidates, which could make it difficult for us to sell profitably, if approved.

If we are unable to obtain and maintain patent protection for our current or any future drug candidates, or if the scope of the patent protection obtained is not sufficiently broad,
we may not be able to compete effectively in our markets.

We may be involved in lawsuits to protect or enforce our patents, the patents of our licensors or our other intellectual property rights, which could be expensive, time consuming
and unsuccessful.

We do not have our own manufacturing capabilities and will rely on third parties to produce clinical and commercial supplies of our current and any future drug candidates.

We intend to rely on third parties to conduct, supervise and monitor our preclinical studies and clinical trials, and if those third parties perform in an unsatisfactory manner, it
may harm our business.

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COVID-19 could adversely impact our business, including our clinical trials and access to capital.

We may need to expand our organization, and we may experience difficulties in managing this growth, which could disrupt our operations.

We may be subject to numerous and varying privacy and security laws, and our failure to comply could result in penalties and reputational damage.

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PART I

Item 1. BUSINESS

Overview

We are a biopharmaceutical company focused on developing impactful medicines for patients and families living with rare neurological disorders. We believe
these disorders represent an attractive area for drug development as the understanding of the underlying biology has grown meaningfully over the last few years and today
represent  a  substantial  opportunity  medically  and  commercially.  Based  on  the  rapid  increase  in  scientific  understanding  of  the  role  of  genetics  and  key  biological
pathways relevant to diseases of the brain, we aim to identify, discover and develop novel compounds for the treatment of rare neurological disorders. We have built a
deep knowledge of such diseases, how to treat them and how to develop the clinically meaningful endpoints required for development of a compound in these disorders.
As  a  result  of  this  knowledge,  we  have  developed  a  pipeline  of  first-in-class  compounds  and  programs  and  have  demonstrated  our  model  by  progressing  compounds
through  to  late-stage  development.  We  continue  to  execute  on  our  strategy  to  build  this  pipeline  by  discovering,  in-licensing  and  collaborating  with  leading
biopharmaceutical companies and academic institutions.

Our Focus: Rare Neurological Disorders

Rare neurological disorders are among the most devastating in their impact on patients and their families. Patients suffering from these disorders typically require
full-time care, and yet are among the most underserved. We believe that there are at least 100 neurodevelopmental disorders, epileptic encephalopathies and other related
rare neurological disorders that we may be able to target. These disorders are characterized by impairments in the growth, development and functioning of the brain. Due
to a historical overwhelming preference in the drug industry to develop drugs for broader neurological indications, many of these disorders have no approved therapies.
As a result, recent scientific advancements have been overlooked, which we believe presents us with an opportunity to pursue these indications. These reasons include:

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High  penetrance  linking  genetic  defect  to  disorder  pathology.  Some  rare  neurological  disorders  have  a  genetic  origin  and  typically  have  a  strong
correlation, or penetrance, between the presence of a gene and the manifestation of the corresponding disease pathology. As a result, we believe in those
cases we can develop drug candidates that will be efficacious in patients with a given genetic profile.

Predictive genetic and other models. Recent advances in genetics enable us to employ predictive in vitro and in vivo genetic models of certain of these
disorders. These models allow us to evaluate and observe a drug candidate’s potential activity prior to initiation of clinical trials. Through these models,
we believe we will be able to select the most relevant clinical endpoints for our trials and increase the potential for clinical success.

Overlapping pathophysiology and symptoms. Neurological disorders are often characterized by a number of overlapping symptoms, such as seizures, sleep
disturbances, movement deficiencies and behavioral manifestations. We believe these commonalities will enable us to employ clinical endpoints that may
be translatable from one disorder to another, and to develop drugs that may provide a clinical benefit across multiple indications.

Early observation of proof-of-concept. By employing clinical endpoints that are highly relevant and are designed to detect meaningful clinical benefits, we
anticipate that many of our studies may provide early proof-of-concept in clinical development.

Potential  ability  to  affect  disease  progression.      We  are  focusing  on  disorders  that  are  typically  diagnosed  in  early  childhood  when  the  brain  is  still
developing. We believe that we may be able to meaningfully address symptoms and potentially alter the progression of disease, especially if the drug can
be administered early in life.

Motivated and accessible patient populations.   We are targeting our programs for disorders with motivated and accessible patient populations. We believe
that  the  patients  and  caregivers  affected  by  these  disorders  are  avid  users  of  social  media,  in  order  to  learn  about  and  share  relevant  information  and
experiences. We use digital platforms to efficiently identify new patients for our clinical trials, raise disease awareness and help connect the patient and
caregiver communities.

The Ovid Strategy

Our strategy is to pursue drug discovery and development for rare neurological disorders in a manner that is scientifically driven, patient focused and is coupled
with  an  integrated  and  discipled  approach  to  research,  clinical  development  and  business  development.  As  we  build  on  our  understanding  of  these  rare  neurological
conditions, we gain an appreciation of the way the different molecular mechanisms and pathways underlying these disorders help drive the symptoms patients suffer. This,
in turn, benefits us with the knowledge gained about genetics, relevant molecular pathways, physiological impact and clinical endpoints from one disorder to another,
which we believe will enable us to build a scalable scientific platform and efficient development capabilities. Ovid has set out to be a leader in this field, and by keeping
our focus on neurology, it is our belief that this offers us the potential to produce multiple medicines in the future, and thereby succeed in our mission.

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Scientifically Driven

We  take  a  scientifically  driven  approach  to  identify  promising  drug  candidates  for  our  pipeline.  We  are  building  our  portfolio  based  on  the  existence  of  clear
biological rationales, including a focus on disorders that have, where possible, a direct genetic linkage. We use our deep understanding of the area to identify mechanisms
of action, appropriate targets and initial drug candidates. As we advance our drug candidates into and through the clinical evaluation, we are building on the emerging
body  of  scientific  and  clinical  insights  developed  by  us  and  others  in  the  biopharmaceutical  industry  to  target  these  important  disease  pathways  of  the  brain.  As  we
evaluate data from previous and ongoing preclinical studies and clinical trials, we intend to refine and improve our scientific approach and apply these insights to continue
to build our pipeline and conduct our clinical trials.

In particular, our approach is driven by the following scientific principles:

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identify the genetic origin of the disorder;

develop understanding of gene expression and link to pathophysiology;

target biological pathways or genes for which proof-of-concept has been established via in vitro or animal models;

focus on the pathways and mechanisms that cause the pathology of the disorder and that generate the symptoms that we can target;

target optimal mechanism of action for drug candidates; and

utilize biomarkers if present that can provide evidence of the activity of our drug candidates.

Patient Focused

We are focused on the patient communities affected by the rare neurological disorders we address. We believe this aspect of our approach is critical. Each of these
disorders  affect  small  populations  of  patients,  but  carry  serious  morbidities  and  require  extensive  and  specialized  involvement  from  the  patients’  families,  caregivers,
physicians and patient advocacy groups.

Our strategy is enhanced by the following patient-focused principles:

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develop  close  relationships  with  patients,  caregivers,  families,  disease  foundations  and  key  opinion  leaders,  to  better  understand  the  history  of  these
disorders, raise awareness, identify patients and facilitate enrollment of clinical trials;

identify clinically meaningful endpoints based on input from patients and their physicians and caregivers; and

develop digital capabilities to engage, foster and maintain close relationships with patient communities.

Research and Development Coupled with Business Development

We have built a broad pipeline of potential drug candidates to treat rare neurological disorders.   Initially we in-licensed or partnered drug candidates. More recently
our pipeline has been built through our internal research and development efforts in collaboration with external leaders in the field. The intended result is to develop a
diversified pipeline to mitigate development risk and provide for scientific and medical opportunity. Central to the success of this process is coupling a highly focused and
disciplined effort to link our research effort in key laboratories around the world aimed at discovering and securing relevant assets in selected rare neurological disorders.

As a result, we have built a specialized, scalable and robust infrastructure that we believe will make us a leader in rare neurological disorders and the partner of choice
for leading biopharmaceutical companies or academic institutions that wish to maximize the value of their neurology drug candidates or research platforms in these areas.
This infrastructure spans across critical domains which include but are not exclusive of target discovery, drug delivery and clinical development. If and when our drug
candidates are approved, we also plan to establish over time a focused commercial and distribution network dedicated to rare neurological disorders in the United States
and Europe, where we believe the patient populations and medical specialists are sufficiently concentrated to effectively market our drug candidates. We believe that we
are particularly well positioned to execute on our business development strategy because of both the extensive network of our Chairman and Chief Executive Officer Dr.
Jeremy Levin and other members of our management team, as well as our demonstrated success in collaboration with partners including Takeda.  

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Our Pipeline

Our efforts have already brought two drug candidates from proof of concept and either through pivotal trials or to the initiation of pivotal trials. The following

table sets forth the status and mechanism of action of our drug candidates:

OV935 (soticlestat)

OV935 is being developed in a joint collaboration with Takeda for the treatment of rare epileptic encephalopathies. In January 2017, we entered into a license
and  collaboration  agreement  with  Takeda,  or  the  Takeda  collaboration  agreement,  to  develop  and  commercialize  OV935  (soticlestat  or  TAK-935).  Under  the  Takeda
collaboration agreement, all costs and all profits are shared on a worldwide basis and Ovid leads development and in addition is responsible for commercialization in
North America, Europe and Israel.

In  March  2021,  we  entered  into  a  royalty,  license  and  termination  agreement,  or  the  Takeda  License  and  Termination  Agreement,  with  Takeda  under  which
Takeda will secure global rights at closing from us to develop and commercialize the investigational medicine OV935 for the treatment of developmental and epileptic
encephalopathies, including DS and LGS. Closing of the Takeda License and Termination Agreement is subject to the satisfaction of customary closing conditions. See
“Business—License and Collaboration Agreements—Agreements with Takeda—2021 Royalty, License and Termination Agreement with Takeda” for a discussion of the
terms of the Takeda License and Termination Agreement.

OV935 is a potent, highly selective inhibitor of the enzyme cholesterol 24-hydroxylase, or CH24H. We believe, if approved, OV935 has the potential to become a
first-in-class and only-in-class compound targeting the metabolism of cholesterol in the brain. We believe that OV935 inhibits a key enzyme in cholesterol metabolism
pathway in the brain and may modulate the excitatory signals involved in epilepsy, which may suppress seizures. CH24H is predominantly expressed in the brain, where
it plays a central role in cholesterol homeostasis and neuronal physiology. Recent literature suggests that in addition to its impact on membrane cholesterol homeostasis in
the  central  nervous  system,  modulation  of  CH24H  may  have  an  impact  on  over-activation  of  neurotransmitter  pathways  that  have  been  implicated  in  a  number  of
neurological  disorders,  such  as  epilepsy.  Preclinical  data  suggest  that  inhibition  of  brain  CH24H  indirectly  reduces  glutamatergic  signaling  via  NMDA  receptors  and
modulates glial function and inflammation, which may impact disease pathology and epileptogenesis.

We believe that because OV935 is an inhibitor of CH24H it may modulate the excitatory signals involved in epilepsy, which may suppress seizures. In addition
to these effects on seizures and excitability of the brain, we believe that OV935 may reduce inflammation in and neurotoxic damage to the brain, which may lead to long-
term,  disease  modifying  effect.  As  a  result,  OV935  is  being  developed  in  rare  and  difficult  to  treat  epilepsies  with  the  goal  to  develop  OV935  not  just  as  a  potential
medicine to treat the seizures but also one that may have long-term disease-modifying potential. We believe that OV935 if successful in these areas may have utility in
other  areas  as  well.  OV935  is  initially  being  studied  in  those  suffering  from  severe  and  often  intractable  forms  of  DEE,  including  Dravet  syndrome,  or  DS,  Lennox-
Gastaut syndrome, or LGS, CDKL5 Deficiency Disorder, or CDD, and Duplication 15q, or Dup15q syndrome. There are limited or no therapeutic options in each of these
disorders.

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We have completed multiple trials on OV935 and expect to initiate pivotal phase 3 trials in second quarter of 2021.  Previously we completed a Phase 1b/2a
clinical  trial  of  OV935  in  a  mixed  group  of  adults  with  DEE  and  announced  the  results  in  December  2018.  The  trial  achieved  its  primary  endpoint  of  safety  and
tolerability, dose proportional reduction in a potential plasma biomarker called 24HC, and a robust reduction in seizure frequency (61% at day 92), with two patients
becoming seizure-free at the end of the treatment period. Following this trial and as further discussed below, we reported the initial data from the Phase 2 open-label
extension study (which we refer to as the ENDYMION trial) of OV935 in six patients who previously completed our 12-week Phase 1b/2a clinical trial of OV935 in
adults with DEE.

On August 25, 2020, we, together with Takeda, announced positive topline results from the ELEKTRA trial which was a phase 2 trial in DS and LGS, along with
updated findings from the ENDYMION trial. Based on the trial results of ELEKTRA and after presentation of the data and review of the phase 3 pivotal trial approach
with regulatory authorities in the US (FDA), EU (CHMP), and Japan (PMDA), we expect to initiate two separate multinational Phase 3 pivotal registrational trials in
Dravet syndrome and LGS with OV935 in the second quarter of 2021.

The FDA has granted orphan drug designation for OV935 for the treatment of Dravet syndrome and LGS.

Dravet Syndrome

Dravet syndrome is a severe form of childhood epilepsy largely genetically driven by the mutation of the SCN1A gene that typically presents during the first year
of  life.  Eighty  percent  of  patients  have  a  mutation  of  the  SCN1A-gene.  Children  experience  frequent  seizures,  loss  of  muscle  control,  cognitive  deficits  and,  in
approximately 10% of cases, death before the age of 12 years. Children continue to suffer from seizures and severe cognitive and developmental impairment throughout
their lifetime. While some patients may survive into adulthood, their long-term intellectual development and seizure outcomes are typically extremely poor. The incidence
of Dravet syndrome in the United States ranges from 1 in 15,700 to 1 in 20,900 births.

Lennox-Gastaut Syndrome

Lennox-Gastaut  syndrome  is  a  rare  disorder  that  is  often  diagnosed  between  three  and  five  years  of  age.  Patients  diagnosed  with  Lennox-Gastaut  syndrome
experience  a  multitude  of  seizure  types  that  are  difficult  to  manage  and  have  many  of  the  same  symptomologies  as  other  rare  pediatric  epilepsies.  Lennox-Gastaut
syndrome affects over 30,000 people in the United States with approximately half being children under the age of 18.  Some patients have de novo genetic mutations,
including a mutation of the SCN2A gene. The annual incidence of Lennox-Gastaut syndrome in childhood is estimated to be two per 100,000 children. It is also estimated
that between 1% and 4% of childhood epilepsies are a result of Lennox-Gastaut syndrome.

CDKL5 Deficiency Disorder

Patients with cyclin-dependent kinase-like 5 (CDKL5) mutations present with early epilepsy. In particular, early drug-resistant epilepsy, usually starting in the first
months of life, tends to be the most common feature. Complex partial seizures, infantile spasms, myoclonic, generalized tonic-clonic, and tonic seizures have all been
reported.  Stereotypic  hand  movements,  severe  hypotonia,  and  impaired  psychomotor  development  are  usually  associated  with  CDKL5  mutations  and  common  to  the
general clinical manifestations.

Dup15q syndrome

Duplications of the proximal arm of chromosome 15q11.2-q13.1 result in the genetic condition Dup15q syndrome. Multiple genes including UBE3A from this
region are implicated in the pathogenesis of autism spectrum disorders, epilepsy, and schizophrenia. Increased expression of the UBE3A gene contributes to epilepsy in
Dup15q syndrome and it is thought to be the underlying cause of the autistic features of the syndrome as well. The most devastating feature of Dup15q syndrome is
difficult to control seizures. The most common seizure types are infantile spasm and generalized tonic–clonic seizures followed by atonic, myoclonic, focal-onset, and
tonic seizures. Poorly  controlled  seizures  severely  impact  the  quality  of  life  of  both  affected  individuals  and  their  caregivers.  Current  treatment  options  for  Dup15q
syndrome-associated epilepsy are often ineffective. GABAergic promoting antiepileptics are typically ineffective while broad-spectrum antiepileptic medications such as
valproic acid and rufinamide provide some relief.

OV935 Clinical Data

Phase 1 Trials

OV935 has been tested in 86 healthy volunteers across four Phase 1 trials. Single oral doses of up to 1,350mg of OV935 were well-tolerated. The most frequently
reported adverse events were headache, ECG electrode application site dermatitis and nausea. All reported events were mild with no apparent dose-response. In a 14-day
repeat dosing trial, doses of 100mg QD, 300mg QD and 400mg QD were well-tolerated. One volunteer at the 300mg BID experienced an event of confusional state and
another volunteer at the 600mg QD dose experienced acute psychosis. Both volunteers discontinued the trial at day 11. One volunteer receiving placebo reported events of
nightmares, spatial disorientation, insomnia and dizziness. All AEs resolved with continued dosing through day 15.

4

 
No SAEs were reported. Overall, no safety issues of concern were identified in the Phase 1 trials based on assessments of physical examinations, vital sign measurements,
clinical laboratory values or 12-lead electrocardiogram findings.

The following table summarizes each Phase 1 trial:

Trial
1

   Purpose

Safety and tolerability

   Design

Phase  1,  randomized,  double-blind,  placebo-
controlled, single ascending dose trial

Number of
Volunteers
48

   Dosage

15-1,350mg, oral

2

3

4

Safety and tolerability

Phase  1,  randomized,  double-blind,  placebo-
controlled, multiple ascending dose trial

Brain CH24H enzyme occupancy using positron
emission tomography, or PET

Open-label, non-randomized

40

11

QD,
100-600mg 
and  300mg  BID,  14  days,
oral

50-600mg, oral

Relative  bioavailability  of  tablet  versus  solution
formulation; effect of food

Phase 1, randomized, open-label, single dose trial

9

300mg 
300mg (solution), oral

(tablet), 

oral;

Phase 1b/2a Trial - 2001

The Phase 1b/2a trial of OV935 achieved its primary endpoint of safety and tolerability and showed OV935 was generally well tolerated.  The trial was designed
to have two parts. Part 1 was a randomized, double-blind, placebo-controlled (OV935 vs. placebo with a ratio of 4:1), 30-day phase that included a titration period (20
days: 100 mg, 200 mg twice daily), and treatment period (10 days).

OV935 achieved the primary endpoint of safety and tolerability as measured by incidence of AEs. AEs in patients treated with OV935 were similar to those who
received placebo in Part 1. The majority of AEs in both treatment arms were mild. Overall, the data are consistent with a favorable safety and tolerability profile and
support the continued clinical development of OV935.

AEs  that  occurred  more  frequently  in  the  OV935-treatment  group  versus  the  placebo  group  were:  dysarthria,  insomnia,  lethargy,  seizure  cluster,  and  upper
respiratory infection. Four patients discontinued due to an AE or an SAE in the OV935 treatment arm. Of these, in Part 1, one patient discontinued due to difficulty with
walking and worsening lethargy and a second discontinued due to weakness. In Part 2, one patient discontinued due to a single episode of seizure cluster and a second
experienced multiple seizure clusters.

An increase in seizure frequency was seen in three patients, all of whom were on perampanel. This suggests the potential for a drug-drug interaction between
medicines acting on different glutamatergic receptors. Accordingly, changes in seizure frequency data for the Phase 1b/2a trial are now reported with the inclusion and
exclusion of the three patients on perampanel, respectively.

ENDYMION

ENDYMION  is  a  Phase  2  prospective,  multi-center,  open-label  extension  study  of  OV935  in  patients  with  DEE  who  have  participated  in  a  previous  OV935
clinical study. The primary objective is to assess the long-term safety and tolerability of OV935 over four years of treatment in patients with rare epilepsies. A secondary
endpoint evaluates the effect of OV935 on seizure frequency over time. ENDYMION enrolled eligible patients from the ELEKTRA and ARCADE trials, each discussed
below.  

In September 2019, we announced initial data from the first six patients in ENDYMION who were previously enrolled in the Phase 1b/2a clinical trial of OV935
in adults with DEE and subsequently ceased taking OV935 for a period of between 6 weeks and 12 months. Therefore, in most cases the seizure frequency increased from
the end of the adult DEE trial until they were enrolled in ENDYMION. As shown in Table 1, longer-term data from ENDYMION out to 48 weeks suggest increased
seizure reduction with prolonged treatment of OV935 and is consistent with the believed mechanism of action of OV935. Median seizure frequency reductions were 84%
following 25 to 36 weeks (n=6) and 90% following 37 to 48 weeks (n=4) of treatment.

Table 1: % Reduction from Baseline in Seizure Frequency

Overall median % reduction in seizure frequency from baseline

  Weeks 1-12

  Weeks 13-24

  Weeks 25-36   Weeks 37-48

48%
(n=6)

65%
(n=6)

84%
(n=6)

90%
(n=4)*

5

 
 
  
  
  
  
  
 
 
 
 
 
 
 
 
 
  
  
  
  
 
 
 
 
 
 
 
 
 
  
  
  
  
 
 
 
 
 
 
 
 
 
  
  
  
  
 
 
 
 
  
  
   
  
 
 
 
 
 
% of Patients with ³50% reduction in seizure frequency from baseline

50%

50%

67%

75%

*

At the time of data analysis, two patients had not yet completed 48 weeks of dosing.

Patient  baseline  seizure  frequency  ranged  from  2  to  71  (median=11.5).  In  general,  a  greater  reduction  in  seizure  frequency  was  observed  in  those  with  higher
baseline  seizure  frequency.  In  terms  of  overall  seizure-free  interval  during  treatment,  one  patient  experienced  264  consecutive  days  and  one  patient  experienced  150
consecutive days without a seizure.

In addition to the six patients from the Phase 1b/2a adult DEE trial included in this data analysis, all patients who have completed the ARCADE and ELEKTRA
trials to date have enrolled in ENDYMION. Data from patients who have completed ARCADE, our Phase 2, multi-center, open-label, pilot study evaluating the treatment
of OV935 in patients with epileptic seizures associated with CDD or Dup15q syndrome, are not included the above analysis due to their limited treatment duration in
ENDYMION. Data from patients previously treated in ELEKTRA are not included in the above analysis due to the ELEKTRA trial being double-blinded and placebo-
controlled at the time of the analysis.

Overall, at 48 weeks, safety observations were consistent with the completed Phase 1b/2a clinical trial in adults with DEE. OV935 continues to show a favorable
safety and tolerability profile. The majority of adverse events were mild and comparable with those from the Phase 1b/2a trial. Specifically, adverse events that occurred
included upper abdominal pain, pyrexia, bronchial wall thickening and rales. There was one treatment-related adverse event of nausea. No serious adverse events were
observed.

As discussed below, in August 2020 and September 2020, we announced updated findings from ENDYMION from patients who completed the ELEKTRA and

ARCADE studies, respectively, and elected to enroll in ENDYMION.

ELEKTRA

ELEKTRA was an international, multi-center, randomized, double-blind, placebo-controlled study designed to evaluate treatment with soticlestat in pediatric
patients, aged 2 to 17 years, with highly refractory epileptic seizures associated with convulsive seizures (DS) or drop seizures (LGS). The study consisted of a four- to
six-week screening period to establish baseline seizure frequency, followed by a 20-week double-blind treatment period, including an 8-week dose optimization period
and a 12-week maintenance period. During the 8-week dose optimization period, patients were titrated from 100mg twice daily (BID), to 200mg BID to 300mg BID
(mg/kg dosing for <60 kg) of orally administered soticlestat.

A total of 141 patients were enrolled in ELEKTRA and 126 completed the study. A modified intent-to-treat, or mITT, analysis of 139 patients was performed to
evaluate the efficacy endpoints, which includes any patient who enrolled in the study and received at least one dose of study drug. Patients in the study were allowed to be
on one to four concomitant anti-epileptic drugs, or AEDs, with the majority of patients concomitantly treated with at least three AEDs. The most common AEDs taken by
the patients were valproate, clobazam, levetiracetam and topiramate. Further, all patients who completed ELEKTRA enrolled in the ENDYMION open-label extension
study.

On August 25, 2020, we, together with Takeda, announced positive topline results from ELEKTRA and updated findings from ENDYMION. The ELEKTRA
study achieved its primary endpoint with high statistical significance, demonstrating a 27.8% median reduction from baseline in convulsive seizure (DS) and drop seizure
(LGS) frequency compared to a 3.1% median increase in patients taking placebo during the 12-week maintenance period (median placebo-adjusted reduction=30.5%;
p=0.0007,  based  on  the  efficacy  analysis  set  of  120  patients  with  seizure  data  in  the  maintenance  period).  In  addition,  DS  and  LGS  patients  treated  with  soticlestat
demonstrated a 29.8% median reduction in convulsive seizure (DS) and drop seizure (LGS) frequency compared to 0.0% change in median seizure frequency in patients
taking placebo during the full 20-week treatment period (titration plus maintenance) of the ELEKTRA study (placebo-adjusted reduction=25.1%; p=0.0024). Soticlestat
was generally well-tolerated in the ELEKTRA study and demonstrated a safety profile consistent with those of previous studies, with no new safety signals identified. All
patients who completed the ELEKTRA study elected to enroll into the ENDYMION open-label extension study and findings from ENDYMION were also reported on
August 25, 2020.  The ENDYMION study data of rolled-over ELEKTRA patients support results in the ELEKTRA study. The ENDYMION data indicated maintenance
of effect over 6 months in those patients originally randomized to soticlestat, and similarly reduced seizure frequency as compared to baseline in those patients previously
assigned to the placebo arm. No new safety signals were identified in ENDYMION.

ARCADE

ARCADE  is  a  Phase  2  open-label,  signal-finding  pilot  study  designed  to  inform  the  potential  for  future  development  of  soticlestat  in  CDD  and  Dup15q
syndrome. The study enrolled 20 patients, ages 2 to 55 years, with refractory epileptic seizures associated with CDD (n=12) or Dup15q (n=8) and consisted of a four- to
six-week screening period to establish baseline seizure frequency, followed by a 20-week treatment period, including an eight-week titration/dose optimization period and
a 12-week maintenance period. Patients in the study were allowed to be on one to six concomitant AEDs, with the majority of patients

6

 
 
 
 
 
 
concomitantly treated with at least four AEDs, representing a highly refractory patient population. The primary objective of the ARCADE study was to determine percent
change from baseline in motor seizure frequency during the 12-week maintenance period.  Further, all patients who completed ARCADE enrolled in the ENDYMION
open-label extension study.

On September 30, 2020, we announced results from ARCADE and updated findings from ENDYMION. Together, data from the ARCADE and ENDYMION
studies showed seizure frequency reduction over time. In CDD patients (n=12), median motor seizure frequency reduction was 24% during the 12-week maintenance
period  in  the  ARCADE  study,  increasing  to  a  50%  reduction  in  the  ENDYMION  long-term  extension  study  in  the  five  CDD  patients  who  reached  nine  months  of
continuous treatment. In Dup15q patients (n=8), there was an increase in median motor seizure frequency in the ARCADE study during the 12-week maintenance period;
however, longer-term data from the four Dup15q patients who reached nine months of continuous treatment showed a 74% reduction in median motor seizure frequency.
Soticlestat was generally well tolerated in both studies and continues to demonstrate a favorable safety profile. We believe the results are encouraging and next steps are
being evaluated with Takeda.

OV101 (gaboxadol)

To  date,  we  have  been  developing  OV101  for  the  treatment  of  Angelman  syndrome  and  Fragile  X  syndrome,  two  neurodevelopmental  disorders  that  are
characterized by similar symptoms. In December 2020, we reported the primary endpoint of the Pivotal Phase 3 trial in pediatric individuals with Angelman syndrome
(the NEPTUNE trial) was not achieved. Based on the results of the NEPTUNE trial, further development of OV101, other than the ongoing long-term extension study
with Angelman syndrome patients who had previously been in a trial for OV101 (the ELARA trial), is currently on hold. The data from all trials is under review and
further development of OV101, if any, will be the subject of full analysis of this data.

Angelman  syndrome  and  Fragile  X  syndrome  have  overlapping  symptoms,  including  sleep  disorder,  aberrant  behavior,  anxiety  and  cognitive  or  intellectual
disabilities thought to be caused by decreased tonic inhibition, an important mechanism whereby it is believed that the brain distinguishes signal from noise. Both of these
disorders are typically diagnosable in early childhood and require full-time care for the patients affected. In September 2016, the FDA granted orphan drug designation
for OV101 for the treatment of Angelman syndrome; in October 2017 the FDA granted orphan drug designation for OV101 for the treatment of Fragile X syndrome; in
December 2017 the FDA granted fast track designation for the treatment of Angelman syndrome; and in March 2018, the FDA granted fast track designation for the
treatment of Fragile X syndrome.  In June 2019, the European Commission granted OV101 orphan drug designation for the treatment of Angelman syndrome based on
the results of the STARS clinical trial.

OV101 and Tonic Inhibition

Tonic  inhibition  is  a  critical  physiological  regulatory  mechanism  that  allows  a  healthy  human  brain  to  decipher  excitatory  and  inhibitory  neurological  signals
correctly without being overloaded. Defects of this system are thought to play a role in multiple disease states, including Angelman syndrome, Fragile X syndrome and
insomnia. Because of its unique mode of action, OV101 represents a promising compound targeting this mechanism.

Decreased tonic inhibition results in an imbalance in the ratio of excitation to inhibition. If tonic inhibition is reduced, the brain becomes inundated with signals
and  loses  the  ability  to  separate  background  noise  from  critical  information.  This  imbalance  disrupts  normal  brain  functioning,  including  sensory  processing  and
integration.  Disruption  of  tonic  inhibition  can  lead  to  a  multiplicity  of  symptoms  including,  but  not  limited  to,  sleep  abnormalities,  motor  deficiencies,  behavioral
manifestations, delayed development, intellectual disability and severe speech impairment.  By  modulating  tonic  inhibition,  OV101  may  have  the  potential  to  alleviate
important symptoms and provide a meaningful clinical benefit to patients across several disorders.

We  believe  that  OV101  modulates  tonic  inhibition.  Disruption  of  tonic  inhibition  can  lead  to  a  multiplicity  of  symptoms  including,  but  not  limited  to,  sleep
abnormalities,  motor  deficiencies,  behavioral  manifestations,  delayed  development,  intellectual  disability  and  severe  speech  impairment.  We  believe  modulating  tonic
inhibition may have a meaningful clinical impact in patients with Angelman syndrome and Fragile X syndrome.

7

 
Angelman Syndrome

Overview.     Angelman  syndrome  is  a  rare  genetic  disorder  that  is  typically  diagnosed  in  the  United  States  after  one  year  of  age  when  parents  notice  severe
developmental delays or the child suffers seizures. Characteristic features of this disorder include delayed development, intellectual disability, severe speech impairment,
problems  with  movement  and  balance,  seizures,  sleep  disorders  and  anxiety.  Individual  patients  with  Angelman  syndrome  can  have  varied  symptoms,  including  the
inability to walk or control motor movement, which can limit their ability to handle daily functions such as feeding, dressing or bathing. These patients are also often
hyperactive,  leading  to  various  behavioral  problems.  Angelman  syndrome  symptoms,  such  as  poor  sleeping  patterns,  can  lead  to  serious  consequences,  including
increased  frequency  of  seizures  and  exacerbation  of  behavioral  manifestations.  Different  patients  with  identical  genetic  defects  can  show  different  degrees  of  these
symptoms.  Most  Angelman  syndrome  patients  require  full-time  care  and  are  unable  to  live  independently,  which  can  represent  a  substantial  emotional  and  financial
burden on their families. In addition, Angelman syndrome has been associated with poor parental sleep and high parental stress.

According to the National Organization for Rare Disorders, the approximate prevalence of Angelman syndrome is between 1 in 12,000 and 1 in 20,000 people.
There are currently no approved therapies in the United States or ex-US specifically for the treatment of Angelman syndrome. No standard of care exists for Angelman
syndrome, and current therapeutic options are symptomatic, suggesting a high unmet clinical need. Given the likely high burden of Angelman syndrome, new treatments
targeting the aetiology of the syndrome that result in even small improvements in features of the syndrome may be clinically meaningful for patients and their families.

Fragile X Syndrome

Overview.      Fragile  X  syndrome  is  a  genetic  condition  that  results  in  intellectual  disability,  anxiety  disorders,  behavioral  and  learning  challenges  and  various
physical  disabilities.  Patients  with  Fragile  X  syndrome  exhibit  autism-like  symptoms,  including  cognitive  impairment,  anxiety,  mood  swings,  hyperactivity,  attention
deficit and heightened sensitivity to various stimuli, such as sound. The severity of an individual patient’s impairment can range from mild learning disabilities to more
severe cognitive or intellectual disabilities. Fragile X syndrome is one of the most commonly inherited intellectual disability disorders. Children with Fragile X syndrome
also often have unusual sleep patterns and may have difficulty with routine activities such as feeding and dressing. The challenges presented by Fragile X syndrome often
extend beyond the patient and can lead to significant hardships on the emotional and financial health of their families.

Fragile X syndrome is caused by mutations in the fragile X mental retardation gene, or FMR1 gene. FMR1 is a gene that leads to the synthesis of the fragile X
mental retardation protein, FMRP, which is needed for normal brain development. The FMR1 gene normally contains in its sequence between 5 and 44 copies of a short,
repeated motif, or recurring pattern in DNA. In Fragile X syndrome, there are more than 200 copies of this motif in the FMR1 gene, a genetic change that prevents the
synthesis of FMRP. Patients with intermediate numbers of repeats are able to make some FMRP and have milder symptoms.

According  to  the  National  Fragile  X  Foundation,  Fragile  X  syndrome  affects  approximately  1  in  3,600  to  4,000  males  and  1  in  4,000  to  6,000  females.  The
average age of diagnosis of Fragile X syndrome is approximately three years. Currently, there are no approved therapies for the treatment of Fragile X syndrome. The
current standard of care for the psychiatric challenges of Fragile X syndrome is tailored to each patient and may include antipsychotics, antidepressants and drugs to treat
attention deficit and sleep disorders. Special education and symptomatic treatments for anxiety and irritability are often employed to lessen the burden of illness. Fragile
X syndrome patients also may experience seizures, which are treated with traditional anticonvulsants.

We have conducted a number of clinical trials with OV101. In 2017, we completed a successful Phase 1 clinical trial in adolescent patients with Angelman and
Fragile X syndrome. In 2018, we completed a Phase 2 trial of OV101 in adults and adolescents with Angelman syndrome, which we refer to as the STARS clinical trial.
The STARS clinical trial achieved its primary endpoint of safety and tolerability and showed statistically significant improvement in the once-daily OV101 dosing group
on the pre-specified physician-rated Clinical Global Impressions-Improvement, or CGI-I, exploratory endpoint as well as improvements in relevant symptoms such as
sleep, motor function and behavior.

Based on the results of the NEPTUNE trial, further development of OV101, other than the ELARA trial, is currently on hold. The data is under review and further

development, if any, will be the subject of full analysis of the data from this trial together with the data from ELARA.

Angelman Syndrome

STARS

In July of 2018, we completed the Phase 2 STARS trial, a 12-week, double blind, placebo-controlled study in adults and adolescents with Angelman syndrome
that randomized 88 patients aged 13 to 49 years. The study achieved its primary endpoint of safety and tolerability with a similar incidence of adverse events, or AEs,
across  the  OV101  and  placebo  treatment  arms.  The  investigational  medicine  showed  a  favorable  safety  profile  and  was  well  tolerated  in  adults  and  adolescents  with
Angelman syndrome through the 12 weeks of treatment. The most common AEs reported in the trial were vomiting, somnolence, irritability, aggression, and pyrexia.
Serious adverse events, or SAEs, of seizure were reported in two patients with a previous history of seizures: one patient

8

 
in the once-daily, QD, dose group experienced a seizure that was deemed unrelated to study drug; one patient experienced a seizure in the twice-daily, BID, dose group
that was assessed as possibly related to study drug by the investigator.  At the prespecified efficacy analysis at 12 weeks of treatment, OV101 QD and BID dose groups
showed a statistically significant improvement compared to placebo in the CGI-I. CGI-I was ranked first in the prespecified hierarchy of the statistical analysis plan. Data
from the full analysis indicate that OV101 positively impacts several relevant clinical features of Angelman syndrome (global functioning, sleep, motor disruption). We
met with the FDA in November 2018 to discuss OV101 as part of our End of Phase 2 Meeting.

NEPTUNE

Following the End of Phase 2 Meeting, we initiated the NEPTUNE trial and enrolled our first pediatric patient in September 2019. NEPTUNE was a randomized,
double-blind, placebo-controlled, Phase 3 study that enrolled and treated 97 pediatric patients diagnosed with Angelman syndrome, four to 12 years of age, and seven
patients  diagnosed  with  Angelman  syndrome  ages  two  to  three  years  for  safety  and  pharmacokinetic  evaluation  only.  The  study  was  designed  to  assess  the  effects  of
treatment with OV101 (oral, once-daily dosing) versus placebo over 12 weeks. The sole primary endpoint was change in overall score on the Clinical Global Impression-
Improvement-Angelman  syndrome,  or  CGI-I-AS,  scale.  Secondary  endpoints  included  sleep,  communication,  motor  function,  socialization,  daily  living  skills  and
behaviour domains.

The primary endpoint of the NEPTUNE study was not achieved. Patients given OV101 showed a 0.7-point improvement in CGI-I-AS over baseline while placebo
also showed a 0.8-point improvement in CGI-I-AS (p=NS). Secondary endpoints continue to be evaluated, although initial results show no difference between OV101
and placebo.

OV101 was well-tolerated, with no significant safety issues observed. We plan to complete a full analysis of the results of the NEPTUNE study and discuss these
results with the FDA to determine next steps, if any, for the program. We will continue to offer study drug to patients enrolled in the open-label extension trial, ELARA,
pending further analysis of the NEPTUNE study.

ELARA

Based on the STARS clinical trial data, we also initiated ELARA, an open-label extension trial which enrolled its first patient in February 2019, and enrollment is

ongoing. We expect to report data from the ELARA study in the first half of 2021.

Based on the results of the NEPTUNE trial, further development of OV101, other than the ELARA trial, is currently on hold. The data is under review and further

development, if any, will be the subject of full analysis of the data from this trial together with the data from ELARA.

Fragile X Syndrome

ROCKET

In May 2020, we completed a Phase 2 trial evaluating OV101 in adolescent and young male adults with Fragile X syndrome, which we refer to as the ROCKET
clinical trial. The trial met its primary objective and OV101 appeared to be well tolerated over 12 weeks of treatment with no serious adverse events reported across all
three  dose  cohorts.  OV101  demonstrated  a  statistically  significant  effect  on  secondary  behavioral  endpoints  in  the  three  combined  study  groups  as
follows:  26.2%  mean  improvement  in  the  Aberrant  Behavior  Checklist  for  Fragile  X  (ABC-CFXS)  total  score  from  baseline  to  week  12  (p=0.002);  and
a 21.6% mean improvement in the Anxiety, Depression and Mood Scale (ADAMS) total score from baseline to week 12 (p=0.004). Statistically significant improvements
were also observed across various ABC-FXS and ADAMS subscales. In addition, OV101 demonstrated a statistically significant mean reduction of 0.4 in the Clinical
Global Impressions Scale-Severity (CGI-S) total score (p=0.002) from baseline to week 12.

SKYROCKET

We  also  initiated  the  SKYROCKET  study  in  the  fourth  quarter  of  2018.    SKYROCKET  was  a  12-week,  non-drug  study  to  assess  the  suitability  of  several
behavioral scales in individuals with Fragile X syndrome. The trial was an observational study designed to provide additional data on the key endpoints that are being
explored in the ROCKET trial as well as provide contextual data on the benefit offered by the standard of care. The participating clinicians and caregivers were aware that
the trial was non-interventional. The mean changes from baseline to week 12 were evaluated in the ABC total and subscale scores, the ADAMS subscale scores, and the
CGI-S subscale scores as well as the mean change in CGI-I score at week 12. Other exploratory scales were also assessed. High variability was seen among caregiver-
administered assessments (ABC-c, ADAMS) compared to clinician-assessed scales (CGI-I, CGI-S). The caregiver-administered assessments showed a placebo response
as  seen  with  previous  Fragile  X  syndrome  trials.  In  these  other  trials,  placebo  response  rates  were  highly  variable.  Therefore,  the  SKYROCKET  trial  data  will  help
inform future study design, including potential endpoints and measures to mitigate placebo response.  

Based on the results of the NEPTUNE trial, development of OV101 in Fragile X syndrome is under review to enable us to fully understand the ramifications if any,

for any potential future trial in Fragile X syndrome.

9

 
Previous Clinical Development of OV101 in Insomnia

We acquired worldwide rights to OV101 from H. Lundbeck A/S, or Lundbeck, in March 2015. Prior to the acquisition, Lundbeck filed an investigational new
drug application, or IND, with the FDA for the treatment of insomnia. Pursuant to this IND, Lundbeck and Merck & Co., Inc., or Merck, partnered to conduct several
Phase 3 trials for primary insomnia between 2004 and 2007. Over the course of the development of OV101, over 4,000 adults were administered OV101, resulting in an
OV101 exposure of approximately 950 patient years. These trials were primarily randomized, placebo-controlled short-term and long-term safety and efficacy clinical
studies,  using  classic  sleep  parameters  such  as  total  sleep  time,  time  to  sleep  onset,  wakefulness  after  sleep  onset,  and  number  of  nocturnal  awakenings  as  clinical
endpoints.

The Phase 3 program consisted of three trials: two 3-month placebo-controlled trials conducted in the United States and one 2-week trial conducted in Europe and
Canada, each evaluating OV101 against placebo and the active comparator, zolpidem (Ambien). The primary endpoints of the trials included total sleep time and time-to-
sleep onset and the secondary endpoints included number of nocturnal awakenings, wakefulness after sleep onset and daytime function. In Phase 3 trials, which were
conducted for durations of up to 12 months, OV101 was observed to have efficacy that was largely comparable to zolpidem (Ambien) on several sleep metrics. In the first
3-month trial, a dose of 15mg of OV101 met both of the primary endpoints as well as the secondary endpoints at week one and month three compared to placebo. In the
second 3-month trial, the same dose met only total sleep time and number of awakenings at week one, but significance was lost after adjusting for multiplicity at month
three.  The  2-week  trial  met  all  primary  endpoints  and  wakefulness  after  sleep  onset,  for  15mg  of  OV101  at  weeks  one  and  two.  Additionally,  subjects  who  were
administered  OV101  showed  no  evidence  of  withdrawal  symptoms  or  rebound  insomnia  after  discontinuation  of  short-term  treatment,  whereas  transient  rebound
insomnia was observed in subjects receiving zolpidem. In addition, clear differences were observed between OV101 and zolpidem from a sleep architecture perspective.
OV101 has shown consistent increases in slow wave sleep compared to zolpidem with no significant effect on stage 2 or REM sleep in healthy adult, elderly subjects. It is
believed  that  slow  wave  sleep  is  important  for  encoding  long-term,  fact-based  memories.  Slow  wave  sleep  has  been  associated  with  physical  changes  in  neuronal
connections.

Safety and Tolerability

Overall, OV101 was observed to be well-tolerated in adult patients aged 18-64 years in the Phase 2 and Phase 3 insomnia trials at doses of 5mg to 15mg given as evening
doses. Success in these previous trials does not ensure that our clinical trials in OV101 will generate the same results or otherwise provide adequate data to demonstrate the
efficacy and safety of OV101. The most common reported adverse events were headache, nausea, vomiting, somnolence and dizziness. In general, the adverse events appeared to
be dose-related. The majority of the serious adverse events observed were considered to not be related to treatment with OV101. One SAE, fatigue, was considered by Lundbeck
and Merck as probably related to OV101 treatment. Among the nine SAEs considered by Lundbeck and Merck to be possibly related to OV101 treatment, there were three cases
of fainting and one case each of: radius fracture, abnormal QRS axis, transient ischemic attack, non-cardiac chest pain, unresponsive to stimuli and atrial fibrillation. Across trials
there were no apparent clinical trends regarding SAEs with respect to frequency, distribution across system organ classes or preferred terms. Also, there were no apparent clinical
differences versus placebo. In the Phase 3 trials at the 15mg dose, at least one SAE was observed in 1.3% of subjects at two weeks and 3 months and 3.0% of subjects at 12
months versus 0.0% to 1.0% on placebo over the same time frame.

Consistent with the clinical development of other insomnia drugs, the FDA requested that Lundbeck and Merck conduct a series of preclinical and clinical abuse
studies as part of their development program. In preclinical studies, OV101 demonstrated low abuse potential. In one clinical trial, the abuse potential of OV101 was
investigated  in  doses  up  to  45mg  in  male  and  female  subjects  with  a  history  of  hypnotic/sedative  abuse  and  other  drug  abuse.  Safety  results  showed  that  OV101
administered at doses of 30mg and 45mg in women and 45mg in men was not tolerated in this population of drug abusers, contrary to previous experience with the same
doses in healthy volunteers. This indicated that a history of drug abuse decreased tolerability to OV101 in these subjects. Adverse events that were associated with a dose-
dependent lack of tolerability in this trial included psychiatric, nervous system, musculoskeletal and gastrointestinal disorders.

In 2007, following the completion of all clinical trials for OV101 in insomnia, Lundbeck and Merck discontinued the development program for insomnia, and

announced that the overall clinical profile did not support further development of OV101 for insomnia.

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Early-stage Research Programs

OV329 (GABA aminotransferase inhibitor) is a preclinical compound being developed by us for the treatment of seizures associated with Tuberous Sclerosis
Complex  and  Infantile  Spasms.  OV329  functions  by  substantially  reducing  the  activity  of  GABA  aminotransferase  (GABA-AT),  a  key  enzyme  responsible  for  the
degradation of the brain’s major inhibitory neurotransmitter, GABA. OV329 leads to increased concentrations of GABA by inhibiting its metabolism. Given that epilepsy
is  characterized  by  excessive  neuronal  excitation,  the  increased  levels  of  GABA  may  suppress  this  excitatory  signaling  and  may  reduce  seizures.  If  successful,  we
anticipate OV329 could be used to treat seizures associated with Tuberous Sclerosis Complex and Infantile Spasms and we are currently assessing this approach in the
pre-clinical setting. In December 2016, we entered into a license agreement with Northwestern University, or Northwestern, pursuant to which Northwestern granted us
an exclusive, worldwide license to patent rights in certain inventions, or the Northwestern Patent Rights, which relate to a specific compound and related methods of use
for such compound, along with certain Know-How related to the practice of the inventions claimed in the Northwestern Patents.

OV882 is a short hairpin RNA (shRNA-551) we are evaluating as a potential disease-modifying gene therapy for Angelman syndrome. The most common
cause of Angelman syndrome is the loss of functional UBE3A protein due to a defect in the maternal copy of the UBE3A gene. Our aim is to develop a disease-modifying
noncoding RNA vector that reduces expression of UBE3A-antisense and restores UBE3A expression via the paternal gene copy. We are in early stages of our research.
This research program is being conducted in collaboration with the University of Connecticut School of Medicine

In June 2020, we began a strategic research collaboration with Columbia University Irving Medical Center, or Columbia, to advance genetic based therapies
for  a  range  of  rare  neurological  conditions,  complementary  of  our  pipeline.  This  collaboration  provides  us  with  the  potential  to  expand  our  future  drug  development
portfolio  and  impact  individuals  living  with  rare  genetic  neurological  conditions  by  working  closely  with  the  Precision  Medicine  Resource  in  the  Irving  Institute  at
Columbia.  Our  first  research  program  with  Columbia  is  OV815  and  focuses  on  the  kinesin-family  of  proteins  and  KIF1A-associated  neurological  disorder  (KAND),
under this research and translational development alliance, Columbia will align its expertise in rare disease genetics and deep clinical understanding of rare neurological
diseases with our discovery, translational, and clinical development expertise in neurodevelopmental disorders and rare epilepsies.

License and Collaboration Agreements

      Collaboration Agreement with Angelini Pharma

On July 9, 2020, we entered into the Angelini License Agreement with Angelini, pursuant to which we granted to Angelini exclusive rights to develop and
commercialize OV101, a selective agonist of the GABAA receptor, for the treatment of Angelman syndrome in the European Economic Area as well as Switzerland, the
United Kingdom, Russia and Turkey, or the European Territory.  The licenses granted to Angelini include sublicenses under the Lundbeck Agreement, as well as licenses
under our patents and know-how covering OV101.  Angelini will be responsible for conducting any clinical trials necessary to obtain regulatory approval for OV101 for
Angelman syndrome in the European Territory, and we will be responsible for bearing a portion of the costs for such trials.  We will also be responsible, at our expense,
for the completion of certain ongoing clinical trials for OV101, to the extent applicable to obtaining regulatory approval for OV101 in the European Territory.  Angelini
has the exclusive right, at its election, to develop and commercialize OV101 for the treatment of Fragile X Syndrome in the European Territory.  The parties may also
mutually agree to pursue additional indications for OV101 in the European Territory, and in such case, Angelini would have the exclusive rights to commercialize in such
additional indications. Angelini is required to use commercially reasonable efforts to conduct development activities for OV101, and following regulatory approval, to
commercialize OV101 in each approved indication.

In  conjunction  with  the  entry  into  the  Angelini  License  Agreement,  the  parties  entered  into  a  separate  supply  agreement,  pursuant  to  which  we  will  be
responsible  for  supply  of  OV101  to  Angelini  for  development  and  commercialization  in  the  European  Territory,  through  Angelini’s  existing  supply  relationship  with
Lundbeck.    The  Angelini  License  Agreement  also  provides  for  a  transfer,  at  Angelini’s  expense,  of  the  relevant  manufacturing  technology  from  us  and  Lundbeck  to
Angelini, in order to enable Angelini to assume responsibility for its own manufacture and supply of OV101 in the future.

Under the Angelini License Agreement, Angelini made an upfront payment and a milestone payment related to the transfer of a specified amount of compound
and related information to the Company of $25.0 million during the year ended December 31, 2020.  Angelini will be required to make additional milestone payments to
us upon the completion of the specified components of the technology transfer and achievement of specified regulatory milestones for OV101 in Angelman syndrome of
up to $55.0 million in the aggregate, as well as up to €162.5 million ($199.9 million) in sales milestone payments for achievement of specified levels of net sales in the
European Territory.  In addition, Angelini will be required to pay tiered royalties on net sales by Angelini, its affiliates or sublicensees at double-digit percentages above
the teens, subject to certain reductions and offsets.  Royalties will be payable on a product-by-product and country-by-country basis until the latest of the expiration of the
licensed patents covering such product in such country, the expiration of market exclusivity for such product in such country, and fifteen years from first commercial sale
of such product in such country.

11

 
 
 
Either party may terminate the Angelini License Agreement for an uncured material breach of the other party or in the case of insolvency.  We may terminate
the  Angelini  License  Agreement  if  Angelini  challenges  any  of  the  licensed  patents.   Angelini  may  terminate  the  Angelini  License  Agreement  for  convenience  during
specified notice periods, which are determined based upon whether the product has been commercially launched in the European Territory.

License Agreement with H. Lundbeck A/S

In  March  2015,  we  entered  into  a  license  agreement  with  Lundbeck,  which  we  subsequently  amended  in  May  2019,  or  the  Lundbeck  agreement,  pursuant  to
which  we  obtained  from  Lundbeck  an  exclusive  (subject  to  certain  reserved  non-commercial  rights),  worldwide  license  to  develop,  manufacture,  and  commercialize
OV101,  also  known  as  gaboxadol,  for  the  treatment  of  human  disease.  Under  the  Lundbeck  agreement,  we  are  responsible  for  and  will  use  commercially  reasonable
efforts  to  carry  out  all  future  development  and  commercialization  of  OV101.  Initially,  we  will  purchase  OV101  compound  from  Lundbeck’s  existing  inventory  at  a
specified price. Following the depletion of the existing inventory, we may purchase the compound from a third party or, if the parties agree, Lundbeck may continue to
supply the compound to us. We are also obligated to make certain manufacturing-related payments to Lundbeck, including for its preparation of a drug master file for
OV101.

In connection with the Lundbeck agreement, we issued 489,756 shares of our common stock to Lundbeck. We also agreed to pay to Lundbeck milestone
payments up to an aggregate of $189.0 million upon the achievement of certain global development, regulatory and sales milestone events. Pursuant to the Lundbeck
agreement, the first milestone payment is $1.0 million, which is due upon the successful completion of the first Phase 3 trial for a product in which OV101 is an active
ingredient.  In addition, if we successfully develop and commercialize OV101, we will be obligated to pay to Lundbeck tiered royalties based on single-digit and low-
double digit percentage of net sales of OV101, subject to certain reductions for generic product sales and for royalties paid for licenses to third party intellectual property.
If  Lundbeck  manufactures  OV101  compound  for  us  after  the  expiration  of  the  royalty  term,  we  will  pay  to  Lundbeck,  in  addition  to  the  fully  burdened  cost  of  such
manufacture, a low, single-digit manufacturing royalty on the net sales of OV101 manufactured by Lundbeck.

The Lundbeck agreement will continue until the expiration of all relevant royalty terms and may be earlier terminated by either party for the other party’s uncured
material breach or insolvency. In addition, we can terminate the Lundbeck agreement upon advance notice for convenience at any time prior to first regulatory approval of
OV101. If the Lundbeck agreement is terminated by us for convenience or by Lundbeck for our breach or insolvency, the OV101 compound will revert to Lundbeck and
we will grant Lundbeck an exclusive license to develop and commercialize OV101; such license will be royalty-bearing if we filed an application for regulatory approval
prior  to  termination.  If  we  terminate  the  Lundbeck  agreement  for  Lundbeck’s  breach  or  insolvency,  our  license  will  continue  and  our  obligations  to  make  royalty
payments to Lundbeck and to share Asian Partner payments with Lundbeck will continue but we will not be obligated to make further milestone payments to Lundbeck or
to purchase any additional quantities of OV101 compound from Lundbeck’s existing inventory.

Agreements with Takeda

2017 License and Collaboration Agreement with Takeda

In  January  2017,  we  entered  into  the  Takeda collaboration agreement with  Takeda.  All  activities  of  the  collaboration  regarding  OV935  will  be  guided  by  the
Takeda/Ovid “One Team” concept, an integrated and interdisciplinary team from both companies devoted to the successful advancement of OV935 across rare epilepsy
syndromes.  Pursuant  to  the  Takeda  collaboration  agreement,  we  will  take  the  lead  in  nonclinical  and  clinical  development  activities  and  commercialization  of  the
compound  OV935  and  products  containing  this  compound  (as  well  as  certain  other  similar  compounds,  including  any  prodrug  where  TAK-935  is  the  primary
pharmacologically active metabolite) for the treatment of certain rare neurological diseases in the United States, Canada, the European Union and Israel. Takeda will take
the lead in commercialization of OV935 in Japan and has the option to lead in Asia and the rest of the world, or the Takeda Territory. While we and Takeda have agreed to
initially focus on certain rare neurological disorders, the scope of the collaboration may in the future include other mutually agreed upon rare neurological disorders.

Under  the  Takeda  collaboration  agreement,  Takeda  granted  to  us  an  exclusive  license  in  our  territory  under  certain  patents  and  other  intellectual  property
controlled  by  Takeda  to  commercialize  OV935  and  products  containing  OV935  for  the  treatment  of  certain  rare  neurological  disorders.  Takeda  also  granted  to  us  a
worldwide,  co-exclusive  license  to  develop,  manufacture  and  otherwise  exploit  (but  not  commercialize)  OV935  and  products  containing  OV935  for  the  treatment  of
certain rare neurological disorders.

Under the Takeda collaboration agreement, we granted to Takeda an exclusive license in the Takeda Territory under certain patents and other intellectual property
controlled  by  us  to  commercialize  OV935  and  products  containing  OV935  for  the  treatment  of  certain  rare  neurological  disorders.  We  also  granted  to  Takeda  a
worldwide,  co-exclusive  license  to  develop,  manufacture  and  otherwise  exploit  (but  not  commercialize)  OV935  and  products  containing  OV935  for  the  treatment  of
certain rare neurological disorders and a co-exclusive license in certain countries to commercialize OV935 and products containing OV935 for the treatment of certain
rare neurological disorders that are subsequently included in the collaboration.

12

 
 
We  and  Takeda  are  collaborating  in  the  development  of  OV935.  Pursuant  to  the  terms  of  the  Takeda  collaboration  agreement,  each  party  is  required  to  use
commercially reasonable efforts to develop OV935 for the treatment of certain rare neurological disorders in accordance with a mutually agreed upon development plan.
We are primarily responsible for activities related to the development of OV935, and as such Takeda will transition certain development activities to us. Takeda is initially
responsible for regulatory activities in all countries (excluding Israel). We are initially responsible for regulatory activities in Israel, and, upon regulatory approval in the
United States, Canada, and the European Union, we will assume responsibility for further regulatory activities in such jurisdictions.

We and Takeda are collaborating in the commercialization of OV935. Pursuant to the terms of the Takeda collaboration agreement, each party is required to use
commercially reasonable efforts to commercialize OV935 for the treatment of certain rare neurological disorders in its territory. We are responsible for commercialization
of OV935 in the United States, Canada, the European Union and Israel, and Takeda is responsible for commercialization of OV935 in Japan and has the first right to elect
to commercialize the products in the Takeda Territory. Additionally, Takeda has the right to jointly commercialize the products with us in the United States and/or the
European Union for any additional mutually agreed upon rare neurological indication.

Under the Takeda collaboration agreement, we and Takeda initially share equally all development and commercialization costs and expenses prior to launch of a
product and all revenues and commercialization costs and expenses after launch. In the event that we and Takeda agree to expand the scope of the collaboration to include
additional rare neurological disorders, either party may elect not to fund all or a portion of the development of such indication, in which case such party’s overall share of
revenues and commercialization costs and expenses after launch of a product may be reduced under certain circumstances.

During  the  period  commencing  on  the  effective  date  of  the  Takeda  collaboration  agreement,  we  and  Takeda  have  both  agreed  that  we  will  not,  directly  or
indirectly, and will cause all of our respective affiliates, not to, alone or with others, commercialize any competing product in the field of rare neurological disorders. For
these purposes, a competing product is any product or compound directed against CH24H as its primary, intended mode of action. If, during such period, we or any of our
affiliates is acquired by a third party that is commercializing a competing product, then we must divest our interest or terminate the commercialization of the competing
product or cause our affiliate to do so.

The Takeda collaboration agreement will expire upon the cessation of commercialization of the products by both us and Takeda. Either party may terminate the
Takeda  collaboration  agreement  as  a  result  of  the  other  party’s  uncured  material  breach  or  insolvency,  for  safety  reasons,  or,  after  completion  of  the  first  proof  of
mechanism clinical trial, for convenience. Takeda may terminate the Takeda collaboration agreement for our (or our sublicensee’s) challenge to the patents licensed under
the Takeda collaboration agreement. If the agreement is terminated by Takeda for our material breach, bankruptcy or patent challenge or by us for convenience or safety
reasons, our rights to the products will cease, we will transition all activities related to the products to Takeda, and we will grant Takeda an exclusive, royalty-bearing
license under certain patents and other intellectual property controlled by us to commercialize OV935 and products containing OV935 for the treatment of certain rare
neurological disorders. If the agreement is terminated by us for Takeda’s material breach or bankruptcy or by Takeda for convenience or safety reasons, Takeda’s rights to
the  products  will  cease,  Takeda  will  transition  all  activities  related  to  the  products  to  us,  and  Takeda  will  grant  us  an  exclusive,  royalty-bearing  license  under  certain
patents  and  other  intellectual  property  controlled  by  Takeda  to  commercialize  OV935  and  products  containing  OV935  for  the  treatment  of  certain  rare  neurological
disorders.

Under the Takeda collaboration agreement, in the event of an acquisition of us by certain types of acquirers prior to the final dosing of a patient in the first Phase 3
trial, Takeda would have the right to elect to take over all development and commercialization activities with respect to the products, so long as Takeda at such time has
(or will have) sufficient commercial infrastructure to commercialize the products. Even if Takeda exercises such right to take over all development and commercialization
activities  with  respect  to  the  products,  we  and  Takeda  will  continue  to  share  equally  all  development  and  commercialization  costs  and  expenses  prior  to  launch  of  a
product and all revenues and commercialization costs and expenses after launch, unless otherwise set forth in the agreement.

In connection with the Takeda collaboration agreement and in consideration of certain license rights granted to us by Takeda, we issued 1,781,996 shares of our
Series B-1 convertible preferred stock to Takeda. The shares of Series B-1 preferred stock held by Takeda automatically converted into 1,781,996 shares of our common
stock in May 2017. Under the Takeda collaboration agreement, we are obligated to pay Takeda future payments if and when certain milestones are achieved. Upon the
first patient enrollment in the first Phase 3 trial for the first of the initial disorders we and Takeda are focusing on, we are obligated to issue to Takeda the number of
unregistered shares of our common stock equal to the lesser of (a) 8% of our outstanding capital stock on the issuance date or (b) $50.0 million divided by the applicable
share price, unless certain events occur. In the event such payment would cause Takeda to own over 19.99% of our outstanding capital stock or other events occur, such
payment must be paid in cash. The remaining potential global commercial and regulatory milestone payments equal approximately $35.0 million and can be satisfied in
cash or unregistered shares of our common stock at our election.

2021 Royalty, License and Termination Agreement with Takeda

On March 2, 2021, we entered into a royalty, license and termination agreement, or the Takeda License and Termination Agreement, with Takeda, relating to the
Takeda  collaboration  agreement  described  above.  Under  the  terms  of  the  Takeda  License  and  Termination  Agreement,  upon  closing  of  the  transaction,  the  Takeda
collaboration agreement will be terminated by mutual agreement, and Takeda will secure rights to our 50% global share in OV935 (soticlestat), and an exclusive license
under our relevant intellectual property rights, in exchange for an upfront payment, development and commercial milestone payments, and royalties.  Takeda will

13

 
assume all responsibility for, and costs of, both development and commercialization of soticlestat following closing. At closing, we will receive an upfront payment of
$196.0  million  and  are  eligible  to  receive  up  to  an  additional  $660.0  million  in  development,  regulatory  and  sales  milestones.    In  addition,  if  soticlestat  achieves
regulatory approval, we will receive tiered royalties on net sales of soticlestat at percentages ranging from the low double-digits up to 20%, subject to standard reductions
in certain circumstances.  Royalties are payable on a country-by-country and product-by-product basis during the period beginning on the date of the first commercial sale
of such product in such country and ending on the later to occur of the expiration of patent rights covering the product in such country and a specified anniversary of such
first  commercial  sale.  The  Takeda collaboration  agreement  will  remain  in  effect  until  Takeda’s  cessation  of  commercialization  of  soticlestat.    We  expect  to  close  the
Takeda  License  and  Termination  Agreement  in  the  first  half  of  2021,  subject  to  the  satisfaction  of  customary  closing  conditions,  including  regulatory  review  by  the
appropriate regulatory agencies under the Hart-Scott-Rodino Antitrust Improvements Act of 1976, as amended. The Takeda License and Termination Agreement may be
terminated upon the mutual agreement of the parties, or by either Takeda or the Company, if the closing has not occurred on or before May 14, 2021. 

Northwestern License

In December 2016, we entered into a license agreement with Northwestern, pursuant to which Northwestern granted us an exclusive, worldwide license to patent
rights in certain inventions, or the Northwestern Patent Rights, which relate to a specific compound and related methods of use for such compound, along with certain
Know-How related to the practice of the inventions claimed in the Northwestern Patents.

Under the Northwestern agreement, we were granted exclusive rights to research, develop, manufacture and commercialize products utilizing the Northwestern
Patent Rights for all uses. We have agreed that we will not use the Northwestern Patent Rights to develop any products for the treatment of cancer, but Northwestern may
not grant rights in the technology to others for use in cancer. We also have an option, exercisable during the term of the agreement to an exclusive license under certain
intellectual  property  rights  covering  novel  compounds  with  the  same  or  similar  mechanism  of  action  as  the  primary  compound  that  is  the  subject  of  the  license
agreement.  Northwestern has retained the right, on behalf of itself and other non-profit institutions, to use the Northwestern Patent Rights and practice the inventions
claimed therein for educational and research purposes and to publish information about the inventions covered by the Northwestern Patent Rights.  

Upon entry into the Northwestern agreement, we paid an upfront non-creditable one-time license issuance fee of $75,000, and we are required to pay an annual
license maintenance fee of $20,000, which will be creditable against any royalties payable to Northwestern following first commercial sale of licensed products under the
agreement.  We are responsible for all ongoing costs of filing, prosecuting and maintaining the Northwestern Patents, but we also have the right to control such activities
using our own patent counsel.  In consideration for the rights granted to us under the Northwestern agreement, we are required to pay to Northwestern up to an aggregate
of  $5.3  million  upon  the  achievement  of  certain  development  and  regulatory  milestones  for  the  first  product  covered  by  the  Northwestern  Patents,  and,  upon
commercialization  of  any  such  products,  will  be  required  to  pay  to  Northwestern  a  tiered  royalty  on  net  sales  of  such  products  by  the  Company,  its  affiliates  or
sublicensees,  at  percentages  in  the  low  to  mid-single-digits,  subject  to  standard  reductions  and  offsets.    Our  royalty  obligations  continue  on  a  product-by-product  and
country-by-country basis until the later of the expiration of the last-to-expire valid claim in a licensed patent covering the applicable product in such country and 10 years
following  the  first  commercial  sale  of  such  product  in  such  country.    If  Ovid  sublicenses  a  Northwestern  Patent  Right,  it  will  be  obligated  to  pay  to  Northwestern  a
specified percentage of sublicense revenue received by us, ranging from the high single digits to the low-teens.  

The  Northwestern  agreement  requires  that  we  use  commercially  reasonable  efforts  to  develop  and  commercialize  at  least  one  product  that  is  covered  by  the

Northwestern Patent Rights.  

Unless  earlier  terminated,  the  Northwestern  agreement  will  remain  in  force  until  the  expiration  of  our  payment  obligations  thereunder.    We  have  the  right  to
terminate the agreement for any reason upon prior written notice or for an uncured material breach by Northwestern.  Northwestern may terminate the agreement for our
uncured material breach or insolvency.

Sales and Marketing

Given our stage of development, we have not yet established a commercial organization or distribution capabilities, however, in November 2019 we hired a Chief
Commercial  Officer  to  begin  planning  to  establish  a  commercial  organization.  We  plan  to  build  focused  capabilities  in  the  United  States  and  European  Union  to
commercialize our development programs focused on rare disorders of the brain. In other markets for which commercialization may be less capital efficient for us, we
may selectively pursue strategic collaborations with third parties in order to maximize the commercial potential of our drug candidates.

Manufacturing and Supply

We currently outsource all manufacturing, and we intend to use our collaborators and contract manufacturers for the foreseeable future. However, certain members

of our management have broad experience in manufacturing, which we believe may provide a competitive advantage.

14

 
Competition

We believe Sage Therapeutics, Inc., Marinus Pharmaceuticals, Inc. and Zynerba Pharmaceuticals, Inc. are our most direct competitors with respect to OV101 in
Angelman syndrome and Fragile X syndrome. Biogen Inc. in collaboration with Ionis Pharmaceuticals, Inc., Roche Holding AG, PTC Therapeutics, Inc. and Ultragenyx
Pharmaceutical Inc. in collaboration with GeneTx Biotherapeutics LLC are working on genetic approaches to Angelman syndrome.

We believe Zogenix, Inc., GW Pharmaceuticals plc, Sage Therapeutics, Inc., Marinus Pharmaceuticals, Inc., Zynerba Pharmaceuticals, Inc., Stoke Therapeutics,

Inc. and PTC Therapeutics, Inc. are our most direct competitors with respect to OV935.

Drug development is highly competitive and subject to rapid and significant technological advancements. Our ability to compete will significantly depend upon
our ability to complete necessary clinical trials and regulatory approval processes, and effectively market any drug that we may successfully develop. Our current and
potential future competitors include pharmaceutical and biotechnology companies, academic institutions and government agencies. The primary competitive factors that
will  affect  the  commercial  success  of  any  drug  candidate  for  which  we  may  receive  marketing  approval  include  efficacy,  safety  and  tolerability  profile,  dosing
convenience, price, coverage and reimbursement. Many of our existing or potential competitors have substantially greater financial, technical and human resources than
we do and significantly greater experience in the discovery and development of drug candidates, as well as in obtaining regulatory approvals of those drug candidates in
the United States and in foreign countries.

Our current and potential future competitors also have significantly more experience commercializing drugs that have been approved for marketing. Mergers and

acquisitions in the pharmaceutical and biotechnology industries could result in even more resources being concentrated among a small number of our competitors.

Accordingly, our competitors may be more successful than us in obtaining regulatory approval for therapies and in achieving widespread market acceptance of
their  drugs.  It  is  also  possible  that  the  development  of  a  cure  or  more  effective  treatment  method  for  the  disorders  we  are  targeting  by  a  competitor  could  render  our
current  or  future  drug  candidates  non-competitive  or  obsolete  or  reduce  the  demand  for  our  drug  candidates  before  we  can  recover  our  development  and
commercialization expenses.

Intellectual Property

Our commercial success depends in part on our ability to obtain and maintain proprietary protection for our current and future drug candidates, novel discoveries,
product development technologies and know-how, to operate without infringing on the proprietary rights of others and to prevent others from infringing our proprietary
rights. Our policy is to seek to protect our proprietary position by, among other methods, filing or in-licensing U.S. and foreign patents and patent applications related to
technology, inventions and improvements that are important to the development and implementation of our business. We also rely on trademarks, trade secrets, copyright
protection, know-how, continuing technological innovation and potential in-licensing opportunities to develop and maintain our proprietary position. For example, the
proprietary map of disease-relevant biological pathways underlying orphan disorders of the brain that we developed would not be appropriate for patent protection and, as
a result, we rely on trade secrets to protect this aspect of our business.

While we seek broad coverage under our existing patent applications, there is always a risk that an alteration to the product or process may provide sufficient basis
for a competitor to avoid infringement claims. In addition, the coverage claimed in a patent application can be significantly reduced before a patent is issued and courts
can  reinterpret  patent  scope  after  issuance.  Moreover,  many  jurisdictions  including  the  United  States  permit  third  parties  to  challenge  issued  patents  in  administrative
proceedings, which may result in further narrowing or even cancellation of patent claims. Moreover, we cannot provide any assurance that any patents will be issued from
our pending or any future applications or that any potentially issued patents will adequately protect our intellectual property.

We  currently  own  issued  U.S.  patents  directed  to  treatment  of  Angelman  syndrome  and  Fragile  X  syndrome  with  OV101  that  expire  in  2035,  excluding  any
regulatory extensions. We also have exclusively licensed a portfolio of issued U.S. and international patents from Lundbeck directed to polymorphic forms of OV101 and
their preparation, and these patents expire on dates ranging from 2025 to 2028. In addition, we have exclusively licensed from Lundbeck an issued U.S. patent that will
expire in 2036 and a pending application directed to an OV101 manufacturing processes that, if issued, would have a statutory expiration in 2036. We have also filed, and
own, multiple patent families directed to methods of treatment and formulations with OV101. Additional issued patents and pending applications are directed to methods
of treating neurodegenerative diseases and developmental disorders. We are seeking or will seek patent protection for these inventions in numerous countries and regions
including, among others, Europe, Australia, Canada, Mexico, Israel, Japan, China, and Korea.

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We  licensed  from  Takeda  a  portfolio  of  U.S.  and  international  patents  and  applications  directed  to  the  OV935  composition  of  matter,  and  these  patents  and

applications expire in 2032, excluding any regulatory extensions.

Individual patents extend for varying periods depending on the date of filing of the patent application or the date of patent issuance and the legal term of patents in
the  countries  in  which  they  are  obtained.  Generally,  utility  patents  issued  for  applications  filed  in  the  United  States  are  granted  a  term  of  20  years  from  the  earliest
effective filing date of a non-provisional patent application. In addition, in certain instances, a patent term can be extended to recapture a portion of the U.S. Patent and
Trademark Office, or the USPTO, delay in issuing the patent as well as a portion of the term effectively lost as a result of the FDA regulatory review period. However, as
to  the  FDA  component,  the  restoration  period  cannot  be  longer  than  five  years  and  the  total  patent  term  including  the  restoration  period  must  not  exceed  14  years
following  FDA  approval.  The  duration  of  foreign  patents  varies  in  accordance  with  provisions  of  applicable  local  law,  but  typically  is  also  20  years  from  the  earliest
effective filing date. The actual protection afforded by a patent may vary on a product-by-product basis, from country to country and can depend upon many factors,
including the type of patent, the scope of its coverage, the availability of regulatory-related extensions, the availability of legal remedies in a particular country and the
validity and enforceability of the patent.

Furthermore, we rely upon trade secrets and know-how and continuing technological innovation to develop and maintain our competitive position. We seek to
protect our proprietary information, in part, using confidentiality agreements with our employees and consultants and any potential commercial partners and collaborators
and invention assignment agreements with our employees. We also have or intend to implement confidentiality agreements or invention assignment agreements with our
selected  consultants  and  any  potential  commercial  partners.  These  agreements  are  designed  to  protect  our  proprietary  information  and,  in  the  case  of  the  invention
assignment agreements, to grant us ownership of technologies that are developed through a relationship with a third party. These agreements may be breached, and we
may not have adequate remedies for any breach. In addition, our trade secrets may otherwise become known or be independently discovered by competitors. To the extent
that our commercial partners, collaborators, employees and consultants use intellectual property owned by others in their work for us, disputes may arise as to the rights in
related or resulting know-how and inventions.

Our commercial success will also depend in part on not infringing upon the proprietary rights of third parties. It is uncertain whether the issuance of any third-
party patent would require us to alter our development or commercial strategies, or our drugs or processes, obtain licenses or cease certain activities. Our breach of any
license agreements or failure to obtain a license to proprietary rights that we may require to develop or commercialize our future drugs may have an adverse impact on us.
Since  patent  applications  in  the  United  States  and  certain  other  jurisdictions  are  maintained  in  secrecy  for  18  months  or  potentially  longer,  and  since  publication  of
discoveries  in  the  scientific  or  patent  literature  often  lags  behind  actual  discoveries,  we  cannot  be  certain  of  the  priority  of  inventions  covered  by  pending  patent
applications. Moreover, we may have to participate in Interference, Derivation, Reexam, Post-Grant Review, Inter Partes Review, or Opposition proceedings brought by
third parties or declared by the USPTO.

Government Regulation

The  FDA  and  regulatory  authorities  in  state  and  local  jurisdictions  and  in  other  countries  impose  substantial  and  burdensome  requirements  upon  companies
involved in the clinical development, manufacture, marketing and distribution of drugs, such as those we are developing. These agencies and other federal, state and local
entities  regulate,  among  other  things,  the  research  and  development,  testing,  manufacture,  quality  control,  safety,  effectiveness,  labeling,  storage,  record  keeping,
approval, advertising and promotion, distribution, post-approval monitoring and reporting, sampling and export and import of drugs and drug candidates.

U.S. Government Regulation

In  the  United  States,  the  FDA  regulates  drugs  under  the  Federal  Food,  Drug,  and  Cosmetic  Act,  or  FDCA,  and  its  implementing  regulations.  The  process  of
obtaining  regulatory  approvals  and  the  subsequent  compliance  with  applicable  federal,  state,  local  and  foreign  statutes  and  regulations  requires  the  expenditure  of
substantial time and financial resources. Failure to comply with the applicable U.S. requirements at any time during the product development process, approval process or
after approval, may subject an applicant to a variety of administrative or judicial sanctions, such as the FDA’s refusal to approve pending New Drug Applications (NDAs)
or Biologics License Applications (BLAs), withdrawal of an approval, imposition of a clinical hold, issuance of warning letters, product recalls, product seizures, total or
partial suspension of production or distribution, injunctions, fines, refusals of government contracts, restitution, disgorgement or civil or criminal penalties.

The process required by the FDA before a drug product may be marketed in the United States generally involves the following:

•

•

•

completion  of  preclinical  laboratory  tests,  animal  studies  and  formulation  studies  in  compliance  with  the  FDA’s  good  laboratory  practice,  or  GLP,
regulations.

submission to the FDA of an IND which must become effective before human clinical trials may begin.

approval by an independent institutional review board, or IRB, at each clinical site before each trial may be initiated.

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•

•

•

•

•

performance of adequate and well controlled human clinical trials in accordance with good clinical practice, or GCP, requirements to establish the safety
and efficacy of the proposed drug product for each indication.

submission to the FDA of an NDA or BLA.

satisfactory completion of an FDA advisory committee review, if applicable.

satisfactory completion of an FDA inspection of the manufacturing facility or facilities at which the product is produced to assess compliance with current
good manufacturing practice, or cGMP, requirements and to assure that the facilities, methods and controls are adequate to preserve the drug’s identity,
strength, quality and purity; and

FDA review and approval of the NDA or BLA.

Preclinical Studies

Preclinical studies include laboratory evaluation of product chemistry, toxicity and formulation, as well as animal studies to assess potential safety and efficacy.
An  IND  sponsor  must  submit  the  results  of  the  preclinical  tests,  together  with  manufacturing  information,  analytical  data  and  any  available  clinical  data  or  literature,
among other things, to the FDA as part of an IND. Some preclinical testing may continue even after the IND is submitted. An IND automatically becomes effective 30
days after receipt by the FDA, unless before that time the FDA raises concerns or questions related to one or more proposed clinical trials and places the clinical trial on a
clinical hold. In such a case, the IND sponsor and the FDA must resolve any outstanding concerns before the clinical trial can begin. As a result, submission of an IND
may not result in the FDA allowing clinical trials to commence.

Clinical Trials

Clinical trials involve the administration of the investigational new drug to human patients under the supervision of qualified investigators in accordance with
GCP requirements, which include the requirement that all research patients provide their informed consent in writing for their participation in any clinical trial. Clinical
trials are conducted under protocols detailing, among other things, the objectives of the trial, the parameters to be used in monitoring safety and the effectiveness criteria
to be evaluated. A protocol for each clinical trial and any subsequent protocol amendments must be submitted to the FDA as part of the IND. In addition, an IRB at each
institution  participating  in  the  clinical  trial  must  review  and  approve  the  plan  for  any  clinical  trial  before  it  commences  at  that  institution.  Information  about  certain
clinical trials must be submitted within specific timeframes to the National Institutes of Health, or NIH, for public dissemination on their www.clinicaltrials.gov website.

Human clinical trials are typically conducted in three sequential phases, which may overlap or be combined:

•

•

•

Phase 1 clinical trial: The drug is initially introduced into healthy human volunteers or patients with the target disease or condition and tested for safety,
dosage tolerance, absorption, metabolism, distribution, excretion and, if possible, to gain an early indication of its effectiveness.

Phase 2 clinical trial: The drug is administered to a limited patient population to identify possible adverse effects and safety risks, to preliminarily evaluate
the efficacy of the product for specific targeted diseases and to determine dosage tolerance and optimal dosage.

Phase  3  clinical  trial:  The  drug  is  administered  to  an  expanded  patient  population,  generally  at  geographically  dispersed  clinical  trial  sites,  in  well
controlled clinical trials to generate enough data to statistically evaluate the efficacy and safety of the product for approval, to establish the overall risk-
benefit profile of the product, and to provide adequate information for the labeling of the product.

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Progress reports detailing the results of the clinical trials must be submitted at least annually to the FDA and more frequently if serious adverse events occur. Each
of Phase 1, Phase 2 and Phase 3 clinical trials may not be completed successfully within any specified period, or at all. Furthermore, the FDA or the sponsor may suspend
or terminate a clinical trial at any time on various grounds, including a finding that the research patients are being exposed to an unacceptable health risk. Similarly, an
IRB can suspend or terminate approval of a clinical trial at its institution if the clinical trial is not being conducted in accordance with the IRB’s requirements or if the
drug has been associated with unexpected serious harm to patients.

Marketing Approval

Assuming successful completion of the required clinical testing, the results of the preclinical studies and clinical trials, together with detailed information relating
to the product’s chemistry, manufacture, controls and proposed labeling, among other things, are submitted to the FDA as part of an NDA or BLA requesting approval to
market the product for one or more indications. In most cases, the submission of an NDA or BLA is subject to a substantial application user fee. Under the Prescription
Drug User Fee Act, or PDUFA, guidelines that are currently in effect, the FDA has a goal of ten months from the date of “filing” of a standard NDA for a new molecular
entity to review and act on the submission. This review typically takes twelve months from the date the NDA is submitted to FDA because the FDA has approximately
two months to make a “filing” decision.

The FDA conducts a preliminary review of all NDAs within the first 60 days after submission, before accepting them for filing, to determine whether they are
sufficiently complete to permit substantive review. The FDA may request additional information rather than accept an NDA for filing. In this event, the application must
be resubmitted with the additional information. The resubmitted application is also subject to review before the FDA accepts it for filing. Once the submission is accepted
for filing, the FDA begins an in-depth substantive review. The FDA reviews an NDA to determine, among other things, whether the drug is safe and effective and whether
the facility in which it is manufactured, processed, packaged or held meets standards designed to assure the product’s continued safety, quality and purity.

In addition, under the Pediatric Research Equity Act of 2003, or PREA, as amended and reauthorized, certain must contain data that are adequate to assess the
safety  and  effectiveness  of  the  drug  for  the  claimed  indications  in  all  relevant  pediatric  subpopulations,  and  to  support  dosing  and  administration  for  each  pediatric
subpopulation for which the product is safe and effective. The FDA may, on its own initiative or at the request of the applicant, grant deferrals for submission of some or
all pediatric data until after approval of the product for use in adults, or full or partial waivers from the pediatric data requirements.

The FDA also may require submission of a risk evaluation and mitigation strategy, or REMS, plan to ensure that the benefits of the drug outweigh its risks. The
REMS plan could include medication guides, physician communication plans, assessment plans, or elements to assure safe use, such as restricted distribution methods,
patient registries, or other risk minimization tools.  

The FDA may refer an application for a novel drug to an advisory committee. An advisory committee is a panel of independent experts, including clinicians and
other scientific experts, that reviews, evaluates and provides a recommendation as to whether the application should be approved and under what conditions. The FDA is
not bound by the recommendations of an advisory committee, but it considers such recommendations carefully when making decisions.

Before  approving  an  NDA  or  BLA,  the  FDA  typically  will  inspect  the  facility  or  facilities  where  the  product  is  manufactured.  The  FDA  will  not  approve  an
application unless it determines that the manufacturing processes and facilities are in compliance with cGMP requirements and adequate to assure consistent production
of the product within required specifications. Additionally, before approving an NDA or BLA, the FDA may inspect one or more clinical trial sites to assure compliance
with GCP requirements.

After  evaluating  the  application  and  all  related  information,  including  the  advisory  committee  recommendation,  if  any,  and  inspection  reports  regarding  the
manufacturing facilities and clinical trial sites, the FDA may issue an approval letter, or, in some cases, a complete response letter. A complete response letter generally
contains a statement of specific conditions that must be met in order to secure final approval of the NDA or BLA and may require additional clinical or preclinical testing
in order for FDA to reconsider the application. Even with submission of this additional information, the FDA ultimately may decide that the application does not satisfy
the regulatory criteria for approval. If and when those conditions have been met to the FDA’s satisfaction, the FDA will typically issue an approval letter. An approval
letter authorizes commercial marketing of the drug with specific prescribing information for specific indications.

Even if the FDA approves a product, it may limit the approved indications for use of the product, require that particular contraindications, warnings or precautions
be  included  in  the  product  labeling,  require  that  post-approval  studies,  including  Phase  4  clinical  trials,  be  conducted  to  further  assess  a  drug’s  safety  after  approval,
require testing and surveillance programs to monitor the product after commercialization, or impose other conditions, including distribution and use restrictions or other
risk management mechanisms under a REMS, which can materially affect the potential market and profitability of the product. The FDA may prevent or limit further
marketing of a product based on the results of post-marketing studies or surveillance programs. After approval, some types of changes to the approved product, such as
adding new indications, manufacturing changes, and additional labeling claims, are subject to further testing requirements and FDA review and approval.

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Orphan Drug Act

Under the Orphan Drug Act of 1983, the FDA may grant orphan designation to a drug or biologic intended to treat a rare disease or condition, which is generally a
disease or condition that affects fewer than 200,000 individuals in the United States, or more than 200,000 individuals in the United States and for which there is no
reasonable expectation that the cost of developing and making available in the United States a drug for this type of disease or condition will be recovered from sales in the
United States for that drug. Orphan drug designation must be requested before submitting an NDA or BLA. After the FDA grants orphan drug designation, the name of
the sponsor, identity of the drug or biologic and its potential orphan use are disclosed publicly by the FDA. The orphan drug designation does not shorten the duration of
the regulatory review or approval process, but does provide certain advantages, such as a waiver of PDUFA fees, enhanced access to FDA staff and potential waiver of
pediatric research requirements.

If a product that has orphan drug designation subsequently receives the first FDA approval for the disease for which it has such designation, the product is entitled
to orphan product exclusivity, which means that the FDA may not approve any other applications, including a full NDA or BLA, or an abbreviated NDA (ANDA) or
Biosimilar  application,  to  market  a  drug  or  biologic  with  the  same  active  moiety  for  the  same  indication  for  seven  years,  except  in  limited  circumstances,  such  as  a
showing of clinical superiority to the product with orphan drug exclusivity. Orphan drug exclusivity does not prevent FDA from approving a different drug or biologic for
the same disease or condition, or the same drug or biologic for a different disease or condition. Among the other benefits of orphan drug designation are tax credits for
certain research and a waiver of the application user fee. A designated orphan drug may not receive orphan drug exclusivity if it is approved for a use that is broader than
the  indication  for  which  it  received  orphan  designation.  In  addition,  exclusive  marketing  rights  in  the  United  States  may  be  lost  if  the  FDA  later  determines  that  the
request for designation was materially defective or if the manufacturer is unable to assure sufficient quantities of the product to meet the needs of patients with the rare
disease or condition.

Fast Track Designation

The  FDA  is  required  to  facilitate  the  development  and  expedite  the  review  of  pharmaceutical  products  that  are  intended  for  the  treatment  of  a  serious  or  life-
threatening condition for which there is no effective treatment, and which demonstrate the potential to address unmet medical needs for the condition. Under the fast-track
program, the sponsor of a new drug candidate may request the FDA to designate the product for a specific indication as a fast-track product concurrent with or after the
filing  of  the  IND  for  the  product  candidate.  The  FDA  must  determine  if  the  product  candidate  qualifies  for  fast-track  designation  within  60  days  after  receipt  of  the
sponsor’s request.

In  addition  to  other  benefits,  such  as  the  ability  to  have  more  frequent  interactions  with  the  FDA,  the  agency  may  initiate  review  of  sections  of  a  fast-track
product’s NDA or BLA before the application is complete. This rolling review is available if the applicant provides and the FDA approves a schedule for the submission
of the remaining information and the applicant pays applicable user fees. However, the FDA’s PDUFA review period for a fast-track application does not begin until the
last section of the application is submitted. In addition, the fast-track designation may be withdrawn by the FDA if the agency believes that the designation is no longer
supported by data emerging in the clinical trial process.

Post-Approval Requirements

Drugs  manufactured  or  distributed  pursuant  to  FDA  approvals  are  subject  to  pervasive  and  continuing  regulation  by  the  FDA,  including,  among  other  things,
requirements relating to recordkeeping, periodic reporting, product sampling and distribution, advertising and promotion and reporting of adverse experiences with the
product. After approval, most changes to the approved product, such as adding new indications or other labeling claims are subject to prior FDA review and approval.
There  also  are  continuing,  annual  user  fee  requirements  for  any  marketed  products  and  the  establishments  at  which  such  products  are  manufactured,  as  well  as  new
application fees for supplemental applications with clinical data.

The FDA may impose a number of post-approval requirements as a condition of approval of a marketing authorization. For example, the FDA may require post-

marketing testing, including Phase 4 clinical trials, and surveillance to further assess and monitor the product’s safety and effectiveness after commercialization.

In addition, drug manufacturers and other entities involved in the manufacture and distribution of approved drugs are required to register their establishments with
the FDA and state agencies and are subject to periodic unannounced inspections by the FDA and these state agencies for compliance with cGMP requirements. Changes
to  the  manufacturing  process  are  strictly  regulated  and  often  require  prior  FDA  approval  before  being  implemented.  FDA  regulations  also  require  investigation  and
correction of any deviations from cGMP requirements and impose reporting and documentation requirements upon the sponsor and any third-party manufacturers that the
sponsor may decide to use. Accordingly, manufacturers must continue to expend time, money, and effort in the area of production and quality control to maintain cGMP
compliance.

Once  an  approval  is  granted,  the  FDA  may  withdraw  the  approval  if  compliance  with  regulatory  requirements  and  standards  is  not  maintained  or  if  problems
occur  after  the  product  reaches  the  market.  Later  discovery  of  previously  unknown  problems  with  a  product,  including  adverse  events  of  unanticipated  severity  or
frequency, or with manufacturing processes, or failure to comply with regulatory requirements, may result in mandatory revisions to the approved labeling to add new
safety information; imposition of

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post-market studies or clinical trials to assess new safety risks; or imposition of distribution or other restrictions under a REMS program. Other potential consequences
include, among other things:

•

•

•

•

•

restrictions on the marketing or manufacturing of the product, complete withdrawal of the product from the market or product recalls.

fines, warning letters or holds on post-approval clinical trials;

refusal of the FDA to approve related pending applications or supplements to approved applications, or suspension or revocation of product approvals;

product seizure or detention, or refusal to permit the import or export of products; or

injunctions or the imposition of civil or criminal penalties.

The  FDA  strictly  regulates  marketing,  labeling,  advertising  and  promotion  of  products  that  are  placed  on  the  market.  Drugs  may  be  promoted  only  for  the
approved indications and in accordance with the provisions of the approved label. The FDA and other agencies actively enforce the laws and regulations prohibiting the
promotion of off-label uses, and a company that is found to have improperly promoted off-label uses may be subject to significant liability.

Coverage and Reimbursement

Sales of our drug candidates, if approved, will depend, in part, on the extent to which such products will be covered by third-party payors, such as government
health  care  programs,  commercial  insurance  and  managed  healthcare  organizations.  These  third-party  payors  are  increasingly  limiting  coverage  or  reducing
reimbursements  for  medical  products  and  services.  In  addition,  the  U.S.  government,  state  legislatures,  and  foreign  governments  have  continued  implementing  cost-
containment programs, including price controls, restrictions on reimbursement and requirements for substitution of generic products. Third-party payors decide which
therapies they will pay for and establish reimbursement levels. Third-party payors often rely upon Medicare coverage policy and payment limitations in setting their own
coverage and reimbursement policies. Further, no uniform policy for coverage and reimbursement exists in the United States. Therefore, decisions regarding the extent of
coverage and amount of reimbursement to be provided for any drug candidates that we develop will be made on a payor-by-payor basis. Each payor determines whether
or not it will provide coverage for a therapy, what amount it will pay the manufacturer for the therapy, and on what tier of its formulary it will be placed. The position on a
payor’s list of covered drugs, or formulary, generally determines the co-payment that a patient will need to make to obtain the therapy and can strongly influence the
adoption of such therapy by patients and physicians. Adoption of price controls and cost-containment measures, and adoption of more restrictive policies in jurisdictions
with existing controls and measures, could further limit our net revenue and results. Decreases in third-party reimbursement for our drug candidates or a decision by a
third-party payor to not cover our drug candidates could reduce physician usage of our drug candidates, once approved, and have a material adverse effect on our sales,
results of operations and financial condition. Coverage policies and third-party payor reimbursement rates may change at any time. Therefore, even if favorable coverage
and reimbursement status is attained, less favorable coverage policies and reimbursement rates may be implemented in the future.

Other Healthcare Laws

Because of our current and future arrangements with healthcare professionals, principal investigators, consultants, customers and third-party payors, we will also
be subject to healthcare regulation and enforcement by the federal government and the states and foreign governments in which we will conduct our business, including
our clinical research, proposed sales, marketing and educational programs. Failure to comply with these laws, where applicable, can result in the imposition of significant
civil, criminal, and administrative penalties.

The U.S. laws that may affect our ability to operate, among others, include: the federal Health Insurance Portability and Accountability Act of 1996, or HIPAA, as
amended  by  the  Health  Information  Technology  for  Economic  and  Clinical  Health  Act,  which  governs  the  conduct  of  certain  electronic  healthcare  transactions  and
protects the security and privacy of protected health information; certain state laws governing the privacy and security of health information in certain circumstances,
some  of  which  are  more  stringent  than  HIPAA  and  many  of  which  differ  from  each  other  in  significant  ways  and  may  not  have  the  same  effect,  thus  complicating
compliance  efforts;  the  federal  Anti-Kickback  Statute,  which  prohibits,  among  other  things,  individuals  or  entities  from  knowingly  and  willfully  soliciting,  receiving,
offering or paying remuneration, directly or indirectly, in exchange for or to induce either the referral of an individual for, or the purchase, order or recommendation of,
any good or service for which payment may be made under federal healthcare programs such as the Medicare and Medicaid programs; federal false claims laws and civil
monetary  penalty  laws,  which  prohibit,  among  other  things,  individuals  or  entities  from  knowingly  presenting,  or  causing  to  be  presented,  claims  for  payment  from
Medicare,  Medicaid,  or  other  third-party  payors  that  are  false  or  fraudulent;  federal  criminal  laws  that  prohibit  executing  a  scheme  to  defraud  any  healthcare  benefit
program  or  making  false  statements  relating  to  healthcare  matters;  the  Physician  Payments  Sunshine  Act,  which  requires  certain  manufacturers  of  drugs,  devices,
biologics, and medical supplies to report annually to the U.S. Department of Health and Human Services information related to payments and other transfers of value to
physicians (defined to include doctors, dentists, optometrists, podiatrists and chiropractors) and teaching hospitals, and ownership and investment

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interests held by physicians and their immediate family members. Beginning in 2022, applicable manufacturers also will be required to report such information regarding
their  payments  and  other  transfers  of  value  to  physician  assistants,  nurse  practitioners, clinical  nurse  specialists,  anesthesiologist  assistants,  certified  registered  nurse
anesthetists and certified nurse midwives during the previous year.

In addition, many states have similar laws and regulations, such as anti-kickback and false claims laws that may be broader in scope and may apply regardless of
payor, in addition to items and services reimbursed under Medicaid and other state programs. Additionally, to the extent that our product is sold in a foreign country, we
may be subject to similar foreign laws.

Healthcare Reform

Current  and  future  legislative  proposals  to  further  reform  healthcare  or  reduce  healthcare  costs  may  result  in  lower  reimbursement  for  our  products.  The  cost
containment measures that payors and providers are instituting and the effect of any healthcare reform initiative implemented in the future could significantly reduce our
revenues from the sale of our products.

