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Assembly Biosciences, Inc.

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FY2020 Annual Report · Assembly Biosciences, Inc.
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331 Oyster Point Boulevard

4th Floor

South San Francisco, CA 94080

assemblybio.com

2020 Annual Report

Passionate about making a  
profound impact on patients’ lives

Assembly Bio is an ambitious clinical stage biopharmaceutical company 
with cutting-edge therapeutic product candidates capable of improving 
the lives of millions living with chronic hepatitis B virus (HBV) infection 
around the world.

DEAR FELLOW STOCKHOLDERS,

2020 was one of the most uniquely difficult years in recent 

history as the world was — and continues to be — gripped 

by the COVID-19 global health crisis. We witnessed the 

commitment and perseverance of countless life science 

companies that, within just one year, launched thousands 

of clinical trials to evaluate treatment approaches and 

delivered three vaccines. I am proud to be among the 

biotech companies focused in virology and now even 

more impassioned to accomplish what Assembly 

Biosciences has always believed to be possible — freeing 

patients from the burden of lifelong treatment for chronic 

hepatitis B virus (HBV) infection.

At Assembly Bio, 2020 was a year of significant progress 

and also one of learning. 

We had hoped that our lead core 

inhibitor (CI) product, vebicorvir (VBR), 

in combination with standard-of-care 

improving  current chronic suppressive 

therapy. This decision was made after 

internal and external discussions and 

nucleos(t)ide (Nrtl) therapy, would achieve 

analyses, including those with HBV experts, 

an improvement in sustained virologic 

the FDA and, with respect to China, our 

response (SVR) off-treatment versus NrtI 

partner BeiGene. Seeking to address the 

alone, given the safety and deeper viral 

most significant unmet need for HBV 

suppression demonstrated in our Phase 2 

patients — a finite treatment designed to 

studies. We also believed that if we could 

cure — provides us the greatest potential to 

bring a cure to more than 270 million 

patients today, we owed it to them to 

create value for the company's stockholders, 

while leveraging the expertise and passion 

explore that. Though the study did not 

of our management and entire organization. 

achieve a favorable SVR result, we recognize 

that the insights from this trial further 

inform our work and the HBV field as a 

With our focused strategy, the partnerships we 

established in 2020 and cash to fund operations 

whole. More recently, we also updated our 

into 2023, we are well positioned to continue 

pipeline strategy to now focus solely on 

advancing our portfolio of HBV core inhibitor 

the pursuit of finite and curative therapies 

clinical candidates and growing our pipeline 

and forgo registrational studies aimed at 

of discovery programs toward this goal.

Passionate about making a  

profound impact on patients’ lives

Assembly Bio is an ambitious clinical stage biopharmaceutical company 

with cutting-edge therapeutic product candidates capable of improving 

the lives of millions living with chronic hepatitis B virus (HBV) infection 

around the world.

DEAR FELLOW STOCKHOLDERS,

2020 was one of the most uniquely difficult years in recent 
history as the world was — and continues to be — gripped 
by the COVID-19 global health crisis. We witnessed the 
commitment and perseverance of countless life science 
companies that, within just one year, launched thousands 
of clinical trials to evaluate treatment approaches and 
delivered three vaccines. I am proud to be among the 
biotech companies focused in virology and now even 
more impassioned to accomplish what Assembly 
Biosciences has always believed to be possible — freeing 
patients from the burden of lifelong treatment for chronic 
hepatitis B virus (HBV) infection.

At Assembly Bio, 2020 was a year of significant progress 
and also one of learning. 

We had hoped that our lead core 
inhibitor (CI) product, vebicorvir (VBR), 
in combination with standard-of-care 
nucleos(t)ide (Nrtl) therapy, would achieve 
an improvement in sustained virologic 
response (SVR) off-treatment versus NrtI 
alone, given the safety and deeper viral 
suppression demonstrated in our Phase 2 
studies. We also believed that if we could 
bring a cure to more than 270 million 
patients today, we owed it to them to 
explore that. Though the study did not 
achieve a favorable SVR result, we recognize 
that the insights from this trial further 
inform our work and the HBV field as a 
whole. More recently, we also updated our 
pipeline strategy to now focus solely on 
the pursuit of finite and curative therapies 
and forgo registrational studies aimed at 

improving  current chronic suppressive 
therapy. This decision was made after 
internal and external discussions and 
analyses, including those with HBV experts, 
the FDA and, with respect to China, our 
partner BeiGene. Seeking to address the 
most significant unmet need for HBV 
patients — a finite treatment designed to 
cure — provides us the greatest potential to 
create value for the company's stockholders, 
while leveraging the expertise and passion 
of our management and entire organization. 

With our focused strategy, the partnerships we 
established in 2020 and cash to fund operations 
into 2023, we are well positioned to continue 
advancing our portfolio of HBV core inhibitor 
clinical candidates and growing our pipeline 
of discovery programs toward this goal.

Our HBV Program:  
Where We Are Today

POTENT NEXT-GENERATION  
CORE INHIBITORS

•  ABI-H2158 (2158): Phase 2 study 
is ongoing with interim data 
anticipated in the second half  
of 2021. 

•  ABI-H3733 (3733): Phase 1a study 
completed in healthy subjects.

•  Fourth Core Inhibitor Candidate: 
New candidate on track to be 
nominated during the first half  
of 2021 with a potential best-in-
class profile. 

PROOF-OF-CONCEPT COMBINATION 
STUDIES WITH OTHER 
COMPLEMENTARY MECHANISMS

•  VBR + NrtI + interferon (peg-IFNα): 

Phase 2a initiated.

•  VBR + NrtI + RNAi: Phase 2 initiated. 

•  Additional Combinations: Further 
potential studies are under review 
to build upon the VBR + NrtI 
antiviral backbone by evaluating 
the addition of one or more 
complementary mechanisms  
of action.

RESEARCH PROGRAMS ON NEW 
TARGETS

•  Core Protein cccDNA Disruptors: 
Complementary to our portfolio of 
core inhibitors. 

•  Novel HBV Targets: Initiation of 

two additional internal programs 
evaluating differentiated and 
undisclosed targets.

Updated Pipeline Strategy: Three 
Key Components to Drive Progress

Our HBV pipeline of core inhibitors is 
comprised of the most advanced and 
potentially best-in-class core inhibitors 
in development. We believe that core 
inhibitors administered with NrtI will form 
the backbone for finite and curative HBV 
combination therapies, and this approach is 
central to the three key components of our 
updated pipeline strategy:  

•  Data-driven advancement of our core 

inhibitor candidates. We have three core 
inhibitors in various stages of clinical 
development, VBR, ABI-H2128 and 
ABI-H3733, as well as a fourth discovery 
compound that we plan to nominate 
during the first half of 2021. With different 
chemical scaffolds, each candidate offers 
a unique profile and opportunity to more 
deeply suppress viral replication and 
prevent the formation of new cccDNA. The 
ultimate goal is to choose the best core 
inhibitors to move forward in future studies 
of finite and curative combinations. 

•  Advancement of proof-of-concept 

In 2020, we also accomplished a number of 

multi-drug combination studies. With 
a favorable safety profile and Phase 2 
data already in hand, we are initially 
evaluating VBR combined with Nrtl as the 
antiviral backbone in triple-combination 
studies with a third mechanism in 
treating patients with chronic HBV. We 
initiated two of these studies during the 
first quarter of 2021, one with Arbutus 
Biopharma’s GalNAc delivered RNAi 
therapeutic candidate, AB-729, and the 
other with interferon. 

•  Expansion of our discovery programs, 

both internally and externally. During the 

•  Initiating a Phase 2 