For example, implementation of the Patient Protection and Affordable Care Act, as amended by the Health Care and Education Reconciliation Act, collectively
the  Affordable  Care  Act,  or  the  PPACA,  has  substantially  changed  healthcare  financing  and  delivery  by  both  governmental  and  private  insurers,  and  significantly
impacted  the  pharmaceutical  industry.  The  PPACA,  among  other  things,  established  an  annual,  nondeductible  fee  on  any  entity  that  manufactures  or  imports  certain
specified  branded  prescription  drugs  and  biologic  agents,  revised  the  methodology  by  which  rebates  owed  by  manufacturers  to  the  state  and  federal  government  for
covered  outpatient  drugs  under  the  Medicaid  Drug  Rebate  Program  are  calculated,  increased  the  minimum  Medicaid  rebates  owed  by  most  manufacturers  under  the
Medicaid  Drug  Rebate  Program,  extended  the  Medicaid  Drug  Rebate  program  to  utilization  of  prescriptions  of  individuals  enrolled  in  Medicaid  managed  care
organizations, provided incentives to programs that increase the federal government’s comparative effectiveness research and created a licensure frame work for follow-
on  biologic  products.  Since  its  enactment  there  have  been  executive,  judicial  and  Congressional  challenges  to  certain  aspects  of  the  PPACA.  For  example,  President
Trump has signed several Executive Orders and other directives designed to delay the implementation of certain provisions of the PPACA or otherwise circumvent some
of the requirements for health insurance mandated by the PPACA. Concurrently, Congress considered legislation to repeal or repeal and replace all or part of the PPACA.
While Congress has not passed comprehensive repeal legislation, several bills affecting the implementation of certain taxes under the PPACA have been signed into law.
The Tax Cuts and Jobs Act of 2017 includes a provision repealing, effective January 1, 2019, the tax-based shared responsibility payment imposed by the PPACA on
certain individuals who fail to maintain qualifying health coverage for all or part of a year that is commonly referred to as the “individual mandate”. Additionally, the
2020 federal spending package permanently eliminated, effective January 1, 2020, the PPACA-mandated “Cadillac” tax on high-cost employer-sponsored health coverage
and medical device tax and, effective January 1, 2021, also eliminated the health insurer tax. Further, the Bipartisan Budget Act of 2018, or the BBA, among other things,
amends the PPACA, effective January 1, 2019, to increase from 50 percent to 70 percent the point-of-sale discount that is owed by pharmaceutical manufacturers who
participate in Medicare Part D and to close the coverage gap in most Medicare drug plans, commonly referred to as the “donut hole.” Moreover, on December 14, 2018, a
Texas U.S. District Court Judge ruled that the PPACA is unconstitutional in its entirety because the “individual mandate” was repealed by Congress as part of the Tax Act.
Additionally, on December 18, 2019, the U.S. Court of Appeals for the 5th Circuit upheld the District Court ruling that the individual mandate was unconstitutional and
remanded  the  case  back  to  the  District  Court  to  determine  whether  the  remaining  provisions  of  the  PPACA  are  invalid  as  well.  The  U.S.  Supreme  Court  is  currently
reviewing this case, but it is unknown when a decision will be reached. Although the Supreme Court has not yet ruled on the constitutionality of the PPACA, on January
28, 2021, President Biden issued an executive order to initiate a special enrollment period from February 15, 2021 through May 15, 2021 for purposes of obtaining health
insurance coverage through the PPACA marketplace. The executive order also instructs certain governmental agencies to review and reconsider their existing policies and
rules  that  limit  access  to  healthcare,  including  among  others,  reexamining  Medicaid  demonstration  projects  and  waiver  programs  that  include  work  requirements,  and
policies that create barriers to obtaining access to health insurance coverage through Medicaid or the PPACA. It is unclear how the Supreme Court ruling, other such
litigation, and the healthcare reform measures of the Biden administration will impact the PPACA.

In addition, other legislative changes have been proposed and adopted since the PPACA was enacted. In August 2011, then President Obama signed into law the
Budget  Control  Act  of  2011,  which,  among  other  things,  created  the  Joint  Select  Committee  on  Deficit  Reduction  to  recommend  to  Congress  proposals  for  spending
reductions. The Joint Select Committee did not achieve a targeted deficit reduction of at least $1.2 trillion for the years 2013 through 2021, triggering the legislation’s
automatic reduction to several government programs. This includes reductions to Medicare payments to providers of 2% per fiscal year, which went into effect in April
2013 and, due to subsequent legislative amendments, including the BBA, will remain in effect through 2030 unless additional Congressional action is taken. However,
COVID-19 relief support legislation suspended the 2% Medicare sequester from May 1, 2020 through March 31, 2021. Additionally,  in  January  2013,  then  President
Obama signed into law the American Taxpayer Relief Act of 2012, which, among other things, reduced Medicare payments to several providers and increased the statute
of limitations period for the government to recover overpayments to providers from three to five years. Further, there has been heightened governmental scrutiny over the
manner  in  which  manufacturers  set  prices  for  their  marketed  products.  For  example,  there  have  been  presidential  executive  orders  and  several  recent  Congressional
inquiries and proposed and enacted federal and state legislation designed to, among other things, bring more transparency to drug pricing, review the relationship between
pricing and

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manufacturer patient programs, and reform government program reimbursement methodologies for drug products.  It  is  unclear  whether  the  Biden  administration  will
work to reverse these measures or pursue similar policy initiatives.  

We  expect  that  additional  federal  and  state,  as  well  as  foreign,  healthcare  reform  measures  will  be  adopted  in  the  future,  particularly  in  light  of  the  new
presidential  administration,  any  of  which  could  result  in  reduced  demand  for  our  products  or  additional  pricing  pressure.  Further,  it  is  possible  that  additional
governmental action is taken in response to the COVID-19 pandemic.

Employees and Human Capital Resources

As of December 31, 2020, we had 67 full-time employees, 40 of whom were primarily engaged in research and development activities and 16 of whom had an

MD or PhD degree.

Our  human  capital  resources  objectives  include,  as  applicable,  identifying,  recruiting,  retaining,  incentivizing  and  integrating  our  existing  and  additional
employees. The principal purposes of our equity incentive plans are to attract, retain and motivate selected employees, consultants and directors through the granting of
equity-based  compensation  awards  and  cash-based  compensation  awards,  in  order  to  increase  stockholder  value  and  the  success  of  our  company  by  motivating  such
individuals to perform to the best of their abilities and achieve our objectives.

Facilities

We  lease  the  space  for  our  principal  executive  offices,  which  are  located  at  1460  Broadway,  New  York,  New  York,  on  a  monthly  basis.  We  believe  that  our

facilities are adequate to meet our current needs.

Corporate and Other Information

We were incorporated in Delaware in April 2014. Our principal executive offices are located at 1460 Broadway, Suite 15021 New York, New York 10036 and our
telephone number is (646) 661-7661. Our corporate website address is www.ovidrx.com. Information contained on or accessible through our website is not a part of this
Annual Report, and the inclusion of our website address in this Annual Report is an inactive textual reference only.

We file electronically with the Securities and Exchange Commission, or the SEC, our annual reports on Form 10-K, Annual reports on Form 10-Q, current reports
on  Form  8-K,  and  amendments  to  those  reports  filed  or  furnished  pursuant  to  Section  13(a)  or  15(d)  of  the  Exchange  Act.  We  make  available  on  our  website  at
www.ovidrx.com under “Investors,” free of charge, copies of these reports as soon as reasonably practicable after filing or furnishing these reports with the SEC.

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Item 1A. Risk Factors

An investment in our securities involves a high degree of risk. You should carefully consider the following information about these risks, together with the other
information appearing elsewhere in this Annual Report on Form 10-K, including our audited condensed financial statements and related notes hereto, before deciding to
invest in our common stock. The occurrence of any of the following risks could have a material adverse effect on our business, financial condition, results of operations
and future growth prospects or cause our actual results to differ materially from those contained in forward-looking statements we have made in this report and those we
may make from time to time. In these circumstances, the market price of our common stock could decline and you may lose all or part of your investment. We cannot
assure you that any of the events discussed below will not occur. In addition, such risks may be amplified by the COVID-19 pandemic and its potential impact on Ovid’s
business and the global economy.

Risks Related to Our Financial Position and Need for Additional Capital

We have incurred significant operating losses since inception and expect to continue to incur substantial operating losses for the foreseeable future. These factors
raise substantial doubt about our ability to continue as a going concern if we are unsuccessful raising additional capital.

Since  inception  in  April  2014,  we  have  incurred  significant  operating  losses.  Our  net  loss  was  $81.0  million  for  the  year  ended  December  31,  2020.  As  of
December  31,  2020,  we  had  an  accumulated  deficit  of  $294.2  million.  We  expect  to  continue  to  incur  significant  expenses  and  increasing  operating  losses  for  the
foreseeable future. Since inception, we have devoted substantially all of our efforts to research and preclinical and clinical development of our drug candidates, as well as
hiring  employees  and  building  our  infrastructure.  It  could  be  several  years,  if  ever,  before  we  have  a  commercialized  drug.  The  net  losses  we  incur  may  fluctuate
significantly from quarter to quarter and year to year. We anticipate that our expenses will increase substantially if, and as, we:

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continue the ongoing and planned preclinical and clinical development of our drug candidates;

continue to build a portfolio of drug candidates through the acquisition or in-license of drugs, drug candidates or technologies;

initiate preclinical studies and clinical trials for any additional drug candidates that we may pursue in the future;

experience further delays in our preclinical studies and clinical trials due to the ongoing COVID-19 pandemic;

seek marketing approvals for our current and future drug candidates that successfully complete clinical trials;

establish a sales, marketing and distribution infrastructure to commercialize any drug candidate for which we may obtain marketing approval;

develop, maintain, expand and protect our intellectual property portfolio;

implement operational, financial and management systems; and

attract, hire and retain additional administrative, clinical, regulatory and scientific personnel.

Management  has  identified  certain  conditions  or  events,  which,  considered  in  the  aggregate,  raise  substantial  doubt  about  our  ability  to  continue  as  a  going
concern, including the risk that we will be unable to raise adequate additional capital to fund our operations through at least the 12 months following the filing date of the
this annual report on Form 10-K. Substantial doubt about our ability to continue as a going concern may create negative reactions to the price of our common stock. If we
are unable to raise capital, we may be required to delay, reduce the scope of or eliminate research and development programs, or obtain funds through arrangements with
collaborators or others that may require us to relinquish rights to certain drug candidates that we might otherwise seek to develop or commercialize independently. In
addition, if we are unable to continue as a going concern, we may have to liquidate our assets and may receive less than the value at which those assets are carried on our
financial statements, and it is likely that investors will lose all or a part of their investment. Further, the perception that we may be unable to continue as a going concern
may impede our ability to pursue strategic opportunities or operate our business due to concerns regarding our ability to discharge our contractual obligations.

Even  if  we  do  achieve  profitability,  we  may  not  be  able  to  sustain  or  increase  profitability  on  a  quarterly  or  annual  basis.  Our  failure  to  become  and  remain
profitable would decrease the value of our company and could impair our ability to raise capital, maintain our research and development efforts, expand our business or
continue our operations.

We have never generated any revenue from drug sales. Our operating history may make it difficult to evaluate the success of our business to date and to assess our
future viability.

Our operations have consumed substantial amounts of cash since our inception in April 2014, primarily due to organizing and staffing our company, business
planning,  raising  capital,  acquiring  assets  and  undertaking  the  development  of  OV101  and  OV935.  We  have  not  yet  demonstrated  the  ability  to,  obtain  marketing
approvals, manufacture a commercial-scale drug or conduct sales and

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marketing activities necessary for successful commercialization. Consequently, any predictions about our future success or viability may not be as accurate as they could
be if we had more experience developing drug candidates.

Our ability to generate revenue from drug sales and achieve profitability depends on our ability, alone or with any current or future collaborative partners, to
successfully complete the development of, and obtain the regulatory approvals necessary to commercialize, our current and future drug candidates. We do not anticipate
generating revenue from drug sales for the next several years, if ever. Our ability to generate revenue from drug sales depends heavily on our, or any current or future
collaborators’, success in the following areas, including but not limited to:

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timely and successfully completing preclinical and clinical development of our current and future drug candidates;

obtaining regulatory approvals for our current and future drug candidates for which we successfully complete clinical trials;

launching  and  commercializing  any  drug  candidates  for  which  we  obtain  regulatory  approval  by  establishing  a  sales  force,  marketing  and  distribution
infrastructure or, alternatively, collaborating with a commercialization partner;

qualifying  for  coverage  and  adequate  reimbursement  by  government  and  third-party  payors  for  any  drug  candidates  for  which  we  obtain  regulatory
approval, both in the United States and internationally;

developing, validating and maintaining a commercially viable, sustainable, scalable, reproducible and transferable manufacturing process for our current
and future drug candidates that is compliant with current good manufacturing practices, (“cGMP”);

establishing  and  maintaining  supply  and  manufacturing  relationships  with  third  parties  that  can  provide  an  adequate  amount  and  quality  of  drugs  and
services to support clinical development, as well as the market demand for our current and future drug candidates, if approved;

obtaining market acceptance, if and when approved, of our current or any future drug candidates as a viable treatment option by physicians, patients, third-
party payors and others in the medical community;

effectively addressing any competing technological and market developments;

implementing additional internal systems and infrastructure, as needed;

negotiating favorable terms in any collaboration, licensing or other arrangements into which we may enter and performing our obligations pursuant to such
arrangements;

our ability to obtain and maintain orphan drug exclusivity for any of our current and future drug candidates for which we obtain regulatory approval;

maintaining, protecting and expanding our portfolio of intellectual property rights, including patents, trade secrets and know-how;

avoiding and defending against third-party interference or infringement claims; and

securing appropriate pricing in the United States, the European Union and other countries.

We expect our financial condition and operating results to continue to fluctuate from quarter to quarter and year to year due to a variety of factors, many of which
are beyond our control. We will need to eventually transition from a company with a research and development focus to a company capable of undertaking commercial
activities. We may encounter unforeseen expenses, difficulties, complications and delays and may not be successful in such a transition. 

We will require additional capital to finance our operations, which may not be available on acceptable terms, if at all. Failure to obtain this necessary capital when
needed may force us to delay, limit or terminate certain of our drug development efforts or other operations.

Our operations have consumed substantial amounts of cash since our inception. We expect our expenses to increase in connection with our ongoing and planned
activities,  particularly  as  we  continue  to  develop  and  commercialize  our  drug  candidates,  in  addition  to  costs  associated  with  the  acquisition  or  in-licensing  of  any
additional drug candidates we may pursue. Our expenses could increase beyond expectations if the FDA or other regulatory authorities require us to perform clinical and
other studies in addition to those that we currently anticipate. In addition, if we obtain marketing approval for our drug candidates, we expect to incur significant expenses
related to manufacturing, marketing, sales and distribution. Furthermore, we expect to continue to incur additional costs associated with operating as a public company.

As of December 31, 2020, our cash and cash equivalents were $72.0 million and we had an accumulated deficit of $294.2 million. Management has identified
certain conditions or events, which, considered in the aggregate, raise substantial doubt about our ability to continue as a going concern, including the risk that we will be
unable to raise adequate additional capital to fund our

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operations through at least the 12 months following the filing date of this annual report on Form 10-K. Substantial doubt about our ability to continue as a going concern
may create negative reactions to the price of our common stock. If we are unable to raise capital, we may be required to delay, reduce the scope of or eliminate research
and development programs, or obtain funds through arrangements with collaborators or others that may require us to relinquish rights to certain drug candidates that we
might otherwise seek to develop or commercialize independently. In addition, if we are unable to continue as a going concern, we may have to liquidate our assets and
may  receive  less  than  the  value  at  which  those  assets  are  carried  on  our  financial  statements,  and  it  is  likely  that  investors  will  lose  all  or  a  part  of  their  investment.
Further, the perception that we may be unable to continue as a going concern may impede our ability to pursue strategic opportunities or operate our business due to
concerns regarding our ability to discharge our contractual obligations.

We will require more capital in order to continue our preclinical and clinical activities, to obtain regulatory approval and for the commercialization of our current
or future drug candidates. Any additional capital raising efforts may divert our management from their day-to-day activities, which may adversely affect our ability to
develop  and  commercialize  our  current  and  future  drug  candidates.  The  COVID-19  pandemic  has  already  resulted  in  a  significant  disruption  of  global  financial
markets.  If the disruption persists and deepens, we could experience an inability to access additional capital.  If we do not raise additional capital in sufficient amounts, or
on terms acceptable to us, we may be prevented from pursuing development and commercialization efforts, which will harm our business, operating results and prospects.

Raising  additional  capital  or  acquiring  or  licensing  assets  by  issuing  equity  or  debt  securities  may  cause  dilution  to  our  stockholders,  and  raising  funds  through
lending and licensing arrangements may restrict our operations or require us to relinquish proprietary rights.

Until such time as we can generate substantial revenue from drug sales, if ever, we expect to finance our cash needs through a combination of equity and debt
financings, strategic alliances, and license and development agreements in connection with any collaborations. We do not have any committed external source of funds.
To the extent that we issue additional equity securities, our stockholders may experience substantial dilution, and the terms of these securities may include liquidation or
other preferences that adversely affect your rights as a stockholder. In addition, we may issue equity or debt securities as consideration for obtaining rights to additional
compounds. For example, in our arrangement with Takeda, upon the achievement of a certain development milestone, we will be obligated to issue to Takeda additional
securities equal to up to 8% of our outstanding capital stock in certain situations which will dilute our stockholders. In addition, further dilution may occur if we elect to
issue shares of common stock to Takeda as payment for the remaining potential global commercial and regulatory milestone payments, which aggregate to approximately
$35.0 million. In March 2021, we entered into a royalty, license and termination agreement (“Takeda License and Termination Agreement”) with Takeda under which
Takeda will secure global rights at closing from us to develop and commercialize the investigational medicine OV935 for the treatment of developmental and epileptic
encephalopathies,  including  DS  and  LGS.  Closing  of  the  Takeda  License  and  Termination  Agreement  is  subject  to  satisfaction  of  customary  closing  conditions.  See
“Business—License and Collaboration Agreements—Agreements with Takeda—2021 Royalty, License and Termination Agreement with Takeda” for a discussion of the
terms of the Takeda License and Termination Agreement.

Debt  and  equity  financings,  if  available,  may  involve  agreements  that  include  covenants  limiting  or  restricting  our  ability  to  take  specific  actions,  such  as
redeeming our shares, making investments, issuing additional equity, incurring additional debt, making capital expenditures, declaring dividends or placing limitations on
our ability to acquire, sell or license intellectual property rights and other operating restrictions that could negatively impact our ability to conduct our business. If we
raise additional capital through future collaborations, strategic alliances or third-party licensing arrangements, we may have to relinquish valuable rights to our intellectual
property, future revenue streams, research programs or drug candidates, or grant licenses on terms that may not be favorable to us. For example, on July 9, 2020, we
entered  into  a  collaboration  and  license  agreement  (the  “Angelini  License  Agreement”)  with  Angelini  Pharma  Rare  Diseases  AG,  pursuant  to  which  we  granted  to
Angelini exclusive rights to develop and commercialize OV101 in the European Economic Area as well as Switzerland, the United Kingdom, Russia and Turkey.  The
licenses granted to Angelini include sublicenses under our existing license agreement with H. Lundbeck A/S (“Lundbeck”), as well as licenses under our patents and
know-how covering OV101.

If  we  are  unable  to  raise  additional  capital  when  needed,  we  may  be  required  to  delay,  limit,  reduce  or  terminate  our  drug  development  or  future

commercialization efforts, or grant rights to develop and market drug candidates that we would otherwise develop and market ourselves.

Our ability to use our net operating loss (“NOL”) carryforwards and certain other tax attributes to offset future taxable income may be subject to limitation.

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Our NOL carryforwards could expire unused and be unavailable to offset future income tax liabilities because of their limited duration or because of restrictions
under U.S. tax law. Our federal NOLs generated in tax years beginning on or before December 31, 2017 are permitted to be carried forward for only 20 years under
applicable U.S. tax law.  Under the Tax Cuts and Jobs Act, or the Tax Act, as modified by the Coronavirus Aid, Relief, and Economic Security Act, or the CARES Act,
federal NOLs incurred in taxable years beginning after December 31, 2017 may be carried forward indefinitely, but the utilization of such federal NOLs incurred in the
taxable year beginning after December 31, 2020 is limited. It is uncertain how various states will respond to the Tax Act and CARES Act.

In addition, under Section 382 and Section 383 of the Internal Revenue Code of 1986, as amended, and corresponding provisions of state law, if a corporation
undergoes an “ownership change,” its ability to use its pre-change NOL carryforwards and other pre-change tax attributes (such as research tax credits) to offset its post-
change income may be limited. A Section 382 “ownership change” generally occurs if one or more stockholders or groups of stockholders who own at least 5% of our
stock  increase  their  ownership  by  more  than  50  percentage  points  (by  value)  over  their  lowest  ownership  percentage  over  a  rolling  three-year  period.  We  may  have
experienced ownership changes in the past and may experience ownership changes in the future as a result of shifts in our stock ownership (some of which are outside our
control). As a result, if we earn net taxable income, our ability to use our pre-change NOLs to offset such taxable income may be subject to limitations. Similar provisions
of state tax law may also apply to limit our use of accumulated state tax attributes. In addition, at the state level, there may be periods during which the use of NOLs is
suspended or otherwise limited, which could accelerate or permanently increase state taxes owed.

Consequently, even if we achieve profitability, we may not be able to utilize a material portion of our NOL carryforwards and certain other tax attributes, which

could have a material adverse effect on cash flow and results of operations.

Risks Related to the Development and Commercialization of Our Drug Candidates

Our future success is dependent on the successful clinical development, regulatory approval and commercialization of our current and future drug candidates. If we,
or our licensees, are not able to obtain required regulatory approvals, we will not be able to commercialize our drug candidates, and our ability to generate revenue
will be adversely affected.

We  do  not  have  any  drugs  that  have  received  regulatory  approval.  Our  business  is  dependent  on  our  ability  to  successfully  complete  preclinical  and  clinical
development  of,  obtain  regulatory  approval  for,  and,  if  approved,  successfully  commercialize  our  current  and  future  drug  candidates  in  a  timely  manner.  Activities
associated  with  the  development  and  commercialization  of  our  current  and  future  drug  candidates  are  subject  to  comprehensive  regulation  by  the  FDA  and  other
regulatory agencies in the United States and similar regulatory authorities outside the United States. Failure to obtain regulatory approval in the United States or other
jurisdictions would prevent us from commercializing and marketing our current and future drug candidates. An inability to effectively develop and commercialize our
current and future drug candidates, whether due to the impacts of the ongoing COVID-19 pandemic or otherwise, could have an adverse effect on our business, financial
condition, results of operations and growth prospects.

Further, activities associated with the development and commercialization of our current and future drug candidates are subject to comprehensive regulation by
the FDA and other regulatory agencies in the United States and similar regulatory authorities outside the United States. Failure to obtain regulatory approval in the United
States or other jurisdictions would prevent us from commercializing and marketing our current and future drug candidates.

Even if we obtain approval from the FDA and comparable foreign regulatory authorities for our current and future drug candidates, any approval might contain
significant  limitations  related  to  use  restrictions  for  specified  age  groups,  warnings,  precautions  or  contraindications,  or  may  be  subject  to  burdensome  post-approval
study or risk management requirements. If we are unable to obtain regulatory approval, or any approval contains significant limitations, we may not be able to obtain
sufficient  funding  or  generate  sufficient  revenue  to  continue  the  development  of  that  drug  candidate  or  any  other  drug  candidate  that  we  may  in-license,  develop  or
acquire in the future.  In certain circumstances, including under our license agreement with Angelini for OV101, our third-party licensees are responsible for obtaining
regulatory approvals in the countries covered by the license, and we are dependent on their efforts in order to achieve the necessary approvals in order to commercialize
our products.  If Angelini, or any future licensees fail to perform their obligations to develop and obtain regulatory approvals for the licensed products, we may not be
able to commercialize our products in the affected countries, or our ability to do so may be substantially delayed.

Furthermore, even if we obtain regulatory approval for our current and future drug candidates, we will still need to develop a commercial organization, establish a
commercially  viable  pricing  structure  and  obtain  approval  for  adequate  reimbursement  from  third-party  and  government  payors.  If  we  are  unable  to  successfully
commercialize our current and future drug candidates, we may not be able to generate sufficient revenue to continue our business.

Because the results of preclinical studies or earlier clinical trials are not necessarily predictive of future results, our drug candidates may not have favorable results
in planned or future preclinical studies or clinical trials, or may not receive regulatory approval.

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Success in preclinical testing and early clinical trials does not ensure that subsequent clinical trials will generate similar results or otherwise provide adequate
data to demonstrate the efficacy and safety of a drug candidate. Frequently, drug candidates that have shown promising results in early clinical trials have subsequently
suffered  significant  setbacks  in  later  clinical  trials.  For  instance,  our  STARS  trial  was  the  first  clinical  trial  evaluating  efficacy  of  OV101  in  patients  with  Angelman
syndrome and OV101 has not been evaluated in a clinical trial to treat Fragile X syndrome. We may be unable to demonstrate efficacy in any future trials, including any
future clinical trials of OV101 to treat Angelman syndrome. For instance, in December 2020, we reported the primary endpoint of the NEPTUNE study was not achieved.
Based on the results of the NEPTUNE trial, further development of OV101, other than the ELARA trial, is currently on hold. Similarly, our Phase 1b/2a adult study in
OV935 showed exploratory signals of efficacy in seizure frequency reduction, but we may be unable to demonstrate efficacy in future trials in patients with DEE, or the
related indications of Dravet syndrome, Lennox-Gastaut  syndrome,  CDKL5  Deficiency  Disorder  or  Duplication  15q  (“Dup15q”)  syndrome,  and  the  FDA  has  not  yet
made any determination regarding safety and efficacy of OV935 in any of these indications. The results from preclinical studies of OV101 and OV935 in animal models
and the results from our STARS clinical trial of OV101 in patients with Angelman syndrome and clinical trials of OV101 in patients with primary insomnia may not be
predictive of the effects of these compounds in later stage clinical trials. Our approach of targeting the extrasynaptic GABAA receptor with OV101, and cholesterol 24-
hydroxylase (CH24H) with OV935, are both novel and unproven, and as such, the cost and time needed to develop OV101 and OV935 is difficult to predict  and  our
efforts  may  not  be  successful.  If  we  do  not  observe  favorable  results  in  clinical  trials  of  one  of  our  drug  candidates,  we  may  decide  to  delay  or  abandon  clinical
development of that drug candidate. Any such delay or abandonment could harm our business, financial condition, results of operations and prospects.

Interim topline and preliminary results from our clinical trials that we announce or publish from time to time may change as more patient data become available and
are subject to audit and verification procedures, which could result in material changes in the final data.

From time to time, we have and may in the future publish or report preliminary or interim data from our clinical trials, such as the initial data we announced from
the ENDYMION open label extension trial for OV935 in September 2019, which involved data from the first six patients enrolled in that extension trial which showed
promising  signs  of  efficacy  over  the  treatment  period,  or  the  topline  data  from  the  ELEKTRA  trial  for  OV935  in  August  2020.  Preliminary  or  interim  data  from  our
clinical trials and those of our partners may not be indicative of the final results of the trial and are subject to the risk that one or more of the clinical outcomes may
materially change as patient enrollment continues and/or more patient data become available. Preliminary or topline results also remain subject to audit and verification
procedures that may result in the final data being materially different from the preliminary data we previously published or reported. As a result, preliminary or interim
data should be considered carefully and with caution until final data are available. Differences between preliminary or interim data and final data could significantly harm
our business prospects and may cause the trading price of our common stock to fluctuate significantly.

We may encounter substantial delays in our clinical trials or we may fail to demonstrate safety and efficacy to the satisfaction of applicable regulatory authorities.

Before obtaining marketing approval from regulatory authorities for the sale of our drug candidates, we must conduct extensive clinical trials to demonstrate the
safety  and  efficacy  of  the  drug  candidate  for  its  intended  indications.  Clinical  trials  are  expensive,  time-consuming  and  uncertain  as  to  outcome.  Further,  delays  and
interruptions to ongoing trials related to the COVID-19 pandemic may also increase the duration and costs of such trials. We cannot guarantee that any clinical trials will
be conducted as planned or completed on schedule, if at all. A failure of one or more clinical trials can occur at any stage of testing. Events that may prevent successful or
timely completion of clinical development include:

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delays in reaching a consensus with regulatory authorities on trial design;

delays in reaching agreement on acceptable terms with prospective clinical research organizations (“CROs”) and clinical trial sites;

delays in opening investigational sites;

delays or difficulty in recruiting and enrollment of suitable patients to participate in our clinical trials, whether as a result of the COVID-19 pandemic or
otherwise;

imposition of a clinical hold by regulatory authorities because of a serious adverse event, concerns with a class of drug candidates or after an inspection of
our clinical trial operations or trial sites;

delays in having patients complete participation in a trial or return for post-treatment follow-up;

occurrence of serious adverse events associated with the drug candidate that are viewed to outweigh its potential benefits;

changes in regulatory requirements and guidance that require amending or submitting new clinical protocols; or

business interruptions resulting from geo-political actions, including war and terrorism, or natural disasters and public health epidemics.

In addition, our clinical trials may be affected by the COVID-19 pandemic.

Clinical site initiation and patient enrollment may be delayed due to prioritization of hospital resources toward the COVID-19 pandemic. Patients may not be able
to comply with clinical trial protocols if quarantines impede patient movement or interrupt healthcare services. Similarly, our ability to recruit and retain patients and
principal investigators and site staff who, as healthcare providers, may have heightened exposure to COVID-19, could be limited, which in turn could adversely impact
our clinical trial operations. Additionally, we may experience interruption of key clinical trial activities, such as clinical trial site monitoring, due to limitations on travel,
quarantines or social distancing protocols imposed or recommended by federal or state governments, employers and others in connection with the ongoing COVID-19
pandemic. As a result of the COVID-19 pandemic, we have faced and may continue to face delays in meeting our anticipated timelines for our ongoing and planned
clinical trials.

Further, clinical endpoints for certain diseases we are targeting, such as Angelman syndrome and Fragile X syndrome, have not been established, and accordingly
we may have to develop new modalities or modify existing endpoints to measure efficacy, which may increase the time it takes for us to commence or complete clinical
trials. In addition, we believe investigators in this area may be inexperienced in conducting trials in this area due to the current lack of drugs to treat these disorders, which
may result in increased time and expense to train investigators and open clinical sites.

Any inability to successfully complete preclinical and clinical development could result in additional costs to us or impair our ability to generate revenue from
future drug sales and regulatory and commercialization milestones. In addition, if we make manufacturing or formulation changes to our drug candidates, we may need to
conduct additional testing to bridge our modified drug candidate to earlier versions. Clinical trial delays could also shorten any periods during which we may have the
exclusive right to commercialize our drug candidates, if approved, or allow our competitors to bring comparable drugs to market before we do, which could impair our
ability to successfully commercialize our drug candidates and may harm our business, financial condition, results of operations and prospects.

Additionally, if the results of our clinical trials are inconclusive or if there are safety concerns or serious adverse events associated with our drug candidates, we

may:

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be delayed in obtaining marketing approval, if at all;

obtain approval for indications or patient populations that are not as broad as intended or desired;

obtain approval with labeling that includes significant use or distribution restrictions or safety warnings;

be subject to additional post-marketing testing requirements;

be required to perform additional clinical trials to support approval or be subject to additional post-marketing testing requirements;

have  regulatory  authorities  withdraw,  or  suspend,  their  approval  of  the  drug  or  impose  restrictions  on  its  distribution  in  the  form  of  a  modified  risk
evaluation and mitigation strategy (“REMS”);

be subject to the addition of labeling statements, such as warnings or contraindications;

be sued; or

experience damage to our reputation.

Our  drug  development  costs  will  also  increase  if  we  experience  delays  in  testing  or  obtaining  marketing  approvals.  We  do  not  know  whether  any  of  our

preclinical studies or clinical trials will begin as planned, need to be restructured or be completed on schedule, if at all.

Further, we, the FDA or an institutional review board (“IRB”) may suspend our clinical trials at any time if it appears that we or our collaborators are failing to
conduct a trial in accordance with regulatory requirements, including the FDA’s current Good Clinical Practice (“GCP) regulations, that we are exposing participants to
unacceptable  health  risks,  or  if  the  FDA  finds  deficiencies  in  our  investigational  new  drug  (“IND”)  applications  or  the  conduct  of  these  trials.  Therefore,  we  cannot
predict with any certainty the schedule for commencement and completion of future clinical trials. If we experience delays in the commencement or completion of our
clinical trials, or if we terminate a clinical trial prior to completion, the commercial prospects of our drug candidates could be negatively impacted, and our ability to
generate revenues from our drug candidates may be delayed.

Angelman syndrome has no treatments approved by the U.S. Food and Drug Administration, and the primary clinical endpoint, CGI-I-AS, has not previously been
used as a sole primary endpoint in a pivotal clinical trial.

Angelman  syndrome  is  characterized  by  a  variety  of  signs  and  symptoms,  such  as  delayed  development,  intellectual  disability,  severe  speech  impairment,
problems with movement and balance, seizures, sleep disorders and anxiety. In order to obtain a broad indication for treatment of Angelman syndrome from the FDA, we
may need to demonstrate efficacy on several of the key symptoms of Angelman syndrome. If we fail to do so, our clinical development may be delayed and/or our label
may be limited. In December 2020, we reported the primary endpoint of the NEPTUNE study was not achieved. Based  on  the  results  of  the  NEPTUNE  trial,  further
development of OV101, other than the ELARA trial, is currently on hold.

We may need to develop a new liquid formulation of OV101 for use in infant patients if our existing formulation in capsules that can be opened and sprinkled on
semi-solid foods is not acceptable to the regulatory authorities, and we may be unable to successfully develop an appropriate liquid formulation

Our existing formulation of OV101 is an oral capsule. We have recently developed lower strength capsules that can be opened and sprinkled on applesauce or
similar  semi-solid  foods.  However,  we  may  need  to  develop  an  oral  liquid  formulation  of  OV101  for  use  in  very  young  pediatric  patients.  While  we  have  begun
developing this formulation, we do not know if our efforts will be successful or if the FDA will agree that the new formulation is comparable to our current formulation.
We may experience manufacturing problems that may affect solubility or stability, or we may discover that the new formulation is less effective than an oral capsule. In
addition, we will need to conduct bridging studies to demonstrate that the new formulation is equivalent to our oral capsule, which could result in delays in development
and additional costs.

If  we  are  not  successful  in  discovering,  developing  and  commercializing  additional  drug  candidates,  our  ability  to  expand  our  business  and  achieve  our  strategic
objectives would be impaired.

A key element of our strategy is to develop and potentially commercialize a portfolio of drug candidates to treat rare neurological disorders. We intend to do so
by  in-licensing  and  entering  into  collaborations  with  leading  biopharmaceutical  companies  or  academic  institutions  for  new  drug  candidates.  Identifying  new  drug
candidates  requires  substantial  technical,  financial  and  human  resources,  whether  or  not  any  drug  candidates  are  ultimately  identified.  Our  approach  to  business
development, including our efforts to map the biological pathways related to orphan disorders of the brain and our relationships among the pharmaceutical industry, may
not result in viable drug candidates for clinical development. The COVID-19 pandemic could also impact our ability to do in person due diligence, negotiations and other
interactions to identify new opportunities. Even if we identify drug candidates that initially show promise, we may fail to in-license or acquire these assets and may also
fail to successfully develop and commercialize such drug candidates for many reasons, including the following:

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the research methodology used may not be successful in identifying potential drug candidates;

competitors may develop alternatives that render any drug candidate we develop obsolete;

any drug candidate we develop may nevertheless be covered by third parties’ patents or other exclusive rights;

a drug candidate may, on further study, be shown to have harmful side effects or other characteristics that indicate it is unlikely to be effective or otherwise
does not meet applicable regulatory criteria;

a drug candidate may not be capable of being produced in commercial quantities at an acceptable cost, or at all; and

a drug candidate may not be accepted as safe and effective by physicians, patients, the medical community or third-party payors.

We have limited financial and management resources and, as a result, we may forego or delay pursuit of opportunities with other drug candidates or for other
indications that later prove to have greater market potential. Our resource allocation decisions may cause us to fail to capitalize on viable commercial drugs or profitable
market opportunities. If we do not accurately evaluate the commercial potential or target market for a particular drug candidate, we may relinquish valuable rights to that
drug candidate through collaboration, licensing or other royalty arrangements in circumstances under which it would have been more advantageous for us to retain sole
development and commercialization rights to such drug candidate.

If we are unsuccessful in identifying and developing additional drug candidates or are unable to do so, our key growth strategy and business will be harmed.

Clinical trials are very expensive, time-consuming and difficult to design and implement.

Our drug candidates will require clinical testing before we are prepared to submit a new drug application (“NDA”) for regulatory approval. We cannot predict
with any certainty if or when we might submit an NDA for regulatory approval for any of our drug candidates or whether any such NDA will be approved by the FDA.
Human clinical trials are very expensive and difficult to design and implement, in part because they are subject to rigorous regulatory requirements. For instance, the FDA
may not agree with our proposed endpoints for any future clinical trial of our drug candidates, which may delay the commencement of our clinical trials. In addition, we
may not succeed in developing and validating disease-relevant clinical endpoints based on insights regarding biological pathways for the disorders we are studying. The
clinical  trial  process  is  also  time-consuming.  We  estimate  that  the  successful  completion  of  clinical  trials  of  our  drug  candidates  will  take  at  least  several  years  to
complete, if not longer. Furthermore, failure can occur at any stage and we could encounter problems that cause us to abandon or repeat clinical trials.

Enrollment  and  retention  of  patients  in  clinical  trials  is  an  expensive  and  time-consuming  process  and  could  be  made  more  difficult  or  rendered  impossible  by
multiple factors outside our control.

Identifying  and  qualifying  patients  to  participate  in  our  clinical  trials  is  critical  to  our  success.  The  number  of  patients  suffering  from  Angelman  syndrome,
Fragile  X  syndrome  and  DEE,  such  as  Dravet  syndrome,  Lennox-Gastaut  syndrome,  Dup15q  syndrome  and  CDKL5  deficiency  disorder  is  small  and  has  not  been
established with precision. If the actual number of patients with these disorders is smaller than we anticipate, we may encounter difficulties in enrolling patients in our
clinical trials, thereby delaying or preventing development and approval of our drug candidates. Even once enrolled we may be unable to retain a sufficient number of
patients to complete any of our trials. Patient enrollment and retention in clinical trials depends on many factors, including the size of the patient population, the nature of
the trial protocol, the existing body of safety and efficacy data, the number and nature of competing treatments and ongoing clinical trials of competing therapies for the
same indication, the proximity of patients to clinical sites and the eligibility criteria for the trial, any such enrollment issues could cause delays or prevent development
and approval of our drug candidates. Because we are focused on addressing rare neurological disorders, there are limited patient pools from which to draw in order to
complete our clinical trials in a timely and cost-effective manner. Furthermore, our efforts to build relationships with patient communities may not succeed, which could
result in delays in patient enrollment in our clinical trials. In addition, any negative results we may report in clinical trials of our drug candidate may make it difficult or
impossible to recruit and retain patients in other clinical trials of that same drug candidate. Delays or failures in planned patient enrollment or retention may result in
increased costs, program delays or both, which could have a harmful effect on our ability to develop our drug candidates, or could render further development impossible.
For example, the impact of public health pandemics, such as COVID-19, may delay or prevent patients from enrolling or from receiving treatment in accordance with the
protocol and the required timelines, which could delay our clinical trials, or prevent us or our partners from completing our clinical trials at all, and harm our ability to
obtain approval for such product candidate. In addition, we may rely on CROs and clinical trial sites to ensure proper and timely conduct of our future clinical trials and,
while we intend to enter into agreements governing their services, we will be limited in our ability to compel their actual performance.

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Our drug candidates may cause undesirable side effects or have other properties that could delay or prevent their regulatory approval, limit the commercial potential
or result in significant negative consequences following any potential marketing approval.

During the conduct of clinical trials, patients report changes in their health, including illnesses, injuries and discomforts, to their doctor. Often, it is not possible to
determine whether or not the drug candidate being studied caused these conditions. Regulatory authorities may draw different conclusions or require additional testing to
confirm these determinations, if they occur. In addition, it is possible that as we test our drug candidates in larger, longer and more extensive clinical programs, or as use
of these drug candidates becomes more widespread if they receive regulatory approval, illnesses, injuries, discomforts and other adverse events that were observed in
earlier trials, as well as conditions that did not occur or went undetected in previous trials, will be reported by subjects. Many times, side effects are only detectable after
investigational drugs are tested in large-scale, Phase 3 trials or, in some cases, after they are made available to patients on a commercial scale after approval. For example,
in one of the trials conducted by Lundbeck, there were reports of hallucinations in drug abusers at 30mg and 45mg doses of OV101, which are higher than the 10mg and
15mg doses that were effective for insomnia. In addition, some patients treated with OV101 in the Lundbeck Phase 3 trials experienced headaches, nausea and dizziness.
In the STARS study, the most frequent adverse events for OV101 treated arms that were greater than placebo arm included pyrexia, rash, seizure, enuresis, myoclonic
epilepsy, otitis media and viral infection. Patients in our ongoing or planned clinical trials may experience similar or other adverse events after treatment with OV101. In
the Phase 1b/2a OV935 trial, adverse events that occurred more frequently in the OV935-treatment group versus the placebo group were dysarthria, insomnia, lethargy,
seizure cluster, and upper respiratory infection. If additional clinical experience indicates that any of our current drug candidates, including OV101 and OV935, or any
future drug candidates has adverse events or causes serious or life-threatening adverse events, the development of that drug candidate may fail or be delayed, or, if the
drug candidate has received regulatory approval, such approval may be revoked, which would harm our business, prospects, operating results and financial condition.

Moreover, if we elect, or are required, to delay, suspend or terminate any clinical trial of our drug candidates, the commercial prospects of our drug candidates
may be harmed and our ability to generate revenue through their sale may be delayed or eliminated. Any of these occurrences may harm our business, financial condition
and prospects significantly.

Additionally, if any of our drug candidates receive marketing approval, the FDA could require us to include a black box warning in our label or adopt REMS to
ensure that the benefits outweigh its risks, which may include, among other things, a medication guide outlining the risks of the drug for distribution to patients and a
communication plan to health care practitioners. Furthermore, if we or others later identify undesirable side effects caused by our drug candidates, several potentially
significant negative consequences could result, including:

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regulatory authorities may suspend or withdraw approvals of such drug candidate;

regulatory authorities may require additional warnings on the label;

we may be required to change the way a drug candidate is administered or conduct additional clinical trials;

we could be sued and held liable for harm caused to patients;

we may need to conduct a recall; and

our reputation may suffer.

Any  of  these  events  could  prevent  us  from  achieving  or  maintaining  market  acceptance  of  our  drug  candidates  and  could  significantly  harm  our  business,

prospects, financial condition and results of operations.

If  the  market  opportunities  for  our  drug  candidates  are  smaller  than  we  believe  they  are,  even  assuming  approval  of  a  drug  candidate,  our  business  may  suffer.
Because  the  patient  populations  in  the  market  for  our  drug  candidates  may  be  small,  we  must  be  able  to  successfully  identify  patients  and  acquire  a  significant
market share to achieve profitability and growth.

We focus our research and drug development on treatments for rare neurological disorders. Given the small number of patients who have the disorders that we are
targeting, our eligible patient population and pricing estimates may differ significantly from the actual market addressable by our drug candidates. Our projections of both
the  number  of  people  who  have  these  disorders,  as  well  as  the  subset  of  people  with  these  disorders  who  have  the  potential  to  benefit  from  treatment  with  our  drug
candidates, are based on our beliefs and estimates. These estimates have been derived from a variety of sources, including the scientific literature, patient foundations, or
market research, and may prove to be incorrect. Further, new studies may change the estimated incidence or prevalence of these disorders. The number of patients may
turn out to be lower than expected. Likewise, the potentially addressable patient population for each of our drug candidates may be limited or may not be amenable to
treatment  with  our  drug  candidates,  and  new  patients  may  become  increasingly  difficult  to  identify  or  gain  access  to,  which  would  adversely  affect  our  results  of
operations and our business. 

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We face substantial competition, which may result in others developing or commercializing drugs before or more successfully than us.

The  development  and  commercialization  of  new  drugs  is  highly  competitive.  We  face  competition  with  respect  to  our  current  drug  candidates  and  will  face
competition  with  respect  to  any  other  drug  candidates  that  we  may  seek  to  develop  or  commercialize  in  the  future,  from  major  pharmaceutical  companies,  specialty
pharmaceutical companies and biotechnology companies worldwide. There are a number of large pharmaceutical and biotechnology companies that currently market and
sell  drugs  or  are  pursuing  the  development  of  drug  candidates  for  the  treatment  of  the  indications  that  we  are  pursuing.  Potential  competitors  also  include  academic
institutions,  government  agencies  and  other  public  and  private  research  organizations  that  conduct  research,  seek  patent  protection  and  establish  collaborative
arrangements for research, development, manufacturing and commercialization.

More  established  companies  may  have  a  competitive  advantage  over  us  due  to  their  greater  size,  resources  and  institutional  experience.  In  particular,  these
companies have greater experience and expertise in securing reimbursement, government contracts, relationships with key opinion leaders, conducting testing and clinical
trials,  obtaining  and  maintaining  regulatory  approvals  and  distribution  relationships  to  market  products,  and  marketing  approved  drugs.  These  companies  also  have
significantly greater research and marketing capabilities than we do. If we are not able to compete effectively against existing and potential competitors, our business and
financial condition may be harmed.

As  a  result  of  these  factors,  our  competitors  may  obtain  regulatory  approval  of  their  drugs  before  we  are  able  to,  which  may  limit  our  ability  to  develop  or
commercialize our drug candidates. Our competitors may also develop therapies that are safer, more effective, more widely accepted and cheaper than ours, and may also
be  more  successful  than  us  in  manufacturing  and  marketing  their  drugs.  These  appreciable  advantages  could  render  our  drug  candidates  obsolete  or  non-competitive
before we can recover the expenses of such drug candidates’ development and commercialization.

Mergers and acquisitions in the pharmaceutical and biotechnology industries may result in even more resources being concentrated among a smaller number of
our competitors. Smaller and other early-stage companies may also prove to be significant competitors, particularly through collaborative arrangements with large and
established companies. These third parties compete with us in recruiting and retaining qualified scientific, management and commercial personnel, establishing clinical
trial sites and subject registration for clinical trials, as well as in acquiring technologies complementary to, or necessary for, our programs.

Even if our current or future drug candidates receive marketing approval, they may fail to achieve market acceptance by physicians, patients, third-party payors or
others in the medical community necessary for commercial success.

Even if our current or future drug candidates receive marketing approval, they may fail to gain sufficient market acceptance by physicians, patients, third-party
payors and others in the medical community. If they do not achieve an adequate level of acceptance, we may not generate significant drug revenue and may not become
profitable. The degree of market acceptance of our current or future drug candidates, if approved for commercial sale, will depend on a number of factors, including but
not limited to:

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the efficacy and potential advantages compared to alternative treatments and therapies;

the safety profile of our drug candidate compared to alternative treatments and therapies;

effectiveness of sales and marketing efforts;

the strength of our relationships with patient communities;

the cost of treatment in relation to alternative treatments and therapies, including any similar generic treatments;

our ability to offer such drug for sale at competitive prices;

the convenience and ease of administration compared to alternative treatments and therapies;

the willingness of the target patient population to try new therapies and of physicians to prescribe these therapies;

the strength of marketing and distribution support;

the availability of third-party coverage and adequate reimbursement;

the prevalence and severity of any side effects; and

any restrictions on the use of the drug together with other medications.

Our efforts to educate physicians, patients, third-party payors and others in the medical community on the benefits of our drug candidates may require significant
resources and may never be successful. Such efforts may require more resources than are typically required due to the complexity and uniqueness of our drug candidates.
Because we expect sales of our drug candidates, if approved, to

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generate substantially all of our drug revenues for the foreseeable future, the failure of our drugs to find market acceptance would harm our business and could require us
to seek additional financing.

If  we  are  unable  to  establish  sales  and  marketing  capabilities,  or  enter  into  agreements  with  third  parties  to  market  and  sell  our  current  or  any  future  drug
candidates, we may be unable to generate any revenue from drug sales.

To successfully commercialize any drug candidate that may result from our development programs, we will need to build out our sales and marketing capabilities,
either  on  our  own  or  with  others.  The  establishment  and  development  of  our  own  commercial  team  or  the  establishment  of  a  contract  sales  force  to  market  any  drug
candidate we may develop will be expensive and time-consuming and could delay any drug launch. Moreover, we cannot be certain that we will be able to successfully
develop this capability. We may seek to enter into additional collaborations with other entities to utilize their established marketing and distribution capabilities, but we
may be unable to enter into such agreements on favorable terms, if at all. If any current or future collaborators do not commit sufficient resources to commercialize our
drug candidates, or we are unable to develop the necessary capabilities on our own, we will be unable to generate sufficient revenue to sustain our business. We compete
with  many  companies  that  currently  have  extensive,  experienced  and  well-funded  marketing  and  sales  operations  to  recruit,  hire,  train  and  retain  marketing  and  sales
personnel. We also face competition in our search for third parties to assist us with the sales and marketing efforts of our current and future drug candidates. Without an
internal  team  or  the  support  of  a  third  party  to  perform  marketing  and  sales  functions,  we  may  be  unable  to  compete  successfully  against  these  more  established
companies.

Even if we obtain and maintain approval for our current or future drug candidates from the FDA, we may never obtain approval for our current or future drug
candidates outside of the United States, which would limit our market opportunities and could harm our business.

Approval of a drug candidate in the United States by the FDA does not ensure approval of such drug candidate by regulatory authorities in other countries or
jurisdictions, and approval by one foreign regulatory authority does not ensure approval by regulatory authorities in other foreign countries or by the FDA. Sales of our
current and future drug candidates outside of the United States will be subject to foreign regulatory requirements governing clinical trials and marketing approval. Even if
the FDA grants marketing approval for a drug candidate, comparable regulatory authorities of foreign countries also must approve the manufacturing and marketing of the
drug  candidate  in  those  countries.  Approval  procedures  vary  among  jurisdictions  and  can  involve  requirements  and  administrative  review  periods  different  from,  and
more onerous than, those in the United States, including additional preclinical studies or clinical trials. In many countries outside the United States, a drug candidate must
be approved for reimbursement before it can be approved for sale in that country. In some cases, the price that we intend to charge for any drug candidates, if approved, is
also subject to approval. Obtaining approval for our current and future drug candidates in the European Union from the European Commission following the opinion of
the EMA, if we choose to submit a marketing authorization application there, would be a lengthy and expensive process. Even if a drug candidate is approved, the FDA or
the European Commission, as the case may be, may limit the indications for which the drug may be marketed, require extensive warnings on the drug labeling or require
expensive  and  time-consuming  additional  clinical  trials  or  reporting  as  conditions  of  approval.  Obtaining  foreign  regulatory  approvals  and  compliance  with  foreign
regulatory  requirements  could  result  in  significant  delays,  difficulties  and  costs  for  us  and  could  delay  or  prevent  the  introduction  of  our  current  and  future  drug
candidates in certain countries. In certain cases, including under our license with Angelini, which covers the European Economic Area as well as Switzerland, the United
Kingdom, Russia and Turkey, we are dependent on third parties to obtain such foreign regulatory approvals, and any delay or failure of performance of such third parties
could  delay  or  prevent  our  ability  to  commercialize  our  products  in  the  affected  countries.  Due  to  the  ongoing  COVID-19  pandemic,  it  is  possible  that  we  could
experience  delays  in  the  timing  of  our  interactions  with  regulatory  authorities  due  to  absenteeism  by  governmental  employees,  inability  to  conduct  planned  physical
inspections  related  to  regulatory  approval,  or  the  diversion  of  regulatory  authority  efforts  and  attention  to  approval  of  other  therapeutics  or  other  activities  related  to
COVID-19,  which  could  delay  anticipated  approval  decisions  and  otherwise  delay  or  limit  our  ability  to  make  planned  regulatory  submissions  or  obtain  new  product
approvals.

Further,  clinical  trials  conducted  in  one  country  may  not  be  accepted  by  regulatory  authorities  in  other  countries.  Also,  regulatory  approval  for  our  drug
candidates may be withdrawn. If we fail to comply with the regulatory requirements, our target market will be reduced and our ability to realize the full market potential
of our current and future drug candidates will be harmed and our business, financial condition, results of operations and prospects could be harmed.

If we seek approval to commercialize our current or future drug candidates outside of the United States, in particular in the European Union and Israel, a variety of
risks associated with international operations could harm our business.

If  we  seek  approval  of  our  current  or  future  drug  candidates  outside  of  the  United  States,  we  expect  that  we  will  be  subject  to  additional  risks  in

commercialization including:

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different regulatory requirements for approval of therapies in foreign countries;

reduced protection for intellectual property rights;

the potential requirement of additional clinical studies in international jurisdictions;

unexpected changes in tariffs, trade barriers and regulatory requirements;

economic weakness, including inflation, or political instability in particular foreign economies and markets;

compliance with tax, employment, immigration and labor laws for employees living or traveling abroad;

foreign currency fluctuations, which could result in increased operating expenses and reduced revenues, and other obligations incident to doing business in
another country;

foreign reimbursement, pricing and insurance regimes;

workforce uncertainty in countries where labor unrest is more common than in the United States;

production shortages resulting from any events affecting raw material supply or manufacturing capabilities abroad; and

business interruptions resulting from geopolitical actions, including war and terrorism or natural disasters and public health pandemics, such as COVID-
19;

We  have  no  prior  experience  in  these  areas.  In  addition,  there  are  complex  regulatory,  tax,  labor  and  other  legal  requirements  imposed  by  both  the  European
Union,  Israel  and  many  of  the  individual  countries  in  and  outside  of  Europe  with  which  we  will  need  to  comply.  Many  biopharmaceutical  companies  have  found  the
process of marketing their own products in foreign countries to be very challenging.

Product liability lawsuits against us could cause us to incur substantial liabilities and could limit commercialization of any drug candidate that we may develop.

We face an inherent risk of product liability exposure related to the testing of our current and any future drug candidates in clinical trials and may face an even
greater risk if we commercialize any drug candidate that we may develop. If we cannot successfully defend ourselves against claims that any such drug candidates caused
injuries, we could incur substantial liabilities. Regardless of merit or eventual outcome, liability claims may result in:

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decreased demand for any drug candidate that we may develop;

loss of revenue;

substantial monetary awards to trial participants or patients;

significant time and costs to defend the related litigation;

withdrawal of clinical trial participants;

the inability to commercialize any drug candidate that we may develop; and

injury to our reputation and significant negative media attention.

Although we maintain product liability insurance coverage, such insurance may not be adequate to cover all liabilities that we may incur. We anticipate that we
will need to increase our insurance coverage each time we commence a clinical trial and if we successfully commercialize any drug candidate. Insurance coverage is
increasingly expensive. We may not be able to maintain insurance coverage at a reasonable cost or in an amount adequate to satisfy any liability that may arise.

Risks Related to Licensing and Collaboration Arrangements

We are heavily dependent on our relationship with Takeda for the development and commercialization of OV935. Any disruption in our relationship with Takeda
could lead to delays in, or the termination of, the development of OV935, which would materially harm our business.

We  are  jointly  developing  OV935  with  Takeda  pursuant  to  the  Takeda  collaboration,  which  also  granted  us  intellectual  property  rights  to  OV935.  The
development and commercialization of OV935 is highly dependent upon our relationship with Takeda, including Takeda’s submission of the IND to the FDA. If for any
reason  the  Takeda  collaboration  is  terminated,  or  we  otherwise  lose  the  intellectual  property  rights  to  OV935,  our  business  would  be  adversely  affected.  The  Takeda
collaboration  imposes  on  us  rights  and  obligations,  including  but  not  limited  to  exclusivity,  territorial  rights,  development,  commercialization,  funding,  payment,
diligence, sublicensing, insurance and intellectual property protection. After a negotiated time period, each party has the right to

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terminate the license for convenience upon six to twelve months’ notice to the other party, which would result in us being unable to co-develop and sell OV935. Further,
if we breach any material obligations, or use the intellectual property licensed to us in an unauthorized manner, we may be required to pay damages to Takeda, and Takeda
may have the right to terminate the license. Takeda could also breach its obligations under the agreement or may not commit a sufficient amount of resources to satisfy its
obligations,  which  would  result  in  the  development  of  OV935  being  materially  delayed  or  terminated.  In  March  2021,  we  entered  into  the  Takeda  License  and
Termination Agreement under  which  Takeda  will  secure  global  rights  at  closing  from  us  to  develop  and  commercialize  the  investigational  medicine  OV935  for  the
treatment of developmental and epileptic encephalopathies, including DS and LGS. Closing of the Takeda License and Termination Agreement is subject to satisfaction of
customary closing conditions. See “Business—License and Collaboration Agreements—Agreements with Takeda—2021 Royalty,  License  and  Termination  Agreement
with Takeda” for a discussion of the terms of the Takeda License and Termination Agreement.

We are dependent on our relationship with Angelini for the development and commercialization of OV101 in European Economic Area as well as Switzerland, the
United  Kingdom,  Russia  and  Turkey.  Any  disruption  in  our  relationship  with  Angelini  could  lead  to  delays  in  the  development  and  achievement  of  regulatory
approval in these countries, which would materially harm our business.

Under our license agreement with Angelini, Angelini obtained exclusive rights to develop and commercialize OV101 in the European Economic Area as well as
Switzerland, the United Kingdom, Russia and Turkey. The development and commercialization of OV101 is highly dependent upon our relationship with Angelini, and
on  Angelini’s  performance  of  its  obligations  under  the  agreement,  including  with  respect  to  the  preparation  and  submission  of  applications  for  marketing  approval  in
Europe and the other licensed countries. If for any reason Angelini fails to perform its obligations, we may not be able to achieve regulatory approval for OV101 in the
licensed countries, or may be materially delayed in doing so, and our business would be adversely affected.

We may be required to make significant payments in connection with our licenses of OV101 from Lundbeck and OV935 from Takeda.

We  acquired  rights  to  OV101,  pursuant  to  a  license  agreement  with  Lundbeck  in  March  2015  (the  “Lundbeck  Agreement”),  as  amended  on  May  10,  2019.
Under  the  Lundbeck  Agreement,  as  amended,  we  are  subject  to  significant  obligations,  including  payment  obligations  upon  achievement  of  specified  milestones  and
royalties  on  drug  sales,  as  well  as  other  material  obligations.  We  are  obligated  to  pay  Lundbeck  milestone  payments  up  to  an  aggregate  of  $189.0  million  upon  the
achievement of certain development, regulatory and sales milestone events. In addition, we are obligated to pay Lundbeck tiered royalties based on net sales of OV101. If
these payments become due under the terms of the Lundbeck agreement, we may not have sufficient funds available to meet our obligations and our development efforts
may be harmed.

We  also  acquired  rights  to  OV935  pursuant  to  a  license  and  collaboration  agreement  with  Takeda  (the  “Takeda  collaboration”)  in  January  2017.  Under  the
Takeda collaboration, we are obligated to pay Takeda future payments upon achievement of specified milestones. Upon the first patient enrollment in the first Phase 3 trial
for the first of the initial indications we and Takeda are focusing on pursuant to the Takeda collaboration, we are obligated to issue to Takeda the number of unregistered
shares of our common stock equal to the lesser of (i) 8% of our outstanding capital stock on the issuance date or (ii) $50.0 million divided by the applicable share price,
unless certain events occur. The remaining potential global commercial and regulatory milestone payments equal approximately $35.0 million and can be satisfied in cash
or  unregistered  shares  of  our  common  stock  at  our  election,  unless  certain  events  occur  in  which  Takeda  can  require  us  to  pay  such  payments  in  cash.  In  the  event  a
payment settled in shares of our common stock would cause Takeda to own over 19.99% of our outstanding capital stock or other events occur, such payment must be
paid in cash. If these payments become due under the terms of the Takeda collaboration and we can only pay, or choose to pay, these payments in cash, we may not have
sufficient  funds  available  to  meet  our  obligations  and  our  development  efforts  may  be  harmed.  In  March  2021,  we  entered  into  the  Takeda  License  and  Termination
Agreement under  which  Takeda  will  secure  global  rights  at  closing  from  us  to  develop  and  commercialize  the  investigational  medicine  OV935  for  the  treatment  of
developmental and epileptic encephalopathies, including DS and LGS. Closing of the Takeda License and Termination Agreement is subject to satisfaction of customary
closing conditions. See “Business—License and Collaboration Agreements—Agreements with Takeda—2021 Royalty, License and Termination Agreement with Takeda”
for a discussion of the terms of the Takeda License and Termination Agreement.

Risks  associated  with  the  in-licensing  or  acquisition  of  drug  candidates  could  cause  substantial  delays  in  the  preclinical  and  clinical  development  of  our  drug
candidates.

Prior to March 2015, we had no involvement with or control over the preclinical and clinical research and development of OV101. We have relied on Lundbeck
or  its  prior  licensee  to  have  conducted  such  research  and  development  in  accordance  with  the  applicable  protocol,  legal,  regulatory  and  scientific  standards,  having
accurately reported the results of all clinical trials conducted prior to our acquisition of OV101 and having correctly collected and interpreted the data from these trials. If
the research and development processes or the results of the development programs prior to our acquisition of OV101 prove to be unreliable, this could result in increased
costs and delays in the development of OV101, which could adversely affect any future revenue from this drug candidate.

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Similarly, we acquired rights to OV935 from Takeda in January 2017. Because we were not involved in the development of OV935 prior to January 2017, we
may experience difficulties in the transition of certain development activities from Takeda and its affiliates to us, which may result in delays in clinical trials, as well as
problems in our development efforts. In March 2021, we entered into the Takeda License and Termination Agreement under which Takeda will secure global rights at
closing from us to develop and commercialize the investigational medicine OV935 for the treatment of developmental and epileptic encephalopathies, including DS and
LGS. Closing of the Takeda License and Termination Agreement is subject to satisfaction of customary closing conditions. See “Business—License and Collaboration
Agreements—Agreements  with  Takeda—2021  Royalty,  License  and  Termination  Agreement  with  Takeda”  for  a  discussion  of  the  terms  of  the  Takeda  License  and
Termination Agreement.

We may also acquire or in-license additional drug candidates for preclinical or clinical development in the future as we continue to build our pipeline. The risks
associated  with  acquiring  or  in-licensing  current  or  future  drug  candidates  could  result  in  delays  in  the  commencement  or  completion  of  our  preclinical  studies  and
clinical trials, if ever, and our ability to generate revenues from our drug candidates may be delayed.

We may be required to relinquish important rights to and control over the development and commercialization of our drug candidates to any future collaborators.

Our current and future collaborations could subject us to a number of risks, including:

we may be required to undertake the expenditure of substantial operational, financial and management resources;

we may be required to issue equity securities that would dilute our stockholders’ percentage of ownership;

we may be required to assume substantial actual or contingent liabilities;

we may not be able to control the amount and timing of resources that our strategic collaborators devote to the development or commercialization of our
drug candidates;

strategic collaborators may delay clinical trials, provide insufficient funding, terminate a clinical trial or abandon a drug candidate, repeat or conduct new
clinical trials or require a new version of a drug candidate for clinical testing;

strategic collaborators may not pursue further development and commercialization of products resulting from the strategic collaboration arrangement or
may elect to discontinue research and development programs;

strategic collaborators may not commit adequate resources to the marketing and distribution of our drug candidates, limiting our potential revenues from
these products;

we rely on our current collaborators to manufacture drug substance and drug product and may do so with respect to future collaborators, which could result
in disputes or delays;

disputes may arise between us and our strategic collaborators that result in the delay or termination of the research, development or commercialization of
our drug candidates or that result in costly litigation or arbitration that diverts management’s attention and consumes resources;

strategic collaborators may experience financial difficulties;

strategic collaborators may not properly maintain or defend our intellectual property rights or may use our proprietary information in a manner that could
jeopardize or invalidate our proprietary information or expose us to potential litigation;

business combinations or significant changes in a strategic collaborator’s business strategy may also adversely affect a strategic collaborator’s willingness
or ability to complete its obligations under any arrangement;

strategic  collaborators  could  decide  to  move  forward  with  a  competing  drug  candidate  developed  either  independently  or  in  collaboration  with  others,
including our competitors; and

strategic collaborators could terminate the arrangement or allow it to expire, which would delay the development and may increase the cost of developing
our drug candidates.

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We may explore additional strategic collaborations that may never materialize or may fail.

Our business strategy is based on acquiring or in-licensing compounds directed at rare neurological disorders. As a result, we intend to periodically explore a
variety of possible additional strategic collaborations in an effort to gain access to additional drug candidates or resources. At the current time, we cannot predict what
form such a strategic collaboration might take. We are likely to face significant competition in seeking appropriate strategic collaborators, and strategic collaborations can
be complicated and time consuming to negotiate and document. We may not be able to negotiate strategic collaborations on acceptable terms, or at all. We are unable to
predict when, if ever, we will enter into any additional strategic collaborations because of the numerous risks and uncertainties associated with establishing them.

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Risks Related to Regulatory Compliance

Our relationships with customers, physicians, and third-party payors may be subject, directly or indirectly, to federal and state healthcare fraud and abuse laws, false
claims laws, health information privacy and security laws, and other healthcare laws and regulations. If we are unable to comply, or have not fully complied, with
such laws, we could face substantial penalties.

Healthcare  providers  and  third-party  payors  in  the  United  States  and  elsewhere  will  play  a  primary  role  in  the  recommendation  and  prescription  of  any  drug
candidates for which we obtain marketing approval. Our current and future arrangements with healthcare professionals, principal investigators, consultants, customers and
third-party payors may subject us to various federal and state fraud and abuse laws and other healthcare laws, including, without limitation, the federal Anti-Kickback
Statute,  the  federal  civil  and  criminal  false  claims  laws  and  the  law  commonly  referred  to  as  the  Physician  Payments  Sunshine  Act  and  regulations.  These  laws  will
impact, among other things, our clinical research, proposed sales, marketing and educational programs. In addition, we may be subject to patient privacy laws by both the
federal government and the states in which we conduct or may conduct our business. The laws that will affect our operations include, but are not limited to:

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the federal Anti-Kickback Statute, which prohibits, among other things, persons or entities from knowingly and willfully soliciting, receiving, offering or
paying any remuneration (including any kickback, bribe or rebate), directly or indirectly, overtly or covertly, in cash or in kind, in return for the purchase,
recommendation,  leasing  or  furnishing  of  an  item  or  service  reimbursable  under  a  federal  healthcare  program,  such  as  the  Medicare  and  Medicaid
programs. This statute has been interpreted to apply to arrangements between pharmaceutical manufacturers on the one hand, and prescribers, purchasers
and formulary managers on the other. The Patient Protection and Affordable Care Act, as amended by the Health Care and Education Reconciliation Act
(collectively,  the  “PPACA”),  amended  the  intent  requirement  of  the  federal  Anti-Kickback  Statute.  A  person  or  entity  no  longer  needs  to  have  actual
knowledge of this statute or specific intent to violate it in order to have committed a violation;

federal civil and criminal false claims laws, including, without limitation, the False Claims Act, and civil monetary penalty laws which prohibit, among
other things, individuals or entities from knowingly presenting, or causing to be presented, claims for payment or approval from Medicare, Medicaid or
other government payors that are false or fraudulent or making a false statement to avoid, decrease or conceal an obligation to pay money to the federal
government. The PPACA provides, and recent government cases against pharmaceutical and medical device manufacturers support, the view that federal
Anti-Kickback Statute violations and certain marketing practices, including off-label promotion, may implicate the False Claims Act;

the  federal  Health  Insurance  Portability  and  Accountability  Act  of  1996  (“HIPAA”),  which  created  additional  federal  criminal  statutes  that  prohibit  a
person from knowingly and willfully executing a scheme or making false or fraudulent statements to defraud any healthcare benefit program, regardless of
the payor (e.g., public or private);

HIPAA, as amended by the Health Information Technology for Economic and Clinical Health Act (“HITECH”), and their implementing regulations, and
as amended again by the final HIPAA omnibus rule, Modifications to the HIPAA Privacy, Security, Enforcement, and Breach Notification Rules Under
HITECH  and  the  Genetic  Information  Nondiscrimination  Act;  Other  Modifications  to  HIPAA,  published  in  January  2013,  which  imposes  certain
requirements relating to the privacy, security and transmission of individually identifiable health information without appropriate authorization by entities
subject  to  the  rule,  such  as  health  plans,  healthcare  clearinghouses  and  certain  healthcare  providers,  known  as  covered  entities,  and  their  respective
business associates, individuals or entities that perform certain services on behalf of a covered entity that involves the use or disclosure of individually
identifiable health information and their subcontractors that use, disclose or otherwise process individually identifiable health information;

Physician Payments Sunshine Act, which is part of the PPACA, that require certain manufacturers of drugs, devices, biologics and medical supplies for
which  payment  is  available  under  Medicare,  Medicaid  or  the  Children’s  Health  Insurance  Program,  with  specific  exceptions,  to  report  annually  to  the
Centers  for  Medicare  &  Medicaid  Services  (“CMS”),  information  related  to:  (i)  payments  or  other  “transfers  of  value”  made  to  physicians  (defined  to
include doctors, dentists, optometrists, podiatrists and chiropractors) and teaching hospitals; and (ii) ownership and investment interests held by physicians
and  their  immediate  family  members  which  will  be  expanded  beginning  in  2022,  to  require  applicable  manufacturers  to  report  information  regarding
payments and other transfers of value provided to physician assistants, nurse practitioners, clinical nurse specialists, anesthesiologist assistants, certified
registered nurse anesthetists and certified nurse midwives during the previous year;

state and foreign law equivalents of each of the above federal laws, state laws that require manufacturers to report information related to payments and
other transfers of value to physicians and other healthcare providers or marketing expenditures and/or information regarding drug pricing, state laws that
require pharmaceutical companies to comply with the pharmaceutical industry’s voluntary compliance guidelines and the relevant compliance guidance
promulgated by the federal government or to adopt compliance programs as prescribed by state laws and regulations, or that otherwise restrict payments
that may be made to healthcare providers, state laws and regulations that require drug manufacturers to file reports relating to drug pricing and marketing
information, and state and local laws that require the registration of pharmaceutical sales representatives; and

state  and  foreign  laws  that  govern  the  privacy  and  security  of  health  information  in  some  circumstances,  many  of  which  differ  from  each  other  in
significant ways and often are not preempted by HIPAA, thus complicating compliance efforts.

Because of the breadth of these laws and the narrowness of the statutory exceptions and regulatory safe harbors available, it is possible that some of our business

activities could be subject to challenge under one or more of such laws.

It  is  possible  that  governmental  authorities  will  conclude  that  our  business  practices  may  not  comply  with  current  or  future  statutes,  regulations  or  case  law
involving  applicable  fraud  and  abuse  or  other  healthcare  laws  and  regulations.  If  our  operations  are  found  to  be  in  violation  of  any  of  these  laws  or  any  other
governmental regulations that may apply to us, we may be subject to significant civil, criminal and administrative penalties, damages, fines, disgorgement, imprisonment,
exclusion from participation in government funded healthcare programs, such as Medicare and Medicaid, additional reporting requirements and oversight if we become
subject  to  a  corporate  integrity  agreement  or  similar  agreement  to  resolve  allegations  of  non-compliance  with  these  laws  and  the  curtailment  or  restructuring  of  our
operations.

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The risk of our being found in violation of these laws is increased by the fact that many of them have not been fully interpreted by the regulatory authorities or the
courts,  and  their  provisions  are  open  to  a  variety  of  interpretations.  Efforts  to  ensure  that  our  business  arrangements  with  third  parties  will  comply  with  applicable
healthcare laws and regulations will involve substantial costs. Any action against us for violation of these laws, even if we successfully defend against it, could cause us to
incur significant legal expenses and divert our management’s attention from the operation of our business. The shifting compliance environment and the need to build and
maintain  robust  and  expandable  systems  to  comply  with  multiple  jurisdictions  with  different  compliance  and/or  reporting  requirements  increases  the  possibility  that  a
healthcare company may run afoul of one or more of the requirements.

Coverage and adequate reimbursement may not be available for our current or any future drug candidates, which could make it difficult for us to sell profitably, if
approved.

Market  acceptance  and  sales  of  any  drug  candidates  that  we  commercialize,  if  approved,  will  depend  in  part  on  the  extent  to  which  coverage  and  adequate
reimbursement  for  these  drugs  and  related  treatments  will  be  available  from  third-party  payors,  including  government  health  administration  authorities,  managed  care
organizations and other private health insurers. Third-party payors decide which therapies they will pay for and establish reimbursement levels. Third-party payors often
rely  upon  Medicare  coverage  policy  and  payment  limitations  in  setting  their  own  coverage  and  reimbursement  policies.  However,  decisions  regarding  the  extent  of
coverage  and  amount  of  reimbursement  to  be  provided  for  any  drug  candidates  that  we  develop  will  be  made  on  a  payor-by-payor  basis.  One  third-party  payor’s
determination to provide coverage for a drug does not assure that other payors will also provide coverage, and adequate reimbursement, for the drug. Additionally, a third-
party payor’s decision to provide coverage for a therapy does not imply that an adequate reimbursement rate will be approved. Each third-party payor determines whether
or not it will provide coverage for a therapy, what amount it will pay the manufacturer for the therapy, and on what tier of its formulary it will be placed. The position on a
third-party  payor’s  list  of  covered  drugs,  or  formulary,  generally  determines  the  co-payment  that  a  patient  will  need  to  make  to  obtain  the  therapy  and  can  strongly
influence  the  adoption  of  such  therapy  by  patients  and  physicians.  Patients  who  are  prescribed  treatments  for  their  conditions  and  providers  prescribing  such  services
generally  rely  on  third-party  payors  to  reimburse  all  or  part  of  the  associated  healthcare  costs.  Patients  are  unlikely  to  use  our  drugs  unless  coverage  is  provided  and
reimbursement is adequate to cover a significant portion of the cost of our drugs.

A primary trend in the U.S. healthcare industry and elsewhere is cost containment. Third-party payors have attempted to control costs by limiting coverage and
the amount of reimbursement for particular medications. We cannot be sure that coverage and reimbursement will be available for any drug that we commercialize and, if
reimbursement is available, what the level of reimbursement will be. Inadequate coverage and reimbursement may impact the demand for, or the price of, any drug for
which we obtain marketing approval. If coverage and adequate reimbursement are not available, or are available only to limited levels, we may not be able to successfully
commercialize our current and any future drug candidates that we develop. Further, coverage policies and third-party payor reimbursement rates may change at any time.
Even if favorable coverage and reimbursement status is attained, less favorable coverage policies and reimbursement rates may be implemented in the future.

Healthcare legislative reform measures may have a negative impact on our business and results of operations.

In  the  United  States  and  some  foreign  jurisdictions,  there  have  been,  and  continue  to  be,  several  legislative  and  regulatory  changes  and  proposed  changes
regarding the healthcare system that could prevent or delay marketing approval of drug candidates, restrict or regulate post-approval activities, and affect our ability to
profitably sell any drug candidates for which we obtain marketing approval.

Among policy makers and payors in the United States and elsewhere, there is significant interest in promoting changes in healthcare systems with the stated goals
of containing healthcare costs, improving quality and/or expanding access. In the United States, the pharmaceutical industry has been a particular focus of these efforts
and has been significantly affected by major legislative initiatives. In March 2010, the PPACA was passed, which substantially changed the way healthcare is financed by
both the government and private insurers, and significantly impacts the U.S. pharmaceutical industry.

There  have  been  executive,  judicial,  Congressional  and  executive  branch  challenges  to  certain  aspects  of  the  PPACA.  For  example,  President  Trump  signed
Executive Orders and other directives designed to delay the implementation of certain provisions of the PPACA or otherwise circumvent some of the requirements for
health insurance mandated by the PPACA.  Concurrently, Congress considered legislation to repeal or repeal and replace all or part of the PPACA. While Congress has
not passed comprehensive repeal legislation, it has enacted laws that modify certain provisions of the PPACA such as removing penalties, starting January 1, 2019, for not
complying with the PPACA’s individual mandate to carry health insurance, delaying the implementation of certain PPACA-mandated fees, and increasing the point-of-
sale discount that is owed by pharmaceutical manufacturers who participate in Medicare Part D.  Additionally, the 2020 federal spending package permanently eliminated,
effective January 1, 2020, the PPACA-mandated “Cadillac” tax on high-cost employer-sponsored health coverage and medical device tax and, effective January 1, 2021,
also  eliminated  the  health  insurer  tax.  On  December  14,  2018,  a  Texas  U.S.  District  Court  Judge  ruled  that  the  PPACA  is  unconstitutional  in  its  entirety  because  the
“individual mandate” was repealed by Congress as part of the Tax Cuts and Jobs Act of 2017. On December 18, 2019, the U.S. Court of Appeals for the 5th Circuit
upheld the District Court ruling that the individual mandate was

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unconstitutional and remanded the case back to the District Court to determine whether the remaining provisions of the PPACA are invalid as well. The United States
Supreme Court is currently reviewing this case, but it is unknown when a decision will be reached. Although the Supreme Court has not yet ruled on the constitutionality
of the PPACA, on January 28, 2021, President Biden issued an executive order to initiate a special enrollment period from February 15, 2021 through May 15, 2021 for
purposes  of  obtaining  health  insurance  coverage  through  the  PPACA  marketplace.  The  executive  order  also  instructs  certain  governmental  agencies  to  review  and
reconsider their existing policies and rules that limit access to healthcare, including among others, reexamining Medicaid demonstration projects and waiver programs
that include work requirements, and policies that create barriers to obtaining access to health insurance coverage through Medicaid or the PPACA. It is unclear how the
Supreme Court ruling, other such litigation and the healthcare reform measures of the Biden administration will impact the PPACA and our business.  

Other legislative changes have been proposed and adopted since the PPACA was enacted. These changes include aggregate reductions to Medicare payments to
providers of up to 2% per fiscal year pursuant to the Budget Control Act of 2011, which began in 2013, and due to subsequent legislative amendments to the statute,
including the BBA, will remain in effect through 2030 unless additional Congressional action is taken. However, COVID-19 relief legislation suspended the 2% Medicare
sequester from May 1, 2020 through March 31, 2021. The American Taxpayer Relief Act of 2012, among other things, further reduced Medicare payments to several
providers, including hospitals and cancer treatment centers, and increased the statute of limitations period for the government to recover overpayments to providers from
three to five years.

Additional changes that may affect our business include the expansion of new programs such as Medicare payment for performance initiatives for physicians
under the Medicare Access and CHIP Reauthorization Act of 2015 (“MACRA”), which ended the use of the statutory formula and established a quality payment program,
also referred to as the Quality Payment Program. In November 2019, CMS issued a final rule finalizing the changes to the Quality Payment Program. At this time, the full
impact to overall physician reimbursement as a result of the introduction of the Quality Payment Program remains unclear.

Also, there has been heightened governmental scrutiny recently over the manner in which drug manufacturers set prices for their marketed products, which have
resulted in several Congressional inquiries and proposed and enacted federal and state legislation designed to, among other things, bring more transparency to product
pricing, review the relationship between pricing and manufacturer patient programs, and reform government program reimbursement methodologies for drug products. At
the federal level, the Trump administration used several means to propose or implement drug pricing reform, including through federal budget proposals, executive orders
and policy initiatives. For example, on July 24, 2020 and September 13, 2020, the Trump administration announced several executive orders related to prescription drug
pricing that attempt to implement several of the administration’s proposals. The FDA also released a final rule, effective November 30, 2020, implementing a portion of
the  importation  executive  order  providing  guidance  for  states  to  build  and  submit  importation  plans  for  drugs  from  Canada.  Further,  on  November  20,  2020,  HHS
finalized a regulation removing safe harbor protection for price reductions from pharmaceutical manufacturers to plan sponsors under Part D, either directly or through
pharmacy benefit managers, unless the price reduction is required by law. The implementation of the rule has been delayed by the Biden administration from January 1,
2022 to January 1, 2023 in response to ongoing litigation. The rule also creates a new safe harbor for price reductions reflected at the point-of-sale, as well as a new safe
harbor for certain fixed fee arrangements between pharmacy benefit managers and manufacturers, the implementation of which have also been delayed pending review by
the  Biden  administration  until  March  22,  2021.  On  November  20,  2020,  CMS  issued  an  interim  final  rule  implementing  President  Trump’s  Most  Favored  Nation
executive order, which would tie Medicare Part B payments for certain physician-administered drugs to the lowest price paid in other economically advanced countries,
effective  January  1,  2021.  On  December  28,  2020,  the  United  States  District  Court  in  Northern  California  issued  a  nationwide  preliminary  injunction  against
implementation of the interim final rule. It is unclear whether the Biden administration will work to reverse these measures or pursue similar policy initiatives. At the state
level, legislatures have increasingly passed and implemented regulations designed to control pharmaceutical and biological product pricing, including pricing, including
price or patient reimbursement constraints, discounts, restrictions on certain product access and marketing cost disclosure and transparency measures, and, in some cases,
designed  to  encourage  importation  from  other  countries  and  bulk  purchasing.  We  expect  that  these  and  other  healthcare  reform  measures  that  may  be  adopted  in  the
future,  may  result  in  more  rigorous  coverage  criteria  and  in  additional  downward  pressure  on  the  price  that  we  receive  for  any  approved  drug.  Any  reduction  in
reimbursement from Medicare or other government programs may result in a similar reduction in payments from private payors. The implementation of cost containment
measures or other healthcare reforms may prevent us from being able to generate revenue, attain profitability, or commercialize our drugs.

It is possible that additional governmental action is taken in response to the ongoing COVID-19 pandemic.

We may not be able to obtain or maintain orphan drug designations or exclusivity for our drug candidates, which could limit the potential profitability of our drug
candidates.

Regulatory authorities in some jurisdictions, including the United States, may designate drugs for relatively small patient populations as orphan drugs. Under the
Orphan Drug Act of 1983, the FDA may designate a drug as an orphan drug if it is a drug intended to treat a rare disease or condition, which is generally defined as a
patient population of fewer than 200,000 individuals in the United States. Generally, if a drug with an orphan drug designation subsequently receives the first marketing
approval for an indication for which it receives the designation, then the drug is entitled to a period of marketing exclusivity that precludes the

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applicable  regulatory  authority  from  approving  another  marketing  application  for  the  same  drug  for  the  same  indication  for  the  exclusivity  period  except  in  limited
situations. For purposes of small molecule drugs, the FDA defines “same drug” as a drug that contains the same active moiety and is intended for the same use as the drug
in question. A designated orphan drug may not receive orphan drug exclusivity if it is approved for a use that is broader than the indication for which it received orphan
designation.

For  OV101,  the  FDA  granted  orphan  drug  designation  for  OV101  for  the  treatment  of  Angelman  syndrome  and  for  the  treatment  of  Fragile  X  syndrome  in
September  2016  and  October  2017,  respectively.  The  EMA  granted  orphan  designation  for  OV101  for  the  treatment  of  Angelman  syndrome  in  June  2019.  The  FDA
granted orphan drug designation for OV935 for the treatment of Dravet syndrome and Lennox-Gastaut syndrome both in December 2017. We intend to pursue orphan
drug designation for OV101 in additional indications, pending our further analysis of the NEPTUNE trial data and analysis of data from ELARA, for OV935 in additional
indications, pending closing of the Takeda License and Termination Agreement, and for potential other future drug candidates. Obtaining orphan drug designations is
important to our business strategy; however, obtaining an orphan drug designation can be difficult and we may not be successful in doing so. Even if we were to obtain
orphan drug designation for a drug candidate, we may not obtain orphan exclusivity and that exclusivity may not effectively protect the drug from the competition of
different  drugs  for  the  same  condition,  which  could  be  approved  during  the  exclusivity  period.  Additionally,  after  an  orphan  drug  is  approved,  the  FDA  could
subsequently approve another application for the same drug for the same indication if the FDA concludes that the later drug is shown to be safer, more effective or makes
a  major  contribution  to  patient  care.  Orphan  drug  exclusive  marketing  rights  in  the  United  States  also  may  be  lost  if  the  FDA  later  determines  that  the  request  for
designation  was  materially  defective  or  if  the  manufacturer  is  unable  to  assure  sufficient  quantity  of  the  drug  to  meet  the  needs  of  patients  with  the  rare  disease  or
condition. The failure to obtain an orphan drug designation for any drug candidates we may develop, the inability to maintain that designation for the duration of the
applicable  period,  or  the  inability  to  obtain  or  maintain  orphan  drug  exclusivity  could  reduce  our  ability  to  make  sufficient  sales  of  the  applicable  drug  candidate  to
balance our expenses incurred to develop it, which would have a negative impact on our operational results and financial condition.

We have received Fast Track designations for OV101 for the treatment of Angelman syndrome and Fragile X syndrome, but such designations may not actually lead
to a faster development or regulatory review or approval process.

The  FDA  granted  Fast  Track  designations  to  OV101  for  the  treatment  of  Angelman  syndrome  and  Fragile  X  syndrome  in  December  2017  and  March  2018,
respectively. If a drug is intended for the treatment of a serious condition and nonclinical or clinical data demonstrate the potential to address unmet medical need for such
condition, a sponsor may apply for FDA Fast Track designation. Even though we received Fast Track designations for OV101, such Fast Track designations do not ensure
that we will receive marketing approval or that approval will be granted within any particular timeframe for any of these fast track-designated indications. We may not
experience a faster development or regulatory review or approval process with Fast Track designation compared to conventional FDA procedures. In addition, the FDA
may withdraw Fast Track designation if it believes that the designation is no longer supported by data from our clinical development program. Fast Track designation
alone does not guarantee qualification for the FDA’s priority review procedures.

Although the FDA has granted Rare Pediatric Disease Designation for OV101 for the treatment of Angelman Syndrome, an NDA for OV101, if approved, may not
meet the eligibility criteria for a priority review voucher.

Rare Pediatric Disease Designation has been granted for OV101 for the treatment of Angelman Syndrome. In 2012, Congress authorized the FDA to award
priority  review  vouchers  to  sponsors  of  certain  rare  pediatric  disease  product  applications.  This  provision  is  designed  to  encourage  development  of  new  drug  and
biological products for prevention and treatment of certain rare pediatric diseases. Specifically, under this program, a sponsor who receives an approval for a drug or
biologic for a “rare pediatric disease” may qualify for a voucher that can be redeemed to receive a priority review of a subsequent marketing application for a different
product. The sponsor of a rare pediatric disease drug product receiving a priority review voucher may transfer (including by sale) the voucher to another sponsor. The
voucher may be further transferred any number of times before the voucher is used, as long as the sponsor making the transfer has not yet submitted the application. The
FDA  may  also  revoke  any  priority  review  voucher  if  the  rare  pediatric  disease  drug  for  which  the  voucher  was  awarded  is  not  marketed  in  the  U.S.  within  one  year
following  the  date  of  approval.  For  the  purposes  of  this  program,  a  “rare  pediatric  disease”  is  a  (a)  serious  or  life-threatening  disease  in  which  the  serious  or  life-
threatening manifestations primarily affect individuals aged from birth to 18 years, including age groups often called neonates, infants, children, and adolescents; and
(b) rare disease or conditions within the meaning of the Orphan Drug Act. Congress has only authorized the Rare Pediatric Disease Priority Review Voucher program
until September 30, 2024. However, if a drug candidate receives Rare Pediatric Disease Designation before September 30, 2024, it is eligible to receive a voucher if it is
approved before September 30, 2026.

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However, OV101 for the treatment of Angelman Syndrome may not be approved by that date, or at all, and, therefore, we may not be in a position to obtain a
priority  review  voucher  prior  to  expiration  of  the  program,  unless  Congress  further  reauthorizes  the  program.  Additionally,  designation  of  a  drug  for  a  rare  pediatric
disease does not guarantee that an NDA will meet the eligibility criteria for a rare pediatric disease priority review voucher at the time the application is approved. Finally,
a Rare Pediatric Disease Designation does not lead to faster development or regulatory review of the product, or increase the likelihood that it will receive marketing
approval. We may or may not realize any benefit from receiving designation or a voucher.

Even if we obtain regulatory approval for our current or future drug candidates, they will remain subject to ongoing regulatory oversight.

Even  if  we  obtain  any  regulatory  approval  for  our  current  or  future  drug  candidates,  such  approvals  will  be  subject  to  ongoing  regulatory  requirements  for
manufacturing,  labeling,  packaging,  storage,  advertising,  promotion,  sampling,  record-keeping  and  submission  of  safety  and  other  post-market  information.  Any
regulatory approvals that we receive for our current or future drug candidates may also be subject to a REMS, limitations on the approved indicated uses for which the
drug may be marketed or to the conditions of approval, or contain requirements for potentially costly post-marketing testing, including Phase 4 trials, and surveillance to
monitor the quality, safety and efficacy of the drug.

In  addition,  drug  manufacturers  and  their  facilities  are  subject  to  payment  of  user  fees  and  continual  review  and  periodic  inspections  by  the  FDA  and  other
regulatory authorities for compliance with cGMP requirements and adherence to commitments made in the NDA or foreign marketing application. If we, or a regulatory
authority, discover previously unknown problems with a drug, such as adverse events of unanticipated severity or frequency, or problems with the facility where the drug
is manufactured or if a regulatory authority disagrees with the promotion, marketing or labeling of that drug, a regulatory authority may impose restrictions relative to that
drug, the manufacturing facility or us, including requesting a recall or requiring withdrawal of the drug from the market or suspension of manufacturing.

If we fail to comply with applicable regulatory requirements following approval of our current or future drug candidates, a regulatory authority may:

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issue an untitled letter or warning letter asserting that we are in violation of the law;

seek an injunction or impose administrative, civil or criminal penalties or monetary fines;

suspend or withdraw regulatory approval;

suspend any ongoing clinical trials;

refuse to approve a pending NDA or comparable foreign marketing application (or any supplements thereto) submitted by us or our strategic partners;

restrict the marketing or manufacturing of the drug;

seize or detain the drug or otherwise require the withdrawal of the drug from the market;

refuse to permit the import or export of drug candidates; or

refuse to allow us to enter into supply contracts, including government contracts.

Moreover, the FDA strictly regulates the promotional claims that may be made about drug products. In particular, a product may not be promoted for uses that are
not approved by the FDA as reflected in the product’s approved labeling. The FDA and other agencies actively enforce the laws and regulations prohibiting the promotion
of off-label uses, and a company that is found to have improperly promoted off-label uses may be subject to significant civil, criminal and administrative penalties.

Any  government  investigation  of  alleged  violations  of  law  could  require  us  to  expend  significant  time  and  resources  in  response  and  could  generate  negative
publicity. The occurrence of any event or penalty described above may inhibit our ability to commercialize our current or future drug candidates and harm our business,
financial condition, results of operations and prospects.

In addition, the FDA’s policies, and those of equivalent foreign regulatory agencies, may change and additional government regulations may be enacted that could
cause changes to or delays in the drug review process, or suspend or restrict regulatory approval of our drug candidates. We cannot predict the likelihood, nature or extent
of government regulation that may arise from future legislation or administrative action, either in the United States or abroad. If we are slow or unable to adapt to changes
in existing requirements or the adoption of new requirements or policies, or if we are not able to maintain regulatory compliance, we may lose any marketing approval
that we may have obtained and we may not achieve or sustain profitability, which would harm our business, financial condition, results of operations and prospects. 

Risks Related to Our Intellectual Property

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If  we  are  unable  to  obtain  and  maintain  patent  protection  for  our  current  or  any  future  drug  candidates,  or  if  the  scope  of  the  patent  protection  obtained  is  not
sufficiently broad, we may not be able to compete effectively in our markets.

We  rely  upon  a  combination  of  patents,  trade  secret  protection  and  confidentiality  agreements  to  protect  the  intellectual  property  related  to  our  development
programs and drug candidates. Our success depends in large part on our ability to obtain and maintain patent protection in the United States and other countries with
respect to our current and any future drug candidates. We seek to protect our proprietary position by filing patent applications in the United States and abroad related to
our current and future development programs and drug candidates. The patent prosecution process is expensive and time-consuming, and we may not be able to file and
prosecute all necessary or desirable patent applications at a reasonable cost or in a timely manner.

Pursuant  to  the  Lundbeck  Agreement,  as  amended,  we  obtained  an  exclusive,  worldwide  license  to  develop,  manufacture  and  commercialize  OV101  for  the
treatment of human disease. However, the Lundbeck Agreement, as amended, permits Lundbeck and certain other entities to manufacture and research OV101 and, in
certain situations, to perform additional non-commercial activities involving OV101, all of which could result in new patentable inventions concerning the manufacture or
use  of  OV101.  While  the  Lundbeck  Agreement,  as  amended,  prohibits  Lundbeck  from  filing  certain  patent  applications  regarding  OV101  and  obligates  Lundbeck  to
include certain newly filed patents in the license granted to us, if new patents issue that cover valuable methods for making or using OV101, we would be prohibited from
employing such methods to manufacture or use OV101 unless we obtain a license to such patents.

It is also possible that we will fail to identify patentable aspects of our research and development output before it is too late to obtain patent protection. The patent
applications that we own or in-license may fail to result in issued patents with claims that cover our current or any future drug candidates in the United States or in other
foreign countries. There is no assurance that all of the potentially relevant prior art relating to our patents and patent applications has been found, which can invalidate a
patent or prevent a patent from issuing from a pending patent application. Even if patents do successfully issue and even if such patents cover our current or any future
drug candidates, third parties may challenge their validity, enforceability or scope, which may result in such patents being narrowed, invalidated, or held unenforceable.
Any successful opposition to these patents or any other patents owned by or licensed to us could deprive us of rights necessary for the successful commercialization of
any drug candidates or companion diagnostic that we may develop. Further, if we encounter delays in regulatory approvals, the period of time during which we could
market a drug candidate and companion diagnostic under patent protection could be reduced. 

If the patent applications we hold or have in-licensed with respect to our development programs and drug candidates fail to issue, if their breadth or strength of
protection is threatened, or if they fail to provide meaningful exclusivity for our current or any future drug candidates, it could dissuade companies from collaborating
with us to develop drug candidates, and threaten our ability to commercialize, future drugs. Any such outcome could have a negative effect on our business.

The patent position of biotechnology and pharmaceutical companies generally is highly uncertain, involves complex legal and factual questions and has in recent
years been the subject of much litigation. In addition, the laws of foreign countries may not protect our rights to the same extent as the laws of the United States. For
example, European patent law restricts the patentability of methods of treatment of the human body more than United States law does. Publications of discoveries in
scientific literature often lag behind the actual discoveries, and patent applications in the United States and other jurisdictions are typically not published until 18 months
after filing, or in some cases not at all. Therefore, we cannot know with certainty whether we were the first to make the inventions claimed in our owned or licensed
patents or pending patent applications, or that we were the first to file for patent protection of such inventions. As a result, the issuance, scope, validity, enforceability and
commercial value of our patent rights are highly uncertain. Our pending and future patent applications may not result in patents being issued which protect our technology
or  drugs,  in  whole  or  in  part,  or  which  effectively  prevent  others  from  commercializing  competitive  technologies  and  drugs.  Changes  in  either  the  patent  laws  or
interpretation of the patent laws in the United States and other countries may diminish the value of our patents or narrow the scope of our patent protection.

Recent patent reform legislation could increase the uncertainties and costs surrounding the prosecution of our patent applications and the enforcement or defense
of  our  issued  patents.  On  December  16,  2011,  the  Leahy-Smith  America  Invents  Act  (the  “Leahy-Smith  Act”)  was  signed  into  law.  The  Leahy-Smith  Act  includes  a
number  of  significant  changes  to  United  States  patent  law.  These  include  provisions  that  affect  the  way  patent  applications  are  prosecuted  and  may  also  affect  patent
litigation.  The  United  States  Patent  Office  recently  developed  new  regulations  and  procedures  to  govern  administration  of  the  Leahy-Smith  Act,  and  many  of  the
substantive  changes  to  patent  law  associated  with  the  Leahy-Smith  Act,  and  in  particular,  the  first  to  file  provisions,  only  became  effective  on  March  16,  2013.
Accordingly, it is not clear what, if any, impact the Leahy-Smith Act will have on the operation of our business. However, the Leahy-Smith Act and its implementation
could increase the uncertainties and costs surrounding the prosecution of our patent applications and the enforcement or defense of our issued patents, all of which could
harm our business and financial condition.

Moreover, we may be subject to a third-party pre-issuance submission of prior art to the U.S. Patent and Trademark Office (the “USPTO”) or become involved in

opposition, derivation, reexamination, inter partes review, post-grant review or interference

43

 
proceedings challenging our patent rights or the patent rights of others. An adverse determination in any such submission, proceeding or litigation could reduce the scope
of, or invalidate, our patent rights, allow third parties to commercialize our technology or drugs and compete directly with us, without payment to us, or result in our
inability to manufacture or commercialize drugs without infringing third-party patent rights. In addition, if the breadth or strength of protection provided by our patents
and patent applications is threatened, it could dissuade companies from collaborating with us to license, develop or commercialize current or future drug candidates.

The issuance of a patent is not conclusive as to its inventorship, scope, validity or enforceability, and our owned and licensed patents may be challenged in the
courts  or  patent  offices  in  the  United  States  and  abroad.  An  adverse  determination  in  any  such  challenges  may  result  in  loss  of  exclusivity  or  in  patent  claims  being
narrowed,  invalidated  or  held  unenforceable,  in  whole  or  in  part,  which  could  limit  our  ability  to  stop  others  from  using  or  commercializing  similar  or  identical
technology  and  drugs,  or  limit  the  duration  of  the  patent  protection  of  our  technology  and  drugs.  Moreover,  patents  have  a  limited  lifespan.  In  the  United  States,  the
natural expiration of a patent is generally 20 years from the earliest filing date of a non-provisional patent application. Various extensions may be available; however, the
life of a patent, and the protection it affords, is limited. Without patent protection for our current or future drug candidates, we may be open to competition from generic
versions of such drugs. Given the amount of time required for the development, testing and regulatory review of new drug candidates, patents protecting such candidates
might expire before or shortly after such candidates are commercialized. As a result, our owned and licensed patent portfolio may not provide us with sufficient rights to
exclude others from commercializing drugs similar or identical to ours.

We may be unable to prevent third parties from selling, making, promoting, manufacturing, or distributing alternative polymorphic forms of OV101.

We currently have issued patents directed to polymorphic forms of OV101. These patents would not prevent a third-party from creating, making and marketing
alternative  polymorphic  forms  that  fall  outside  the  scope  of  these  patent  claims.  There  can  be  no  assurance  that  any  such  alternative  polymorphic  forms  will  not  be
therapeutically equivalent and/or commercially feasible. In the event an alternative polymorphic form of OV101 is developed and approved for use in indications that we
may seek approval for, the marketability and commercial success of OV101, if approved, could be materially harmed.

Obtaining  and  maintaining  our  patent  protection  depends  on  compliance  with  various  procedural,  document  submission,  fee  payment  and  other  requirements
imposed by government patent agencies, and our patent protection could be reduced or eliminated for non-compliance with these requirements.

Periodic maintenance fees, renewal fees, annuity fees and various other government fees on patents and/or applications will be due to be paid to the USPTO and
various government patent agencies outside of the United States over the lifetime of our owned and licensed patents and/or applications and any patent rights we may own
or license in the future. We rely on our outside counsel or our licensing partners to pay these fees due to non-U.S. patent agencies. The USPTO and various non-U.S.
government patent agencies require compliance with several procedural, documentary, fee payment and other similar provisions during the patent application process. We
employ  reputable  law  firms  and  other  professionals  to  help  us  comply  and  we  are  also  dependent  on  our  licensors  to  take  the  necessary  action  to  comply  with  these
requirements with respect to our licensed intellectual property. In many cases, an inadvertent lapse can be cured by payment of a late fee or by other means in accordance
with  the  applicable  rules.  There  are  situations,  however,  in  which  non-compliance  can  result  in  abandonment  or  lapse  of  the  patent  or  patent  application,  resulting  in
partial or complete loss of patent rights in the relevant jurisdiction. In such an event, potential competitors might be able to enter the market and this circumstance could
harm our business.

Patent terms may be inadequate to protect our competitive position on our drug candidates for an adequate amount of time.

Given the amount of time required for the development, testing and regulatory review of new drug candidates such as OV101, patents protecting such candidates
might  expire  before  or  shortly  after  such  candidates  are  commercialized.  We  expect  to  seek  extensions  of  patent  terms  in  the  United  States  and,  if  available,  in  other
countries where we are prosecuting patents. In the United States, the Drug Price Competition and Patent Term Restoration Act of 1984 permits a patent term extension of
up  to  five  years  beyond  the  normal  expiration  of  the  patent,  which  is  limited  to  the  approved  indication  (or  any  additional  indications  approved  during  the  period  of
extension). However, the applicable authorities, including the FDA and the USPTO in the United States, and any equivalent regulatory authority in other countries, may
not agree with our assessment of whether such extensions are available, and may refuse to grant extensions to our patents, or may grant more limited extensions than we
request. If this occurs, our competitors may be able to take advantage of our investment in development and clinical trials by referencing our clinical and preclinical data
and launch their drug earlier than might otherwise be the case.

Intellectual property rights do not necessarily address all potential threats to our business.

The  degree  of  future  protection  afforded  by  our  intellectual  property  rights  is  uncertain  because  intellectual  property  rights  have  limitations,  and  may  not

adequately protect our business. The following examples are illustrative:

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others may be able to make compounds or formulations that are similar to our drug candidates but that are not covered by the claims of any patents, should
they issue, that we own or control;

we or any strategic partners might not have been the first to make the inventions covered by the issued patents or pending patent applications that we own
or control;

we might not have been the first to file patent applications covering certain of our inventions;

others  may  independently  develop  similar  or  alternative  technologies  or  duplicate  any  of  our  technologies  without  infringing  our  intellectual  property
rights;

it is possible that our pending patent applications will not lead to issued patents;

issued  patents  that  we  own  or  control  may  not  provide  us  with  any  competitive  advantages,  or  may  be  held  invalid  or  unenforceable  because  of  legal
challenges;

our  competitors  might  conduct  research  and  development  activities  in  the  United  States  and  other  countries  that  provide  a  safe  harbor  from  patent
infringement  claims  for  certain  research  and  development  activities,  as  well  as  in  countries  where  we  do  not  have  patent  rights  and  then  use  the
information learned from such activities to develop competitive drugs for sale in our major commercial markets;

we may not develop additional proprietary technologies that are patentable; and

the patents of others may have an adverse effect on our business.

The  proprietary  map  of  disease-relevant  biological  pathways  underlying  orphan  disorders  of  the  brain  that  we  developed  would  not  be  appropriate  for  patent

protection and, as a result, we rely on trade secrets to protect this aspect of our business.

Third parties may initiate legal proceedings alleging that we are infringing their intellectual property rights, the outcome of which would be uncertain and could
have a negative impact on the success of our business.

Our  commercial  success  depends,  in  part,  upon  our  ability  and  the  ability  of  our  current  or  future  collaborators  to  develop,  manufacture,  market  and  sell  our
current  and  any  future  drug  candidates  and  use  our  proprietary  technologies  without  infringing  the  proprietary  rights  and  intellectual  property  of  third  parties.  The
biotechnology and pharmaceutical industries are characterized by extensive and complex litigation regarding patents and other intellectual property rights. We may in the
future become party to, or be threatened with, adversarial proceedings or litigation regarding intellectual property rights with respect to our current and any future drug
candidates and technology, including interference proceedings, post grant review and inter partes review before the USPTO. Third parties may assert infringement claims
against  us  based  on  existing  patents  or  patents  that  may  be  granted  in  the  future,  regardless  of  their  merit. There  is  a  risk  that  third  parties  may  choose  to  engage  in
litigation with us to enforce or to otherwise assert their patent rights against us. Even if we believe such claims are without merit, a court of competent jurisdiction could
hold that these third-party patents are valid, enforceable and infringed, which could have a negative impact on our ability to commercialize our current and any future
drug candidates.  In order to successfully challenge the validity of any such U.S. patent in federal court, we would need to overcome a presumption of validity. As this
burden  is  a  high  one  requiring  us  to  present  clear  and  convincing  evidence  as  to  the  invalidity  of  any  such  U.S.  patent  claim,  there  is  no  assurance  that  a  court  of
competent jurisdiction would invalidate the claims of any such U.S. patent. If we are found to infringe a third party’s valid and enforceable intellectual property rights, we
could be required to obtain a license from such third party to continue developing, manufacturing and marketing our drug candidate(s) and technology. However, we may
not be able to obtain any required license on commercially reasonable terms or at all. Even if we were able to obtain a license, it could be non-exclusive, thereby giving
our competitors and other third parties access to the same technologies licensed to us, and it could require us to make substantial licensing and royalty payments. We
could be forced, including by court order, to cease developing, manufacturing and commercializing the infringing technology or drug candidate. In addition, we could be
found liable for monetary damages, including treble damages and attorneys’ fees, if we are found to have willfully infringed a patent or other intellectual property right. A
finding  of  infringement  could  prevent  us  from  manufacturing  and  commercializing  our  current  or  any  future  drug  candidates  or  force  us  to  cease  some  or  all  of  our
business operations, which could materially harm our business. Claims that we have misappropriated the confidential information or trade secrets of third parties could
have a similar negative impact on our business, financial condition, results of operations and prospects.  See the section herein titled “Legal Proceedings” for additional
information.

We may be subject to claims asserting that our employees, consultants or advisors have wrongfully used or disclosed alleged trade secrets of their current or former
employers or claims asserting ownership of what we regard as our own intellectual property.

Certain of our employees, consultants or advisors are currently, or were previously, employed at universities or other biotechnology or pharmaceutical companies,
including  our  competitors  or  potential  competitors.  Although  we  try  to  ensure  that  our  employees,  consultants  and  advisors  do  not  use  the  proprietary  information  or
know-how of others in their work for us, we may be subject to claims that these individuals or we have used or disclosed intellectual property, including trade secrets or
other proprietary

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information, of any such individual’s current or former employer. Litigation may be necessary to defend against these claims. If we fail in defending any such claims, in
addition  to  paying  monetary  damages,  we  may  lose  valuable  intellectual  property  rights  or  personnel.  Even  if  we  are  successful  in  defending  against  such  claims,
litigation could result in substantial costs and be a distraction to management.

In addition, while it is our policy to require our employees and contractors who may be involved in the conception or development of intellectual property to
execute agreements assigning such intellectual property to us, we may be unsuccessful in executing such an agreement with each party who, in fact, conceives or develops
intellectual property that we regard as our own. The assignment of intellectual property rights may not be self-executing or the assignment agreements may be breached,
and  we  may  be  forced  to  bring  claims  against  third  parties,  or  defend  claims  that  they  may  bring  against  us,  to  determine  the  ownership  of  what  we  regard  as  our
intellectual property.

We may be involved in lawsuits to protect or enforce our patents, the patents of our licensors or our other intellectual property rights, which could be expensive, time
consuming and unsuccessful.

Competitors  may  infringe  or  otherwise  violate  our  patents,  the  patents  of  our  licensors  or  our  other  intellectual  property  rights.  To  counter  infringement  or
unauthorized use, we may be required to file legal claims, which can be expensive and time-consuming. In addition, in an infringement proceeding, a court may decide
that a patent of ours or our licensors is not valid or is unenforceable, or may refuse to stop the other party from using the technology at issue on the grounds that our
patents do not cover the technology in question. An adverse result in any litigation or defense proceedings could put one or more of our patents at risk of being invalidated
or interpreted narrowly and could put our patent applications at risk of not issuing. The initiation of a claim against a third party may also cause the third party to bring
counter claims against us such as claims asserting that our patents are invalid or unenforceable. In patent litigation in the United States, defendant counterclaims alleging
invalidity or unenforceability are commonplace. Grounds for a validity challenge could be an alleged failure to meet any of several statutory requirements, including lack
of novelty, obviousness, non-enablement or lack of statutory subject matter. Grounds for an unenforceability assertion could be an allegation that someone connected with
prosecution of the patent withheld relevant material information from the USPTO, or made a materially misleading statement, during prosecution. Third parties may also
raise  similar  validity  claims  before  the  USPTO  in  post-grant  proceedings  such  as  ex  parte  reexaminations,  inter  partes  review,  or  post-grant  review,  or  oppositions  or
similar proceedings outside the United States, in parallel with litigation or even outside the context of litigation. The outcome following legal assertions of invalidity and
unenforceability is unpredictable. We cannot be certain that there is no invalidating prior art, of which we and the patent examiner were unaware during prosecution. For
the patents and patent applications that we have licensed, we may have limited or no right to participate in the defense of any licensed patents against challenge by a third
party. If a defendant were to prevail on a legal assertion of invalidity or unenforceability, we would lose at least part, and perhaps all, of any future patent protection on
our current or future drug candidates. Such a loss of patent protection could harm our business.

We may not be able to prevent, alone or with our licensors, misappropriation of our intellectual property rights, particularly in countries where the laws may not
protect  those  rights  as  fully  as  in  the  United  States.  Our  business  could  be  harmed  if  in  litigation  the  prevailing  party  does  not  offer  us  a  license  on  commercially
reasonable terms. Any litigation or other proceedings to enforce our intellectual property rights may fail, and even if successful, may result in substantial costs and distract
our management and other employees.

Furthermore,  because  of  the  substantial  amount  of  discovery  required  in  connection  with  intellectual  property  litigation,  there  is  a  risk  that  some  of  our
confidential information could be compromised by disclosure during this type of litigation. There could also be public announcements of the results of hearings, motions
or other interim proceedings or developments. If securities analysts or investors perceive these results to be negative, it could have an adverse effect on the price of our
common stock.

Changes  in  U.S.  patent  law  or  the  patent  law  of  other  countries  or  jurisdictions  could  diminish  the  value  of  patents  in  general,  thereby  impairing  our  ability  to
protect our current and any future drug candidates.

The United States has recently enacted and implemented wide-ranging patent reform legislation. The U.S. Supreme Court has ruled on several patent cases in
recent years, either narrowing the scope of patent protection available in certain circumstances or weakening the rights of patent owners in certain situations. In addition
to increasing uncertainty with regard to our ability to obtain patents in the future, this combination of events has created uncertainty with respect to the value of patents,
once obtained. Depending on actions by the U.S. Congress, the federal courts, and the USPTO, the laws and regulations governing patents could change in unpredictable
ways that would weaken our ability to obtain new patents or to enforce patents that we have licensed or that we might obtain in the future. Similarly, changes in patent
law and regulations in other countries or jurisdictions or changes in the governmental bodies that enforce them or changes in how the relevant governmental authority
enforces patent laws or regulations may weaken our ability to obtain new patents or to enforce patents that we have licensed or that we may obtain in the future. 

We may not be able to protect our intellectual property rights throughout the world, which could negatively impact our business.

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Filing,  prosecuting  and  defending  patents  covering  our  current  and  any  future  drug  candidates  throughout  the  world  would  be  prohibitively  expensive.
Competitors  may  use  our  technologies  in  jurisdictions  where  we  have  not  obtained  patent  protection  to  develop  their  own  drugs  and,  further,  may  export  otherwise
infringing drugs to territories where we may obtain patent protection, but where patent enforcement is not as strong as that in the United States. These drugs may compete
with our drugs in jurisdictions where we do not have any issued or licensed patents and any future patent claims or other intellectual property rights may not be effective
or sufficient to prevent them from so competing.

Reliance on third parties requires us to share our trade secrets, which increases the possibility that a competitor will discover them or that our trade secrets will be
misappropriated or disclosed.

If we rely on third parties to manufacture or commercialize our current or any future drug candidates, or if we collaborate with additional third parties for the
development  of  our  current  or  any  future  drug  candidates,  we  must,  at  times,  share  trade  secrets  with  them.  We  may  also  conduct  joint  research  and  development
programs  that  may  require  us  to  share  trade  secrets  under  the  terms  of  our  research  and  development  partnerships  or  similar  agreements.  We  seek  to  protect  our
proprietary  technology  in  part  by  entering  into  confidentiality  agreements  and,  if  applicable,  material  transfer  agreements,  consulting  agreements  or  other  similar
agreements  with  our  advisors,  employees,  third-party  contractors  and  consultants  prior  to  beginning  research  or  disclosing  proprietary  information.  These  agreements
typically limit the rights of the third parties to use or disclose our confidential information, including our trade secrets. Despite the contractual provisions employed when
working with third parties, the need to share trade secrets and other confidential information increases the risk that such trade secrets become known by our competitors,
are inadvertently incorporated into the technology of others, or are disclosed or used in violation of these agreements. Given that our proprietary position is based, in part,
on our know-how and trade secrets, a competitor’s discovery of our trade secrets or other unauthorized use or disclosure could have an adverse effect on our business and
results of operations.

In addition, these agreements typically restrict the ability of our advisors, employees, third-party contractors and consultants to publish data potentially relating to
our  trade  secrets.  Despite  our  efforts  to  protect  our  trade  secrets,  our  competitors  may  discover  our  trade  secrets,  either  through  breach  of  our  agreements  with  third
parties, independent development or publication of information by any third-party collaborators. A competitor’s discovery of our trade secrets would harm our business.

Risks Related to Our Dependence on Third Parties

We do not have our own manufacturing capabilities and will rely on third parties to produce clinical and commercial supplies of our current and any future drug
candidates.

We do not own or operate, and we do not expect to own or operate, facilities for drug manufacturing, storage and distribution, or testing. We will be dependent on
third  parties  to  manufacture  the  clinical  supplies  of  our  drug  candidates.  The  drug  substance  for  OV101  was  manufactured  by  Lundbeck.  We  believe  that  the  drug
substance transferred from Lundbeck under the Lundbeck Agreement will be sufficient for us to complete our ongoing and future clinical trials. Until the closing of the
Takeda License and Termination Agreement, we will also continue to rely on Takeda to provide the drug product supply for our planned clinical trials of OV935.

Further, we also will rely on third-party manufacturers to supply us with sufficient quantities of our drug candidates, including OV101 and OV935, to be used, if
approved, for commercialization. Any significant delay in the supply of a drug candidate, or the raw material components thereof, for an ongoing clinical trial due to the
need  to  replace  a  third-party  manufacturer  could  considerably  delay  completion  of  our  clinical  trials,  product  testing  and  potential  regulatory  approval  of  our  drug
candidates.

Further, our reliance on third-party manufacturers entails risks to which we would not be subject if we manufactured drug candidates ourselves including:

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inability to meet our drug specifications and quality requirements consistently;

delay or inability to procure or expand sufficient manufacturing capacity;

issues related to scale-up of manufacturing;

costs and validation of new equipment and facilities required for scale-up;

failure to comply with cGMP and similar foreign standards;

inability to negotiate manufacturing agreements with third parties under commercially reasonable terms, if at all;

termination or nonrenewal of manufacturing agreements with third parties in a manner or at a time that is costly or damaging to us;

reliance on single sources for drug components;

lack of qualified backup suppliers for those components that are currently purchased from a sole or single source supplier;

operations of our third-party manufacturers or suppliers could be disrupted by conditions unrelated to our business or operations, including the bankruptcy
of the manufacturer or supplier; and

carrier disruptions or increased costs that are beyond our control.

Any of these events could lead to clinical trial delays, failure to obtain regulatory approval or impact our ability to successfully commercialize our current or any
future  drug  candidates  once  approved.  Some  of  these  events  could  be  the  basis  for  FDA  action,  including  injunction,  request  for  recall,  seizure,  or  total  or  partial
suspension of production.

We intend to rely on third parties to conduct, supervise and monitor our preclinical studies and clinical trials, and if those third parties perform in an unsatisfactory
manner, it may harm our business.

We do not currently have the ability to independently conduct any clinical trials. We intend to rely on CROs and clinical trial sites to ensure the proper and timely
conduct of our preclinical studies and clinical trials, and we expect to have limited influence over their actual performance. We intend to rely upon CROs to monitor and
manage  data  for  our  clinical  programs,  as  well  as  the  execution  of  future  nonclinical  studies.  We  expect  to  control  only  certain  aspects  of  our  CROs’  activities.
Nevertheless, we will be responsible for ensuring that each of our preclinical studies or clinical trials are conducted in accordance with the applicable protocol, legal,
regulatory and scientific standards and our reliance on the CROs does not relieve us of our regulatory responsibilities.

We and our CROs will be required to comply with good laboratory practices (“GLPs”) and good clinical practices (“GCPs”), which are regulations and guidelines
enforced  by  the  FDA  and  are  also  required  by  the  Competent  Authorities  of  the  Member  States  of  the  European  Economic  Area  and  comparable  foreign  regulatory
authorities  in  the  form  of  International  Conference  on  Harmonization  guidelines  for  any  of  our  drug  candidates  that  are  in  preclinical  and  clinical  development.  The
regulatory  authorities  enforce  GCPs  through  periodic  inspections  of  trial  sponsors,  principal  investigators  and  clinical  trial  sites.  Although  we  will  rely  on  CROs  to
conduct GCP-compliant clinical trials, we remain responsible for ensuring that each of our GLP preclinical studies and clinical trials is conducted in accordance with its
investigational plan and protocol and applicable laws and regulations, and our reliance on the CROs does not relieve us of our regulatory responsibilities. If we or our
CROs fail to comply with GCPs, the clinical data generated in our clinical trials may be deemed unreliable and the FDA or comparable foreign regulatory authorities may
require  us  to  perform  additional  clinical  trials  before  approving  our  marketing  applications.  Accordingly,  if  our  CROs  fail  to  comply  with  these  regulations  or  fail  to
recruit a sufficient number of subjects, we may be required to repeat clinical trials, which would delay the regulatory approval process.

While we will have agreements governing their activities, our CROs will not be our employees, and we will not control whether or not they devote sufficient time
and resources to our future clinical and nonclinical programs. These CROs may also have relationships with other commercial entities, including our competitors, for
whom  they  may  also  be  conducting  clinical  trials,  or  other  drug  development  activities  which  could  harm  our  business.  We  face  the  risk  of  potential  unauthorized
disclosure  or  misappropriation  of  our  intellectual  property  by  CROs,  which  may  reduce  our  trade  secret  protection  and  allow  our  potential  competitors  to  access  and
exploit our proprietary technology. If our CROs do not successfully carry out their contractual duties or obligations, fail to meet expected deadlines, or if the quality or
accuracy of the clinical data they obtain is compromised due to the failure to adhere to our clinical protocols or regulatory requirements or for any other reasons, our
clinical trials may be extended, delayed or terminated, and we may not be able to obtain regulatory approval for, or successfully commercialize any drug candidate that
we develop. As a result, our financial results and the commercial prospects for any drug candidate that we develop would be harmed, our costs could increase, and our
ability to generate revenue could be delayed.

If our relationship with these CROs terminates, we may not be able to enter into arrangements with alternative CROs or do so on commercially reasonable terms.

Switching or adding additional CROs involves substantial cost and requires management time and

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focus. In addition, there is a natural transition period when a new CRO commences work. As a result, delays occur, which can negatively impact our ability to meet our
desired clinical development timelines. Though we intend to carefully manage our relationships with our CROs, there can be no assurance that we will not encounter
challenges or delays in the future or that these delays or challenges will not have a negative impact on our business, financial condition and prospects.

In  addition,  principal  investigators  for  our  clinical  trials  may  serve  as  scientific  advisors  or  consultants  to  us  from  time  to  time  and  receive  compensation  in
connection with such services. Under certain circumstances, we may be required to report some of these relationships to the FDA. The FDA may conclude that a financial
relationship between us and a principal investigator has created a conflict of interest or otherwise affected interpretation of the trial. The FDA may therefore question the
integrity of the data generated at the applicable clinical trial site and the utility of the clinical trial itself may be jeopardized. This could result in a delay in approval, or
rejection, of our marketing applications by the FDA and may ultimately lead to the denial of marketing approval of our current and future drug candidates. 

If our contemplated royalty, license and repurchase agreement with Takeda is not successfully closed or if we fail to realize the benefits we anticipate from such
strategic alliance, it may harm our business.

In March 2021, we entered into the Takeda License and Termination Agreement under which Takeda will secure global rights at closing from us to develop and

commercialize the investigational medicine OV935 for the treatment of developmental and epileptic encephalopathies, including DS and LGS.

Under the Takeda collaboration, Takeda received equity in us and was eligible to receive up to $85.0 million in payments for regulatory milestones, including the

initiation of Phase 3 clinical trials. Since signing the agreement, we led global development of OV935.

Should we close the Takeda License and Termination Agreement, all rights in OV935 will be owned by Takeda, or exclusively licensed to Takeda by us.  Takeda
will  assume  sole  responsibility  for  further  worldwide  development  and  commercialization,  and  we  will  no  longer  have  any  financial  obligation  to  Takeda  under  the
original collaboration agreement, including for milestone payments or any future development and commercialization costs.  Under the Takeda License and Termination
Agreement we will be eligible to receive an upfront payment of $196.0 million at closing and eligible to receive up to an additional $660.0 million upon Takeda achieving
development, regulatory and sales milestones. In addition, we would be entitled to receive tiered royalties beginning in the low double-digits, and up to 20% on sales of
OV935, if approved and commercialized.

We expect to close the Takeda License and Termination Agreement in the first half of 2021, subject to the satisfaction of customary closing conditions, including
regulatory review by the appropriate regulatory agencies under the Hart-Scott-Rodino Antitrust Improvements Act of 1976, as amended (“HSR Act”). We cannot assure
you  that  such  closing  conditions  will  be  satisfied  or  that  the  post-closing  filing  will  be  approved  by  the  appropriate  regulatory  agencies  under  the  HSR  Act.  If  the
regulatory agencies do not approve our filing, such agencies may request us to rescind the transactions related to the Takeda License and Termination Agreement. If we
fail to close the Takeda License and Termination Agreement, then we will not be entitled to any of the payments described above, and the current terms of collaboration
and related risks will remain in effect and our business and financial condition may be harmed.

Risks Related to Our Business Operations, Employee Matters and Managing Growth

COVID-19 could adversely impact our business, including our clinical trials and access to capital.

The ongoing COVID-19 pandemic has resulted in travel and other restrictions in order to reduce the spread of the disease, including state and local orders across
the  country,  which,  among  other  things,  direct  individuals  to  shelter  at  their  places  of  residence,  direct  businesses  and  governmental  agencies  to  cease  non-essential
operations at physical locations, prohibit certain non-essential gatherings, and order cessation of non-essential travel. In response to these public health directives and
orders, we have implemented work-from-home policies for all employees. Our current plans to return to the office remain fluid as federal, state and local guidelines, rules
and regulations continue to evolve. The effects of the executive orders, the shelter-in-place orders and our work-from-home policies may negatively impact productivity,
disrupt our business and delay our clinical programs and timelines, the magnitude of which will depend, in part, on the length and severity of the restrictions and other
limitations  on  our  ability  to  conduct  our  business  in  the  ordinary  course.  These  and  similar,  and  perhaps  more  severe,  disruptions  in  our  operations  could  negatively
impact our business, operating results and financial condition.

Quarantines, shelter-in-place and similar government orders related to COVID-19 may adversely impact our business operations and the business operations of
our contract research organizations conducting our clinical trials and our third-party manufacturing facilities in the United States and other countries. In particular, some
of  our  third-party  manufacturers  which  we  use  for  the  supply  of  materials  for  product  candidates  or  other  materials  necessary  to  manufacture  product  to  conduct
preclinical studies and clinical trials are located in countries affected by COVID-19, and should they experience disruptions, such as temporary closures or

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suspension of services, we would likely experience delays in advancing these tests and trials. Currently, we expect no material impact on the clinical supply of any of our
product candidates.

In addition, our clinical trials may be affected by the COVID-19 pandemic.

Clinical site initiation and patient enrollment may be delayed due to prioritization of hospital resources toward the COVID-19 pandemic. Some patients may not
be willing or able to comply with clinical trial protocols if quarantines impede patient movement or interrupt healthcare services. Similarly, our ability to recruit and retain
patients  and  principal  investigators  and  site  staff  who,  as  healthcare  providers,  may  have  heightened  exposure  to  COVID-19  and  adversely  impact  our  clinical  trial
operations. As a result of the COVID-19 pandemic, we have faced and may continue to face delays in meeting our anticipated timelines for our ongoing and planned
clinical trials.

The spread of COVID-19, which has caused a broad impact globally, may materially affect us economically. While the potential economic impact brought by,
and the duration of, COVID-19 may be difficult to assess or predict, a widespread pandemic could result in significant disruption of global financial markets, reducing our
ability to access capital, which could in the future negatively affect our liquidity. In addition, a recession or market correction resulting from the spread of COVID-19
could materially affect our business and the value of our common stock.

The global pandemic of COVID-19 continues to rapidly evolve. The extent to which the COVID-19 pandemic impacts our business, our clinical development
and regulatory efforts will depend on future developments that are highly uncertain and cannot be predicted with confidence, such as the duration of the outbreak, travel
restrictions, quarantines, social distancing requirements and business closures in the United States and other countries, and business disruptions, and the effectiveness of
actions taken in the United States and other countries to contain and treat the disease.  Accordingly, we do not yet know the full extent of potential delays or impacts on
our business, our clinical and regulatory activities, healthcare systems or the global economy as a whole.  However, these impacts could adversely affect our business,
financial condition, results of operations and growth prospects.

In addition, to the extent the ongoing COVID-19 pandemic adversely affects our business and results of operations, it may also have the effect of heightening

many of the other risks and uncertainties described in this ‘‘Risk Factors’’ section.

We are highly dependent on the services of our senior management team, including our Chairman and Chief Executive Officer, Dr. Jeremy Levin, and if we are not
able to retain these members of our management team or recruit and retain additional management, clinical and scientific personnel, our business will be harmed.

We are highly dependent on our senior management team, including our Chairman and Chief Executive Officer, Dr. Levin. The employment agreements we
have with these officers do not prevent such persons from terminating their employment with us at any time. The loss of the services of any of these persons could impede
the achievement of our research, development and commercialization objectives.

In addition, we are dependent on our continued ability to attract, retain and motivate highly qualified additional management, clinical and scientific personnel. If
we are not able to retain our management and to attract, on acceptable terms, additional qualified personnel necessary for the continued development of our business, we
may not be able to sustain our operations or grow.  This risk may be further amplified given the particularly competitive hiring market in New York City, the location of
our corporate headquarters.

We  may  not  be  able  to  attract  or  retain  qualified  personnel  in  the  future  due  to  the  intense  competition  for  qualified  personnel  among  biotechnology,
pharmaceutical and other businesses. Many of the other pharmaceutical companies that we compete against for qualified personnel and consultants have greater financial
and other resources, different risk profiles and a longer history in the industry than we do. They also may provide more diverse opportunities and better chances for career
advancement. Some of these characteristics may be more appealing to high-quality candidates and consultants than what we have to offer. If we are unable to continue to
attract, retain and motivate high-quality personnel and consultants to accomplish our business objectives, the rate and success at which we can discover and develop drug
candidates and our business will be limited and we may experience constraints on our development objectives.

Our  future  performance  will  also  depend,  in  part,  on  our  ability  to  successfully  integrate  newly  hired  executive  officers  into  our  management  team  and  our
ability to develop an effective working relationship among senior management. Our failure to integrate these individuals and create effective working relationships among
them  and  other  members  of  management  could  result  in  inefficiencies  in  the  development  and  commercialization  of  our  drug  candidates,  harming  future  regulatory
approvals, sales of our drug candidates and our results of operations. Additionally, we do not currently maintain “key person” life insurance on the lives of our executives
or any of our employees.

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We may need to expand our organization, and we may experience difficulties in managing this growth, which could disrupt our operations.

As of December 31, 2020, we had 67 full-time employees. As our development and commercialization plans and strategies develop, we expect to need additional
managerial, operational, sales, marketing, financial, legal and other resources. Our management may need to divert a disproportionate amount of its attention away from
our day-to-day operations and devote a substantial amount of time to managing these growth activities. We may not be able to effectively manage the expansion of our
operations, which may result in weaknesses in our infrastructure, operational inefficiencies, loss of business opportunities, loss of employees and reduced productivity
among  remaining  employees.  Our  expected  growth  could  require  significant  capital  expenditures  and  may  divert  financial  resources  from  other  projects,  such  as  the
development of our current and potential future drug candidates. If our management is unable to effectively manage our growth, our expenses may increase more than
expected, our ability to generate and grow revenue could be reduced and we may not be able to implement our business strategy. Our future financial performance, our
ability to commercialize drug candidates, develop a scalable infrastructure and compete effectively will depend, in part, on our ability to effectively manage any future
growth.

Our employees, principal investigators, consultants and commercial partners may engage in misconduct or other improper activities, including non-compliance with
regulatory standards and requirements and insider trading.

We  are  exposed  to  the  risk  that  our  employees,  consultants,  distributors,  and  collaborators  may  engage  in  fraudulent  or  illegal  activity.  Misconduct  by  these
parties  could  include  intentional,  reckless  or  negligent  conduct  or  disclosure  of  unauthorized  activities  to  us  that  violates  the  regulations  of  the  FDA  and  non-U.S.
regulators, including those laws requiring the reporting of true, complete and accurate information to such regulators, manufacturing standards, healthcare fraud and abuse
laws and regulations in the United States and abroad or laws that require the true, complete and accurate reporting of financial information or data. In particular, sales,
marketing and business arrangements in the healthcare industry, including the sale of pharmaceuticals, are subject to extensive laws and regulations intended to prevent
fraud, misconduct, kickbacks, self-dealing and other abusive practices. These laws and regulations may restrict or prohibit a wide range of pricing, discounting, marketing
and  promotion,  sales  commission,  customer  incentive  programs  and  other  business  arrangements.  It  is  not  always  possible  to  identify  and  deter  misconduct  by  our
employees and other third parties, and the precautions we take to detect and prevent this activity may not be effective in controlling unknown or unmanaged risks or
losses or in protecting us from governmental investigations or other actions or lawsuits stemming from a failure to comply with these laws or regulations. Further, because
of the work from home policies we implemented due to COVID-19, information that is normally protected, including company confidential information, may be less
secure.  If  actions  are  instituted  against  us  and  we  are  not  successful  in  defending  ourselves  or  asserting  our  rights,  those  actions  could  result  in  the  imposition  of
significant fines or other sanctions, including the imposition of civil, criminal and administrative penalties, damages, monetary fines, imprisonment, possible exclusion
from  participation  in  Medicare,  Medicaid  and  other  federal  healthcare  programs,  additional  reporting  obligations  and  oversight  if  we  become  subject  to  a  corporate
integrity agreement or other agreement to resolve allegations of non-compliance with these laws, contractual damages, reputational harm, diminished profits and future
earnings  and  curtailment  of  operations,  any  of  which  could  adversely  affect  our  ability  to  operate  our  business  and  our  results  of  operations.  Whether  or  not  we  are
successful in defending against such actions or investigations, we could incur substantial costs, including legal fees, and divert the attention of management in defending
ourselves against any of these claims or investigations.

Significant disruptions of our information technology systems or data security incidents could result in significant financial, legal, regulatory, business and
reputational harm to us.

We  are  increasingly  dependent  on  information  technology  systems  and  infrastructure,  including  mobile  technologies,  to  operate  our  business.  In  the  ordinary
course of our business, we collect, store, process and transmit large amounts of sensitive information, including intellectual property, proprietary business information,
personal information and other confidential information. It is critical that we do so in a secure manner to maintain the confidentiality, integrity and availability of such
sensitive information. We have also outsourced elements of our operations (including elements of our information technology infrastructure) to third parties, and as a
result, we manage a number of third-party vendors who may or could have access to our computer networks or our confidential information. In addition, many of those
third  parties  in  turn  subcontract  or  outsource  some  of  their  responsibilities  to  third  parties.  While  all  information  technology  operations  are  inherently  vulnerable  to
inadvertent  or  intentional  security  breaches,  incidents,  attacks  and  exposures,  the  accessibility  and  distributed  nature  of  our  information  technology  systems,  and  the
sensitive information stored on those systems, make such systems potentially vulnerable to unintentional or malicious, internal and external attacks on our technology
environment. In addition, due to the COVID-19 pandemic, we have enabled all of our employees to work remotely, which may make us more vulnerable to cyberattacks.
Potential vulnerabilities can be exploited from inadvertent or intentional actions of our employees, third-party vendors, business partners, or by malicious third parties.
Attacks of this nature are increasing in their frequency, levels of persistence, sophistication and intensity, and are being conducted by sophisticated and organized groups
and individuals with a wide range of motives (including, but not limited to, industrial espionage) and expertise, including organized criminal groups, “hacktivists,” nation
states and others. In addition to the extraction of sensitive information, such attacks could include the deployment of harmful malware, ransomware, denial-of-service
attacks, social engineering and other means to affect service reliability and threaten the

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confidentiality, integrity and availability of information. In addition, the prevalent use of mobile devices increases the risk of data security incidents.

Significant disruptions of our, our third-party vendors’ and/or business partners’ information technology systems or other similar data security incidents could
adversely  affect  our  business  operations  and/or  result  in  the  loss,  misappropriation,  and/or  unauthorized  access,  use  or  disclosure  of,  or  the  prevention  of  access  to,
sensitive  information,  which  could  result  in  financial,  legal,  regulatory,  business  and  reputational  harm  to  us.  In  addition,  information  technology  system  disruptions,
whether  from  attacks  on  our  technology  environment  or  from  computer  viruses,  natural  disasters,  terrorism,  war  and  telecommunication  and  electrical  failures,  could
result in a material disruption of our development programs and our business operations. For example, the loss of clinical trial data from completed or future clinical trials
could result in delays in our regulatory approval efforts and significantly increase our costs to recover or reproduce the data.

There is no way of knowing with certainty whether we have experienced any data security incidents that have not been discovered. While we have no reason to
believe this to be the case, attackers have become very sophisticated in the way they conceal access to systems, and many companies that have been attacked are not
aware  that  they  have  been  attacked.  Any  event  that  leads  to  unauthorized  access,  use  or  disclosure  of  personal  information,  including  but  not  limited  to  personal
information  regarding  our  patients  or  employees,  could  disrupt  our  business,  harm  our  reputation,  compel  us  to  comply  with  applicable  federal  and/or  state  breach
notification  laws  and  foreign  law  equivalents,  subject  us  to  time  consuming,  distracting  and  expensive  litigation,  regulatory  investigation  and  oversight,  mandatory
corrective  action,  require  us  to  verify  the  correctness  of  database  contents,  or  otherwise  subject  us  to  liability  under  laws,  regulations  and  contractual  obligations,
including  those  that  protect  the  privacy  and  security  of  personal  information.  This  could  result  in  increased  costs  to  us,  and  result  in  significant  legal  and  financial
exposure and/or reputational harm. In addition, any failure or perceived failure by us or our vendors or business partners to comply with our privacy, confidentiality or
data security-related legal or other obligations to third parties, or any further security incidents or other inappropriate access events that result in the unauthorized access,
release  or  transfer  of  sensitive  information,  which  could  include  personally  identifiable  information,  may  result  in  governmental  investigations,  enforcement  actions,
regulatory fines, litigation, or public statements against us by advocacy groups or others, and could cause third parties, including clinical sites, regulators or current and
potential partners, to lose trust in us or we could be subject to claims by third parties that we have breached our privacy- or confidentiality-related obligations, which
could materially and adversely affect our business and prospects. Moreover, data security incidents and other inappropriate access can be difficult to detect, and any delay
in  identifying  them  may  lead  to  increased  harm  of  the  type  described  above.  While  we  have  implemented  security  measures  intended  to  protect  our  information
technology systems and infrastructure, there can be no assurance that such measures will successfully prevent service interruptions or security incidents.

We may be subject to numerous and varying privacy and security laws, and our failure to comply could result in penalties and reputational damage.

We  are  subject  to  laws  and  regulations  covering  data  privacy  and  the  protection  of  personal  information  including  health  information.  The  legislative  and
regulatory landscape for privacy and data protection continues to evolve, and there has been an increasing focus on privacy and data protection issues which may affect
our business. In the U.S., we may be subject to state security breach notification laws, state health information privacy laws and federal and state consumer protections
laws which impose requirements for the collection, use, disclosure and transmission of personal information. Each of these laws is subject to varying interpretations by
courts and government agencies, creating complex compliance issues for us. If we fail to comply with applicable laws and regulations we could be subject to penalties or
sanctions, including criminal penalties if we knowingly obtain individually identifiable health information from a covered entity in a manner that is not authorized or
permitted by HIPAA or for aiding and abetting the violation of HIPAA.

Numerous other countries have, or are developing, laws governing the collection, use and transmission of personal information as well. EU member states and
other  jurisdictions  have  adopted  data  protection  laws  and  regulations,  which  impose  significant  compliance  obligations.  For  example,  in  May  2016,  the  EU  formally
adopted  the  General  Data  Protection  Regulation,  or  GDPR,  which  applies  to  all  EU  member  states  as  of  May  25,  2018  and  replaces  the  former  EU  Data  Protection
Directive. The regulation introduces new data protection requirements in the EU and imposes substantial fines for breaches of the data protection rules. The GDPR must
be  implemented  into  national  laws  by  the  EU  member  states  imposes  strict  obligations  and  restrictions  on  the  ability  to  collect,  analyze,  and  transfer  personal  data,
including  health  data  from  clinical  trials  and  adverse  event  reporting.  Data  protection  authorities  from  different  EU  member  states  have  interpreted  the  privacy  laws
differently, which adds to the complexity of processing personal data in the EU, and guidance on implementation and compliance practices are often updated or otherwise
revised. Any failure to comply with the rules arising from the GDPR and related national laws of EU member states could lead to government enforcement actions and
significant penalties against us, and adversely impact our operating results. The GDPR will increase our responsibility and liability in relation to personal data that we
process and we may be required to put in place additional mechanisms ensuring compliance with EU data protection rules.

Additionally, California enacted the California Consumer Privacy Act (the “CCPA”) legislation that has been dubbed the first “GDPR-like” law in the United

States. The CCPA gives California residents expanded rights to access and delete their personal

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information,  opt  out  of  certain  personal  information  sharing  and  receive  detailed  information  about  how  their  personal  information  is  used  by  requiring  covered
companies  to  provide  new  disclosures  to  California  consumers  (as  that  term  is  broadly  defined)  and  provide  such  consumers  new  ways  to  opt-out  of  certain  sales  of
personal information. The CCPA provides for civil penalties for violations, as well as a private right of action for data breaches that is expected to increase data breach
litigation.  The CCPA may increase our compliance costs and potential liability.

Risks Related to Being a Public Company

We are an “emerging growth company” and a “smaller reporting company” and the reduced disclosure requirements applicable to such companies may make our
common stock less attractive to investors.

We are an emerging growth company (“EGC”), as defined in the Jumpstart Our Business Startups Act of 2012 (the “JOBS Act”). We will remain an EGC until the
earlier of: (i) the last day of the fiscal year in which we have total annual gross revenues of $1.07  billion or more; (ii) December 31, 2022, the last day of the fiscal year
following the fifth anniversary of the date of the completion of our IPO; (iii) the date on which we have issued more than $1.0  billion in nonconvertible debt during the
previous three years; or (iv) the date on which we are deemed to be a large accelerated filer under the rules of the Securities and Exchange Commission (“SEC”). For so
long as we remain an EGC, we are permitted and intend to rely on exemptions from certain disclosure requirements that are applicable to other public companies that are
not emerging growth companies. These exemptions include:

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not being required to comply with the auditor attestation requirements of Section 404 of the Sarbanes-Oxley Act of 2002 (“Section 404”);

not being required to comply with any requirement that may be adopted by the Public Company Accounting Oversight Board regarding mandatory audit
firm rotation or a supplement to the auditor’s report providing additional information about the audit and the financial statements;

being  permitted  to  provide  only  two  years  of  audited  financial  statements,  in  addition  to  any  required  unaudited  interim  financial  statements,  with
correspondingly reduced “Management’s Discussion and Analysis of Financial Condition and Results of Operations” disclosure;

reduced disclosure obligations regarding executive compensation arrangements; and

exemptions from the requirements of holding a nonbinding advisory vote on executive compensation and stockholder approval of any golden parachute
payments not previously approved.

We currently intend to take advantage of some, but not all, of the reduced regulatory and reporting requirements that will be available to us so long as we qualify
as an EGC. For example, our independent registered public accounting firm will not be required to provide an attestation report on the effectiveness of our internal control
over financial reporting so long as we qualify as an EGC, which may increase the risk that material weaknesses or significant deficiencies in our internal control over
financial  reporting  go  undetected.  Likewise,  so  long  as  we  qualify  as  an  EGC,  we  may  elect  not  to  provide  you  with  certain  information,  including  certain  financial
information and certain information regarding compensation of our executive officers, that we would otherwise have been required to provide in filings we make with the
SEC, which may make it more difficult for investors and securities analysts to evaluate our company. We cannot predict if investors will find our common stock less
attractive because we may rely on these exemptions. If some investors find our common stock less attractive as a result, there may be a less active trading market for our
common stock, and our stock price may be more volatile and may decline.

In addition, the JOBS Act provides that an EGC may take advantage of an extended transition period for complying with new or revised accounting standards.
This allows an EGC to delay the adoption of certain accounting standards until those standards would otherwise apply to private companies. We have irrevocably elected
not to avail ourselves of this exemption from new or revised accounting standards and, therefore, we will be subject to the same new or revised accounting standards as
other public companies that are not an EGC. 

We are also a smaller reporting company as defined in the Exchange Act. We may continue to be a smaller reporting company even after we are no longer an
emerging growth company. We may take advantage of certain of the scaled disclosures available to smaller reporting companies and will be able to take advantage of
these scaled disclosures for so long as (i) our voting and non-voting common stock held by nonaffiliates is less than $250.0 million measured on the last business day of
our second fiscal quarter or (ii) our annual revenue is less than $100.0 million during the most recently completed fiscal year and our voting and non-voting common
stock held by non-affiliates is less than $700.0 million measured on the last business day of our second fiscal quarter.

We  will  continue  to  incur  increased  costs  as  a  result  of  operating  as  a  public  company,  and  our  management  will  devote  substantial  time  to  new  compliance
initiatives.

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As a public company, and particularly after we are no longer an EGC, we will incur significant legal, accounting and other expenses that we did not incur as a
private company. In addition, the Sarbanes-Oxley Act of 2002 and rules subsequently implemented by the SEC and The Nasdaq Stock Market LLC have imposed various
requirements  on  public  companies,  including  establishment  and  maintenance  of  effective  disclosure  and  financial  controls  and  corporate  governance  practices.  Our
management and other personnel devote a substantial amount of time to these and other compliance initiatives. Moreover, these rules and regulations will continue to
increase our legal and financial compliance costs and will make some activities more time-consuming and costly.

If we fail to maintain an effective system of internal control over financial reporting in the future, we may not be able to accurately report our financial condition,
results of operations or cash flows, which may adversely affect investor confidence in us and, as a result, the value of our common stock.

The Sarbanes-Oxley Act requires, among other things, that we maintain effective internal controls for financial reporting and disclosure controls and procedures.
We are required, under Section 404, to furnish a report by management on, among other things, the effectiveness of our internal control over financial reporting. This
assessment will need to include disclosure of any material weaknesses identified by our management in our internal control over financial reporting. A material weakness
is a deficiency, or combination of deficiencies, in internal control over financial reporting that results in more than a reasonable possibility that a material misstatement of
annual  or  interim  financial  statements  will  not  be  prevented  or  detected  on  a  timely  basis.  Section  404  also  generally  requires  an  attestation  from  our  independent
registered public accounting firm on the effectiveness of our internal control over financial reporting. However, for as long as we remain an emerging growth company as
defined in the JOBS Act, we intend to take advantage of the exemption permitting us not to comply with the independent registered public accounting firm attestation
requirement.

Our compliance with Section 404 will require that we incur substantial expense and expend significant management efforts. We currently do not have an internal
audit  group,  and  we  will  need  to  hire  additional  accounting  and  financial  staff  with  appropriate  public  company  experience  and  technical  accounting  knowledge  and
compile the system and process documentation necessary to perform the evaluation needed to comply with Section 404. We may not be able to complete our evaluation,
testing and any required remediation in a timely fashion. During the evaluation and testing process, if we identify one or more material weaknesses in our internal control
over financial reporting, we will be unable to assert that our internal control over financial reporting is effective. We cannot assure you that there will not be material
weaknesses or significant deficiencies in our internal control over financial reporting in the future. Any failure to maintain internal control over financial reporting could
severely inhibit our ability to accurately report our financial condition, results of operations or cash flows. If we are unable to conclude that our internal control over
financial reporting is effective, or if our independent registered public accounting firm determines we have a material weakness or significant deficiency in our internal
control over financial reporting once that firm begins its Section 404 reviews, we could lose investor confidence in the accuracy and completeness of our financial reports,
the  market  price  of  our  common  stock  could  decline,  and  we  could  be  subject  to  sanctions  or  investigations  by  The  Nasdaq  Stock  Market  LLC,  the  SEC  or  other
regulatory  authorities.  Failure  to  remedy  any  material  weakness  in  our  internal  control  over  financial  reporting,  or  to  implement  or  maintain  other  effective  control
systems required of public companies, could also restrict our future access to the capital markets.

Risks Related to the Ownership of Our Common Stock and Other General Matters

The market price of our common stock may be volatile and fluctuate substantially, which could result in substantial losses for our common stock.

The market price of our common stock is likely to be volatile. The stock market in general and the market for biopharmaceutical or pharmaceutical companies in
particular, has experienced extreme volatility that has often been unrelated to the operating performance of particular companies, including very recently in connection
with  the  ongoing  COVID-19  pandemic,  which  has  resulted  in  decreased  stock  prices  for  many  companies  notwithstanding  the  lack  of  a  fundamental  change  in  their
underlying  business  models  or  prospects.  Broad  market  and  industry  factors,  including  potentially  worsening  economic  conditions  and  other  adverse  effects  or
developments relating to the ongoing COVID-19 pandemic, may negatively affect the market price of our common stock, regardless of our actual operating performance.
As a result of this volatility, you may lose all or part of your investment in our common stock since you might be unable to sell your shares at or above the price you paid
for the shares. The market price for our common stock may be influenced by many factors, including:

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results of clinical trials of our current and any future drug candidates or those of our competitors;

the success of competitive drugs or therapies;

regulatory or legal developments in the United States and other countries;

developments or disputes concerning patent applications, issued patents or other proprietary rights;

the recruitment or departure of key personnel;

the level of expenses related to our current and any future drug candidates or clinical development programs;

the results of our efforts to discover, develop, acquire or in-license additional drug candidates;

actual or anticipated changes in estimates as to financial results, development timelines or recommendations by securities analysts;

our inability to obtain or delays in obtaining adequate drug supply for any approved drug or inability to do so at acceptable prices;

disputes  or  other  developments  relating  to  proprietary  rights,  including  patents,  litigation  matters  and  our  ability  to  obtain  patent  protection  for  our
technologies;

significant lawsuits, including patent or stockholder litigation;

variations in our financial results or those of companies that are perceived to be similar to us;

changes in the structure of healthcare payment systems;

market conditions in the pharmaceutical and biotechnology sectors;

general economic, industry and market conditions; and

the other factors described in this “Risk Factors” section.

In  addition,  in  the  past,  stockholders  have  initiated  class  action  lawsuits  against  companies  following  periods  of  volatility  in  the  market  prices  of  these

companies’ stock. Such litigation, if instituted against us, could cause us to incur substantial costs and divert management’s attention and resources.

There is no public market for our Series A convertible preferred stock.

There is no established public trading market for our Series A convertible preferred stock, and we do not expect a market to develop. In addition, we do not
intend to apply for listing of the Series A convertible preferred stock on any national securities exchange or other nationally recognized trading system. Without an active
market, the liquidity of the Series A convertible preferred stock will be limited.

We may sell additional equity or debt securities or enter into other arrangements to fund our operations, which may result in dilution to our stockholders and impose
restrictions or limitations on our business.

Until  we  can  generate  a  sufficient  amount  of  revenue  from  our  products,  if  ever,  we  expect  to  finance  future  cash  needs  through  public  or  private  equity  or
debt  offerings.  In  November  2020,  we  filed  a  shelf  registration  statement  on  Form  S-3  (Registration  No.  333-250054)  that  allows  us  to  sell  up  to  an  aggregate  of
$250.0  million  of  our  common  stock,  preferred  stock,  debt  securities  and/or  warrants  (the  “S-3  Registration  Statement”),  which  includes  a  prospectus  covering  the
issuance and sale of up to $75.0 million of common stock pursuant to an at-the-market (“ATM”) offering program. As of December 31, 2020, we had $250.0 million
available under our S-3 Registration Statement, including $75.0 million available pursuant to our ATM program. Financing activities may have an adverse impact on our
stockholders’ rights as well as on our operations, and such additional funding may not be available on reasonable terms, if at all. If we raise additional funds through the
issuance  of  additional  debt  or  equity  securities,  it  may  result  in  dilution  to  our  existing  stockholders  and/or  increased  fixed  payment  obligations.  Furthermore,  these
securities may have rights senior to those of our common stock and could contain covenants that would restrict our operations and potentially impair our competitiveness,
such as redeeming our shares, making investments, issuing additional equity, limitations on our ability to incur additional debt, limitations on our ability to acquire, sell or
license intellectual property rights and other operating restrictions that could adversely impact our ability to conduct our business. Additionally, if we seek funds through
arrangements with collaborative partners, these arrangements may require us to relinquish rights to some of our technologies or product candidates or otherwise agree to
terms unfavorable to us. Any of these events could significantly harm our business, financial condition and prospects.

You will be diluted by any conversions of outstanding Series A convertible preferred stock and exercises of outstanding options.

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As of December 31, 2020, we had outstanding options to purchase an aggregate of 10,403,420 shares of our common stock at a weighted average exercise price of
$5.26 per share and 3,250,000 shares of common stock issuable upon conversion of outstanding Series A convertible preferred stock for no additional consideration. Such
Series A convertible preferred stock is convertible any time at the option of the holder thereof subject to the beneficial ownership limitations described in Note 6 to the
financial statements contained in this Annual Report on Form 10-K. The exercise of such options and conversion of the Series A convertible preferred stock for shares of
our common stock will result in further dilution of your investment and could negatively affect the market price of our common stock. In addition, you may experience
further dilution if we issue common stock, or securities convertible into common stock, in the future. As a result of this dilution, you may receive significantly less than
the full purchase price you paid for the shares in the event of liquidation.

Concentration of ownership of our common stock among our executive officers, directors and principal stockholders may prevent new investors from influencing
significant corporate decisions.

Based upon our shares of our common stock outstanding as of March 8, 2021, our executive officers, directors and stockholders who owned more than 5% of

our outstanding common stock, in the aggregate, beneficially own shares representing approximately 35.54% of our outstanding common stock.

Takeda,  a  greater  than  5%  holder,  may  receive  additional  securities  upon  the  achievement  of  certain  development,  commercial  and  regulatory  milestones
pursuant to the Takeda collaboration. Specifically, we will be obligated to issue additional securities to Takeda equal to the lesser of 8% of our outstanding capital stock or
$50.0 million unless certain events occur, and may issue, at our discretion, additional securities to Takeda upon the achievement of other milestones. Further, pursuant to
the Series B-1 preferred stock purchase agreement entered into with Takeda in January 2017, or the Takeda stock purchase agreement, Takeda has agreed to, among other
things, (i) a standstill provision, (ii) restrictions on its ability to sell or otherwise transfer it shares of our stock, (iii) vote its shares on certain matters in accordance with
the holders of a majority of shares of our common stock and (iv) restrictions on the percentage of our outstanding common stock it may own.

If our executive officers, directors and stockholders who owned more than 5% of our outstanding common stock acted together, they may be able to significantly
influence  all  matters  requiring  stockholder  approval,  including  the  election  and  removal  of  directors  and  approval  of  any  merger,  consolidation  or  sale  of  all  or
substantially  all  of  our  assets.  The  concentration  of  voting  power,  Takeda  standstill  provisions,  voting  obligations  and  transfer  restrictions  could  delay  or  prevent  an
acquisition of our company on terms that other stockholders may desire or result in the management of our company in ways with which other stockholders disagree with.

If securities analysts do not publish research or reports about our business or if they publish negative evaluations of our stock, the price of our stock could decline.

The trading market for our common stock relies, in part, on the research and reports that industry or financial analysts publish about us or our business.  We do
currently have research coverage offered by several industry or financial analysts. If one or more of the analysts covering our business downgrade their evaluations of our
stock, the price of our stock could decline. If one or more of these analysts cease to cover our stock, we could lose visibility in the market for our stock, which in turn
could cause our stock price to decline.

Because we do not anticipate paying any cash dividends on our capital stock in the foreseeable future, capital appreciation, if any, will be your sole source of gain.

We have never declared or paid cash dividends on our capital stock. We currently intend to retain all of our future earnings, if any, to finance the growth and
development of our business. In addition, the terms of any future debt agreements may preclude us from paying dividends. As a result, capital appreciation, if any, of our
common stock will be your sole source of gain for the foreseeable future.

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Provisions in our corporate charter documents and under Delaware law could make an acquisition of us, which may be beneficial to our stockholders, more difficult
and may prevent attempts by our stockholders to replace or remove our current management.

Provisions in our corporate charter and our bylaws may discourage, delay or prevent a merger, acquisition or other change in control of us that stockholders may
consider favorable, including transactions in which you might otherwise receive a premium for your shares. These provisions also could limit the price that investors
might  be  willing  to  pay  in  the  future  for  shares  of  our  common  stock,  thereby  depressing  the  market  price  of  our  common  stock.  In  addition,  because  our  board  of
directors is responsible for appointing the members of our management team, these provisions may frustrate or prevent any attempts by our stockholders to replace or
remove our current management by making it more difficult for stockholders to replace members of our board of directors. Among other things, these provisions:

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establish a classified board of directors such that not all members of the board are elected at one time;

allow the authorized number of our directors to be changed only by resolution of our board of directors;

limit the manner in which stockholders can remove directors from the board;

establish advance notice requirements for stockholder proposals that can be acted on at stockholder meetings and nominations to our board of directors;

require that stockholder actions must be effected at a duly called stockholder meeting and prohibit actions by our stockholders by written consent;

limit who may call stockholder meetings;

authorize our board of directors to issue preferred stock without stockholder approval, which could be used to institute a stockholder rights plan, or so-
called “poison pill,” that would work to dilute the stock ownership of a potential hostile acquirer, effectively preventing acquisitions that have not been
approved by our board of directors; and

require the approval of the holders of at least 66 2/3% of the votes that all our stockholders would be entitled to cast to amend or repeal certain provisions
of our charter or bylaws.

Moreover,  because  we  are  incorporated  in  Delaware,  we  are  governed  by  the  provisions  of  Section  203  of  the  Delaware  General  Corporation  Law,  which
prohibits  a  person  who  owns  in  excess  of  15%  of  our  outstanding  voting  stock  from  merging  or  combining  with  us  for  a  period  of  three  years  after  the  date  of  the
transaction in which the person acquired in excess of 15% of our outstanding voting stock, unless the merger or combination is approved in a prescribed manner.

Additionally, the Takeda standstill provisions and transfer restrictions in the Takeda Stock Purchase Agreement may delay or prevent a merger, acquisition or

other change in control of us that stockholders may consider favorable, including transactions in which you might otherwise receive a premium for your shares.

We may be subject to securities litigation, which is expensive and could divert management attention.

The market price of our common stock may be volatile.  For example, on August 25, 2020, we announced the topline results of our ELEKTRA clinical trial, and
our stock experienced a material decline.  In the past, companies that have experienced volatility in the market price of their stock have been subject to securities class
action litigation. We may be the target of this type of litigation in the future. Securities litigation against us could result in substantial costs and divert our management’s
attention from other business concerns, which could seriously harm our business.

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Some  provisions  of  our  charter  documents  and  Delaware  law  may  have  anti-takeover  effects  that  could  discourage  an  acquisition  of  us  by  others,  even  if  an
acquisition would benefit our stockholders and may prevent attempts by our stockholders to replace or remove our current management.

Provisions in our amended and restated certificate of incorporation and amended and restated bylaws, as well as provisions of Delaware law, could make it more
difficult for a third party to acquire us or increase the cost of acquiring us, even if doing so would benefit our stockholders, or remove our current management. These
provisions include:

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authorizing the issuance of “blank check” preferred stock, the terms of which we may establish and shares of which we may issue without stockholder
approval;

prohibiting cumulative voting in the election of directors, which would otherwise allow for less than a majority of stockholders to elect director candidates;

prohibiting stockholder action by written consent, thereby requiring all stockholder actions to be taken at a meeting of our stockholders;

eliminating the ability of stockholders to call a special meeting of stockholders; and

establishing  advance  notice  requirements  for  nominations  for  election  to  the  board  of  directors  or  for  proposing  matters  that  can  be  acted  upon  at
stockholder meetings.

These  provisions  may  frustrate  or  prevent  any  attempts  by  our  stockholders  to  replace  or  remove  our  current  management  by  making  it  more  difficult  for
stockholders  to  replace  members  of  our  board  of  directors,  who  are  responsible  for  appointing  the  members  of  our  management.  Because  we  are  incorporated  in
Delaware, we are governed by the provisions of Section 203 of the Delaware General Corporation Law (the “DGCL”), which may discourage, delay or prevent someone
from acquiring us or merging with us whether or not it is desired by or beneficial to our stockholders. Under the DGCL, a corporation may not, in general, engage in a
business combination with any holder of 15% or more of its capital stock unless the holder has held the stock for three years or, among other things, the board of directors
has approved the transaction. Any provision of our amended and restated certificate of incorporation or amended and restated bylaws or Delaware law that has the effect
of delaying or deterring a change of control could limit the opportunity for our stockholders to receive a premium for their shares of our common stock and could also
affect the price that some investors are willing to pay for our common stock.

If we engage in future acquisitions or strategic partnerships, this may increase our capital requirements, dilute our stockholders, cause us to incur debt or assume
contingent liabilities and subject us to other risks.

Our business plan is to continue to evaluate various acquisitions and strategic partnerships, including licensing or acquiring complementary drugs, intellectual

property rights, technologies, or businesses. Any potential acquisition or strategic partnership may entail numerous risks, including:

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increased operating expenses and cash requirements;

the assumption of additional indebtedness or contingent liabilities;

assimilation of operations, intellectual property and drugs of an acquired company, including difficulties associated with integrating new personnel;

the diversion of our management’s attention from our existing drug programs and initiatives in pursuing such a strategic partnership, merger or acquisition;

retention of key employees, the loss of key personnel, and uncertainties in our ability to maintain key business relationships;

risks and uncertainties associated with the other party to such a transaction, including the prospects of that party and their existing drugs or drug candidates
and regulatory approvals; and

our inability to generate revenue from acquired technology and/or drugs sufficient to meet our objectives in undertaking the acquisition or even to offset
the associated acquisition and maintenance costs.

In addition, if we engage in future acquisitions or strategic partnerships, we may issue dilutive securities, assume or incur debt obligations, incur large one-time
expenses  and  acquire  intangible  assets  that  could  result  in  significant  future  amortization  expense.  Moreover,  we  may  not  be  able  to  locate  suitable  acquisition
opportunities and this inability could impair our ability to grow or obtain access to technology or drugs that may be important to the development of our business.

Sales of a substantial number of shares of our common stock in the public market could cause the market price of our common stock to drop significantly.

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Sales of a substantial number of shares of our common stock in the public market could occur at any time. These sales, or the perception in the market that the
holders of a large number of shares intend to sell shares, could reduce the market price of our common stock. Some of the holders of our securities have rights, subject to
certain conditions, to require us to file registration statements covering their shares or to include their shares in registration statements that we may file for ourselves or
other stockholders. Registration of these shares would result in the shares becoming freely tradable without restriction under the Securities Act except for shares held by
our affiliates. Any sales of securities by these stockholders could have a material adverse effect on the trading price of our common stock.

Item 1B. Unresolved Staff Comments

None.

Item 2. Properties

We  lease  the  space  for  our  principal  executive  offices,  which  are  located  at  1460  Broadway,  New  York,  New  York,  on  a  monthly  basis.  We  believe  that  our

facilities are adequate to meet our current needs.

Item 3. Legal Proceedings

We are not currently subject to any material legal proceedings.

Item 4. Mine Safety Disclosures

Not applicable.

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PART II

Item 5. Market for Registrant’s Common Equity, Related Stockholder Matters and Issuer Purchases of Equity Securities

Market Information

Our common stock began trading on The Nasdaq Global Select Market on May 5, 2017, under the symbol “OVID.”

Comparative Stock Performance Graph

The following performance graph and related information shall not be deemed “soliciting material” or to be “filed” with the SEC, nor shall such information be
incorporated  by  reference  into  any  future  filing  under  the  Securities  Act  or  Exchange  Act.  The  following  graph  shows  a  comparison  from  May  5,  2017  (the  date  our
common stock commenced trading on the Nasdaq Global Select Market) through December 31, 2020, of the cumulative total return for our common stock, the Nasdaq
Composite Index, and the Nasdaq Biotechnology.

The graph assumes an initial investment of $100 on May 5, 2017. The comparisons in the graph are not intended to forecast or be indicative of possible future

performance of our common stock.

Holders of Record

As of March 8, 2021, we had approximately 11 holders of record of our common stock. Certain shares are held in “street” name and accordingly, the number of
beneficial owners of such shares is not known or included in the foregoing number. This number of holders of record also does not include stockholders whose shares
may be held in trust by other entities.

Dividend Policy

We have never declared or paid any cash dividends on our common stock. We currently intend to retain future earnings to fund the development and growth of our
business. We do not expect to pay any cash dividends in the foreseeable future. Any future determination to pay dividends will be made at the discretion of our board of
directors  and  will  depend  on  then-existing  conditions,  including  our  financial  conditions,  operating  results,  contractual  restrictions,  capital  requirements,  business
prospects and other factors our board of directors may deem relevant.

Recent Sales of Unregistered Securities

None.

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Item 6.  Selected Financial Data

This item is no longer required as we have elected to early adopt the changes to Item 301 of Regulation S-K contained in SEC Release No. 33-10890.

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Item 7. Management’s Discussion and Analysis of Financial Condition and Results of Operations

The following discussion and analysis should be read in conjunction with our financial statements and related notes included elsewhere in this Annual Report on
Form 10-K. This discussion and analysis and other parts of this Annual Report on Form 10-K contain forward-looking statements based upon current beliefs, plans and
expectations that involve risks, uncertainties and assumptions, such as statements regarding our plans, objectives, expectations, intentions and projections. Our actual
results and the timing of selected events could differ materially from those anticipated in these forward-looking statements as a result of several factors, including those
set forth under “Risk Factors” and elsewhere in this Annual Report on Form 10-K. You should carefully read the “Risk Factors” section of this Annual Report on Form
10-K  to  gain  an  understanding  of  the  important  factors  that  could  cause  actual  results  to  differ  materially  from  our  forward-looking  statements.  Please  also  see  the
section entitled “Special Note Regarding Forward-Looking Statements.”

Overview

We are a biopharmaceutical company focused on developing impactful medicines for patients and families living with rare neurological disorders. We believe
these disorders represent an attractive area for drug development as the understanding of the underlying biology has grown meaningfully over the last few years and today
represent  a  substantial  opportunity  medically  and  commercially.  Based  on  the  rapid  increase  in  scientific  understanding  of  the  role  of  genetics  and  key  biological
pathways relevant to diseases of the brain, we aim to identify, discover and develop novel compounds for the treatment of rare neurological disorders. We have built a
deep knowledge of such diseases, how to treat them and how to develop the clinically meaningful endpoints required for development of a compound in these disorders.
As  a  result  of  this  knowledge,  we  have  developed  a  pipeline  of  first-in-class  compounds  and  programs  and  have  demonstrated  our  model  by  progressing  compounds
through  to  late-stage  development.  We  continue  to  execute  on  our  strategy  to  build  this  pipeline  by  discovering  in-licensing  and  collaborating  with  leading
biopharmaceutical companies and academic institutions.

Our latest pipeline includes two late-stage programs and several earlier stage programs.

Since  our  inception  in  April  2014,  we  have  devoted  substantially  all  of  our  efforts  to  organizing  and  planning  our  business,  building  our  management  and

technical team, acquiring operating assets and raising capital.

During the year ended December 31, 2020, we generated $12.6 million of license and other revenue through our Collaboration and License Agreement, or the
Angelini License Agreement, with Angelini Pharma Rare Diseases AG, or Angelini, and have otherwise funded our business primarily through the sale of our capital
stock.  Through  December  31,  2020,  we  have  raised  net  proceeds  of  $275.4  million  from  the  sale  of  our  convertible  preferred  stock  and  our  common  stock.  As  of
December 31, 2020, we had $72.0 million in cash and cash equivalents. We recorded net losses of $81.0 million and $60.5 million for the years ended December 31, 2020
and 2019, respectively. As of December 31, 2020, we had an accumulated deficit of $294.2 million.

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We expect to continue to incur significant expenses and increasing operating losses for at least the next several years. Our net losses may fluctuate significantly
from  period  to  period,  depending  on  the  timing  of  our  planned  clinical  trials  and  expenditures  on  our  other  research  and  development  and  commercial  development
activities. We expect our expenses will increase substantially over time as we:

•

•

•

•

•

•

•

•

continue the ongoing and planned preclinical and clinical development of our drug candidates;

build a portfolio of drug candidates through the development, acquisition or in-license of drugs, drug candidates or technologies;

initiate preclinical studies and clinical trials for any additional drug candidates that we may pursue in the future;

seek marketing approvals for our current and future drug candidates that successfully complete clinical trials;

establish a sales, marketing and distribution infrastructure to commercialize any drug candidate for which we may obtain marketing approval;

develop, maintain, expand and protect our intellectual property portfolio;

implement operational, financial and management systems; and

attract, hire and retain additional administrative, clinical, regulatory, manufacturing, commercial and scientific personnel.

Recent Developments

Royalty, License and Termination Agreement with Takeda

On March 2, 2021, we entered into a royalty, license and termination agreement, or the Takeda License and Termination Agreement, with Takeda, relating to the
Takeda collaboration agreement described above in Item 1. Business section. Under the terms of the Takeda License and Termination Agreement, upon closing of the
transaction, the Takeda collaboration agreement will be terminated by mutual agreement, and Takeda will secure rights to our 50% global share in soticlestat, and an
exclusive  license  under  our  relevant  intellectual  property  rights,  in  exchange  for  an  upfront  payment,  development  and  commercial  milestone  payments,  and
royalties.  Takeda will assume all responsibility for, and costs of, both development and commercialization of soticlestat following closing. At closing, we will receive an
upfront payment of $196.0 million and are eligible to receive up to an additional $660.0 million in development, regulatory and sales milestones.  In addition, if soticlestat
achieves regulatory approval, we will receive tiered royalties on net sales of soticlestat at percentages ranging from the low double-digits up to 20%, subject to standard
reductions  in  certain  circumstances.    Royalties  are  payable  on  a  country-by-country  and  product-by-product  basis  during  the  period  beginning  on  the  date  of  the  first
commercial sale of such product in such country and ending on the later to occur of the expiration of patent rights covering the product in such country and a specified
anniversary  of  such  first  commercial  sale.  The  Takeda  License  and  Termination  Agreement  will  remain  in  effect  until  Takeda’s  cessation  of  commercialization  of
soticlestat.    We  expect  to  close  the  Takeda  License  and  Termination  Agreement  in  the  first  half  of  2021,  subject  to  the  satisfaction  of  customary  closing  conditions,
including regulatory review by the appropriate regulatory agencies under the Hart-Scott-Rodino Antitrust Improvements Act of 1976, as amended. The Takeda License
and Termination Agreement may be terminated upon the mutual agreement of the parties, or by either Takeda or the Company, if the closing has not occurred on or before
May 14, 2021. 

COVID-19 Update

We  have  implemented  business  continuity  plans  designed  to  address  and  mitigate  the  impact  of  the  ongoing  COVID-19  pandemic  on  our  employees  and  our
business. We continue to operate normally with the exception of enabling all of our employees to work productively at home and abiding by travel restrictions issued by
federal, state and local governments. Our current plans to return to the office remain fluid as federal, state and local guidelines, rules and regulations continue to evolve.

Financial Operations Overview

Revenue

We have generated limited revenue under the Angelini License Agreement and expect to recognize additional revenue as we satisfy our performance obligations.
We have not generated any revenue from commercial drug sales and do not expect to generate any further revenue unless or until we obtain regulatory approval of and
commercialize one or more of our current or future drug candidates. In the future, we may also seek to generate revenue from a combination of research and development
payments, license fees and other upfront or milestone payments.

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Research and Development Expenses

Research and development expenses consist primarily of costs incurred for our research activities, including our product discovery efforts and the development of

our product candidates, which include, among other things:

•

•

•

•

•

•

•

employee-related expenses, including salaries, benefits and stock-based compensation expense;

fees paid to consultants for services directly related to our drug development and regulatory effort;

expenses  incurred  under  agreements  with  contract  research  organizations,  as  well  as  contract  manufacturing  organizations  and  consultants  that  conduct
preclinical studies and clinical trials;

costs associated with preclinical activities and development activities;

costs associated with technology and intellectual property licenses;

milestone payments and other costs under licensing agreements; and

depreciation expense for assets used in research and development activities.

Costs incurred in connection with research and development activities are expensed as incurred. Costs for certain development activities, such as clinical trials, are
recognized  based  on  an  evaluation  of  the  progress  to  completion  of  specific  tasks  using  data  such  as  patient  enrollment,  clinical  site  activations  or  other  information
provided to us by our vendors.

Research and development activities are and will continue to be central to our business model. We expect our research and development expenses to increase for
the foreseeable future as we advance our current and future drug candidates through preclinical studies and clinical trials. The process of conducting preclinical studies
and clinical trials necessary to obtain regulatory approval is costly and time-consuming. It is difficult to determine with certainty the duration and costs of any preclinical
study  or  clinical  trial  that  we  may  conduct.  The  duration,  costs  and  timing  of  clinical  trial  programs  and  development  of  our  current  and  future  drug  candidates  will
depend on a variety of factors that include, but are not limited to, the following:

•

•

•

•

•

•

•

•

•

•

•

number of clinical trials required for approval and any requirement for extension trials;

per patient trial costs;

number of patients who participate in the clinical trials;

number of sites included in the clinical trials;

countries in which the clinical trial is conducted;

length of time required to enroll eligible patients;

number of doses that patients receive;

drop-out or discontinuation rates of patients;

potential additional safety monitoring or other studies requested by regulatory agencies;

duration of patient follow-up; and

efficacy and safety profile of the drug candidate.

In addition, the probability of success for any of our current or future drug candidates will depend on numerous factors, including competition, manufacturing
capability and commercial viability. We will determine which programs to pursue and how much to fund each program in response to the scientific and clinical success of
each drug candidate, as well as an assessment of each drug candidate’s commercial potential.

General and Administrative Expenses

General and administrative expenses consist primarily of employee-related expenses, including salaries, benefits and stock-based compensation expense, related
to  our  executive,  finance,  business  development  and  support  functions.  Other  general  and  administrative  expenses  include  costs  associated  with  operating  as  a  public
company described below, travel expenses, conferences, professional fees for auditing, tax and legal services and facility-related costs.

Other Income, Net

Other income consists of interest income earned on our cash and cash equivalents maintained in money market funds and prior short-term investments that

were maintained in U.S. treasury notes.

64

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Results of Operations

Comparison of the Years Ended December 31, 2020 and 2019

The following table summarizes the results of our operations for the periods indicated:

Revenue:
    License and other revenue
Operating expenses:
    Research and development
    General and administrative
          Total operating expenses
Loss from operations
Other income, net
Net loss

  Year Ended     Year Ended        
  December 31,

    December 31,

2020

2019
(in thousands)

Change $

  $

12,617    $

-    $

12,617 

63,417     
30,631     
94,048     
(81,431)    
395     
(81,036)   $

42,157     
19,252     
61,409     
(61,409)    
948     
(60,461)   $

21,260 
11,379 
32,639 
(20,022)
(553)
(20,575)

  $

Revenue

Total revenue was $12.6 million for the year ended December 31, 2020 as a result of revenue recorded in connection with the Angelini License Agreement. We

did not generate any revenue during the year ended December 31, 2019.

Research and Development Expenses

Preclinical and development expenses
Payroll and payroll-related expenses
Other expenses
Total research and development

Year Ended
December 31,
2020

Year Ended
December 31,
2019
(in thousands)

Change $

  $

  $

43,612    $
15,439     
4,366     
63,417    $

27,034    $
11,496     
3,627     
42,157    $

16,578 
3,943 
739 
21,261

Research and development expenses were $63.4 million for the year ended December 31, 2020 compared to $42.2 million for the year ended December 31, 2019.
The increase of $21.3 million was primarily due to an increase in development activities related to our ongoing development programs. During the year ended December
31, 2020, total research and development expenses consisted of $43.6 million in preclinical and development expenses, including a credit of $0.7 million representing
costs  reimbursable  to  the  Company  from  Takeda  in  respect  of  the  Takeda  collaboration,  $15.4  million  in  payroll  and  payroll-related  expenses,  of  which  $2.8  million
related to stock-based compensation, and $4.4 million in other expenses.  During the year ended December 31, 2019, total research and development expenses consisted
of $27.0 million in preclinical and development expenses, including a credit of $4.7 million representing costs reimbursed to us from Takeda in respect of the Takeda
collaboration, $11.5 million in payroll and payroll-related expenses, of which $2.4 million related to stock-based compensation, and $3.6 million in other expenses.

General and Administrative Expenses

Payroll and payroll-related expenses
Legal and professional fees
General office expenses
Total general and administrative

Year Ended
December 31,
2020

Year Ended
December 31,
2019
(in thousands)

Change $

  $

  $

13,390    $
13,824     
3,417     
30,631    $

9,888    $
5,623     
3,741     
19,252    $

3,502 
8,201 
(324)
11,379

General and administrative expenses were $30.6 million for the year ended December 31, 2020 compared to $19.3 million for the year ended December 31, 2019.
The increase of $11.4 million primarily consisted of increases in legal fees, compliance and pre-commercialization expenses and professional fees of $8.2 million and
payroll-related expenses of $3.5 million.

Other Income, Net

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Other income includes interest income of $0.4 million for the year ended December 31, 2020 and $0.9 million for the year ended December 31, 2019.

Income Taxes

There was no provision for income taxes for the years ended December 31, 2020 and 2019 because we have historically incurred operating losses and we maintain
a full valuation allowance against our net deferred tax assets.  The valuation allowance was approximately $89.8 million and $76.5 million at December 31, 2020 and
2019, respectively.

Liquidity and Capital Resources

Overview

As of December 31, 2020, we had total cash, cash equivalents and short-term investments of $72.0 million as compared to $76.7 million as of December 31, 2019.

On  July  9,  2020,  we  entered  into  the  Angelini  License  Agreement  with  Angelini,  pursuant  to  which  we  granted  to  Angelini  exclusive  rights  to  develop  and
commercialize OV101 in the European Territory.  Under the Angelini License Agreement, Angelini made an upfront payment and a milestone payment related to the
transfer of a specified amount of compound and related information to the Company of $25.0 million during the year ended December 31, 2020. In addition, Angelini will
be  required  to  make  additional  milestone  payments  to  us  upon  the  completion  of  the  specified  components  of  the  technology  transfer,  and  achievement  of  specified
regulatory  milestones  for  OV101  in  Angelman  syndrome  of  up  to  $55.0  million  in  the  aggregate,  as  well  as  up  to  €162.5  million  ($199.9  million)  in  sales  milestone
payments for achievement of specified levels of net sales in the European Territory.  Angelini also will be required to pay tiered royalties on net sales by Angelini, its
affiliates or sublicensees at double-digit percentages above the teens, subject to certain standard reductions and offsets.

In  November  2020,  we  filed  a  new  shelf  registration  statement  on  Form  S-3  (Registration  No.  333-250054)  that  allows  us  to  sell  up  to  an  aggregate  of
$250.0  million  of  our  common  stock,  preferred  stock,  debt  securities  and/or  warrants  (the  “S-3  Registration  Statement”),  which  includes  a  prospectus  covering  the
issuance and sale of up to $75.0 million of common stock pursuant to an at-the-market (“ATM”) offering program. As of December 31, 2020, we had $250.0 million
available under our S-3 Registration Statement, including $75.0 million available pursuant to our ATM program.

In August 2020, we sold 6,250,000 shares of our common stock at a public offering price of $8.00 per share, for net proceeds of $46.7 million, after deducting

underwriting discounts and commissions and other offering expenses payable by us, or the August 2020 Offering.

In February 2019, we sold 13,993,778 shares of our common stock and 2,500 shares of Series A Convertible Preferred Stock at a public offering price of $2.00
and $2,000 per share, respectively, for net proceeds of $30.5 million, after deducting underwriting discounts and commissions and other offering expenses payable by us,
or the February 2019 Offering. In October and November 2019, we sold 10,350,000 shares of our common stock, which included the full exercise of the underwriters’
option to purchase additional shares, and 4,000 shares of Series A Convertible Preferred Stock at a public offering price of $2.50 and $2,500 per share, respectively, for
net proceeds of $33.5 million after deducting underwriting discounts and commissions and other offering expenses payable by us, or the October 2019 Offering.

During the year ended December 31, 2019, we sold 6,893,888 shares of our common stock under our previous ATM program for net proceeds of $22.3 million

after deducting sales agent commissions and other offering expenses payable by us, or the ATM Offering.

Similar to other development-stage biotechnology companies, we have generated limited revenue, which has been through the Angelini License Agreement.  We
have incurred losses and experienced negative operating cash flows since our inception and anticipate that we will continue to incur losses for at least the next several
years. We incurred net losses of approximately $81.0 million and $60.5 million for the year ended December 31, 2020 and 2019, respectively. As of December 31, 2020,
we had an accumulated deficit of $294.2 million and working capital of $52.8 million.

Management  has  identified  these  conditions  or  events,  which,  considered  in  the  aggregate,  raise  substantial  doubt  about  our  ability  to  continue  as  a  going
concern, including the risk that we will be unable to raise adequate additional capital to fund operations through at least the next 12 months from the date of filing of this
Annual Report on Form 10-K.  Management’s response to these conditions and events is that the successful closing of the Takeda License and Termination Agreement
with Takeda (see note 12 of our Consolidated Financial Statements) will provide the liquidity needed to alleviate the substantial doubt referred to above.  As described in
note  12  of  our  Consolidated  Financial  Statements,  there  are  certain  conditions  to  close  the  Takeda  License  and  Termination  Agreement,  however,  management  has
determined that the likelihood of not closing in the first half of 2021 is remote. In the event that we are unable to close the Takeda License and Termination Agreement,
we will need to raise additional capital in order to

66

 
 
alleviate substantial doubt about our ability to continue as a going concern. The failure to raise capital as and when needed could have a negative impact on our financial
condition  and  ability  to  pursue  our  business  strategy.    If  we  are  unable  to  raise  capital,  we  may  be  required  to  delay,  reduce  the  scope  of  or  eliminate  research  and
development programs, or obtain funds through arrangements with collaborators or others that may require us to relinquish rights to certain drug candidates that we might
otherwise seek to develop or commercialize independently.

In addition to the proceeds we expect to receive upon closing of the Takeda License and Termination Agreement, we plan to finance our cash needs through
either equity offerings, debt financings, collaborations, strategic alliances, or licensing agreements or a combination of any such transactions. To the extent that we raise
additional capital through future equity offerings or debt financings, ownership interests may be diluted, and the terms of these securities may include liquidation or other
preferences that adversely affect your rights as a common stockholder. Debt and equity financings, if available, may involve agreements that include covenants limiting or
restricting our ability to take specific actions, such as incurring additional debt, making capital expenditures or declaring dividends. There can be no assurance that such
financings will be obtained on terms acceptable to us, if at all. The ongoing COVID-19 pandemic continues to rapidly evolve and has already resulted in a significant
disruption  of  global  financial  markets.    If  the  disruption  persists  and  deepens,  we  could  experience  an  inability  to  access  additional  capital,  which  could  in  the  future
negatively affect our operations. If we raise additional funds through collaborations, strategic alliances or licensing agreements with third parties for one or more of our
current or future drug candidates, we may be required to relinquish valuable rights to our technologies, future revenue streams, research programs or drug candidates or to
grant licenses on terms that may not be favorable to us. Our failure to raise capital as and when needed would have a material adverse effect on our financial condition
and our ability to pursue our business strategy.

Cash Flows

The following table summarizes our cash flows for the periods indicated:

Net cash provided by (used in):
Operating activities
Investing activities
Financing activities
Net increase in cash and cash equivalents

Net Cash Used in Operating Activities

Year Ended
December 31,
2020

Year Ended
December 31,
2019

(in thousands)

(51,584)   $
34,648     
47,072     
30,136    $

(51,091)
(30,041)
86,539 
5,407

  $

  $

Net cash used in operating activities was $51.6 million for the year ended December 31, 2020, which consisted of a net loss of $81.0 million offset by a net of
$29.5  million  of  non-cash  charges  and  indirect  cash  changes,  primarily  related  to  $7.5  million  of  stock-based  compensation  expense  and  $12.4  million  of  deferred
revenue. Net cash used in operating activities was $51.1 million for the year ended December 31, 2019, which consisted of a net loss of $60.5 million offset by a net of
$9.4 million of non-cash charges and indirect cash changes, primarily related to $5.2 million of stock-based compensation expense.

Net Cash Provided by (Used in) Investing Activities

Net cash provided by investing activities was $34.6 million for the year ended December 31, 2020, compared to $30.0 million used in investing activities for the
year ended December 31, 2019. The change in net cash provided by investing activities was primarily due to the higher maturities of short-term investments during the
year ended December 31, 2020 compared to net purchases during the year ended December 31, 2019.

Net Cash Provided by Financing Activities

Net cash provided by financing activities of $47.0 million for the year ended December 31, 2020 was primarily due to the net proceeds from the August 2020
Offering. Net cash provided by financing activities of $86.5 million for the year ended December 31, 2019 was primarily due to the net proceeds from the February 2019
Offering, October 2019 Offering and ATM Offering.

Contractual Obligations and Commitments

As of December 31, 2020, we agreed to continue certain studies that were ongoing at the time of signing the Angelini License Agreement.  In March 2021, we
entered  into  the  Takeda  License  and  Termination  Agreement  under  which  Takeda  will  secure  global  rights  at  closing  from  us  to  develop  and  commercialize  the
investigational  medicine  OV935  for  the  treatment  of  developmental  and  epileptic  encephalopathies,  including  DS  and  LGS.  Closing  of  the  Takeda  License  and
Termination Agreement is subject to satisfaction of customary closing conditions, including regulatory review by the appropriate regulatory agencies under the HSR Act.
We had no other material contractual obligations or commitments. We had no long-term debt or leases and no material non-cancelable

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purchase commitments with service providers, as we have generally contracted on a cancelable, purchase order basis. We excluded any potential contingent payments
upon the achievement by us of clinical, regulatory and commercial events, as applicable, or royalty payments that we may be required to make under license agreements
we  have  entered  into  with  various  entities  pursuant  to  which  we  have  in-licensed  certain  intellectual  property  as  contractual  obligations  or  commitments,  including
agreements with H. Lundbeck A/S, Northwestern, and our Takeda license agreement. Pursuant to these license agreements, we have agreed to make milestone payments
up to an aggregate of $279.3 million upon the achievement of certain development, regulatory and sales milestones. We excluded these contingent payments given that
the timing, probability, and amount, if any, of such payments cannot be reasonably estimated at this time.

Off-Balance Sheet Arrangements

We did not have during the periods presented, and we do not currently have, any off-balance sheet arrangements, as defined in the rules and regulations of the

SEC.

Emerging Growth Company Status and Smaller Reporting Company Status

We are an “emerging growth company,” as defined in the Jumpstart Our Business Startups Act of 2012, or the JOBS Act, and may remain an emerging growth
company until December 31, 2022. For so long as we remain an emerging growth company, we are permitted and intend to rely on exemptions from certain disclosure
requirements that are applicable to other public companies that are not emerging growth companies. These exemptions include:

•

•

•

reduced disclosure about our executive compensation arrangements;

no non-binding stockholder advisory votes on executive compensation or golden parachute arrangements; and

exemption from the auditor attestation requirement in the assessment of our internal control over financial reporting.

We have taken advantage of reduced reporting requirements in this Annual Report on Form 10-K and may continue to do so until such time that we are no longer
an emerging growth company. We will remain an “emerging growth company” until the earliest of (a) the last day of the fiscal year in which we have total annual gross
revenues of $1.07 billion or more, (b) December 31, 2022, the last day of the fiscal year following the fifth anniversary of the completion of the our IPO, (c) the date on
which we have issued more than $1.0 billion in nonconvertible debt during the previous three years or (d) the date on which we are deemed to be a large accelerated filer
under the rules of the SEC. Section 107 of the JOBS Act provides that an emerging growth company can take advantage of the extended transition period for complying
with new or revised accounting standards. We have irrevocably elected not to avail ourselves of this extended transition period and, as a result, we will adopt new or
revised accounting standards on the relevant dates on which adoption of such standards is required for other public companies.

In addition, we are also a smaller reporting company as defined in the Exchange Act. We may continue to be a smaller reporting company even after we are no
longer  an  emerging  growth  company.  We  may  take  advantage  of  certain  of  the  scaled  disclosures  available  to  smaller  reporting  companies  and  will  be  able  to  take
advantage of these scaled disclosures for so long as (i) our voting and non-voting common stock held by non-affiliates is less than $250.0 million measured on the last
business day of our second fiscal quarter or (ii) our annual revenue is less than $100.0 million during the most recently completed fiscal year and our voting and non-
voting common stock held by non-affiliates is less than $700.0 million measured on the last business day of our second fiscal quarter.

Critical Accounting Policies and Estimates

Our  management’s  discussion  and  analysis  of  financial  condition  and  results  of  operations  is  based  on  our  financial  statements,  which  have  been  prepared  in
accordance  with  accounting  principles  generally  accepted  in  the  United  States.  The  preparation  of  these  financial  statements  requires  us  to  make  estimates  and
assumptions that affect the reported amounts of assets and liabilities and the disclosure of contingent assets and liabilities at the date of the financial statements, as well as
the  revenue  and  expenses  incurred  during  the  reported  periods.  On  an  ongoing  basis,  we  evaluate  our  estimates  and  judgments,  including  those  related  to  accrued
expenses  and  stock-based  compensation.  We  base  our  estimates  on  historical  experience  and  on  various  other  factors  that  we  believe  are  reasonable  under  the
circumstances,  the  results  of  which  form  the  basis  for  making  judgments  about  the  carrying  value  of  assets  and  liabilities  that  are  not  apparent  from  other  sources.
Changes  in  estimates  are  reflected  in  reported  results  for  the  period  in  which  they  become  known.  Actual  results  may  differ  from  these  estimates  under  different
assumptions or conditions.

During the year ended December 31, 2020, we recognized revenue.  In addition, see Note 2 of our Consolidated Financial Statements under the heading “Recent

Accounting Pronouncements” for new accounting pronouncements or changes to the accounting pronouncements during the year ended December 31, 2020.

Accrued Clinical Expenses

When preparing our consolidated financial statements, we are required to estimate our accrued clinical expenses. This process involves reviewing open contracts
and communicating with our personnel to identify services that have been performed on our behalf and estimating the level of service performed and the associated cost
incurred for the service when we have not yet been invoiced or

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otherwise notified of actual cost. Payments under some of the contracts we have with third parties depend on factors, such as successful enrollment of certain numbers of
patients, site initiation and the completion of clinical trial milestones.

When accruing clinical expenses, we estimate the time period over which services will be performed and the level of effort to be expended in each period. If
possible, we obtain information regarding unbilled services directly from our service providers. However, we may be required to estimate the cost of these services based
only on information available to us. If we underestimate or overestimate the cost associated with a trial or service at a given point in time, adjustments to research and
development expenses may be necessary in future periods. Historically, our estimated accrued clinical expenses have approximated actual expense incurred.

Stock-Based Compensation

We account for stock-based compensation awards in accordance with the Financial Accounting Standards Board Accounting Standards Codification, or ASC,
Topic 718, Compensation—Stock Compensation,  or  ASC  718  (see  Note  2  of  our Consolidated Financial Statements). ASC 718 requires all stock-based compensation
awards to be recognized as expense based on their grant date fair values. We recognized expenses over the requisite service period, which is generally the vesting period
of  the  award  under  the  straight-line  method.    We  account  for  forfeitures  as  they  occur.  We  record  the  expense  for  stock-based  compensation  awards  subject  to
performance-based  milestone  vesting  over  the  remaining  service  period  when  management  determines  that  achievement  of  the  milestone  is  probable.  Management
evaluates when the achievement of a performance-based milestone is probable based on the expected satisfaction of the performance conditions at each reporting date.

We measure the grant-date fair value based on the Black-Scholes option-pricing model, which uses subjective assumptions and other inputs.  These assumptions

and inputs include:

•

•

•

•

Expected Volatility.  Due  to  the  lack  of  sufficient  volatility  data,  the  expected  volatility  is  estimated  using  weighted  average  measures  of  the  historical
volatility of a representative group of small, publicly traded drug development companies at a similar stage of development as ourselves.  

Expected Term. The expected term of the options outstanding is determined using the “simplified” method for “plain vanilla” options based on the mid-
point between the vesting date and the end of the contractual term as prescribed by Staff Accounting Bulletin No. 107, Share-Based Payment.  

Risk-Free Interest Rate. The risk-free interest rate is based on U.S. Treasury notes with remaining terms similar to the expected term of the option.

Expected  Dividends.    The  dividend  yield  assumption  is  zero  since  we  have  never  paid  cash  dividends  and  do  not  plan  to  pay  cash  dividends  in  the
foreseeable future.

Revenue Recognition

We recognize revenue under sublicense agreements in accordance with the ASC 606. We currently have one such agreement, the Angelini License Agreement.
The terms of the agreement within this scope may contain multiple performance obligations, including but not limited to licenses and research and development activities.
ASC 606 requires that we evaluate these agreements to determine the distinct performance obligations. Non-refundable, up-front fees that are not contingent on any future
performance and require no consequential continuing involvement by us, are recognized as revenue when the license term commences and the licensed data, technology
or product is delivered. We defer recognition of non-refundable upfront fees if the performance obligations are not satisfied.

Prior  to  recognizing  revenue,  we  make  estimates  of  the  transaction  price,  including  variable  consideration  that  is  subject  to  a  constraint.  Amounts  of  variable
consideration are included in the transaction price to the extent that it is probable that a significant reversal in the amount of cumulative revenue recognized will not occur
when  the  uncertainty  associated  with  the  variable  consideration  is  subsequently  resolved.  Variable  consideration  may  include  all  or  portions  of  upfront  license  fees,
payments  for  research  and  development  activities,  reimbursement  of  certain  third-party  costs,  payments  based  upon  the  achievement  of  specified  milestones,  royalty
payments based on product sales derived from collaboration and other payments.

If there are multiple distinct performance obligations, we allocate the transaction price to each distinct performance obligation based on its relative standalone
selling price. For the Angelini License Agreement, the transaction price was allocated based on the standalone selling prices of the license and ongoing trials. The portion
of  the  upfront  payment  allocated  to  the  license  was  recognized  in  full  as  it  was  non-refundable  and  not  contingent  on  any  future  performance  and  requires  no
consequential continuing involvement by the Company. Revenue related to ongoing trials is recognized by measuring the progress toward complete satisfaction of the
performance obligations over time based on the portion of estimated total trial costs to be incurred. Milestone payments are considered contingent variable consideration
which are not accounted for until the contingencies are met.

69

 
 
 
 
 
 
 
Item 7A. Quantitative and Qualitative Disclosures About Market Risk.

The primary objectives of our investment activities are to ensure liquidity and to preserve capital. As of December 31, 2020, we had cash and cash equivalents of
$72.0 million that were held in an interest-bearing money market account. Our primary exposure to market risk is interest rate sensitivity, which is affected by changes in
the general level of U.S. interest rates. Due to the short-term maturities of our cash equivalents and the low risk profile of our investments, an immediate 100 basis point
change in interest rates would not have a material effect on the fair market value of our cash equivalents. To minimize the risk in the future, we intend to maintain our
portfolio of cash equivalents in institutional market funds that are comprised of U.S. Treasury and U.S. Treasury-backed repurchase agreements.

Item 8. Financial Statements and Supplementary Data

Our financial statements, together with the report of our independent registered public accounting firm, appear in this Annual Report on Form 10-K beginning on

page F-1.

Item 9. Changes in and Disagreements with Accountants on Accounting and Financial Disclosure

None.

Item 9A. Controls and Procedures.

Management’s Evaluation of our Disclosure Controls and Procedures

We maintain disclosure controls and procedures that are designed to ensure that information required to be disclosed in the reports that we file or submit under the
Securities Exchange Act of 1934, as amended (the “Exchange Act”) is (1) recorded, processed, summarized, and reported within the time periods specified in the SEC’s
rules  and  forms  and  (2)  accumulated  and  communicated  to  our  management,  including  our  principal  executive  officer  and  principal  financial  officer,  to  allow  timely
decisions regarding required disclosure.

As of December 31, 2020, our management, with the participation of our principal executive officer and principal financial officer, evaluated the effectiveness of
our  disclosure  controls  and  procedures  (as  defined  in  Rules  13a-15(e)  and  15d-15(e)  under  the  Exchange  Act).  Our  management  recognizes  that  any  controls  and
procedures,  no  matter  how  well  designed  and  operated,  can  provide  only  reasonable  assurance  of  achieving  their  objectives,  and  management  necessarily  applies  its
judgment in evaluating the cost-benefit relationship of possible controls and procedures. Our principal executive officer and principal financial officer have concluded
based upon the evaluation described above that, as of December 31, 2020 our disclosure controls and procedures were effective at the reasonable assurance level.

Management’s Annual Report on Internal Control over Financial Reporting

Our management is responsible for establishing and maintaining adequate internal control over financial reporting, as defined in Rules 13a-15(f) and 15d-15(f) of
the Exchange Act. Our management, under the supervision and with the participation of our Chief Executive Officer and Principal Financial and Accounting Officer,
conducted  an  evaluation  of  the  effectiveness  of  our  internal  control  over  financial  reporting  as  of  December  31,  2020  based  on  the  framework  in  Internal  Control-
Integrated Framework issued by the Committee of Sponsoring Organizations of the Treadway Commission (2013 Framework). Based on the results of its evaluation,
management concluded that our internal control over financial reporting was effective as of December 31, 2020.

Attestation Report of the Registered Public Accounting Firm

This Annual Report on Form 10-K does not include an attestation report of our registered public accounting firm due to an exemption established by the JOBS

Act for “emerging growth companies.”

Changes in Internal Control over Financial Reporting

There have been no changes in our internal control over financial reporting during our most recent quarter ended December 31, 2020 that materially affected, or

are reasonably likely to materially affect, our internal control over financial reporting.

Item 9B.  Other Information.

None.

70

 
Item 10. Directors, Executive Officers, and Corporate Governance

PART III

The  information  required  by  this  item  is  incorporated  by  reference  to  the  information  set  forth  in  the  sections  titled  “Proposal  1  –  Election  of  Directors,”

“Executive Officers,” and “Information Regarding the Board and Corporate Governance” and “Delinquent Section 16(a) Reports,” if any, in our 2021 Proxy Statement.

Item 11. Executive Compensation

The information required by this item is incorporated by reference to the information set forth in the section titled “Executive Officer and Director Compensation”

in our 2021 Proxy Statement.

Item 12. Security Ownership of Certain Beneficial Owners and Management and Related Stockholder Matters

The  information  required  by  this  item  is  incorporated  by  reference  to  the  information  set  forth  in  the  section  titled  “Security  Ownership  of  Certain  Beneficial

Owners and Management and “Equity Compensation Plan Information” in our 2021 Proxy Statement.

Item 13. Certain Relationships and Related Transactions and Director Independence

The  information  required  by  this  item  is  incorporated  by  reference  to  the  information  set  forth  in  the  section  titled  “Transactions  with  Related  Persons”  and

“Information Regarding the Board and Corporate Governance – Board Independence” in our 2021 Proxy Statement.

Item 14. Principal Accountant Fees and Services

The information required by this item is incorporated by reference to the information set forth in the section titled “Independent Registered Public Accounting

Firm Fees” and “Pre-Approval Policies and Procedures” contained in our 2021 Proxy Statement.

71

 
PART IV

Item 15. Exhibits, Financial Statements and Schedules

(a)(1) Financial Statements.

The response to this portion of Item 15 is set forth under Item 8 hereof.

(a)(2) Financial Statement Schedules.

All schedules have been omitted because they are not required or because the required information is given in the Financial Statements or Notes thereto.

(a)(3) Exhibits.

The exhibits listed below are filed as part of this Annual Report on Form 10-K.

Number

  Description

3.1

3.2

3.3

4.1

4.2

4.3

4.4

10.1+

10.2+

10.3+

10.4+

10.5+

10.6+

Amended and Restated Certificate of Incorporation (incorporated herein by reference to Exhibit 3.1 to the Company’s Current Report on Form 8-K (File
No. 001-38085), filed with the Commission on May 10, 2017).

Corrected Amended and Restated Certificate of Designation of Series A Convertible Preferred Stock (incorporated herein by reference to Exhibit 3.1 to
the Company’s Current Report on Form 8-K (File No. 001-38085), filed with the Commission on September 24, 2019).

Amended and Restated Bylaws (incorporated herein by reference to Exhibit 3.2 to the Company’s Current Report on Form 8-K (File No. 001-38085),
filed with the Commission on May 10, 2017).

Form of Common Stock Certificate of the Company (incorporated herein by reference to Exhibit 4.1 to the Company’s Registration Statement on Form
S-1/A (File No. 333-217245), filed with the Commission on April 25, 2017).

Second Amended and Restated Investors’ Rights Agreement, by and among the Company and certain of its stockholders, dated January 6, 2017
(incorporated herein by reference to Exhibit 4.2 to the Company’s Registration Statement on Form S-1 (File No. 333-217245), filed with the
Commission on April 10, 2017).

Description of the Securities of Ovid Therapeutics Inc. (incorporated herein by reference to Exhibit 4.3 to the Company’s Annual Report on Form 10-K
(File No. 001-38085), filed with the Commission on March 12, 2020).

Form of Series A Preferred Stock Certificate (incorporated herein by reference to Exhibit 4.1 to the Company’s Current Report on Form 8-K (File No.
001-38085), filed with the Commission on February 21, 2019).

Form of Indemnity Agreement by and between the Company and its directors and officers (incorporated herein by reference to Exhibit 10.1 to the
Company’s Registration Statement on Form S-1 (File No. 333-217245), filed with the Commission on April 10, 2017).

2017 Equity Incentive Plan (incorporated herein by reference to Exhibit 4.12 to the Company’s Registration Statement on Form S-8 (File No. 001-
38085), filed with the Commission on May 22, 2017).

Forms of Option Grant Notice and Option Agreement under 2017 Equity Incentive Plan (incorporated herein by reference to Exhibit 10.3 to the
Company’s Registration Statement on Form S-1 (File No. 333-217245), filed with the Commission on April 10, 2017).

2014 Equity Incentive Plan, as amended (incorporated herein by reference to Exhibit 10.5 to the Company’s Registration Statement on Form S-1 (File
No. 333-217245), filed with the Commission on April 10, 2017).

Amendment to 2014 Equity Incentive Plan, effective as of March 9, 2015 (incorporated herein by reference to Exhibit 10.6 to the Company’s
Registration Statement on Form S-1 (File No. 333-217245), filed with the Commission on April 10, 2017).

Amendment to 2014 Equity Incentive Plan, effective as of June 4, 2015 (incorporated herein by reference to Exhibit 10.7 to the Company’s Registration
Statement on Form S-1 (File No. 333-217245), filed with the Commission on April 10, 2017).

72

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
10.7+

10.8+

10.9+

10.10+

10.11+

10.12+

10.13+

10.14+

10.15+

10.16+

10.17+

10.18+

10.19+

10.20†

10.21†

10.22†

10.23†

10.24^

Amendment to 2014 Equity Incentive Plan, effective as of July 28, 2015 (incorporated herein by reference to Exhibit 10.8 to the Company’s Registration
Statement on Form S-1 (File No. 333-217245), filed with the Commission on April 10, 2017).

Amendment to 2014 Equity Incentive Plan, effective as of February 11, 2016 (incorporated herein by reference to Exhibit 10.9 to the Company’s
Registration Statement on Form S-1 (File No. 333-217245), filed with the Commission on April 10, 2017).

Form of Restricted Stock Purchase Agreement under the 2014 Equity Incentive Plan (incorporated herein by reference to Exhibit 10.10 to the
Company’s Registration Statement on Form S-1 (File No. 333-217245), filed with the Commission on April 10, 2017).

Form of Stock Option Agreement—Early Exercise under the 2014 Equity Incentive Plan (incorporated herein by reference to Exhibit 10.11 to the
Company’s Registration Statement on Form S-1 (File No. 333-217245), filed with the Commission on April 10, 2017).

Forms of Stock Option Agreement under the 2014 Equity Incentive Plan (incorporated herein by reference to Exhibit 10.12 to the Company’s
Registration Statement on Form S-1 (File No. 333-217245), filed with the Commission on April 10, 2017).

2017 Employee Stock Purchase Plan (incorporated herein by reference to Exhibit 4.14 to the Company’s Registration Statement on Form S-8 (File No.
001-38085), filed with the Commission on May 22, 2017).

Non-Employee Director Compensation Plan (incorporated herein by reference to Exhibit 10.13 to the Company’s Annual Report on Form 10-K (File
No. 001-38085), filed with the Commission on March 12, 2020).

Executive Employment Agreement between the Registrant and Jeremy M. Levin, dated June 5, 2015 (incorporated herein by reference to Exhibit 10.13
to the Company’s Registration Statement on Form S-1 (File No. 333-217245), filed with the Commission on April 10, 2017).

Second Amended and Restated Executive Employment Agreement between the Company and Amit Rakhit, effective November 1, 2019 (incorporated
herein by reference to Exhibit 10.15 to the Company’s Annual Report on Form 10-K (File No. 001-38085), filed with the Commission on March 12,
2020.

Third Amended and Restated Executive Employment Agreement between the Company and Tim Daly, effective December 18, 2019 (incorporated
herein by reference to Exhibit 10.16 to the Company’s Annual Report on Form 10-K (File No. 001-38085), filed with the Commission on March 12,
2020.

  Executive Employment Agreement between the Company and Jeff Rona, effective September 30, 2020

  Executive Employment Agreement between the Company and Jason Tardio, effective October 21, 2019

  Amended and Restated Executive Employment Agreement between the Company and Thomas Perone, effective January 1, 2020

License Agreement by and between H. Lundbeck A/S and the Company, dated March 25, 2015 (incorporated herein by reference to Exhibit 10.16 to the
Company’s Registration Statement on Form S-1 (File No. 333-217245), filed with the Commission on May 2, 2017).

Collaboration and License Agreement, by and between the Company and Takeda Pharmaceutical Company Limited, effective January 6, 2017
(incorporated herein by reference to Exhibit 10.18 to the Company’s Registration Statement on Form S-1 (File No. 333-217245), filed with the
Commission on April 10, 2017).

Series B-1 Preferred Stock Purchase Agreement, by and between the Company and Takeda Pharmaceutical Company Limited, dated January 6, 2017
(incorporated herein by reference to Exhibit 10.19 to the Company’s Registration Statement on Form S-1 (File No. 333-217245), filed with the
Commission on April 10, 2017).

License Agreement by and between Northwestern University and the Company, dated December 15, 2016.  (incorporated herein by reference to Exhibit
10.19 to the Company’s Annual Report on Form 10-K (File No. 001-38085), filed with the Commission on April 10, 2017).

First Amendment to License Agreement, by and between H. Lundbeck A/S and the Company, dated May 10, 2019 (incorporated herein by reference to
Exhibit 10.1 to the Company’s Current Report on Form 8-K/A (File No. 001-38085), filed with the Commission on June 17, 2019).

73

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
10.25†

  Collaboration and License Agreement, by and between the Company and Angelini Pharma Rare Diseases AG, dated July 9, 2020.

23.1

24.1

31.1

31.2

  Consent of Independent Registered Public Accounting Firm.

  Power of Attorney (included on the signature page to this report).

  Certification of Principal Executive Officer Pursuant to Rules 13a-14(a) and 15d-14(a) under the Securities Exchange Act of 1934, as Adopted Pursuant

to Section 302 of the Sarbanes-Oxley Act of 2002.

  Certification of Principal Financial Officer Pursuant to Rules 13a-14(a) and 15d-14(a) under the Securities Exchange Act of 1934, as Adopted Pursuant

to Section 302 of the Sarbanes-Oxley Act of 2002.

32.1*

  Certification of Principal Executive Officer and Principal Financial Officer Pursuant to 18 U.S.C. Section 1350, as Adopted Pursuant to Section 906 of

the Sarbanes-Oxley Act of 2002.

101.INS

  XBRL Instance Document

101.SCH

  XBRL Taxonomy Extension Schema Document

101.CAL

  XBRL Taxonomy Extension Calculation Linkbase Document

101.DEF

  XBRL Taxonomy Extension Definition Linkbase Document

101.LAB

  XBRL Taxonomy Extension Label Linkbase Document

101.PRE

  XBRL Taxonomy Extension Presentation Linkbase Document

*

+
†
^

Furnished herewith and not deemed to be “filed” for purposes of Section 18 of the Securities Exchange Act of 1934, as amended (the “Exchange Act”), and shall
not be deemed to be incorporated by reference into any filing under the Securities Act of 1933, as amended, or the Exchange Act (whether made before or after
the date of the Form 10-K), irrespective of any general incorporation language contained in such filing.
Indicates a management contract or compensatory plan.
Confidential treatment has been granted for certain portions of this exhibit. These portions have been omitted and filed separately with the SEC.
Pursuant to Item 601(b)(10)(iv) of Regulation S-K promulgated by the Securities and Exchange Commission, certain portions of this exhibit have been redacted.
The Registrant hereby agrees to furnish supplementally to the Securities and Exchange Commission, upon its request, an unredacted copy of this exhibit.

Item 16. Form 10-K Summary

Not applicable.

74

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Pursuant to the requirements of the Securities Exchange Act of 1934, the registrant has duly caused this report on Form 10-K to be signed on its behalf by the

undersigned thereunto duly authorized.

SIGNATURES

Date: March 15, 2021

Date: March 15, 2021

  OVID THERAPEUTICS INC.

By:  /s/ Jeremy M. Levin
   Jeremy M. Levin
  Chief Executive Officer

(Principal Executive Officer)

By:  /s/ Timothy Daly
  Timothy Daly

Executive Vice President, Finance, Corporate Controller &
Treasurer
(Principal Financial and Accounting Officer)

POWER OF ATTORNEY

Each person whose individual signature appears below hereby authorizes and appoints Jeremy M. Levin, DPhil, MB BChir and Timothy Daly, and each of them, with
full power of substitution and resubstitution and full power to act without the other, as his or her true and lawful attorney-in-fact and agent to act in his or her name, place
and stead and to execute in the name and on behalf of each person, individually and in each capacity stated below, and to file any and all amendments to this report on
Form 10-K, and to file the same, with all exhibits thereto, and other documents in connection therewith, with the Securities and Exchange Commission, granting unto said
attorneys-in-fact and agents, and each of them, full power and authority to do and perform each and every act and thing, ratifying and confirming all that said attorneys-
in-fact and agents or any of them or their or his or her substitute or substitutes may lawfully do or cause to be done by virtue thereof.

Pursuant to the requirements of the Securities Exchange Act of 1934, this report has been signed below by the following persons on behalf of the registrant and in the

capacities and on the dates indicated.

Signature

Title

/s/ Jeremy M. Levin, DPhil, MB BChir
Jeremy M. Levin, DPhil, MB BChir

Chief Executive Officer and Director
(Principal Executive Officer)

/s/ Timothy Daly
Timothy Daly

/s/ Karen Bernstein, PhD
Karen Bernstein, PhD

/s/ Barbara Duncan
Barbara Duncan

/s/ Bart Friedman
Bart Friedman

/s/ Douglas Williams, PhD
Douglas Williams, PhD

Executive Vice President, Finance and Corporate Controller
(Principal Financial and Accounting Officer)

Director

Director

Director

Director

75

Date

March 15, 2021

March 15, 2021

March 15, 2021

March 15, 2021

March 15, 2021

March 15, 2021

 
 
 
 
 
 
 
   
 
 
 
 
 
 
 
 
    
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
OVID THERAPEUTICS INC.

Index to Consolidated Financial Statements

Report of Independent Registered Public Accounting Firm
Consolidated Balance Sheets
Consolidated Statements of Operations
Consolidated Statements of Comprehensive Loss
Consolidated Statements of Changes in Stockholders’ Equity
Consolidated Statements of Cash Flows
Notes to Consolidated Financial Statements

F-1

F-2  
F-3  
F-4  
F-5  
F-6  
F-7  
F-8–F-23  

 
 
 
 
 
 
 
 
 
 
Report of Independent Registered Public Accounting Firm

To the Stockholders and Board of Directors 
Ovid Therapeutics Inc.:

Opinion on the Consolidated Financial Statements

We have audited the accompanying consolidated balance sheets of Ovid Therapeutics Inc. and subsidiary (the Company) as of December 31, 2020 and 2019, the related
consolidated statements of operations, comprehensive loss, changes in stockholders’ equity, and cash flows for the years then ended, and the related notes (collectively,
the consolidated financial statements). In our opinion, the consolidated financial statements present fairly, in all material respects, the financial position of the Company
as of December 31, 2020 and 2019, and the results of its operations and its cash flows for the years then ended, in conformity with U.S. generally accepted accounting
principles.

Basis for Opinion

These consolidated financial statements are the responsibility of the Company’s management. Our responsibility is to express an opinion on these consolidated
financial statements based on our audits. We are a public accounting firm registered with the Public Company Accounting Oversight Board (United States) (PCAOB)
and are required to be independent with respect to the Company in accordance with the U.S. federal securities laws and the applicable rules and regulations of the
Securities and Exchange Commission and the PCAOB.

We conducted our audits in accordance with the standards of the PCAOB. Those standards require that we plan and perform the audit to obtain reasonable assurance
about whether the consolidated financial statements are free of material misstatement, whether due to error or fraud. The Company is not required to have, nor were
we engaged to perform, an audit of its internal control over financial reporting. As part of our audits, we are required to obtain an understanding of internal control
over financial reporting but not for the purpose of expressing an opinion on the effectiveness of the Company’s internal control over financial reporting. Accordingly,
we express no such opinion.

Our audits included performing procedures to assess the risks of material misstatement of the consolidated financial statements, whether due to error or fraud, and
performing procedures that respond to those risks. Such procedures included examining, on a test basis, evidence regarding the amounts and disclosures in the
consolidated financial statements. Our audits also included evaluating the accounting principles used and significant estimates made by management, as well as
evaluating the overall presentation of the consolidated financial statements. We believe that our audits provide a reasonable basis for our opinion.

/s/ KPMG LLP

We have served as the Company’s auditor since 2015.

New York, New York
March 15, 2021

F-2

 
 
 
 
 
PART I—FINANCIAL INFORMATION

OVID THERAPEUTICS INC.
Consolidated Balance Sheets

Assets

Item 1. Financial Statements.

Current assets:

Cash and cash equivalents
Short-term investments
Related party receivable
Prepaid expenses and other current assets

Total current assets

Long-term prepaid expenses
Security deposit
Property and equipment, net
Other assets

Total assets

Liabilities and Stockholders' Equity

Current liabilities:

Accounts payable
Accrued expenses
Related party payable
Deferred revenue - current
Total current liabilities
Related party payable - noncurrent
Deferred revenue, net of current portion

Total liabilities

Stockholders' equity:

December 31,
2020

December 31,
2019

  $

72,033,930    $

-   
141,763   
2,667,508   
74,843,201   

477,171   
150,626   
135,620   
318,900   
75,925,518    $

5,446,206    $
12,032,685   
2,370,992   
2,212,892   
22,062,775   
61,200   
10,169,887   
32,293,862   

  $

  $

41,897,144 
34,841,969 
1,131,146 
1,942,933 
79,813,192 

359,539 
135,390 
68,363 
467,247 
80,843,731 

3,256,098 
7,266,706 
10,804 
- 
10,533,608 
286,562 
- 
10,820,170 

Preferred stock, $0.001 par value; 10,000,000 shares authorized; Series A convertible preferred stock, 10,000 shares
designated, 3,250 and 7,762 shares issued and outstanding at December 31, 2020 and 2019, respectively
Common stock, $0.001 par value; 125,000,000 shares authorized; 65,743,170 and 54,710,322 shares issued and
outstanding at December 31, 2020 and 2019, respectively
Additional paid-in-capital
Accumulated other comprehensive income
Accumulated deficit

Total stockholders' equity

Total liabilities and stockholders' equity

3   

8 

65,743   
337,758,007   
-   
(294,192,097)  
43,631,656   
75,925,518    $

54,711 
283,122,894 
2,469 
(213,156,521)
70,023,561 
80,843,731

  $

See accompanying notes to these consolidated financial statements

F-3

 
 
 
 
 
 
 
 
 
 
 
 
     
   
   
 
 
   
   
   
 
   
 
   
 
   
 
 
 
 
 
 
   
   
   
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
   
   
 
     
   
   
 
 
   
   
   
 
   
 
   
 
   
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
   
   
 
 
 
   
   
   
 
 
   
   
   
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
OVID THERAPEUTICS INC.
Consolidated Statements of Operations

Revenue:

License and other revenue

Operating expenses:

Research and development
General and administrative
Total operating expenses

Loss from operations
Other income, net
Net loss

Net loss attributable to common stockholders

Net loss per share attributable to common stockholders, basic and diluted

Weighted-average common shares outstanding basic and diluted

For the Year Ended
December 31,
2020

For the Year Ended
December 31,
2019

  $

12,617,221    $

- 

63,417,394 
30,630,804 
94,048,198 
(81,430,977)
395,401 
(81,035,576)

(81,035,576)

 $

 $

(1.39)   $

42,157,641 
19,251,826 
61,409,467 
(61,409,467)
948,224 
(60,461,243)

(60,461,243)

(1.54)

58,451,293 

39,217,223  

 $

 $

  $

See accompanying notes to these consolidated financial statements

F-4

 
 
 
 
   
 
 
 
 
 
 
 
   
   
   
 
 
   
   
   
 
  
  
  
  
  
  
  
  
  
  
   
   
 
OVID THERAPEUTICS INC.
Consolidated Statements of Comprehensive Loss

Net loss
Other comprehensive (loss) income:

Unrealized (loss) gain on available-for-sale securities

Comprehensive loss

For the Year
Ended
December 31,
2020

For the Year
Ended
December 31,
2019

 $

(81,035,576)  $

(60,461,243)

(2,469)   
(81,038,045)  $

4,298 
(60,456,945)

 $

See accompanying notes to these consolidated financial statements

F-5

 
 
 
 
   
 
 
 
 
 
 
    
 
    
 
  
 
 
 
OVID THERAPEUTICS INC.
Consolidated Statement of Changes in Stockholders’ Equity

Balance, December 31, 2019
ATM costs
Issuance of common stock from employee stock purchase plan
Issuance of common stock from exercise of stock options
Conversion of series A convertible preferred stock to common stock
Proceeds from August 2020 Offering, net of underwriting costs and
commissions
Stock-based compensation expense
Other comprehensive loss
Net loss
Balance, December 31, 2020

Balance, December 31, 2018
Proceeds from February Offering, net of underwriting costs and
commissions
Issuance of common stock from employee stock purchase plan
Conversion of common stock to series A convertible preferred stock
Proceeds from October Offering, net of underwriting costs and
commissions
Proceeds from ATM Offerings, net of underwriting costs and
commissions
Stock-based compensation expense
Other comprehensive income
Net loss
Balance, December 31, 2019

Convertible
Preferred Stock

Common Stock

  Shares  
  7,762 
- 
- 
- 

  (4,512)  

  Amount  
8 
  $
- 
- 
- 
(5)  

- 
- 
- 
- 
  3,250 

  $

- 
- 
- 
- 
3 

Shares
  54,710,322 
- 
105,464 
165,384 
4,512,000 

6,250,000 
- 
- 
- 
  65,743,170 

Additional
Paid-In
Capital
  $ 283,122,894 

(114,936)  
203,361 
300,656 

(4,507)  

  Amount
  $

54,711 
- 
105 
165 
4,512 

Accumulated
Other
Comprehensive 
  Income/(Loss)  
2,469 
  $
- 
- 

  Accumulated  
Deficit

Total

  $ (213,156,521)   $ 70,023,561 
(114,936)
- 
203,466 
- 
300,821 
- 

- 

6,250 
- 
- 
- 
65,743 

46,725,185 
7,525,354 
- 
- 
  $ 337,758,007 

  $

  $

(2,469)  

- 
- 
- 

  46,731,435 
7,525,354 
(2,469)
  (81,035,576)
  $ (294,192,097)   $ 43,631,656 

(81,035,576)  

- 

- 
- 

- 
- 

Convertible
Preferred Stock

Common Stock

  Shares  
- 

  Amount  
- 
  $

Shares
  24,654,114 

  Amount
  $

24,654 

Additional
Paid-In
Capital
  $ 191,477,598 

Accumulated
Other
Comprehensive 
  Income/(Loss)  
  $

  Accumulated  
Deficit

Total

(1,829)   $ (152,695,278)   $ 38,805,145 

  2,500 
- 
  1,262 

  4,000 

- 
- 
- 
- 
  7,762 

  $

3 
- 
1 

4 

- 
- 
- 
- 
8 

  13,993,778 
80,542 
(1,262,000)  

13,994 
81 
(1,262)  

30,506,838 
131,814 
1,261 

  10,350,000 

10,350 

33,519,919 

6,893,888 
- 
- 
- 
  54,710,322 

  $

6,894 
- 
- 
- 
54,711 

22,279,672 
5,205,792 
- 
- 
  $ 283,122,894 

  $

- 
- 
- 

- 

- 
- 
4,298 
- 
2,469 

- 
- 
- 

- 

  30,520,835 
131,895 
- 

  33,530,273 

- 
- 
- 

  22,286,566 
5,205,792 
4,298 
  (60,461,243)
  $ (213,156,521)   $ 70,023,561 

(60,461,243)  

See accompanying notes to these consolidated financial statements

F-6

 
 
 
 
 
 
 
 
 
 
 
 
   
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
     
       
       
       
       
       
       
       
 
 
 
 
 
 
 
 
 
   
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
     
       
       
       
       
       
       
       
 
 
     
       
       
       
       
       
       
       
 
 
OVID THERAPEUTICS INC.
Consolidated Statements of Cash Flows

Year Ended
December 31,
2020

Year Ended
December 31,
2019

  $

(81,035,576)   $

(60,461,243)

Cash flows from operating activities:

Net loss
Adjustments to reconcile net loss to cash used in operating activities:

Stock-based compensation expense
Depreciation and amortization expense
Change in accrued interest and accretion of discount on short-term
investments
Change in operating assets and liabilities:

Prepaid expenses and other current assets
Security deposit
Related party receivable
Long-term prepaid expenses
Accounts payable
Accrued expenses
Deferred revenue
Related party payable

Net cash used in operating activities

Cash flows from investing activities:

Purchases of short-term investments
Proceeds from maturities of short-term investments
Purchase of property and equipment
Software development and other assets

Net cash provided by (used in) investing activities

Cash flows from financing activities:

Proceeds from August 2020 Offering, net of offering expenses
Proceeds from February and October 2019 Offerings, net of offering
expenses
Proceeds from ATM Offerings, net of offering expenses
ATM costs
Proceeds from employee stock purchase plan
Proceeds from exercise of options

Net cash provided by financing activities

Net increase in cash and cash equivalents
Cash and cash equivalents, at beginning of period
Cash and cash equivalents, at end of period

Non-cash investing and financing activities:

Software development and other costs in accrued expenses and accounts
payable
Offering costs in accrued expenses and accounts payable

  $

  $
  $

7,525,354     
306,848     

5,205,792 
255,002 

(199,408)    

(29,633)

(724,575)    
(15,236)    
989,383     
(117,632)    
2,333,716     
4,835,607     
12,382,779     
2,134,826     
(51,583,914)    

224,458 
(13,235)
(531,042)
2,438,022 
(653,953)
2,177,844 
- 
297,366 
(51,090,622)

(9,961,092)    
45,000,000     
(127,240)    
(263,440)    
34,648,228     

(34,797,004)
5,000,000 
(57,156)
(186,889)
(30,041,049)

46,731,435     

- 

-     
-     
(163,250)    
203,466     
300,821     
47,072,472     

64,120,736 
22,286,566 
- 
131,895 
- 
86,539,197 

30,136,786     
41,897,144     
72,033,930    $

5,407,526 
36,489,618 
41,897,144 

—    $
21,314    $

164,922 
69,628

See accompanying notes to these consolidated financial statements

F-7

 
 
 
   
 
 
 
 
 
 
     
       
 
     
       
 
   
   
   
     
       
 
   
   
   
   
   
   
   
   
   
 
     
       
 
     
       
 
   
   
   
   
   
 
     
       
 
     
       
 
   
   
   
   
   
   
   
 
     
       
 
   
   
 
     
       
 
     
       
 
 
 
 
NOTE 1 – NATURE OF OPERATIONS

OVID THERAPEUTICS, INC.
NOTES TO CONSOLIDATED FINANCIAL STATEMENTS

Ovid Therapeutics Inc. (the “Company”) was incorporated under the laws of the state of Delaware on April 1, 2014 and maintains its principal executive office in New
York,  New  York.  The  Company  commenced  operations  on  April  1,  2014  (date  of  inception).  The  Company  is  a  biopharmaceutical  company  focused  exclusively  on
developing impactful medicines for patients and families living with rare neurological disorders.

Since its inception, the Company has devoted substantially all of its efforts to business development, research and development, recruiting management and technical
staff, and raising capital, and has financed its operations through issuance of convertible preferred stock (“Preferred Stock”), common stock and other equity instruments.
The  Company  is  subject  to  risks  and  uncertainties  common  to  early-stage  companies  in  the  biotechnology  industry,  including,  but  not  limited  to,  development  and
regulatory success, development by competitors of new technological innovations, dependence on key personnel, protection of proprietary technology, compliance with
government regulations, and ability to secure additional capital to fund operations.

Historically, the Company’s major sources of cash have been comprised of proceeds from various public and private offerings of its capital stock and interest income. As
of December 31, 2020, the Company had approximately $72.0 million in cash and cash equivalents. Since inception, the Company has generated $12.6 million in revenue
as part of the Company’s license and collaboration agreement (the “Angelini License Agreement”) with Angelini Pharma Rare Diseases AG (“Angelini”). The Company
has incurred recurring losses, has experienced recurring negative operating cash flows and requires significant cash resources to execute its business plans. The Company
has an accumulated deficit of $294.2 million as of December 31, 2020, working capital of $52.8 million and had cash outflows from operating activities of $51.6 million
for the year ended December 31, 2020.

The Company has incurred operating losses since inception and expects to continue to incur net losses for at least the next several years and ongoing operations are highly
dependent on the Company’s ability to obtain additional sources of funding. Management has identified these conditions or events, which, considered in the aggregate,
raise substantial doubt about our ability to continue as a going concern, including the risk that the Company will be unable to raise adequate additional capital to fund
operations through at least the next 12 months from the date of filing of this Annual Report on Form 10-K.  Management’s response to these conditions and events is that
the successful closing of the Takeda License and Termination Agreement with Takeda (see note 12) will provide the liquidity needed to alleviate the substantial doubt
referred to above.  As described in note 12, there are certain conditions to close the Takeda License and Termination Agreement, however management has determined
that the likelihood of not closing in the first half of 2021 is remote.  

We  have  implemented  business  continuity  plans  designed  to  address  and  mitigate  the  impact  of  the  COVID-19  pandemic  on  our  business.    The  extent  to  which  the
ongoing COVID-19 pandemic impacts our business, our clinical development and regulatory efforts, our corporate development objectives and the value of and market
for our common stock, will depend on future developments that are highly uncertain and cannot be predicted with confidence at this time, such as the ultimate duration of
the pandemic, travel restrictions, quarantines, social distancing and business closure requirements in the U.S., Europe and other countries, and the effectiveness of actions
taken globally to contain and treat the disease.  The global economic slowdown, the overall disruption of global healthcare systems and the other risks and uncertainties
associated with the pandemic could have a material adverse effect on our business, financial condition, results of operations and growth prospects.

In addition, we are subject to other challenges and risks specific to our business and our ability to execute on our strategy, as well as risks and uncertainties common to
companies in the pharmaceutical industry with development and commercial operations, including, without limitation, risks and uncertainties associated with: obtaining
regulatory  approval  of  our  late-stage  product  candidates;  delays  or  problems  in  the  supply  of  our  products,  loss  of  single  source  suppliers  or  failure  to  comply  with
manufacturing  regulations;  identifying,  acquiring  or  in-licensing  additional  products  or  product  candidates;  pharmaceutical  product  development  and  the  inherent
uncertainty of clinical success; and the challenges of protecting and enhancing our intellectual property rights; complying with applicable regulatory requirements.  In
addition, to the extent the ongoing COVID-19 pandemic adversely affects our business and results of operations, it may also have the effect of heightening many of the
other risks and uncertainties discussed above.

NOTE 2 – SUMMARY OF SIGNIFICANT ACCOUNTING POLICIES

(A) Basis of Presentation and Consolidation

The accompanying consolidated financial statements have been prepared in conformity with accounting principles generally accepted in the United States of America
(“GAAP”) and include the accounts of Ovid Therapeutics Inc. and its wholly-owned subsidiary, Ovid Therapeutics Hong Kong Limited.  All intercompany transactions
and balances have been eliminated in consolidation.

F-8

 
 
 
 
 
 
(B) Use of Estimates

The preparation of financial statements in conformity with GAAP requires management to make estimates and assumptions that affect the reported amounts of assets and
liabilities and disclosure of contingent assets and liabilities at the date of the financial statements and the reported amounts of expenses during the reporting period. Actual
results could differ materially from those estimates.

(C) Risks and Uncertainties

The Company is subject to risks common to companies in the development stage including, but not limited to, dependency on the clinical and commercial success of its
drug  candidates,  ability  to  obtain  regulatory  approval  of  its  drug  candidates,  the  need  for  substantial  additional  financing  to  achieve  its  goals,  uncertainty  of  broad
adoption of its approved products, if any, by physicians and consumers, and significant competition and untested manufacturing capabilities.

(D) Deferred Transaction Costs

Deferred transaction costs, primarily consisted of direct incremental legal, accounting, and other fees related to the Company’s offering of its capital stock are capitalized
as incurred. The deferred transaction costs are offset against proceeds upon the consummation of an offering.

(E) Comprehensive Loss

Comprehensive  loss  includes  net  loss  as  well  as  other  changes  in  stockholders’  equity  that  result  from  transactions  and  economic  events  other  than  those  with
stockholders.

(F) Collaboration Arrangement

License and Collaboration Agreement with Takeda Pharmaceutical Company Limited

Under the terms of the current license and collaboration agreement with Takeda Ovid and Takeda are sharing 50/50 in the drug development, the Company records 50%
of the development costs in research and development.  When Ovid incurs the majority of the costs and Takeda transfers a payment to Ovid to equalize the costs, Ovid
records the participation by Takeda as a reduction of its research and development expenses, as the parties under the collaboration are sharing in the costs and the payment
represents reimbursement of costs by Takeda. When Takeda incurs the majority of the costs and Ovid transfers a payment to Takeda (to equalize the costs), Ovid records
the participation in Takeda’s expenses as research and development costs in its statement of operations, as Ovid and Takeda are sharing in the research and development
activities and this participation represents Ovid’s share of the research and development costs in the specific period.

(G) Cash and Cash Equivalents

The Company’s cash and cash equivalents consist of cash held in checking accounts and money market funds. The Company considers all highly liquid investments with
an original maturity date of three months or less to be cash and cash equivalents. Accounts held at U.S. financial institutions are insured by the FDIC up to $250,000.
Cash balances could exceed insured amounts at any given time.

(H) Short-term Investments

Short-term investments consist of debt securities with maturities greater than three months from the date of purchase.  The Company classifies all of its investments as
available-for-sale securities. Debt securities are recorded at fair value with unrealized gains and losses included in other comprehensive income (loss) as a component of
stockholders’ equity until realized. Realized gains and losses, amortization and accretion of premiums and discounts are included within net loss.

(I) Property and Equipment

Property and equipment are stated at cost and depreciated over their estimated useful lives of three years using the straight-line method. Repairs and maintenance costs are
expensed. The Company reviews the recoverability of all long-lived assets, including the related useful life, whenever events or changes in circumstances indicate that the
carrying amount of a long-lived asset might not be recoverable.

(J) Research and Development Expenses

The  Company  expenses  the  cost  of  research  and  development  as  incurred.  Research  and  development  expenses  comprise  costs  incurred  in  performing  research  and
development activities, including clinical trial costs, manufacturing costs for both clinical and pre-clinical materials as well as other contracted services, license fees, and
other  external  costs.  Nonrefundable  advance  payments  for  goods  and  services  that  will  be  used  in  future  research  and  development  activities  are  expensed  when  the
activity is performed or when the goods have been received, rather than when the cost is incurred, in accordance with ASC 730, Research and Development.

F-9

 
 
 
 
 
 
 
 
 
 
 
 
 
(K) Stock-Based Compensation

The Company accounts for its stock-based compensation in accordance with ASC 718, Compensation—Stock Compensation, which establishes accounting for stock-
based  awards  granted  to  employees  for  services  and  requires  companies  to  expense  the  estimated  fair  value  of  these  awards  over  the  requisite  service  period.  The
Company estimates the fair value of all awards granted using the Black-Scholes valuation model. Key inputs and assumptions include the expected term of the option,
stock price volatility, risk-free interest rate, dividend yield, stock price and exercise price. Many of the assumptions require significant judgment and any changes could
have a material impact in the determination of stock-based compensation expense. The Company elected an accounting policy to record forfeitures as they occur. The
Company recognizes employee stock-based compensation expense based on the fair value of the award on the date of the grant. The compensation expense is recognized
over the vesting period under the straight-line method.

The Company accounts for options awards granted to nonemployee consultants and directors in accordance with ASU 2018-07, Compensation – Stock Compensation
(Topic  718):  Improvements  to  Nonemployee  Share-Based  Payment  Accounting.  The  fair  value  of  the  option  issued  or  committed  to  be  issued  is  used  to  measure  the
transaction, as this is more reliable than the fair value of the services received. The fair value is measured at the value of the Company’s common stock award at the
earlier of the date that the commitment for performance by the counterparty has been reached or the counterparty’s performance is complete.

(L) Fair Value of Financial Instruments

Financial Accounting Standards Board (“FASB”) guidance specifies a hierarchy of valuation techniques based on whether the inputs to those valuation techniques are
observable  or  unobservable.  Observable  inputs  reflect  market  data  obtained  from  independent  sources,  while  unobservable  inputs  reflect  market  assumptions.  The
hierarchy  gives  the  highest  priority  to  unadjusted  quoted  prices  in  active  markets  for  identical  assets  or  liabilities  (Level  1  measurement)  and  the  lowest  priority  to
unobservable inputs (Level 3 measurement). 
The three levels of the fair value hierarchy are as follows:

•

•

•

Level 1—Unadjusted quoted prices in active markets for identical assets or liabilities that the reporting entity has the ability to access at the measurement
date.  Level  1  primarily  consists  of  financial  instruments  whose  value  is  based  on  quoted  market  prices  such  as  exchange-traded  instruments  and  listed
equities.  The  Company’s  Level  1  assets  consisted  of  money  market  funds  and  short-term  investments  totaling  $70.1  million  and  $76.2  million  as  of
December 31, 2020 and 2019, respectively.

Level 2—Inputs other than quoted prices included within Level 1 that are observable for the asset or liability, either directly or indirectly (e.g., quoted
prices of similar assets or liabilities in active markets, or quoted prices for identical or similar assets or liabilities in markets that are not active). Level 2
includes  financial  instruments  that  are  valued  using  models  or  other  valuation  methodologies.  The  Company  had  no  Level  2  assets  or  liabilities  as  of
December 31, 2020 and 2019.

Level 3—Unobservable inputs for the asset or liability. Financial instruments are considered Level 3 when their fair values are determined using pricing
models, discounted cash flows or similar techniques and at least one significant model assumption or input is unobservable. The Company had no Level 3
assets or liabilities as of December 31, 2020 and 2019.

The carrying amounts reported in the balance sheets for cash and cash equivalents, related-party receivables, other current assets, accounts payable, accrued expenses, and
current related-party payables approximate their fair value based on the short-term maturity of these instruments.

(M) Income Taxes

The Company accounts for income taxes under the asset and liability method, which requires deferred tax assets and liabilities to be recognized for the estimated future
tax consequences attributable to differences between financial statement carrying amounts and respective tax bases of existing assets and liabilities, as well as for net
operating loss carryforwards and research and development credit. Valuation allowances are provided if it is more likely than not that some portion or all of the deferred
tax assets will not be realized.  The impact of a change in the tax laws is recorded in the period in which the law is enacted.

(N) Net Loss Per Common Share

Basic and diluted net loss per common share is determined by dividing net loss attributable to common stockholders by the weighted-average common shares outstanding
during the period. For all periods presented, stock options have been excluded from the calculation because their effect would be anti-dilutive. Therefore, the weighted-
average shares outstanding used to calculate both basic and diluted loss per common share are the same. Under the terms of the Series A Preferred Stock issued in 2019,
Preferred  stockholders  do  not  share  in  losses  of  the  Company  and  have  no  obligation  to  fund  losses  or  transfer  assets.    Since  there  is  a  loss,  diluted  EPS  should  be
computed in the same manner as basic EPS and because no potential common shares shall be included in the computation of any diluted per-share amounts when a loss
exists, the Series A Preferred Stock should be excluded from the computation of basic and diluted EPS.

F-10

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
The following potentially dilutive securities have been excluded from the computations of diluted weighted-average shares outstanding as they would be anti-dilutive:

Stock options to purchase common stock
Series A convertible preferred stock

(O) Segment Data

For the Year Ended December 31,

2020
10,403,420   
3,250   

2019
7,405,295 
7,762

The Company manages its operations as a single segment for the purposes of assessing performance and making operating decisions.

(P) Retirement Plan

The Company maintains a 401(k)-retirement plan for its employees that is intended to qualify under Sections 401(a) and 501(a) of the U.S. Internal Revenue Code of
1986,  as  amended  (“Code”).  The  Company  provides  all  active  employees  with  a  100%  matching  contribution  equal  to  3%  of  an  employee’s  eligible  compensation
deferred and 50% matching contributions on employee contributions that are between 3% and 5% of an employee’s eligible compensation deferred. These safe harbor
contributions vest immediately.  For the years ended December 31, 2020 and 2019 the Company contributed $321,000 and $285,000, respectively.

(Q) Revenue Recognition

Under ASC 606, an entity recognizes revenue when its customer obtains control of promised goods or services, in an amount that reflects the consideration that the entity
expects  to  receive  in  exchange  for  those  goods  or  services.  In  applying  ASC  606,  the  Company  performs  the  following  five  steps:  (i)  identify  the  contract(s)  with  a
customer; (ii) identify the promises and performance obligations in the contract; (iii) determine the transaction price; (iv) allocate the transaction price to the performance
obligations in the contract; and (v) recognize revenue when (or as) it satisfies the performance obligations. The Company only applies the five-step model to contracts
when it is probable that it will collect the consideration to which it is entitled in exchange for the goods or services we transfer to the customer. At contract inception, once
the  contract  is  determined  to  be  within  the  scope  of  ASC  606,  the  Company  assesses  the  goods  or  services  promised  within  each  contract,  determines  those  that  are
performance obligations and assesses whether each promised good or service is distinct. The Company then recognizes as revenue the amount of the transaction price that
is allocated to the respective performance obligation when (or as) the performance obligation is satisfied.

Prior to recognizing revenue, the Company makes estimates of the transaction price, including variable consideration that is subject to a constraint. Amounts of variable
consideration are included in the transaction price to the extent that it is probable that a significant reversal in the amount of cumulative revenue recognized will not occur
and when the uncertainty associated with the variable consideration is subsequently resolved.

If there are multiple distinct performance obligations, the Company allocates the transaction price to each distinct performance obligation based on its relative standalone
selling price. The standalone selling price is generally determined using expected cost and comparable transactions. Revenue for performance obligations recognized over
time is recognized by measuring the progress toward complete satisfaction of the performance obligations using an input measure.

Non-refundable  upfront  fees  allocated  to  licenses  that  are  not  contingent  on  any  future  performance  and  require  no  consequential  continuing  involvement  by  the
Company, are recognized as revenue when the license term commences and the licensed data, technology or product is delivered. The Company defers recognition of
upfront license fees if the performance obligations are not satisfied.

(R) Recent Accounting Pronouncements

Recent accounting standards which have been adopted

In June 2016, the FASB issued ASU No. 2016-13, Financial Instruments – Credit Losses (Topic 326): Measurement of Credit Losses on Financial Instruments.  This new
standard requires the measurement and recognition of expected credit losses for financial assets held at amortized cost, including loans and trade and other receivables.
ASU 2016-13 replaces the existing incurred loss impairment model with an expected loss methodology, which will result in more timely recognition of credit losses. The
standard also amends the impairment model for available-for-sale debt securities and requires entities to determine whether all or a portion of the unrealized loss on an
available-for-sale  debt  security  is  a  credit  loss.  Under  the  new  guidance,  an  entity  recognizes  an  allowance  for  credit  losses  on  available-for-sale  debt  securities  as  a
contra-account to the amortized cost basis rather than as a direct reduction of the amortized cost basis of the investment, as was previously required. ASU 2016-13 is
effective for annual reporting periods, and interim periods within those years, beginning after December 15, 2019. As of December 31, 2020, the Company did not hold
any debt securities with

F-11

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
credit losses, nor does it have any trade receivables. The adoption of this standard effective January 1, 2020 did not have a material impact on the Company’s consolidated
financial statements.

On August 29, 2018, the FASB issued ASU No. 2018-15, Intangibles – Goodwill and Other - Internal-Use Software (Subtopic 350-40) - which amends ASC 350-40 to
address a customer’s accounting for implementation costs incurred in a cloud computing arrangement (“CCA”) that is a service contract. ASU No. 2018-15 aligns the
accounting for costs incurred to implement a CCA that is a service arrangement with the guidance on capitalizing costs associated with developing or obtaining internal-
use software. Specifically, the ASU amends ASC 350 to include in its scope implementation costs of a CCA that is a service contract and clarifies that a customer should
apply ASC 350-40 to determine which implementation costs should be capitalized in a CCA that is considered a service contract. According to the standard the balance
sheet line item for the presentation of capitalized implementation costs should be the same as that for the prepayment of fees related to the hosting arrangement and the
manner in which an entity classifies the cash flows related to capitalized implementation costs should be the same as that in which it classifies the cash flows for the fees
related  to  the  hosting  arrangement.  ASU  2018-15  is  effective  for  the  Company  for  fiscal  years  beginning  after  December  15,  2019,  including  interim  periods  therein.
Entities are permitted to apply either a retrospective or prospective transition approach to adopt the guidance. The adoption of this standard effective January 1, 2020 did
not have a material impact on the Company’s consolidated financial statements and was adopted prospectively.

On  November  5,  2018,  the  FASB  issued  ASU  2018-18,  Collaborative  Arrangements  (Topic  808),  -  which  amends  ASC  808  to  clarify  when  transactions  between
participants  in  a  collaborative  arrangement  under  ASC  808  are  within  the  scope  of  the  FASB’s  new  revenue  standard,  ASU  2014-09  (codified  in  ASC  606).  The
amendments  require  the  application  of  ASC  606  existing  guidance  to  determine  the  units  of  account  that  are  distinct  in  a  collaborative  arrangement  for  purposes  of
identifying transactions with customers. If a unit of account within the collaborative arrangement is distinct and is with a customer, an entity shall apply the guidance in
Topic 606 to that unit of account. In a transaction between collaborative participants, an entity is precluded by ASU 2018-18 from presenting a transaction together with
“revenue  from  contracts  with  customers”  unless  the  unit  of  account  is  within  the  scope  of  ASC  606  and  the  entity  applies  the  guidance  in  ASC  606  to  such  unit  of
account. The amended guidance is effective for public business entities for fiscal years beginning after December 15, 2019, and interim periods within those fiscal years.
The retrospective adoption of this standard effective January 1, 2020 did not have a material impact on the Company’s consolidated financial statements.

In  October  2020,  the  FASB  issued  ASU  2020-10,  Codification  Improvements,  which  updates  various  codification  topics  by  clarifying  or  improving  disclosure
requirements. ASU 2020-10 is effective for annual and interim periods beginning after December 15, 2020. The Company early adopted ASU 2020-10 for the reporting
period ending December 31, 2020. The adoption of this update did not have a material effect on the Company s consolidated financial statements.

NOTE 3 – CASH EQUIVALENTS AND SHORT-TERM INVESTMENTS

All short-term investments are classified as available-for-sale. The following tables summarize the fair value of cash, cash equivalents, and short-term investments, as
well as gross unrealized holding gains and losses as of December 31, 2020 and December 31, 2019:

  Cash
  Money market funds
Total cash and cash equivalents

  U.S. treasury notes
Total short-term investments

  $

  $

  $
  $

Amortized

December 31, 2020

Gross
unrealized

Gross
unrealized

cost
1,977,320    $
70,056,610     
72,033,930    $

    holding gains     holding losses    
-    $
-     
-    $

-    $
-     
-    $

Fair

value
1,977,320 
70,056,610 
72,033,930 

-    $
-    $

-    $
-    $

-     
-    $

- 
- 

F-12

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
 
     
       
       
       
 
 
     
       
       
       
 
  Cash
  Money market funds
Total cash and cash equivalents

  U.S. treasury notes
Total short-term investments

  $

  $

  $
  $

December 31, 2019

Gross
unrealized

Gross
unrealized

Amortized

cost

501,537    $
41,395,607     
41,897,144    $

    holding gains     holding losses    
-    $
-     
-    $

-    $
-     
-    $

Fair

value

501,537 
41,395,607 
41,897,144 

34,839,500    $
34,839,500    $

2,469    $
2,469    $

-     
-    $

34,841,969 
34,841,969 

The Company did not hold any securities that were in an unrealized loss position for more than 12 months as of December 31, 2020 and 2019.

There were no material realized gains or losses on available-for-sale securities during the years ended December 31, 2020 and 2019. 

NOTE 4 – PROPERTY AND EQUIPMENT AND INTANGIBLE ASSETS

Property and equipment is summarized as follows:

Furniture and equipment
Less accumulated depreciation
Total property, plant and equipment, net

December 31,
2020

December 31,
2019

  $

  $

320,957    $
(185,337)    
135,620    $

193,717 
(125,354)
68,363  

Depreciation expense was $60,000 and $39,000 for the years ended December 31, 2020 and 2019 respectively.

Intangible assets, net of accumulated amortization, were $319,000 and $467,000 as of December 31, 2020 and December 31, 2019, respectively, and are included in other
assets. Amortization expense was $247,000 and $216,000 for the years ended December 31, 2020 and 2019, respectively.

NOTE 5 – ACCRUED EXPENSES

Accrued expenses consist of the following:

Clinical trials accrual
Payroll and bonus accrual
Professional fees accrual
Other

Total

December 31,
2020
4,175,497    $
3,845,441   
3,846,211   
165,536   
12,032,685    $

December 31,
2019
3,235,527 
2,728,495 
1,070,589 
232,095 
7,266,706  

  $

  $

NOTE 6 – STOCKHOLDERS’ EQUITY AND PREFERRED STOCK

The  Company’s  capital  structure  consists  of  common  stock  and  Preferred  Stock.  Pursuant  to  the  Company’s  amended  and  restated  certificate  of  incorporation,  as
amended, the Company is authorized to issue up to 125,000,000 shares of common stock and 10,000,000 shares of Preferred Stock. The Company has designated 10,000
of the 10,000,000 authorized shares of Preferred Stock as non-voting Series A Convertible Preferred Stock (“Series A Preferred Stock”).

The holders of common stock are entitled to one vote for each share held. The holders of common stock have no preemptive or other subscription rights, and there are no
redemption  or  sinking  fund  provisions  with  respect  to  such  shares.  Subject  to  preferences  that  may  apply  to  any  outstanding  series  of  Preferred  Stock,  holders  of  the
common stock are entitled to receive ratably any dividends declared on a non-cumulative basis. Shares of Series A Preferred Stock will be entitled to receive dividends at
a rate equal to (on an as-if-converted-to-common stock basis), and in the same form and manner as, dividends actually paid on shares of common stock. The common
stock is subordinate to all series of Preferred Stock with respect to rights upon liquidation, winding up and dissolution of the Company. The holders of common stock are
entitled to liquidation proceeds after all liquidation preferences for the Preferred Stock are satisfied.

F-13

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
 
     
       
       
       
 
 
     
       
       
       
 
 
 
 
 
 
 
 
 
 
 
   
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
In June 2018, the Company entered into a sales agreement (the “2018 ATM agreement”) with Cowen and Company, LLC (“Cowen”) under which the Company offered
and sold in “at the market offerings,” from time to time at its sole discretion, shares of its common stock having an aggregate offering price of up to $50.0 million through
Cowen acting as sales agent. During the year ended December 31, 2019, the Company sold 6,893,888 shares of its common stock under the 2018 ATM agreement for net
proceeds of $22.3 million after deducting sales agent commissions and other offering expenses payable by the Company, (the “ATM Offerings”).

In November 2020, the Company entered into a new sales agreement (the “2020 ATM agreement”) with Cowen and under which the Company may offer and sell in “at
the market offerings,” from time to time at its sole discretion, shares of its common stock having an aggregate offering price of up to $75.0 million through Cowen acting
as sales agent.

There  were  3,250  and  7,762  shares  of  Series  A  Preferred  Stock  outstanding  as  of  December  31,  2020  and  December  31,  2019,  respectively.  Each  share  of  Series  A
Preferred Stock is convertible into 1,000 shares of common stock at any time at the holder’s option. However, the holder will be prohibited, subject to certain exceptions,
from converting shares of Series A Preferred Stock into shares of common stock if, as a result of such conversion, the holder, together with its affiliates, would own more
than, at the written election of the holder, either 9.99% or 14.99% of the total number of shares of common stock then issued and outstanding, which percentage may be
changed at the holder’s election to any other number less than or equal to 19.99% upon 61 days’ notice to the Company; provided, however, that effective 61 days after
delivery of such notice, such beneficial ownership limitations shall not be applicable to any holder that beneficially owns either 10.0% or 15.0%, as applicable based on
the holder’s initial written election noted above, of the total number of shares of common stock issued and outstanding immediately prior to delivery of such notice. In the
event  of  a  liquidation,  dissolution,  or  winding  up  of  the  Company,  holders  of  Series  A  Preferred  Stock  will  receive  a  payment  equal  to  $0.001  per  share  of  Series  A
Preferred Stock before any proceeds are distributed to the holders of common stock.

In December 2020, entities affiliated with Biotechnology Value Fund, L.P. elected to convert an aggregate of 2,256 shares of Series A Preferred Stock owned by such
holders into an aggregate of 2,256,000 shares of the Company’s common stock.

In August 2020, the Company sold 6,250,000 shares of its common stock at a public offering price of $8.00 per share, for net proceeds of $46.7 million after deducting
underwriting discounts and commissions and other offering expenses payable by the Company, (the “August 2020 Offering”).

In May 2020, entities affiliated with Biotechnology Value Fund, L.P. elected to convert an aggregate of 2,256 shares of Series A Preferred Stock owned by such holders
into an aggregate of 2,256,000 shares of the Company’s common stock.

In  October  and  November  2019,  the  Company  sold  10,350,000  shares  of  its  common  stock,  which  included  the  full  exercise  of  the  underwriters’  option  to  purchase
additional shares, and 4,000 shares of Series A Preferred Stock at a public offering price of $2.50 and $2,500 per share, respectively, for net proceeds of $33.5 million
after deducting underwriting discounts and commissions and other offering expenses payable by the Company, (the “October 2019 Offering”).

In  September  2019,  the  Company  entered  into  an  exchange  agreement  with  entities  affiliated  with  Biotechnology  Value  Fund,  L.P.  (the  “Exchanging  Stockholders”),
pursuant to which the Company exchanged an aggregate of 1,262,000 shares of the Company’s common stock owned by the Exchanging Stockholders for an aggregate of
1,262  shares  of  the  Company’s  Series  A  Preferred  Stock  (the  “Exchange  Shares”).  The  Exchange  Shares  were  issued  without  registration  under  the  Securities  Act  of
1933, as amended, in reliance on the exemption from registration contained in Section 3(a)(9) of the Securities Act. 

In February 2019, the Company sold 13,993,778 shares of its common stock and 2,500 shares of Series A Preferred Stock at a public offering price of $2.00 and $2,000
per share, respectively, for net proceeds of $30.5 million after deducting underwriting discounts and commission and other offering expenses payable by the Company
(the “February 2019 Offering”).

Dividends

No dividends on the common stock shall be declared and paid unless dividends on the Preferred Stock have been declared and paid. Through December 31, 2020, the
Company has not declared any dividends.

NOTE 7 – STOCK-BASED COMPENSATION

On August 29, 2014, the Company’s Board of Directors adopted and approved the 2014 Equity Incentive Plan (the “2014 Plan”), which authorized the Company to grant
shares of common stock in the form of incentive stock options, nonstatutory stock options, stock appreciation rights, restricted stock and restricted stock units. The types
of stock-based awards, including share purchase rights amount, terms, and exercisability provisions of grants are determined by the Company’s Board of Directors.

The Company's Board of Directors adopted, and the Company's stockholders approved the 2017 equity incentive plan (“2017 Plan”), which became effective immediately
prior to the execution of the underwriting agreement related to the IPO on May 4, 2017. The initial reserve of shares of common stock that may be issued under the 2017
Plan was 3,052,059 shares. The 2017 Plan provides

F-14

 
 
 
 
 
 
 
 
 
 
 
 
for the grant of incentive stock options, non-statutory stock options, restricted stock awards, restricted stock unit awards, stock appreciation rights, performance-based
stock  awards,  and  other  forms  of  stock-based  awards.   Additionally,  the  2017  Plan  provides  for  the  grant  of  performance  cash  awards.  The  Company's  employees,
officers, directors and consultants and advisors are eligible to receive awards under the 2017 Plan.  Upon the adoption of the 2017 Plan, no further awards will be granted
under the 2014 Plan. Pursuant to the terms of the 2017 Plan, on each January 1st, the plan limit shall be increased by the lesser of (x) 5% of the number of shares of
common  stock  outstanding  as  of  the  immediately  preceding  December  31  and  (y)  such  lesser  number  as  the  Board  of  Directors  may  determine  in  its  discretion. On
January 1, 2019, an additional 1,232,705 shares were reserved for issuance under the 2017 Plan. As of December 31, 2019, there were 2,199,765 shares of the Company’s
common stock reserved for issuance under the 2017 Plan. On January 1, 2020, an additional 2,735,516  shares  were  reserved  for  issuance  under  the  2017  Plan.  As  of
December 31, 2020, there were 1,771,772 shares of the Company’s common stock reserved for issuance under the 2017 Plan.

The  Company's  Board  of  Directors  adopted,  and  the  Company's  stockholders  approved  the  2017  employee  stock  purchase  plan  (the  “2017  ESPP”),  which  became
effective immediately prior to the execution of the underwriting agreement related to the IPO on May 4, 2017. The initial reserve of shares of common stock that may be
issued under the 2017 ESPP was 279,069 shares. On September 20, 2017, the Company’s Compensation Committee approved an offering period under the 2017 ESPP,
which began on October 20, 2017. The ESPP allows employees to purchase common stock of the Company at a 15% discount to the market price on designated purchase
dates. During the years ended December 31, 2020 and 2019, 105,464 and 80,542 shares were purchased under the ESPP and the Company recorded expense of $152,973
and $109,319, respectively. The number of shares of common stock reserved for issuance under the 2017 ESPP will automatically increase on January 1 of each year,
beginning on January 1, 2018 and continuing through and including January 1, 2027, by the lesser of (i) 1% of the total number of shares of the Company’s capital stock
outstanding on December 31 of the preceding calendar year, (ii) 550,000 shares or (iii) such lesser number of shares determined by our Board. On January 1, 2019, an
additional 246,541 shares were reserved for issuance under the 2017 ESPP. No shares were reserved for issuance under the 2017 ESPP during the year ended December
31, 2020. As of December 31, 2020, there were 553,552 shares of the Company’s common stock reserved for issuance under the 2017 ESPP.

Unless specified otherwise in an individual option agreement, stock options granted under the 2014 Plan and 2017 Plan generally have a ten-year term and a four-year
graded vesting period. The vesting requirement is generally conditioned upon the grantee’s continued service with the Company during the vesting period. Once vested,
all  awards  are  exercisable  from  the  date  of  grant  until  they  expire.  The  option  grants  are  non-transferable.  Vested  options  generally  remain  exercisable  for  90  days
subsequent to the termination of the option holder’s service with the Company. In the event of option holder’s death or disability while employed by or providing service
to the Company, the exercisable period extends to 12 months.

Performance-based option awards generally have similar vesting terms, with vesting occurring on the date the performance condition is achieved and expire in accordance
to the specific terms of the agreement. At December 31, 2020, there were 125,000 performance-based options outstanding and unvested that include options to vest upon
the achievement of certain research and development milestones. 

F-15

 
The fair value of options granted during the years ended December 31, 2020 and 2019 was estimated using the Black-Scholes option valuation model. The inputs for the
Black-Scholes option valuation model require management’s significant assumptions and are detailed in the table below. The risk-free interest rates were based on the rate
for  U.S.  Treasury  securities  at  the  date  of  grant  with  maturity  dates  approximately  equal  to  the  expected  life  at  the  grant  date.  The  expected  life  was  based  on  the
simplified method in accordance with the SEC Staff Accounting Bulletin No. Topic 14D. The expected volatility was estimated based on historical volatility information
of peer companies that is publicly available.

All assumptions used to calculate the grant date fair value of nonemployee options are generally consistent with the assumptions used for options granted to employees. In
the event the Company terminates any of its consulting agreements, the unvested options underlying the agreements would also be cancelled.

The  Company  granted  10,000  and  175,000  stock  options  to  nonemployee  consultants  for  services  rendered  during  the  years  ended  December  31,  2020  and  2019,
respectively.  There  were  32,500  and  145,204  unvested  nonemployee  options  outstanding  as  of  December  31,  2020  and  2019,  respectively.  Total  expense  recognized
related to the nonemployee stock options for the years ended December 31, 2020 and 2019 was $257,431 and $51,666, respectively. During the year ended December 31,
2019,  the  Company  recognized  a  credit  of  $17,000  related  to  the  nonemployee  stock  options  including  the  modification  of  certain  options  in  connection  with
the  separation  and  consulting  agreement  with  Dr.  During  (see  Note  11).  Total  unrecognized  compensation  expenses  related  to  the  nonemployee  stock  options  was
$186,823 as of December 31, 2020. During the years ended December 31, 2020, and 2019, the Company recognized $115,240 and zero, respectively, in expenses for
nonemployee performance-based option awards.

The Company granted 3,573,160 and 3,372,513 stock options to employees during the years ended December 31, 2020 and 2019, respectively. There were 4,975,262 and
3,963,544 unvested employee options outstanding as of December 31, 2020 and 2019, respectively. Total expense recognized related to the employee stock options for the
years ended December 31, 2020 and 2019 was $7.1 million and $5.0 million, respectively. Total unrecognized compensation expense related to employee stock options
was  $12.2  million  as  of  December  31,  2020.  During  the  years  ended  December  31,  2020  and  2019,  the  Company  recognized  $2,340,808  and  $9,391  in  expenses  for
employee performance-based option awards.

The Company’s stock-based compensation expense was recognized in operating expenses as follows:

Research and development
General and administrative

Total

Stock options
Employee Stock Purchase Plan

Total

For the Year Ended December 31,

2020
2,779,758 
4,745,596 
7,525,354 

 $

 $

2019
2,391,909 
2,813,883 
5,205,792

For the Year Ended December 31,

2020
7,372,381 
152,973 
7,525,354 

 $

 $

2019
5,096,473 
109,319 
5,205,792

  $

  $

  $

  $

The fair value of employee options granted during the years ended December 31, 2020 and 2019, respectively, was estimated by utilizing the following assumptions:

Volatility
Expected term in years
Dividend rate
Risk-free interest rate
Fair value of option on grant date

F-16

For the Year Ended December 31,

2020
Weighted
Average

2019
Weighted
Average

81.48%   

5.88 
0.00%   
0.58%   
 $
2.62 

81.87%
6.07 
0.00%
2.04%
2.26

  $

 
 
 
 
 
 
 
 
 
 
   
  
 
 
 
 
 
 
 
 
 
 
 
   
  
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
   
  
   
   
 
 
The  fair  value  of  nonemployee  options  granted  and  remeasured  during  the  years  ended  December  31,  2020  and  2019,  respectively,  was  estimated  by  utilizing  the
following assumptions:

Volatility
Expected term in years
Dividend rate
Risk-free interest rate
Fair value of option on grant date

For the Year Ended December 31,

2020
Weighted
Average

2019
Weighted
Average

74.37%   

5.64 
0.00%   
2.32%   
 $
1.18 

74.56%
5.30 
0.00%
2.37%
1.07

  $

The following table summarizes the number of options outstanding and the weighted average exercise price:

Options Outstanding at December 31, 2018

Vested and exercisable at December 31, 2018

Granted
Exercised
Forfeited
Options Outstanding December 31, 2019

Vested and exercisable at December 31, 2019

Granted
Exercised
Forfeited

Options Outstanding December 31, 2020

Vested and exercisable at December 31, 2020

  Weighted  
Average
Exercise
Price

  Weighted  
Average
  Remaining  
  Contractual  
  Life in Years  

  Aggregate
Intrinsic
Value

8.10     

7.88     

2.93     
-     
6.43     
5.82     

7.93     

3.93     
1.82     
5.00     
5.26     
6.45     

7.89    $

153,485 

7.20    $

153,485 

9.56     

8.01    $ 4,488,930 

6.53    $

356,443 

9.68     
-     

7.59    $

652,438 

6.13    $

445,599

  Number of

Shares
4,714,383    $

2,337,931    $

3,547,513     

- 

(856,601)    
7,405,295    $

3,296,547    $

3,583,160     
(165,384)   
(415,526)    
    10,403,420    $
5,395,658    $

At December 31, 2020, there was $12.3 million of unamortized share–based compensation expense, which is expected to be recognized over a remaining average vesting
period of 3.04 years.

NOTE 8 – INCOME TAXES

At December 31, 2020, the Company has available approximately $238.6 million and $186.7 million of unused NOL carryforwards for federal and state tax purposes,
respectively, that may be applied against future taxable income. The Company also has approximately $165.4 million of unused NOL carryforwards for New York City
purposes. The NOL carryforwards will begin to expire in the year 2035 if not utilized prior to that date. There is no provision for income taxes because the Company has
historically incurred operating losses and maintains a full valuation allowance against its net deferred tax assets. The valuation allowance increased by approximately
$13.3 million and $22.5 million during the years 2020 and 2019, respectively.

The Company may be subject to the NOL utilization provisions of Section 382 of the Code. The effect of an ownership change would be the imposition of an annual
limitation  on  the  use  of  NOL  carryforwards  attributable  to  periods  before  the  change.  The  amount  of  the  annual  limitation  depends  upon  the  value  of  the  Company
immediately before the change, changes to the Company’s capital during a specified period prior to the change, and the federal published interest rate. The Company has
not completed a Section 382 analysis to determine if a change in ownership has occurred. Until an analysis is completed, there can be no assurance that the existing net
operating loss carry-forwards or credits are not subject to significant limitation.

The Company’s reserves related to taxes are based on a determination of whether and how much of a tax benefit taken by the Company in its tax filings or positions is
more likely than not to be realized following resolution of any potential contingencies related to the tax benefit. For the years ended December 31, 2020 and 2019, the
Company had no unrecognized tax benefits or related interest and penalties accrued. The Company has not yet conducted a study of research and development credit
carryforwards. This study may result in an adjustment to the Company’s research and development credit carryforwards; however, until a study is completed, and any
adjustment is known, no amounts are being presented as an uncertain tax position. A full valuation allowance has been provided against the Company’s research and
development credits and, if an adjustment is required, this adjustment would be offset by an adjustment to the valuation allowance. Thus, there would be no impact to the
balance  sheet  or  statement  of  operations  if  an  adjustment  were  required.  The  Company  would  recognize  both  accrued  interest  and  penalties  related  to  unrecognized
benefits in income tax

F-17

 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
   
  
   
   
 
 
 
 
   
 
 
   
 
 
   
 
 
 
   
 
 
 
 
   
 
 
 
   
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
   
   
  
   
  
      
  
   
      
  
   
   
   
  
   
  
   
      
  
   
 
 
 
 
 
expense. The Company’s uncertain tax positions yet to be determined would be related to years that remain subject to examination by relevant tax authorities. Since the
Company is in a loss carryforward position, the Company is generally subject to examination by the U.S. federal, state and local income tax authorities for all tax years in
which a loss carryforward is available.

The tax effects of temporary differences that gave rise to significant portions of the deferred tax assets and liabilities were as follows:

Deferred tax assets/liabilities:

Net operating loss carryovers
Research and development tax credits
Share-based compensation
Accrued compensation
Depreciation
Charitable contributions
Intangible assets

Total gross deferred tax assets/liabilities
Valuation allowance
Net deferred tax assets (liabilities)

December 31,

2020

2019

  $

  $

74,064,673    $
5,458,004   
4,978,370   
514,316   
(29,760)  
87,120   
4,742,031   
89,814,754 
(89,814,754)   
-    $

57,288,334 
3,351,315 
6,606,889 
898,067 
(22,026)
132,072 
8,208,519 
76,463,170 
(76,463,170)
-  

A reconciliation of the statutory U.S. Federal rate to the Company’s effective tax rate is as follows:

Federal income tax benefit at statutory rate

State income tax, net of federal benefit (1)
Permanent items
Change in valuation allowance
Research and development tax credits
Other

Effective income tax (benefit) expense rate

December 31,

2020

2019

(21.00)    
6.15 
0.75 
16.72 
(2.64)    
0.02 

0%    

(21.00)
(13.80)
0.50 
37.14 
(2.67)
(0.17)
0%

(1) Inclusive of $5.8 million deferred tax benefit due to change in apportionment

NOTE 9 – COMMITMENTS AND CONTINGENCIES

License Agreements

On  March  26,  2015,  the  Company  entered  into  an  exclusive  agreement  with  H.  Lundbeck  A/S  (“Lundbeck”)  for  a  worldwide  perpetual  licensing  right  related  the
research, development and commercialization of OV101. On May 10, 2019, the parties amended the license agreement.

Pursuant to the Lundbeck license agreement, as amended, the Company agreed to make milestone payments totaling up to $189.0 million upon the achievement of certain
development, regulatory and sales milestones. The first payment of $1.0 million is due upon the successful completion of the first Phase 3 trial for a product in which
OV101 is an active ingredient. In addition, the agreement calls for the Company to pay royalties for an initial term based on a low double-digit percentage of sales and
provides for the reduction of royalties in certain limited circumstances.  As of December 31, 2020, none of these contingent payments were considered probable.

In  December  2016,  the  Company  entered  into  a  license  agreement  with  Northwestern  University,  or  Northwestern,  pursuant  to  which  Northwestern  granted  us  an
exclusive, worldwide license to patent rights in certain inventions, or the Northwestern Patent Rights, which relate to a specific compound and related methods of use for
such compound, along with certain Know-How related to the practice of the inventions claimed in the Northwestern Patents.  

Under the Northwestern agreement, the Company was granted exclusive rights to research, develop, manufacture and commercialize products utilizing the Northwestern
Patent  Rights  for  all  uses.  The  Company  has  agreed  that  it  will  not  use  the  Northwestern  Patent  Rights  to  develop  any  products  for  the  treatment  of  cancer,  but
Northwestern may not grant rights in the technology to others for use in cancer. The Company also has an option, exercisable during the term of the agreement to an
exclusive license under certain intellectual property rights covering novel compounds with the same or similar mechanism of action as the primary compound that is

F-18

 
 
 
 
 
 
 
 
 
 
 
 
 
   
   
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
  
 
 
 
 
 
 
 
 
 
 
 
   
   
   
   
   
   
   
   
   
   
   
 
   
  
   
  
 
 
 
   
 
     
 
 
 
 
the subject of the license agreement.  Northwestern has retained the right, on behalf of itself and other non-profit institutions, to use the Northwestern Patent Rights and
practice  the  inventions  claimed  therein  for  educational  and  research  purposes  and  to  publish  information  about  the  inventions  covered  by  the  Northwestern  Patent
Rights.  

Upon entry into the Northwestern agreement, the Company paid an upfront non-creditable one-time license issuance fee of $75,000, and is required to pay an annual
license maintenance fee of $20,000, which will be creditable against any royalties payable to Northwestern following first commercial sale of licensed products under the
agreement.   The  Company  is  responsible  for  all  ongoing  costs  of  filing,  prosecuting  and  maintaining  the  Northwestern  Patents,  but  also  has  the  right  to  control  such
activities using its own patent counsel.  In consideration for the rights granted to the Company under the Northwestern agreement, the Company is required to pay to
Northwestern up to an aggregate of $5.3 million upon the achievement of certain development and regulatory milestones for the first product covered by the Northwestern
Patents, and, upon commercialization of any such products, will be required to pay to Northwestern a tiered royalty on net sales of such products by the Company, its
affiliates  or  sublicensees,  at  percentages  in  the  low  to  mid  single-digits,  subject  to  standard  reductions  and  offsets.   The  Company’s  royalty  obligations  continue  on  a
product-by-product and country-by-country basis until the later of the expiration of the last-to-expire valid claim in a licensed patent covering the applicable product in
such  country  and  10  years  following  the  first  commercial  sale  of  such  product  in  such  country.    If  the  Company  sublicenses  a  Northwestern  Patent  Right,  it  will  be
obligated to pay to Northwestern a specified percentage of sublicense revenue received by the Company, ranging from the high single digits to the low-teens.  

The Northwestern agreement requires that the Company use commercially reasonable efforts to develop and commercialize at least one product that is covered by the
Northwestern Patent Rights.  

Unless earlier terminated, the Northwestern agreement will remain in force until the expiration of the Company’s payment obligations thereunder.  The Company has the
right to terminate the agreement for any reason upon prior written notice or for an uncured material breach by Northwestern.  Northwestern may terminate the agreement
for the Company’s uncured material breach or insolvency.

As of December 31, 2020, none of these contingent payments were considered probable.

Contingencies

Liabilities for loss contingencies arising from claims, assessments, litigation, fines, and penalties and other sources are recorded when it is probable that a liability has
been incurred and the amount can be reasonably estimated. Legal costs incurred in connection with loss contingencies are expensed as incurred. The Company is not
currently involved in any legal matters arising in the normal course of business.

Under  the  terms  of  their  respective  employment  agreements,  each  of  our  named  executive  officers  is  eligible  to  receive  severance  payments  and  benefits  upon  a
termination  without  “cause”  or  due  to  “permanent  disability,”  or  upon  “resignation  for  good  reason,”  contingent  upon  the  named  executive  officer’s  delivery  to  the
Company of a satisfactory release of claims, and subject to the named executive officer’s compliance with non-competition and non-solicitation restrictive covenants for
two years following the termination date.

Pursuant to the Northwestern agreement, Northwestern granted the Company an exclusive license to certain patent rights and know-how, including a patent application
covering  a  specified  composition  of  matter  (the  “Patent  Application”).    Northwestern  previously  entered  into  a  license  agreement  with  Catalyst  Pharmaceuticals,  Inc.
(“Catalyst”), dated August 27, 2009, pursuant to which Northwestern granted Catalyst rights under certain intellectual property rights covering a different composition of
matter (the “Catalyst License”).  In addition, the Company is a party to a confidential disclosure agreement with Catalyst, dated September 16, 2016 (the “CDA”). On
June 25, 2018, Catalyst sent a letter to Northwestern and the Company alleging, among other things, that Northwestern breached the Catalyst License by licensing the
Patent Application to the Company. Catalyst’s letter also asserted that the Company had breached its obligations under the CDA by allegedly failing to disclose that the
Company  had  a  license  to  the  Patent  Application,  and  that  a  further  breach  would  occur  if  the  Company  makes  any  use  of  information  obtained  under  the  CDA  in
connection with its development program arising from the rights granted under the license agreement.  Catalyst has asserted that the combined conduct of Northwestern
and the Company gives rise to various claims, including breach of contract, fraud, and tortious interference. The Company believes that Catalyst’s claims are without
merit and responded by letter dated June 28, 2018, which denies any and all liability to Catalyst, and further denies that Catalyst has been damaged in any way. On May
20, 2019, the Company entered into a Settlement Agreement with Catalyst (the “Settlement Agreement”), pursuant to which Catalyst released the Company from any and
all claims, known or unknown, arising from or related to the dispute between Catalyst and Northwestern, the license agreement, and/or the claims that Catalyst asserted
against the Company in the June 25, 2018 letter.  Under the Settlement Agreement the Company retains all rights and privileges previously granted to the Company under
the Northwestern license agreement.

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NOTE 10 – COLLABORATION AGREEMENT

Angelini Collaboration

On  July  9,  2020,  the  Company  entered  into  the  Angelini  License  Agreement  with  Angelini,  pursuant  to  which  the  Company  granted  to  Angelini  exclusive  rights  to
develop and commercialize OV101, a selective agonist of the GABAA receptor, for the treatment of Angelman syndrome in the European Economic Area as well as
Switzerland, the United Kingdom, Russia and Turkey (the “European Territory”).  The licenses granted to Angelini include sublicenses under the Lundbeck Agreement,
as  well  as  licenses  under  the  Company’s  patents  and  know-how  covering  OV101.   Angelini  will  be  responsible  for  conducting  any  clinical  trials  necessary  to  obtain
regulatory  approval  for  OV101  for  Angelman  syndrome  in  the  European  Territory,  and  the  Company  will  be  responsible  for  bearing  a  portion  of  the  costs  for  such
trials.    The  Company  will  also  be  responsible,  at  its  expense,  for  the  completion  of  certain  ongoing  clinical  trials  for  OV101,  to  the  extent  applicable  to  obtaining
regulatory approval for OV101 in the European Territory.  Angelini has the exclusive right, at its election, to develop and commercialize OV101 for the treatment of
Fragile X Syndrome in the European Territory.  The parties may also mutually agree to pursue additional indications for OV101 in the European Territory, and in such
case, Angelini would have the exclusive rights to commercialize in such additional indications. Angelini is required to use commercially reasonable efforts to conduct
development activities for OV101, and following regulatory approval, to commercialize OV101 in each approved indication.

In  conjunction  with  the  entry  into  the  Angelini  License  Agreement,  the  parties  entered  into  a  separate  supply  agreement,  pursuant  to  which  the  Company  will  be
responsible  for  supply  of  OV101  to  Angelini  for  development  and  commercialization  in  the  European  Territory,  through  its  existing  supply  relationship  with
Lundbeck.    The  Angelini  License  Agreement  also  provides  for  a  transfer,  at  Angelini’s  expense,  of  the  relevant  manufacturing  technology  from  the  Company  and
Lundbeck to Angelini, in order to enable Angelini to assume responsibility for its own manufacture and supply of OV101 in the future.

Under  the  Angelini  License  Agreement,  Angelini  made  an  upfront  payment  and  a  milestone  payment  related  to  the  transfer  of  a  specified  amount  of  compound  and
related information to the Company of $25.0 million during the year ended December 31, 2020.  Angelini will be required to make additional milestone payments to the
Company  upon  the  completion  of  the  specified  components  of  the  technology  transfer  and  achievement  of  specified  regulatory  milestones  for  OV101  in  Angelman
syndrome of up to $55.0 million in the aggregate, as well as up to €162.5 million ($199.9 million) in sales milestone payments for achievement of specified levels of net
sales  in  the  European  Territory.    In  addition,  Angelini  will  be  required  to  pay  tiered  royalties  on  net  sales  by  Angelini,  its  affiliates  or  sublicensees  at  double-digit
percentages above the teens, subject to certain standard reductions and offsets.  Royalties will be payable on a product-by-product and country-by-country basis until the
latest of the expiration of the licensed patents covering such product in such country, the expiration of market exclusivity for such product in such country, and fifteen
years from first commercial sale of such product in such country.

Either party may terminate the Angelini License Agreement for an uncured material breach of the other party or in the case of insolvency.  The Company may terminate
the Angelini License Agreement if Angelini challenges any of the licensed patents.  Angelini may terminate the Angelini License Agreement for convenience on specified
notice periods, which are determined based upon whether the product has been commercially launched in the European Territory.

The  Company  identified  the  following  material  promises  under  the  Angelini  License  Agreement:  (1)  licensing  of  intellectual  property  with  respect  to  OV101  (2)
completion of certain ongoing trials (3) transfer of a specified amount of compound and related information (4) potential for funding 35% of the cost for Angelini future
trials limited to $7.0 million and (5) completion of the manufacturing process technology transfer.

The Company determined that the $7.0 million represents a potential payment to a customer and should be deferred. The transfer of compound and related information is
considered a contingent milestone payment that will be recognized upon acceptance by Angelini of the milestone which was achieved and recognized in December 2020.
The Company further determined that the license and the completion of ongoing trials are distinct from each other, as each has value without the other.

The Company determined the transaction price is equal to the up-front fee of $20.0 million. The transaction price was allocated based on the standalone selling price of
the license, the ongoing trials and $7.0 million for potential future trials.

Upon the transfer of the specified amount of compound and related information and acceptance by Angelini, Angelini was required to and made a $5.0 million payment.
This performance obligation was determined to be variable consideration which was constrained and not considered part of the upfront transaction price allocation.

Angelini will be required to make a separate $5.0 million tech transfer payment towards the $55.0 million aggregate tech transfer and regulatory milestone payments upon
the successful completion of the manufacturing process technology transfer. The Company earning this is fully dependent on performance and cooperation of Angelini
and Lundbeck in implementing the Technology Transfer. At this time, the Company cannot estimate if or when this milestone-related performance obligation might be
achieved.

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During the year ended December 31, 2020, the Company recognized $6.1 million of license revenue and $1.5 million relating to the progress of the ongoing trials as well
as  $5.0  million  for  the  transfer  of  the  specified  amount  of  compound  and  related  information.  The  portion  of  the  upfront  payment  allocated  to  License  Revenue  was
recognized in full as it was non-refundable and not contingent on any future performance and requires no consequential continuing involvement by the Company. The
Company did not have any such revenue during the year ended December 31, 2019. In addition, the Company recorded deferred revenue in the amount of approximately
$12.4  million  as  of  December  31,  2020  which  will  be  recognized  over  the  term  of  the  ongoing  trials  based  on  the  portion  of  total  estimated  expenses  incurred.  The
Company has classified deferred revenue as current or noncurrent based on the expected timing of such expenses.

Takeda Collaboration

On January 6, 2017, the Company entered into a license and collaboration agreement with Takeda, pursuant to which Takeda granted the Company an exclusive license to
commercialize the compound TAK-935, which the Company refers to as OV935, in certain territories, and a co-exclusive worldwide license, together with Takeda, to
develop OV935. In consideration of certain license rights granted to the Company pursuant to the Takeda collaboration, the Company issued 1,781,996 shares of its Series
B-1 Preferred Stock, pursuant to a Series B-1 preferred stock purchase agreement entered into on January 6, 2017, at an ascribed price per share of $14.513 on January 6,
2017 for an aggregate fair value of $25.9 million, which was recorded as research and development expense at the date of the transaction. The 1,781,996 shares of Series
B-1 Preferred Stock held by Takeda automatically converted into 1,781,996 shares of the Company’s common stock upon the completion of its IPO in 2017. Under the
Takeda collaboration, the Company is obligated to pay Takeda future payments if and when certain milestones are achieved. Upon the first patient enrollment in the first
Phase 3 trial for the first of the initial indications the Company and Takeda are focusing on in the Takeda collaboration, the Company is obligated to issue to Takeda the
number of unregistered shares of the Company’s common stock equal to the lesser of (a) 8% of the Company outstanding capital stock on the issuance date or (b) $50.0
million divided by the applicable share price, unless certain events occur. In the event such payment would cause Takeda to own over 19.99% of our outstanding capital
stock or other events occur, such payment must be paid in cash.   The  remaining  potential  global  commercial  and  regulatory  milestone  payments  equal  approximately
$35.0 million and can be satisfied in cash or unregistered shares of the Company’s common stock at its election, unless certain events occur. As of December 31, 2020,
none of these contingent payments have been triggered.  During the year ended December 31, 2020, the Company recognized $0.7 million in research and development
expenses representing research and development expenses reimbursable to the Company from Takeda, of which $0.1 million was included in related party receivable as of
December  31,  2020  and  $2.1  million  was  included  in  related  party  payable  as  of  December  31,  2020.    During  the  year  ended  December  31,  2019,  the  Company
recognized  a  credit  in  research  and  development  expenses  of  $4.7  million  representing  costs  reimbursable  to  the  Company  from  Takeda,  of  which  $1.1  million  was
included in related party receivable as of December 31, 2019.   

The  Takeda  collaboration  will  expire  upon  the  cessation  of  commercialization  of  the  products  by  both  the  Company  and  Takeda.  Either  party  may  terminate  the  Takeda
collaboration because of the other party’s uncured material breach or insolvency, for safety reasons, or, after completion of the first proof of mechanism clinical trial, for
convenience.  Takeda  may  terminate  the  Takeda  collaboration  for  the  Company’s  (or  the  Company’s  sublicensee’s)  challenge  to  the  patents  licensed  under  the  Takeda
collaboration. If the collaboration is terminated by Takeda for material breach by the Company, bankruptcy or patent challenge or by the Company for convenience or safety
reasons, the Company’s rights to the products will cease, the Company will transition all activities related to the products to Takeda, and the Company will grant Takeda an
exclusive, royalty-bearing license under certain patents and other intellectual property controlled by the Company to commercialize OV935 and products containing OV935
for  the  treatment  of  certain  rare  neurological  disorders.  If  the  collaboration  is  terminated  by  the  Company  for  Takeda’s  material  breach  or  bankruptcy  or  by  Takeda  for
convenience  or  safety  reasons,  Takeda’s  rights  to  the  products  will  cease,  Takeda  will  transition  all  activities  related  to  the  products  to  us,  and  Takeda  will  grant  us  an
exclusive, royalty-bearing license under certain patents and other intellectual property controlled by Takeda to commercialize OV935 and products containing OV935 for the
treatment of certain rare neurological disorders.

In March 2021, the Company entered into a royalty, license and termination agreement with Takeda (see note 12).

NOTE 11 – RELATED PARTY TRANSACTIONS

As part of the Company’s collaboration agreement with Takeda the Company recognized a long-term liability representing long-term prepaid expenses to be reimbursed
to Takeda.

On March 24, 2019, the Company entered into a separation and consulting agreement with Dr. Matthew During in connection with Dr. During’s resignation as President
and Chief Scientific Officer with the Company effective as of April 1, 2019. Pursuant to the separation and consulting agreement, Dr. During agreed to non-solicit and
non-compete covenants through such time as he remains a consultant to the Company, as well as a general release of claims in connection therewith. Dr. During agreed to
a three-year consulting arrangement, pursuant to which he will be paid, amongst other specific milestone and meeting related fees, $150,000 per year for his role as the
Chairman  of  the  Company’s  Scientific  Advisory  Board  and  $150,000  per  year  for  other  advisory  and  consulting  services.  Further,  Dr.  During  was  granted  options  to
acquire 100,000 shares of common stock at an exercise price of $1.76 per share, the fair market value on April 1, 2019, which options shall vest in full upon completion
of a specific clinical milestone, subject to Dr.

F-21

 
 
 
 
During’s continued service through such vesting date. In the event such option does not vest by December 31, 2020, the stock option will expire. Provided further, in
recognition of Dr. During’s service on the Scientific Advisory Board, Dr. During was granted options to acquire 75,000 shares of common stock at an exercise price equal
to $1.76  per  share,  the  fair  market  value  on  April  1,  2019. Either  Dr.  During  or  the  Company  may  terminate  the  consulting  arrangements  pursuant  to  the  Consulting
Agreement in accordance with its terms, at any time and for any reason, upon thirty (30) days written notice to the other party. Upon such termination, the Company will
have no further obligations to Dr. During, including any obligation to pay further consulting fees.

In February 2019, the Company issued and sold an aggregate of 6,325,000 shares of common stock and 2,500 shares of Series A Preferred Stock to entities affiliated with
Takeda, a collaboration partner and an existing stockholder, entities affiliated with Biotechnology Value Fund, L.P., an existing stockholder, and Dr. Jeremy M. Levin, its
Chief Executive Officer and Chairman, for aggregate gross proceeds of $17.7 million.

In October and November 2019, the Company issued and sold an aggregate of 4,058,000 shares of common stock and 2,000 shares of Series A Preferred Stock to entities
affiliated with Takeda, a collaboration partner and an existing stockholder, entities affiliated with Biotechnology Value Fund, L.P., an existing stockholder, and Dr. Jeremy
M. Levin, its Chief Executive Officer and Chairman, for aggregate gross proceeds of $10.2 million.

In September 2019, the Company entered into an exchange agreement with the Exchanging Stockholders pursuant to which the Company exchanged an aggregate of
1,262,000 shares of the Company’s common stock owned by the Exchanging Stockholders for an aggregate of 1,262 shares of the Company’s Series A Preferred Stock.

In May 2020, entities affiliated with Biotechnology Value Fund, L.P. elected to convert an aggregate of 2,256 shares of Series A Preferred Stock owned by such holders
into an aggregate of 2,256,000 shares of the Company’s common stock.

In August 2020, the Company issued and sold an aggregate of 1,250,000 shares of common stock to entities affiliated with Biotechnology Value Fund, L.P., an existing
stockholder for aggregate gross proceeds of $10.0 million.

In December 2020, entities affiliated with Biotechnology Value Fund, L.P. elected to convert an aggregate of 2,256 shares of Series A Preferred Stock owned by such
holders into an aggregate of 2,256,000 shares of the Company’s common stock.   

NOTE 12 – SUBSEQUENT EVENTS

Equity Awards

From January 1, 2021 through the date of the filing of this Form 10-K, the Company has granted option awards for an aggregate of 643,600 shares of common stock to
employees with a weighted average exercise price of $3.18.

Royalty, License and Termination Agreement with Takeda

In March 2021, the Company entered into a royalty, license and termination agreement (the “Takeda License and Termination Agreement”) with Takeda under which
Takeda will secure rights to the Company’s 50% global share in soticlestat, and an exclusive license under our relevant intellectual property rights and global rights at
closing  from  the  Company  to  develop  and  commercialize  the  investigational  medicine  OV935  for  the  treatment  of  developmental  and  epileptic  encephalopathies,
including Dravet syndrome and Lennox-Gastaut syndrome.

Under the Takeda License and Termination Agreement, all rights in OV935 will be owned by Takeda, or exclusively licensed to Takeda by the Company.  Takeda will
assume sole responsibility for further worldwide development and commercialization, and the Company will no longer have any financial obligation to Takeda under the
original  collaboration  agreement,  including  for  milestone  payments  or  any  future  development  and  commercialization  costs.  Should  the  Company  close  the  Takeda
License and Termination Agreement, the Company will receive an upfront payment of $196.0 million at closing and will be eligible to receive up to an additional $660.0
million upon achieving development, regulatory and sales milestones. In addition, the Company would be entitled receive tiered royalties beginning in the low double-
digits, and up to 20% on sales of OV935, if approved and commercialized.

The  Company  expects  to  close  the  Takeda  License  and  Termination  Agreement  in  the  first  half  of  2021,  subject  to  the  satisfaction  of  closing  conditions,  including
regulatory review by the appropriate regulatory agencies under the Hart-Scott-Rodino Antitrust Improvements Act of 1976, as amended. Either party may terminate the
agreement if it does not close by May 14, 2021.

F-22

 
 
 
 
 
 
 
 
 
 
 
 
EXECUTIVE EMPLOYMENT AGREEMENT

Exhibit 10.17

This EXECUTIVE EMPLOYMENT AGREEMENT (this “Agreement”) is entered into as of the 30th day of September, 2020, between
Jeff Rona (“Executive”) and OVID THERAPEUTICS INC. (the “Company”). Certain capitalized terms used in this Agreement are defined in Section
6.

WHEREAS, the Company is a biopharmaceutical company;

WHEREAS,  the  Company  desires  to  employ  Executive  in  the  position  set  forth  below,  and  wishes  to  provide  Executive  with  certain

compensation and benefits in return for such services, as set forth in this Agreement; and

WHEREAS,  Executive  wishes  to  be  employed  by  the  Company  and  to  provide  personal  services  to  the  Company  in  return  for  certain

compensation and benefits, as set forth in this Agreement.

NOW, THEREFORE, in consideration of the mutual promises contained herein and for other good and valuable consideration, the receipt

and sufficiency of which is hereby acknowledged, the Company and Executive agree as follows:

1.  TERMS OF EMPLOYMENT

1.1.

Position, Duties and Location.  Executive’s anticipated start date is September 30, 2020, (“Start Date”) or such other date
as mutually agreed upon by the parties. Executive shall initially serve as Chief Business Officer reporting to the Company’s CEO.  Executive shall perform
those  duties  and  responsibilities  as  are  customary  for  such  position  and  as  may  be  directed  by  the  Company  and  the  Board  from  time  to  time.  During
Executive’s employment with the Company, Executive shall devote Executive’s best efforts and substantially all of Executive’s business time and attention
to the business of the Company, except for approved vacation periods and reasonable periods of illness or other incapacities permitted by the Company’s
general employment policies.  Executive’s primary office location will be the Niwot, CO, the Executive will spend time at the Company’s New York office
as required and expenses will be reimbursed under the Company’s reimbursement policy.  Notwithstanding the foregoing, the Company reserves the right
to reasonably require Executive to perform Executive’s duties at places other than Executive’s primary office location from time to time, and to require
reasonable  business  travel.    During  Executive’s  employment  with  the  Company,  Executive  shall  not  engage  in  any  activity  that  conflicts  with  or  is
detrimental to the Company’s best interests, as determined by the CEO.  

Executive may participate as Advisor and Board Member to Applied Immunotherapeutic and Brooklyn Defender Service (non-profit) and in wind down
activities  with  Danforth  Advisors  and  their  clients  for  90  days  after  the  date  of  this  agreement  (the “Activities”), provided  that  Executive  obtains  their
manager’s prior written consent, and that none of the following activities involve activities in the area of neurology, detract from Ovid’s reputation, impact
Executive’s  full  time  duties  to  the  Company,  or  could  reasonably  result  in  the  disclosure  or  use  of  the  Company’s  proprietary  or  confidential
information.  The manager may rescind their consent to Executive’s participation in the Activities, or participation in other business or public activities, if
the manager, in their sole discretion, determines that such activities compromise or threaten to compromise the Company’s business interests or conflict
with Executive’s duties to the Company.

1.2.

Employment  Term.    Executive  will  be  employed  by  the  Company  on  an  “at-will”  basis.    This  means  that  either  the

Company or Executive may terminate Executive’s employment at any time, for

Office: (646) 661-7661 | Fax: (646) 661-4027

Suite 15021, New York, NY 10036

 
 
 
 
 
any reason, with or without Cause, and with or without advance notice (provided that (a) Resignation for Good Reason (as defined below) requires certain
advanced notice by Executive of Executive’s termination of employment as set forth below and (b) as a professional courtesy, Executive agrees to provide
the  Company  with  at  least  sixty  (60)  days  advance  written  notice  of  a  voluntary  resignation  by  Executive  that  is  not  a  Resignation  for  Good
Reason).  Subject to the terms herein, it also means that Executive’s job title, duties, responsibilities, reporting level, compensation and benefits, as well as
the  Company’s  personnel  policies  and  procedures,  may  be  changed  with  or  without  notice  at  any  time  in  the  Company’s  sole  discretion.   This  at-will
employment relationship shall not be modified by any conflicting actions or representations of any Company employee or other party before or during the
term of Executive’s employment.   

1.3.

Compensation.

a)

Annual  Base  Salary.      Executive’s  annual  base  salary  shall  be  paid  at  the  rate  of  $425,000  per  year
(“Annual Base Salary”),  payable  in  equal  installments,  less  applicable  payroll  deductions  and  withholdings,  on  the  Company’s  ordinary  payroll  cycle.
Executive’s Annual Base Salary shall be subject to annual review by the Board and may be adjusted from time to time.  As an exempt salaried employee,
Executive will be required to work the Company’s normal business hours, and such additional time as appropriate for Executive’s work assignments and
position, and Executive will not be entitled to overtime compensation.

Benefits.  Executive  will  be  eligible  to  participate  in  all  of  the  Company’s  employee  benefits  and  benefit
plans that the Company generally makes available to its full-time employees and executives in accordance with the terms and conditions of the benefit
plans and applicable policies as in effect from time to time.  

b)

c)

Bonus.  Executive  shall  be  eligible  to  earn  an  annual  performance  bonus  of  up  to  forty  percent  (40%)  of
Executive’s Annual Base Salary (the “Target Performance Bonus”).  The Target Performance Bonus shall be based upon the Company’s assessment of
Executive’s attainment of written Company and individual objectives as set by the Company in its sole discretion.  The Company may increase the Target
Performance Bonus in its sole discretion.  Bonus payments, if any, shall be subject to applicable payroll deductions and withholdings.  Following the close
of each calendar year, the Company shall determine whether Executive has earned a Target Performance Bonus, and the amount of any such bonus, based
on the achievement of such objectives.  Executive must be an employee of the Company in good standing on the Target Performance Bonus payment date
to be eligible to receive a Target Performance Bonus, and no partial or prorated bonuses shall be provided.  The Target Performance Bonus, if earned, shall
be paid on or before March 15th of the calendar year after the applicable bonus year.  Executive’s bonus eligibility is subject to change in the discretion of
the Company.   If Executive’s start date with the Company falls within the fourth quarter, the Executive will not be eligible for a target bonus for that
calendar year.  

d)

Equity Compensation. Subject to the approval of the Board, at the next meeting of the Board following
the Start Date, Executive will be issued an option to purchase one three hundred twenty-five thousand (325,000) shares of the Company’s common stock
(the “Option”). The Option will be evidenced by a stock option agreement and be subject to the terms and conditions of the Company’s 2017 Equity
Incentive Plan (the “Equity Plan”). The exercise price per share of the Option will be equal to the per share fair market value of the Company’s common
stock on the date the Option is granted, as defined under the Equity Plan. The vesting schedule of the Option will be as follows: twenty-five percent
(25%) of the shares of the Company’s common stock subject to the Option will vest on the one year anniversary of the Start Date, and one thirty-sixth
(1/36th) of the remaining shares of the Company’s common stock subject to the Option will vest each month thereafter on the same day of the month as

RONA - 2

 
 
the Executive’s date of hire (and if there is no corresponding day, on the last day of the month), so long as Executive remains an employee, consultant,
director or officer of the Company, and subject to the terms and conditions of the stock option agreement and the Equity Plan. Subject to the approval of
the Board, the stock option agreement shall provide that upon a Change in Control Termination, the vesting and exercisability of the Option shall be
accelerated in full. At the discretion of the Board, Executive will be eligible to receive additional options to purchase shares of the Company’s common
stock.

1.4.

Reimbursement  of  Expenses.    Subject  to  Section  4.8(c),  the  Company  shall  reimburse  Executive  for  Executive’s
necessary  and  reasonable  business  expenses  incurred  in  connection  with  Executive’s  duties  in  accordance  with  the  Company’s  generally  applicable
expense reimbursement policies as in effect from time to time.  

1.5.

Indemnification  Agreement.  Executive  and  Company  shall  enter  into  an  Indemnity  Agreement  (the  “Indemnification

Agreement”), which shall be effective as of the Start Date and is incorporated herein by reference.  

1.6.

Compliance with Confidentiality Agreement and Company Policies.  Executive shall execute and abide by all terms
and provisions of the Confidentiality Agreement to be signed on or prior to the Start Date (or any successor agreement thereto), attached hereto as Exhibit
A.  Executive  shall  also  abide  by  all  terms  and  provisions  of  the  Company’s  Code  of  Business  Conduct  and  Ethics,  attached  hereto  as  Exhibit  D.  In
addition, Executive is required to abide by the Company’s policies and procedures, including but not limited to the Company’s Employee Handbook, as
adopted or modified from time to time within the Company’s discretion; provided, however, that in the event the terms of this Agreement differ from or
are in conflict with the Company’s general employment policies or practices, this Agreement shall control.  

2.  COVERED TERMINATION SEVERANCE BENEFITS

2.1.

Severance Benefits.  Upon a Covered Termination, then subject to Section 4 below and Executive’s continued compliance

with the terms of this Agreement, the Company shall provide Executive with the severance benefits set forth in this Section 2 (the “Severance Benefits”).

2.2.

Salary Payment.  The Company shall pay Executive, as cash severance, (i) Executive’s Monthly Base Salary, multiplied
by (ii) the number of months in the Covered Termination Severance Period, less applicable payroll deductions and withholdings (the “Severance”). The
Severance shall be paid (except as set forth in Section 4) in equal installments on the Company’s ordinary payroll cycle commencing on the first regularly-
scheduled payroll date occurring on or after the Release Deadline Date (as set forth in Section 4.1).

2.3.

Health Continuation Payments.

a)

The Company will pay Executive on the first day of each month a fully taxable cash payment equal to the
applicable  premium  for  Executive,  her  spouse  and  any  dependents  for  the  group  health  plan  maintained  by  the  Company  for  the  month  in  which  the
Covered Termination occurs, subject to applicable tax withholdings but grossed up for all taxes owed by the Executive on such payment, for the duration
of the Covered Termination Benefits Period. Such coverage shall be counted as coverage pursuant to COBRA. The Company shall have no obligation in
respect of any premium payments following the effective date of the Executive’s coverage by a health insurance plan of a subsequent employer. Executive
shall be required to notify the Company immediately if Executive becomes covered by a health insurance plan of a subsequent employer.

of state law, and (ii) any applicable insurance premiums that are paid by the

b)

For purposes of this Section 2.3, (i) references to COBRA shall be deemed to include analogous provisions

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Company shall not include any amounts payable by Executive under a Code Section 125 health care reimbursement plan, which amounts, if any, are the
sole responsibility of Executive.

3.  CHANGE IN CONTROL SEVERANCE BENEFITS

3.1.

Change  in  Control  Severance  Benefits.    Upon  a  Change  in  Control  Termination,  then  subject  to  Section  4  below  and
Executive’s continued compliance with the terms of this Agreement, the Company shall provide Executive with the severance benefits set forth in this
Section 3 (the “Change in Control Severance Benefits”).  

3.2.

Salary Payment.  The Company shall pay Executive, as cash severance, (i) Executive’s Monthly Base Salary, multiplied
by (ii) the number of months in the Change in Control Severance Period, less applicable payroll deductions and withholdings (the “Change  in  Control
Severance”). The Change in Control Severance shall be paid (except as set forth in Section 4) in equal installments on the Company’s ordinary payroll
cycle commencing on the first regularly-scheduled payroll date occurring on or after the Release Deadline Date.  

3.3.

Health Continuation Payments.

a)The Company will pay Executive on the first day of each month a fully taxable cash payment equal to the applicable premium
for  Executive,  her  spouse  and  any  dependents  for  the  group  health  plan  maintained  by  the  Company  for  the  month  in  which  the  Change  in  Control
Termination occurs, subject to applicable tax withholdings but grossed up for all taxes owed by the Executive on such payment, for the duration of the
Change in Control Benefits Period. Such coverage shall be counted as coverage pursuant to COBRA. The Company shall have no obligation in respect of
any premium payments following the effective date of the Executive’s coverage by a health insurance plan of a subsequent employer. Executive shall be
required to notify the Company immediately if Executive becomes covered by a health insurance plan of a subsequent employer.

For purposes of this Section 3.3, (i) references to COBRA shall be deemed to include analogous provisions
of state law, and (ii) any applicable insurance premiums that are paid by the Company shall not include any amounts payable by Executive under a Code
Section 125 health care reimbursement plan, which amounts, if any, are the sole responsibility of Executive.

b)

3.4.

Change in Control Termination Vesting Acceleration Benefits.  Upon a Change in Control Termination, (i) the vesting
and  exercisability  of  all  outstanding  options  to  purchase  the  Company’s  common  stock  (or  stock  appreciation  rights  or  other  rights  with  respect  to  the
stock  of  the  Company  issued  pursuant  to  any  equity  incentive  plan  of  the  Company)  that  are  held  by  Executive  on  the  Termination  Date  shall  be
accelerated in full, (ii) each such option shall be exercisable and to the extent not exercised, expire on the latest date permitted under the Equity Plan and
(iii)  any  reacquisition  or  repurchase  rights  held  by  the  Company  with  respect  to  common  stock  issued  or  issuable  (or  with  respect  to  other  rights  with
respect to the stock of the Company issued or issuable) pursuant to any other stock award granted to Executive pursuant to any equity incentive plan of the
Company shall lapse.

4.  LIMITATIONS AND CONDITIONS ON BENEFITS

4.1.

Release  Prior  to  Payment  of  Severance  Benefits  and  Change  in  Control  Severance  Benefits.    The  receipt  of  any
Severance Benefits or Change in Control Severance Benefits pursuant to this Agreement is subject to Executive signing and not revoking a separation
agreement and general release of claims (the “Release”), in substantially the form attached hereto and incorporated herein as Exhibit B or Exhibit C, as
appropriate, and subject to any further modifications as determined in the Company’s discretion, which Release must become effective and irrevocable no
later than the sixtieth (60th) day following Executive’s Termination Date (the “Release Deadline Date”).  If the Release does not become

RONA - 4

 
 
 
 
effective  and  irrevocable  by  the  Release  Deadline  Date,  Executive  will  forfeit  any  right  to  any  Severance  Benefits  or  Change  in  Control  Severance
Benefits under this Agreement.  In no event will Severance Benefits or Change in Control Severance Benefits be paid or provided until after the Release
Deadline  Date.    On  the  first  regularly-scheduled  payroll  date  occurring  on  or  after  the  Release  Deadline  Date,  the  Company  will  pay  Executive  the
Severance or Change in Control Severance amount that Executive would otherwise have received on or prior to such date but for the delay in payment
related to the effectiveness of the Release, with the balance of the Severance or Change in Control Severance amount being paid as originally scheduled.
The  Company  may  modify  the  Release  in  its  discretion  to  comply  with  changes  in  applicable  law  at  any  time  prior  to  Executive’s  execution  of  such
Release.

4.2.

Return of Company Property.  Not later than the Termination Date, or earlier if requested by the Company, Executive
shall  return  to  the  Company  all  documents  (and  all  copies  thereof)  and  other  property  belonging  to  the  Company  that  Executive  has  in  his  or  her
possession  or  control.  The  documents  and  property  to  be  returned  include,  but  are  not  limited  to,  all  files,  correspondence,  email,  memoranda,  notes,
notebooks,  records,  plans,  forecasts,  reports,  studies,  analyses,  compilations  of  data,  proposals,  agreements,  financial  information,  research  and
development information, marketing information, operational and personnel information, databases, computer-recorded information, tangible property and
equipment (including, but not limited to, computers, facsimile machines, mobile telephones and servers), credit cards, entry cards, identification badges
and  keys,  and  any  materials  of  any  kind  which  contain  or  embody  any  proprietary  or  confidential  information  of  the  Company  (and  all  reproductions
thereof in whole or in part). Executive agrees to make a diligent search to locate any such documents, property and information. If Executive has used any
personally owned computer, server or e-mail system to receive, store, review, prepare or transmit any Company confidential or proprietary data, materials
or  information,  then  within  ten  (10)  business  days  after  the  Termination  Date,  or  earlier  if  requested  by  the  Company,  Executive  shall  provide  the
Company with a computer-useable copy of all such information and then permanently delete and expunge such confidential or proprietary information
from those systems. Executive agrees to provide the Company with a certification that the necessary copying and/or deletion is done.

4.3.

Cooperation and Continued Compliance with Restrictive Covenants.

a)

After the Termination Date, Executive shall cooperate fully with the Company, at reasonable times as agreed
between  Executive  and  the  Company,  in  connection  with  its  actual  or  contemplated  defense,  prosecution  or  investigation  of  any  existing  or  future
litigation, arbitrations, mediations, claims, demands, audits, government or regulatory inquiries, or other matters arising from events, acts or failures to act
that occurred during the time period in which Executive was employed by the Company (including any period of employment with an entity acquired by
the Company). Such cooperation includes, without limitation, being available upon reasonable notice, without subpoena, to provide accurate and complete
advice,  assistance  and  information  to  the  Company,  including  offering  and  explaining  evidence,  providing  truthful  and  accurate  sworn  statements,  and
participating  in  discovery  and  trial  preparation  and  testimony.  Executive  also  agrees  to  promptly  send  the  Company  copies  of  all  correspondence  (for
example, but not limited to, subpoenas) received by Executive in connection with any such legal proceedings, unless Executive is expressly prohibited by
law from so doing.  Nothing in this Agreement prohibits Executive from responding accurately and fully to any request for information if required by legal
process  or  in  connection  with  a  government  investigation.    In  addition,  nothing  in  this  Agreement  is  intended  to  prohibit  or  restrain  Executive  in  any
manner  from  making  disclosures  that  are  protected  under  the  whistleblower  provisions  of  federal  law  or  regulation  or  under  other  applicable  law  or
regulation.  The Company will reimburse Executive for reasonable out-of-pocket expenses incurred in connection with any such cooperation (excluding
foregone wages, salary or other compensation) within

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thirty  (30)  days  of  Executive’s  timely  presentation  of  appropriate  documentation  thereof,  in  accordance  with  the  Company’s  standard  reimbursement
policies  and  procedures.  The  Company  will  reasonably  accommodate  Executive’s  scheduling  needs  with  respect  to  any  such  cooperation  after  the
Termination Date.

b)

After the Termination Date, Executive shall continue to abide by Executive’s continuing obligations under

the Confidentiality Agreement.

c)

From  the  Start  Date  and  through  and  including  the  Change  in  Control  Severance  Period  or  Covered
Termination Severance Period as defined below, or, if Executive is Terminated with Cause, for one year after Executive’s Termination Date, whichever is
applicable,  Executive  shall  not,  without  the  Company’s  prior  written  consent,  whether  directly  or  indirectly  be  employed,  under  contract  with,  provide
services to or on behalf of, or be involved with any business or organization (whether “for profit” or  “not-for-profit”), or applicable Division thereof (as
defined  below),  which  researches,  develops,  creates,  manufactures,  designs  and/or  sells  compounds  and/or  related  pharmaceuticals,  medicines  and/or
therapies  to  treat  rare  or  orphan  neurological  conditions  or  diseases,  and/or  otherwise  competes  with  products  and/or  services  then  under  research  or
development by or offered or sold by the Company in the same therapeutic category.  Nothing in Section 4.3(c) shall prohibit Executive from investing as
a less than one percent (1%) shareholder in securities of any company listed on a national securities exchange or quoted on an automated quotation system.

d)

From the Start Date until twelve (12) months after Termination Date, Executive shall not hire or retain, or
attempt to hire or retain, any of the Company’s then-existing board members, employees, advisors, consultants, collaborators, investigators or agents and
shall not induce any such to give up employment with or to cease providing services to the Company, and shall not otherwise interfere with, or attempt to
interfere with, the relationship of any such person with the Company; or attempt in any manner to solicit, persuade or induce any Client of the Company to
terminate, reduce or refrain from renewing or extending its contractual or other relationship with the Company in regard to the purchase of products or
services  marketed  or  sold  by  the  Company,  or  to  become  a  Client  of  or  enter  into  any  contractual  or  other  relationship  with  Executive  or  any  other
individual, person or entity in regard to the purchase of products or services similar or identical to those marketed or sold by the Company.

e)

Executive acknowledges and agrees that Executive’s obligations under this Section 4.3 are an essential part
of the consideration Executive is providing hereunder in exchange for which and in reliance upon which the Company has agreed to provide the payments
and benefits under this Agreement. Executive further acknowledges and agrees that Executive’s violation of this Section 4.3 inevitably would involve use
or  disclosure  of  the  Company’s  proprietary  and  confidential  information.  If  it  is  determined  by  a  court  of  competent  jurisdiction  in  any  state  that  any
restriction in this Section 4.3 is excessive in duration or scope or is unreasonable or unenforceable under the laws of that state, it is the intention of the
parties that such restriction may be modified or amended by the court to render it enforceable to the maximum extent permitted by the law of that state.

4.4.

Parachute Payments.

a)

Parachute  Payment  Limitation.    If  any  payment  or  benefit  (including  payments  and  benefits  pursuant  to  this
Agreement)  Executive  would  receive  in  connection  with  a  Change  in  Control  from  the  Company  or  otherwise  (“Payment”)  would  (i)  constitute  a
“parachute  payment”  within  the  meaning  of  Section  280G  of  the  Code,  and  (ii)  but  for  this  paragraph,  be  subject  to  the  excise  tax  imposed  by
Section 4999 of the Code (the “Excise Tax”), then the Company shall cause to be determined, before any amounts of the Payment are paid to Executive,
which of the following two alternative forms of payment shall be paid to Executive: (A) payment in full of the entire amount of the Payment (a “Full

RONA - 6

 
 
Payment”), or (B) payment of only a part of the Payment so that Executive receives the largest payment possible without the imposition of the Excise Tax
(a “Reduced Payment”). A Full Payment shall be made in the event that the amount received by the Executive on a net after-tax basis is greater than what
would be received by the Executive on a net after-tax basis if the Reduced Payment were made, otherwise a Reduced Payment shall be made. If a Reduced
Payment is made, (i) the Payment shall be paid only to the extent permitted under the Reduced Payment alternative, and Executive shall have no rights to
any  additional  payments  and/or  benefits  constituting  the  Payment,  and  (ii)  reduction  in  payments  and/or  benefits  shall  occur  in  the  following  order:
(A) reduction of cash payments; (B) cancellation of accelerated vesting of equity awards other than stock options; (C) cancellation of accelerated vesting
of stock options; and (D) reduction of other benefits paid to Executive. In the event that acceleration of compensation from Executive’s equity awards is to
be reduced, such acceleration of vesting shall be canceled in the reverse order of the date of grant.

b)

The independent registered public accounting firm engaged by the Company for general audit purposes as
of the day prior to the effective date of the Change in Control shall make all determinations required to be made under this Section 4.4. If the independent
registered public accounting firm so engaged by the Company is serving as accountant or auditor for the individual, entity or group effecting the Change in
Control, the Company shall appoint a nationally recognized independent registered public accounting firm to make the determinations required hereunder.
The  Company  shall  bear  all  expenses  with  respect  to  the  determinations  by  such  independent  registered  public  accounting  firm  required  to  be  made
hereunder.

c)

The  independent  registered  public  accounting  firm  engaged  to  make  the  determinations  hereunder  shall
provide its calculations, together with detailed supporting documentation, to the Company and Executive within fifteen (15) calendar days after the date on
which Executive’s right to a Payment is triggered (if requested at that time by the Company or Executive) or such other time as requested by the Company
or Executive. If the independent registered public accounting firm determines that no Excise Tax is payable with respect to a Payment, either before or
after  the  application  of  the  Reduced  Amount,  it  shall  furnish  the  Company  and  Executive  with  an  opinion  reasonably  acceptable  to  Executive  that  no
Excise Tax will be imposed with respect to such Payment. Any good faith determinations of the accounting firm made hereunder shall be final, binding
and conclusive upon the Company and Executive.

4.5.

Certain  Reductions  and  Offsets.   To  the  extent  that  any  federal,  state  or  local  laws,  including,  without  limitation,  the
Worker Adjustment and Retraining Notification Act or any other so-called “plant closing” laws, require the Company to give advance notice or make a
payment  of  any  kind  to  Executive  because  of  Executive’s  involuntary  termination  due  to  a  layoff,  reduction  in  force,  plant  or  facility  closing,  sale  of
business, change in control or any other similar event or reason, the benefits payable under this Agreement shall be correspondingly reduced. The benefits
provided  under  this  Agreement  are  intended  to  satisfy  any  and  all  statutory  obligations  that  may  arise  out  of  Executive’s  involuntary  termination  of
employment for the foregoing reasons, and the parties shall construe and enforce the terms of this Agreement accordingly.

4.6.

Mitigation.  Except as otherwise specifically provided herein, Executive shall not be required to mitigate damages or the
amount  of  any  payment  provided  under  this  Agreement  by  seeking  other  employment  or  otherwise,  nor  shall  the  amount  of  any  payment  or  benefit
provided  for  under  this  Agreement  be  reduced  by  any  compensation  earned  by  Executive  as  a  result  of  employment  by  another  employer  or  by  any
retirement  benefits  received  by  Executive  after  the  date  of  a  Covered  Termination  or  Change  in  Control  Termination  (except  as  expressly  provided  in
Sections 2.3 and 3.3 above).

RONA - 7

 
 
4.7.

Indebtedness of Executive. If Executive is indebted to the Company on the effective date of a Covered Termination  or
Change in Control Termination Date, the Company reserves the right to offset any Severance Benefits or Change in Control Severance Benefits under this
Agreement by the amount of such indebtedness, subject to the requirements of Section 409A of the Code and applicable law.

4.8.

Application of Section 409A.

a)

Separation from Service.  Notwithstanding any provision to the contrary in this Agreement, no amount deemed deferred
compensation  subject  to  Section  409A  of  the  Code  shall  be  payable  pursuant  to  Section  2  or  Section  3  unless  Executive’s  termination  of  employment
constitutes a “separation from service” with the Company within the meaning of Section 409A of the Code and the Department of Treasury Regulations
and  other  guidance  promulgated  thereunder  and,  except  as  provided  under  Section  4.8(b)  hereof,  any  such  amount  shall  not  be  paid,  or  in  the  case  of
installments,  commence  payment,  until  the  first  regularly-scheduled  payroll  date  occurring  on  or  after  the  sixtieth  (60th)  day  following  Executive’s
separation  from  service.  Any  installment  payments  that  would  have  been  made  to  Executive  during  the  sixty  (60)  day  period  immediately  following
Executive’s separation from service but for the preceding sentence shall be paid to Executive on the first regularly-scheduled payroll date occurring on or
after the sixtieth (60th) day after Executive’s separation from service and the remaining payments shall be made as provided in this Agreement.

b)

Specified Executive.  Notwithstanding any provision to the contrary in this Agreement, if Executive is deemed at the time
of  his  or  her  separation  from  service  to  be  a  “specified  employee”  for  purposes  of  Section  409A(a)(2)(B)(i)  of  the  Code,  to  the  extent  delayed
commencement of any portion of the benefits to which Executive is entitled under this Agreement is required in order to avoid a prohibited distribution
under Section 409A(a)(2)(B)(i) of the Code, such portion of Executive’s benefits shall not be provided to Executive prior to the earlier of (i) the expiration
of the six (6)-month period measured from the date of Executive’s “separation from service” with the Company (as such term is defined in the Treasury
Regulations  issued  under  Section  409A  of  the  Code)  or  (ii)  the  date  of  Executive’s  death.  Upon  the  first  business  day  following  the  expiration  of  the
applicable Code Section 409A(a)(2)(B)(i) period, all payments deferred pursuant to this Section 4.8(b) shall be paid in a lump sum to Executive, and any
remaining payments due under this Agreement shall be paid as otherwise provided herein.

c)

Expense Reimbursements.    To  the  extent  that  any  reimbursement  payable  pursuant  to  this  Agreement  is  subject  to  the
provisions of Section 409A of the Code, any such reimbursement payable to Executive pursuant to this Agreement shall be paid to Executive no later than
December 31 of the year following the year in which the expense was incurred; the amount of expenses reimbursed in one year shall not affect the amount
eligible  for  reimbursement  in  any  subsequent  year;  and  Executive’s  right  to  reimbursement  under  this  Agreement  will  not  be  subject  to  liquidation  or
exchange for another benefit.

Installments.    For  purposes  of  Section  409A  of  the  Code  (including,  without  limitation,  for  purposes  of  Treasury
Regulation Section 1.409A-2(b)(2)(iii)), Executive’s right to receive any installment payments under this Agreement shall be treated as a right to receive a
series of separate payments and, accordingly, each such installment payment shall at all times be considered a separate and distinct payment.

d)

4.9.

Tax Withholding. All  payments  under  this  Agreement  shall  be  subject  to  applicable  withholding  for  federal,  state  and

local income and employment taxes.

4.10.

No Duplication of Severance Benefits. The Severance Benefits and Change in Control Severance Benefits provided in

Section 2 and Section 3 are mutually exclusive of each other, and in no

RONA - 8

 
 
event shall Executive receive any Severance Benefits or Change in Control Severance Benefits pursuant to both Section 2 and Section 3.  

5.  TERMINATION WITH CAUSE OR BY VOLUNTARY RESIGNATION; OTHER RIGHTS AND BENEFITS

5.1.

Termination  for  Cause;  Resignation  Without  Good  Reason;  Death  or  Disability.    If,  at  any  time,  the  Company
terminates Executive’s employment with the Company for Cause, or upon a voluntary resignation by Executive that is not a Resignation for Good Reason,
or Executive’s employment terminates for any reason not entitling Executive to the Severance Benefits or Change in Control Severance Benefits, or if
Executive’s employment terminates as a result of Executive’s death or disability (other than a Permanent Disability in the case of a Covered Termination),
then  the  Company  shall  have  no  further  obligation  to  Executive  hereunder  except  for  the  payment  or  provision,  as  applicable,  of  (i)  the  portion  of  the
Annual Base Salary accrued through Executive’s last day of employment, (ii) all unreimbursed expenses (if any), subject to Sections 1.4 and 4.8(c), and
(iii) any unused vacation (if applicable) accrued through Executive’s last day of employment.  Under these circumstances, Executive will not be entitled to
any other form of compensation, including any Severance Benefits or Change in Control Severance Benefits, other than Executive’s rights to the vested
portion of Executive’s Option and any other rights to which Executive is entitled under the Company’s benefit programs.    

5.2.

Other  Rights  and  Benefits.  Nothing  in  this  Agreement  shall  prevent  or  limit  Executive’s  continuing  or  future
participation  in  any  benefit,  bonus,  incentive  or  other  plans,  programs,  policies  or  practices  provided  by  the  Company  and  for  which  Executive  may
otherwise qualify, nor shall anything herein limit or otherwise affect such rights as Executive may have under other agreements with the Company except
as  provided  in  Section  4  and  Section  5.1  above.  Except  as  otherwise  expressly  provided  herein,  amounts  that  are  vested  benefits  or  that  Executive  is
otherwise  entitled  to  receive  under  any  plan,  policy,  practice  or  program  of  the  Company  at  or  subsequent  to  the  date  of  a  Change  in  Control  shall  be
payable in accordance with such plan, policy, practice or program.

6.  DEFINITIONS

For purposes of this Agreement, the following definitions shall apply:

6.1.“Board” means the Board of Directors of the Company, or the compensation committee thereof, as determinations or responsibilities may

be delegated by the Board to the compensation committee.

6.2.

“Cause”  shall  mean  a  determination  by  the  Company  based  upon  reasonably  available  information  of  Executive’s:  (i)
unauthorized use or disclosure of the Company’s confidential information or trade secrets; (ii) material breach of any agreement to which the Executive
and the Company are a party; (iii) material failure to comply with the Company’s written policies or rules; (iv) conviction of, or plea of “guilty” or “no
contest”  to,  a  felony  under  the  laws  of  the  United  States  or  any  State;  (v)  negligence  or  willful  misconduct  relating  to  Executive’s  performance  of  her
duties on behalf of the Company; (vi) continuing failure to perform material and lawful assigned duties after receiving thirty (30) days’ written notification
of the failure from the Company if such breach is not cured (if curable) during that thirty (30) day period; (vii) failure to cooperate in good faith with a
governmental  or  internal  investigation  of  the  Company  or  its  directors,  officers  or  employees,  if  the  Company  has  requested  Executive’s  cooperation
without prejudice or personal liability to Executive; (viii) violation of employee or ethical guidelines including, without limitation, violations of business
practices and ethics commonly in place in similar companies in the United States; or (ix) violation of the Company code of conduct and/or any contractual
code of conduct to which the Company is obligated.

RONA - 9

 
 
 
 
6.3.
more of the following events:

“Change  in  Control”  means  the  occurrence,  in  a  single  transaction  or  in  a  series  of  related  transactions,  of  any  one  or

a)

Any natural person, entity or group within the meaning of Section 13(d) or 14(d) of the Securities Exchange Act of 1934, as
amended (“Exchange Act Person”), becomes the owner, directly or indirectly, of securities of the Company representing more than fifty percent (50%) of
the  combined  voting  power  of  the  Company’s  then  outstanding  securities  other  than  by  virtue  of  a  merger,  consolidation  or  similar  transaction.
Notwithstanding the foregoing, a Change in Control shall not be deemed to occur (i) on account of the acquisition of securities of the Company by any
institutional investor, any affiliate thereof or any other Exchange Act Person that acquires the Company’s securities in a transaction or series of related
transactions that are primarily a private financing transaction for the Company or (ii) solely because the level of ownership held by any Exchange Act
Person  (the  “Subject  Person”)  exceeds  the  designated  percentage  threshold  of  the  outstanding  voting  securities  as  a  result  of  a  repurchase  or  other
acquisition of voting securities by the Company reducing the number of shares outstanding, provided that if a Change in Control would occur (but for the
operation of this sentence) as a result of the acquisition of voting securities by the Company, and after such share acquisition, the Subject Person becomes
the  owner  of  any  additional  voting  securities  that,  assuming  the  repurchase  or  other  acquisition  had  not  occurred,  increases  the  percentage  of  the  then
outstanding voting securities owned by the Subject Person over the designated percentage threshold, then a Change in Control shall be deemed to occur;

b)

There  is  consummated  a  merger,  consolidation  or  similar  transaction  involving,  directly  or  indirectly,  the  Company  if,
immediately after the consummation of such merger, consolidation or similar transaction, the stockholders of the Company immediately prior thereto do
not  own,  directly  or  indirectly,  either  (i)  outstanding  voting  securities  representing  more  than  fifty  percent  (50%)  of  the  combined  outstanding  voting
power of the surviving entity in such merger, consolidation or similar transaction or (ii) more than fifty percent (50%) of the combined outstanding voting
power of the parent of the surviving entity in such merger, consolidation or similar transaction; or

c)

There is consummated a sale, lease, license or other disposition of all or substantially all of the consolidated assets of the
Company and its subsidiaries, other than a sale, lease, license or other disposition of all or substantially all of the consolidated assets of the Company and
its subsidiaries to an entity, more than fifty percent (50%) of the combined voting power of the voting securities of which are owned by stockholders of the
Company in substantially the same proportion as their ownership of the Company immediately prior to such sale, lease, license or other disposition.

The term Change in Control shall not include a sale of assets, merger or other transaction effected exclusively for the purpose of changing the
domicile of the Company. Notwithstanding the foregoing or any other provision of this Agreement, the definition of Change in Control (or any analogous
term) in an individual written agreement between the Company or any affiliate and the participant shall supersede the foregoing definition with respect to
stock awards subject to such agreement (it being understood, however, that if no definition of Change in Control or any analogous term is set forth in such
an individual written agreement, the foregoing definition shall apply).

6.4.

6.5.

“Change in Control Benefits Period” means the period of twelve (12) months commencing on the Termination Date.

“Change in Control Severance Period” means the period of twelve (12) months commencing on the Termination Date.

6.6.

  “Change  in  Control  Termination”  means  an  “Involuntary  Termination  Without  Cause”  or  “Resignation  for  Good
Reason,” either of which occurs within three (3) months prior to or upon or within twelve (12) months following the closing of a Change in Control or
Dissolution Event, provided that

RONA - 10

 
 
any such termination is a “separation from service” within the meaning of Treasury Regulation Section 1.409A-1(h).  Death and disability shall not be
deemed Change in Control Terminations.

6.7.

6.8.

6.9.

“COBRA” means the Consolidated Omnibus Budget Reconciliation Act of 1985, as amended.

“Code” means the Internal Revenue Code of 1986, as amended.

“Company”  means  Ovid  Therapeutics  Inc.  or,  following  a  Change  in  Control,  the  surviving  entity  resulting  from  such

transaction, or any subsequent surviving entity resulting from any subsequent Change in Control.

6.10.

“Confidentiality Agreement”  means  Senior  Executive  Confidential  Information  and  Invention  Assignment  Agreement

with the Company, (or any successor agreement thereto).

6.11.

  “Covered  Termination”  means  an  “Involuntary  Termination  Without  Cause”  or  “Resignation  for  Good  Reason,”
provided that any such termination is a “separation from service” within the meaning of Treasury Regulation Section 1.409A-1(h). Death and disability,
other  than  a  Permanent  Disability,  shall  not  be  deemed  Covered  Terminations.    If  an  Involuntary  Termination  Without  Cause  or  Resignation  for  Good
Reason qualifies as a Change in Control Termination, it shall not constitute a Covered Termination.  

Date.

6.12.

6.13.

6.14.

“Covered Termination Benefits Period” means the period of twelve (12) months commencing on the Termination Date.

“Covered  Termination  Severance  Period”  means  the  period  of  twelve  (12)  months  commencing  on  the  Termination

“Dissolution  Event”  means  the  stockholders  of  the  Company  approve  or  the  Board  approves  a  plan  of  complete

dissolution or liquidation of the Company, or a complete dissolution or liquidation of the Company shall otherwise occur.

6.15.

“Involuntary Termination Without Cause” means Executive’s dismissal or discharge by the Company for reasons other
than  Cause  and  other  than  as  a  result  of  death  or  disability;  provided, however,  that  for  purposes  of  a  Covered  Termination,  Involuntary  Termination
Without Cause shall include Executive’s dismissal or discharge by the Company for reasons of Permanent Disability.

6.16.

  “Monthly  Base  Salary”  means  1/12th  of  Executive’s  Annual  Base  Salary  (excluding  incentive  pay,  premium  pay,
commissions,  overtime,  bonuses  and  other  forms  of  variable  compensation)  as  in  effect  on  the  date  of  a  Covered  Termination  or  Change  in  Control
Termination.

6.17.

“Permanent Disability” means total and permanent disability as defined in Code Section 22(e)(3).

6.18.

“Resignation for Good Reason” means Executive’s resignation from all employee positions Executive then holds with
the  Company  within  ninety  (90)  days  following  any  of  the  following  events  taken  without  Executive’s  consent,  provided  Executive  has  given  the
Company written notice of such event within thirty (30) days after the first occurrence of such event and the Company has not cured such event within
thirty (30) days thereafter:

a)

A material decrease in Executive’s Annual Base Salary, other than in connection with a decrease in compensation for all

comparable executives of the Company;

b)

A relocation of Executive’s principal place of work outside of a fifty (50) mile radius of its current location; or

RONA - 11

 
 
c)

The Company’s material breach of this Agreement.

6.19.

“Termination Date” means the effective date of a Change in Control Termination, a Covered Termination, a termination

for Cause or any other circumstance under which the employment relationship between Executive and the Company terminates, as applicable.

6.20.

“Division” shall mean only that part, unit or therapeutic category of a larger entity that is competitive with the Company,

but not an entire company itself, if other divisions, units or therapeutic categories of such larger company are not competitive with the Company.

6.21.

"Client"  shall  mean  (A)  anyone  who  is  a  client  of  the  Company  as  of,  or  at  any  time  during  the  one-year  period
immediately preceding, the termination of Executive’s employment, but only if Executive had a direct relationship with, supervisory responsibility for or
otherwise were involved with such client during Executive’s employment with the Company; and (B) any prospective client to whom the Company made
a  new  business  presentation  (or  similar  offering  of  services)  at  any  time  during  the  one-year  period  immediately  preceding,  or  six-month  period
immediately following, Executive’s employment termination (but only if initial discussions between the Company and such prospective client relating to
the rendering of services occurred prior to the termination date, and only if Executive participated in or supervised such presentation and/or its preparation
or the discussions leading up to it).

6.22.

“Solicit”  shall  mean:  (A)  active  solicitation  of  any  Client  or  Company  employee,  board  member,  advisor,  consultant,
collaborator,  investigator  or  agents;  (B)  the  provision  of  information  regarding  any  Client  or  Company  employee,  board  member,  advisor,  consultant,
collaborator, investigator or agents to any third party where such information could be useful to such third party in attempting to obtain business from such
Client or attempting to hire any such Company employee; (C) participation in any meetings, discussions, or other communications with any third party
regarding any Client or Company employee, board member, advisor, consultant, collaborator, investigator or agents where the purpose or effect of such
meeting,  discussion  or  communication  is  to  obtain  business  from  such  Client  or  employ  such  Company  employee;  and  (D)  any  other  passive  use  of
information  about  any  Client  or  Company  employee,  board  member,  advisor,  consultant,  collaborator,  investigator  or  agents  which  has  the  purpose  or
effect of assisting a third party or causing harm to the business of the Company.

7.  GENERAL PROVISIONS

7.1.

Employment  Status.    This  Agreement  does  not  constitute  a  contract  of  employment  or  impose  upon  Executive  any
obligation  to  remain  as  an  employee,  or  impose  on  the  Company  any  obligation  (i)  to  retain  Executive  as  an  employee,  (ii)  to  change  the  status  of
Executive as an at-will employee or (iii) to change the Company’s policies regarding termination of employment.

7.2.

Notices. Any notices provided hereunder must be in writing, and such notices or any other written communication shall be
deemed effective upon the earlier of personal delivery (including personal delivery by facsimile or email transmission (to a facsimile number or email
address designated in advance by the receiving party)) or the third day after mailing by first class mail, to the Company at its primary office location and to
Executive at Executive’s address as listed in the Company’s payroll records. Any payments made by the Company to Executive under the terms of this
Agreement shall be delivered to Executive either in person or at the address as listed in the Company’s payroll records.

7.3.

Severability. Whenever possible, each provision of this Agreement will be interpreted in such manner as to be effective
and  valid  under  applicable  law,  but  if  any  provision  of  this  Agreement  is  determined  to  be  invalid,  illegal  or  unenforceable  in  any  respect  under  any
applicable law or rule in any jurisdiction, such invalidity, illegality or unenforceability will not affect any other provision or any other

RONA - 12

 
 
 
jurisdiction, and the provision in question shall be modified so as to be rendered enforceable in a manner consistent with the intent of the parties insofar as
possible under applicable law.

7.4.

Waiver. If either party should waive any breach of any provisions of this Agreement, he, she or it shall not thereby be

deemed to have waived any preceding or succeeding breach of the same or any other provision of this Agreement.

7.5.

Complete  Agreement.  This  Agreement,  together  with  Exhibits  A  thru  D,  the  Confidentiality  Agreement  and  the
Indemnification Agreement, forms the complete and exclusive statement of Executive’s employment agreement with the Company, and supersedes and
replaces any other agreements or promises made to Executive by anyone, whether oral or written (including but not limited to the Prior Agreement).

7.6.

Amendment or Termination of Agreement; Continuation of Agreement. Except for those changes expressly reserved
to the Company’s or the Board’s discretion in this Agreement, this Agreement may be changed or terminated only upon the mutual written consent of the
Company and Executive. The written consent of the Company to a change or termination of this Agreement must be signed by an executive officer of the
Company (other than Executive) after such change or termination has been approved by the Board. Unless so terminated, this Agreement shall continue in
effect for as long as Executive continues to be employed by the Company or by any surviving entity following any Change in Control. For the avoidance
of any doubt, if, following a Change in Control, Executive continues to be employed by the surviving entity without a Change in Control Termination and
the  surviving  entity  then  undergoes  a  Change  in  Control,  following  which  Executive  is  terminated  by  the  subsequent  surviving  entity  in  a  Change  in
Control Termination, Executive shall receive the benefits described in Section 3 hereof.  

7.7.

Counterparts. This Agreement may be executed in separate counterparts, any one of which need not contain signatures of
more than one party, but all of which taken together will constitute one and the same Agreement.  Facsimile and electronic image copies of signatures shall
be equivalent to original signatures.  

7.8.

Headings. The headings of the Sections hereof are inserted for convenience only and shall not be deemed to constitute a

part hereof nor to affect the meaning thereof.

7.9.

Successors and Assigns. This Agreement is intended to bind and inure to the benefit of and be enforceable by Executive,
and  the  Company,  and  any  surviving  entity  resulting  from  a  Change  in  Control  and  upon  any  other  person  who  is  a  successor  by  merger,  acquisition,
consolidation  or  otherwise  to  the  business  formerly  carried  on  by  the  Company,  and  their  respective  successors,  assigns,  heirs,  executors  and
administrators, without regard to whether or not such person actively assumes any rights or duties hereunder; provided, however, that Executive may not
assign any duties hereunder and may not assign any rights hereunder without the written consent of the Company, which consent shall not be withheld
unreasonably.

7.10.

Choice of Law. This Agreement shall be construed and enforced in accordance with the laws of the State of New York

without regard to conflicts of law principles. 

7.11.

Arbitration.    To  ensure  the  rapid  and  economical  resolution  of  any  disputes  that  may  arise  under  or  relate  to  this
Agreement or Executive’s employment relationship, Executive and the Company agree that, unless otherwise prohibited by applicable law, any and all
disputes,  claims,  or  causes  of  action,  in  law  or  equity,  arising  from  or  relating  to  the  performance,  enforcement,  execution,  or  interpretation  of  this
Agreement, Executive’s employment with the Company, or the termination of Executive’s employment (collectively, “Claims”), shall be resolved by final,
binding, and (to the extent permitted by

RONA - 13

 
 
law) confidential arbitration before a single arbitrator in New York, New York.  Executive and the Company agree that they shall resolve all such Claims
in accordance with the provisions of Section 12 of the Confidential Information and Invention Assignment Agreement attached hereto as Exhibit A.    

7.12.

Construction of Agreement. In the event of a conflict between the text of this Agreement and any summary, description

or other information regarding this Agreement, the text of this Agreement shall control.

7.13.

Circular  230  Disclaimer.  THE  FOLLOWING  DISCLAIMER  IS  PROVIDED  IN  ACCORDANCE  WITH  THE
INTERNAL  REVENUE  SERVICE’S  CIRCULAR  230  (21  C.F.R.  PART  10).  ANY  TAX  ADVICE  CONTAINED  IN  THIS  AGREEMENT  IS
INTENDED TO BE PRELIMINARY, FOR DISCUSSION PURPOSES ONLY AND NOT FINAL. ANY SUCH ADVICE IS NOT INTENDED
TO BE USED FOR MARKETING, PROMOTING OR RECOMMENDING ANY TRANSACTION OR FOR THE USE OF ANY PERSON IN
CONNECTION WITH THE PREPARATION OF ANY TAX RETURN. ACCORDINGLY, THIS ADVICE IS NOT INTENDED OR WRITTEN
TO  BE  USED,  AND  IT  CANNOT  BE  USED,  BY  ANY  PERSON  FOR  THE  PURPOSE  OF  AVOIDING  TAX  PENALTIES  THAT  MAY  BE
IMPOSED ON SUCH PERSON.

REVIEWED, UNDERSTOOD AND ACCEPTED:

OVID THERAPEUTICS INC.

EXECUTIVE

By:
Name:
Title:

Suzanne K. Wakamoto
SVP, Human Resources

By: 
Name: 

Jeffrey Rona

RONA - 14

 
 
 
 
 
 
 
 
 
 
 
 
148402431 v2

Rona - D-1

 
 
 
 
EXECUTIVE EMPLOYMENT AGREEMENT

Exhibit 10.18

This EXECUTIVE EMPLOYMENT AGREEMENT (this “Agreement”) is entered into as of the 21st day of October, 2019, between Jason

Tardio (“Executive”) and OVID THERAPEUTICS INC. (the “Company”). Certain capitalized terms used in this Agreement are defined in Section 6.

WHEREAS, the Company is a biopharmaceutical company;

WHEREAS,  the  Company  desires  to  employ  Executive  in  the  position  set  forth  below,  and  wishes  to  provide  Executive  with  certain

compensation and benefits in return for such services, as set forth in this Agreement; and

WHEREAS,  Executive  wishes  to  be  employed  by  the  Company  and  to  provide  personal  services  to  the  Company  in  return  for  certain

compensation and benefits, as set forth in this Agreement.

NOW, THEREFORE, in consideration of the mutual promises contained herein and for other good and valuable consideration, the receipt

and sufficiency of which is hereby acknowledged, the Company and Executive agree as follows:

1.  TERMS OF EMPLOYMENT

1.1.

Position, Duties and Location.  Executive’s anticipated start date is November 18, 2019, (“Start Date”) or such other date
as mutually agreed upon by the parties. Executive shall initially serve as Chief Commercial Officer reporting to the Company’s Chief Medical Officer and
Head of Research & Development, Amit Rakhit, MD, MBA (“Manager”).  Executive shall perform those duties and responsibilities as are customary for
such position and as may be directed by the Company and the Board from time to time. During Executive’s employment with the Company, Executive
shall devote Executive’s best efforts and substantially all of Executive’s business time and attention to the business of the Company, except for approved
vacation periods and reasonable periods of illness or other incapacities permitted by the Company’s general employment policies.  Executive’s primary
office  location  will  be  the  Company’s  offices  in  New  York,  New  York.    Notwithstanding  the  foregoing,  the  Company  reserves  the  right  to  reasonably
require  Executive  to  perform  Executive’s  duties  at  places  other  than  Executive’s  primary  office  location  from  time  to  time,  and  to  require  reasonable
business travel.  During Executive’s employment with the Company, Executive shall not engage in any activity that conflicts with or is detrimental to the
Company’s best interests, as determined by the CEO.  

Executive may participate in side activities such as board or committee member, advisor or consultant (the “Activities”), provided that Executive obtains
Manager’s prior written consent, which consent shall not be unreasonably withheld, and that none of the following activities involve activities in the area
of neurology, detract from Ovid’s reputation, impact Executive’s full time duties to the Company, or could reasonably result in the disclosure or use of the
Company’s proprietary or confidential information.  The Manager may rescind the consent to Executive’s participation in the Activities, or participation in
other  business  or  public  activities,  if  the  Manager  in  his  sole  discretion,  determines  that  such  activities  compromise  or  threaten  to  compromise  the
Company’s business interests or conflict with Executive’s duties to the Company.

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Exhibit 10.18

1.2.

Employment  Term.    Executive  will  be  employed  by  the  Company  on  an  “at-will”  basis.    This  means  that  either  the
Company or Executive may terminate Executive’s employment at any time, for any reason, with or without Cause, and with or without advance notice
(provided  that  (a)  Resignation  for  Good  Reason  (as  defined  below)  requires  certain  advanced  notice  by  Executive  of  Executive’s  termination  of
employment as set forth below and (b) as a professional courtesy, Executive agrees to provide the Company with at least sixty (60) days advance written
notice of a voluntary resignation by Executive that is not a Resignation for Good Reason).  Subject to the terms herein, it also means that Executive’s job
title, duties, responsibilities, reporting level, compensation and benefits, as well as the Company’s personnel policies and procedures, may be changed with
or without notice at any time in the Company’s sole discretion.  This at-will employment relationship shall not be modified by any conflicting actions or
representations of any Company employee or other party before or during the term of Executive’s employment.   

1.3.

Compensation.

a)

Annual  Base  Salary.      Executive’s  annual  base  salary  shall  be  paid  at  the  rate  of  $400,000  per  year
(“Annual Base Salary”),  payable  in  equal  installments,  less  applicable  payroll  deductions  and  withholdings,  on  the  Company’s  ordinary  payroll  cycle.
Executive’s Annual Base Salary shall be subject to annual review by the Board and may be adjusted from time to time.  As an exempt salaried employee,
Executive will be required to work the Company’s normal business hours, and such additional time as appropriate for Executive’s work assignments and
position, and Executive will not be entitled to overtime compensation.

b)

Benefits.  Executive  will  be  eligible  to  participate  in  all  of  the  Company’s  employee  benefits  and  benefit
plans that the Company generally makes available to its full-time employees and executives in accordance with the terms and conditions of the benefit
plans and applicable policies as in effect from time to time.  In accordance with the Company’s policies and procedures, as in effect from time to time,
Executive will be eligible to accrue twenty (20) days of paid time off per year.

c)

Bonus. Executive shall be eligible to earn an annual performance bonus of up to thirty five percent (35%) of
Executive’s Annual Base Salary (the “Target Performance Bonus”).  The Target Performance Bonus shall be based upon the Company’s assessment of
Executive’s attainment of written Company and individual objectives as set by the Company in its sole discretion.  The Company may increase the Target
Performance Bonus in its sole discretion.  Bonus payments, if any, shall be subject to applicable payroll deductions and withholdings.  Following the close
of each calendar year, the Company shall determine whether Executive has earned a Target Performance Bonus, and the amount of any such bonus, based
on the achievement of such objectives.  Executive must be an employee of the Company in good standing on the Target Performance Bonus payment date
to be eligible to receive a Target Performance Bonus, and no partial or prorated bonuses shall be provided.  The Target Performance Bonus, if earned, shall
be paid on or before March 15th of the calendar year after the applicable bonus year.  Executive’s bonus eligibility is subject to change in the discretion of
the Company.     If Executive’s  start date with the Company falls within the fourth quarter, the Executive will not  be eligible for a target bonus for that
calendar year.  

d)

Equity Compensation. Subject to the approval of the Board, at the next meeting of the Board following
the Start Date, Executive will be issued an option to purchase one hundred twenty five thousand (125,000) shares of the Company’s common stock (the
“Option”).  The  Option  will  be  evidenced  by  a  stock  option  agreement  and  be  subject  to  the  terms  and  conditions  of  the  Company’s  2017  Equity
Incentive Plan (the “Equity Plan”). The exercise price per share of the Option will be equal

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148402431 v2

 
 
 
Exhibit 10.18

to  the  per  share  fair  market  value  of  the  Company’s  common  stock  on  the  date  the  Option  is  granted,  as  defined  under  the  Equity  Plan.  The  vesting
schedule of the Option will be as follows: twenty-five percent (25%) of the shares of the Company’s common stock subject to the Option will vest on the
one year anniversary of the Start Date, and one thirty-sixth (1/36th) of the remaining shares of the Company’s common stock subject to the Option will
vest each month thereafter on the same day of the month as the Executive’s date of hire (and if there is no corresponding day, on the last day of the
month), so long as Executive remains an employee, consultant, director or officer of the Company, and subject to the terms and conditions of the stock
option agreement and the Equity Plan. Subject to the approval of the Board, the stock option agreement shall provide that upon a Change in Control
Termination, the vesting and exercisability of the Option shall be accelerated in full. At the discretion of the Board, Executive will be eligible to receive
additional options to purchase shares of the Company’s common stock.

e)

Sign-on Bonus.  Within  thirty  (30)  days  of  the  commencement  of  Executive’s  employment,  the  Company
will pay Executive a sign-on bonus in the amount of $110,000.  Should Executive resign from the Company or be terminated by the Company with Cause
within one (1) year of the commencement of Executive’s employment, Executive agrees to reimburse the Company pro rata for the amount of the sign-on
bonus.  This reimbursement will be due to the Company within thirty (30) days of Executive’s last day of employment.

1.4.

Reimbursement  of  Expenses.    Subject  to  Section  4.8(c),  the  Company  shall  reimburse  Executive  for  Executive’s
necessary  and  reasonable  business  expenses  incurred  in  connection  with  Executive’s  duties  in  accordance  with  the  Company’s  generally  applicable
expense reimbursement policies as in effect from time to time.  

1.5.

Indemnification  Agreement.  Executive  and  Company  shall  enter  into  an  Indemnity  Agreement  (the  “Indemnification

Agreement”), which shall be effective as of the Start Date and is incorporated herein by reference.  

1.6.

Compliance with Confidentiality Agreement and Company Policies.  Executive shall execute and abide by all terms
and provisions of the Confidentiality Agreement to be signed on or prior to the Start Date (or any successor agreement thereto), attached hereto as Exhibit
A.  Executive  shall  also  abide  by  all  terms  and  provisions  of  the  Company’s  Code  of  Business  Conduct  and  Ethics,  attached  hereto  as  Exhibit  D.  In
addition, Executive is required to abide by the Company’s policies and procedures, including but not limited to the Company’s Employee Handbook, as
adopted or modified from time to time within the Company’s discretion; provided, however, that in the event the terms of this Agreement differ from or
are in conflict with the Company’s general employment policies or practices, this Agreement shall control.  

2.  COVERED TERMINATION SEVERANCE BENEFITS

2.1.

Severance Benefits.  Upon a Covered Termination, then subject to Section 4 below and Executive’s continued compliance

with the terms of this Agreement, the Company shall provide Executive with the severance benefits set forth in this Section 2 (the “Severance Benefits”).

2.2.

Salary Payment.  The Company shall pay Executive, as cash severance, (i) Executive’s Monthly Base Salary, multiplied
by (ii) the number of months in the Covered Termination Severance Period, less applicable payroll deductions and withholdings (the “Severance”). The
Severance shall be paid (except as set forth in Section 4) in equal installments on the Company’s ordinary payroll cycle commencing on the first regularly-
scheduled payroll date occurring on or after the Release Deadline Date (as set forth in Section 4.1).

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148402431 v2

 
 
 
 
Exhibit 10.18

2.3.

Health Continuation Payments.

a)

The Company will pay Executive on the first day of each month a fully taxable cash payment equal to the
applicable  premium  for  Executive,  her  spouse  and  any  dependents  for  the  group  health  plan  maintained  by  the  Company  for  the  month  in  which  the
Covered Termination occurs, subject to applicable tax withholdings but grossed up for all taxes owed by the Executive on such payment, for the duration
of the Covered Termination Benefits Period. Such coverage shall be counted as coverage pursuant to COBRA. The Company shall have no obligation in
respect of any premium payments following the effective date of the Executive’s coverage by a health insurance plan of a subsequent employer. Executive
shall be required to notify the Company immediately if Executive becomes covered by a health insurance plan of a subsequent employer.

For purposes of this Section 2.3, (i) references to COBRA shall be deemed to include analogous provisions
of state law, and (ii) any applicable insurance premiums that are paid by the Company shall not include any amounts payable by Executive under a Code
Section 125 health care reimbursement plan, which amounts, if any, are the sole responsibility of Executive.

b)

3.  CHANGE IN CONTROL SEVERANCE BENEFITS

3.1.

Change  in  Control  Severance  Benefits.    Upon  a  Change  in  Control  Termination,  then  subject  to  Section  4  below  and
Executive’s continued compliance with the terms of this Agreement, the Company shall provide Executive with the severance benefits set forth in this
Section 3 (the “Change in Control Severance Benefits”).  

3.2.

Salary Payment.  The Company shall pay Executive, as cash severance, (i) Executive’s Monthly Base Salary, multiplied
by (ii) the number of months in the Change in Control Severance Period, less applicable payroll deductions and withholdings (the “Change  in  Control
Severance”). The Change in Control Severance shall be paid (except as set forth in Section 4) in equal installments on the Company’s ordinary payroll
cycle commencing on the first regularly-scheduled payroll date occurring on or after the Release Deadline Date.  

3.3.

Health Continuation Payments.

a)The Company will pay Executive on the first day of each month a fully taxable cash payment equal to the applicable premium
for  Executive,  her  spouse  and  any  dependents  for  the  group  health  plan  maintained  by  the  Company  for  the  month  in  which  the  Change  in  Control
Termination occurs, subject to applicable tax withholdings but grossed up for all taxes owed by the Executive on such payment, for the duration of the
Change in Control Benefits Period. Such coverage shall be counted as coverage pursuant to COBRA. The Company shall have no obligation in respect of
any premium payments following the effective date of the Executive’s coverage by a health insurance plan of a subsequent employer. Executive shall be
required to notify the Company immediately if Executive becomes covered by a health insurance plan of a subsequent employer.

For purposes of this Section 3.3, (i) references to COBRA shall be deemed to include analogous provisions
of state law, and (ii) any applicable insurance premiums that are paid by the Company shall not include any amounts payable by Executive under a Code
Section 125 health care reimbursement plan, which amounts, if any, are the sole responsibility of Executive.

b)

3.4.

Change in Control Termination Vesting Acceleration Benefits.  Upon a Change in Control Termination, (i) the vesting
and  exercisability  of  all  outstanding  options  to  purchase  the  Company’s  common  stock  (or  stock  appreciation  rights  or  other  rights  with  respect  to  the
stock of the Company issued

Tardio - D-4

148402431 v2

 
 
 
 
Exhibit 10.18

pursuant to any equity incentive plan of the Company) that are held by Executive on the Termination Date shall be accelerated in full, (ii) each such option
shall be exercisable and to the extent not exercised, expire on the latest date permitted under the Equity Plan and (iii) any reacquisition or repurchase rights
held by the Company with respect to common stock issued or issuable (or with respect to other rights with respect to the stock of the Company issued or
issuable) pursuant to any other stock award granted to Executive pursuant to any equity incentive plan of the Company shall lapse.

4.  LIMITATIONS AND CONDITIONS ON BENEFITS

4.1.

Release  Prior  to  Payment  of  Severance  Benefits  and  Change  in  Control  Severance  Benefits.    The  receipt  of  any
Severance Benefits or Change in Control Severance Benefits pursuant to this Agreement is subject to Executive signing and not revoking a separation
agreement and general release of claims (the “Release”), in substantially the form attached hereto and incorporated herein as Exhibit B or Exhibit C, as
appropriate, and subject to any further modifications as determined in the Company’s discretion, which Release must become effective and irrevocable no
later than the sixtieth (60th) day following Executive’s Termination Date (the “Release Deadline Date”).  If the Release does not become effective and
irrevocable by the Release Deadline Date, Executive will forfeit any right to any Severance Benefits or Change in Control Severance Benefits under this
Agreement.  In no event will Severance Benefits or Change in Control Severance Benefits be paid or provided until after the Release Deadline Date.  On
the first regularly-scheduled payroll date occurring on or after the Release Deadline Date, the Company will pay Executive the Severance or Change in
Control Severance amount that Executive would otherwise have received on or prior to such date but for the delay in payment related to the effectiveness
of the Release, with the balance of the Severance or Change in Control Severance amount being paid as originally scheduled. The Company may modify
the Release in its discretion to comply with changes in applicable law at any time prior to Executive’s execution of such Release.

4.2.

Return of Company Property.  Not later than the Termination Date, or earlier if requested by the Company, Executive
shall  return  to  the  Company  all  documents  (and  all  copies  thereof)  and  other  property  belonging  to  the  Company  that  Executive  has  in  his  or  her
possession  or  control.  The  documents  and  property  to  be  returned  include,  but  are  not  limited  to,  all  files,  correspondence,  email,  memoranda,  notes,
notebooks,  records,  plans,  forecasts,  reports,  studies,  analyses,  compilations  of  data,  proposals,  agreements,  financial  information,  research  and
development information, marketing information, operational and personnel information, databases, computer-recorded information, tangible property and
equipment (including, but not limited to, computers, facsimile machines, mobile telephones and servers), credit cards, entry cards, identification badges
and  keys,  and  any  materials  of  any  kind  which  contain  or  embody  any  proprietary  or  confidential  information  of  the  Company  (and  all  reproductions
thereof in whole or in part). Executive agrees to make a diligent search to locate any such documents, property and information. If Executive has used any
personally owned computer, server or e-mail system to receive, store, review, prepare or transmit any Company confidential or proprietary data, materials
or  information,  then  within  ten  (10)  business  days  after  the  Termination  Date,  or  earlier  if  requested  by  the  Company,  Executive  shall  provide  the
Company with a computer-useable copy of all such information and then permanently delete and expunge such confidential or proprietary information
from those systems. Executive agrees to provide the Company with a certification that the necessary copying and/or deletion is done.

4.3.

Cooperation and Continued Compliance with Restrictive Covenants.

a)

After the Termination Date, Executive shall cooperate fully with the Company, at reasonable times as agreed

between Executive and the Company, in connection with its actual or

148402431 v2

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Exhibit 10.18

contemplated defense, prosecution or investigation of any existing or future litigation, arbitrations, mediations, claims, demands, audits, government or
regulatory inquiries, or other matters arising from events, acts or failures to act that occurred during the time period in which Executive was employed by
the  Company  (including  any  period  of  employment  with  an  entity  acquired  by  the  Company).  Such  cooperation  includes,  without  limitation,  being
available  upon  reasonable  notice,  without  subpoena,  to  provide  accurate  and  complete  advice,  assistance  and  information  to  the  Company,  including
offering  and  explaining  evidence,  providing  truthful  and  accurate  sworn  statements,  and  participating  in  discovery  and  trial  preparation  and  testimony.
Executive also agrees to promptly send the Company copies of all correspondence (for example, but not limited to, subpoenas) received by Executive in
connection  with  any  such  legal  proceedings,  unless  Executive  is  expressly  prohibited  by  law  from  so  doing.    Nothing  in  this  Agreement  prohibits
Executive  from  responding  accurately  and  fully  to  any  request  for  information  if  required  by  legal  process  or  in  connection  with  a  government
investigation.    In  addition,  nothing  in  this  Agreement  is  intended  to  prohibit  or  restrain  Executive  in  any  manner  from  making  disclosures  that  are
protected  under  the  whistleblower  provisions  of  federal  law  or  regulation  or  under  other  applicable  law  or  regulation.    The  Company  will  reimburse
Executive  for  reasonable  out-of-pocket  expenses  incurred  in  connection  with  any  such  cooperation  (excluding  foregone  wages,  salary  or  other
compensation)  within  thirty  (30)  days  of  Executive’s  timely  presentation  of  appropriate  documentation  thereof,  in  accordance  with  the  Company’s
standard  reimbursement  policies  and  procedures.  The  Company  will  reasonably  accommodate  Executive’s  scheduling  needs  with  respect  to  any  such
cooperation after the Termination Date.

the Confidentiality Agreement.

b)

After the Termination Date, Executive shall continue to abide by Executive’s continuing obligations under

c)

From  the  Start  Date  and  through  and  including  the  Change  in  Control  Severance  Period  or  Covered
Termination Severance Period as defined below, or, if Executive is Terminated with Cause, for one year after Executive’s Termination Date, whichever is
applicable,  Executive  shall  not,  without  the  Company’s  prior  written  consent,  whether  directly  or  indirectly  be  employed,  under  contract  with,  provide
services to or on behalf of, or be involved with any business or organization (whether “for profit” or  “not-for-profit”), or applicable Division thereof (as
defined  below),  which  researches,  develops,  creates,  manufactures,  designs  and/or  sells  compounds  and/or  related  pharmaceuticals,  medicines  and/or
therapies  to  treat  rare  or  orphan  neurological  conditions  or  diseases,  and/or  otherwise  competes  with  products  and/or  services  then  under  research  or
development by or offered or sold by the Company in the same therapeutic category.  Nothing in Section 4.3(c) shall prohibit Executive from investing as
a less than one percent (1%) shareholder in securities of any company listed on a national securities exchange or quoted on an automated quotation system.

d)

From the Start Date until twelve (12) months after Termination Date, Executive shall not hire or retain, or
attempt to hire or retain, any of the Company’s then-existing board members, employees, advisors, consultants, collaborators, investigators or agents and
shall not induce any such to give up employment with or to cease providing services to the Company, and shall not otherwise interfere with, or attempt to
interfere with, the relationship of any such person with the Company; or attempt in any manner to solicit, persuade or induce any Client of the Company to
terminate, reduce or refrain from renewing or extending its contractual or other relationship with the Company in regard to the purchase of products or
services  marketed  or  sold  by  the  Company,  or  to  become  a  Client  of  or  enter  into  any  contractual  or  other  relationship  with  Executive  or  any  other
individual, person or entity in regard to the purchase of products or services similar or identical to those marketed or sold by the Company.

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Exhibit 10.18

e)

Executive acknowledges and agrees that Executive’s obligations under this Section 4.3 are an essential part
of the consideration Executive is providing hereunder in exchange for which and in reliance upon which the Company has agreed to provide the payments
and benefits under this Agreement. Executive further acknowledges and agrees that Executive’s violation of this Section 4.3 inevitably would involve use
or  disclosure  of  the  Company’s  proprietary  and  confidential  information.  If  it  is  determined  by  a  court  of  competent  jurisdiction  in  any  state  that  any
restriction in this Section 4.3 is excessive in duration or scope or is unreasonable or unenforceable under the laws of that state, it is the intention of the
parties that such restriction may be modified or amended by the court to render it enforceable to the maximum extent permitted by the law of that state.

4.4.

Parachute Payments.

a)

Parachute  Payment  Limitation.    If  any  payment  or  benefit  (including  payments  and  benefits  pursuant  to  this
Agreement)  Executive  would  receive  in  connection  with  a  Change  in  Control  from  the  Company  or  otherwise  (“Payment”)  would  (i)  constitute  a
“parachute  payment”  within  the  meaning  of  Section  280G  of  the  Code,  and  (ii)  but  for  this  paragraph,  be  subject  to  the  excise  tax  imposed  by
Section 4999 of the Code (the “Excise Tax”), then the Company shall cause to be determined, before any amounts of the Payment are paid to Executive,
which of the following two alternative forms of payment shall be paid to Executive: (A) payment in full of the entire amount of the Payment (a “Full
Payment”), or (B) payment of only a part of the Payment so that Executive receives the largest payment possible without the imposition of the Excise Tax
(a “Reduced Payment”). A Full Payment shall be made in the event that the amount received by the Executive on a net after-tax basis is greater than what
would be received by the Executive on a net after-tax basis if the Reduced Payment were made, otherwise a Reduced Payment shall be made. If a Reduced
Payment is made, (i) the Payment shall be paid only to the extent permitted under the Reduced Payment alternative, and Executive shall have no rights to
any  additional  payments  and/or  benefits  constituting  the  Payment,  and  (ii)  reduction  in  payments  and/or  benefits  shall  occur  in  the  following  order:
(A) reduction of cash payments; (B) cancellation of accelerated vesting of equity awards other than stock options; (C) cancellation of accelerated vesting
of stock options; and (D) reduction of other benefits paid to Executive. In the event that acceleration of compensation from Executive’s equity awards is to
be reduced, such acceleration of vesting shall be canceled in the reverse order of the date of grant.

b)

The independent registered public accounting firm engaged by the Company for general audit purposes as
of the day prior to the effective date of the Change in Control shall make all determinations required to be made under this Section 4.4. If the independent
registered public accounting firm so engaged by the Company is serving as accountant or auditor for the individual, entity or group effecting the Change in
Control, the Company shall appoint a nationally recognized independent registered public accounting firm to make the determinations required hereunder.
The  Company  shall  bear  all  expenses  with  respect  to  the  determinations  by  such  independent  registered  public  accounting  firm  required  to  be  made
hereunder.

c)

The  independent  registered  public  accounting  firm  engaged  to  make  the  determinations  hereunder  shall
provide its calculations, together with detailed supporting documentation, to the Company and Executive within fifteen (15) calendar days after the date on
which Executive’s right to a Payment is triggered (if requested at that time by the Company or Executive) or such other time as requested by the Company
or Executive. If the independent registered public accounting firm determines that no Excise Tax is payable with respect to a Payment, either before or
after  the  application  of  the  Reduced  Amount,  it  shall  furnish  the  Company  and  Executive  with  an  opinion  reasonably  acceptable  to  Executive  that  no
Excise Tax will be imposed with respect to such Payment. Any

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Exhibit 10.18

good faith determinations of the accounting firm made hereunder shall be final, binding and conclusive upon the Company and Executive.

4.5.

Certain  Reductions  and  Offsets.   To  the  extent  that  any  federal,  state  or  local  laws,  including,  without  limitation,  the
Worker Adjustment and Retraining Notification Act or any other so-called “plant closing” laws, require the Company to give advance notice or make a
payment  of  any  kind  to  Executive  because  of  Executive’s  involuntary  termination  due  to  a  layoff,  reduction  in  force,  plant  or  facility  closing,  sale  of
business, change in control or any other similar event or reason, the benefits payable under this Agreement shall be correspondingly reduced. The benefits
provided  under  this  Agreement  are  intended  to  satisfy  any  and  all  statutory  obligations  that  may  arise  out  of  Executive’s  involuntary  termination  of
employment for the foregoing reasons, and the parties shall construe and enforce the terms of this Agreement accordingly.

4.6.

Mitigation.  Except as otherwise specifically provided herein, Executive shall not be required to mitigate damages or the
amount  of  any  payment  provided  under  this  Agreement  by  seeking  other  employment  or  otherwise,  nor  shall  the  amount  of  any  payment  or  benefit
provided  for  under  this  Agreement  be  reduced  by  any  compensation  earned  by  Executive  as  a  result  of  employment  by  another  employer  or  by  any
retirement  benefits  received  by  Executive  after  the  date  of  a  Covered  Termination  or  Change  in  Control  Termination  (except  as  expressly  provided  in
Sections 2.3 and 3.3 above).

4.7.

Indebtedness of Executive. If Executive is indebted to the Company on the effective date of a Covered Termination or
Change in Control Termination Date, the Company reserves the right to offset any Severance Benefits or Change in Control Severance Benefits under this
Agreement by the amount of such indebtedness, subject to the requirements of Section 409A of the Code and applicable law.

4.8.

Application of Section 409A.

a)

Separation from Service.  Notwithstanding any provision to the contrary in this Agreement, no amount deemed deferred
compensation  subject  to  Section  409A  of  the  Code  shall  be  payable  pursuant  to  Section  2  or  Section  3  unless  Executive’s  termination  of  employment
constitutes a “separation from service” with the Company within the meaning of Section 409A of the Code and the Department of Treasury Regulations
and  other  guidance  promulgated  thereunder  and,  except  as  provided  under  Section  4.8(b)  hereof,  any  such  amount  shall  not  be  paid,  or  in  the  case  of
installments,  commence  payment,  until  the  first  regularly-scheduled  payroll  date  occurring  on  or  after  the  sixtieth  (60th)  day  following  Executive’s
separation  from  service.  Any  installment  payments  that  would  have  been  made  to  Executive  during  the  sixty  (60)  day  period  immediately  following
Executive’s separation from service but for the preceding sentence shall be paid to Executive on the first regularly-scheduled payroll date occurring on or
after the sixtieth (60th) day after Executive’s separation from service and the remaining payments shall be made as provided in this Agreement.

b)

Specified Executive.  Notwithstanding any provision to the contrary in this Agreement, if Executive is deemed at the time
of  his  or  her  separation  from  service  to  be  a  “specified  employee”  for  purposes  of  Section  409A(a)(2)(B)(i)  of  the  Code,  to  the  extent  delayed
commencement of any portion of the benefits to which Executive is entitled under this Agreement is required in order to avoid a prohibited distribution
under Section 409A(a)(2)(B)(i) of the Code, such portion of Executive’s benefits shall not be provided to Executive prior to the earlier of (i) the expiration
of the six (6)-month period measured from the date of Executive’s “separation from service” with the Company (as such term is defined in the Treasury
Regulations  issued  under  Section  409A  of  the  Code)  or  (ii)  the  date  of  Executive’s  death.  Upon  the  first  business  day  following  the  expiration  of  the
applicable Code Section 409A(a)(2)(B)(i)

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Exhibit 10.18

period,  all  payments  deferred  pursuant  to  this  Section  4.8(b)  shall  be  paid  in  a  lump  sum  to  Executive,  and  any  remaining  payments  due  under  this
Agreement shall be paid as otherwise provided herein.

c)

Expense Reimbursements.    To  the  extent  that  any  reimbursement  payable  pursuant  to  this  Agreement  is  subject  to  the
provisions of Section 409A of the Code, any such reimbursement payable to Executive pursuant to this Agreement shall be paid to Executive no later than
December 31 of the year following the year in which the expense was incurred; the amount of expenses reimbursed in one year shall not affect the amount
eligible  for  reimbursement  in  any  subsequent  year;  and  Executive’s  right  to  reimbursement  under  this  Agreement  will  not  be  subject  to  liquidation  or
exchange for another benefit.

Installments.    For  purposes  of  Section  409A  of  the  Code  (including,  without  limitation,  for  purposes  of  Treasury
Regulation Section 1.409A-2(b)(2)(iii)), Executive’s right to receive any installment payments under this Agreement shall be treated as a right to receive a
series of separate payments and, accordingly, each such installment payment shall at all times be considered a separate and distinct payment.

d)

4.9.

Tax Withholding. All  payments  under  this  Agreement  shall  be  subject  to  applicable  withholding  for  federal,  state  and

local income and employment taxes.

4.10.

No Duplication of Severance Benefits. The Severance Benefits and Change in Control Severance Benefits provided in
Section  2  and  Section  3  are  mutually  exclusive  of  each  other,  and  in  no  event  shall  Executive  receive  any  Severance  Benefits  or  Change  in  Control
Severance Benefits pursuant to both Section 2 and Section 3.  

5.  TERMINATION WITH CAUSE OR BY VOLUNTARY RESIGNATION; OTHER RIGHTS AND BENEFITS

5.1.

Termination  for  Cause;  Resignation  Without  Good  Reason;  Death  or  Disability.    If,  at  any  time,  the  Company
terminates Executive’s employment with the Company for Cause, or upon a voluntary resignation by Executive that is not a Resignation for Good Reason,
or Executive’s employment terminates for any reason not entitling Executive to the Severance Benefits or Change in Control Severance Benefits, or if
Executive’s employment terminates as a result of Executive’s death or disability (other than a Permanent Disability in the case of a Covered Termination),
then  the  Company  shall  have  no  further  obligation  to  Executive  hereunder  except  for  the  payment  or  provision,  as  applicable,  of  (i)  the  portion  of  the
Annual Base Salary accrued through Executive’s last day of employment, (ii) all unreimbursed expenses (if any), subject to Sections 1.4 and 4.8(c), and
(iii) any unused vacation (if applicable) accrued through Executive’s last day of employment.  Under these circumstances, Executive will not be entitled to
any other form of compensation, including any Severance Benefits or Change in Control Severance Benefits, other than Executive’s rights to the vested
portion of Executive’s Option and any other rights to which Executive is entitled under the Company’s benefit programs.    

5.2.

Other  Rights  and  Benefits.  Nothing  in  this  Agreement  shall  prevent  or  limit  Executive’s  continuing  or  future
participation  in  any  benefit,  bonus,  incentive  or  other  plans,  programs,  policies  or  practices  provided  by  the  Company  and  for  which  Executive  may
otherwise qualify, nor shall anything herein limit or otherwise affect such rights as Executive may have under other agreements with the Company except
as  provided  in  Section  4  and  Section  5.1  above.  Except  as  otherwise  expressly  provided  herein,  amounts  that  are  vested  benefits  or  that  Executive  is
otherwise  entitled  to  receive  under  any  plan,  policy,  practice  or  program  of  the  Company  at  or  subsequent  to  the  date  of  a  Change  in  Control  shall  be
payable in accordance with such plan, policy, practice or program.

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Exhibit 10.18

6.  DEFINITIONS

For purposes of this Agreement, the following definitions shall apply:

6.1.“Board” means the Board of Directors of the Company, or the compensation committee thereof, as determinations or responsibilities may

be delegated by the Board to the compensation committee.

6.2.

“Cause”  shall  mean  a  determination  by  the  Company  based  upon  reasonably  available  information  of  Executive’s:  (i)
unauthorized use or disclosure of the Company’s confidential information or trade secrets; (ii) material breach of any agreement to which the Executive
and the Company are a party; (iii) material failure to comply with the Company’s written policies or rules; (iv) conviction of, or plea of “guilty” or “no
contest”  to,  a  felony  under  the  laws  of  the  United  States  or  any  State;  (v)  negligence  or  willful  misconduct  relating  to  Executive’s  performance  of  her
duties on behalf of the Company; (vi) continuing failure to perform material and lawful assigned duties after receiving thirty (30) days’ written notification
of the failure from the Company if such breach is not cured (if curable) during that thirty (30) day period; (vii) failure to cooperate in good faith with a
governmental  or  internal  investigation  of  the  Company  or  its  directors,  officers  or  employees,  if  the  Company  has  requested  Executive’s  cooperation
without prejudice or personal liability to Executive; (viii) violation of employee or ethical guidelines including, without limitation, violations of business
practices and ethics commonly in place in similar companies in the United States; or (ix) violation of the Company code of conduct and/or any contractual
code of conduct to which the Company is obligated.

6.3.
more of the following events:

“Change  in  Control”  means  the  occurrence,  in  a  single  transaction  or  in  a  series  of  related  transactions,  of  any  one  or

a)

Any natural person, entity or group within the meaning of Section 13(d) or 14(d) of the Securities Exchange Act of 1934, as
amended (“Exchange Act Person”), becomes the owner, directly or indirectly, of securities of the Company representing more than fifty percent (50%) of
the  combined  voting  power  of  the  Company’s  then  outstanding  securities  other  than  by  virtue  of  a  merger,  consolidation  or  similar  transaction.
Notwithstanding the foregoing, a Change in Control shall not be deemed to occur (i) on account of the acquisition of securities of the Company by any
institutional investor, any affiliate thereof or any other Exchange Act Person that acquires the Company’s securities in a transaction or series of related
transactions that are primarily a private financing transaction for the Company or (ii) solely because the level of ownership held by any Exchange Act
Person  (the  “Subject  Person”)  exceeds  the  designated  percentage  threshold  of  the  outstanding  voting  securities  as  a  result  of  a  repurchase  or  other
acquisition of voting securities by the Company reducing the number of shares outstanding, provided that if a Change in Control would occur (but for the
operation of this sentence) as a result of the acquisition of voting securities by the Company, and after such share acquisition, the Subject Person becomes
the  owner  of  any  additional  voting  securities  that,  assuming  the  repurchase  or  other  acquisition  had  not  occurred,  increases  the  percentage  of  the  then
outstanding voting securities owned by the Subject Person over the designated percentage threshold, then a Change in Control shall be deemed to occur;

b)

There  is  consummated  a  merger,  consolidation  or  similar  transaction  involving,  directly  or  indirectly,  the  Company  if,
immediately after the consummation of such merger, consolidation or similar transaction, the stockholders of the Company immediately prior thereto do
not  own,  directly  or  indirectly,  either  (i)  outstanding  voting  securities  representing  more  than  fifty  percent  (50%)  of  the  combined  outstanding  voting
power of the surviving entity in such merger, consolidation or similar transaction or (ii) more than fifty percent (50%) of the combined outstanding voting
power of the parent of the surviving entity in such merger, consolidation or similar transaction; or

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Exhibit 10.18

c)

There is consummated a sale, lease, license or other disposition of all or substantially all of the consolidated assets of the
Company and its subsidiaries, other than a sale, lease, license or other disposition of all or substantially all of the consolidated assets of the Company and
its subsidiaries to an entity, more than fifty percent (50%) of the combined voting power of the voting securities of which are owned by stockholders of the
Company in substantially the same proportion as their ownership of the Company immediately prior to such sale, lease, license or other disposition.

The term Change in Control shall not include a sale of assets, merger or other transaction effected exclusively for the purpose of changing the
domicile of the Company. Notwithstanding the foregoing or any other provision of this Agreement, the definition of Change in Control (or any analogous
term) in an individual written agreement between the Company or any affiliate and the participant shall supersede the foregoing definition with respect to
stock awards subject to such agreement (it being understood, however, that if no definition of Change in Control or any analogous term is set forth in such
an individual written agreement, the foregoing definition shall apply).

6.4.

6.5.

“Change in Control Benefits Period” means the period of twelve (12) months commencing on the Termination Date.

“Change in Control Severance Period” means the period of twelve (12) months commencing on the Termination Date.

6.6.

  “Change  in  Control  Termination”  means  an  “Involuntary  Termination  Without  Cause”  or  “Resignation  for  Good
Reason,” either of which occurs within three (3) months prior to or upon or within twelve (12) months following the closing of a Change in Control or
Dissolution  Event,  provided  that  any  such  termination  is  a  “separation  from  service”  within  the  meaning  of  Treasury  Regulation  Section  1.409A-
1(h).  Death and disability shall not be deemed Change in Control Terminations.

6.7.

6.8.

6.9.

“COBRA” means the Consolidated Omnibus Budget Reconciliation Act of 1985, as amended.

“Code” means the Internal Revenue Code of 1986, as amended.

“Company”  means  Ovid  Therapeutics  Inc.  or,  following  a  Change  in  Control,  the  surviving  entity  resulting  from  such

transaction, or any subsequent surviving entity resulting from any subsequent Change in Control.

6.10.

“Confidentiality Agreement”  means  Senior  Executive  Confidential  Information  and  Invention  Assignment  Agreement

with the Company, (or any successor agreement thereto).

6.11.

  “Covered  Termination”  means  an  “Involuntary  Termination  Without  Cause”  or  “Resignation  for  Good  Reason,”
provided that any such termination is a “separation from service” within the meaning of Treasury Regulation Section 1.409A-1(h). Death and disability,
other  than  a  Permanent  Disability,  shall  not  be  deemed  Covered  Terminations.    If  an  Involuntary  Termination  Without  Cause  or  Resignation  for  Good
Reason qualifies as a Change in Control Termination, it shall not constitute a Covered Termination.  

6.12.

6.13.

Date.

148402431 v2

“Covered Termination Benefits Period” means the period of twelve (12) months commencing on the Termination Date.

“Covered  Termination  Severance  Period”  means  the  period  of  twelve  (12)  months  commencing  on  the  Termination

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Exhibit 10.18

6.14.

“Dissolution  Event”  means  the  stockholders  of  the  Company  approve  or  the  Board  approves  a  plan  of  complete

dissolution or liquidation of the Company, or a complete dissolution or liquidation of the Company shall otherwise occur.

6.15.

“Involuntary Termination Without Cause” means Executive’s dismissal or discharge by the Company for reasons other
than  Cause  and  other  than  as  a  result  of  death  or  disability;  provided, however,  that  for  purposes  of  a  Covered  Termination,  Involuntary  Termination
Without Cause shall include Executive’s dismissal or discharge by the Company for reasons of Permanent Disability.

6.16.

  “Monthly  Base  Salary”  means  1/12th  of  Executive’s  Annual  Base  Salary  (excluding  incentive  pay,  premium  pay,
commissions,  overtime,  bonuses  and  other  forms  of  variable  compensation)  as  in  effect  on  the  date  of  a  Covered  Termination  or  Change  in  Control
Termination.

6.17.

“Permanent Disability” means total and permanent disability as defined in Code Section 22(e)(3).

6.18.

“Resignation for Good Reason” means Executive’s resignation from all employee positions Executive then holds with
the  Company  within  ninety  (90)  days  following  any  of  the  following  events  taken  without  Executive’s  consent,  provided  Executive  has  given  the
Company written notice of such event within thirty (30) days after the first occurrence of such event and the Company has not cured such event within
thirty (30) days thereafter:

comparable executives of the Company;

a)

A material decrease in Executive’s Annual Base Salary, other than in connection with a decrease in compensation for all

b)

c)

A relocation of Executive’s principal place of work outside of a fifty (50) mile radius of its current location; or

The Company’s material breach of this Agreement.

6.19.

“Termination Date” means the effective date of a Change in Control Termination, a Covered Termination, a termination

for Cause or any other circumstance under which the employment relationship between Executive and the Company terminates, as applicable.

6.20.

“Division” shall mean only that part, unit or therapeutic category of a larger entity that is competitive with the Company,

but not an entire company itself, if other divisions, units or therapeutic categories of such larger company are not competitive with the Company.

6.21.

"Client"  shall  mean  (A)  anyone  who  is  a  client  of  the  Company  as  of,  or  at  any  time  during  the  one-year  period
immediately preceding, the termination of Executive’s employment, but only if Executive had a direct relationship with, supervisory responsibility for or
otherwise were involved with such client during Executive’s employment with the Company; and (B) any prospective client to whom the Company made
a  new  business  presentation  (or  similar  offering  of  services)  at  any  time  during  the  one-year  period  immediately  preceding,  or  six-month  period
immediately following, Executive’s employment termination (but only if initial discussions between the Company and such prospective client relating to
the rendering of services occurred prior to the termination date, and only if Executive participated in or supervised such presentation and/or its preparation
or the discussions leading up to it).

6.22.

“Solicit”  shall  mean:  (A)  active  solicitation  of  any  Client  or  Company  employee,  board  member,  advisor,  consultant,
collaborator,  investigator  or  agents;  (B)  the  provision  of  information  regarding  any  Client  or  Company  employee,  board  member,  advisor,  consultant,
collaborator, investigator or agents to any third party where such information could be useful to such third party in attempting to obtain business from such
Client or attempting to hire any such Company employee; (C) participation in any meetings, discussions, or other communications with any third party
regarding any Client or Company employee, board member, advisor, consultant, collaborator, investigator

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Exhibit 10.18

or  agents  where  the  purpose  or  effect  of  such  meeting,  discussion  or  communication  is  to  obtain  business  from  such  Client  or  employ  such  Company
employee;  and  (D)  any  other  passive  use  of  information  about  any  Client  or  Company  employee,  board  member,  advisor,  consultant,  collaborator,
investigator or agents which has the purpose or effect of assisting a third party or causing harm to the business of the Company.

7.  GENERAL PROVISIONS

7.1.

Employment  Status.    This  Agreement  does  not  constitute  a  contract  of  employment  or  impose  upon  Executive  any
obligation  to  remain  as  an  employee,  or  impose  on  the  Company  any  obligation  (i)  to  retain  Executive  as  an  employee,  (ii)  to  change  the  status  of
Executive as an at-will employee or (iii) to change the Company’s policies regarding termination of employment.

7.2.

Notices. Any notices provided hereunder must be in writing, and such notices or any other written communication shall be
deemed effective upon the earlier of personal delivery (including personal delivery by facsimile or email transmission (to a facsimile number or email
address designated in advance by the receiving party)) or the third day after mailing by first class mail, to the Company at its primary office location and to
Executive at Executive’s address as listed in the Company’s payroll records. Any payments made by the Company to Executive under the terms of this
Agreement shall be delivered to Executive either in person or at the address as listed in the Company’s payroll records.

7.3.

Severability. Whenever possible, each provision of this Agreement will be interpreted in such manner as to be effective
and  valid  under  applicable  law,  but  if  any  provision  of  this  Agreement  is  determined  to  be  invalid,  illegal  or  unenforceable  in  any  respect  under  any
applicable law or rule in any jurisdiction, such invalidity, illegality or unenforceability will not affect any other provision or any other jurisdiction, and the
provision in question shall be modified so as to be rendered enforceable in a manner consistent with the intent of the parties insofar as possible under
applicable law.

7.4.

Waiver. If either party should waive any breach of any provisions of this Agreement, he, she or it shall not thereby be

deemed to have waived any preceding or succeeding breach of the same or any other provision of this Agreement.

7.5.

Complete  Agreement.  This  Agreement,  together  with  Exhibits  A  thru  D,  the  Confidentiality  Agreement  and  the
Indemnification Agreement, forms the complete and exclusive statement of Executive’s employment agreement with the Company, and supersedes and
replaces any other agreements or promises made to Executive by anyone, whether oral or written (including but not limited to the Prior Agreement).

7.6.

Amendment or Termination of Agreement; Continuation of Agreement. Except for those changes expressly reserved
to the Company’s or the Board’s discretion in this Agreement, this Agreement may be changed or terminated only upon the mutual written consent of the
Company and Executive. The written consent of the Company to a change or termination of this Agreement must be signed by an executive officer of the
Company (other than Executive) after such change or termination has been approved by the Board. Unless so terminated, this Agreement shall continue in
effect for as long as Executive continues to be employed by the Company or by any surviving entity following any Change in Control. For the avoidance
of any doubt, if, following a Change in Control, Executive continues to be employed by the surviving entity without a Change in Control Termination and
the surviving entity then

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Exhibit 10.18

undergoes  a  Change  in  Control,  following  which  Executive  is  terminated  by  the  subsequent  surviving  entity  in  a  Change  in  Control  Termination,
Executive shall receive the benefits described in Section 3 hereof.  

7.7.

Counterparts. This Agreement may be executed in separate counterparts, any one of which need not contain signatures of
more than one party, but all of which taken together will constitute one and the same Agreement.  Facsimile and electronic image copies of signatures shall
be equivalent to original signatures.  

7.8.

Headings. The headings of the Sections hereof are inserted for convenience only and shall not be deemed to constitute a

part hereof nor to affect the meaning thereof.

7.9.

Successors and Assigns. This Agreement is intended to bind and inure to the benefit of and be enforceable by Executive,
and  the  Company,  and  any  surviving  entity  resulting  from  a  Change  in  Control  and  upon  any  other  person  who  is  a  successor  by  merger,  acquisition,
consolidation  or  otherwise  to  the  business  formerly  carried  on  by  the  Company,  and  their  respective  successors,  assigns,  heirs,  executors  and
administrators, without regard to whether or not such person actively assumes any rights or duties hereunder; provided, however, that Executive may not
assign any duties hereunder and may not assign any rights hereunder without the written consent of the Company, which consent shall not be withheld
unreasonably.

7.10.

Choice of Law. This Agreement shall be construed and enforced in accordance with the laws of the State of New York

without regard to conflicts of law principles. 

7.11.

Arbitration.    To  ensure  the  rapid  and  economical  resolution  of  any  disputes  that  may  arise  under  or  relate  to  this
Agreement or Executive’s employment relationship, Executive and the Company agree that, unless otherwise prohibited by applicable law, any and all
disputes,  claims,  or  causes  of  action,  in  law  or  equity,  arising  from  or  relating  to  the  performance,  enforcement,  execution,  or  interpretation  of  this
Agreement, Executive’s employment with the Company, or the termination of Executive’s employment (collectively, “Claims”), shall be resolved by final,
binding, and (to the extent permitted by law) confidential arbitration before a single arbitrator in New York, New York.  Executive and the Company agree
that  they  shall  resolve  all  such  Claims  in  accordance  with  the  provisions  of  Section  12  of  the  Confidential  Information  and  Invention  Assignment
Agreement attached hereto as Exhibit A.    

7.12.

Construction of Agreement. In the event of a conflict between the text of this Agreement and any summary, description

or other information regarding this Agreement, the text of this Agreement shall control.

7.13.

Circular  230  Disclaimer.  THE  FOLLOWING  DISCLAIMER  IS  PROVIDED  IN  ACCORDANCE  WITH  THE
INTERNAL  REVENUE  SERVICE’S  CIRCULAR  230  (21  C.F.R.  PART  10).  ANY  TAX  ADVICE  CONTAINED  IN  THIS  AGREEMENT  IS
INTENDED TO BE PRELIMINARY, FOR DISCUSSION PURPOSES ONLY AND NOT FINAL. ANY SUCH ADVICE IS NOT INTENDED
TO BE USED FOR MARKETING, PROMOTING OR RECOMMENDING ANY TRANSACTION OR FOR THE USE OF ANY PERSON IN
CONNECTION WITH THE PREPARATION OF ANY TAX RETURN. ACCORDINGLY, THIS ADVICE IS NOT INTENDED OR WRITTEN
TO  BE  USED,  AND  IT  CANNOT  BE  USED,  BY  ANY  PERSON  FOR  THE  PURPOSE  OF  AVOIDING  TAX  PENALTIES  THAT  MAY  BE
IMPOSED ON SUCH PERSON.

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SIGNATURE PAGE TO FOLLOW

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REVIEWED, UNDERSTOOD AND ACCEPTED:

OVID THERAPEUTICS INC.

EXECUTIVE

Suzanne K. Wakamoto
SVP, Human Resources

By:
Name:
Title:

148402431 v2

By: 
Name: 

Jason Tardio

Exhibit 10.18

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Exhibit 10.19

AMENDED AND RESTATED EXECUTIVE EMPLOYMENT AGREEMENT

Thomas Perone (“Executive”) is currently employed by OVID THERAPEUTICS INC. (the “Company”) as its General Counsel, Corporate Secretary
and Chief Compliance Officer pursuant to the terms of an Executive Employment Agreement with the Company effective March 11, 2019 (the “Prior
Agreement”).   Executive and the Company hereby agree to this amended agreement.   The terms and conditions set forth in this AMENDED AND
RESTATED EXECUTIVE EMPLOYMENT AGREEMENT (this “Agreement”) shall become effective as of January 1, 2020 (the “Effective Date”)
and shall supersede and replace the terms and conditions set forth in the Prior Agreement.  Certain bolded terms used in this Agreement are defined in
Section 6.  

WHEREAS, the Company is a biopharmaceutical company;

WHEREAS,  the  Company  desires  to  employ  Executive  in  the  position  set  forth  below,  and  wishes  to  provide  Executive  with  certain

compensation and benefits in return for such services, as set forth in this Agreement; and

WHEREAS,  Executive  wishes  to  be  employed  by  the  Company  and  to  provide  personal  services  to  the  Company  in  return  for  certain

compensation and benefits, as set forth in this Agreement.

NOW, THEREFORE, in consideration of the mutual promises contained herein and for other good and valuable consideration, the receipt

and sufficiency of which is hereby acknowledged, the Company and Executive agree as follows:

1.  TERMS OF EMPLOYMENT

1.1.

Position,  Duties  and  Location.    Executive  shall  initially  serve  as  General  Counsel,  Corporate  Secretary  and  Chief
Compliance Officer reporting to the Company’s Chief Executive Officer.  Executive shall perform those duties and responsibilities as are customary for
such position and as may be directed by the Company and the Board from time to time. During Executive’s employment with the Company, Executive
shall devote Executive’s best efforts and substantially all of Executive’s business time and attention to the business of the Company, except for approved
vacation periods and reasonable periods of illness or other incapacities permitted by the Company’s general employment policies.  Executive’s primary
office location will be the Company’s offices in New York City, NY.  Notwithstanding the foregoing, the Company reserves the right to reasonably require
Executive  to  perform  Executive’s  duties  at  places  other  than  Executive’s  primary  office  location  from  time  to  time,  and  to  require  reasonable  business
travel.    During  Executive’s  employment  with  the  Company,  Executive  shall  not  engage  in  any  activity  that  conflicts  with  or  is  detrimental  to  the
Company’s best interests, as determined by the CEO.  

Executive  may  participate  as  in  side  activities  such  as  board  or  committee  member,  advisor  or  consultant  (the  “Activities”),  provided  that  Executive
obtains  their  manager’s  prior  written  consent,  and  that  none  of  the  following  activities  involve  activities  in  the  area  of  neurology,  detract  from  Ovid’s
reputation,  impact  Executive’s  full  time  duties  to  the  Company,  or  could  reasonably  result  in  the  disclosure  or  use  of  the  Company’s  proprietary  or
confidential information.  The manager may rescind their consent to Executive’s participation in the Activities, or participation in other business or public
activities, if the manager, in their

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1946726.1 29165-0001-000

D-1

 
 
 
 
sole discretion, determines that such activities compromise or threaten to compromise the Company’s business interests or conflict with Executive’s duties
to the Company.

1.2.

Employment  Term.    Executive  will  be  employed  by  the  Company  on  an  “at-will”  basis.    This  means  that  either  the
Company or Executive may terminate Executive’s employment at any time, for any reason, with or without Cause, and with or without advance notice
(provided  that  (a)  Resignation  for  Good  Reason  (as  defined  below)  requires  certain  advanced  notice  by  Executive  of  Executive’s  termination  of
employment as set forth below and (b) as a professional courtesy, Executive agrees to provide the Company with at least sixty (60) days advance written
notice of a voluntary resignation by Executive that is not a Resignation for Good Reason).  Subject to the terms herein, it also means that Executive’s job
title, duties, responsibilities, reporting level, compensation and benefits, as well as the Company’s personnel policies and procedures, may be changed with
or without notice at any time in the Company’s sole discretion.  This at-will employment relationship shall not be modified by any conflicting actions or
representations of any Company employee or other party before or during the term of Executive’s employment.   

1.3.

Compensation.

a)

Annual  Base  Salary.      Executive’s  annual  base  salary  shall  be  paid  at  the  rate  of  $440,000  per  year
(“Annual Base Salary”),  payable  in  equal  installments,  less  applicable  payroll  deductions  and  withholdings,  on  the  Company’s  ordinary  payroll  cycle.
Executive’s Annual Base Salary shall be subject to annual review by the Board and may be adjusted from time to time.  As an exempt salaried employee,
Executive will be required to work the Company’s normal business hours, and such additional time as appropriate for Executive’s work assignments and
position, and Executive will not be entitled to overtime compensation.

Benefits.  Executive  will  be  eligible  to  participate  in  all  of  the  Company’s  employee  benefits  and  benefit
plans that the Company generally makes available to its full-time employees and executives in accordance with the terms and conditions of the benefit
plans and applicable policies as in effect from time to time.  

b)

c)

Bonus.  Executive  shall  be  eligible  to  earn  an  annual  performance  bonus  of  up  to  thirty  percent  40%  of
Executive’s Annual Base Salary (the “Target Performance Bonus”).  The Target Performance Bonus shall be based upon the Company’s assessment of
Executive’s attainment of written Company and individual objectives as set by the Company in its sole discretion.  The Company may increase the Target
Performance Bonus in its sole discretion.  Bonus payments, if any, shall be subject to applicable payroll deductions and withholdings.  Following the close
of each calendar year, the Company shall determine whether Executive has earned a Target Performance Bonus, and the amount of any such bonus, based
on the achievement of such objectives.  Executive must be an employee of the Company in good standing on the Target Performance Bonus payment date
to be eligible to receive a Target Performance Bonus, and no partial or prorated bonuses shall be provided.  The Target Performance Bonus, if earned, shall
be paid on or before March 15th of the calendar year after the applicable bonus year.  Executive’s bonus eligibility is subject to change in the discretion of
the Company.   If Executive’s  start date with the Company falls within the fourth quarter, the Executive will not  be eligible for a target bonus for that
calendar year.  

Equity Compensation., Executive shall be granted options to purchase shares of the Company’s common
stock (the “Option”)  as  determined  by  Management  and  approved  by  the  Compensation  Committee.  The  Option  will  be  evidenced  by  a  stock  option
agreement and be subject to

d)

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the terms and conditions of the Company’s 2017 Equity Incentive Plan (the “Equity Plan”). The exercise price per share of the Option will be equal to
the  per  share  fair  market  value  of  the  Company’s  common  stock  on  the  date  the  Option  is  granted,  as  defined  under  the  Equity  Plan.  The  vesting
schedule of the Option will be as follows: twenty-five percent (25%) of the shares of the Company’s common stock subject to the Option will vest on the
one year anniversary of the Start Date, and one thirty-sixth (1/36th) of the remaining shares of the Company’s common stock subject to the Option will
vest each month thereafter on the same day of the month as the Executive’s date of hire (and if there is no corresponding day, on the last day of the
month), so long as Executive remains an employee, consultant, director or officer of the Company, and subject to the terms and conditions of the stock
option agreement and the Equity Plan. Subject to the approval of the Board, the stock option agreement shall provide that upon a Change in Control
Termination, the vesting and exercisability of the Option shall be accelerated in full. At the discretion of the Board, Executive will be eligible to receive
additional options to purchase shares of the Company’s common stock.

e)

Any raise or bonus connected with performance in you first calendar year of service will be prorated from
your start date. Ongoing Stock Option Grants are awarded at the Company’s discretion; eligible Ovidians typically are awarded these grants in the first
quarter. New Ovidians who start in the fourth quarter are not eligible for a raise or bonus for that calendar year and are not eligible for the Ongoing Grant
awarded in first quarter of the following year.

1.4.

Reimbursement  of  Expenses.    Subject  to  Section  4.8(c),  the  Company  shall  reimburse  Executive  for  Executive’s
necessary  and  reasonable  business  expenses  incurred  in  connection  with  Executive’s  duties  in  accordance  with  the  Company’s  generally  applicable
expense reimbursement policies as in effect from time to time.  

1.5.

Indemnification  Agreement.  Executive  and  Company  shall  enter  into  an  Indemnity  Agreement  (the  “Indemnification

Agreement”), which shall be effective as of the Start Date and is incorporated herein by reference.  

1.6.

Compliance with Confidentiality Agreement and Company Policies.  Executive shall execute and abide by all terms
and provisions of the Confidentiality Agreement to be signed on or prior to the Start Date (or any successor agreement thereto), attached hereto as Exhibit
A.  Executive  shall  also  abide  by  all  terms  and  provisions  of  the  Company’s  Code  of  Business  Conduct  and  Ethics,  attached  hereto  as  Exhibit  D.  In
addition, Executive is required to abide by the Company’s policies and procedures, including but not limited to the Company’s Employee Handbook, as
adopted or modified from time to time within the Company’s discretion; provided, however, that in the event the terms of this Agreement differ from or
are in conflict with the Company’s general employment policies or practices, this Agreement shall control.  

2.  COVERED TERMINATION SEVERANCE BENEFITS

2.1.

Severance Benefits.  Upon a Covered Termination, then subject to Section 4 below and Executive’s continued compliance

with the terms of this Agreement, the Company shall provide Executive with the severance benefits set forth in this Section 2 (the “Severance Benefits”).

2.2.

Salary Payment.  The Company shall pay Executive, as cash severance, (i) Executive’s Monthly Base Salary, multiplied
by (ii) the number of months in the Covered Termination Severance Period, less applicable payroll deductions and withholdings (the “Severance”). The
Severance shall be paid (except as set forth in Section 4) in equal installments on the Company’s ordinary payroll cycle

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commencing on the first regularly-scheduled payroll date occurring on or after the Release Deadline Date (as set forth in Section 4.1).

2.3.

Health Continuation Payments.

a)

The Company will pay Executive on the first day of each month a fully taxable cash payment equal to the
applicable  premium  for  Executive,  her  spouse  and  any  dependents  for  the  group  health  plan  maintained  by  the  Company  for  the  month  in  which  the
Covered Termination occurs, subject to applicable tax withholdings but grossed up for all taxes owed by the Executive on such payment, for the duration
of the Covered Termination Benefits Period. Such coverage shall be counted as coverage pursuant to COBRA. The Company shall have no obligation in
respect of any premium payments following the effective date of the Executive’s coverage by a health insurance plan of a subsequent employer. Executive
shall be required to notify the Company immediately if Executive becomes covered by a health insurance plan of a subsequent employer.

For purposes of this Section 2.3, (i) references to COBRA shall be deemed to include analogous provisions
of state law, and (ii) any applicable insurance premiums that are paid by the Company shall not include any amounts payable by Executive under a Code
Section 125 health care reimbursement plan, which amounts, if any, are the sole responsibility of Executive.

b)

3.  CHANGE IN CONTROL SEVERANCE BENEFITS

3.1.

Change  in  Control  Severance  Benefits.    Upon  a  Change  in  Control  Termination,  then  subject  to  Section  4  below  and
Executive’s continued compliance with the terms of this Agreement, the Company shall provide Executive with the severance benefits set forth in this
Section 3 (the “Change in Control Severance Benefits”).  

3.2.

Salary Payment.  The Company shall pay Executive, as cash severance, (i) Executive’s Monthly Base Salary, multiplied
by (ii) the number of months in the Change in Control Severance Period, less applicable payroll deductions and withholdings (the “Change  in  Control
Severance”). The Change in Control Severance shall be paid (except as set forth in Section 4) in equal installments on the Company’s ordinary payroll
cycle commencing on the first regularly-scheduled payroll date occurring on or after the Release Deadline Date.  

3.3.

Health Continuation Payments.

a)The Company will pay Executive on the first day of each month a fully taxable cash payment equal to the applicable premium
for  Executive,  her  spouse  and  any  dependents  for  the  group  health  plan  maintained  by  the  Company  for  the  month  in  which  the  Change  in  Control
Termination occurs, subject to applicable tax withholdings but grossed up for all taxes owed by the Executive on such payment, for the duration of the
Change in Control Benefits Period. Such coverage shall be counted as coverage pursuant to COBRA. The Company shall have no obligation in respect of
any premium payments following the effective date of the Executive’s coverage by a health insurance plan of a subsequent employer. Executive shall be
required to notify the Company immediately if Executive becomes covered by a health insurance plan of a subsequent employer.

For purposes of this Section 3.3, (i) references to COBRA shall be deemed to include analogous provisions
of state law, and (ii) any applicable insurance premiums that are paid by the Company shall not include any amounts payable by Executive under a Code
Section 125 health care reimbursement plan, which amounts, if any, are the sole responsibility of Executive.

b)

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3.4.

Change in Control Termination Vesting Acceleration Benefits.  Upon a Change in Control Termination, (i) the vesting
and  exercisability  of  all  outstanding  options  to  purchase  the  Company’s  common  stock  (or  stock  appreciation  rights  or  other  rights  with  respect  to  the
stock  of  the  Company  issued  pursuant  to  any  equity  incentive  plan  of  the  Company)  that  are  held  by  Executive  on  the  Termination  Date  shall  be
accelerated in full, (ii) each such option shall be exercisable and to the extent not exercised, expire on the latest date permitted under the Equity Plan and
(iii)  any  reacquisition  or  repurchase  rights  held  by  the  Company  with  respect  to  common  stock  issued  or  issuable  (or  with  respect  to  other  rights  with
respect to the stock of the Company issued or issuable) pursuant to any other stock award granted to Executive pursuant to any equity incentive plan of the
Company shall lapse.

4.  LIMITATIONS AND CONDITIONS ON BENEFITS

4.1.

Release  Prior  to  Payment  of  Severance  Benefits  and  Change  in  Control  Severance  Benefits.    The  receipt  of  any
Severance Benefits or Change in Control Severance Benefits pursuant to this Agreement is subject to Executive signing and not revoking a separation
agreement and general release of claims (the “Release”), in substantially the form attached hereto and incorporated herein as Exhibit B or Exhibit C, as
appropriate, and subject to any further modifications as determined in the Company’s discretion, which Release must become effective and irrevocable no
later than the sixtieth (60th) day following Executive’s Termination Date (the “Release Deadline Date”).  If the Release does not become effective and
irrevocable by the Release Deadline Date, Executive will forfeit any right to any Severance Benefits or Change in Control Severance Benefits under this
Agreement.  In no event will Severance Benefits or Change in Control Severance Benefits be paid or provided until after the Release Deadline Date.  On
the first regularly-scheduled payroll date occurring on or after the Release Deadline Date, the Company will pay Executive the Severance or Change in
Control Severance amount that Executive would otherwise have received on or prior to such date but for the delay in payment related to the effectiveness
of the Release, with the balance of the Severance or Change in Control Severance amount being paid as originally scheduled. The Company may modify
the Release in its discretion to comply with changes in applicable law at any time prior to Executive’s execution of such Release.

4.2.

Return of Company Property.  Not later than the Termination Date, or earlier if requested by the Company, Executive
shall  return  to  the  Company  all  documents  (and  all  copies  thereof)  and  other  property  belonging  to  the  Company  that  Executive  has  in  his  or  her
possession  or  control.  The  documents  and  property  to  be  returned  include,  but  are  not  limited  to,  all  files,  correspondence,  email,  memoranda,  notes,
notebooks,  records,  plans,  forecasts,  reports,  studies,  analyses,  compilations  of  data,  proposals,  agreements,  financial  information,  research  and
development information, marketing information, operational and personnel information, databases, computer-recorded information, tangible property and
equipment (including, but not limited to, computers, facsimile machines, mobile telephones and servers), credit cards, entry cards, identification badges
and  keys,  and  any  materials  of  any  kind  which  contain  or  embody  any  proprietary  or  confidential  information  of  the  Company  (and  all  reproductions
thereof in whole or in part). Executive agrees to make a diligent search to locate any such documents, property and information. If Executive has used any
personally owned computer, server or e-mail system to receive, store, review, prepare or transmit any Company confidential or proprietary data, materials
or  information,  then  within  ten  (10)  business  days  after  the  Termination  Date,  or  earlier  if  requested  by  the  Company,  Executive  shall  provide  the
Company with a computer-useable copy of all such information and then permanently delete and expunge such confidential or proprietary information
from those systems. Executive agrees to provide the Company with a certification that the necessary copying and/or deletion is done.

4.3.

Cooperation and Continued Compliance with Restrictive Covenants.

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a)

After the Termination Date, Executive shall cooperate fully with the Company, at reasonable times as agreed
between  Executive  and  the  Company,  in  connection  with  its  actual  or  contemplated  defense,  prosecution  or  investigation  of  any  existing  or  future
litigation, arbitrations, mediations, claims, demands, audits, government or regulatory inquiries, or other matters arising from events, acts or failures to act
that occurred during the time period in which Executive was employed by the Company (including any period of employment with an entity acquired by
the Company). Such cooperation includes, without limitation, being available upon reasonable notice, without subpoena, to provide accurate and complete
advice,  assistance  and  information  to  the  Company,  including  offering  and  explaining  evidence,  providing  truthful  and  accurate  sworn  statements,  and
participating  in  discovery  and  trial  preparation  and  testimony.  Executive  also  agrees  to  promptly  send  the  Company  copies  of  all  correspondence  (for
example, but not limited to, subpoenas) received by Executive in connection with any such legal proceedings, unless Executive is expressly prohibited by
law from so doing.  Nothing in this Agreement prohibits Executive from responding accurately and fully to any request for information if required by legal
process  or  in  connection  with  a  government  investigation.    In  addition,  nothing  in  this  Agreement  is  intended  to  prohibit  or  restrain  Executive  in  any
manner  from  making  disclosures  that  are  protected  under  the  whistleblower  provisions  of  federal  law  or  regulation  or  under  other  applicable  law  or
regulation.  The Company will reimburse Executive for reasonable out-of-pocket expenses incurred in connection with any such cooperation (excluding
foregone  wages,  salary  or  other  compensation)  within  thirty  (30)  days  of  Executive’s  timely  presentation  of  appropriate  documentation  thereof,  in
accordance  with  the  Company’s  standard  reimbursement  policies  and  procedures.  The  Company  will  reasonably  accommodate  Executive’s  scheduling
needs with respect to any such cooperation after the Termination Date.

the Confidentiality Agreement.

b)

After the Termination Date, Executive shall continue to abide by Executive’s continuing obligations under

c)

From  the  Start  Date  and  through  and  including  the  Change  in  Control  Severance  Period  or  Covered
Termination Severance Period as defined below, or, if Executive is Terminated with Cause, for one year after Executive’s Termination Date, whichever is
applicable,  Executive  shall  not,  without  the  Company’s  prior  written  consent,  whether  directly  or  indirectly  be  employed,  under  contract  with,  provide
services to or on behalf of, or be involved with any business or organization (whether “for profit” or  “not-for-profit”), or applicable Division thereof (as
defined  below),  which  researches,  develops,  creates,  manufactures,  designs  and/or  sells  compounds  and/or  related  pharmaceuticals,  medicines  and/or
therapies  to  treat  rare  or  orphan  neurological  conditions  or  diseases,  and/or  otherwise  competes  with  products  and/or  services  then  under  research  or
development by or offered or sold by the Company in the same therapeutic category.  Nothing in Section 4.3(c) shall prohibit Executive from investing as
a less than one percent (1%) shareholder in securities of any company listed on a national securities exchange or quoted on an automated quotation system.

d)

From the Start Date until twelve (12) months after Termination Date, Executive shall not hire or retain, or
attempt to hire or retain, any of the Company’s then-existing board members, employees, advisors, consultants, collaborators, investigators or agents and
shall not induce any such to give up employment with or to cease providing services to the Company, and shall not otherwise interfere with, or attempt to
interfere with, the relationship of any such person with the Company; or attempt in any manner to solicit, persuade or induce any Client of the Company to
terminate, reduce or refrain from renewing or extending its contractual or other relationship with the Company in regard to the purchase of products or
services  marketed  or  sold  by  the  Company,  or  to  become  a  Client  of  or  enter  into  any  contractual  or  other  relationship  with  Executive  or  any  other
individual, person or entity in regard to the purchase of products or services similar or identical to those marketed or sold by the Company.

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e)

Executive acknowledges and agrees that Executive’s obligations under this Section 4.3 are an essential part
of the consideration Executive is providing hereunder in exchange for which and in reliance upon which the Company has agreed to provide the payments
and benefits under this Agreement. Executive further acknowledges and agrees that Executive’s violation of this Section 4.3 inevitably would involve use
or  disclosure  of  the  Company’s  proprietary  and  confidential  information.  If  it  is  determined  by  a  court  of  competent  jurisdiction  in  any  state  that  any
restriction in this Section 4.3 is excessive in duration or scope or is unreasonable or unenforceable under the laws of that state, it is the intention of the
parties that such restriction may be modified or amended by the court to render it enforceable to the maximum extent permitted by the law of that state.

4.4.

Parachute Payments.

a)

Parachute  Payment  Limitation.    If  any  payment  or  benefit  (including  payments  and  benefits  pursuant  to  this
Agreement)  Executive  would  receive  in  connection  with  a  Change  in  Control  from  the  Company  or  otherwise  (“Payment”)  would  (i)  constitute  a
“parachute  payment”  within  the  meaning  of  Section  280G  of  the  Code,  and  (ii)  but  for  this  paragraph,  be  subject  to  the  excise  tax  imposed  by
Section 4999 of the Code (the “Excise Tax”), then the Company shall cause to be determined, before any amounts of the Payment are paid to Executive,
which of the following two alternative forms of payment shall be paid to Executive: (A) payment in full of the entire amount of the Payment (a “Full
Payment”), or (B) payment of only a part of the Payment so that Executive receives the largest payment possible without the imposition of the Excise Tax
(a “Reduced Payment”). A Full Payment shall be made in the event that the amount received by the Executive on a net after-tax basis is greater than what
would be received by the Executive on a net after-tax basis if the Reduced Payment were made, otherwise a Reduced Payment shall be made. If a Reduced
Payment is made, (i) the Payment shall be paid only to the extent permitted under the Reduced Payment alternative, and Executive shall have no rights to
any  additional  payments  and/or  benefits  constituting  the  Payment,  and  (ii)  reduction  in  payments  and/or  benefits  shall  occur  in  the  following  order:
(A) reduction of cash payments; (B) cancellation of accelerated vesting of equity awards other than stock options; (C) cancellation of accelerated vesting
of stock options; and (D) reduction of other benefits paid to Executive. In the event that acceleration of compensation from Executive’s equity awards is to
be reduced, such acceleration of vesting shall be canceled in the reverse order of the date of grant.

b)

The independent registered public accounting firm engaged by the Company for general audit purposes as
of the day prior to the effective date of the Change in Control shall make all determinations required to be made under this Section 4.4. If the independent
registered public accounting firm so engaged by the Company is serving as accountant or auditor for the individual, entity or group effecting the Change in
Control, the Company shall appoint a nationally recognized independent registered public accounting firm to make the determinations required hereunder.
The  Company  shall  bear  all  expenses  with  respect  to  the  determinations  by  such  independent  registered  public  accounting  firm  required  to  be  made
hereunder.

c)

The  independent  registered  public  accounting  firm  engaged  to  make  the  determinations  hereunder  shall
provide its calculations, together with detailed supporting documentation, to the Company and Executive within fifteen (15) calendar days after the date on
which Executive’s right to a Payment is triggered (if requested at that time by the Company or Executive) or such other time as requested by the Company
or Executive. If the independent registered public accounting firm determines that no Excise Tax is payable with respect to a Payment, either before or
after  the  application  of  the  Reduced  Amount,  it  shall  furnish  the  Company  and  Executive  with  an  opinion  reasonably  acceptable  to  Executive  that  no
Excise Tax will be imposed with respect to such Payment. Any

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good faith determinations of the accounting firm made hereunder shall be final, binding and conclusive upon the Company and Executive.

4.5.

Certain  Reductions  and  Offsets.   To  the  extent  that  any  federal,  state  or  local  laws,  including,  without  limitation,  the
Worker Adjustment and Retraining Notification Act or any other so-called “plant closing” laws, require the Company to give advance notice or make a
payment  of  any  kind  to  Executive  because  of  Executive’s  involuntary  termination  due  to  a  layoff,  reduction  in  force,  plant  or  facility  closing,  sale  of
business, change in control or any other similar event or reason, the benefits payable under this Agreement shall be correspondingly reduced. The benefits
provided  under  this  Agreement  are  intended  to  satisfy  any  and  all  statutory  obligations  that  may  arise  out  of  Executive’s  involuntary  termination  of
employment for the foregoing reasons, and the parties shall construe and enforce the terms of this Agreement accordingly.

4.6.

Mitigation.  Except as otherwise specifically provided herein, Executive shall not be required to mitigate damages or the
amount  of  any  payment  provided  under  this  Agreement  by  seeking  other  employment  or  otherwise,  nor  shall  the  amount  of  any  payment  or  benefit
provided  for  under  this  Agreement  be  reduced  by  any  compensation  earned  by  Executive  as  a  result  of  employment  by  another  employer  or  by  any
retirement  benefits  received  by  Executive  after  the  date  of  a  Covered  Termination  or  Change  in  Control  Termination  (except  as  expressly  provided  in
Sections 2.3 and 3.3 above).

4.7.

Indebtedness of Executive. If Executive is indebted to the Company on the effective date of a Covered Termination or
Change in Control Termination Date, the Company reserves the right to offset any Severance Benefits or Change in Control Severance Benefits under this
Agreement by the amount of such indebtedness, subject to the requirements of Section 409A of the Code and applicable law.

4.8.

Application of Section 409A.

a)

Separation from Service.  Notwithstanding any provision to the contrary in this Agreement, no amount deemed deferred
compensation  subject  to  Section  409A  of  the  Code  shall  be  payable  pursuant  to  Section  2  or  Section  3  unless  Executive’s  termination  of  employment
constitutes a “separation from service” with the Company within the meaning of Section 409A of the Code and the Department of Treasury Regulations
and  other  guidance  promulgated  thereunder  and,  except  as  provided  under  Section  4.8(b)  hereof,  any  such  amount  shall  not  be  paid,  or  in  the  case  of
installments,  commence  payment,  until  the  first  regularly-scheduled  payroll  date  occurring  on  or  after  the  sixtieth  (60th)  day  following  Executive’s
separation  from  service.  Any  installment  payments  that  would  have  been  made  to  Executive  during  the  sixty  (60)  day  period  immediately  following
Executive’s separation from service but for the preceding sentence shall be paid to Executive on the first regularly-scheduled payroll date occurring on or
after the sixtieth (60th) day after Executive’s separation from service and the remaining payments shall be made as provided in this Agreement.

b)

Specified Executive.  Notwithstanding any provision to the contrary in this Agreement, if Executive is deemed at the time
of  his  or  her  separation  from  service  to  be  a  “specified  employee”  for  purposes  of  Section  409A(a)(2)(B)(i)  of  the  Code,  to  the  extent  delayed
commencement of any portion of the benefits to which Executive is entitled under this Agreement is required in order to avoid a prohibited distribution
under Section 409A(a)(2)(B)(i) of the Code, such portion of Executive’s benefits shall not be provided to Executive prior to the earlier of (i) the expiration
of the six (6)-month period measured from the date of Executive’s “separation from service” with the Company (as such term is defined in the Treasury
Regulations  issued  under  Section  409A  of  the  Code)  or  (ii)  the  date  of  Executive’s  death.  Upon  the  first  business  day  following  the  expiration  of  the
applicable Code Section 409A(a)(2)(B)(i)

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period,  all  payments  deferred  pursuant  to  this  Section  4.8(b)  shall  be  paid  in  a  lump  sum  to  Executive,  and  any  remaining  payments  due  under  this
Agreement shall be paid as otherwise provided herein.

c)

Expense Reimbursements.    To  the  extent  that  any  reimbursement  payable  pursuant  to  this  Agreement  is  subject  to  the
provisions of Section 409A of the Code, any such reimbursement payable to Executive pursuant to this Agreement shall be paid to Executive no later than
December 31 of the year following the year in which the expense was incurred; the amount of expenses reimbursed in one year shall not affect the amount
eligible  for  reimbursement  in  any  subsequent  year;  and  Executive’s  right  to  reimbursement  under  this  Agreement  will  not  be  subject  to  liquidation  or
exchange for another benefit.

Installments.    For  purposes  of  Section  409A  of  the  Code  (including,  without  limitation,  for  purposes  of  Treasury
Regulation Section 1.409A-2(b)(2)(iii)), Executive’s right to receive any installment payments under this Agreement shall be treated as a right to receive a
series of separate payments and, accordingly, each such installment payment shall at all times be considered a separate and distinct payment.

d)

4.9.

Tax Withholding. All  payments  under  this  Agreement  shall  be  subject  to  applicable  withholding  for  federal,  state  and

local income and employment taxes.

4.10.

No Duplication of Severance Benefits. The Severance Benefits and Change in Control Severance Benefits provided in
Section  2  and  Section  3  are  mutually  exclusive  of  each  other,  and  in  no  event  shall  Executive  receive  any  Severance  Benefits  or  Change  in  Control
Severance Benefits pursuant to both Section 2 and Section 3.  

5.  TERMINATION WITH CAUSE OR BY VOLUNTARY RESIGNATION; OTHER RIGHTS AND BENEFITS

5.1.

Termination  for  Cause;  Resignation  Without  Good  Reason;  Death  or  Disability.    If,  at  any  time,  the  Company
terminates Executive’s employment with the Company for Cause, or upon a voluntary resignation by Executive that is not a Resignation for Good Reason,
or Executive’s employment terminates for any reason not entitling Executive to the Severance Benefits or Change in Control Severance Benefits, or if
Executive’s employment terminates as a result of Executive’s death or disability (other than a Permanent Disability in the case of a Covered Termination),
then  the  Company  shall  have  no  further  obligation  to  Executive  hereunder  except  for  the  payment  or  provision,  as  applicable,  of  (i)  the  portion  of  the
Annual Base Salary accrued through Executive’s last day of employment, (ii) all unreimbursed expenses (if any), subject to Sections 1.4 and 4.8(c), and
(iii) any unused vacation (if applicable) accrued through Executive’s last day of employment.  Under these circumstances, Executive will not be entitled to
any other form of compensation, including any Severance Benefits or Change in Control Severance Benefits, other than Executive’s rights to the vested
portion of Executive’s Option and any other rights to which Executive is entitled under the Company’s benefit programs.    

5.2.

Other  Rights  and  Benefits.  Nothing  in  this  Agreement  shall  prevent  or  limit  Executive’s  continuing  or  future
participation  in  any  benefit,  bonus,  incentive  or  other  plans,  programs,  policies  or  practices  provided  by  the  Company  and  for  which  Executive  may
otherwise qualify, nor shall anything herein limit or otherwise affect such rights as Executive may have under other agreements with the Company except
as  provided  in  Section  4  and  Section  5.1  above.  Except  as  otherwise  expressly  provided  herein,  amounts  that  are  vested  benefits  or  that  Executive  is
otherwise  entitled  to  receive  under  any  plan,  policy,  practice  or  program  of  the  Company  at  or  subsequent  to  the  date  of  a  Change  in  Control  shall  be
payable in accordance with such plan, policy, practice or program.

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6.  DEFINITIONS

For purposes of this Agreement, the following definitions shall apply:

6.1.“Board” means the Board of Directors of the Company, or the compensation committee thereof, as determinations or responsibilities may

be delegated by the Board to the compensation committee.

6.2.

“Cause”  shall  mean  a  determination  by  the  Company  based  upon  reasonably  available  information  of  Executive’s:  (i)
unauthorized use or disclosure of the Company’s confidential information or trade secrets; (ii) material breach of any agreement to which the Executive
and the Company are a party; (iii) material failure to comply with the Company’s written policies or rules; (iv) conviction of, or plea of “guilty” or “no
contest”  to,  a  felony  under  the  laws  of  the  United  States  or  any  State;  (v)  negligence  or  willful  misconduct  relating  to  Executive’s  performance  of  her
duties on behalf of the Company; (vi) continuing failure to perform material and lawful assigned duties after receiving thirty (30) days’ written notification
of the failure from the Company if such breach is not cured (if curable) during that thirty (30) day period; (vii) failure to cooperate in good faith with a
governmental  or  internal  investigation  of  the  Company  or  its  directors,  officers  or  employees,  if  the  Company  has  requested  Executive’s  cooperation
without prejudice or personal liability to Executive; (viii) violation of employee or ethical guidelines including, without limitation, violations of business
practices and ethics commonly in place in similar companies in the United States; or (ix) violation of the Company code of conduct and/or any contractual
code of conduct to which the Company is obligated.

6.3.
more of the following events:

“Change  in  Control”  means  the  occurrence,  in  a  single  transaction  or  in  a  series  of  related  transactions,  of  any  one  or

a)

Any natural person, entity or group within the meaning of Section 13(d) or 14(d) of the Securities Exchange Act of 1934, as
amended (“Exchange Act Person”), becomes the owner, directly or indirectly, of securities of the Company representing more than fifty percent (50%) of
the  combined  voting  power  of  the  Company’s  then  outstanding  securities  other  than  by  virtue  of  a  merger,  consolidation  or  similar  transaction.
Notwithstanding the foregoing, a Change in Control shall not be deemed to occur (i) on account of the acquisition of securities of the Company by any
institutional investor, any affiliate thereof or any other Exchange Act Person that acquires the Company’s securities in a transaction or series of related
transactions that are primarily a private financing transaction for the Company or (ii) solely because the level of ownership held by any Exchange Act
Person  (the  “Subject  Person”)  exceeds  the  designated  percentage  threshold  of  the  outstanding  voting  securities  as  a  result  of  a  repurchase  or  other
acquisition of voting securities by the Company reducing the number of shares outstanding, provided that if a Change in Control would occur (but for the
operation of this sentence) as a result of the acquisition of voting securities by the Company, and after such share acquisition, the Subject Person becomes
the  owner  of  any  additional  voting  securities  that,  assuming  the  repurchase  or  other  acquisition  had  not  occurred,  increases  the  percentage  of  the  then
outstanding voting securities owned by the Subject Person over the designated percentage threshold, then a Change in Control shall be deemed to occur;

b)

There  is  consummated  a  merger,  consolidation  or  similar  transaction  involving,  directly  or  indirectly,  the  Company  if,
immediately after the consummation of such merger, consolidation or similar transaction, the stockholders of the Company immediately prior thereto do
not  own,  directly  or  indirectly,  either  (i)  outstanding  voting  securities  representing  more  than  fifty  percent  (50%)  of  the  combined  outstanding  voting
power of the surviving entity in such merger, consolidation or similar transaction or (ii) more than fifty percent (50%) of the combined outstanding voting
power of the parent of the surviving entity in such merger, consolidation or similar transaction; or

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c)

There is consummated a sale, lease, license or other disposition of all or substantially all of the consolidated assets of the
Company and its subsidiaries, other than a sale, lease, license or other disposition of all or substantially all of the consolidated assets of the Company and
its subsidiaries to an entity, more than fifty percent (50%) of the combined voting power of the voting securities of which are owned by stockholders of the
Company in substantially the same proportion as their ownership of the Company immediately prior to such sale, lease, license or other disposition.

The term Change in Control shall not include a sale of assets, merger or other transaction effected exclusively for the purpose of changing the
domicile of the Company. Notwithstanding the foregoing or any other provision of this Agreement, the definition of Change in Control (or any analogous
term) in an individual written agreement between the Company or any affiliate and the participant shall supersede the foregoing definition with respect to
stock awards subject to such agreement (it being understood, however, that if no definition of Change in Control or any analogous term is set forth in such
an individual written agreement, the foregoing definition shall apply).

6.4.

6.5.

“Change in Control Benefits Period” means the period of twelve (12) months commencing on the Termination Date.

“Change in Control Severance Period” means the period of twelve (12) months commencing on the Termination Date.

6.6.

  “Change  in  Control  Termination”  means  an  “Involuntary  Termination  Without  Cause”  or  “Resignation  for  Good
Reason,” either of which occurs within three (3) months prior to or upon or within twelve (12) months following the closing of a Change in Control or
Dissolution  Event,  provided  that  any  such  termination  is  a  “separation  from  service”  within  the  meaning  of  Treasury  Regulation  Section  1.409A-
1(h).  Death and disability shall not be deemed Change in Control Terminations.

6.7.

6.8.

6.9.

“COBRA” means the Consolidated Omnibus Budget Reconciliation Act of 1985, as amended.

“Code” means the Internal Revenue Code of 1986, as amended.

“Company”  means  Ovid  Therapeutics  Inc.  or,  following  a  Change  in  Control,  the  surviving  entity  resulting  from  such

transaction, or any subsequent surviving entity resulting from any subsequent Change in Control.

6.10.

“Confidentiality Agreement”  means  Senior  Executive  Confidential  Information  and  Invention  Assignment  Agreement

with the Company, (or any successor agreement thereto).

6.11.

  “Covered  Termination”  means  an  “Involuntary  Termination  Without  Cause”  or  “Resignation  for  Good  Reason,”
provided that any such termination is a “separation from service” within the meaning of Treasury Regulation Section 1.409A-1(h). Death and disability,
other  than  a  Permanent  Disability,  shall  not  be  deemed  Covered  Terminations.    If  an  Involuntary  Termination  Without  Cause  or  Resignation  for  Good
Reason qualifies as a Change in Control Termination, it shall not constitute a Covered Termination.  

6.12.

6.13.

Date.

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“Covered Termination Benefits Period” means the period of twelve (12) months commencing on the Termination Date.

“Covered  Termination  Severance  Period”  means  the  period  of  twelve  (12)  months  commencing  on  the  Termination

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6.14.

“Dissolution  Event”  means  the  stockholders  of  the  Company  approve  or  the  Board  approves  a  plan  of  complete

dissolution or liquidation of the Company, or a complete dissolution or liquidation of the Company shall otherwise occur.

6.15.

“Involuntary Termination Without Cause” means Executive’s dismissal or discharge by the Company for reasons other
than  Cause  and  other  than  as  a  result  of  death  or  disability;  provided, however,  that  for  purposes  of  a  Covered  Termination,  Involuntary  Termination
Without Cause shall include Executive’s dismissal or discharge by the Company for reasons of Permanent Disability.

6.16.

  “Monthly  Base  Salary”  means  1/12th  of  Executive’s  Annual  Base  Salary  (excluding  incentive  pay,  premium  pay,
commissions,  overtime,  bonuses  and  other  forms  of  variable  compensation)  as  in  effect  on  the  date  of  a  Covered  Termination  or  Change  in  Control
Termination.

6.17.

“Permanent Disability” means total and permanent disability as defined in Code Section 22(e)(3).

6.18.

“Resignation for Good Reason” means Executive’s resignation from all employee positions Executive then holds with
the  Company  within  ninety  (90)  days  following  any  of  the  following  events  taken  without  Executive’s  consent,  provided  Executive  has  given  the
Company written notice of such event within thirty (30) days after the first occurrence of such event and the Company has not cured such event within
thirty (30) days thereafter:

comparable executives of the Company;

a)

A material decrease in Executive’s Annual Base Salary, other than in connection with a decrease in compensation for all

b)

c)

A relocation of Executive’s principal place of work outside of a fifty (50) mile radius of its current location; or

The Company’s material breach of this Agreement.

6.19.

“Termination Date” means the effective date of a Change in Control Termination, a Covered Termination, a termination

for Cause or any other circumstance under which the employment relationship between Executive and the Company terminates, as applicable.

6.20.

“Division” shall mean only that part, unit or therapeutic category of a larger entity that is competitive with the Company,

but not an entire company itself, if other divisions, units or therapeutic categories of such larger company are not competitive with the Company.

6.21.

"Client"  shall  mean  (A)  anyone  who  is  a  client  of  the  Company  as  of,  or  at  any  time  during  the  one-year  period
immediately preceding, the termination of Executive’s employment, but only if Executive had a direct relationship with, supervisory responsibility for or
otherwise were involved with such client during Executive’s employment with the Company; and (B) any prospective client to whom the Company made
a  new  business  presentation  (or  similar  offering  of  services)  at  any  time  during  the  one-year  period  immediately  preceding,  or  six-month  period
immediately following, Executive’s employment termination (but only if initial discussions between the Company and such prospective client relating to
the rendering of services occurred prior to the termination date, and only if Executive participated in or supervised such presentation and/or its preparation
or the discussions leading up to it).

6.22.

“Solicit”  shall  mean:  (A)  active  solicitation  of  any  Client  or  Company  employee,  board  member,  advisor,  consultant,
collaborator,  investigator  or  agents;  (B)  the  provision  of  information  regarding  any  Client  or  Company  employee,  board  member,  advisor,  consultant,
collaborator, investigator or agents to any third party where such information could be useful to such third party in attempting to obtain business from such
Client or attempting to hire any such Company employee; (C) participation in any meetings, discussions, or other communications with any third party
regarding any Client or Company employee, board member, advisor, consultant, collaborator, investigator

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or  agents  where  the  purpose  or  effect  of  such  meeting,  discussion  or  communication  is  to  obtain  business  from  such  Client  or  employ  such  Company
employee;  and  (D)  any  other  passive  use  of  information  about  any  Client  or  Company  employee,  board  member,  advisor,  consultant,  collaborator,
investigator or agents which has the purpose or effect of assisting a third party or causing harm to the business of the Company.

7.  GENERAL PROVISIONS

7.1.

Employment  Status.    This  Agreement  does  not  constitute  a  contract  of  employment  or  impose  upon  Executive  any
obligation  to  remain  as  an  employee,  or  impose  on  the  Company  any  obligation  (i)  to  retain  Executive  as  an  employee,  (ii)  to  change  the  status  of
Executive as an at-will employee or (iii) to change the Company’s policies regarding termination of employment.

7.2.

Notices. Any notices provided hereunder must be in writing, and such notices or any other written communication shall be
deemed effective upon the earlier of personal delivery (including personal delivery by facsimile or email transmission (to a facsimile number or email
address designated in advance by the receiving party)) or the third day after mailing by first class mail, to the Company at its primary office location and to
Executive at Executive’s address as listed in the Company’s payroll records. Any payments made by the Company to Executive under the terms of this
Agreement shall be delivered to Executive either in person or at the address as listed in the Company’s payroll records.

7.3.

Severability. Whenever possible, each provision of this Agreement will be interpreted in such manner as to be effective
and  valid  under  applicable  law,  but  if  any  provision  of  this  Agreement  is  determined  to  be  invalid,  illegal  or  unenforceable  in  any  respect  under  any
applicable law or rule in any jurisdiction, such invalidity, illegality or unenforceability will not affect any other provision or any other jurisdiction, and the
provision in question shall be modified so as to be rendered enforceable in a manner consistent with the intent of the parties insofar as possible under
applicable law.

7.4.

Waiver. If either party should waive any breach of any provisions of this Agreement, he, she or it shall not thereby be

deemed to have waived any preceding or succeeding breach of the same or any other provision of this Agreement.

7.5.

Complete  Agreement.  This  Agreement,  together  with  Exhibits  A  thru  D,  the  Confidentiality  Agreement  and  the
Indemnification Agreement, forms the complete and exclusive statement of Executive’s employment agreement with the Company, and supersedes and
replaces any other agreements or promises made to Executive by anyone, whether oral or written (including but not limited to the Prior Agreement).

7.6.

Amendment or Termination of Agreement; Continuation of Agreement. Except for those changes expressly reserved
to the Company’s or the Board’s discretion in this Agreement, this Agreement may be changed or terminated only upon the mutual written consent of the
Company and Executive. The written consent of the Company to a change or termination of this Agreement must be signed by an executive officer of the
Company (other than Executive) after such change or termination has been approved by the Board. Unless so terminated, this Agreement shall continue in
effect for as long as Executive continues to be employed by the Company or by any surviving entity following any Change in Control. For the avoidance
of any doubt, if, following a Change in Control, Executive continues to be employed by the surviving entity without a Change in Control Termination and
the surviving entity then

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undergoes  a  Change  in  Control,  following  which  Executive  is  terminated  by  the  subsequent  surviving  entity  in  a  Change  in  Control  Termination,
Executive shall receive the benefits described in Section 3 hereof.  

7.7.

Counterparts. This Agreement may be executed in separate counterparts, any one of which need not contain signatures of
more than one party, but all of which taken together will constitute one and the same Agreement.  Facsimile and electronic image copies of signatures shall
be equivalent to original signatures.  

7.8.

Headings. The headings of the Sections hereof are inserted for convenience only and shall not be deemed to constitute a

part hereof nor to affect the meaning thereof.

7.9.

Successors and Assigns. This Agreement is intended to bind and inure to the benefit of and be enforceable by Executive,
and  the  Company,  and  any  surviving  entity  resulting  from  a  Change  in  Control  and  upon  any  other  person  who  is  a  successor  by  merger,  acquisition,
consolidation  or  otherwise  to  the  business  formerly  carried  on  by  the  Company,  and  their  respective  successors,  assigns,  heirs,  executors  and
administrators, without regard to whether or not such person actively assumes any rights or duties hereunder; provided, however, that Executive may not
assign any duties hereunder and may not assign any rights hereunder without the written consent of the Company, which consent shall not be withheld
unreasonably.

7.10.

Choice of Law. This Agreement shall be construed and enforced in accordance with the laws of the State of New York

without regard to conflicts of law principles. 

7.11.

Arbitration.    To  ensure  the  rapid  and  economical  resolution  of  any  disputes  that  may  arise  under  or  relate  to  this
Agreement or Executive’s employment relationship, Executive and the Company agree that, unless otherwise prohibited by applicable law, any and all
disputes,  claims,  or  causes  of  action,  in  law  or  equity,  arising  from  or  relating  to  the  performance,  enforcement,  execution,  or  interpretation  of  this
Agreement, Executive’s employment with the Company, or the termination of Executive’s employment (collectively, “Claims”), shall be resolved by final,
binding, and (to the extent permitted by law) confidential arbitration before a single arbitrator in New York, New York.  Executive and the Company agree
that  they  shall  resolve  all  such  Claims  in  accordance  with  the  provisions  of  Section  12  of  the  Confidential  Information  and  Invention  Assignment
Agreement attached hereto as Exhibit A.    

7.12.

Construction of Agreement. In the event of a conflict between the text of this Agreement and any summary, description

or other information regarding this Agreement, the text of this Agreement shall control.

7.13.

Circular  230  Disclaimer.  THE  FOLLOWING  DISCLAIMER  IS  PROVIDED  IN  ACCORDANCE  WITH  THE
INTERNAL  REVENUE  SERVICE’S  CIRCULAR  230  (21  C.F.R.  PART  10).  ANY  TAX  ADVICE  CONTAINED  IN  THIS  AGREEMENT  IS
INTENDED TO BE PRELIMINARY, FOR DISCUSSION PURPOSES ONLY AND NOT FINAL. ANY SUCH ADVICE IS NOT INTENDED
TO BE USED FOR MARKETING, PROMOTING OR RECOMMENDING ANY TRANSACTION OR FOR THE USE OF ANY PERSON IN
CONNECTION WITH THE PREPARATION OF ANY TAX RETURN. ACCORDINGLY, THIS ADVICE IS NOT INTENDED OR WRITTEN
TO  BE  USED,  AND  IT  CANNOT  BE  USED,  BY  ANY  PERSON  FOR  THE  PURPOSE  OF  AVOIDING  TAX  PENALTIES  THAT  MAY  BE
IMPOSED ON SUCH PERSON.

148402431 v2

Perone - D-14

 
 
 
 
 
 
REVIEWED, UNDERSTOOD AND ACCEPTED:

OVID THERAPEUTICS INC.

EXECUTIVE

By:
Name:

Suzanne K. Wakamoto

Title:

SVP, Human Resources

148402431 v2

By: 
Name: 

Title:

Thomas Perone

General Counsel, Corporate Secretary and Chief Compliance
Officer

Perone - D-15

 
 
 
 
 
 
 
 
 
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

Exhibit 10.25

COLLABORATION AND LICENSE AGREEMENT

THIS COLLABORATION AND LICENSE AGREEMENT (the “Agreement”) is entered into as of July 8, 2020 (the “Effective Date”), by and
between  OVID  THERAPEUTICS  INC.,  a  Delaware  company  having  an  address  at  1460  Broadway,  Suite  15021  New  York,  NY  10036,  USA
(“Ovid”) and ANGELINI PHARMA RARE DISEASES AG, a Swiss company under direction and control of Angelini Pharma S.p.A. and having an
address at Consulting GmbH Sumpfstrasse 26 6312 Steinhausen, Zurich, Switzerland (“Licensee”).  Ovid and Licensee may be referred to
herein individually as a “Party” or collectively as the “Parties”.  

RECITALS

WHEREAS,  Ovid,  a  biopharmaceutical  company,  owns  or  controls  certain  patents,  know-how,  and  other  intellectual  property
relating  to  its  proprietary  compound  known  as  OV101,  a  selective  agonist  of  the  GABAA  receptor,  including  certain  intellectual  property
rights in-licensed from H. Lundbeck A/S, which Ovid has been developing for the treatment of Angelman syndrome and Fragile X syndrome
and potentially other Rare Diseases indications;

WHEREAS,  Licensee  is  a  subsidiary,  100%  under  direction  and  control  of  Angelini  Pharma  S.p.A.,  an  Italian  pharmaceutical

company, which is experienced in the development and commercialization of pharmaceutical products; and

WHEREAS, Licensee and Ovid desire to form a collaboration for the continued development and commercialization of OV101, with

the status of Orphan Medicine and with Final Label 1a, 1b and/or 2, all on the terms and conditions set forth below.

NOW, THEREFORE, in consideration of the foregoing premises and the mutual covenants contained herein, and for other good and

valuable consideration, the receipt and sufficiency of which are hereby acknowledged, Ovid and Licensee hereby agree as follows:

AGREEMENT

1.

DEFINITIONS

1.1

1.2

“Additional Development Activities” has the meaning set forth in Section 4.3(a).

“Additional  Indications”  means  any  Rare  Diseases  Indication  other  than  the  Initial  Indication  and  the  Second

Indication that has been submitted to and approved by the CGB.

1.3

“Additional  Pivotal  Trial”  means  the  additional  Phase  3  Clinical  Trial  of  the  Product  for  the  Initial  Indication,  if
required by the EMA or by Licensee at its own discretion, for the purpose of seeking or maintaining MAA Approval of the Product for the
Initial Indication in the Licensee Territory, as described in Exhibit H.

1.4

“Affiliate” means, with respect to any party, any entity that, directly or indirectly through one or more intermediaries,
controls, is controlled by, or is under common control with such party, but for only so long as such control exists.  As used in this Section 1.4,
“control” means (a) to possess, directly or indirectly, the power to direct the management or policies of an entity, whether through ownership
of voting securities, by contract relating to voting rights or corporate

1

 
 
governance; or (b) direct or indirect beneficial ownership of more than fifty percent (50%) (or such lesser percentage which is the maximum
allowed to be owned by a foreign corporation in a particular jurisdiction) of the voting share capital or other equity interest in such entity.

1.5

“Allocated Quantity of Compound” means [***] of the Compound in Ovid’s control as of the Effective Date, which
Ovid has agreed, under the Supply Agreement, to allocate exclusively for the purpose of fulfilling Licensee’s or Licensee Affiliate’s Purchase
Orders under the Supply Agreement.

1.6

1.7

1.8

“Allowable Increases” has the meaning set forth in Section 4.5(b).

“Amended Development Budget” has the meaning set forth in Section 4.2.

“Amended Development Plan” has the meaning set forth in Section 4.2.

1.9

“Angelini  Commercially  Reasonable  Efforts”  means,  with  respect  to  Licensee  and  its  obligations  under  this
Agreement,  commercially  reasonable  efforts  and  resources  as  commonly  used  by  a  similar  size  pharmaceutical  company  to  Develop  and
Commercialize a product controlled by Licensee or to which it has exclusive rights, which product is at similar stage in its development or
product life and is of similar market potential taking into account efficacy, safety, approved and/or anticipated labelling, the competitiveness
of  alternative  products  sold  by  Third  Parties  in  the  marketplace,  the  patent  and  other  proprietary  position  of  the  product,  likelihood  of
regulatory  approval  given  the  regulatory  structure  involved,  the  profitability  of  the  product,  [***]  and  other  relevant  factors,  including
technical, legal, scientific and/or medical factors. Commercially Reasonable Efforts shall be determined on a country-by-country basis and
indication-by-indication  basis  for  a  particular  Product,  and  it  is  anticipated  that  the  level  of  effort  will  change  over  the  time,  reflecting
changes in the status of the Product and the country(s) involved. [***].

1.10

“Applicable Laws” means the applicable provisions (including Data Protection Legislation) of any and all national,
supranational,  regional,  state  and  local  laws,  treaties,  statutes,  rules,  regulations,  administrative  codes,  guidance,  ordinances,  judgments,
decrees,  directives,  injunctions,  orders,  permits  (including  MAAs)  of  or  from  any  court,  Regulatory  Authority,  or  governmental  agency  or
authority having jurisdiction over or related to the subject item.

1.11

1.12

“Auditor” has the meaning set forth in Section 9.4.

“Calendar  Quarter”  means  each  respective  period  of  three  (3)  consecutive  months  ending  on  March  31,  June  30,

September 30, and December 31.

1.13

“Calendar Year” means each respective period of twelve (12) consecutive months ending on December 31.

1.14

“cGCP”  means  the  current  good  clinical  practice  standards  as  set  out  in  (a)  ICH  Harmonized  Guidance  on  current
Good  Clinical  Practice  (CPMP/ICH/135/95),  (b)  U.S.  21  C.F.R.  Parts  50,  54,  56,  58,  210,  211  and  312,  and  (c)  the  equivalent  law  or
regulation in any other applicable jurisdiction in the Territory, each as may be amended from time to time.

2
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
1.15

“cGLP” means current good laboratory practice standards promulgated or endorsed by the FDA, as defined in U.S. 21

C.F.R. Part 58 (or such other comparable regulatory standards in jurisdictions outside the U.S.), as may be amended from time to time.

1.16

“cGMP” means the current standards for systems to assure the proper design, monitoring, and control of processes and
facilities to be used for the manufacture, processing, packing, or holding of a drug as specified by applicable laws of the relevant countries at
the  time  of  manufacturing  conducted  in  accordance  with  this  Agreement,  defined  under  (a)  U.S.  21  C.F.R.  Parts  210  and  211  and  (b)  the
equivalent law or regulation in any other applicable jurisdiction in the Territory, each as may be amended from time to time.

1.17

1.18

“Claim” has the meaning set forth in Section 12.3.

“Clawback”  means  post  sales  clawback  policies  applied  to  manufacturers,  requiring  them  to  pass  a  part  of  their

revenues in respect of a product to a national health service or other Governmental Authority.

1.19

“Clinical Trial” or “Clinical Trials” means Phase 1 Clinical Trial, Phase 2 Clinical Trial, Phase 3 Clinical Trial, or

Phase 4 Clinical Trial, as the context dictates.

1.20

“Collaboration Governance Board” or “CGB” has the meaning set forth in Section 3.1.

1.21

“Combination  Product”  means  any  pharmaceutical  product  containing  the  Compound  as  an  active  pharmaceutical
ingredient  in  combination  with  one  or  more  other  therapeutically  active  ingredients,  in  any  and  all  forms,  presentations,  dosages,  and
formulations.

1.22

“Commercialization” means the conduct of all activities undertaken before and after Regulatory Approval relating to
the  promotion,  sales,  marketing,  medical  and  patient  support  and  services,  and  distribution  (including  importing,  exporting,  transporting,
customs clearance, warehousing, invoicing, handling, and delivering Products to customers) of Products in the Field, including sales force
efforts,  detailing,  advertising,  market  research,  market  access  (including  price  and  reimbursement  activities),  medical  education  and
information services, publication, scientific and medical affairs, advisory and collaborative activities with opinion leaders and professional
societies  including  symposia,  marketing,  sales  force  training,  and  sales  (including  receiving,  accepting  and  filling  Product  orders)  and
distribution.  “Commercialize” and “Commercializing” have correlative meanings.

1.23

1.24

1.25

medicines.

“Commercialization Plan” has the meaning set forth in Section 6.2.

“Committee” means the CGB, JPT, or any other subcommittee established by the CGB, as applicable.

“Committee for Medicinal Products for Human Use (CHMP)” means the EMA committee responsible for human

1.26

“Competing Acquirer” means a Third Party that, as of the closing date of the applicable transaction, is engaged in

[***] of products, other than Products, for [***].

3
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
1.27

“Competing  Product”  means  any  product  or  compound,  other  than  the  Compound  and  Products  and  the  Current

Licensee Pipeline Products, (a) [***], or (b) [***].

1.28

“Compound”  means  the  δ-selective  extrasynaptic  GABAA  receptor  agonist  known  internally  by  Ovid  as  OV101,

having the chemical structure set forth in Exhibit A.

1.29

1.30

“Compound Invention” has the meaning set forth in Section 10.1(b)(i).

“Compounding” or “Compounding Activities” means [***].

1.31
dated as of July 8, 2019.

“Confidentiality  Agreement”  means  that  certain  Confidential  Disclosure  Agreement  between  Ovid  and  Licensee

1.32

“Confidential  Information”  means  all  Know-How  and  other  proprietary  scientific,  marketing,  financial,  or
commercial information or data that is generated by or on behalf of a Party or its Affiliates or which one Party or any of its Affiliates has
supplied  or  otherwise  made  available  to  the  other  Party  or  its  Affiliates,  whether  made  available  orally,  in  writing,  or  in  electronic  form,
including information comprising or relating to concepts, discoveries, inventions, data, designs, or formulae in relation to this Agreement;
provided  that  all  Ovid  Technology  will  be  deemed  Ovid’s  Confidential  Information,  all  Licensee  Technology  will  be  deemed  Licensee’s
Confidential Information, and all Joint Inventions and Joint Patents will be deemed both Parties’ Confidential Information.

1.33

“Control” or “Controlled” means, with respect to any Know-How, Patents, or other intellectual property rights, the
legal authority or right (whether by ownership, license, or otherwise, but without taking into account any rights granted by one Party to the
other Party pursuant to this Agreement) of a Party to grant access, a license, or a sublicense of or under such Know-How, Patents, or other
intellectual  property  rights  to  another  Party,  or  to  otherwise  disclose  proprietary  or  trade  secret  information  to  such  other  Party,  without
breaching the terms of any agreement with a Third Party, or misappropriating the proprietary or trade secret information of a Third Party.

1.34

“Cost of Goods”  means,  with  respect  to  the  Drug  Product,  the  fully  burdened  cost  to  manufacture  and  supply  such
Drug Product, which means: (a) in the case of products and services acquired from Third Parties, [***]; and (b) in the case of manufacturing
services performed by a Party or its Affiliates, including manufacturing services to support products and services acquired from Third Parties
as contemplated in subsection (a), [***].

1.35

“Current Licensee Pipeline Products” means, in each case as of the Effective Date, Licensee’s pipeline for products

related to (a) [***], (b) [***], and (c) [***], in each case as better defined in Exhibit I.

1.36

“Data” means any and all scientific, technical, test, marketing, or sales data pertaining to any Product that is generated
by or on behalf of Ovid, Licensee, and their respective Affiliates and (sub)licensees, including research data, clinical pharmacology data, pre-
clinical data, clinical data, clinical study reports, or submissions made in association with an IND or MAA with respect to any Product.  

4
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
1.37

“Data Protection Legislation” means all applicable legislation relating to the protection and processing of personal
data,  data  privacy  and  the  privacy  of  electronic  communications  in  any  relevant  jurisdiction,  including  the  General  Data  Protection
Regulation ((EU) 2016/679), and any national implementing laws, regulations and secondary legislation, as amended or updated from time to
time.

1.38

toxicology,
“Development”  means  all  non-clinical  and  clinical  drug  development  activities, 
pharmacological,  and  other  non-clinical  efforts,  statistical  analysis,  the  performance  of  Clinical  Trials,  including  the  Manufacturing  of  the
Products for use in the Clinical Trials, Manufacturing Development or other activities reasonably necessary in order to obtain or maintain
Regulatory  Approval  of  Products  in  the  Field  in  the  Territory,  as  detailed  in  a  Development  Plan  for  the  Products.  “Development”  shall
exclude all Commercialization activities. When used as a verb, “Develop” means to engage in Development activities.

including 

1.39

“Development  Budget”  means  the  initial  reasonably  detailed  budget  estimated  by  the  Parties  for  all  Development

activities set forth in the Development Plan.

1.40

“Development Costs” means the costs incurred by a Party or for its account or by the Parties jointly, during the Term
and pursuant to this Agreement, that are specifically directed (or reasonably allocable) to the Development of a Product.  The Development
Costs  shall  include  amounts  that  a  Party  pays  to  Third  Parties  involved  in  the  Development  of  a  Product  (at  cost),  and  all  internal  costs
(calculated  on  an  FTE  basis  at  the  then-current  FTE  Rate)  and  out-of-pocket  costs  incurred  by  or  on  account  of  a  Party  in  performing
Development in accordance with the Development Plan.  For clarity, [***].

1.41

1.42

1.43

“Development Plan” means the initial plan of Development activities for the Product set forth in Exhibit C.

“Drug Product” means the Compound, filled and finished into unit doses, but not packaged or labelled.

“Elara Trial” means the open-label extension study for patients with Angelman Syndrome who have previously been

enrolled in a Clinical Trial of the Product (including the Neptune Trial) as of the Effective Date, as further described in Exhibit J.  [***].

1.44

“EMA” means the European Medicines Agency, and any successor agency or authority having substantially the same

function.

1.45

“Executive Officers” means the [***] of Ovid and the [***] of Licensee.

1.46

“Export  Control  Laws”  means  all  applicable  U.S.  laws  and  regulations  relating  to  (a)  sanctions  and  embargoes
imposed  by  the  Office  of  Foreign  Assets  Control  of  the  U.S.  Department  of  Treasury  or  (b)  the  export  or  re-export  of  commodities,
technologies, or services, including the Export Administration Act of 1979, 24 U.S.C. §§ 2401-2420, the International Emergency Economic
Powers Act, 50 U.S.C. §§ 1701-1706, the Trading with the Enemy Act, 50 U.S.C. §§ 1 et. seq., the Arms Export Control Act, 22 U.S.C. §§
2778 and 2779, and the

5
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
International Boycott Provisions of Section 999 of the U.S. Internal Revenue Code of 1986, in each case, as amended.

1.47

“Extended  Commercialization  Term”  means  the  period  commencing  on  the  expiration  of  the  Royalty  Term  and
continuing for so long as Ovid continues to supply to Licensee or Licensee Affiliate the Product under the terms of the Lundbeck License
Agreement.

1.48

“FCPA” means the U.S. Foreign Corrupt Practices Act (15 U.S.C. Section 78dd-1, et. seq.), as amended.

1.49
same function.

“FDA” means the U.S. Food and Drug Administration, and any successor agency or authority having substantially the

1.50

“Field” means the treatment of (a) the Initial Indication, (b) the Second Indication (subject to Section 4.2(e)) and (c)
any  Additional  Indication(s)  for  which  the  Parties  agree  to  incorporate  Additional  Development  Activities  into  the  Development  Plan  and
Development Budget in accordance with Section 4.3.

1.51

“Final Label” refers to the information regarding an approved Indication and population target that is included with a

prescription drug as approved by an applicable Regulatory Authority.

1.52

1.53

1.54

years of age or more.

“Final Label 1a” means the Final Label for a population from two (2) years of age up to twelve (12) years of age.

“Final Label 1b” means the Final Label for a population from four (4) years of age up to twelve (12) years of age.

“Final Label 2” means the Final Label for the population from twelve (12) years of age up to, at least seventeen (17)

1.55

“First Commercial Sale” means, on a Product-by-Product and country-by-country basis, the first sale of such Product
in such country by Licensee or its Affiliates or Sublicensees to a Third Party after Regulatory Approval for such Product has been obtained in
such country.  

1.56

“FTE” means the equivalent of a full-time individual’s work for a twelve (12) month period, consisting of a total of
[***] hours per year of dedicated effort.  Any person who devotes more or less than [***] hours per year on the applicable activities shall be
treated as an FTE on a pro-rata basis, based upon the actual number of hours worked by such person on such activities, divided by [***].  For
clarity, the hours spent by temporary workers and contractors on applicable activities may be treated as FTE on a pro-rata basis.

1.57

“FTE Rate” means an initial rate of (a) with respect to Ovid’s personnel, [***] per FTE per year and (b) with respect
to Licensee’s personnel, [***] per FTE per year, which rates shall apply through [***].  Thereafter, the FTE Rate shall be changed annually
on  a  Calendar  Year  basis  to  reflect  any  year-to-year  percentage  increase  or  decrease  (as  the  case  may  be)  (i)  with  respect  to  Ovid,  in  the
Consumer Price Index for All Urban Consumers for the U.S., as published by the U.S. Department of Labor, Bureau of Labor Statistics, and
(ii) with respect to Licensee, in

6
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
the Italy Consumer Price Index as  published  by  the  Italian  National  Statistical  Institute  (both  changes  based  on  the  change  from  the  most
recent applicable index available as of the Effective Date to the most recent applicable index available as of the date of the calculation of such
revised FTE Rate).

1.58

“Generic  Product”  means,  (a)  any  pharmaceutical  product  which  has  received  Regulatory  Approval  [***]  of  the
Product;  and/or  (b)  any  other  pharmaceutical  product,  approved  under  an  Abbreviated  New  Drug  Application,  or  ANDA,  in  the  United
States, under Section 505(b)(2) of the Food Drug and Cosmetic Act, or similar regulatory pathways outside of the U.S., in any case, with the
Product as the reference product.

1.59

“Generic  Product  Competition”  with  respect  to  a  Product,  on  a  country-by-country  basis,  Generic  Product
Competition shall exist if [***] there are one or more Generic Products sold [***] in such country and the sales of such Generic Product(s)
account for [***] or more of the sales revenue of the Product and its Generic Product(s) in the given country during such [***] as determined
by reference to applicable sales data obtained from IMS Health, Verispan, or from such other reputable source for such sales data as may be
used  and  relied  upon  by  the  Parties  from  time  to  time,  provided  however  if  sale  of  such  Generic  Product(s)  [***],  Generic  Product
Competition shall no longer exist.

1.60

  “Governmental  Authority”  means  any  national,  international,  federal,  state,  provincial,  or  local  government,  or
political  subdivision  thereof,  or  any  multinational  organization,  or  any  authority,  agency,  or  commission  entitled  to  exercise  any
administrative, executive, judicial, legislative, police, regulatory, or taxing authority or power, or any court or tribunal (or any department,
bureau or division thereof, or any governmental arbitrator or arbitral body).

1.61

“ICH”  means  the  International  Conference  on  Harmonization  (of  Technical  Requirements  for  Registration  of

Pharmaceuticals for Human Use).

1.62

“IND”  means  an  application  filed  with  a  Regulatory  Authority  for  authorization  to  commence  Clinical  Trials,
including  (a)  an  Investigational  New  Drug  Application  or  any  successor  application  or  procedure  filed  with  the  FDA,  (b)  a  Clinical  Trial
Application or any successor application or procedure filed with the EMA, (c) any equivalent of the applications in (a) and (b) in countries or
regulatory jurisdictions outside the U.S. and EU, and (d) all supplements, amendments, variations, extensions, and renewals thereof that may
be filed with respect to the foregoing.

1.63

1.64

1.65

1.66

“Indemnitee” has the meaning set forth in Section 12.3.

“Indemnitor” has the meaning set forth in Section 12.3.

“Independent Development Activities” has the meaning set forth in Section 4.3(d).

“Independent Development Costs” has the meaning set forth in Section 8.2(b).

7
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
1.67

“Indication” means a separate and distinct disease, disorder, illness, or health condition and all of its associated signs,
symptoms, stages, or progression (including precursor conditions), in each case for which a separate MAA may be filed.  Subpopulations or
patients with a primary disease or condition, however stratified (including stratification by stages or progression, particular combinations of
symptoms  associated  with  the  primary  disease  or  condition,  prior  treatment  courses,  response  to  prior  treatment,  family  history,  clinical
history, phenotype, or other stratification) shall not be deemed to be separate “Indications” for the purposes of this Agreement.

1.68

“Initial Indication” means Angelman syndrome (AS).

1.69

“International  Transparency  Reporting  Requirements  for  Europe”  means  EFPIA  consolidated  Code  for
Pharmaceutical Companies to report transfers of value related to HCPs: donations and grants, contribution to costs related to events, fees for
service and consultancy, research and development.

1.70

“Inventions” means all inventions, whether or not patentable, discovered, made, conceived, or reduced to practice in

the course of activities contemplated by this Agreement.

1.71

1.72

1.73

1.74

“JPT” has the meaning set forth in Section 3.2.

“Joint Development Activities” has the meaning set forth in Section 4.2(d).

“Joint Inventions” has the meaning set forth in Section 10.1(b)(ii).

“Joint Patents” has the meaning set forth in Section 10.1(b)(ii).

1.75

“Know-How” means all technical and scientific information, know-how, and data, including inventions, discoveries,
trade  secrets,  specifications,  instructions,  processes,  formulae,  compositions  of  matter,  cells,  cell  lines,  assays,  animal  models,  and  other
physical, biological, or chemical materials, expertise, and other technology applicable to development, registration, use, or marketing or to
methods  of  assaying  or  testing  them,  and  including  all  biological,  chemical,  pharmacological,  biochemical,  toxicological,  pharmaceutical,
physical,  and  analytical  safety,  nonclinical,  and  clinical  data,  regulatory  documents,  data  and  filings,  instructions,  processes,  formulae,
expertise, and information relevant to the research, development, use, importation, offering for sale, or sale of, or which may be useful in
studying, testing, developing, Products.  Know-How excludes Patents.  

1.76

1.77

“Licensee Data” has the meaning set forth in Section 10.1(a).

“Licensee Indemnitee” has the meaning set forth in Section 12.1.

1.78

“Licensee  Know-How”  means  all  Know-How  that  Licensee  or  its  Affiliate(s)  Controls  as  of  the  Effective  Date  or
during  the  Term,  including  any  Joint  Inventions,  that  is  necessary  or  reasonably  useful  for  the  research,  Development,  manufacture,  use,
importation,  offer  for  sale,  or  sale  of  the  Compound  or  any  Product  in  the  Field.    For  clarity,  subject  to  Section 8.2(b)  in  the  case  of  any
Licensee Data generated as a result of Licensee’s Independent Development Activities, the Licensee Know‑How includes the Licensee Data.

8
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
1.79

“Licensee Patents” means all Patents that Licensee or its Affiliate(s) Controls as of the Effective Date or during the
Term  (including  any  Joint  Patents)  that  would  be  infringed,  absent  a  license  or  other  right  to  practice  granted  under  such  Patents,  by  the
research, Development, manufacture, use, importation, offer for sale, or sale of any Compound or Product (considering patent applications to
be issued with the then-pending claims and considering Joint Patents as if owned solely by Licensee or its Affiliate).

1.80

“Licensee Technology” means the Licensee Know-How and the Licensee Patents, including Licensee’s interest in the

Joint Inventions and Joint Patents.

1.81

“Licensee  Territory”  or  “Licensed  Territory”  means  Austria,  Belgium,  Bulgaria,  Croatia,  Cyprus,  Czechia,
Denmark, Estonia, Finland, France, Germany, Greece, Hungary, Iceland, Ireland, Italy, Latvia, Liechtenstein, Lithuania, Luxembourg, Malta,
Netherlands, Norway, Poland, Portugal, Romania, Russia, Slovakia, Slovenia, Spain, Sweden, Switzerland, Turkey, and the United Kingdom.

1.82

1.83

“Licensee Territory Development Activities” has the meaning set forth in Section 4.2(b).

“Losses” has the meaning set forth in Section 12.1.

1.84

“Lundbeck  License  Agreement”  means  the  License  Agreement  by  and  between  Ovid  and  H.  Lundbeck  A/S
(“Lundbeck”)  dated  25  March,  2015,  and  amended  on  July  7,  2020  to  clarify  certain  sights  of  sublicensees  upon  termination  of  such
agreement (such amendment, the “Lundbeck Sublicense Amendment”).

1.85

“MAA” means a marketing authorization application or equivalent application, and all amendments and supplements
thereto, filed with the applicable Regulatory Authority in any country or jurisdiction.  For clarity, MAA does not include any application for
Pricing and Reimbursement Approval.

1.86

“MAA Approval”  means  approval  of  an  MAA  by  the  applicable  Regulatory  Authority  for  marketing  and  sale  of  a

Product in the applicable country or jurisdiction, but excluding any Pricing and Reimbursement Approval.

1.87

“Major European Market” means [***].

1.88

Manufacturing  Development”  means  any  of  the  following  with  respect  to  the  Compound  or  a  Product:
manufacturing process development, process improvements and any analytical development or validation associated with such development
or improvements.

1.89

“Market  Exclusivity”  means  any  exclusive  marketing  rights  or  data  exclusivity  rights  conferred  by  a  Regulatory
Authority with respect to a Product other than patents, including Directive 2001/83/EC and 2004/27/EC (as amended) in the EU and rights
equivalent  to  those  conferred  in  the  U.S.  under  the  Hatch-Waxman  Act  or  the  FDA  Modernization  Act  of  1997  (including  pediatric
exclusivity).

9
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
1.90

“Medical  Affairs”  or  “Medical  Affairs  Activities”  means  activities  designed  to  ensure  or  improve  appropriate
medical  use  of,  conduct  medical  education  of,  or  further  research  regarding,  the  Product,  including  by  way  of  example:    (a)  activities  of
medical  scientific  liaisons/medical  advisors  who,  among  their  other  functions,  may:  (i)  conduct  service  based  medical  activities  including
providing input and assistance with consultancy meetings, proposing investigators for clinical trials sponsored or co-sponsored by a Party or
Affiliate,  and  providing  input  in  the  design  of  such  trials  and  other  research  related  activities;  and/or  (ii)  deliver  non-promotional
communications  and  conduct  non-promotional  activities;  (b)  grants  to  support  continuing  medical  education,  symposia,  or  Third  Party
research related to the Product; (c) development, publication, and dissemination of original and literature review data relating to the Products;
(d) medical information services provided in response to inquiries communicated via sales representatives or received by letter, phone call, or
email;  (e)  conducting  advisory  board  meetings,  international  advisory  board  activities,  or  other  consultant  programs,  including  the
engagement  of  key  opinion  leaders  and  health  care  professional  in  individual  or  group  advisory  and  consulting  arrangements;  and  (f)  the
evaluation of applications submitted for support of investigator-initiated trials.  

1.91

“Neptune Trial” means the Phase 3 Clinical Trial of the Product for Angelman Syndrome ongoing as of the Effective

Date and for which Ovid is the sponsor, as further described in Exhibit J.

“Net Sales”  means,  with  respect  to  any  Product,  the  aggregate  gross  amount  invoiced  by  Licensee,  its  Affiliates,  or
Sublicensees for the sale of the Product to a Third Party, less the following deductions to the extent allowed and actually taken on such sales:

1.92

Sublicensee’s customers, including handling charges and insurance premiums relating thereto;

(a)

transportation charges relating to the Product to the extent actually invoiced to Licensee’s, its Affiliate’s, or

to the Product and any other equivalent governmental charges imposed on the importation, use, or sale of the Product;

(b)

sales taxes, excise taxes, use taxes, VAT, and duties paid by Licensee, its Affiliate, or Sublicensee in relation

(c)
and other rebates or fees;

(d)

(e)

(f)

Payments).

government-mandated  rebates  (including  any  Paybacks  or  Clawbacks  charged  with  respect  to  the  Product)

customary trade, quantity, and case discounts allowed on the Product;

allowances or credits to customers on account of retrospective price reductions affecting the Product; and

customary  rebates  (including  confidential  discount  agreements  Success  Fee  and  Performance  based

The transfer of Product between Licensee and its Affiliates and Sublicensees shall not be considered a sale unless
the Affiliate or Sublicensee is a bona fide purchaser at fair market value for resale.  If the Affiliate or Sublicensee
is not an end user, Net Sales shall be determined based

10
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
on  the  invoiced  sale  price  by  the  Affiliate  or  Sublicensee  to  the  first  Third  Party  trade  purchaser,  less  the
deductions allowed under this Section 1.92.  Disposal of Product for or use of Product in Clinical Studies or as
free samples in quantities common in the industry for this sort of Product shall not give rise to any deemed sale
under this definition.

Net Sales shall be calculated and accounted for in accordance with accounting standards during the Term (i.e., IFRS), consistently applied.

If Product is sold for other than cash payment, Net Sales of the Product shall be deemed to be the cash value of such other payment.

If the Product is sold as part of a Combination Product, Net Sales of such Product shall be deemed to be an amount equal to the following:

(X divided by Y) multiplied by Z,

where “X”  is  the  average  sales  price  during  the  applicable  reporting  period  achieved  for  the  relevant  Product  in  the
country in which such sale occurred when the Product contains only the Compound and no other active pharmaceutical
ingredient;

“Y”  is  the  sum  of  the  average  sales  price  as  a  single  entity  during  the  applicable  reporting  period  achieved  in  that
country (as applicable) of each product included in the Combination Product when such product is sold as a separate
product and not as part of a Combination Product; and

“Z” is the single price at which the relevant Combination Product was actually sold.

In the event that no separate sale of either (a) the Product comprising the Compound as the sole active pharmaceutical ingredient,
or  (b)  a  product  containing  the  other  active  pharmaceutical  ingredient(s)  included  in  the  Combination  Product,  are  made  during  the
accounting period in which the sale was made or if the price for a particular therapeutically active ingredient cannot otherwise be determined
for an accounting period, Net Sales allocable to the Product shall be determined by mutual agreement of the Parties prior to the end of the
accounting period in question based on an equitable method of determining the same that takes into account, in the Territory, variations in
potency, the relative contribution of each therapeutically active ingredient in the Combination Product, and relative value to the end user of
each  therapeutically  active  ingredient;  provided,  that  if  the  Parties  cannot  reach  mutual  agreement  prior  to  the  end  of  the  applicable
accounting period, such matter shall be resolved in accordance with Article 15.

1.93

“Orphan Drug Designation”  means  a  status  assigned  to  a  medicine  intended  for  use  against  a  rare  condition.  The
medicine  must  fulfil  certain  criteria  for  designation  as  an  orphan  medicine  so  that  it  can  benefit  from  incentives  such  as  protection  from
competition once on the market.

1.94

“Orphan Drug Designation of the Product” means the EMA orphan drug designation obtained for the Product.

11
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
1.95

“Orphan Medicine” means a medicine that continues to meet the criteria for maintaining its orphan status in parallel

with the assessment of an application for marketing authorisation by the European Medicines Agency (EMA).

1.96

“Ovid  Commercially  Reasonable  Efforts”  means,  with  respect  to  Ovid  and  its  obligations  under  this  Agreement,
commercially reasonable efforts and resources as commonly used by a similar size pharmaceutical company to Develop and Commercialize a
product controlled by Ovid or to which it has exclusive rights, which product is at similar stage in its development or product life and is of
similar market potential taking into account efficacy, safety, approved and/or anticipated labelling, the competitiveness of alternative products
sold by Third Parties in the marketplace, the patent and other proprietary position of the product, likelihood of regulatory approval given the
regulatory  structure  involved,  the  profitability  of  the  product,  [***],  and  other  relevant  factors,  including  technical,  legal,  scientific  and/or
medical factors. Commercially Reasonable Efforts shall be determined on a country-by-country basis and indication-by-indication basis for a
particular Product, and it is anticipated that the level of effort will change over the time, reflecting changes in the status of the Product and the
country(s) involved.

1.97

1.98

“Ovid Data” has the meaning set forth in Section 10.1(a).

“Ovid Indemnitee” has the meaning set forth in Section 12.2.

1.99

“Ovid Know-How” means all Know-How that Ovid Controls as of the Effective Date or, subject to Section  2.7(b),
during the Term, including any Joint Inventions, that is necessary or reasonably useful for the Development, use, importation, offer for sale,
or sale of any Compound or Product in the Field in the Licensee Territory.  For clarity, any Ovid Data generated during Ovid’s Independent
Development  Activities  will  be  included  within  the  Ovid  Know‑How  following  reimbursement  by  Licensee  of  its  share  of  Development
Costs in accordance with Section 8.2(b).

1.100

“Ovid Ongoing Trials” means the Rocket Trial, Elara Trial, and Neptune Trial.

1.101

“Ovid Patents” means all Patents in the Licensee Territory that Ovid Controls as of the Effective Date or, subject to
Section 2.7(b), during the Term (including any Joint Patents) that would be infringed, absent a license or other right to practice granted under
such Patents, by the Development, use, importation, offer for sale, or sale of any Compound or Product in the Field in the Licensee Territory
(considering patent applications to be issued with the then-pending claims and considering Joint Patents as if owned solely by Ovid).  The
Ovid Patents existing as of the Effective Date are set forth in Exhibit B.

1.102
Inventions and Joint Patents.

“Ovid  Technology”  means  the  Ovid  Know‑How  and  the  Ovid  Patents,  including  Ovid’s  interest  in  the  Joint

1.103

1.104

“Ovid Territory” means the world outside the Licensee Territory.

“Paediatric  Investigational  Plan  (PIP)”  is  the  development  plan  aimed  at  ensuring  that  the  necessary  data  are

obtained through studies in children, to support the

12
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
authorisation of a medicine for use in children. Any Applicants must obtain EMA approval of the PIP before MAA.

1.105

“Patents”  means  (a)  all  patents,  certificates  of  invention,  applications  for  certificates  of  invention,  priority  patent
filings, provisional patent applications and patent applications, and (b) any renewals, divisions, or continuations (in whole or in part) of any
of such patents, certificates of invention and patent applications, and any all patents or certificates of invention issuing thereon, and any and
all reissues, reexaminations, extensions, supplementary protection certificates, divisions, renewals, substitutions, confirmations, registrations,
revalidations, revisions, and additions of or to any of the foregoing.

1.106

“Payback” means payback policies which require manufacturers to pay back a share of their revenue in respect of a

product, if a prespecified budget ceiling for public pharmaceutical expenditures is exceeded.

1.107

“Pharmacovigilance Agreement” has the meaning set forth in Section 5.4.

1.108

“Phase 1 Clinical Trial” means a human clinical trial of a pharmaceutical product that satisfies the requirements for
a  Phase  1  study  as  defined  in  21  CFR  §  312.21(a)  (or  any  amended  or  successor  regulations),  regardless  of  where  such  clinical  trial  is
conducted.

1.109

“Phase 2 Clinical Trial” means a human clinical trial of a pharmaceutical product that satisfies the requirements for
a  Phase  2  study  as  defined  in  21  CFR  §  312.21(b)  (or  any  amended  or  successor  regulations),  regardless  of  where  such  clinical  trial  is
conducted.

1.110

“Phase 3 Clinical Trial” means a human clinical trial of a pharmaceutical product for an indication on a sufficient
number of subject that is designed to establish that the pharmaceutical product is safe and efficacious for its intended use, and to determine
warnings, precautions and adverse reactions that are associated with the pharmaceutical product in the dosage range to be described, and to
support Regulatory Authority to market such Product in patients having the indication being studied and that satisfies the requirements for a
Phase  3  study  as  defined  in  21  CFR  §  312.21(c)  (or  any  amended  or  successor  regulations),  regardless  of  where  such  clinical  trial  is
conducted.

1.111

“Phase 4 Clinical Trial” means a product support clinical trial of a Product that is commenced after receipt of MAA
Approval  in  the  country  where  such  trial  is  conducted.  Phase  4  Clinical  Trial  may  include  epidemiological  studies,  modeling  and
pharmacoeconomic studies, and post-marketing surveillance trials.

1.112

“PIP  Compliance  Check”  means  that  PIP  has  been  checked  by  EMA  for  compliance  with  all  the  measures

mentioned in the PIP decision, including the timelines for the conduct of the studies or collection of the data.

1.113

“Pricing and Reimbursement Approval” means, with respect to a Product, the approval, agreement, determination,
or decision of any applicable Governmental Authority establishing the price or reimbursement level for such Product, as required in a given
country or jurisdiction prior to sale of such Product in such country or jurisdiction.

13
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
1.114

“Product”  means  any  pharmaceutical  product  containing  the  Compound  as  an  active  ingredient,  alone  or  in
combination with one or more other active pharmaceutical ingredients, in any form, presentation, dosage, or formulation, and for any mode of
administration.

1.115

1.116

1.117

1.118

“Product Infringement” has the meaning set forth in Section 10.3(a).

“Promotional Materials” has the meaning set forth in Section 6.4(c).

“Proposal” has the meaning set forth in Section 4.3.

“Proposing Party” has the meaning set forth in Section 4.3.

1.119

“Public Official or Entity” means (a) any officer, employee (including physicians, hospital administrators, or other
healthcare  professionals),  agent,  representative,  department,  agency,  de  facto  official,  representative,  corporate  entity,  instrumentality,  or
subdivision of any government, military, or international organization, including any ministry or department of health or any state-owned or
affiliated company or hospital, or (b) any candidate for political office, any political party, or any official of a political party.

1.120

1.121

“Rare Disease” means a disease that affects one person per two thousand (2,000).

“Recall” has the meaning set forth in Section 5.7.

1.122

“Regulatory  Approval”  means,  with  respect  to  a  country  or  jurisdiction,  any  and  all  approvals  (including  MAA
Approval  and,  if  required  by  Applicable  Law,  Pricing  and  Reimbursement  Approval),  licenses,  registrations,  permits,  notifications  and
authorizations (or waivers) of any Regulatory Authority that are necessary for the manufacture, use, storage, import, transport, promotion,
marketing, distribution, offer for sale, sale, or other commercialization of a Product in such country or jurisdiction.

1.123

“Regulatory Authority” means any Governmental Authority that has responsibility in its applicable jurisdiction over
the  testing,  development,  manufacture,  use,  storage,  import,  transport,  promotion,  marketing,  distribution,  offer  for  sale,  sale,  or  other
commercialization of pharmaceutical products in a given jurisdiction.  For countries where Pricing and Reimbursement Approval is required,
Regulatory Authority shall also include any Governmental Authority whose grant of Pricing and Reimbursement Approval of the Product is
required.  

1.124

“Regulatory  Filing”  means  all  applications,  filings,  submissions,  approvals,  licenses,  registrations,  permits,
notifications, and authorizations (or waivers) with respect to the testing, Development, manufacture, or Commercialization of any Product
made to or received from any Regulatory Authority in a given country, including INDs and MAAs.

1.125

1.126

“Regulatory Meeting” has the meaning set forth in Section 5.1(c)(ii).

“Regulatory Milestone Event” has the meaning set forth in Section 8.3(a).

14
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
1.127

“Rocket Trial” means the Phase 2 Clinical Trial of the Product for Fragile X Syndrome ongoing as of the Effective

Date and for which Ovid is the sponsor, as further described in Exhibit J.

1.128

“Safety Data”  means  Data  related  solely  to  any  adverse  drug  experiences  and  serious  adverse  drug  experience  as
such  information  is  reportable  to  Regulatory  Authorities.    Safety  Data  also  includes  “adverse  events”,  “adverse  drug  reactions”,  and
“unexpected  adverse  drug  reactions”  as  defined  in  the  ICH  Harmonised  Tripartite  Guideline  for  Clinical  Safety  Data  Management:
Definitions and Standards for Expedited Reporting.

1.129

“SEC”  means  the  U.S.  Securities  and  Exchange  Commission,  or  any  successor  entity  or  its  foreign  equivalent,  as

applicable.

1.130

1.131

1.132

“Safety Reason” has the meaning set forth in Section 4.15.

“Sales Milestone Event” has the meaning set forth in Section 8.4(a).

“Scientific  Advice”  means  any  report  of  the  advice  provided  by  EMA  to  medicine  developers  on  the  most

appropriate way to generate robust evidence on a medicine’s benefits and risks.

1.133

1.134

“Second Indication” means Fragile X syndrome (FXS).

“Second  Indication  Opt-In”  means  the  election  by  Licensee,  following  the  Licensee’s  exercise  of  the  Second

Indication Opt-Out, to resume the Licensee’s rights granted to Licensee according to Section 2.1 with respect to the Second Indication.

1.135

“Second  Indication  Opt-Out”  means  the  election  by  Licensee,  in  accordance  with  the  terms  hereof,  not  to

participate in Development and/or Commercialization activities for the Product for the Second Indication.

1.136

“Segregate” means, with respect to a Competing Product, to [***] segregate the Development, Manufacturing and
Commercialization of such Competing Product in the Field from Development, Manufacture and Commercialization activities with respect to
Compounds and Products under this Agreement, including [***]; provided that, [***].

1.137

“Sponsor” means the Party that takes the ultimate responsibility for the initiation, performance, and management of,

including financing or arranging the financing for, the applicable Clinical Trial.

1.138

“Sublicensee” means a Third Party to whom Licensee grants a sublicense to Develop, use, import, promote, offer for

sale, or sell any Product in the Field in the Licensee Territory.  In no event shall Ovid or any of its Affiliates be deemed a Sublicensee.

1.139

“Success Fee” or “Performance Based Payments”  means  the  returned  part  of  the  Product-generated  revenues  for
those  cases  where  outcomes  are  not  meeting  pre-defined  clinical  goals  set  by  National  Health  Authority  (e.g.QoL  Gain,  Survival,
Progression, Course of Disease Modification).

15
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
1.140

1.141

“Sunshine Reporting Laws” has the meaning set forth in Section 5.8.

“Supply Agreement” means the supply agreement between Ovid and Licensee attached hereto as Exhibit K.

1.142

“Take the Lead” means, with the respect to a particular Party and a particular activity, that such Party is primarily
responsible  for,  and  has  the  authority  to  make,  all  day-to-day  operational  decisions,  in  accordance  with  the  Development  Plan  and
Commercialization Plan and the terms of this Agreement; provided that [***]; and provided further that [***].  For clarity, [***].

1.143

“Technology Transfer Completion Date” means the earlier of (a) the date on which the activities [***], as set forth

in the Technology Transfer Plan, has been completed, but for clarity, excluding [***] and (b) the [***].

1.144

1.145

1.146

1.147

“Technology Transfer Agreement” has the meaning set forth in Section 11.4(e).

“Technology Transfer Plan” has the meaning set forth in Section 11.4(e).

“Term” has the meaning set forth in Section 14.1.

“Third Party” means any entity other than Ovid or Licensee or an Affiliate of Ovid or Licensee.

1.148

“Threshold Price Sale” means, on a Product-by-Product and country-by-country basis, the first sale of such Product
in  such  country  (after  Regulatory  Approval  for  such  Product  has  been  obtained  in  such  country)  for  which  Licensee  or  its  Affiliate  or
Sublicensee, as applicable, invoices a Third Party (a) [***], or (b) [***].

1.149

1.150

“Total Supply Price” means, for any Product, [***].

“U.S.” means the United States of America, including its territories and possessions (including Puerto Rico).

1.151

“Valid Claim” means (a) a claim of an issued and unexpired patent that has not been revoked or held unenforceable,
unpatentable, or invalid by a decision of a court or other governmental agency of competent jurisdiction that is not appealable or has not been
appealed within the time allowed for appeal, and that has not been abandoned, disclaimed, denied, or admitted to be invalid or unenforceable
through  reissue,  re-examination,  or  disclaimer  or  otherwise,  or  (b)  a  claim  of  a  pending  patent  application  that  has  not  been  cancelled,
withdrawn, or abandoned or finally rejected by an administrative agency action from which no appeal can be taken.

2.

GRANT OF LICENSES

2.1

Licenses Granted to Licensee.  Subject to the terms and conditions of this Agreement, Ovid hereby grants to Licensee,

during the Term:

16
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
(a)

an exclusive (even as to Ovid, except as expressly set forth herein), royalty-bearing license, with the right to
grant sublicenses (through multiple tiers) solely as provided in Section 2.2, under the Ovid Technology to use and have used, sell, offer for
sale, import, and otherwise Commercialize and have Commercialized (but not to make or have made, unless otherwise provided herein) the
Products in the Field in the Licensee Territory;

a  non-exclusive  license,  with  the  right  to  grant  sublicenses  (through  multiple  tiers)  solely  as  provided  in
Section  2.2,  under  the  Ovid  Technology  to  Develop  (but  not  to  make  or  have  made  unless  otherwise  provided  herein)  the  Products  on  a
worldwide basis in accordance with the Development Plan, and to use the Products for that purpose; and

(b)

(c)

a non-exclusive, royalty-bearing license, with the right to grant sublicenses (through multiple tiers) solely as
provided in Section 2.2, under the Ovid Technology to make or have made the Products solely for use in the Field in the Licensee Territory in
accordance with the licenses granted in Sections 2.1(a) and 2.1(b), provided that, for clarity, Licensee’s rights under any Patents and Know-
How Controlled by Lundbeck that are included within the Ovid Technology shall be subject to the completion of the Technology Transfer and
the terms of the Lundbeck License Agreement; and

(d)

solely as and to the extent provided in Section 14.5, an exclusive (even as to Ovid, except as expressly set
forth herein), royalty-bearing license, with the right to grant sublicenses (through multiple tiers) solely as provided in Section 2.2, under the
Ovid  Technology  to  Develop,  have  developed,  use  and  have  used,  sell,  offer  for  sale,  import,  and  otherwise  Commercialize  and  have
Commercialized the Products in the Field in the Licensee Territory.

2.2

Sublicenses.  Licensee shall have the right to grant sublicenses under the licenses granted in Section 2.1:

provided that such sublicense will terminate if such sublicensee no longer qualifies as an Affiliate of Licensee.

(a)

to  an  Affiliate  of  Licensee  without  Ovid’s  express  prior  written  consent  but  with  written  notice  to  Ovid,

(b)
unreasonably withheld, conditioned or delayed).

to a Third Party other than as set forth in Section 2.2(a) with Ovid’s express prior written consent (not to be

All sublicenses granted under the licenses granted in Section 2.1 shall be in writing and shall be subject
to, and consistent with, the terms and conditions of this Agreement and shall provide that any such Sublicensee
(including  any  distributor)  shall  not  further  sublicense  except  with  the  written  consent  of  Licensee  and
Ovid.  Licensee shall ensure that each agreement with a Sublicensee grants Ovid all rights with respect to Data,
Inventions,  and  Regulatory  Filings  made  or  generated  by  such  Sublicensee  as  if  such  Data,  Inventions,  and
Regulatory Filings were made or generated by Licensee. Licensee shall be responsible for the compliance of its
Affiliates,  Sublicensees  (including  any  distributors),  and  subcontractors  with  the  terms  and  conditions  of  this
Agreement.  Licensee shall provide written notice to Ovid of each sublicense granted to a Third Party hereunder,
specifying the name of the Sublicensee, the territory, and the duration of the sublicense.

17
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or confidential.

 
2.3

Reserved Rights.  Ovid hereby expressly reserves:

whether directly or through one or more licensees or subcontractors; and

(a)

the right under the Ovid Technology to exercise its rights and perform its obligations under this Agreement,

granted in Section 2.1.

(b)

all rights to practice, and to grant licenses under, the Ovid Technology outside of the scope of the licenses

2.4

Licenses  Granted  to  Ovid.  Subject  to  the  terms  and  conditions  of  this  Agreement,  including  Section  2.8,  Licensee

hereby grants to Ovid:

the Licensee Technology to use, sell, offer for sale, import, and otherwise Commercialize the Products in the Ovid Territory; and

(a)

a non-exclusive, royalty-free, fully paid-up license, with the right to sublicense (through multiple tiers), under

a non-exclusive, worldwide, royalty-free, fully paid-up license, with the right to sublicense (through multiple
tiers), under the Licensee Technology to (i) Develop the Compound and Products on a worldwide basis under the Development Plan, and (ii)
to make and have made the Compound and Products anywhere in the world.

(b)

2.5

No  Implied  Licenses;  Negative  Covenant.    Except  as  set  forth  in  this  Agreement,  neither  Party  shall  acquire  any
license or other intellectual property interest, by implication or otherwise, under or to any Patents, Know-How, or other intellectual property
owned or controlled by the other Party.  Neither Party shall, nor shall it permit any of its Affiliates or (sub)licensees to, practice any Patents or
Know-How licensed to it by the other Party outside the scope of the licenses granted to it under this Agreement.

2.6

Disclosure of Know-How.  For as long as the Parties are conducting Development activities under the Development
Plan, upon Licensee’s written request no more frequently than [***], Ovid shall disclose and make available to Licensee, in electronic form
where  possible,  all  Ovid  Know-How  that  comes  into  existence  after  the  Effective  Date  and  that  was  not  previously  provided  to  Licensee,
promptly  after  the  earlier  of  the  development,  making,  conception,  or  reduction  to  practice  of  such  Ovid  Know-How.    For  as  long  as  the
Parties  are  conducting  Development  activities  under  the  Development  Plan,  upon  Ovid’s  written  request  no  more  frequently  than  [***],
Licensee shall, and shall cause its Affiliates to, disclose and make available to Ovid, in electronic form where possible, any Licensee Know-
How not previously  provided  to  Ovid, promptly  after  the  earlier  of  the  development, making, conception, or reduction to practice of such
Licensee Know-How.  The CGB shall establish a mechanism for the reciprocal disclosure of such Know-How.

2.7

Third Party Licenses.  

Notice. Licensee shall promptly notify Ovid if it becomes aware of any Third Party Know-How or Patent that
is necessary or reasonably useful to Develop, make, have made, use, sell, offer for sale, or import the Compound or Product in the Field in the
Licensee Territory, and [***].

(a)

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or confidential.

 
(b)

Sublicense  under  Third  Party  License.    If  Ovid  enters  into  any  agreement  with  a  Third  Party  after  the
Effective Date that includes a license from such Third Party to Ovid under any Know-How or Patents that are necessary to Develop, use, sell,
offer for sale, or import the Products in the Field in the Licensee Territory, and Ovid has the right to grant a sublicense under such Know-How
or  Patents  to  Licensee,  then  Ovid  shall  notify  Licensee  and  identify  the  relevant  Know-How  or  Patents  and  provide  Licensee  with  the
substantive terms of the applicable Third Party license agreement to Licensee, in each case to the extent applicable to the rights that would be
sublicensed to Licensee.  Such Know-How and Patents, to the extent falling within the definition of Ovid Technology, will be sublicensed to
Licensee only if Licensee provides Ovid with written notice in which (i) Licensee consents to adding such Patents and Know-How to the
definition of Ovid Technology and (ii) Licensee acknowledges in writing that its sublicense under such license agreement is subject to the
terms and conditions of such license agreement.

Licensee Restriction.  Except with the prior written consent of Ovid, Licensee shall not obtain a license to
any Third Party Patent or Know-How that is necessary to Develop, make, have made, use, sell, offer for sale, or import the Products in the
Ovid Territory.

(c)

2.8

Exclusivity.

Exclusivity.  Subject to Section 2.8(c), for the period starting from the Effective Date and for [***] in the
Licensee Territory, neither Party shall, directly or indirectly (including through an Affiliate or a Third Party), develop or commercialize any
Competing Product that is directed to the treatment of the Initial Indication or Second Indication in the Licensee Territory.

(a)

(b)

Competing Program Exclusivity.  If a Third Party becomes an assignee of this Agreement from a Party, or
becomes  an  Affiliate  of  a  Party  after  the  Effective  Date  through  merger,  acquisition,  consolidation,  or  other  similar  transaction,  and  such
Third Party, as of the closing date of such transaction, is engaged in the development or commercialization of a Competing Product in the
Licensee  Territory  (a  “Competing Program”),  then  such  Competing  Program  shall  not  be  a  breach  of  Section 2.8(a),  so  long  as  (i)  such
Third Party, or such Party or its Affiliates, [***], and (ii) [***] such Competing Product.  [***] of such Competing Program.  

Territory  Exclusivity.    During  the  Term,  Licensee  shall  not,  directly  or  indirectly  (including  through  an
Affiliate  or  a  Third  Party),  Commercialize  the  Product  in  the  Ovid  Territory.  Ovid  shall  not,  directly  or  indirectly  (including  through  an
Affiliate or a Third Party), Commercialize the Product in the Licensee Territory, except as provided in Section 2.3(a).

(c)

(d)

Effect of Triggering Acquisition. In the event of an acquisition of Ovid by a Competing Acquirer that closes
prior to [***] (a “Triggering Acquisition”), then Ovid shall provide notice to Licensee of such Triggering Acquisition within [***] after the
date upon which the Triggering Acquisition closes or otherwise becomes effective. On or before the date that is [***] after the date on which
Licensee receives notice of a Triggering Acquisition, Licensee shall have the right to elect to Take the Lead on any or all then current Joint
Development Activities and future Licensee activities in the Licensee Territory, [***] remaining in full force and effect. For sake of clarity,
[***].

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or confidential.

 
2.9

Licensee’s access to Ovid Data, Know-How and Patents

Ovid hereby agrees to provide to Licensee, within [***] following the Effective Date, a list of (a) [***] the
Ovid  Know-How  [***]  and  (b)  [[***]  the  Compound  and/or  Product  necessary  for  Licensee’s  Development,  use,  manufacture,  and
Commercialization of the Product in the Field in the Licensee Territory, [***].

(a)

control that relate to [***].

(b)

Promptly  following  the  Effective  Date,  Ovid  shall  transfer  to  Licensee  information  in  its  possession  and

From time to time during the Term, and at no additional cost to Licensee (subject to Section 4.5), Ovid shall
provide to Licensee [***] the Ovid Know-How solely relating to the Compound and/or the Product, reasonably requested by Licensee and
necessary for Licensee’s Development, use, manufacture, and Commercialization of the Product.

(c)

(d)

Ovid hereby agrees that, [***] following the Effective Date, Ovid will provide to Licensee the Ovid Know-
How  [***]  for  Licensee  to  Develop,  manufacture,  use,  and  Commercialize  the  Compound  and  the  Product  in  the  Field  in  the  Licensee
Territory in accordance with the terms of this Agreement. Licensee shall reimburse Ovid all out of pocket costs and reasonable, internal cost
related to such technology transfer.

2.10

Licensee’s Access to Ovid Personnel.  The Parties acknowledge the significant contribution and experience of Ovid
and Ovid employees to the Development, manufacture, use, and Commercialization of the Compound and Product prior the Effective Date
and that these contributions and experience may be valuable to Licensee. Accordingly, Licensee is entitled to meet with employees of Ovid
who hold significant experience or expertise in the Development activities, and manufacture, use, and Commercialization of the Compound
and Product. Licensee shall provide reasonable notice to Ovid requesting such a meeting and Ovid’s approval of date and agenda of meeting
shall not be unreasonably withheld. Each Party shall bear its own cost in relation to such meetings.

3.

GOVERNANCE

3.1

Collaboration  Governance  Board.    As  of  the  Effective  Date,  the  Parties  have  established  a  board  to  govern  their
collaboration under this Agreement (the “Collaboration Governance Board” or the “CGB”), composed of an equal number of up to [***]
employees of each Party, to oversee and guide the strategic direction of the collaboration of the Parties under this Agreement.  The CGB shall
act as a joint consultative body and, to the extent expressly provided herein, a joint decision-making body.  The CGB shall in particular:

overall implementation of the Development Plan;

(a)

review and discuss the strategy for the Development of the Product worldwide, coordinate and oversee the

the Licensee Territory;

(b)

provide a forum for discussion of the Development and Commercialization of the Compound and Products in

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or confidential.

 
against agreed budgets, and discuss and approve any budget overruns;

(c)

monitor  performance  of  Development  activities  in  and  for  the  Licensee  Territory,  including  performance

(d)

(e)

oversee the activities of the JPT, and serve as a forum for resolution of disputes arising at the JPT;

review  and  discuss  any  proposed  amendments  to  the  Development  Plan,  including  corresponding  budgets,

and approve any proposed amendments to Joint Development Activities under the Development Plan;

progress of all Clinical Trials in the Licensee Territory;

(f)

review,  discuss,  and  approve  Clinical  Trial  protocols  for  jointly-conducted  Clinical  Trials,  and  monitor  the

phase Clinical Trial is merited;

(g)

review Clinical Trial Data from jointly-conducted Clinical Trials to determine whether progress to the next

activities directed to Additional Indications;

(h)

review,  discuss,  and  approve  Proposals,  including  amendments  to  the  Development  Plan  with  respect  to

directed to obtaining Regulatory Approval in Additional Indications;

(i)

monitor  and  coordinate  regulatory  strategy  and  activities  for  the  Licensee  Territory,  including  activities

coordinating of pharmacovigilance and safety matters will conducted in accordance with the pharmacovigilance agreement);

(j)

coordinating reporting of pharmacovigilance and safety matters for the Product worldwide (monitoring and

(k)

oversee and coordinate Medical Affairs Activities for the Product in all Indications in the Licensee Territory;

review  and  discuss  the  Commercialization  Plan  for  the  Licensee  Territory,  including  any  amendments
proposed thereto, and oversee the Commercialization of Products in the Licensee Territory in accordance with the global commercialization
strategy for Products;

(l)

Products in the Licensee Territory and discuss potential international pricing reference by relevant Regulatory Authorities;

(m)

provide  a  forum  for  discussion  regarding  launch  sequencing,  pricing  and  reimbursement  strategy  for

13.4;

(n)

(o)

(p)

oversee the manufacturing and supply strategy and monitor supply of Products for the Licensee Territory;    

oversee and facilitate the Parties’ communications and activities with respect to publications under Section

establish joint subcommittees  as  it  deems  necessary  or  advisable  to  further  the purpose of this Agreement,

including as set forth in Section 3.7; and

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or confidential.

 
perform such other functions as appropriate to further the purposes of this Agreement, as expressly set forth
in  this  Agreement  or  allocated  to  it  by  the  Parties’  written  agreement,  including  providing  financial  oversight  of  the  activities  conducted
pursuant to this Agreement.

(q)

3.2

Joint Project Team.  No later than [***] following the Effective Date, the Parties will establish a cross-functional joint
project  team  (the  “JPT”),  composed  of  an  equal  number  of  up  to  [***]  employees  of  each  Party,  to  (a)  design  and  implement  the
Development Plan (subject to CGB review and approval), and (b) oversee the commercial strategy and Commercialization of the Products in
the Licensee Territory.  The JPT shall in particular:

on such activities;

(a)

(b)

oversee the conduct of activities under the Development Plan in the Licensee Territory and report to the CGB

provide a forum for, and facilitate communications between the Parties with respect to the Development of

Products in the Licensee Territory, including sharing of Data in accordance with Section 4.7;

(c)

(d)

prepare and submit to the CGB for approval protocols for jointly-conducted Clinical Trials;

prepare  amendments  to  the  Development  Plan  as  needed  (including  corresponding  changes  to  the

Development Budget) and submit such amendments to the CGB for approval;

(e)

review and discuss Proposals and make recommendations to the CGB with respect thereto;

review and discuss the CMC components of the Regulatory Filings in the Licensee Territory, and oversee and
coordinate  the  manufacture  and  supply  of  Drug  Product  to  Licensee  for  use  in  Clinical  Trials  for  which  Licensee  is  the  Sponsor  in  the
Licensee Territory;

(f)

(g)
commercialization in the Licensee Territory;

prepare  and  submit  to  the  CGB  for  approval  a  plan  for  manufacture  and  supply  of  Drug  Product  for

strategy for Products, and provide comments thereto;

(h)

review  the  Commercialization  Plan  prepared  by  Licensee  for  alignment  with  the  global  commercialization

(i)

(j)

the Development of Products.

monitor the conduct of Commercialization of Products in the Licensee Territory; and

perform such other functions as may be appropriate to further the purposes of this Agreement with respect to

3.3

Committee Membership and Meetings.

sufficient seniority within the applicable Party to make

(a)

Committee Members.  Each Committee representative shall have appropriate knowledge and expertise and

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or confidential.

 
decisions  arising  within  the  scope  of  such  Committee’s  responsibilities.    Each  Party  may  replace  its  representatives  on  a  Committee  on
written notice to the other Party.  The CGB chairperson shall be one of the representatives appointed by Ovid.  The chairperson of the JPT
shall alternate between one of the representatives appointed by Ovid and one of the representatives appointed by Licensee.  The chairperson
shall prepare and circulate agendas to Committee members at least [***] before each Committee meeting and shall direct the preparation of
reasonably  detailed  notes  for  each  such  Committee  meeting,  which  shall  be  approved  by  the  chairperson  and  circulated  to  Committee
members  within  [***]  after  such  meeting.    If  not  determined  as  of  the  Effective  Date,  the  Parties  shall  determine  their  respective  initial
members of each Committee promptly following the Effective Date.

(b)

Meetings.    Each  Committee  shall  hold  meetings  at  such  times  as  it  elects  to  do  so,  but  in  no  event  shall
meetings of the JPT be held less frequently than [***], and meetings of the CGB once every [***].  The first CGB meeting and first JPT
meeting  shall  be  held  within  [***]  after  the  Effective  Date.    Committee  meetings  may  be  held  in  person  or  by  audio  or  video
teleconference.  In-person Committee meetings shall be held at locations alternately selected by the Parties.  Each Party shall be responsible
for all of its own expenses of participating in any Committee meeting.  No action taken at any Committee meeting shall be effective unless at
least one (1) representative of each Party is participating.  In addition, upon written notice to the other Party, either Party may request that a
special  ad  hoc  meeting  of  a  Committee  be  convened  for  the  purpose  of  resolving  any  disputes  in  connection  with,  or  for  the  purpose  of
reviewing or making a decision pertaining to any material subject-matter within the scope of such Committee, the review or resolution of
which cannot be reasonably postponed until the following scheduled Committee meeting.  Such ad hoc meeting shall be convened at such
time as may be mutually agreed by the Parties, but no later than [***] following the notification date of request that such meeting be held.    

(c)

Non-Member Attendance.  Each Party may from time to time invite a reasonable number of participants, in
addition to its representatives, to attend Committee meetings in a non‑voting capacity; provided that if either Party intends to have any Third
Party (including any consultant) attend such a meeting, such Party shall provide reasonable prior written notice to the other Party and obtain
the other Party’s approval for such Third Party to attend such meeting, which approval shall not be unreasonably withheld or delayed.  Such
Party  shall  ensure  that  such  Third  Party  is  bound  by  written  confidentiality  and  non-use  obligations  consistent  with  the  terms  of  this
Agreement.

3.4

Decision-Making.

(a)

All decisions of a Committee shall be made by unanimous vote, with each Party’s representatives collectively
having  one  (1)  vote.    If  after  reasonable  discussion  and  good  faith  consideration  of  each  Party’s  view  on  a  particular  matter,  the
representatives of the Parties cannot reach an agreement as to such matter within [***] after such matter was first considered, then if such
disagreement arose within the JPT, it shall be referred to the CGB for resolution.  If the CGB cannot resolve such matter within a further
[***], or if the disagreement first arose within the CGB, then prior to any formal dispute resolution process such issue shall be referred to the
Executive Officers for resolution.  

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or confidential.

 
then:

(b)

If the Executive Officers cannot resolve such matter within [***] after such matter has been referred to them,

(i)

Ovid  shall  have  the  final  decision  making  authority,  which  shall  be  exercised  in  its  reasonable
discretion,  with  respect  to  (A)  Ovid’s  Independent  Development  Activities,  (B)  the  Ovid  Ongoing  Trials,  (C)  all  manufacturing  matters
outside  the  Licensee  Territory,  and  (D)  Joint  Development  Activities  necessary  for  obtaining  Regulatory  Approvals  for  Products  in  any
Indication  in  the  Licensee  Territory  for  which  Ovid  is  the  sponsor  (including  any  necessary  updates  to  the  Development  Plan  and
Development Budget pursuant to Section 4.2, but subject in all cases to Sections 3.4(b)(i)(1) and 3.4(b)(i)(2)), except for:

(1)

  the  addition  of  new  Clinical  Trials  to  the  Development  Plan  as  Joint  Development

Activities (the cost of which would be shared by the Parties); and

(2)

any material modification to a previously agreed upon Clinical Trial that is set forth in the
Development Plan as Joint Development Activities (unless such modification is required by a Regulatory Authority
or any local or regional IRB/ethics committee, or is reasonably necessary to protect patient safety); for the purpose of
this Section 3.4(b)(i)(2), “material modification” means [***].

(ii)

Licensee  shall  have  the  final  decision  making  authority  with  respect  to  (A)  Joint  Development
Activities necessary for obtaining Regulatory Approvals for Products in any Indication in the Licensee Territory for which Licensee is the
sponsor (including any necessary updates to the Development Plan and Development Budget pursuant to Section 4.2, but subject in all cases
to  Sections  3.4(b)(i)(1)  and  3.4(b)(i)(2)),  (B)  the  determination  of  whether  the  Additional  Pivotal  Trial  is  necessary  to  obtain  Regulatory
Approval in the Licensee Territory (although [***] for the Additional Pivotal Trial) (C) Commercialization of the Product in the Licensee
Territory, (D) Licensee Territory Development Activities and (E) Licensee’s Independent Development Activities in the Licensee Territory,
and (F) Phase 4 Clinical Trials for the Licensee Territory (but subject in all cases to Sections 3.4(b)(i)(1) and 3.4(b)(i)(2)), in each case (A)
through  (F)  provided  that  Licensee’s  exercise  of  any  such  decision  right  does  not  adversely  affect,  the  Development,  manufacture,  or
Commercialization of the Product in the Ovid Territory, and complies with the terms and conditions of this Agreement.  For clarity, [***].

Sections 3.4(b)(i)(1) and (2), and the status quo shall persist with respect to such matter unless and until the Parties are able to agree.

(iii)

Neither  Party  shall  have  the  final  decision  making  authority  with  respect  to  the  matters  in

3.5

Limitations  on  Authority.    Each  Committee  shall  have  only  such  powers  as  are  expressly  assigned  to  it  in  this
Agreement, and such powers shall be subject to the terms and conditions of this Agreement.  Without limiting the generality of the foregoing,
no  Committee  will  have  the  power  to  amend  this  Agreement,  and  no  Committee  decision  may  be  in  contravention  of  any  terms  and
conditions of this Agreement.

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or confidential.

 
3.6

Discontinuation  of  the  Committees.  The  activities  to  be  performed  by  each  Committee  shall  solely  relate  to
governance under this Agreement and are not intended to be or involve the delivery of services.  Each Committee shall continue to exist until
the first to occur of (a) the Parties mutually agree to disband such Committee or (b) Ovid provides written notice to Licensee of its intention
to disband and no longer participate in such Committee. Once the Parties mutually agree or Ovid has provided written notice to disband a
Committee,  such  Committee  shall  have  no  further  obligations  under  this  Agreement  and,  thereafter,  each  Party  shall  designate  a  contact
person for the exchange of information under this Agreement or such exchange of information shall be made through Alliance Managers, and
decisions of such Committee shall be decisions as between the Parties, subject to the other terms and conditions of this Agreement.  [***].

3.7

Alliance Managers. Promptly after the Effective Date, each Party shall appoint an individual who shall be an employee
of such Party having appropriate qualification and experience to act as the alliance manager for such Party (the “Alliance Manager”).  Each
Alliance Manager shall be responsible for coordinating and managing processes and interfacing between the Parties on a day-to-day basis
throughout the Term.  The Alliance Manager will ensure communication to the CGB of all relevant matters raised at the JPT and any other
subcommittee.  Each Alliance Manager shall be permitted to attend meetings of the CGB and JPT, in each case as appropriate and as non-
voting  participants.    The  Alliance  Managers  shall  be  the  primary  contact  for  the  Parties  regarding  the  activities  contemplated  by  this
Agreement and shall facilitate all such activities hereunder.  Each Party may replace its Alliance Manager with an alternative representative at
any time with prior written notice to the other Party.  Any Alliance Manager may designate a substitute to temporarily perform the functions
of  that  Alliance  Manager.    Each  Party  shall  bear  its  own  costs  of  its  Alliance  Manager,  which  costs  shall  be  excluded  from  the  Parties’
respective Development and manufacturing costs (including Cost of Goods) under this Agreement.

3.8

Supply Contacts.  Each Party shall designate one (1) qualified and experienced supply chain professional to serve as
that  Party’s  primary  supply  contact  regarding  the  supply  of  Drug  Product  under  this  Agreement  (“Supply  Contacts”).    Each  Party  may
replace its Supply Contact with an alternative representative at any time with prior written notice to the other Party.  The Supply Contacts
shall be responsible for facilitating information exchange and discussion between the Parties regarding the supply of Drug Product under this
Agreement.   The  Supply  Contacts  shall  have  decision-making  authority  with  respect  to  the  supply  of  Drug  Product  under  this  Agreement
within the guidance of the JPT and subject to the review and approval of the CGB.  Each Party shall bear its own costs of its Supply Contact,
which  costs  shall  be  excluded  from  the  Parties’  respective  Development  and  manufacturing  costs  (including  Cost  of  Goods)  under  this
Agreement.

4.

DEVELOPMENT

4.1

Overview.    Subject  to  the  terms  and  conditions  of  this  Agreement,  the  Parties  will  collaborate  with  respect  to  the
Development of the Compound and Products and share the Data resulting from such collaboration as provided in this Article 4 to facilitate
the Development of the Compound and Products throughout the Licensee Territory and the Ovid Territory.

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or confidential.

 
4.2

Amendments to Development Plan. Any amendment to the Development Plan for the Compound and Products under
this  Agreement,  including  the  Ovid  Ongoing  Trials,  Licensee  Territory  Development  Activities  for  registrational  purposes,  all  Joint
Development Activities, and all Independent Development Activities shall be conducted pursuant to a comprehensive written updated (from
time to time) Development Plan (the “Amended Development Plan”), which shall be incorporated by reference into this Agreement.  The
Amended  Development  Plan  will  include  Clinical  Trials  for  the  Initial  Indications  that  the  Parties  have  agreed  to  conduct  jointly  (unless
modification  is  required  by  a  Regulatory  Authority  or  any  local  or  regional  IRB/ethics  committee,  or  is  reasonably  necessary  to  protect
patient safety), the Clinical Trials for the Second Indication that Ovid may conduct under its sole responsibility and cost if Licensee exercises
the Second Indication Opt-Out and not the Second Indication Opt-In, as well as Clinical Trials for the Additional Indications that the Parties
(through the CGB) mutually agree to conduct and include in accordance with Section 4.3. The Amended Development Plan will also include:

(1)

(2)

(3)

any other Development activities approved by the CGB in accordance with Article 3; and

the PIP for the Initial Indication; and

the Additional Pivotal Trial, if applicable.

The  Amended  Development  Plan  shall  also  set  forth  the  amendments  to  the  detailed  budget  of  the  anticipated  costs  for  all  Development
activities (the “Amended Development Budget”) on a study-by-study or Clinical Trial-by-Clinical Trial basis.  As of the Effective Date, the
Parties have agreed upon an initial Development Plan and Development Budget, attached to this Agreement as Exhibit C.  If the terms of the
Development Plan contradict, or create inconsistencies or ambiguities with, the terms of this Agreement, then the terms of this Agreement
shall govern. In addition, the following shall apply to the Development of the Compound and Products under the Development Plan:

Neptune Trial, Rocket Trial and Elara Trial.  Ovid shall be responsible for, and shall use Commercially
Reasonable Efforts to conduct, at its own expense, (i) the Neptune Trial, (ii) the Rocket Trial, and (iii) the Elara Trial ((i)-(iii) collectively, the
“Ovid Ongoing Trials”).

(a)

PIP.  Ovid  shall  be  responsible  for  the  full  applying  process  to  obtain  EMA  agreement  for  the  Paediatric
Investigational Plan in order to allow the Licensee to submit the MAA for the Product for the Initial Indication in the Licensee Territory. Ovid
shall discuss and agree with the Licensee the PIP before moving forward with the application process.

(b)

(c)

Licensee Territory Development Activities for Initial Indication.  

Licensee shall be solely responsible for and shall use Angelini Commercially Reasonable Efforts to
conduct,  at  its  sole  expense,  all  Development  activities  that  are  exclusively  for  the  benefit  of  one  or  more  countries  within  the  Licensee
Territory for the Initial Indication, including (A) any and all Development activities required or recommended by a

(i)

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or confidential.

 
 
 
 
Regulatory Authority for the exclusive benefit of the Licensee Territory, including any Phase 4 Clinical Trials for the Initial Indication in the
Licensee  Territory,  and  (B)  any  and  all  Development  activities  required  for  any  Pricing  and  Reimbursement  Approval  in  the  Licensee
Territory.

 Licensee shall be solely responsible for the Additional Pivotal Trial, and for the Phase 4 Clinical
Trials  of  the  Product  in  the  Licensee  Territory,  but  Licensee  shall  bear  [***]  and  Ovid  shall  bear  [***]  of  the  Development  Costs  for  the
Development  Activities  for  the  Additional  Pivotal  Trial,  up  to  a  total  amount  of  [***],  and  for  any  Additional  Pivotal  Trial  Development
Costs in excess of [***] Licensee shall bear [***] and Ovid shall bear [***].

(ii)

(iii)

The activities specified in the foregoing subsections (i) and (ii) shall be referred to collectively as
the  “Licensee  Territory  Development  Activities”.    Prior  to  commencing  any  Licensee  Territory  Development  Activities,  Licensee  shall
provide the CGB with a draft workplan therefor, and following review and approval of such Licensee Territory Development activities by the
CGB, such Licensee Territory Development Activities shall be included in and conducted in accordance with the Development Plan, subject
to the oversight of the CGB and JPT as set forth in Article 3.  Notwithstanding anything to the contrary herein, Licensee shall consider in
good faith and incorporate Ovid’s reasonable comments on any proposed Licensee Territory Development Activities.

(d)

Joint Development Activities for Initial Indication and Second Indication. The Development Plan shall
set forth the timeline and details ([***]) of all preclinical (if any) and clinical Development activities ([***]) to be conducted jointly by the
Parties in order to generate Data sufficient to meet the common requirements of the FDA, EMA, and other Regulatory Authorities agreed
upon by the Parties for MAA Approval of the Compound and Products for each of the Initial Indication and eventually and separately for the
Second Indication, ([***]) (such activities, the “Joint Development Activities”).  All Joint Development Activities shall be included in and
conducted in accordance with the Development Plan, subject to the oversight of the CGB and JPT as set forth in Article 3. The Development
Plan shall also set forth the allocation of responsibility for all Joint Development Activities as between the Parties.  All Development Costs
Associated with Joint Development Activities shall be borne in accordance with Section 8.2(a).  

(e)

Second Indication Opt-Out and Second Indication Opt-In.  

(i)

Second  Indication  Opt-Out.  If  Licensee  determines,  at  its  sole  and  absolute  discretion,  within
[***], not to pursue further additional Development activities with respect to the Second Indication, Licensee shall have the right to exercise
the Second Indication Opt-Out, exercisable by written notice to Ovid. The Second Indication Opt-Out shall be effective as of the date of such
notice.  If  Licensee  exercises  the  Second  Indication  Opt-Out,  then  the  definition  of  Field  shall  automatically  be  deemed  to  not  include  the
Second Indication, provided that if Ovid undertakes to submit an MAA for the Product for the Second Indication in the Licensee Territory it
shall do so with a trademark other than the Trademark for the Initial Indication.

Second Indication Opt-In. In any case, after Licensee has made the Second Indication Opt-Out,
Licensee will have the right, at any time as below and for any reason, to exercise the Second Indication Opt-In, exercisable by written notice
to Ovid [***]. The Second

(ii)

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or confidential.

 
Indication  Opt-In  shall  be  effective  as  of  the  date  of  such  notice.    If  Licensee  makes  the  Second  Indication  Opt-In,  then  Licensee  shall
reimburse  to  Ovid  an  amount  equal  to  [***]  of  all  Development  Costs  incurred  by  Ovid  in  the  conduct  of  Development  activities  for  the
Second  Indication  during  the  period  of  Licensee’s  Second  Indication  Opt-Out,  and  [***]  of  all  Development  Costs  incurred  for  such
Development  activities  following  the  Second  Indication  Opt-In.  Then  the  definition  of  Field  shall  automatically  be  deemed  to  include  the
Second Indication

(f)

Regulatory  Filings.    The  Development  Plan  shall  include  a  coordinated  Development  and  regulatory
strategy, including the Parties’ respective roles in the development of the registration dossier and Regulatory Filings for the Products, and the
countries in which Clinical Trials of the Products will occur.  All costs associated with regulatory activities in connection with Regulatory
Filings and obtaining MAA Approval for Products in the Licensee Territory shall be borne solely by Licensee.

(g)

Updates. During the Term (at least on a [***] basis), the JPT shall review the Development Plan and prepare
updates and amendments, as appropriate, to the then-current Development Plan, including budgets, and submit such updates and amendments
to the CGB for review and approval.  If the CGB determines that any pre-clinical studies or Clinical Trials not included in the Development
Plan  are  required  in  order  to  obtain  or  maintain  MAA  Approval  for  a  Product  for  the  Initial  Indication  in  one  or  more  countries  in  the
Licensee  Territory,  then  the  CGB  shall  review  and  approve  an  amendment  to  the  Development  Plan  reflecting  such  additional  studies,
including associated budget.  Such additional Development activities for the Initial Indication shall be either Licensee Territory Development
Activities or Joint Development Activities and the costs of such additional studies shall be borne by the Parties as provided in Section 4.5(a).

4.3

Additional Indications.  

(a)

Proposal.  If either Party (the “Proposing Party”) desires to pursue additional Development of a Product in
order to seek Regulatory Approval of the Product in one or more Additional Indications for the benefit of (a) the Ovid Territory and Licensee
Territory in the case of Ovid, or (b) the Licensee Territory in the case of Licensee, in each case beyond what is set forth in the then-current
Development Plan, then such Party shall provide the other Party (the “Reviewing Party”) with a written detailed plan and budget for such
additional work (the “Proposal”).  Within [***] after the Reviewing Party’s receipt of the Proposal (or at such other time as the Parties may
mutually agree), the JPT shall meet to review and discuss in good faith the Proposal and permit the Reviewing Party an opportunity to ask
questions and request additional information from the Proposing Party related to the Proposal, including whether such Proposal is reasonably
likely to have any adverse effect on the Development or Commercialization of the Product in the Reviewing Party’s territory.  No work under
any Proposal shall proceed unless and until (i) the CGB determines in its reasonable discretion that such Proposal is not likely to adversely
affect  the  Development  or  Commercialization  of  the  Product  in  the  Reviewing  Party’s  territory,  and  (ii)  in  the  case  of  Licensee  as  the
Proposing Party, Ovid consents in writing to such activities being included as Joint Development Activities, or to Licensee performing such
additional Development as Licensee Territory Development Activities (where such Development Activities solely and specifically relate to
the Licensee Territory), or as Independent Development Activities, such consent not to be unreasonably withheld.  For clarity, (i) Licensee’s
final decision

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or confidential.

 
right  under  Section  3.4(b)(ii)  shall  not  apply  to  Licensee  Territory  Development  Activities  proposed  in  connection  of  initiation  of
Development for any Additional Indication, but once Development Activities have been commenced in such Additional Indication in and for
the Licensee Territory, any further Licensee Territory Development Activities proposed by Licensee in respect of such Additional Indication
shall be subject to the process set forth in Section 4.2(b) and (ii) Ovid will not develop in the Licensee Territory any Product in additional
indications other than Rare Diseases without Licensee’s prior written consent. Following each such determination and, if applicable, consent,
the CGB shall incorporate such additional Development activities and the corresponding budget into the Development Plan (the “Additional
Development Activities”).  

(b)

Costs.    If  the  Parties  jointly  agree  to  conduct  Additional  Development  Activities,  such  Additional
Development Activities shall be included in the Development Plan and conducted as Joint Development Activities, subject to the allocation
of responsibility for leading such activities set forth in Section 4.3(c), and the costs of such Joint Development Activities shall be shared as
further  set  forth  in  Section  8.2(a).    Notwithstanding  the  foregoing,  for  Additional  Development  Activities  that  would  otherwise  be  Joint
Development Activities (if the Parties agreed to conduct such activities together), the Reviewing Party may elect, at its discretion, and by
written  notice  delivered  to  the  Proposing  Party  within  [***]  following  the  receipt  of  the  Proposal,  to  opt  out  of  funding  its  share  of  the
Development Costs for such Additional Development Activities.  Upon such an election, such Additional Development Activities shall be
deemed the “Independent Development Activities” of the Proposing Party and the Proposing Party may pursue such work subject to the
remainder of this Section 4.3, and the Development Costs with respect thereto shall be Independent Development Costs subject to Section
8.2(b).  

(c)

Conduct  of  Additional  Development  Activities.    In  general,  except  as  the  Parties  may  agree  in  an
amendment to the Development Plan, including to allocate specific activities to Licensee in the Licensee Territory, (i) Ovid shall be the lead
Party responsible for conducting Additional Development Activities that relate to both the Ovid Territory and the Licensee Territory, provided
that such activities shall be subject to the oversight of the CGB to the extent such activities impact the Licensee Territory, and (ii) Licensee
shall be the lead Party responsible for conducting Additional Development Activities that relate to the Licensee Territory and not the Ovid
Territory.  

(d)

Independent  Development  Activities.    The  CGB  shall  amend  the  Development  Plan  to  include  any
Additional  Development  Activities  in  the  Rare  Diseases  indications  that  are  Independent  Development  Activities,  and  thereafter  the
Proposing Party may conduct such Independent Development Activities, provided that: (i) the Proposing Party shall have the right to make
the  final  decision  in  the  event  of  any  dispute  regarding  the  conduct  of  the  Independent  Development  Activities,  except  to  the  extent  that,
where  the  Proposing  Party  is  Licensee,  Ovid  reasonably  believes  that  Licensee’s  exercise  of  such  right  would  adversely  impact  Ovid’s
Development and Commercialization of Products outside the Licensee Territory, (ii) the Proposing Party shall have the right to make the final
decision in the event of any dispute regarding the conduct of the Independent Development Activities, except to the extent that, where the
Proposing Party is Ovid, Licensee reasonably believes that Ovid’s exercise of such right would adversely impact Licensee’s Development and
Commercialization of Products in the Licensee Territory, (iii) to the extent applicable to the Licensee Territory, Independent Development
Activities shall be conducted in accordance with the amended Development Plan, (iv) the

29
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or confidential.

 
Proposing Party shall provide updates to the CGB with respect to such Independent Development Activities impacting the Licensee Territory
at  each  regularly  scheduled  CGB  meeting,  and  (v)  neither  Party  shall  conduct  any  Independent  Development  Activities  in  a  manner  that
would have any adverse effect on the Development or Commercialization of the Product in either Party’s territory. The Investigator initiated
trials (IIT) proposed to each Party for the Licensee Territory shall be discussed and agreed between the Parties before providing feedback to
the  proposing  Investigator.  The  Party  receiving  the  proposal  will  be  responsible  for  the  costs  to  support  the  IIT  unless  a  different  specific
agreement is entered among the Parties. For sake of clarity, Independent Development Activities shall not include indications other than Rare
Disease.

(e)

Ovid’s  Right  to  Develop.    Notwithstanding  anything  to  the  contrary  herein,  Ovid  shall  have  the  right  to
conduct any Development activities with respect to the Compound or Product in or relating to the Ovid Territory outside the scope of the
Development Plan.  Such Development activities shall be at Ovid’s expense and Licensee shall have the right of reference to the Safety Data
generated in such Development activities as necessary for regulatory purposes without any reimbursement obligation to Ovid.

4.4

Annual  Update  to  Development  Budget.    The  CGB  shall  review,  discuss,  and,  with  respect  to  Joint  Development

Activities, agree upon the subsequent year’s Development Budget on an annual basis no later than [***] of each year.  

4.5

Development Costs.

Licensee  Territory  Development  Costs.    Licensee  shall  be  solely  responsible  for  all  Development  Costs
incurred in connection with Licensee Territory Development Activities, except as provided in Section 4.2(c)(ii) with respect to the Additional
Pivotal Study.

(a)

Joint Development Costs.  The Development Costs associated with all Joint Development Activities that are
shared  by  the  Parties  in  accordance  with  Section  8.2(a)  shall  include  Allowable  Increases.  “Allowable  Increases”  means  increased
Development Costs resulting from [***].

(b)

Section 4.3 shall be solely responsible for all Independent Development Costs as provided in Section 8.2(b).

(c)

Independent Development Costs.   The  Party  conducting  Independent  Development  Activities  pursuant  to

4.6

Development Responsibilities.  Ovid shall be responsible for, and shall use Ovid Commercially Reasonable Efforts in
connection  with,  the  conduct  of  the  Ovid  Ongoing  Trials.    Licensee  shall  be  responsible  for  the  conduct  of  the  Licensee  Territory
Development Activities, other than Additional Pivotal Study which shall be shared by the Parties as set forth in Section 4.2(c)(ii).  The Parties
shall  each  be  responsible  for  the  conduct  of  the  Joint  Development  Activities,  and  the  allocation  of  such  agreed  responsibility  therefore
(including which Party shall be the Sponsor for each applicable Clinical Trial), shall be set forth in the Development Plan.  Each Party shall
have the operational responsibility and be the Sponsor for its own Independent Development Activities.

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or confidential.

 
4.7

Data Exchange and Use.  

General. With respect to all Joint Development Activities, Licensee Territory Development Activities, and
Independent Development Activities (but subject to Section 4.7(c)), each Party shall promptly provide the other Party with [***].  The Parties
shall cooperate [***] to facilitate the sharing of reports, Data, and other information on a routine basis.  

(a)

(b)

Joint Development Activities Data.  Each Party shall have the right to use and reference, without additional
consideration,  any  and  all  Data  generated  by  or  on  behalf  of  the  other  Party  (including  by  any  Sublicensee)  in  the  performance  of  Joint
Development  Activities  for  obtaining  and  maintaining  Regulatory  Approval  for  the  Products  and  Commercializing  the  Products  in  its
territory in accordance with the terms of this Agreement.  Notwithstanding the foregoing, should Licensee fail to obtain the foregoing use and
reference rights from any Sublicensee, Licensee shall not have the right to grant use and access or other rights to such Sublicensee to any
Data or other documentation provided to Licensee by Ovid pursuant to Section 4.7(a).  

(c)

Independent  and  Licensee  Territory  Development  Activities  Data.    The  Party  receiving  Data  resulting
from the other Party’s Independent Development Activities shall have the right to use such Data only to the extent reasonably necessary for
the receiving Party to comply with its regulatory reporting and compliance obligations, including safety reporting obligations.  Licensee shall
have the right to use such Data only to support its own Development, Regulatory Approval, or Commercialization of the Product in the Field
in  such  Party’s  territory  for  the  Initial  Indication  unless  Licensee  reimburses  Ovid  for  Licensee’s  share  of  Development  Costs  pursuant  to
Section 8.2(b). Ovid shall have the right to use Data resulting from the Licensee Territory Development Activities as necessary for Ovid or its
Affiliates or licensees (other than Licensee) to comply with its regulatory reporting and compliance obligations, including safety reporting
obligations, and to support its own Development, Regulatory Approval, or Commercialization of the Product in the Ovid Territory.

(d)
laws of the EU and USA.

Any  data  transfer  between  the  Parties  under  this  Agreement  shall  comply  with  the  applicable  data  privacy

4.8

Diligence.  Each Party shall use its Commercially Reasonable Efforts to perform the Development activities assigned to
such  Party  under  and  in  accordance  with  the  Development  Plan  and  the  Amended  Development  Plan.  In  addition,  Licensee  shall  use
Commercially  Reasonable  Efforts  to  perform  any  Independent  Development  Activities  of  Licensee,  and  Licensee  Territory  Development
Activities and file MAAs and seek and maintain Regulatory Approval (including Pricing and Reimbursement Approval, as applicable) for the
Products throughout the Licensee Territory.

4.9

Compliance.  Each Party shall perform Development activities for the Compound and Products in and for the Licensee
Territory in compliance with all Applicable Laws, including good scientific and clinical practices under the Applicable Laws of the country in
which such activities are conducted.

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or confidential.

 
4.10

Development  Records.    Each  Party  shall  maintain  complete,  current,  and  accurate  records  of  all  Development
activities conducted by it hereunder, and all data and other information resulting from such activities.  Such records shall fully and properly
reflect  all  work  done  and  results  achieved  in  the  performance  of  the  Development  activities  in  good  scientific  manner  appropriate  for
regulatory and patent purposes.  Each Party shall document all non-clinical studies and Clinical Trials and/or Studies in formal written study
reports according to Applicable Laws and national and international guidelines (e.g., ICH, GCP, GLP, and GMP).    

4.11

Development  Reports.    At  each  regularly  scheduled  JPT  meeting,  each  Party  shall  provide  the  JPT  with  regular
reports detailing its Development activities for the Products under this Agreement, and the results of such activities.  In addition, after the
completion  of  any  Clinical  Trial  or  other  study  of  the  Products,  the  Party  responsible  for  the  conduct  of  such  Clinical  Trial  or  study  shall
promptly  provide  the  other  Party  with  a  data  package  consisting  of,  at  a  minimum,  [***],  as  well  as  any  other  Data  specified  in  the
Development Plan or otherwise agreed by the Parties.  The Parties shall discuss the status, progress, and results of each Party’s Development
activities under this Agreement at such JPT meetings.

4.12

Use  of  Subcontractors.  Each  Party  may  perform  its  Development  activities  under  this  Agreement  through  one  or
more subcontractors, provided that (a) such Party will remain responsible for the work allocated to, and payment to, such subcontractors to
the same extent it would if it had done such work itself, (b) each subcontractor undertakes in writing obligations of confidentiality and non-
use  regarding  Confidential  Information  that  are  substantially  the  same  as  those  undertaken  by  the  Parties  pursuant  to  Article 13,  (c)  each
subcontractor agrees in writing to assign all intellectual property developed in the course of performing any such work to such Party (or, in
the event such assignment is not feasible, a license to such intellectual property with the right to sublicense to such other Party), and (d) in the
case of Licensee engaging any subcontractor to conduct significant activities under this Agreement (e.g., a contract research organization to
manage a Clinical Trial), Licensee will be responsible for the selection of the subcontractor and will inform Ovid on the selection process
including  the  criteria  applied  and  shall  first  obtain  Ovid’s  written  consent  to  such  subcontractor,  such  consent  not  to  be  unreasonably
withheld.  The Parties may also subcontract work on terms other than those set forth in this Section 4.12 with the prior approval of the CGB.

4.13

Restrictions.  During  the  Term,  neither  Party  nor  any  of  its  Affiliates  or  Sublicensees  shall,  directly  or  through  any
Third Party, sponsor, conduct, cause to be conducted, otherwise assist in, supply any Product for use in connection with, or otherwise fund
any research or Development of any Product in the Licensee Territory outside the scope of the Development Plan.  For clarity and without
limiting the foregoing, if Licensee wishes to perform or sponsor any study or test on the Compound or Products, including any pre-clinical or
non-clinical  study,  toxicology  study,  CMC-related  study,  or  comparator  study,  Licensee  shall  first  prepare  and  provide  to  Ovid  for  Ovid’s
approval a Proposal detailing such study in accordance with Section 4.3.

4.14

Materials Transfer.    In  order  to  facilitate  the  Development  activities  contemplated  by  this  Agreement,  either  Party
may  provide  to  the  other  Party  certain  biological  materials  or  chemical  compounds  Controlled  by  the  supplying  Party  (collectively,
“Materials”)  for  use  by  the  other  Party  in  furtherance  of  such  Development  activities.    Except  as  otherwise  provided  for  under  this
Agreement, all such Materials delivered to the other Party will remain the sole property of the

32
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or confidential.

 
supplying Party, and will be used only in furtherance of the Development activities conducted in accordance with this Agreement, will not be
used or delivered to or for the benefit of any Third Party, except to subcontractors, without the prior written consent of the supplying Party,
and will be used in compliance with all Applicable Laws.  The Materials supplied under this Agreement must be used with prudence and
appropriate  caution  in  any  experimental  work  because  not  all  of  their  characteristics  may  be  known.    Except  as  expressly  set  forth  in  this
Agreement, THE MATERIALS ARE PROVIDED “AS IS” AND WITHOUT ANY REPRESENTATION OR WARRANTY, EXPRESS OR
IMPLIED,  INCLUDING  WITHOUT  LIMITATION  ANY  IMPLIED  WARRANTY  OF  MERCHANTABILITY  OR  OF  FITNESS  FOR
ANY PARTICULAR PURPOSE OR ANY WARRANTY THAT THE USE OF THE MATERIALS WILL NOT INFRINGE OR VIOLATE
ANY PATENT OR OTHER PROPRIETARY RIGHTS OF ANY THIRD PARTY.

4.15

Suspension  and  Termination  for  Safety  Reasons.  Each  Party  shall  have  the  right,  at  any  time,  to  request  that  the
CGB meet promptly to discuss whether to suspend the continued Development and/or Commercialization of the Products in the Field in the
Licensee  Territory  for  a  period  of  [***]  (the  “Suspension”),  upon  providing  written  notice  to  the  other  Party,  if  such  Party  reasonably
determines in good faith that the Compound or any other Product caused or is likely to cause a safety issue (a “Safety Reason”).  If the CGB
does not come to a consensus with regard to such Safety Reason during the Suspension, either Party may terminate the Agreement (with the
understanding that the other Party shall have the continuing right to Develop and Commercialize the Product; provided, however, that if the
other Party is Licensee and Licensee wishes to continue the Development and Commercialization of the Product, this Agreement shall remain
in force and effect, but the provisions of Section 14.5  shall  apply)  with  immediate  effect,  upon  written  notice  to  the  other  Party  if:  (i)  the
Executive Officers meet (in person or otherwise) within [***] to resolve the dispute in good faith; and (ii) such Executive Officers are unable
to resolve the dispute.

5.

REGULATORY ACTIVITIES

5.1

Regulatory Responsibilities.  

(a)

General.  

(i)

The Development Plan shall set forth the regulatory strategy for seeking Regulatory Approval for
the Compound and Products by the appropriate Regulatory Authorities in the Licensee Territory and Ovid Territory.  Subject to the oversight
of  the  CGB  and  except  as  otherwise  set  forth  in  the  Development  Plan  and  the  remainder  of  this  Section  5.1(a)(i),  each  Party  shall  be
responsible for implementing such regulatory strategy in its territory.  The Development Plan shall also specify which Party shall apply for
and hold Regulatory Filings in each country with respect to the conduct of Development activities, provided that (1) Ovid shall apply for and
hold all Regulatory Filings and Regulatory Approvals for the Ovid Ongoing Trials and Ovid’s Independent Development Activities and (2)
Licensee  shall  apply  for  and  hold  all  Regulatory  Filings  for  the  Licensee  Territory  arising  from  the  Licensee  Territory  Development
Activities, Licensee’s Independent Development Activities, and Joint Development Activities.  Except as otherwise provided herein or in the
Development  Plan  or  required  by  Applicable  Law,  each  Party  shall  (A)  be  responsible  for  the  preparation  and  submission  of  any  and  all
Product

33
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or confidential.

 
registrations  and  MAAs  in  its  territory  and  (B)  own  and  hold  all  such  Regulatory  Filings  (including  Regulatory  Approvals).    For  the
avoidance of doubt, in no event shall Licensee submit any Regulatory Filing for the Product in the Ovid Territory.  

Each Party shall be responsible for the costs of all regulatory activities in its territory, except that
any costs incurred by Ovid in connection with regulatory activities in the Licensee Territory pursuant to Ovid’s Independent Development
Activities shall be Independent Development Costs of Ovid and subject to Section 8.2(b).  

(ii)

Licensee  acknowledges  that  Ovid  may  be  required  from  time  to  time  to  communicate  with
Regulatory Authorities in the Licensee Territory as a result of Development and manufacturing activities in such territory. Ovid shall notify
Licensee as soon as reasonably practicable of such communication with Regulatory Authorities in the Licensee Territory.

(iii)

[***] for the Product for the Initial Indication [***] under this Agreement.

(iv)

Ovid  will  provide  to  Licensee  [***].  Licensee  shall  have  the  right  to  use  such  information  to

(v)

Prior to [***], Ovid will not, without Licensee’s input, (A) withdraw the IND for the Product in
the Licensee Territory for any reason other than a Safety Reason, (B) file an MAA for the Product in the Licensee Territory, or (C) finalize the
PIP  for  the  Initial  Indication.    Prior  to  [***],  Ovid  shall  notify  Licensee  of  any  scheduled  meeting  with  a  Regulatory  Authority  in  the
Licensee  Territory  that  relates  to  the  any  of  the  Ovid  Ongoing  Trials  and,  to  the  extent  permitted  by  Applicable  Law  and  the  relevant
Regulatory Authority, shall permit a representative of Licensee to attend such meeting, at Licensee’s request and expense.  

Initial Indication in the Licensee Territory.

(vi)

Ovid will,  upon  Licensee’s  reasonable  request,  cooperate  with  Licensee  in  [***]  Product  in  the

Advice with the applicable Regulatory Authorities in the Licensee Territory.

(vii)

Ovid shall [***] for the Compound [***].  Licensee shall have the right to perform a Scientific

(b)

Regulatory Filing Right of Reference.  Except as set forth in Section 5.1(c), Ovid shall grant and hereby
grants to Licensee a right of reference and access to all Regulatory Approvals and Regulatory Filings Controlled by Ovid in the Licensee
Territory for the Compound and Product, in each case to the extent necessary  for  Licensee  to  submit  Regulatory  Filings  and  obtain  MAA
Approvals for Products in the Initial Indication in the Licensee Territory.  For the purposes of this Agreement, “right of reference” means the
“right of reference or use” as defined in 21 C.F.R. §314.3(b) and any equivalent regulation outside the U.S., as each may be amended.

(c)

Licensee Regulatory Information Sharing and Right of Reference.  

Licensee shall promptly provide Ovid with copies of any Regulatory Filings prepared (including
any drafts), submitted, or received by Licensee in the Licensee Territory pertaining to the Compound and Products, and Ovid shall have the
right to comment on

(i)

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or confidential.

 
drafts  of  such  Regulatory  Filings.    Licensee  shall  share  with  Ovid  the  following  communications/correspondence  with  any  Regulatory
Authority: (1) [***], (2) [***], and (3) [***] relating to the Compound or Product.  If any Regulatory Filing to be provided under this Section
5.1(c) was originally created in a language other than the English language, then Licensee shall provide an English translation along with the
original  document  to  Ovid.    Licensee  shall  use  Commercially  Reasonable  Efforts  to  grant  to  Ovid  access  and  rights  to  use  any  such
communications with any Regulatory Authority generated by or on behalf of any Sublicensee.  Should Licensee fail to obtain such access and
rights from any Sublicensee despite the application of Commercially Reasonable Efforts, Licensee shall not have the right to grant access or
rights to such Sublicensee to any Regulatory Filing or right of reference granted to Licensee by Ovid pursuant to Section 5.1(b).

(ii)

Licensee  hereby  grants  to  Ovid  a  right  of  reference  to  all  Regulatory  Filings  for  the  Compound
and Products submitted by or on behalf of Licensee.  Ovid may use such right of reference to seek, obtain, and maintain Regulatory Approval
of the Products in the Ovid Territory, except that Ovid may use such right of reference to any Regulatory Filings based on Data resulting from
Licensee’s  Independent  Development  Activities  only  to  comply  with  its  safety  reporting  obligations,  unless  Ovid  reimburses  Licensee  for
such work as set forth in Section 8.2(b).

5.2

Meetings with Regulatory Authorities.  On a current and ongoing basis, each Party (through the JPT) shall provide
the other Party with a list and schedule of any in-person meeting or material teleconference with Regulatory Authorities (or related advisory
committees)  in  the  Licensee  Territory  planned  for  [***]  that  relates  to  the  Development  of  the  Compound  and  Products  under  the
Development Plan in the Licensee Territory (each, a “Regulatory Meeting”).  In addition, each Party shall notify the other Party as soon as
reasonably possible if such Party becomes aware of any additional Regulatory Meetings that become scheduled for such Calendar Quarter
and  will  keep  the  other  Party  informed  of  any  significant  interface  or  communication  with  any  Regulatory  Authority  which  might  affect
efforts  to  obtain  Regulatory  Approval  for  the  Product  in  the  Licensee  Territory.  Each  Party  shall  be  solely  responsible  for  any
communications with any Regulatory Authorities occurring or required in connection with performing its regulatory responsibilities set forth
in  this  Article  5  with  respect  to  the  Product  in  the  Licensee  Territory.  With  respect  to  Regulatory  Meetings  for  which  Licensee  is  the
responsible Party, Ovid shall have the right to comment in preparation for all such Regulatory Meetings and the right, but not the obligation,
to have its representatives attend any such Regulatory Meetings.

5.3

Regulatory  Inspections.    Licensee  shall  permit  the  Regulatory  Authority(ies)  in  the  Ovid  Territory  to  conduct
inspections of Licensee, its Affiliates, and its Sublicensees and subcontractors (including Clinical Trial sites) relating to the Development of
the  Product  under  the  Development  Plan,  and  shall  ensure  that  such  Affiliates  and  Sublicensees  and  subcontractors  permit  such
inspections.  In addition, Licensee shall promptly notify Ovid of any such inspection and shall supply Ovid with all information pertinent
thereto.  Ovid shall have the right to have a representative attend any such inspection. Ovid shall permit the Regulatory Authority(ies) in the
Licensee Territory to conduct inspections of Licensee, its Affiliates, and its Sublicensees and subcontractors (including Clinical Trial sites)
relating to the Development of the Product in the Licensee Territory under the Development Plan, and shall ensure that such Affiliates and
Sublicensees and subcontractors permit such inspections.  In addition, Ovid shall promptly notify the Licensee of any such inspection in the
Licensee Territory and shall supply the Licensee with

35
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
all information pertinent thereto.  The Licensee shall have the right to have a representative attend any such inspection.

5.4

Adverse Event Reporting; Pharmacovigilance Agreement.  [***] after the Effective Date, the Parties shall enter into
a pharmacovigilance agreement setting forth the worldwide pharmacovigilance procedures for the Parties with respect to the Products, such
as  Safety  Data  sharing,  adverse  event  reporting,  and  safety  signal  and  risk  management  (the  “Pharmacovigilance  Agreement”),  which
agreement shall be amended by the Parties from time to time as necessary to comply with any changes in Applicable Laws or any guidance
received  from  Regulatory  Authorities.    Such  procedures  shall  be  in  accordance  with,  and  enable  the  Parties  to  fulfill,  local  and  national
regulatory reporting obligations under Applicable Laws (including, to the extent applicable, those obligations contained in ICH guidelines) to
monitor patients’ safety.  Ovid has established, and shall continue to hold (either by itself or through a vendor engaged by Ovid) the global
safety  database  for  the  Products,  and  shall  maintain  such  global  safety  database  for  so  long  as  such  Product  is  under  Development  or
Commercialization by the Parties.  The Parties envision that Ovid will separately maintain the Product global safety database and Licensee
will maintain its own Product safety database with respect to the Licensee Territory and the Parties will synchronize the Product databases in
accordance  with  the  Pharmacovigilance  Agreement  so  that  they  each  maintain  all  Product  safety  data;  however,  the  Parties  agree  that  the
Ovid global safety database will be the source for all periodic reports. Ovid shall [***] from its database and Licensee will maintain [***] its
own Product safety database. The CGB shall establish a safety subcommittee to draft the Pharmacovigilance Agreement to define the process
for exchanging adverse event reports using the Ovid global safety database, as well as periodic reports, regulatory communication, and other
key elements.  The Parties will collaboratively agree on data cut points for periodic safety reports and Ovid will review and approve all such
reports.  The Parties will jointly review and approve such reports before submission to Regulatory Authorities in the Licensee Territory as
required.    Such  safety  subcommittee  shall  implement  the  Pharmacovigilance  Agreement  and  coordinate  with  respect  to  any  Safety  Data
reporting for the Products to the Regulatory Authorities in the Licensee Territory including,  responding to safety issues, communicating with
Regulatory Authorities related to the Products under any MAA or Regulatory Approval for the Product held by such Party and filed with such
Regulatory  Authorities,  including  maintaining  the  qualified  person  for  Pharmacovigilance  and  individual  case  safety  report  processing,  in
each case at its own cost. Each Party agrees to comply with its respective obligations under the Pharmacovigilance Agreement and to cause
its Affiliates, licensees, and Sublicensees to comply with such obligations.

5.5

No Harmful Actions.  If a Party reasonably believes that the other Party is taking or intends to take any action with
respect to a Product that could reasonably be expected to have a material adverse impact upon the regulatory status of such Product in such
Party’s  territory,  then  such  Party  may  bring  the  matter  to  the  attention  of  the  CGB  and  the  Parties  shall  discuss  in  good  faith  to  promptly
resolve such concern.  

5.6

Notification  of  Threatened  Action.    Each  Party  shall  notify  the  other  Party  within  twenty-four  (24)  hours  of  any
information it receives regarding any threatened or pending action, inspection, or communication by any Regulatory Authority which may
affect the safety or efficacy claims of any Product or the continued Development or Commercialization of any Product.  Upon

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Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
receipt of such information, the Parties shall promptly consult with each other in an effort to arrive at a mutually acceptable procedure for
taking appropriate action.  

5.7

Recalls.  In the event that a recall, withdrawal, or correction (including the dissemination of relevant information) of
any Product in a Party’s territory is required by a Regulatory Authority of competent jurisdiction, or if any Regulatory Authority requires or
advises  either  Party  or  such  Party’s  Affiliates  or  sublicensees  to  distribute  a  “Dear  Doctor”  letter  or  its  equivalent  regarding  use  of  such
Product in a Party’s territory, or if a recall, withdraw, or correction of a Product in its territory is deemed advisable by such Party in its sole
discretion, such Party shall so notify the other Party no later than [***] in advance of the earlier of (a) [***], or (b) [***].  Any such recall,
withdrawal, correction, or dissemination of information (e.g., “Dear Doctor” letter) shall be referred to herein as a “Recall”.  Promptly after
being notified of a Recall, each Party shall provide the other Party with such assistance in connection with such Recall as may be reasonably
requested by such other Party.  All costs and expenses in connection with a Recall [***].  Each Party shall handle exclusively the organization
and  implementation  of  all  Recalls  of  Products  in  its  territory.    Notwithstanding  the  foregoing,  any  Recall  related  to  the  manufacture  and
supply of the Product by Ovid to Licensee shall be governed by the terms and conditions of the Supply Agreement.

5.8

Sunshine Reporting Laws and the International Transparency Reporting Requirements for Europe.  Each Party
acknowledges that the other Party may be subject to federal, state, local, and international laws, regulations, and rules related to the tracking
and  reporting  of  payments  and  transfers  of  value  provided  to  health  care  professionals,  health  care  organizations,  and  other  relevant
individuals  and  entities,  including,  as  applicable,  International  Transparency  Reporting  Requirements  for  Europe  (collectively,  “Sunshine
Reporting Laws”), and agrees to provide the other Party with all information regarding such payments or transfers of value by such Party as
necessary for such other Party to comply in a timely manner with its reporting obligations under the Sunshine Reporting Laws.    

6.

COMMERCIALIZATION

6.1

General.  Subject to the terms and conditions of this Agreement, including this Article 6, Licensee shall have the sole
and exclusive responsibility, at its own expense, for all aspects of the Commercialization of the Products in the Licensee Territory, including
(a) developing and executing a commercial launch and pre-launch plan, (b) negotiating with applicable Governmental Authorities and other
payors  regarding  the  price  and  reimbursement  status  of  the  Products,  (c)  marketing  and  promotion,  (d)  booking  sales  and  distribution  and
performance of related services, (e) handling all aspects of order processing, invoicing and collection, inventory and receivables, (f) providing
customer  support,  including  handling  medical  queries,  and  performing  other  related  functions,  and  (g)  conforming  its  practices  and
procedures  to  Applicable  Laws  applying  to  the  promotion,  sales  and  marketing,  access,  and  distribution  of  the  Products  in  the  Licensee
Territory.  

6.2

Commercialization  Plan.    As  soon  as  reasonably  practicable,  but  no  later  than  [***],  Licensee  shall  prepare  and
present to the CGB a reasonably detailed plan for the Commercialization of the Product in the Licensee Territory (the “Commercialization
Plan”).  The Commercialization Plan will include specific information on a country-by-country basis, as

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or confidential.

 
applicable, and shall be consistent with the global commercialization plan for branding and messaging.  Licensee shall update and amend the
Commercialization Plan [***] following the First Commercial Sale of the Product in the Licensee Territory and present such updates and any
amendments to the CGB for review and discussion.  Subject to the terms of this Agreement and compliance with the Commercialization Plan,
Licensee shall have full Control and authority with respect to the day-to-day Commercialization of the Products and implementation of the
Commercialization Plan.

6.3

 Diligence.  

Products for each and every Indication that receives Regulatory Approval in the Licensee Territory.  

(a)

General.    During  the  Term,  Licensee  shall  use  Commercially  Reasonable  Efforts  to  Commercialize  the

(b)

Product Launch.  Licensee shall use Angelini Commercially Reasonable Efforts to launch the Product for
each  Indication  that  has  received  Regulatory  Approval  and,  if  required  by  Applicable  Law,  Pricing  and  Reimbursement  Approval  in  the
Licensee Territory (including any Indication that received Regulatory Approval as a result of Ovid’s Independent Development Activities).
As applicable, Licensee shall obtain all necessary Pricing and Reimbursement Approvals necessary to list and to launch such Product for such
Indication following receipt of MAA Approval of such Product in a country.  Without limiting the generality of the foregoing, Licensee shall
use Angelini Commercially Reasonable Efforts to launch the Product in each country in the Licensee Territory within [***] after receiving
Regulatory Approval, or, where required by Applicable Law, after the publication of the Pricing and Reimbursement Approval, of the Product
for  an  Indication  from  the  applicable  Regulatory  Authority  in  such  country.    Thereafter,  Licensee  shall  utilize  Commercially  Reasonable
Efforts in the ongoing support for such Product in such country.

(c)

Commercial  Updates.    Licensee  shall  update  the  CGB  on  [***]  basis  regarding  its  Commercialization
activities  with  respect  to  the  Products  in  the  Licensee  Territory.    Each  such  update  shall  be  in  a  form  to  be  agreed  by  the  CGB  and  shall
summarize  Licensee’s  and  its  Affiliates’  and  Sublicensees’  significant  Commercialization  activities  with  respect  to  the  Products  in  the
Licensee  Territory,  and  shall  contain  at  least  such  information  at  a  level  of  detail  reasonably  required  by  Ovid  to  determine  Licensee’s
compliance with its diligence obligations set forth in this Section 6.3.  Such updates shall include Licensee’s sales activities, sales forecasts
for at least the next [***], marketing activities, and Medical Affairs Activities.

6.4

Coordination of Commercialization Activities.

(a)

Generally.    The  Parties,  through  the  CGB  (or  JPT  or  other  designated  team),  shall  update  each  other  on
Commercialization strategies for the Product (e.g., for market and payor research, branding and messaging, international congresses, advisory
boards) in their respective territories, and the Parties shall work together to identify and take advantage of any potential global strategies and
messaging.  The foregoing shall not be construed as requiring either Party to seek the other Party’s consent in connection with such first Party
establishing or implementing any sales, marketing, or medical affairs practices in such first Party’s territory.

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or confidential.

 
(b)

Pricing.  Following  the  CGB  discussion  and  processes,  Licensee  shall  keep  Ovid  timely  informed  on  the
status of any application for Pricing and Reimbursement Approval or material updates to an existing Pricing and Reimbursement Approval in
the  Licensee  Territory,  including  any  discussion  with  a  Regulatory  Authority  with  respect  thereto.  Licensee  and  its  Affiliates  and
Sublicensees shall [***] include a Product, [***] of the Product [***] and the Product [***].

(c)

Sharing  of  Promotional  Materials.    Licensee  shall,  at  its  own  expense,  prepare,  develop,  produce,  or
otherwise  obtain  and  utilize  sales,  promotional,  advertising,  marketing,  website,  educational,  and  training  materials  (the  “Promotional
Materials”) to support its Commercialization activities in the Licensee Territory, and shall ensure that such Promotional Materials, as well as
all  information  contained  therein,  comply  with  all  Applicable  Laws  and  are  consistent  with  the  Regulatory  Approvals  obtained  for  the
Product  in  the  applicable  jurisdiction  in  the  Licensee  Territory.    At  Ovid’s  request,  Licensee  shall  share  samples  of  and  updates  to
Promotional Materials with respect to the Commercialization of the Products with Ovid. If Ovid has such promotional materials available for
the Product for the Ovid Territory prior to the commercial launch of such Product in the Licensee Territory, Ovid will share such materials
with the Licensee upon its request.

the Product in the Ovid Territory at its own expense, with or without Third Party(ies).

(d)

Commercialization in Ovid Territory.    For  clarity,  Ovid  shall  have  the  exclusive  right  to  Commercialize

6.5

Medical Affairs Activities.

(a)

Coordination  of  Global  Medical  Affairs  Activities.    Ovid  shall  be  responsible  for  all  Medical  Affairs
Activities for the Product in the Ovid Territory in accordance with the medical affairs portion of the Development Plan.  Licensee shall be
responsible for Medical Affairs Activities in the Licensee Territory in accordance with the medical affairs portion of the Development Plan,
provided, however, that Ovid shall have the right, but not the obligation, to also conduct Medical Affairs Activities in the Licensee Territory
in global support of the Product, consistent with the medical affairs portion of the Development Plan and in coordination and agreement with
Licensee, such agreement not to be unreasonably withheld, conditioned, or delayed.  Licensee will not undertake Medical Affairs Activities
in the Ovid Territory without Ovid’s prior written consent, to be given on a case-by-case basis in Ovid’s sole discretion.

(b)

Advisory Panels.  To the extent practicable, each Party shall give the other Party written notice at least [***]
in advance of any major market or international level advisory panel meetings with key opinion leaders with respect to the Commercialization
of  the  Products  in  the  Licensee  Territory  and  the  Ovid  Territory  that  are  held,  sponsored,  or  attended  by  either  Party  or  its  Affiliate  or
sublicensee, and each Party shall have the right to attend and participate in such meetings with the consent of the other Party.  

Medical  Information.  Ovid  will  provide  Licensee  with  any  relevant  materials  developed  by  Ovid  for  the
Product  in  the  Ovid  Territory  for  medical  information,  including  reports  of  collected  and  answered  inquires,  which  Licensee  may  use  in
connection with

(c)

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or confidential.

 
medical  affairs  activities  in  the  Licensee  Territory.    For  clarity,  Ovid  shall  provide  such  materials  in  the  form  used  by  Ovid  in  the  Ovid
Territory.

Scientific Training.  At  times  reasonably  agreed  by  the  Parties,  Ovid  will  deliver  the  onboarding  scientific
training to Licensee’s medical and commercial team and to share updates with respect to the Commercialization of the Product.  Each Party
shall bear its own cost in relation to such meetings.

(d)

6.6

Diversion.    To  enforce  the  Parties’  respective  rights  and  obligations  set  forth  in  Sections  2.1,  2.4,  and  2.8  of  the
Agreement, to the extent permitted by Applicable Law, each Party hereby covenants and agrees that it and its Affiliates shall not, and it shall
contractually obligate (and use Commercially Reasonable Efforts to enforce such contractual obligation) its sublicensees not to, directly or
indirectly, promote, market, distribute, import, sell, or have sold any Product, including via the Internet or mail order, to any Third Party or to
any  address  or  Internet  Protocol  address  or  the  like  in  the  other  Party’s  territory.    Neither  Party  shall  engage,  nor  permit  its  Affiliates  and
sublicensees to engage, in any advertising or promotional activities relating to any Product for use directed primarily to customers or other
buyers  or  users  of  such  Product  located  in  any  country  or  jurisdiction  in  the  other  Party’s  territory,  or  solicit  orders  from  any  prospective
purchaser located in any country or jurisdiction in the other Party’s territory.  If a Party or its Affiliates or sublicensees receives any order for
a Product for use from a prospective purchaser located in a country or jurisdiction in the other Party’s territory, such Party shall immediately
refer that order to such other Party and shall not accept any such orders.  Neither Party shall, nor permit its Affiliates and sublicensees to,
deliver or tender (or cause to be delivered or tendered) any Product for use in the other Party’s territory.

6.7

Ovid’s  Right  to  Commercialize.    Notwithstanding  anything  to  the  contrary  herein,  if  Ovid  conducts  Development
activities  for  the  Product  in  the  Licensee  Territory  as  provided  in  Section  2.3(a)  for  any  Additional  Indication(s)  for  which  Licensee  has
elected to not share Development Costs as provided in Section 8.2(a) and/or Section 8.2(b), as applicable, then prior to filing for Regulatory
Approval  for  the  Product  in  any  Additional  Indication,  the  Parties  shall  discuss  in  good  faith  whether  Licensee  wishes  to  include  such
Additional Indication within the Field  and to Commercialize such Product in such Additional Indications.  For clarity, neither Party may file
for  Regulatory  Approval  or  Commercialize  Products  in  (i)  any  Additional  Indication  for  which  Licensee  has  elected  not  to  share
Development Costs or (ii) any additional indication other than Rare Diseases unless the Parties mutually agree to do so.

7.

MANUFACTURE AND SUPPLY

7.1

Upon Licensee’s request, Ovid will manufacture and supply, itself or through a Third Party contract manufacturer, all
Drug  Product  for  use  in  the  Development  and  Commercialization  of  the  Products  under  this  Agreement  and  according  to  the  Supply
Agreement.  All Drug Product supplied by Ovid to Licensee or Licensee Affiliate for use for Development and Commercial purposes shall be
supplied at [***], provided that [***] (“Total Supply Price Threshold”). In case the Total Supply Price will be [***], the Cost of Good for
such Drug Product will be [***] the Total Supply Price Threshold.  For clarity, the Total Supply Price Threshold [***].  Payment shall be due
within [***] after Licensee’s receipt from Ovid of an invoice for such Drug Product.  Drug Product shall be delivered EXW (Incoterms 2020)
at supplier facility (or that

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or confidential.

 
of its Third Party contract manufacturer), and Licensee shall be responsible for all costs of freight, insurance, taxes and duties associated with
shipment of Drug Product to Licensee’s designated delivery point.  Licensee shall be responsible, at its expense, for the final packaging and
labeling of the Product for all countries in the Licensee Territory.  Licensee  shall  also  be  responsible,  at  its  sole  expense,  for  any  specific
manufacturing requirements, such as stability studies or development of finished Product presentations, necessary to obtain MAA Approval
of the Product in the Licensee Territory.  If Licensee is manufacturing Drug Product following the Technology Transfer Completion Date,
Ovid may request, and Licensee or Licensee Affiliate will supply Drug Product to Ovid, on the same terms as set forth above, pursuant to a
mutually agreed supply agreement.  

8.

FINANCIAL PROVISIONS

8.1

Upfront and Technology Transfer Financials.  

of twenty million dollars ($20,000,000) within five (5) business days after the Effective Date.

(a)

Upfront Payment.  Licensee shall make a one-time, non-refundable, non‑creditable upfront payment to Ovid

(b)

Technology Transfer and Compound Delivery Payment.

(i)

Within [***] following (A) the transfer to Licensee of [***], (B) the delivery ([***]) to Licensee
or to Licensee Affiliate of [***] and (C) [***], Licensee shall pay to Ovid a one-time, non-refundable, non-creditable payment of (1) five
million dollars ($5,000,000)  if  [***]  is  transferred  by  Ovid  to  Licensee  before  December  10,  2020,  or  (2)  [***]  if  [***].    Licensee  shall  use
Angelini Commercially Reasonable Efforts to cooperate with Ovid and Lundbeck to implement the foregoing transfers within the timelines
set forth in this Section 8.1(b)(i).

Within  [***]  following  the  Technology  Transfer  Completion  Date,  Licensee  shall  make  a  one-
time, non-refundable, non-creditable technology transfer payment of [***]. Licensee shall use Angelini Commercially Reasonable Efforts to
cooperate with Ovid and Lundbeck to implement the Technology Transfer Agreement within [***] after the Effective Date.

(ii)

8.2

Sharing/Reimbursements of Development Costs.

(a)

Shared Development Costs.   With  respect  to  Joint  Development  Activities  conducted  pursuant  to  Section
4.2(b) or Section 4.3 directed to obtaining Regulatory Approval for any Indication, excluding the Ovid Ongoing Trials, Ovid shall bear [***]
and Licensee shall bear [***] of all Development Costs for such Joint Development Activities.  No later than [***] after the beginning of
each Calendar Quarter during which a Party will perform any Joint Development Activities pursuant to Section 4.2(b) or Section 4.3 in such
Calendar Quarter, such Party shall submit to the other Party a statement setting forth the Development Costs incurred, including the other
Party’s  share  (calculated  in  accordance  with  the  foregoing  sentence)  of  (i)  estimated  Development  Costs  for  the  then  current  quarter;  (ii)
variances from prior invoiced estimates and actual Development Costs; and (iii) Development Costs incurred by or on account of such Party
in the past quarter not previously invoiced.  Such invoice shall include a reasonably detailed report for such Development Costs, including
reasonable supporting documents.  The other Party shall

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or confidential.

 
pay the amount invoiced within [***] after the receipt of the invoice, subject to the other Party’s right to audit the invoicing Party’s records
and books related to such costs as provided in Section 9.4.  If both Parties will perform Joint Development Activities pursuant to Section
4.2(b) or Section 4.3  under  the  Development  Plan  in  such  Calendar  Quarter,  the  Parties  shall  consolidate  the  payments  for  such  Calendar
Quarter into a single payment from one Party to the other Party, as applicable.

(b)

Independent Development Costs.  In general, each Party shall bear all Development Costs incurred by or
on account of such Party in performing its own Independent Development Activities (the “Independent Development Costs”).   After  the
completion of such Independent Development Activities, such Party shall provide the other Party (the “Non-Funding Party”) with a report
of such Independent Development Costs.  If a Non-Funding Party desires to submit any portion of the Data, or reference any portion of a
Regulatory Filing, resulting from Independent Development Activities conducted by the other Party to support any Regulatory Approval in
the Non-Funding Party’s territory, then such Non-Funding Party may notify the other Party in writing of such request at any time following
the completion of such Independent Development Activities.  Within [***] after its receipt of such notice, the Party having conducted such
Independent Development Activities shall submit to the other Party a reasonably detailed invoice for, [***] of the Independent Development
Costs  incurred  [***]  in  connection  with  the  performance  of  such  Independent  Development  Activities,  with  such  invoiced  amount
representing the Non-Funding Party’s base share of Development Costs ([***]), had such Party originally opted in, plus [***], provided that
in no event will either Party be required to pay, as a result of the application of such premium, more than [***] the costs actually incurred in
conducting such Independent Development Activities.  If the Non-Funding Party subsequently uses or references such Data, in whole or in
part to support Regulatory Approval of the Product in the applicable Indication in its territory, then such Party shall notify the conducting
Party in writing of such decision and pay the amount set forth in the invoice within [***] after its submission of a Regulatory Filing including
or referencing such Data.

Internal  Development  Cost.  Each  Party  shall  record  and  calculate  its  Development  Costs  for  the
Development Activities implemented from the Effective Date on an FTE basis at the applicable FTE Rate.  The Parties agree that [***] from
the Effective Date.

(c)

8.3

Development Milestone Payments.

Development Milestones.  Subject to the remainder of this Section 8.3, Licensee shall pay to Ovid the one-
time, non-refundable, non-creditable payments set forth in the table below upon the achievement of the applicable milestone event (whether
by or on behalf of Licensee or its Affiliates or Sublicensees or Ovid or its Affiliates or licensee(s) (other than Licensee)).  

(a)

Regulatory Milestone Event

Regulatory Milestone
Amount
[***]

[***]

[***]

[***]

[***]

[***]

[***]

[***]

[***]

[***]

Notice and Payment.  Each Party shall notify the other Party in writing within [***] after the achievement
of any milestone event set forth in this Section 8.3 by such Party or its Affiliates or Sublicensees.  Licensee shall pay to Ovid the applicable
development milestone payment within [***] after the delivery or receipt of such notice.

(b)

how many times the corresponding Regulatory Milestone Event is achieved.  

(c)

One-time Payment. Each of the above Regulatory Milestone amounts shall only be payable once no matter

(d)

For  clarity,  Licensee  shall  pay  to  Ovid  each  Regulatory  Milestone  amount  the  first  time  that  the

corresponding Regulatory Milestone Event is achieved.

8.4

Sales Milestones Payments.  

(a)

Licensee shall pay to Ovid the one-time, non-refundable, non-creditable payments set forth in the table below
when  the  aggregated  Net  Sales  of  all  Products  in  the  Licensee  Territory  in  any  Calendar  Year  first  reach  the  values  indicated  in  the  table
below.  For clarity, each payment in this Section 8.4  shall  be  payable  once  only  upon  first  achievement  of  the  applicable  milestone  event,
regardless of the number of times such milestone is subsequently achieved.

Aggregate Net Sales of all Products in the

Licensee Territory in a Calendar Year

Sales Milestone
Payment Amount

[***]

[***]

[***]

[***]

[***]

[***]

[***]

[***]

[***]

[***]

 
 
42
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

(b)

Notice and Payment.  As part of the report in Section 9.1, Licensee shall provide written notice to Ovid if
the aggregated Net Sales of all Products in the Licensee Territory in any Calendar Year first reach the values set forth in Section 8.4(a), and
Licensee shall pay to Ovid the corresponding Net Sales milestone payment along with its payment of royalties in accordance with Section
9.1, following the end of the Calendar Quarter in which such Net Sales milestone is achieved.

One-time Payment. Each of the above Sales Milestone amounts shall only be payable once during the Term
of this Agreement no matter how many times the corresponding Sales Milestone Event is achieved.  For clarity, Licensee shall pay to Ovid
each Sales Milestone amount the first time that the corresponding Sales Milestone Event is achieved.

(c)

8.5

Royalty During the Royalty Term.

Royalty Rate. Subject to the remainder of this Section 8.5,  during  the  Royalty  Term,  Licensee  shall  make
quarterly non-refundable, non-creditable royalty payments to  Ovid on the annual Net Sales of all Products sold in the Licensee Territory at
the applicable rate to the relevant portion of annual Net Sales as set forth below:

(a)

Annual Net Sales of all Products in the Licensee

Territory

Royalty Rate

Portion of annual Net Sales up to [***]

Portion of annual Net Sales greater than [***] and
less than or equal to [***]

Portion of annual Net Sales greater than [***] and
less than or equal to [***]

[***]%

[***]%

[***]%

Portion of annual Net Sales greater than [***]

[***]%

For example purposes only, [***].

(b)

Royalty Term. Royalties shall be paid on a Product-by-Product and country-by-country basis in the Licensee
Territory from the First Commercial Sale of such Product in such country by or on behalf of Licensee, its Affiliates, or Sublicensees, until the
last to occur of (i) the expiration of the last‑to‑expire Valid Claim of the Ovid Patents (ii) the expiration of all Market Exclusivity covering
such  Product  in  such  country,  and  (iii)  fifteen  (15)  years  after  the  First  Commercial  Sale  of  such  Product  in  such  country    (the  “Royalty
Term”).

(c)

Royalty Stacking Reduction.  If it is necessary for Licensee to obtain a license from a Third Party
under any Patent in a particular country in the Licensee Territory in order to sell the Compound or the Compound incorporated into a Product
for the Initial Indication or, if Licensee does not exercise the Second Indication Opt-Out, the Second Indication in such country and Licensee
obtains such a license, then solely during the Royalty Term, Licensee may

43
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
 
deduct from the royalty payment that would otherwise have been due pursuant to Section 8.5(a) with respect to Net Sales of such Product in
such country in a particular Calendar Quarter an amount equal to [***] of the royalties paid by Licensee to such Third Party pursuant to such
license on account of the sale of such Product in such country during such Calendar Quarter.

Royalty Floor.    Notwithstanding the  foregoing Sections 8.5(c) and Section  8.7  with  respect  to  any
Product in any Calendar Quarter, the royalties that would otherwise have been due under Section 8.5(a)  with  respect  to  Net  Sales  of  such
Product in the applicable country(ies) during such Calendar Quarter shall not be reduced by more than [***] as a result of all such reductions.

(d)

8.6

Royalties During the Extended Commercialization Term.  During the Extended Commercialization Term, Licensee
shall  pay  to  Ovid  a  quarterly  non-refundable,  non-creditable  royalty  of  [***]  on  the  annual  Net  Sales  of  all  Products  sold  in  the  Licensee
Territory, as calculated by multiplying the foregoing royalty rate by the amount of Net Sales of the Product in the Territory in the applicable
Calendar Quarter.

8.7

Royalty Reduction for Generic Competition. If at any time Generic Product Competition exists in a given country
with  respect  to  a  Product,  then  the  royalty  rate  set  forth  in  Section  8.5(a)  with  respect  to  sales  of  such  Product  in  such  country  shall  be
reduced by [***].  For clarity, if Generic Product Competition ceases to exist, then the royalty rate shall no longer be reduced.

8.8

Upstream License Agreement Payments.  Any and all payments that become due under the Lundbeck
License  Agreement  as  a  result  of  activities  under  this  Agreement,  whether  by  or  on  behalf  of  Ovid  or  by  Licensee  or  its  Affiliate  or
Sublicensee, shall be the responsibility of Ovid and Ovid shall make such payment in accordance with the terms of the Lundbeck License
Agreement.

9.

PAYMENT; RECORDS; AUDITS

9.1

Payment; Reports.  All royalty payments due under this Agreement shall be accompanied by a report setting forth, on a
country-by-country  basis,  Net  Sales  of  the  Products  by  Licensee  and  its  Affiliates  and  Sublicensees  in  the  Licensee  Territory  in  sufficient
detail to permit confirmation of the accuracy of the royalty payment made, including, for each country, the number of Products sold, the gross
sales and Net Sales of Products, including the deductions from gross sales to arrive at Net Sales, the royalty payable, the exchange rates used,
any adjustments to the royalty paid during the Royalty Term pursuant to Section 8.5(c), and whether any Net Sales milestone under Section
8.4 has been achieved.  Within [***] following the end of each Calendar Quarter during the Royalty Term and Extended Commercialization
Term, Licensee shall provide Ovid with the foregoing report and the payment due for such Calendar Quarter.  For clarity, royalty payments
during the Extended Commercialization Term shall not be subject to any offsets or reductions whatsoever, including those set forth in Section
8.5(c).    Prior  to  the  First  Commercial  Sale  of  the  Product  in  the  Licensee  Territory,  the  Parties  will  agree  on  the  form  of  royalty
report.    Licensee  shall  submit  a  single  report  for  all  Net  Sales  during  a  Calendar  Year,  including  all  of  Licensee’s  and  its  Affiliates’  and
Sublicensees’ Net Sales, but shall separately identify the Net Sales and other information applicable to each entity.

44
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
9.2

Exchange  Rate;  Manner  and  Place  of  Payment.    All  references  to  dollars  and  “$”  herein  shall  refer  to  U.S.
dollars.  Unless otherwise specified herein, all payments due under this Agreement shall be payable in U.S. dollars.  When conversion of Net
Sales from any currency other than U.S. dollars is required, such conversion shall be at the exchange rate equal to the conversion rate for the
U.S. dollar for the currency of the country in which the applicable Net Sales were made as published by [***].  All payments owed under this
Agreement  shall  be  made  by  wire  transfer  in  immediately  available  funds  to  a  bank  and  account  designated  in  writing  by  Ovid,  unless
otherwise specified in writing by Ovid.  

9.3

Taxes.

income arising directly or indirectly from the activities of the Parties under this Agreement.  

(a)

Taxes on Income.  Each Party shall be solely responsible for the payment of all taxes imposed on its share of

(b)

Tax Cooperation.   The  Parties  agree  to  cooperate  with  one  another  and  use  reasonable  efforts  to  avoid  or
reduce tax withholding or similar obligations in respect of the milestone payments, royalty payments, and other payments made by Licensee
to Ovid under this Agreement.  To the extent that Licensee is required by Applicable Laws to deduct and withhold taxes on any payment to
Ovid, Licensee shall withhold the amount of such taxes otherwise payable to Ovid and, if and when necessary pay the amounts of such taxes
to the proper Governmental Authority in a timely manner and promptly transmit to Ovid an official tax certificate or other evidence of such
payment  sufficient  to  enable  Ovid  to  claim  such  payment  of  taxes.    Ovid  shall  provide  Licensee  any  tax  forms  that  may  be  reasonably
necessary in order for Licensee to not withhold tax or to withhold tax at a reduced rate under an applicable bilateral income tax treaty, to the
extent legally able to do so.  Ovid shall use reasonable efforts to provide any such tax forms to Licensee in advance of the due date.  Licensee
shall  provide  Ovid  with  reasonable  assistance  to  enable  the  recovery,  as  permitted  by  Applicable  Laws,  of  withholding  taxes  or  similar
obligations resulting from payments made under this Agreement, such recovery to be for the benefit of Ovid.  Licensee shall have the right to
deduct  any  such  tax,  levy,  or  charge  actually  paid  from  payment  due  to  Ovid.    Each  Party  agrees  to  assist  the  other  Party  in  claiming
exemption  from  such  deductions  or  withholdings  under  double  taxation  or  similar  agreement  or  treaty  from  time  to  time  in  force  and  in
minimizing the amount required to be so withheld or deducted.

(c)

Taxes Resulting From Licensee’s Action. If a Party takes any action of its own discretion (not required by a
Regulatory  Authority  and  without  consent  of  the  other  Party),  including  any  assignment,  sublicense,  change  of  place  of  incorporation,  or
failure to comply with Applicable Laws or filing or record retention requirements, which results in a withholding or deduction obligation (a
“Withholding  Tax  Action”),  then  such  Party  shall  pay  the  sum  associated  with  such  Withholding  Tax  Action.    For  clarity,  if  Licensee
undertakes a Withholding Tax Action, then the sum payable by Licensee (in respect of which such deduction or withholding is required to be
made) shall be increased to the extent necessary to ensure that Ovid receives a sum equal to the sum which it would have received had no
such Withholding Tax Action occurred.  If a change in Applicable Laws results in a withholding or deduction obligation absent either Party
taking a Withholding Tax Action, then the amount of such withholding or deduction obligation shall be paid by Licensee to the applicable
Governmental  Authority  on  behalf  of  Ovid,  provided  that  Licensee  shall  assist  Ovid  in  minimizing  or  recovering  such  withholding  or
deduction obligation.  

45
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
The Parties shall use commercially reasonable efforts to invoke the application of any applicable bilateral income tax treaty that would reduce
or eliminate otherwise applicable taxes with respect to payments payable pursuant to this Agreement.

9.4

Records;  Audit.    Each  Party  shall  maintain  complete  and  accurate  records  in  sufficient  detail  in  relation  to  this
Agreement to permit the other Party to confirm the accuracy of the amount of Development Costs to be reimbursed or shared, achievement of
Net Sales milestones, and the amount of royalty and other payments payable under this Agreement.  Each Party will keep such books and
records for at least [***] following the Calendar Year to which they pertain.  Upon reasonable prior notice, such records shall be inspected
during regular business hours at such place or places where such records are customarily kept by an independent certified public accountant
(the “Auditor”) selected by the auditing Party and reasonably acceptable to the audited Party for the sole purpose of verifying for the auditing
Party the accuracy of the financial reports furnished by the audited Party pursuant to this Agreement or of any payments made, or required to
be  made,  by  or  to  the  audited  Party  pursuant  to  this  Agreement.    Before  beginning  its  audit,  the  Auditor  shall  execute  an  undertaking
acceptable to each Party by which the Auditor agrees to keep confidential all information reviewed during the audit.  Such audits may occur
no  more  often  than  [***].    Each  Party  shall  only  be  entitled  to  audit  the  books  and  records  from  the  [***]  in  which  the  audit  request  is
made.  The Auditor shall not disclose the audited Party’s Confidential Information to the auditing Party, and shall only verify the accuracy or
inaccuracy of the financial reports furnished by the audited Party or the amount of payments by such Party under this Agreement, and, in the
case of any inaccuracy, the amount of such inaccuracy.  In the event that the final result of the inspection reveals an undisputed underpayment
or overpayment, the underpaid or overpaid amount shall be settled within [***] after the Auditor’s report.  The auditing Party shall bear the
full  cost  of  such  audit  unless  such  audit  reveals  an  overpayment  to,  or  an  underpayment  by,  the  audited  Party,  which  underpayment  or
overpayment was more than [***], in which case the audited Party shall reimburse the auditing Party for the costs for such audit.  For clarity,
the foregoing audit rights may also be exercised by Ovid on behalf of Lundbeck pursuant to the terms of the Lundbeck License Agreement.  

9.5

Late Payments.  In the event that any payment due under this Agreement is not paid when due in accordance with the
applicable provisions of this Agreement, the payment shall accrue interest from the date due [***]; provided, however, that in no event shall
such rate exceed the maximum legal annual interest rate.  The payment of such interest shall not limit the Party entitled to receive payment
from exercising any other rights it may have as a consequence of the lateness of any payment.  

10.

INTELLECTUAL PROPERTY

10.1

Ownership.  

(a)

Data. All Data generated in connection with any Development or Commercial activities with respect to any
Product conducted solely by or on behalf of Ovid and its Affiliates and licensees (other than Licensee) (the “Ovid Data”) shall be the sole
and  exclusive  property  of  Ovid  or  such  Affiliates  or  licensees,  as  applicable.   All  Data  generated  in  connection  with  any  Development  or
Commercial  activities  with  respect  to  any  Product  conducted  solely  by  or  on  behalf  of  Licensee  or  its  Affiliates  or  Sublicensees  (the
“Licensee Data”) shall be the sole

46
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
and  exclusive  property  of  Licensee  or  such  Affiliates  or  Sublicensees,  as  applicable.    All  Data  generated  in  connection  with  any  Joint
Development Activities or joint Commercial activities with respect to any Product and for which the Parties are sharing Development Costs
pursuant to Section 8.2(a) shall be jointly owned by the Parties.  For clarity, each Party shall have access and right to use and reference the
other Party’s Data as and to the extent set forth in this Agreement.

Inventions.    Inventorship  of  any  Inventions  will  be  determined  in  accordance  with  the  standards  of
inventorship  and  conception  under  U.S.  patent  laws.    The  Parties  will  work  together  to  resolve  any  issues  regarding  inventorship  or
ownership of Inventions.  Ownership of Inventions will be allocated as follows:

(b)

(i)

Ovid shall solely own all data, Inventions, and Patents claiming such Inventions that relate to the
composition,  formulation,  manufacture,  dosing,  new  indications  or  method  of  use  of  the  Compound,  or  any  improvement  of  any  such
composition,  manufacture,  or  use,  including  in  combination  with  other  agents  or  components  (each,  a  “Compound  Invention”).    All
Compound  Inventions  will  be  included  in  the  Ovid  Know-How,  and  Patents  in  the  Licensee  Territory  claiming  such  Inventions  will  be
included in the Ovid Patents.  To the extent that any Compound Invention is made by Licensee, whether solely or jointly with Ovid, Licensee
shall,  and  hereby  does,  transfer  and  assign  to  Ovid,  without  additional  consideration,  all  of  its  right,  title,  and  interest  in  such  Compound
Invention.  To effectuate the foregoing assignment, Licensee shall ensure that all entities and individuals that perform any Development under
this  Agreement  are  under  a  written  or  other  legally  enforceable  obligation  to  assign  all  of  its  right,  title,  and  interest  in  such  Invention  to
Licensee or to an entity that is obligated to assign all right, title, and interest to Licensee.

(ii)

Except  for  Compound  Inventions,  each  Party  shall  solely  own  any  Inventions  made  solely  by  it
and its Affiliates’ employees, agents, or independent contractors, and the Parties shall jointly own any Inventions that are made jointly by
employees, agents, or independent contractors of one Party and its Affiliates together with employees, agents, or independent contractors of
the other Party and its Affiliates (“Joint Inventions”).  All Patents claiming patentable Joint Inventions shall be referred to herein as “Joint
Patents”.  Except to the extent either Party is restricted by the licenses granted to the other Party under this Agreement, each Party shall be
entitled  to  practice,  license,  assign,  and  otherwise  exploit  its  interest  under  the  Joint  Inventions  and  Joint  Patents  without  the  duty  of
accounting or seeking consent from the other Party.  

10.2

Patent Prosecution and Maintenance.  

(a)

Ovid Patents.

(i)

Subject to the remainder of this Section 10.2(a),  and  as  between  the  Parties,  Ovid  shall  have  the
sole  right,  but  not  the  obligation,  to  control  the  preparation,  filing,  prosecution,  and  maintenance  (including  any  interferences,  reissue
proceedings, reexaminations, inter partes review, patent term extensions, applications for supplementary protection certificates, oppositions,
invalidation proceedings and defense of validity or enforceability challenges) of the Ovid Patents (other than Joint Patents) worldwide, using
counsel of its own choice.  Subject to the terms of the Lundbeck License Agreement, Ovid shall (A) keep Licensee informed of material

47
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
progress  with  regard  to  the  preparation,  filing,  prosecution,  and  maintenance  of  the  Ovid  Patents  in  the  Licensee  Territory,  sufficiently  in
advance  for  Licensee  to  be  able  to  review  any  material  documents,  including  content,  timing,  and  jurisdiction  of  the  filing  of  such  Ovid
Patents  in  the  Licensee  Territory,  (B)  consult  with,  and  consider  in  good  faith  the  requests  and  suggestions  of,  Licensee  with  respect  to
strategies for filing, prosecuting, and defending, if any, the Ovid Patents in the Licensee Territory, and (C), [***].

(ii)

In the event that Ovid desires to abandon or cease prosecution or maintenance of any Ovid Patent
in any country in the Licensee Territory, Ovid shall provide reasonable prior written notice to Licensee of such intention to abandon (which
notice shall, to the extent possible, be given no later than [***] prior to the next deadline for any action that must be taken with respect to any
such Ovid Patent in the relevant patent office).  In such case, upon Licensee’s written election provided no later than [***] after such notice
from Ovid, Ovid shall continue prosecution and maintenance of such Ovid Patent at Licensee’s direction and expense.  If Licensee does not
provide such election within [***] after such notice from Ovid, Ovid may, in its sole discretion, continue prosecution and maintenance of
such Ovid Patent or discontinue prosecution and maintenance of such Ovid Patent.

(b)

Licensee Patents.  

(i)

Subject  to  the  remainder  of  this  Section  10.2(b),  Licensee  shall  have  the  first  right,  but  not  the
obligation, to control the preparation, filing, prosecution and maintenance (including any interferences, reissue proceedings, reexaminations,
patent term extensions, applications for supplementary protection certificates, oppositions, invalidation proceedings, and defense of validity
or enforceability challenges) of all Licensee Patents (other than Joint Patents) worldwide, at its sole cost and expense and by counsel of its
own  choice  in  the  Licensee  Territory  and  by  counsel  mutually  agreed  to  by  the  Parties  in  the  Ovid  Territory.    Licensee  shall  keep  Ovid
informed of the status of filing, prosecution, maintenance, and defense, if any, of the Licensee Patents, and Licensee shall consult with, and
consider  in  good  faith  the  requests  and  suggestions  of,  Ovid  with  respect  to  strategies  for  filing,  prosecuting,  and  defending  the  Licensee
Patents.

(ii)

In the event that Licensee desires to abandon or cease prosecution or maintenance of any Licensee
Patent, Licensee shall provide reasonable prior written notice to Ovid of such intention to abandon (which notice shall, to the extent possible,
be  given  no  later  than  [***]  prior  to  the  next  deadline  for  any  action  that  must  be  taken  with  respect  to  any  such  Licensee  Patent  in  the
relevant patent office).  In such case, upon Ovid’s written election provided no later than [***] after such notice from Licensee, Ovid shall
have the right to assume prosecution and maintenance of such Licensee Patent at Ovid’s expense and Licensee shall assign to Ovid all of its
rights, title, and interest in and to such Licensee Patent.  If Ovid does not provide such election within [***] after such notice from Licensee,
Licensee  may,  in  its  sole  discretion,  continue  prosecution  and  maintenance  of  such  Licensee  Patent  or  discontinue  prosecution  and
maintenance of such Licensee Patent.

(c)

Joint Patents.  

(i)
obligation, to prepare, file, prosecute, and maintain (including any

Subject  to  the  remainder  of  this  Section  10.2(c),  Ovid  shall  have  the  first  right,  but  not  the

48
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
interferences, reissue proceedings, reexaminations, patent term extensions, applications for supplementary protection certificates, oppositions,
invalidation proceedings, and defense of validity or enforceability challenges) Joint Patents using a patent counsel selected by Ovid in the
Ovid  Territory  and  counsel  mutually  agreed  to  by  the  Parties  in  the  Licensee  Territory..  Ovid  shall  keep  Licensee  informed  of  material
progress with regard to the preparation, filing, prosecution, maintenance, and defense, if any, of the Joint Patents, including content, timing,
and jurisdiction of the filing of such Joint Patents, and Ovid shall consult with, and consider in good faith the requests and suggestions of,
Licensee with respect to filing, prosecuting, and defending of the Joint Patents in the Licensee Territory.

(ii)

In the event that Ovid desires to abandon or cease prosecution or maintenance of any Joint Patent
in any country in the Licensee Territory, Ovid shall provide reasonable prior written notice to Licensee of such intention to abandon (which
notice shall, to the extent possible, be given no later than sixty (60) days prior to the next deadline for any action that must be taken with
respect to any such Joint Patent in the relevant patent office).  In such case, at Licensee’s sole discretion, upon written notice from Licensee to
Ovid, Licensee may elect to continue prosecution or maintenance of any such Joint Patent at its own expense, and Ovid shall execute such
documents and perform such acts, at Licensee’s expense, as may be reasonably necessary to allow Licensee to continue the prosecution and
maintenance of such Joint Patent in such country in the Licensee Territory.  Any such assignment shall be completed in a timely manner to
allow Licensee to continue prosecution and maintenance of any such Joint Patent and any such Patent so assigned shall cease to be either a
Joint  Patent  or  a  Licensee  Patent  and  shall  no  longer  be  subject  to  the  licenses  and  other  rights  granted  by  Licensee  to  Ovid  under  this
Agreement

(d)

Cooperation. Each Party agrees to cooperate fully in the preparation, filing, prosecution, maintenance, and
defense,  if  any,  of  Patents  under  Section  10.2  and  in  the  obtaining  and  maintenance  of  any  patent  term  extensions  and  supplementary
protection certificates and their equivalents, at its own cost (except as expressly set forth otherwise in this Section 10).    Such  cooperation
includes  (i)  executing  all  papers  and  instruments,  or  requiring  its  employees  or  contractors,  to  execute  such  papers  and  instruments,  so  as
enable  the  other  Party  to  apply  for  and  to  prosecute  patent  applications  in  any  country  as  permitted  by  Section  10.2;  and  (ii)  promptly
informing the other Party of any matters coming to such Party’s attention that may affect the preparation, filing, prosecution, or maintenance
of any such patent application and the obtaining of any patent term extensions or supplementary protection certificates or their equivalents.

10.3

Patent Enforcement.

(a)

Notice.    Each  Party  shall  notify  the  other  within  [***]  of  becoming  aware  of  any  alleged  or  threatened
infringement by a Third Party of any of the Ovid Patents (including Joint Patents) in the Licensee Territory, which infringement adversely
affects or is reasonably expected to adversely affect any Product, including any declaratory judgment, opposition, or similar action alleging
the invalidity, unenforceability, or non-infringement of any of the Ovid Patents (collectively, “Product Infringement”).  

and control any legal action in connection with such

(b)

Enforcement Right.  Ovid shall have the first right to use Ovid Commercially Reasonable Efforts to bring

49
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
Product Infringement at its own expense as it reasonably determines appropriate.  If Ovid (i) decides not to bring such legal action against a
Product  Infringement  (the  decision  of  which  Ovid  shall  inform  Licensee  promptly)  or  (ii)  Ovid  otherwise  fails  to  bring  such  legal  action
against a Product Infringement within [***] after first becoming aware of such Product Infringement, subject to the terms of the Lundbeck
License Agreement, Licensee shall have the right to bring and control any legal action in connection with such Product Infringement at its
own expense as it reasonably determines appropriate after [***] Ovid.

(c)

Collaboration.  Each Party shall provide to the enforcing Party reasonable assistance in such enforcement, at
such enforcing Party’s request and expense, including to be named in such action if required by Applicable Laws to pursue such action.  The
enforcing Party shall keep the other Party regularly informed of the status and progress of such enforcement efforts, shall reasonably consider
the other Party’s comments on any such efforts, including determination of litigation strategy and filing of material papers to the competent
court.  The non-enforcing Party shall be entitled to separate representation in such matter by counsel of its own choice and at its own expense,
but such Party shall at all times cooperate fully with the enforcing Party.  

(d)

Expense and Recovery.  

Except as set forth in Section 10.3(d)(ii),  the  enforcing  Party  shall  be  solely  responsible  for  any
cost  and  expenses  incurred  by  such  Party  as  a  result  of  such  enforcement  action.    If  such  Party  recovers  monetary  damages  in  such
enforcement action, such recovery shall be allocated [***].

(i)

(ii)

Notwithstanding the foregoing, if [***] to bring such action.  If [***], then [***].

(e)

Other Infringement.  Except for Product Infringement as set forth above, each Party shall have the exclusive
right  to  enforce  its  own  Patents  against  any  infringement  anywhere  in  the  world.    For  clarity,  as  between  the  Parties,  Ovid  shall  have  the
exclusive right to enforce (i) the Ovid Patents against any infringement in the Licensee Territory that is not a Product Infringement, and (ii)
the Ovid Patents and Joint Patents against any infringement in the Ovid Territory, in each case at its own expense as it reasonably determines
appropriate, and subject to the terms of the Lundbeck License Agreement. The Parties shall discuss global enforcement strategy for the Ovid
Patents and Licensee Patents, including the defense of validity and enforceability challenges arising from any enforcement action.    

10.4

Infringement of Third Party Rights.  If any Product used or sold by Licensee, its Affiliates, or Sublicensees becomes
the  subject  of  a  Third  Party’s  claim  or  assertion  of  infringement  of  any  intellectual  property  rights  in  a  jurisdiction  within  the  Licensee
Territory,  Licensee  shall  promptly  notify  Ovid  and  the  Parties  shall  promptly  meet  to  consider  the  claim  or  assertion  and  the  appropriate
course of action and may, if appropriate, agree on and enter into a “common interest agreement” wherein the Parties agree to their shared,
mutual interest in the outcome of such potential dispute.  Absent any agreement to the contrary, and subject to claims for indemnification
under Article 12, each Party may defend itself from any such Third Party claim at its own cost and expense, provided that [***].  If [***].

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or confidential.

 
10.5

Trademarks.

(a)

Product  Trademarks.    Ovid  shall  develop  and  adopt  trademarks,  including  trade  names,  trade  dresses,
branding, and logos, to be used for the Products (the “Product Marks”).  Ovid shall own all Product Marks throughout the world and all
goodwill in the Product Marks shall accrue to Ovid.  The Parties shall collaborate to have a global, worldwide trademark to be used on the
Product.  In the event Ovid is unable to obtain or maintain the Product Marks for the Product in the Licensee Territory or in some countries in
the Licensee Territory, the Parties shall collaborate to select such other Product Marks as may be available for registration and marketing of
the Product in those countries. Ovid shall be responsible for the registration, maintenance, defense and enforcement of the Product Marks
using counsel of its own choice in the Ovid Territory and counsel mutually agreed to by the Parties in the Licensee Territory.  Ovid shall keep
Licensee  informed  of  material  progress  with  regard  to  the  registration,  prosecution,  maintenance  and  defense,  if  any,  of  the  Product
Trademarks  in  the  Licensee  Territory,  including  content,  timing,  and  jurisdiction  of  the  filing  of  such  Product  Trademarks  in  the  Licensee
Territory, sufficiently in advance for Licensee to be able to review any material documents, and Ovid shall consult with, and consider in good
faith the requests and suggestions of, Licensee with respect to strategies for filing, prosecuting and defending the Product Trademarks in the
Licensee Territory.

(b)

Trademark License.  Licensee shall use the Product Marks to Commercialize the Product in the Licensee
Territory.    In  addition,  unless  prohibited  by  Applicable  Laws,  Licensee  shall  use  Commercially  Reasonable  Efforts  to  include  Ovid’s
corporate trademark on the packaging and product information of the Products sold in the Licensee Territory to indicate that the Product is
licensed  from  Ovid.    Ovid  hereby  grants  to  Licensee  a  limited,  royalty-free  license  to  use  Ovid’s  corporate  trademark  and  Product  Marks
solely in connection with the Commercialization of the Product in the Licensee Territory under this Agreement.  All use of the Product Marks
and Ovid’s corporate trademark shall comply with Applicable Laws and shall be subject to Ovid’s review and approval.  For clarity, Licensee
shall also include its (or its Affiliate’s or Sublicensee’s, as applicable) corporate logo in the Product sold in the Licensee Territory.

Product  Domain  Names.    In  the  Licensee  Territory,  Licensee  shall  have  the  exclusive  right  to  register
Product Marks as domain names, including all internet domain names under all existing top level domains. This includes as example top level
domains such as .com, .net., .info and country code top level domains such as .dk, .uk and .it.

(c)

11.

REPRESENTATIONS AND WARRANTIES

11.1

Mutual Representations and Warranties.  Each Party represents and warrants to the other that, as of the Effective
Date: (a) it is duly organized and validly existing under the laws of its jurisdiction of incorporation or formation, and has full corporate or
other power and authority to enter into this Agreement and to carry out the provisions hereof, (b) it is duly authorized to execute and deliver
this  Agreement  and  to  perform  its  obligations  hereunder,  and  the  person  or  persons  executing  this  Agreement  on  its  behalf  has  been  duly
authorized to do so by all requisite corporate or partnership action, (c) this Agreement is legally binding upon it, enforceable in accordance
with its terms, and does not conflict with any agreement, instrument, or understanding, oral or written, to which it is a Party or by which it
may  be  bound,  nor  violate  any  material  law  or  regulation  of  any  court,  governmental  body,  or  administrative  or  other  agency  having
jurisdiction

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or confidential.

 
over it, (d) it has the right to grant the licenses granted by it under this Agreement; (e) the execution and delivery of this Agreement and the
performance  of  such  Party’s  obligations  under  this  Agreement  do  not  and  will  not  result  in  the  breach  of,  constitute  a  default,  cause  the
acceleration of performance, require any consent under, or result in the creation of any lien, charge or encumbrance upon any of its property
or assets pursuant to any material instrument or agreement to which it is a party, or by which it or its properties may be bound or affected, as
of the Effective Date; and (f) it is not a party to any agreement, arrangement or understanding with any Third Party which in any significant
way prevents it from fulfilling any its material obligations under the terms of this Agreement.

11.2

Covenants.

(a)

Employees, Consultants, and Contractors.  Each Party covenants that it has obtained or will obtain written
agreements from each of its employees, consultants, and contractors who perform Development activities pursuant to this Agreement, which
agreements will obligate such persons to obligations of confidentiality and non-use and to assign (or, in the case of contractor, grant a license
under) Inventions, in each case in a manner consistent with the provisions of this Agreement.

(b)

Debarment.    Each  Party  represents,  warrants,  and  covenants  to  the  other  Party  that  it  is  not  debarred  or
disqualified under the U.S. Federal Food, Drug and Cosmetic Act, as may be amended, or comparable laws in any country or jurisdiction
other than the U.S., and it does not, and will not during the Term, employ or use the services of any person who is debarred or disqualified, in
connection  with  activities  relating  to  the  Compound  or  any  Product.    In  the  event  that  either  Party  becomes  aware  of  the  debarment  or
disqualification or threatened debarment or disqualification of any person providing services to such Party, including the Party itself or its
Affiliates or Sublicensees, that directly or indirectly relate to activities contemplated by this Agreement, such Party shall immediately notify
the other Party in writing and such Party shall cease employing, contracting with, or retaining any such person to perform any such services.

(c)

Compliance.  Licensee covenants as follows:

its and its Affiliates’ employees and contractors to comply with all Applicable Laws.

(i)

In the performance of its obligations under this Agreement, Licensee shall comply and shall cause

(ii)

Licensee  and  its  and  its  Affiliates’  employees  and  contractors  shall  not,  in  connection  with  the
performance of their respective obligations under this Agreement, directly or indirectly through Third Parties, pay, promise, or offer to pay, or
authorize the payment of, any money or give any promise or offer to give, or authorize the giving of anything of value to a Public Official or
Entity or other person for purpose of obtaining or retaining business for or with, or directing business to, any person, including, Licensee (and
Licensee  represents  and  warrants  that  as  of  the  Effective  Date,  Licensee,  and  to  its  knowledge,  its  and  its  Affiliates’  employees  and
contractors, have not directly or indirectly promised, offered, or provided any corrupt payment, gratuity, emolument, bribe, kickback, illicit
gift, or hospitality or other illegal or unethical benefit to a Public Official or Entity or any other person in connection with the performance of
Licensee’s obligations under this Agreement, and Licensee covenants that it and

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or confidential.

 
its Affiliates’ employees and contractors shall not, directly or indirectly, engage in any of the foregoing).  

Licensee and its Affiliates, and their respective employees and contractors, in connection with the
performance of their respective obligations under this Agreement, (1) shall not violate or cause the violation of the FCPA, Export Control
Laws, or any other Applicable Laws, or otherwise cause any reputational harm to Ovid, and (2) shall immediately notify Ovid if Licensee has
any information or suspicion that there may be a violation of any of the foregoing in connection with activities under this Agreement.

(iii)

In  connection  with  the  performance  of  its  obligations  under  this  Agreement,  Licensee  shall
comply  and  shall  cause  its  and  its  Affiliates’  employees  and  contractors  to  comply  with  Licensee’s  own  anti-corruption  and  anti-bribery
policy, a copy of which has been provided to Ovid prior to the Effective Date.

(iv)

Ovid  will  have  the  right,  upon  reasonable  prior  written  notice  and  during  Licensee’s  regular
business hours, to conduct at its own cost and expenses inspections of and to audit Licensee’s books and records in the event of a suspected
violation or to ensure compliance with the representations, warranties, and covenants of this Section 11.2(c); provided, however, that in the
absence of good cause for such inspections and audits, Ovid may exercise this right no more than annually.

(v)

In the event that Licensee has violated or been suspected of violating any of the representations,
warranties, or covenants in this Section 11.2(c), Licensee will cause its or its Affiliates’ personnel or others working under its direction or
control to submit to periodic training that Licensee will provide on anti-corruption law compliance.

(vi)

Licensee  will,  at  Ovid’s  request,  annually  certify  to  Ovid  in  writing  Licensee’s  compliance,  in
connection  with  the  performance  of  Licensee’s  obligations  under  this  Agreement,  with  the  representations,  warranties,  or  covenants  in
Section 11.2(c), which certification shall be issued by Licensee’s global commercial head for the Product.

(vii)

Ovid shall have the right to suspend or terminate this Agreement in its entirety where there is a
credible  finding,  after  a  reasonable  investigation,  that  Licensee,  its  Affiliates,  or  its  Sublicensees,  in  connection  with  performance  of
Licensee’s obligations under this Agreement, has engaged in chronic or material violations of the FCPA.

(viii)

11.3

Additional Ovid Representations and Warranties.  Ovid represents, warrants, and covenants, on behalf of itself and

its Affiliates, as applicable, to Licensee that, as of the Effective Date:

(a)

to  the  extent  applicable  to  the  performance  of  its  obligations  under  this  Agreement,  Ovid  shall  comply  and

shall cause its and its Affiliates’ employees and contractors to comply with all Applicable Laws;

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or confidential.

 
 
Development, registration, use or Commercialization of the Product in the Licensee Territory;

(b)

Exhibit  B  lists  all  of  the  Ovid  Patents  as  of  the  Effective  Date  that  are  necessary  or  useful  for  the

respect to the Ovid Technology under this Agreement;

(c)

to Ovid’s knowledge, Ovid has the right to grant all rights and licenses it purports to grant to Licensee with

as set forth above, Ovid is not a party to any agreement, arrangement or understanding with any Third Party
which in any manner prevents it from fulfilling or affects its ability to perform any of its obligations under the terms of this Agreement to a
material extent;

(d)

(e)

(f)

Ovid and its Affiliates have not granted any liens or security interests on the Ovid Technology;

Ovid and its Affiliates have not received any written notice from a Third Party that the Development of any

Product conducted by Ovid prior to the Effective Date has infringed any Patents of any Third Party;

Third Party under the Ovid Technology that would conflict with or derogate the licenses or other rights granted to Licensee hereunder;

(g)

Ovid and  its Affiliates have not as of the Effective Date, and will not during the Term, grant any right to any

no  claim  or  action  has  been  brought  or,  to  Ovid’s  knowledge,  threatened  in  writing,  by  any  Third  Party
alleging that the Ovid Patents are invalid or unenforceable, and no Ovid Patent is the subject of any interference, opposition, cancellation, or
other protest proceeding;

(h)

misappropriated the Ovid Technology in the Licensee Territory;

(i)

to  Ovid’s  knowledge,  no  Third  Party  is  infringing  or  misappropriating  or  has  materially  infringed  or

the Effective Date has been conducted in compliance with all Applicable Laws;

(j)

to Ovid’s knowledge, all research and Development of the Product conducted by or on behalf of Ovid prior to

material to the evaluation of the safety, efficacy, and manufacturing process of the Product;

(k)

to Ovid’s knowledge, it has disclosed to Licensee the clinical and non-clinical data in Ovid’s Control that is

to Ovid’s knowledge, there are no issues or information, which to Ovid’s knowledge and reasonable opinion,
are reasonably likely to have a material impact on the Development of the Product that have not been fully disclosed to Licensee in the course
of Licensee’s due diligence;

(l)

to  Ovid’s  knowledge,  the  Ovid  Technology  includes  all  intellectual  property  rights  which  are  reasonably
necessary  for  the  Development,  registration,  manufacture,  use  and  Commercialization  of  the  Product  in  the  Licensee  Territory  as
contemplated by the terms of this Agreement;

(m)

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or confidential.

 
adversely affect the rights granted to Licensee under the Ovid Technology;

(n)

no  litigation  has  been  brought  against  Ovid  or  any  of  its  Affiliate,  or  threatened  in  writing,  which  would

neither Ovid nor any of its Affiliates has granted to any Third Party any right (including any license or option
or other right to obtain a license) to develop or commercialize Product in the Field in the Licensee Territory that would conflict with the rights
granted to Licensee under this Agreement;

(o)

as  set  forth  above,  Ovid  has  not  granted  any  Third  Party  any  license,  option  or  other  right  under  or  with
respect to the Ovid Technology that would conflict with or derogate from the licenses, options and other rights granted to Licensee hereunder;

(p)

encumbrances which would have prevent or impair the grant of such rights;

(q)

Ovid has the right to grant the License under Ovid Know-How specified herein free and clear of any liens or

clear of any liens or encumbrances which would prevent or impair the grant of such rights;

(r)

as set forth above, to Ovid’s knowledge,  it has the right to grant the License specified in Section 2.1 free and

inconsistent with the obligations, rights and licenses granted to Licensee in this Agreement.

(s)

as set forth above, to its knowledge, Ovid has not and will not enter into any agreement that is or would be

of the Compound and/or Product under this Agreement and in compliance with Applicable Law; and

(t)

it will use Ovid Commercially Reasonable Efforts in the conduct of the Development and Commercialization

obligations, rights and licenses granted to Licensee under this Agreement.

(u)

as set forth above, it has to not and will not enter into any agreement that is or would be inconsistent with the

(v)

Ovid:  (i)  has  provided  or  made  available  to  Licensee  all  material  relevant  documents  and  written
communications and materials in its and its Affiliates’ possession or Control from and to any Regulatory Authority in the Licensee Territory
related to the Product; (ii) as of the Effective Date, Ovid and its Affiliates have not received any oral or written communication (including
any notice of inspection, deficiency letter, warning letter or similar notice) from any Regulatory Authority alleging that the Development of
Product by or on behalf of Ovid and its Affiliates is not currently materially in compliance with any and all applicable laws or regulations
implemented by any Regulatory Authority; and (iii) to Ovid’s knowledge, Ovid and its Affiliates have not made, with respect to the Product,
any  untrue  statement  of  material  fact  to  any  Regulatory  Authority,  or  failed  to  disclose  a  material  fact  required  to  be  disclosed  to  such
Regulatory Authority.

11.4

Ovid Covenants Regarding the Lundbeck License Agreement.  Ovid shall make any and all payments that become

due under the Lundbeck License Agreement as a result of any

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or confidential.

 
activity under this Agreement, whether by or on behalf of Ovid or by Licensee or its Affiliate or Sublicensee, in each case in accordance with
the terms of the Upstream License Agreement.

Ovid  is  in  compliance  in  all  material  respects  with  the  Lundbeck  License  Agreement,  and,  to  Licensor’s
knowledge, the other party to the Lundbeck License Agreement is not in breach or default in any respect of the Lundbeck License Agreement
pertaining to the Product.

(a)

In the event that Ovid receives a notice or other communication alleging it is in breach (including a notice or
other  communication  threatening  termination)  of  the  Lundbeck  License  Agreement,  Ovid  shall  promptly  provide  Licensee  with  a  copy  of
such notice.

(b)

Ovid  shall  not  agree  to  any  amendment  or  other  modification  (including  termination)  to  the  Lundbeck
License Agreement in a manner that materially adversely affects the rights sublicensed to Licensee under this Agreement without Licensee’s
prior written consent, such consent not to be unreasonably withheld or delayed.

(c)

(d)

Ovid  and  Licensee  have  negotiated  with  Lundbeck  a  technology  transfer  agreement  (the  “Technology
Transfer Agreement”) for the transfer from Lundbeck to Licensee of Know-How, information, and data owned or controlled by Lundbeck
that is necessary or reasonably useful for the manufacture of the Compound and Drug Product in or for the Licensee Territory and according
to  the  technology  transfer    plan  (the  “Technology  Transfer  Plan”)  as  attached  to  the  Technology  Transfer  Agreement.  Such  Technology
Transfer Agreement shall provide such transfer to be finalized over a period of [***] starting from the Effective Date, provided that such time
period shall be extended to the extent of any delay caused by Licensee or any other factor outside Ovid’s reasonable control, including delays
caused by any force majeure event as described in Section 16.8 of the Agreement.

11.5

Additional Licensee Representations, Warranties, and Covenants.  Licensee represents, warrants, and covenants to
Ovid  that,  as  of  the  Effective  Date,  Licensee  has  not  granted,  and  will  not  grant  during  the  Term,  any  right  to  any  Third  Party  under  the
Licensee Technology that would conflict with the rights granted to Ovid hereunder.  Licensee further represents, warrants, and covenants to
Ovid  that,  as  of  the  Effective  Date,  Licensee  does  not  own  or  control  any  Licensee  Patents.    Licensee  further  represents,  warrants,  and
covenants  to  Ovid  that  Licensee  has  the  personnel,  expertise,  capacity,  resources,  equipment,  and  facilities  necessary  to  implement  the
Technology  Transfer  Plan  in  accordance  with  the  timelines  specified  therein  so  that  such  plan  can  be  completed  over  a  period  of  [***]
following the date such technology transfer is commenced.

11.6

Disclaimer.    Except  as  expressly  set  forth  in  this  Agreement,  THE  TECHNOLOGY  AND  INTELLECTUAL
PROPERTY  RIGHTS  PROVIDED  BY  EACH  PARTY  HEREUNDER  ARE  PROVIDED  “AS  IS”  AND  EACH  PARTY  EXPRESSLY
DISCLAIMS  ANY  AND  ALL  WARRANTIES  OF  ANY  KIND,  EXPRESS  OR  IMPLIED,  INCLUDING  THE  WARRANTIES  OF
DESIGN,  MERCHANTABILITY,  FITNESS  FOR  A  PARTICULAR  PURPOSE,  NONINFRINGEMENT  OF  THE  INTELLECTUAL
PROPERTY  RIGHTS  OF  THIRD  PARTIES,  OR  ARISING  FROM  A  COURSE  OF  DEALING,  USAGE  OR  TRADE  PRACTICES,  IN
ALL CASES WITH RESPECT THERETO.  Without limiting the foregoing, (a) neither Party represents or warrants that any data obtained
from conducting Clinical

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or confidential.

 
 
Trials  in  one  country  or  jurisdiction  will  comply  with  the  laws  and  regulations  of  any  other  country  or  jurisdiction,  and  (b)  neither  Party
represents or warrants the success of any study or test conducted pursuant to this Agreement or the safety or usefulness for any purpose of the
technology it provides hereunder.

12.

INDEMNIFICATION

12.1

Indemnification by Ovid.  Ovid hereby agrees to defend, indemnify, and hold harmless Licensee and its Affiliates and
their respective directors, officers, employees, and agents (each, a “Licensee Indemnitee”) from and against any and all liabilities, expenses,
and  losses  including  any  product  liability,  personal  injury,  property  damage,  including  reasonable  legal  expenses  and  attorneys’  fees
(collectively, “Losses”) to which any Licensee Indemnitee may become subject as a result of any claim, demand, action, or other proceeding
by any Third Party to the extent such Losses arise out of or result from: (a) the Development, use, handling, storage, Commercialization, or
other disposition of any Compound or Product by Ovid or its Affiliates or licensees or the contractors of any of them (excluding any activities
by or on behalf of Licensee or its Affiliates or Sublicensees), (b) the negligence or willful misconduct of any Ovid Indemnitee, or (c) the
breach by Ovid of any warranty, representation, covenant, or agreement made by Ovid in this Agreement; except, in each case (a)-(c), to the
extent such Losses arise out of any activities for which Licensee is obligated to indemnify any Ovid Indemnitee(s) under Section 12.2.

12.2

Indemnification by Licensee.  Licensee hereby agrees to defend, indemnify, and hold harmless Ovid, its Affiliates,
and licensees and their respective directors, officers, employees, and agents (each, a “Ovid Indemnitee”) from and against any and all Losses
to which any Ovid Indemnitee may become subject as a result of any claim, demand, action, or other proceeding by any Third Party to the
extent such Losses arise out of: (a) the Development, use, handling, storage, Commercialization, or other disposition of any Compound or
Product  by  Licensee  or  its  Affiliates  or  Sublicensees  or  the  contractor  of  any  of  them,  (b)  the  negligence  or  willful  misconduct  of  any
Licensee  Indemnitee,  or  (c)  the  breach  by  Licensee  of  any  warranty,  representation,  covenant,  or  agreement  made  by  Licensee  in  this
Agreement; except, in each case (a)-(c), to the extent such Losses arise out of any activities for which Ovid is obligated to indemnify any
Licensee Indemnitee(s) under Section 12.1.

12.3

Procedure.  A  party  that  intends  to  claim  indemnification  under  this  Article  12  (the  “Indemnitee”)  shall  promptly
notify the indemnifying Party (the “Indemnitor”) in writing of any Third Party claim, demand, action, or other proceeding (each, a “Claim”)
in  respect  of  which  the  Indemnitee  intends  to  claim  such  indemnification,  and  the  Indemnitor  shall  have  sole  control  of  the  defense  or
settlement thereof.  The Indemnitee may participate at its expense in the Indemnitor’s defense of and settlement negotiations for any Claim
with counsel of the Indemnitee’s own choice.  The indemnity arrangement in this Article 12 shall not apply to amounts paid in settlement of
any  action  with  respect  to  a  Claim  if  such  settlement  is  effected  without  the  consent  of  the  Indemnitor,  which  consent  shall  not  be
unreasonably withheld or delayed.  The failure to deliver written notice to the Indemnitor within a reasonable time after the commencement
of any action with respect to a Third Party Claim shall only relieve the Indemnitor of its indemnification obligations under this Article 12 if
and to the extent the Indemnitor is actually prejudiced thereby.  The Indemnitee shall cooperate fully with the Indemnitor and its legal

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or confidential.

 
representatives in the investigation of any action with respect to a Claim covered by this indemnification.

12.4

Insurance.  Each Party, at its own expense, hereby agrees and undertakes to maintain insurance policies with respect
to the activities to be made by and obligations assumed by each of the Party in accordance to the provisions of this Agreement. In this respect
the Parties agree to carry out at their sole expense and with a commercially reasonable insurance company, the following liability policies, in
an amount consistent with sound business practice and reasonable in light of its obligations under this Agreement during the Term:

activities under this Agreement, with limits and warranties no less than those required by Applicable Law; and

(a)

Clinical Trial liability policies reasonable for each specific phase and country in which a Party is conducting

(b)

product liability policies with limits at a minimum equivalent to [***] per each occurrence and per year.

The Public and Product liability policies above shall start from the Effective Date and last for a period of [***] after the expiration or the
earlier  termination  of  the  Agreement.  Each  Party  shall  provide  a  certificate  of  insurance  (or  evidence  of  self-insurance)  evidencing  such
coverages  to  the  other  Party  upon  request.    It  is  understood  that  such  policies  shall  not  be  construed  to  create  any  limit  of  either  Party’s
obligations  or  liabilities  with  respect  to  its  indemnification  obligations  hereunder.    In  the  event  of  use  by  either  Party  of  subcontractors,
sublicensees,  or  any  Third  Party  in  the  performance  of  such  Party’s  obligations  under  the  Agreement,  such  Party  shall  ensure  that  its
subcontractor, sublicensee, or Third Party has a proper and adequate general liability or professional liability insurance to cover its risks with
respect to the other Party for damages mentioned above.

12.5

Limitation of Liability.  NEITHER PARTY SHALL BE ENTITLED TO RECOVER FROM THE OTHER PARTY
ANY  SPECIAL,  INCIDENTAL,  CONSEQUENTIAL,  OR  PUNITIVE  DAMAGES,  INCLUDING  LOST  PROFITS,  IN  CONNECTION
WITH THIS AGREEMENT OR ANY LICENSE GRANTED HEREUNDER, REGARDLESS OF ANY NOTICE OF THE POSSIBILITY
OF  SUCH  DAMAGES;  PROVIDED,  HOWEVER,  THAT  THIS  SECTION  12.5  SHALL  NOT  BE  CONSTRUED  TO  LIMIT  EITHER
PARTY’S  INDEMNIFICATION  OBLIGATIONS  UNDER  THIS  ARTICLE  12  OR  DAMAGES  AVAILABLE  AS  A  RESULT  OF  A
BREACH OF A PARTY’S EXCLUSIVITY OBLIGATIONS UNDER SECTION 2.8  OR  CONFIDENTIALITY  OBLIGATIONS  UNDER
ARTICLE 13.  

13.

CONFIDENTIALITY

13.1

Confidential  Information.    Except  to  the  extent  expressly  authorized  by  this  Agreement  or  otherwise  agreed  in
writing by the Parties, the Parties agree that, during the Term and for [***] thereafter, the receiving Party shall keep confidential and shall not
publish  or  otherwise  disclose  and  shall  not  use  for  any  purpose  other  than  as  expressly  provided  for  in  this  Agreement  any  Confidential
Information of the other Party, and both Parties shall keep confidential and, subject to the remainder of this Article 13, shall not publish or
otherwise disclose

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or confidential.

 
the terms of this Agreement.  Each Party may use the other Party’s Confidential Information only to the extent required to accomplish the
purposes of this Agreement, including exercising its rights or performing its obligations under this Agreement.  Each Party will use at least
the same standard of care as it uses to protect proprietary or confidential information of its own (but no less than reasonable care) to ensure
that  its  employees,  agents,  consultants,  contractors,  and  other  representatives  do  not  disclose  or  make  any  unauthorized  use  of  the
Confidential Information of the other Party.  Each Party will promptly notify the other upon discovery of any unauthorized use or disclosure
of the Confidential Information of the other Party.

13.2

Exceptions.    The  obligations  of  confidentiality  and  restriction  on  use  under  Section  13.1  will  not  apply  to  any
information that the receiving Party can prove by competent written evidence: (a) is at the time of disclosure, or thereafter becomes, through
no act or failure to act on the part of the receiving Party, generally known or available to the public; (b) is known by the receiving Party at the
time of receiving such information, other than by previous disclosure of the disclosing Party, or its Affiliates, employees, agents, consultants,
or  contractors;  (c)  is  disclosed  to  the  receiving  Party  without  restriction  by  a  Third  Party  who  has  no  obligation  of  confidentiality  or
limitations on use with respect thereto; or (d) is independently discovered or developed by the receiving Party without the use of or reference
to the Confidential Information belonging to the disclosing Party.

13.3

Authorized Disclosure.  Each Party may disclose Confidential Information belonging to the other Party as expressly

permitted by this Agreement or if and to the extent such disclosure is reasonably necessary in the following instances:

(a)

(b)

filing, prosecuting, and maintaining Patents as permitted by this Agreement;

submitting and maintaining Regulatory Filings for Products that such Party has a license or right to Develop

or Commercialize under this Agreement in a given country or jurisdiction;

(c)

prosecuting and defending litigation as permitted by this Agreement;

(d)
securities exchanges; and

complying  with  applicable  court  orders  or  governmental  regulations,  including  regulations  promulgated  by

(e)

disclosure to its and its Affiliates’ employees, consultants, contractors, agents, licensees, and sublicensees, in
each case on a need-to-know basis in connection with the Development, manufacture, or Commercialization of the Compound and Products
in accordance with the terms of this Agreement, in each case under written obligations of confidentiality and non-use at least as stringent as
those herein;

disclosure to actual and bona fide potential investors, acquirors, licensees, and other financial or commercial
partners solely for the purpose of evaluating or carrying out an actual or potential investment, acquisition, collaboration, or other business
relationship, in each case under written obligations of confidentiality and non-use at least as

(f)

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Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
stringent as those herein, provided that the disclosing Party redacts the financial terms and other provisions of this Agreement that are not
reasonably  required  to  be  disclosed  in  connection  with  such  potential  investment,  acquisition,  collaboration,  or  business  transaction  which
redaction shall be prepared in consultation with the other Party; and

disclosure  to  Third  Party  licensors  of  intellectual  property  that  is  related  to  the  Compound  or  any  Product
(e.g., the Third Party that is party to the Lundbeck License Agreement) for the purpose of meeting reporting obligations under such Third
Party agreement.

(g)

Notwithstanding the foregoing, in the event a Party is required to make a disclosure of the other Party’s Confidential Information
pursuant  to  Section  13.3(c)  or  13.3(d),  it  will,  except  where  impracticable,  give  reasonable  advance  notice  to  the  other  Party  of  such
disclosure,  and  to  the  extent  possible,  at  least  [***]  notice,  and  use  the  same  diligent  efforts  to  secure  confidential  treatment  of  such
Confidential Information as such Party would use to protect its own confidential information, but in no event less than reasonable efforts.  In
any  event,  the  Parties  agree  to  take  all  reasonable  action  to  avoid  disclosure  of  Confidential  Information  hereunder.    Any  information
disclosed pursuant to Section 13.3 shall remain Confidential Information and subject to the restrictions set forth in this Agreement, including
the foregoing provisions of this Section 13.

13.4

Publications.  

(a)

Ovid shall have the right to review and comment on any material proposed for disclosure or publication by
Licensee  regarding  results  of  and  other  information  regarding  Licensee’s  Development  activities  during  the  Term  with  respect  to  the
Compound  and  Product,  whether  by  oral  presentation,  manuscript,  or  abstract.    Before  any  such  material  is  submitted  for  publication,  or
presentation of any such material is made, Licensee shall deliver a complete copy of the material proposed for disclosure to Ovid at least
[***]  prior  to  submitting  the  material  to  a  publisher  or  initiating  any  other  disclosure,  or  as  close  to  these  time  frames  as  reasonably
possible.  Ovid shall review any such material and give its comments to Licensee within [***] of the receipt of such material.  With respect to
oral  presentation  materials  and  abstracts,  Ovid  shall  make  reasonable  efforts  to  expedite  review  of  such  materials  and  abstracts,  and  shall
return  such  items  as  soon  as  practicable  to  Licensee  with  comments,  if  any.    Subject  to  Section  13.4(b),  following  the  expiration  of  the
applicable  time  period  for  review,  Licensee  shall  be  free  to  submit  such  proposed  manuscript  for  publication  or  presentation  materials  for
public disclosure, and does not need to follow this process for subsequent publications or presentations of the same data.    

(b)
or presentation, in Ovid’s reasonable judgment:

If Ovid notifies Licensee within the applicable time period set forth in Section 13.4(a) that such publication

contains an invention for which Ovid desires to obtain patent protection, Licensee shall delay such
publication or presentation for a period of up to [***] (or such other time period agreed by the Parties in writing) to permit the preparation
and filing of a patent application for such invention, or

(i)

(ii)
the commercial value of any Confidential Information disclosed by

contains any Confidential Information of Ovid, or could be expected to have an adverse effect on

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Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
Ovid to Licensee, the Parties shall attempt to agree on revisions to the applicable disclosure so as to preserve both the commercial value of
such Confidential Information and the scientific merit of such disclosure, provided that if and to the extent the Parties are unable to agree,
Licensee shall delete such Confidential Information from the proposed publication or presentation.

13.5

Publicity; Public Disclosures and Public Announcements. Save as permitted in this Section 13.5, neither Party shall
make any public announcement or statement to the public containing Confidential Information of the other Party without the prior consent of
such other Party. On or promptly after the Effective Date, the Parties shall issue a joint public announcement, or either Party may issue its
own  public  announcement,  regarding  the  execution  of  this  Agreement  with  information  substantially  consistent  with  the  information
contained  in  the  form  of  press  release  attached  hereto  as  Exhibit  D.    It  is  understood  that  each  Party  may  desire  or  be  required  to  issue
subsequent press releases relating to this Agreement or activities hereunder.  The Parties agree to consult with each other reasonably and in
good faith with respect to the text and timing of such press releases prior to the issuance thereof, to the extent practicable, and in the case of
any press release Licensee wishes to issue, Licensee shall first obtain Ovid’s written approval of such release.  Notwithstanding the foregoing,
neither Party may unreasonably withhold, condition, or delay consent to such releases by more than [***], and either Party may issue such
press releases or make such disclosures to the SEC or other applicable agency as it determines, based on advice of counsel, is reasonably
necessary to comply with Applicable Laws or for appropriate market disclosure.  Each Party shall provide the other Party with advance notice
of legally required disclosures to the extent practicable, and to the extent possible, at least [***] prior to such disclosure.  The Parties will
consult  with  each  other  on  the  provisions  of  this  Agreement  to  be  redacted  in  any  filings  made  by  a  Party  with  the  SEC  or  as  otherwise
required  by  Applicable  Laws;  provided  that  each  Party  shall  have  the  right  to  make  any  such  filing  as  it  reasonably  determines  necessary
under Applicable Laws.  In addition, following the initial joint press release announcing this Agreement, either Party shall be free to disclose,
without  the  other  Party’s  prior  written  consent,  the  existence  of  this  Agreement,  the  identity  of  the  other  Party,  and  those  terms  of  the
Agreement which have already been publicly disclosed in accordance with.

13.6

Prior Confidentiality Agreement.   As  of  the  Effective  Date,  the  terms  of  this  Article  13  shall  supersede  any  prior
non-disclosure,  secrecy,  or  confidentiality  agreement  between  the  Parties  (or  their  Affiliates)  relating  to  the  subject  of  this  Agreement,
including  the  Confidentiality  Agreement.   Any  information  disclosed  pursuant  to  any  such  prior  agreement  shall  be  deemed  Confidential
Information under this Agreement.

13.7

Equitable Relief.  Given the nature of the Confidential Information and the competitive damage that a Party would
suffer  upon  unauthorized  disclosure,  use,  or  transfer  of  its  Confidential  Information  to  any  Third  Party,  the  Parties  agree  that  monetary
damages may not be a sufficient remedy for any breach of this Article 13.  In addition to all other remedies, a Party shall be entitled to seek
specific performance and injunctive and other equitable relief as a remedy for any breach or threatened breach of this Article 13.

14.

TERM AND TERMINATION

14.1

Term.  This Agreement shall commence on the Effective Date and shall continue until terminated as provided in this

Article 14 (the “Term”).  Notwithstanding anything herein, on

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Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
a Product-by-Product and country-by-country basis, upon the expiration of the Royalty Term the licenses granted to Licensee in Section 2.1
shall  become  perpetual    and  fully  paid-up  with  respect  to  such  Product  in  such  country,  subject  to  Licensee’s  payment  obligations  under
Article 8 during the Extended Commercialization Term, but thereafter shall be on a non-exclusive basis.  

14.2

Termination for Cause.

(a)

Material Breach.    Each  Party  shall  have  the  right  to  terminate  this  Agreement  immediately  in  its  entirety
upon written notice to the other Party if such other Party materially breaches this Agreement and has not cured such breach to the reasonable
satisfaction  of  the  other  Party  within  [***]  after  notice  of  such  breach  from  the  non-breaching  Party.    In  the  event  of  any  dispute,  the
Agreement shall remain in place during the pendency of any such dispute.  

(b)

Insolvency Event.

(i)

Either Party may terminate this Agreement in its entirety upon providing written notice to the other
Party on or after the time that such other Party makes a general assignment for the benefit of creditors, files a petition for relief in bankruptcy,
petitions for or acquiesces in the appointment of any receiver, trustee or similar officer to liquidate or conserve its business or any substantial
part  of  its  assets,  commences  under  the  laws  of  any  jurisdiction  any  proceeding  involving  its  insolvency,  bankruptcy,  reorganization,
adjustment of debt, dissolution, liquidation or any other similar proceeding for the release of financially distressed debtors, or becomes the
involuntary subject of any proceeding or action of the type described above and such proceeding or action remains un-dismissed or un-stayed
for a period of more than [***].  

(ii)

All  rights  and  licenses  granted  under  or  pursuant  to  this  Agreement  are,  and  shall  otherwise  be
deemed to be, for purposes of Section 365(n) of Title 11 of the United States Code and other similar laws in any other jurisdiction outside of
the Territory (collectively, the “Bankruptcy Laws”), licenses of rights to “intellectual property” as defined under the Bankruptcy Laws.  If a
case  is  commenced  during  the  Term  by  or  against  a  Party  under  Bankruptcy  Laws  then,  unless  and  until  this  Agreement  is  rejected  as
provided  pursuant  to  such  Bankruptcy  Laws,  such  Party  (in  any  capacity,  including  debtor-in-possession)  and  its  successors  and  assigns
(including  a  Title  11  trustee)  shall  perform  all  of  the  obligations  in  this  Agreement  intended  to  be  performed  by  such  Party.    If  a  case  is
commenced  during  the  Term  by  or  against  a  Party  under  the  Bankruptcy  Laws,  this  Agreement  is  rejected  as  provided  for  under  the
Bankruptcy Laws, and the non-bankrupt Party elects to retain its rights hereunder as provided for under the Bankruptcy Laws, then the Party
subject to such case under the Bankruptcy Laws (in any capacity, including debtor-in-possession) and its successors and assigns (including a
Title 11 trustee), shall provide to the non-bankrupt Party copies of all Patents and Information necessary for the non-bankrupt Party to [***]
enjoy  its  rights  under  the  terms  of  this  Agreement.   All  rights,  powers  and  remedies  of  the  non-bankrupt  Party  as  provided  herein  are  in
addition to and not in substitution for any and all other rights, powers and remedies now or hereafter existing at law or in equity (including
the Bankruptcy Laws) in the event of the commencement of a case by or against a Party under the Bankruptcy Laws.  [***].

written notice to Licensee if Licensee or any of its

(c)

Patent Challenge.  Ovid shall have the  right  to  terminate  this  Agreement  immediately  in  its  entirety upon

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Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
Affiliates or Sublicensees directly, or indirectly through any Third Party, commences any interference or opposition proceeding with respect
to, challenges the validity or enforceability of, or opposes any extension of or the grant of a supplementary protection certificate with respect
to, any Ovid Patent.  

14.3

Termination without Cause.

Territory, Licensee shall have the right to terminate this Agreement in its entirety without cause [***].

(a)

Prior  to  the  First  Commercial  Sale.    Prior  to  the  First  Commercial  Sale  of  the  Product  in  the  Licensee

Territory, Licensee shall have the right to terminate this Agreement in its entirety without cause [***].

(b)

After  the  First  Commercial  Sale.    Following  the  First  Commercial  Sale  of  the  Product  in  the  Licensee

14.4

Effects  of  Termination.    Upon  any  termination  of  this  Agreement  by  either  Party,  the  following  Sections  14.4(a)
through  14.4(g)  will  apply.    For  clarity,  during  the  pendency  of  any  termination  notice  period,  all  of  the  terms  and  conditions  of  this
Agreement shall remain in effect and the Parties shall continue to perform all of their respective obligations hereunder.  

(a)

Licenses.  Except in the event of (i) termination by Licensee for  an uncured material breach by Ovid, or (ii)
termination  by  Licensee  in  the  circumstances  set  forth  in  Section  14.2(b)(i)  with  respect  to  Ovid,  or  (iii)  Ovid’s  termination  for  Safety
Reason,  the  licenses  granted  by  Licensee  to  Ovid  shall  survive  such  termination  and  shall  automatically  become  worldwide.      All  of  the
licenses granted by Ovid to Licensee shall be automatically terminated.

(b)

Regulatory Materials; Data.    Except  in  the  event  of  (i)  termination  by  Licensee  for  an  uncured  material
breach  by  Ovid,  or  (ii)  termination  by  Licensee  in  the  circumstances  set  forth  in  Section  14.2(b)(i)  with  respect  to  Ovid,  or  (iii)  Ovid’s
termination for Safety Reason (where Licensee elects to continue the Development and Commercialization of the Product), within [***] after
the effective date of such termination, Licensee shall transfer and assign to Ovid, at no cost to Ovid, all Regulatory Filings and Regulatory
Approvals for the Products, Data from all pre-clinical, non-clinical, and clinical studies of the Product conducted by or on behalf of Licensee,
its  Affiliates,  or  Sublicensees,  and  all  pharmacovigilance  data  (including  all  adverse  event  data)  on  the  Products.    In  addition,  at  Ovid’s
request, Licensee shall provide Ovid with reasonable assistance with any inquiries and correspondence with Regulatory Authorities regarding
the Product in the Licensee Territory, such assistance shall be limited to a period of [***] after such termination.

(c)

Development Wind-Down. Except in the event of (i) termination by Licensee for an uncured material breach
by Ovid, or (ii) termination by Licensee in the circumstances set forth in Section 14.2(b)(i) with respect to Ovid, or (iii) Ovid’s termination
for  Safety  Reason  (where  Licensee  elects  to  continue  the  Development  and  Commercialization  of  the  Product),  Licensee  shall  either,  as
directed  by  Ovid,  (i)  wind-down  any  ongoing  Development  activities  (including  any  Clinical  Trials)  of  Licensee  or  its  Affiliates  and
Sublicensees with respect to any Product in the Licensee Territory in an orderly fashion or (ii) promptly transfer such

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Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
Development activities to Ovid or its designee, in each case in compliance with all Applicable Laws.  

(d)

Cost of Ongoing Trials. Except in the event of (i) termination by Licensee for  an uncured material breach
by Ovid, or (ii) termination by Licensee in the circumstances set forth in Section 14.2(b)(i) with respect to Ovid, or (iii) Ovid’s termination
for Safety Reason, if there is any ongoing Clinical Trial of the Product under the Development Plan for which the Parties are sharing costs,
then Licensee shall continue to share the cost of such Clinical Trial until the effective date of termination.  

(e)

Commercial Wind-Down. Except in the event of (i) termination by Licensee for  an uncured material breach
by Ovid, or (ii) termination by Licensee in the circumstances set forth in Section 14.2(b)(i) with respect to Ovid, or (iii) Ovid’s termination
for Safety Reason (where Licensee elects to continue the Development and Commercialization of the Product), Licensee shall, as directed by
Ovid, (A) continue certain ongoing Commercial activities of Licensee and its Affiliates and Sublicensees with respect to any Product in the
Licensee  Territory  for  a  period  of  up  to  [***]  after  the  effective  date  of  termination,  as  determined  by  Ovid,  and  (B)  handoff  such
Commercial activities to Ovid or its designee, on a timetable to be set by Ovid, not to exceed [***] after the effective date of termination, and
in compliance with all Applicable Laws.  During such commercial wind-down period, Licensee shall continue to book sales and pay royalties
to  Ovid  in  accordance  with  Section  8.5.    Except  as  necessary  to  conduct  the  foregoing  activities  as  directed  by  Ovid,  Licensee  shall
immediately  discontinue  its  (and  shall  ensure  that  its  Affiliates  and  Sublicensees  immediately  discontinue  their)  promotion,  marketing,
offering for sale, and servicing of the Product and its use of all Product Marks.  In addition, Licensee shall immediately deliver to Ovid (at
Licensee’s  expense)  all  samples,  demonstration  equipment,  sales  materials,  catalogs,  and  literature  of  Ovid  in  Licensee’s  possession  or
control.  

(f)

Transition Assistance. Except in the event of (i) termination by Licensee for  an uncured material breach by
Ovid, or (ii) termination by Licensee in the circumstances set forth in Section 14.2(b)(i) with respect to Ovid, or (iii) Ovid’s termination for
Safety Reason (where Licensee elects to continue the Development and Commercialization of the Product), Licensee shall, at no cost to Ovid,
provide reasonable consultation and assistance for a period of no more than [***] after the effective date of termination for the purpose of
transferring  or  transitioning  to  Ovid  all  Licensee  Know-How  not  already  in  Ovid’s  possession  and,  at  Ovid’s  request,  all  then-existing
commercial  arrangements,  customer  lists,  and  similar  information  relating  to  the  Products  that  Licensee  is  able,  using  Commercially
Reasonable Efforts, to transfer or transition to Ovid or its designee, in each case, to the extent reasonably necessary for Ovid to continue the
Development or Commercialization of the Compound and Products in the Licensee Territory.  If any such contract between Licensee and a
Third Party is not assignable to Ovid or its designee (whether by such contract’s terms or because such contract does not relate specifically to
the  Products)  but  is  otherwise  reasonably  necessary  for  Ovid  to  continue  the  Development  or  Commercialization  of  the  Compound  and
Products in the Licensee Territory, or if Licensee is performing such work for the Compound and Product itself (and thus there is no contract
to assign), then Licensee shall reasonably cooperate with Ovid to negotiate for the continuation of such services for Ovid from such entity, or
Licensee shall continue to perform such work for Ovid, as applicable, for a reasonable period (not to exceed [***]) after the effective date of
termination at Ovid’s cost until Ovid establishes an alternate, validated source of such services.  

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or confidential.

 
(g)

Remaining Inventories. Except in the event of (i) termination by Licensee for an uncured material breach by
Ovid, or (ii) termination by Licensee in the circumstances set forth in Section 14.2(b)(i) with respect to Ovid, or (iii) Ovid’s termination for
Safety Reason (where Licensee elects to continue the Development and Commercialization of the Product), Ovid shall have the right, at its
discretion,  to  obtain  from  Licensee  any  or  all  of  the  inventory  of  the  Products  held  by  Licensee  as  of  the  date  of  termination,  free  of
charge.  Ovid shall notify Licensee within [***] after the effective date of termination whether Ovid elects to exercise such right.

14.5

Licensee Continuation. If (a) Licensee has the right to terminate this Agreement in its entirety
for an uncured material breach by Ovid, but elects to continue this Agreement in its entirety as modified by this Section 14.5, or (b) Licensee
has  the  right  to  terminate  in  the  circumstances  set  forth  in  Section  14.2(b)(i),  but  elects  to  continue  this  Agreement  as  modified  by  this
Section 14.5, or (c) Ovid elects to terminate this Agreement in its entirety for Safety Reason, but Licensee elects to continue this Agreement
as modified by this Section 14.5, then, except as provided below, effective as of the date Licensee delivers notice of such election to Ovid, the
following shall apply:

i.

Licensee  shall  have  the  right  to  terminate  the  Supply  Agreement,  and  if  Licensee  terminates  the  Supply  Agreement,  Ovid
shall cooperate with Licensee for smooth technology transfer of the manufacturing process if termination occurs prior to the
Technology Transfer Completion Date.

ii. Notwithstanding anything contained in this Agreement to the contrary, Ovid shall cease any and all Development/Regulatory
activities  with  respect  to  the  Product  in  the  Field  in  the  Licensee  Territory  (other  than  the  Ovid  Ongoing  Trials  if  still
ongoing);

iii. All Licensee payment obligations provided in this Agreement shall continue, including those that are accrued and unpaid as

of the date of such election by Licensee, [***];

iv. After  the  effective  date  of  such  election  by  Licensee,  the  licenses  granted  by  Ovid  to  Licensee  in  Section  2.1  under  the
Product Marks, Ovid Know-How and Ovid Patents for the research, the Development, the use, and the Commercialization of
the  Product  in  the  Field  in  the  Licensee  Territory  shall  continue  and  the  Licensee  shall  have  such  rights  to  Develop,
Manufacture and Commercialize any Product in the Field in the Licensee Territory at Licensee’s sole discretion;

v.

The CGB shall coordinate the wind-down of Ovid’s efforts under this Agreement, and Ovid, as soon as reasonably practical
after  the  effective  date  of  such  election,  shall  provide  to  Licensee,  as  applicable  and  to  the  extent  permitted  under  any
applicable  Third  Party  contract,  (1)  any  information,  including  copies  of  all  Clinical  Trial  data  and  results,  and  the  like
developed by or for the benefit of Ovid for a Product in the Field in the Licensee Territory; and (2) other documents to the
extent relating to the Products that are necessary for the continued Development, Commercialization and Manufacture of the
Product  (including  material  documents  and  agreements  relating  to  the  sourcing  and  Manufacture  of  a  Product  for  sale,
promotion,  distribution,  or  use  of  a  Product)  in  the  Field  throughout  the  Licensee  Territory.  Ovid  will  cooperate  with
Licensee to

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Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
 
 
 
 
 
provide a transfer of such material information and documents.  At Licensee’s request, Ovid shall use reasonable efforts to
assign to Licensee any and all agreements to which Ovid, or its Affiliate, and a Third Party are parties, and that solely cover
or govern the Development, Commercialization and Manufacturing activities conducted in connection with a Product in the
Field in the Territory prior to such election by Licensee, or if such assignment is not permitted under the relevant agreement,
(A)  grant  to  Licensee  other  reasonable  rights  to  provide  to  Licensee  the  benefit  of  such  non-assignable  agreement,  at
Licensee’s  expense,  to  the  extent  permitted  under  the  terms  of  such  non-assignable  agreement;  or  (B)  to  the  extent  not
permitted under the terms of such non-assignable agreement, the Parties shall discuss in good faith an alternative solution to
enable Licensee to receive, at Licensee’s expense, the benefit of the terms of such non-assignable agreement. Ovid shall take
such other reasonable actions and execute such other instruments, assignments and documents as may be necessary to effect
the transfer of rights to such Product(s) as described in this Section 14.5(v) hereunder to Licensee;

vi. Ovid shall transfer to Licensee any and all Regulatory Materials directly and solely related to the Product in the Field in the
Licensee Territory, and, upon Licensee’s request, shall make available to Licensee any other relevant information reasonably
requested by Licensee related to such Regulatory Materials;

vii. As  long  as  Licensee  is  not  in  breach  of  this  Agreement  or  the  Lundbeck  License  Agreement  at  the  effective  date  of  such
election,  Licensee  shall  have  the  rights  of  a  non-breaching  sublicensee  set  forth  in  the  Lundbeck  License  Agreement  (as
amended by the Lundbeck Sublicense Amendment) from and after such election;

viii. Licensee  shall  have  no  further  obligation  to  use  Angelini  Commercially  Reasonable  Efforts  with  respect  to  its  obligations

hereunder;

ix. Ovid shall be obliged to bear the costs of the Ovid Ongoing Trials, if still ongoing; and

x.

In lieu of Section 12.1 and Section 12.2, the following shall apply: Licensee hereby agrees to defend, indemnify, and hold
harmless the Ovid Indemnitees from and against any and all Losses to which any Ovid Indemnitee may become subject as a
result  of  any  claim,  demand,  action,  or  other  proceeding  by  any  Third  Party  to  the  extent  such  Losses  arise  out  of:  (A)
Licensee’s decision to continue the Development, Manufacture and Commercialization of Product following Ovid’s cessation
of such activities for Safety Reason, (B)  any Development, use, handling, storage, manufacture, Commercialization, or other
disposition of any Compound or Product by Licensee or its Affiliates or Sublicensees or the contractor of any of them, (C)
the negligence or willful misconduct of any Licensee Indemnitee or Licensee’s Affiliates or Sublicensees, or (D) the breach
by Licensee of any warranty, representation, covenant, or agreement made by Licensee in this Agreement.

14.6

Confidential Information.  Upon expiration or termination of this Agreement in its entirety, except to the extent that a
Party  obtains  or  retains  the  right  to  use  the  other  Party’s  Confidential  Information,  each  Party  shall  promptly  return  to  the  other  Party,  or
delete or destroy,

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or confidential.

 
 
 
 
 
 
 
all relevant records and materials in such Party’s possession or control containing Confidential Information of the other Party; provided that
such Party may keep one copy of such materials for archival purposes only subject to continuing confidentiality obligations.  All Licensee
Data and Regulatory Filings assigned to Ovid upon termination of this Agreement will be deemed Ovid’s Confidential Information and no
longer Licensee’s Confidential Information.

14.7

Survival.  Expiration or termination of this Agreement shall not relieve the Parties of any obligation or right accruing
prior to such expiration or termination.  Except as set forth below or elsewhere in this Agreement, the obligations and rights of the Parties
under the following provisions of this Agreement shall survive expiration or termination of this Agreement.

14.8

Exercise  of  Right  to  Terminate.    All  rights  and  obligations  of  a  Party  accrued  prior  to  the  effective  date  of  a
termination  (including  the  rights  to  receive  reimbursement  for  costs  incurred  prior  to  the  effective  date  of  such  termination  and  payments
accrued or due prior to the effective date of such termination) shall survive such termination.

15.

DISPUTE RESOLUTION

15.1

General.  Except as provided in Sections 3.4 and 9.4, any dispute between the Parties in connection with or relating to

this Agreement or any document or instrument delivered in connection herewith (a “Dispute”) shall be resolved pursuant to this Section 15.

15.2

Executive Officers.  Any Dispute shall first be referred to the Executive Officers of the Parties, who shall confer in
good faith on the resolution of the issue.  Any final decision mutually agreed to by the Executive Officers shall be conclusive and binding on
the Parties.

15.3

Intellectual Property Disputes.  If the Executive Officers are not able to agree on the resolution of a Dispute within
thirty (30) days (or such other period of time as mutually agreed by the Executive Officers) after such Dispute was first referred to them and
such Dispute is with respect to the validity, scope, enforceability, inventorship, or ownership of any Patent, trademark, or other intellectual
property  right  (“IP  Dispute”),  then,  if  a  Party  wishes  to  pursue  further  resolution  of  such  IP  Dispute,  an  action,  claim,  or  proceeding  to
resolve  such  IP  Dispute  shall  be  brought  in  any  court  of  competent  jurisdiction  in  any  country  or  jurisdiction  in  which  such  intellectual
property rights apply.  

15.4

Arbitration.  If the Executive Officers are not able to agree on the resolution of a Dispute within thirty (30) days (or
such  other  period  of  time  as  mutually  agreed  by  the  Executive  Officers)  after  such  Dispute  was  first  referred  to  them,  then,  except  as
otherwise set forth in Section 15.3, if a Party wishes to pursue further resolution of such Dispute, such Dispute shall be finally resolved by
binding  arbitration  in  accordance  with  this  Section  15.4.    Such  Dispute  shall  be  referred  to  and  finally  resolved  by  arbitration  under  the
International Chamber of Commerce (“ICC”) Rules, as then in effect, by a tribunal of three (3) arbitrators.  The seat and legal place of the
arbitration shall be [***].  Each Party shall nominate one arbitrator and the third arbitrator shall be nominated by the two Party-nominated
arbitrators within [***] after the second arbitrator’s appointment.  If a Party does not nominate its arbitrator within [***] following the expiry
of the allotted period, then such arbitrator shall be appointed by the ICC in accordance with its rules.  Any arbitrator appointed by the ICC
shall have at least [***] experience in the pharmaceutical

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or confidential.

 
industry.  The arbitration shall be conducted, and all documents submitted to the arbitrators shall be, in English.  Each Party shall bear its own
legal costs for its counsel and other expenses, and the Parties shall equally share the costs of the arbitration; provided that the arbitral tribunal
shall have the discretion to provide that the losing party is responsible for all or a portion of such arbitration and legal costs, in such case the
arbitral award will so provide.  The arbitrators shall have no power to award damages excluded pursuant to Section 12.5.  In no event shall
the arbitrators assign a value to any issue greater than the greatest value for such issue claimed by either Party or less than the smallest value
for such issue for such item claimed by either Party.  The award shall be final and binding upon the Parties and the Parties undertake to carry
out any award without delay.  Judgment on the award may be entered in any court of competent jurisdiction.  Except to the extent necessary
to confirm, enforce, or challenge an award of the arbitration, to protect or pursue a legal right, or as otherwise required by Applicable Law or
regulation or securities exchange, neither Party nor any arbitrator may disclose the existence, content, or results of any arbitration hereunder
without the prior written consent of both Parties.  Notwithstanding anything to the contrary in the foregoing, in no event shall an arbitration
be initiated after the date when commencement of a legal or equitable proceeding based on the dispute, controversy, or claim would be barred
by the applicable New York statute of limitations.  Any disputes concerning the propriety of the commencement of the arbitration shall be
finally settled by the arbitral tribunal.  

15.5

Interim Relief.  Notwithstanding anything herein to the contrary, nothing in this Article 15 shall preclude either Party
from seeking interim or provisional relief, including a temporary restraining order, preliminary injunction, or other interim equitable relief
concerning  a  Dispute  in  any  court  of  competent  jurisdiction  before  or  after  the  initiation  of  an  arbitration  as  set  forth  in  Section  15.4,  if
necessary to protect the interests of such Party.  This Section 15.5 shall be specifically enforceable.

16.

GENERAL PROVISIONS

16.1

Governing  Law.    This  Agreement,  and  all  questions  regarding  the  existence,  validity,  interpretation,  breach,  or
performance of this Agreement, shall be governed by, and construed and enforced in accordance with, the laws of the State of New York,
United States, without reference to its conflicts of law principles.  

16.2

Entire Agreement; Modification.  This Agreement, including the exhibits, is both a final expression of the Parties’
agreement and a complete and exclusive statement with respect to all of its terms.  This Agreement supersedes all prior and contemporaneous
agreements and communications, whether oral, written, or otherwise, concerning any and all matters contained herein.  This Agreement may
only be modified or supplemented in a writing expressly stated for such purpose and signed by the Parties to this Agreement.

16.3

Relationship  Between  the  Parties.    The  Parties’  relationship,  as  established  by  this  Agreement,  is  solely  that  of
independent contractors.  This Agreement does not create any partnership, joint venture, or similar business relationship between the Parties,
including for all tax purposes.  Neither Party is a legal representative of the other Party, and neither Party can assume or create any obligation,
representation,  warranty,  or  guarantee,  express  or  implied,  on  behalf  of  the  other  Party  for  any  purpose  whatsoever.  The  Parties  (and  any
successor, assignee, transferee,

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or confidential.

 
or  Affiliate  of  a  Party)  shall  (a)  use  commercially  reasonable  efforts  to  structure  the  arrangement  and  activities  contemplated  by  this
Agreement to avoid the arrangement contemplated by this Agreement being treated as a partnership that is engaged in a “United States trade
or business” for United States tax purposes and (b) not treat or report the relationship between the Parties arising under this Agreement as a
partnership for United States tax purposes, without the prior written consent of the other Party unless required by a final “determination” as
defined in Section 1313 of the United States Internal Revenue Code of 1986, as amended.

16.4

Non-Waiver.  The failure of a Party to insist upon strict performance of any provision of this Agreement or to exercise
any right arising out of this Agreement shall neither impair that provision or right nor constitute a waiver of that provision or right, in whole
or in part, in that instance or in any other instance.  Any waiver by a Party of a particular provision or right shall be in writing, shall be as to a
particular matter and, if applicable, for a particular period of time and shall be signed by such Party.

16.5

Assignment. Neither Party may assign or transfer this Agreement or any rights or obligations hereunder without the
prior written consent of the other Party, such consent not to be unreasonably withheld. Any successor or assignee of rights and obligations
permitted hereunder shall, in writing to the other Party, expressly assume performance of such rights and obligations. Notwithstanding the
foregoing, either Party may assign this Agreement and its rights and obligations hereunder without the other Party’s consent:

(a)

 in connection with the transfer or sale, through whatever means, of all or substantially all of its assets or the
business of such Party to which this Agreement relates (whatever by assignment, conveyance, reorganization, merger, assumption, purchase
and sale of stock, by contract or by operation of law, provided that the intellectual property rights of the acquiring party to such transaction (if
other than one of the Parties) shall not be included in the technology licensed under this Agreement; or

assigning Party, the Agreement shall be automatically assigned back to the assigning Party or its successor.  

(b)

to an Affiliate, provided that if the entity to which this Agreement is assigned ceases to be an Affiliate of the

Any permitted assignment shall be binding on the successors and the permitted assigns of a Party. Any assignment or attempted

assignment by either Party in violation of the terms of this Section 16.5 shall be null, void and of no legal effects.

16.6

Severability.  If, for any reason, any part of this Agreement is adjudicated invalid, unenforceable, or illegal by a court
of competent jurisdiction, such adjudication shall not, to the extent feasible, affect or impair, in whole or in part, the validity, enforceability,
or  legality  of  any  remaining  portions  of  this  Agreement.    All  remaining  portions  shall  remain  in  full  force  and  effect  as  if  the  original
Agreement had been executed without the invalidated, unenforceable, or illegal part.  

16.7

Notices.  Any notice to be given under this Agreement must be in writing and delivered either in person, by (a) air mail
(postage prepaid) requiring return receipt, (b) overnight courier, or (c) facsimile confirmed thereafter by any of the foregoing, to the Party to
be notified at

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or confidential.

 
its address(es) given below, or at any address such Party may designate by prior written notice to the other in accordance with this Section
16.7.  Notice shall be deemed sufficiently given for all purposes upon the earliest of:  (i) the date of actual receipt, (ii) if air mailed, five (5)
days after the date of postmark, (iii) if delivered by overnight courier, the next day the overnight courier regularly makes deliveries, or (iv) if
sent by facsimile, the date of confirmation of receipt if during the recipient’s normal business hours, otherwise the next business day.

If to Licensee, notices must be addressed to:

Angelini Pharma Rare Diseases AG
Consulting GmbH Sumpfstrasse 26 6312
Steinhausen, Zurich
Switzerland
Attention: Chief Executive Officer

With a copy to:
Angelini Pharma S.p.A.
Viale Amelia 70, 00181
Roma, Italy
Attention: Enza Maria Cristina Onnis, Global Pharma General Counsel
mail: [***]

If to Ovid, notices must be addressed to:

Ovid Therapeutics
1460 Broadway, Suite 15021
New York, NY 10036
USA
Attention:  Chief Executive Officer

And a copy to:

Attention:  General Counsel

With a copy to (which shall not constitute notice):

Cooley LLP
3175 Hanover Street
Palo Alto, CA 94304
USA
Attention: Laura Berezin

16.8

Force Majeure.  Each Party shall be excused from liability for the failure or delay in performance of any obligation
under  this  Agreement  (other  than  failure  to  make  payment  when  due)  by  reason  of  any  event  beyond  such  Party’s  reasonable  control
including Acts of God, fire, flood, explosion, earthquake, pandemic (including the COVID-19 pandemic), quarantine or similar restrictions,
or other natural forces, war, civil unrest, acts of terrorism, accident, destruction

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or confidential.

 
or  other  casualty,  any  lack  or  failure  of  transportation  facilities,  any  injunction,  order,  proclamation,  demand,  or  requirement  of  any
Governmental Authority [***], any lack or failure of supply of raw materials, or any other event similar to those enumerated above. Such
excuse from liability shall be effective only to the extent and duration of the event(s) causing the failure or delay in performance and provided
that the Party has not caused such event(s) to occur and uses reasonable efforts to overcome such event.  Notice of a Party’s failure or delay in
performance due to force majeure must be given to the other Party within [***] after its occurrence.  All delivery dates under this Agreement
that have been affected by force majeure shall be tolled for the duration of such force majeure.  In no event shall any Party be required to
prevent or settle any labor disturbance or dispute.

16.9

Interpretation.  The headings of clauses contained in this Agreement preceding the text of the sections, subsections,
and paragraphs hereof are inserted solely for convenience and ease of reference only and shall not constitute any part of this Agreement, or
have  any  effect  on  its  interpretation  or  construction.    All  references  in  this  Agreement  to  the  singular  shall  include  the  plural  where
applicable.  Unless otherwise specified, references in this Agreement to any Article shall include all Sections, subsections, and paragraphs in
such Article, references to any Section shall include all subsections and paragraphs in such Section, and references in this Agreement to any
subsection shall include all paragraphs in such subsection.  The word “including” and similar words means including without limitation.  The
word “or” means “and/or” unless the context dictates otherwise because the subjects of the conjunction are, or are intended to be, mutually
exclusive.  The words “herein”, “hereof”, and “hereunder” and other words of similar import refer to this Agreement as a whole and not to
any  particular  Section  or  other  subdivision.    All  references  to  days  in  this  Agreement  mean  calendar  days,  unless  otherwise
specified.  Ambiguities and uncertainties in this Agreement, if any, shall not be interpreted against either Party, irrespective of which Party
may be deemed to have caused the ambiguity or uncertainty to exist.  This Agreement has been prepared in the English language and the
English  language  shall  control  its  interpretation.    In  addition,  all  notices  required  or  permitted  to  be  given  hereunder,  and  all  written,
electronic, oral, or other communications between the Parties regarding this Agreement shall be in the English language.

16.10

Counterparts;  Electronic  or  Facsimile  Signatures.    This  Agreement  may  be  executed  in  any  number  of
counterparts, each of which shall be an original, but all of which together shall constitute one instrument.  This Agreement may be executed
and delivered electronically or by facsimile and upon such delivery such electronic or facsimile signature will be deemed to have the same
effect as if the original signature had been delivered to the other Party.

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or confidential.

{SIGNATURE PAGE FOLLOWS}

 
IN WITNESS WHEREOF, the Parties hereto have caused this COLLABORATION  AND LICENSE AGREEMENT  to  be  executed  and  entered

into by their duly authorized representatives as of the Effective Date.

OVID THERAPEUTICS INC.

By:  /s/ Jeremy Levin
Name:  Jeremy Levin
Title:  Chief Executive Officer

ANGELINI PHARMA RARE DISEASES AG  

By:  /s/ Pierluigi Antonelli
Name:  Pierluigi Antonelli
Title:  Chairman of the BoD

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or confidential.

 
 
 
 
 
 
 
 
 
 
 
 
 
 
List of Exhibits and Schedules

Exhibit A: Compound

Exhibit B: Ovid Patents

Exhibit C: Development Plan

Exhibit D: Press Release

Exhibit E: Technology Transfer Plan

Exhibit F: Documents to be transferred according to Section 8.1(b)(i)

Exhibit G: Other Documents to be transferred

Exhibit H: Description of Additional Pivotal Trial

Exhibit I: Current Licensee Pipeline Products

Exhibit J: Descriptions of Elara Trial, Neptune Trial, and Rocket Trial

Exhibit K: Supply Agreement

Exhibit L: Finished Product Documentation

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or confidential.

 
 
 
Exhibit A
Compound

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or confidential.

 
 
 
 
 
 
 
 
 
 
[***]

Exhibit B
Ovid Patents

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or confidential.

 
 
 
 
 
Exhibit C
Development Plan

[***]

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or confidential.

 
 
 
Exhibit D
Press Release

Ovid Therapeutics and Angelini Pharma Enter into Exclusive License Agreement to Develop, Manufacture and
Commercialize OV101 for the Treatment of Angelman Syndrome in Europe

•

•

•

Angelini Pharma obtains exclusive development, manufacturing and commercialization rights to OV101 (gaboxadol) for the
potential treatment of Angelman syndrome in the European Union and other countries in the European Economic Area,
Switzerland, Turkey and the United Kingdom

Ovid Therapeutics will receive an upfront payment of $20 million and additional payments of up to $212.5 million upon the
achievement of development, manufacturing and sales milestones, in addition to double-digit royalties on net sales if successfully
commercialized

Angelini Pharma will execute the agreement through its new affiliate Angelini Pharma Rare Diseases AG

NEW YORK and ROME, July XX, 2020 -- Ovid Therapeutics Inc. (NASDAQ: OVID, hereinafter “Ovid”), a biopharmaceutical company committed to
developing medicines that transform the lives of people with rare neurological diseases, and Angelini Pharma S.p.A. (hereinafter “Angelini Pharma”), an
Italian family-owned pharmaceutical company committed to helping patients with a constant and prevalent focus on Mental Health, Rare Diseases and
Consumer Health, announced an agreement in which Angelini Pharma will be responsible to develop, manufacture and commercialize OV101 (gaboxadol)
for the potential treatment of Angelman syndrome in the European Union, other countries in the European Economic Area, Switzerland, Turkey and
United Kingdom.  Angelini Pharma will execute the agreement through its new affiliate Angelini Pharma Rare Diseases AG. OV101 is believed to be the
only delta (δ)-selective GABAA receptor agonist in development, and is currently being evaluated in the pivotal Phase 3 NEPTUNE trial in Angelman
syndrome, with topline results expected in the fourth quarter of 2020.

Under the terms of the agreement, Ovid will receive an upfront payment of $20 million and is eligible to receive up to an additional $212.5 million in
payments upon the achievement of development,

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or confidential.

 
 
 
           
 
 
 
 
 
 
 
 
 
 
manufacturing and sales milestones for the initial indication (Angelman syndrome), as well as double-digit royalties on net sales if OV101 is successfully
commercialized. Ovid will retain all U.S. and rest-of-world commercial rights to OV101.

“We are excited to enter into a strategic collaboration with Angelini Pharma with the goal of bringing OV101, if approved, to the Angelman community in
Europe as quickly as possible. Angelini Pharma is an ideal partner for Europe as they have deep regional knowledge, an established infrastructure with a
history of successful product launches, and a commitment to improving the quality of life of the patient communities they serve,” said Jeremy Levin,
DPhil, MB, BChir, Chairman and Chief Executive Officer of Ovid Therapeutics. “Finding the right partners to bring OV101 to the Angelman community
as rapidly as possible is a core part of our global strategy. We believe this partnership with Angelini will help to maximize the potential commercial value
of OV101 and achieve our strategic objectives in this important geography."

“Today is a day that we will remember. Through our collaboration with Ovid Therapeutics, we are laying the foundation to developing innovative health
solutions for rare diseases, in line with Angelini Pharma’s new strategy,” said Pierluigi Antonelli, Angelini Pharma CEO. “The new business unit Angelini
Pharma Rare Diseases AG will contribute to the development, registration, production and, if approved, commercialization in Europe of OV101, Ovid
Therapeutics’ very promising drug being evaluated in a Phase 3 clinical trial for the treatment of Angelman syndrome. As of now, there is no effective
treatment for this rare genetic disease, characterized by severe psychomotor disability, which manifests itself from childhood. Delivering on our
commitment makes us proud both from a scientific perspective and its social impact”. 

"As shareholders and executives of Angelini Holding we continue to invest in the pharma area, which today represents half of our Group's turnover,”
commented the executive vice president Thea Paola Angelini and the CEO Sergio Marullo di Condojanni. “Our global development and
internationalization strategy focuses on business areas with high growth potential. Particularly, we look closely at all the opportunities that can open up,
not only in healthcare, but also in the consumer and machinery sector."

About Angelman Syndrome
Angelman syndrome is a rare genetic condition that is characterized by a variety of signs and symptoms. Characteristic features of this condition include
delayed development, intellectual disability, severe speech impairment, problems with movement and balance, seizures, sleep disorders and anxiety. The
most common cause of Angelman syndrome is the loss of function of the gene that codes for ubiquitin protein ligase E3A (UBE3A), which plays a critical
role in nerve cell communication, resulting in impaired tonic inhibition. Individuals with Angelman syndrome typically have normal lifespans but are
unable to live independently. Therefore, they require constant support from a network of specialists and caregivers. Angelman syndrome affects
approximately 1 in 12,000 to 1 in 20,000 people globally.

There are no approved therapies by the U.S. Food and Drug Administration (FDA), European Medicines Agency or rest–of-world for Angelman
syndrome, and treatment primarily consists of behavioral interventions and pharmacologic management of symptoms.

Angelman syndrome is associated with a reduction in tonic inhibition, a function of the delta (δ)-selective GABAA receptor that allows a human brain to
decipher excitatory and inhibitory neurological

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or confidential.

 
 
 
 
 
 
 
 
signals correctly without being overloaded. If tonic inhibition is reduced, the brain becomes inundated with signals and loses the ability to separate
background noise from critical information.

About OV101 (gaboxadol)
OV101 is believed to be the only delta (δ)-selective GABAA receptor agonist in development and the first investigational drug to specifically target the
disruption of tonic inhibition, a central physiological process of the brain that is thought to be the underlying cause of certain neurodevelopmental
disorders. OV101 has demonstrated in laboratory studies and animal models to selectively activate the δ-subunit of GABAA receptors, which are found in
the extrasynaptic space (outside of the synapse), and thereby impact neuronal activity through modulation of tonic inhibition.

Ovid is developing OV101 for the treatment of Angelman syndrome and Fragile X syndrome to potentially restore tonic inhibition and thereby address
several core symptoms of these conditions. In both these syndromes, the underlying pathophysiology includes disruption of tonic inhibition modulated
through the δ-subunit of GABAA receptors. In preclinical studies, it was observed that OV101 improved symptoms of Angelman syndrome and Fragile X
syndrome. This compound has also previously been tested in more than 4,000 patients (more than 1,000 patient-years of exposure) and was observed to
have favorable safety and bioavailability profiles. Ovid is conducting a pivotal Phase 3 clinical trial with OV101 in Angelman syndrome (NEPTUNE) and
has completed a Phase 2 signal-finding clinical trial with OV101 in Fragile X syndrome (ROCKET).

OV101 has received Rare Pediatric Disease Designation from the FDA for the treatment of Angelman syndrome. The FDA has also granted Orphan Drug
and Fast Track designations for OV101 for both the treatment of Angelman syndrome and Fragile X syndrome. In addition, the European Commission
(EC) has granted orphan drug designation to OV101 for the treatment of Angelman syndrome. The U.S. Patent and Trademark Office has granted Ovid
patents directed to methods of treating Angelman syndrome and Fragile X syndrome using OV101. The issued patents expire in 2035 without regulatory
extensions.

About Ovid Therapeutics
Ovid Therapeutics Inc. is a New York-based biopharmaceutical company using its BoldMedicine® approach to develop medicines that transform the lives
of patients with rare neurological disorders. Ovid has a broad pipeline of potential first-in-class medicines. The Company’s most advanced investigational
medicine, OV101 (gaboxadol), is currently in clinical development for the treatment of Angelman syndrome and Fragile X syndrome. Ovid is also
developing OV935 (soticlestat) in collaboration with Takeda Pharmaceutical Company Limited for the potential treatment of rare developmental and
epileptic encephalopathies (DEE). For more information on Ovid, please visit www.ovidrx.com.

About Angelini Pharma
Angelini Pharma, owned by Angelini Holding, is a pharmaceutical Company committed to helping patients with a constant and prevalent focus on Mental
Health, including Pain, Rare Diseases and Consumer Health. Angelini Pharma has an extensive and recognized R&D programs, "World Class" production
plants  and  international  commercialization  activities  of  active  ingredients  and  market-leading  drugs.  For  further  information,  please  visit
www.angelinipharma.com

About Angelini Holding

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or confidential.

 
 
 
 
 
 
 
 
Angelini Holding is the parent company of an international group operating in the pharmaceutical and consumer goods sectors. Founded in Italy in 1919,
today Angelini group operates in 17 countries with a staff of 5,600 and a turnover of €1,7 billion. In addition to the Pharmaceutical sector, Angelini group
operates in Personal and Home Care business area through Fater, a joint venture with Procter & Gamble, in the Machinery field, again in joint venture
with P&G, with the group operating in automation and robotics for the consumer goods industry Fameccanica, in Perfumery and Skincare and Suncare
with Angelini Beauty and in the Wine sector through Bertani Domains. Angelini Holding has recently entered the Baby food market as well through
MadreNatura, a joint venture with Hero Group, which offers 100% organic baby food products.

Ovid Therapeutics Forward-Looking Statements
This press release includes certain disclosures that contain “forward-looking statements,” including, without limitation, statements regarding: advancing
development of and commercializing OV101, the potential benefits and value of OV101; the anticipated reporting schedule of clinical data for OV101;
and the potential benefits and outcome from this collaboration. You can identify forward-looking statements because they contain words such as “will,”
“appears,” “believes” and “expects.” Forward-looking statements are based on Ovid’s current expectations and assumptions. Because forward-looking
statements relate to the future, they are subject to inherent uncertainties, risks and changes in circumstances that may differ materially from those
contemplated by the forward-looking statements, which are neither statements of historical fact nor guarantees or assurances of future performance.
Important factors that could cause actual results to differ materially from those in the forward-looking statements include uncertainties in the development
and regulatory approval processes, and the fact that initial data from clinical trials may not be indicative, and are not guarantees, of the final results of the
clinical trials and are subject to the risk that one or more of the clinical outcomes may materially change as patient enrollment continues and/or more
patient data become available. Additional risks that could cause actual results to differ materially from those in the forward-looking statements are set
forth in Ovid’s filings with the Securities and Exchange Commission under the caption “Risk Factors”. Such risks may be amplified by the COVID-19
pandemic and its potential impact on Ovid’s business and the global economy. Ovid assumes no obligation to update any forward-looking statements
contained herein to reflect any change in expectations, even as new information becomes available.

Ovid Therapeutics Contacts

Investors and Media:
Ovid Therapeutics Inc.
Investor Relations & Public Relations
irpr@ovidrx.com

Or

Investors:
Steve Klass
Burns McClellan, Inc.
sklass@burnsmc.com
(212) 213-0006

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or confidential.

 
 
 
 
 
 
 
 
Media:
Katie Engleman
1AB
katie@1abmedia.com

Angelini Pharma Contact:
Daniela Poggio
Head of Global Communications Angelini Pharma
+39 348 6558882
daniela.poggio@angelinipharma.com

Angelini Holding Contact:
Institutional & External Relations Director Angelini Holding
+39 348 6707240
alessandra.favilli@angeliniholding.com

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or confidential.

 
 
 
 
 
 
 
 
 
 
[***]

Exhibit E
Technology Transfer Plan

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or confidential.

 
 
 
 
 
Exhibit F
Documents to be transferred according to Section 8.1(b)(i)

[***]

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or confidential.

 
 
 
 
[***]

Exhibit G

Other Documents to be transferred

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or confidential.

 
 
 
 
 
Exhibit H
Description of Additional Pivotal Trial

[To be completed if and when the Additional Pivotal Trial is required by the EMA or by Licensee at its own discretion.] 

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or confidential.

 
 
 
 
 
Exhibit I 
Current Licensee Pipeline Products

[***]

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or confidential.

 
 
 
 
 
Exhibit J
Descriptions of Elara Trial, Neptune Trial, and Rocket Trial

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or confidential.

 
 
 
 
 
 
 
88
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
 
[***]

Exhibit K
Supply Agreement

89
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
 
 
 
 
 
 
 
LIST OF EXHIBITS

Exhibit A:

The Compound

Exhibit B:

Mandatory Estimated Forecast

Exhibit C:

Initial Purchase Order for Allocated Quantity of Compound

90
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
 
 
Exhibit A:

The Compound

91
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
 
 
Exhibit B:

Mandatory Estimated Forecast

[***]

92
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
 
 
 
 
Exhibit C:

Initial Purchase Order for Allocated Quantity of Compound

[***]

93
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
 
 
 
 
 
 
 
 
[***]

Exhibit L

Finished Product Documentation

94
Certain identified information marked with [***] has been excluded from the exhibit because it is both not material and is the type that the registrant treats as private
or confidential.

 
 
 
 
 
Consent of Independent Registered Public Accounting Firm

EXHIBIT 23.1

To Board of Directors
Ovid Therapeutics Inc.:

We consent to the incorporation by reference in the registration statements (Nos. 333-218167, 333-224033, 333-233101, and 333-237098) on Form S-8 and (No. 333-250054) on Form S-3 of
Ovid  Therapeutics  Inc.  of  our  report  dated  March  15,  2021,  with  respect  to  the  consolidated  balance  sheets  of  Ovid  Therapeutics  Inc.  as  of  December  31,  2020  and  2019,  the  related
consolidated  statements  of  operations,  comprehensive  loss,  changes  in  stockholders’  equity,  and  cash  flows  for  the  years  then  ended,  and  the  related  notes,  which  report  appears  in  the
December 31, 2020 annual report on Form 10-K of Ovid Therapeutics Inc.

/s/ KPMG LLP

New York, New York
March 15, 2021

 
 
 
CERTIFICATION PURSUANT TO RULES 13a-14(a) AND 15d-14(a) UNDER THE SECURITIES EXCHANGE ACT OF 1934, AS
ADOPTED PURSUANT TO SECTION 302 OF THE SARBANES-OXLEY ACT OF 2002

Exhibit 31.1

I, Jeremy M. Levin, certify that:

1. I have reviewed this Annual Report on Form 10-K of Ovid Therapeutics Inc.;

2. Based on my knowledge, this report does not contain any untrue statement of a material fact or omit to state a material fact necessary to make the statements
made, in light of the circumstances under which such statements were made, not misleading with respect to the period covered by this report;

3. Based on my knowledge, the financial statements, and other financial information included in this report, fairly present in all material respects the financial
condition, results of operations and cash flows of the registrant as of, and for, the periods presented in this report;

4. The registrant’s other certifying officer(s) and I are responsible for establishing and maintaining disclosure controls and procedures (as defined in Exchange Act
Rules 13a-15(e) and 15d-15(e)) and internal control over financial reporting (as defined in Exchange Act Rules 13a-15(f) and 15d-15(f)) for the registrant and
have:

(a) Designed such disclosure controls and procedures, or caused such disclosure controls and procedures to be designed under our supervision, to ensure
that material information relating to the registrant, including its consolidated subsidiaries, is made known to us by others within those entities, particularly
during the period in which this report is being prepared;

(b) Designed such internal control over financial reporting, or caused such internal control over financial reporting to be designed under our supervision, to
provide reasonable assurance regarding the reliability of financial reporting and the preparation of financial statements for external purposes in accordance
with generally accepted accounting principles;

(c) Evaluated the effectiveness of the registrant’s disclosure controls and procedures and presented in this report our conclusions about the effectiveness of
the disclosure controls and procedures, as of the end of the period covered by this report based on such evaluation; and

(d) Disclosed in this report any change in the registrant's internal control over financial reporting that occurred during the registrant's most recent fiscal
quarter (the registrant's fourth fiscal quarter in the case of an annual report) that has materially affected, or is reasonably likely to materially affect, the
registrant's internal control over financial reporting; and

5. The registrant’s other certifying officer(s) and I have disclosed, based on our most recent evaluation of internal control over financial reporting, to the
registrant’s auditors and the audit committee of the registrant’s board of directors (or persons performing the equivalent functions):

(a) All significant deficiencies and material weaknesses in the design or operation of internal control over financial reporting which are reasonably likely to
adversely affect the registrant’s ability to record, process, summarize and report financial information; and

(b) Any fraud, whether or not material, that involves management or other employees who have a significant role in the registrant’s internal control over
financial reporting.

Date: March 15, 2021

By:

/s/ Jeremy M. Levin
Jeremy M. Levin
Chief Executive Officer
(Principal Executive Officer)

 
 
 
CERTIFICATION PURSUANT TO RULES 13a-14(a) AND 15d-14(a) UNDER THE SECURITIES EXCHANGE ACT OF 1934, AS
ADOPTED PURSUANT TO SECTION 302 OF THE SARBANES-OXLEY ACT OF 2002

Exhibit 31.2

I, Timothy Daly, certify that:

1. I have reviewed this Annual Report on Form 10-K of Ovid Therapeutics Inc.;

2. Based on my knowledge, this report does not contain any untrue statement of a material fact or omit to state a material fact necessary to make the statements
made, in light of the circumstances under which such statements were made, not misleading with respect to the period covered by this report;

3. Based on my knowledge, the financial statements, and other financial information included in this report, fairly present in all material respects the financial
condition, results of operations and cash flows of the registrant as of, and for, the periods presented in this report;

4. The registrant’s other certifying officer(s) and I are responsible for establishing and maintaining disclosure controls and procedures (as defined in Exchange Act
Rules 13a-15(e) and 15d-15(e)) and internal control over financial reporting (as defined in Exchange Act Rules 13a-15(f) and 15d-15(f)) for the registrant and
have:

(a) Designed such disclosure controls and procedures, or caused such disclosure controls and procedures to be designed under our supervision, to ensure
that material information relating to the registrant, including its consolidated subsidiaries, is made known to us by others within those entities, particularly
during the period in which this report is being prepared;

(b) Designed such internal control over financial reporting, or caused such internal control over financial reporting to be designed under our supervision, to
provide reasonable assurance regarding the reliability of financial reporting and the preparation of financial statements for external purposes in accordance
with generally accepted accounting principles;

(c) Evaluated the effectiveness of the registrant’s disclosure controls and procedures and presented in this report our conclusions about the effectiveness of
the disclosure controls and procedures, as of the end of the period covered by this report based on such evaluation; and

(d) Disclosed in this report any change in the registrant's internal control over financial reporting that occurred during the registrant's most recent fiscal
quarter (the registrant's fourth fiscal quarter in the case of an annual report) that has materially affected, or is reasonably likely to materially affect, the
registrant's internal control over financial reporting; and

5. The registrant’s other certifying officer(s) and I have disclosed, based on our most recent evaluation of internal control over financial reporting, to the
registrant’s auditors and the audit committee of the registrant’s board of directors (or persons performing the equivalent functions):

(a) All significant deficiencies and material weaknesses in the design or operation of internal control over financial reporting which are reasonably likely to
adversely affect the registrant’s ability to record, process, summarize and report financial information; and

(b) Any fraud, whether or not material, that involves management or other employees who have a significant role in the registrant’s internal control over
financial reporting.

Date: March 15, 2021

By:

/s/ Timothy Daly
Timothy Daly
Executive Vice President, Finance and Corporate Controller
(Principal Financial Officer and Principal Accounting Officer)

 
 
 
 
CERTIFICATION PURSUANT TO 18 U.S.C. SECTION 1350,
AS ADOPTED PURSUANT TO
SECTION 906 OF THE SARBANES-OXLEY ACT OF 2002

Exhibit 32.1

In connection with the Annual Report on Form 10-K of Ovid Therapeutics Inc. (the “Company”) for the year ended December 31, 2020, as filed with the Securities and
Exchange Commission on the date hereof (the “Report”), each of the undersigned officers of the Company hereby certifies, pursuant to 18 U.S.C. Section 1350, that to his
or her knowledge:

(1) The Report fully complies with the requirements of Section 13(a) or 15(d) of the Securities Exchange Act of 1934; and

(2) The information contained in the Report fairly presents, in all material respects, the financial condition and results of operations of the Company.

Date: March 15, 2021

Date: March 15, 2021

By /s/ Jeremy M. Levin
Jeremy M. Levin
Chief Executive Officer
(Principal Executive Officer)

By /s/ Timothy Daly
Timothy Daly
Executive Vice President, Finance and Corporate Controller
(Principal Financial Officer and Principal Accounting Officer)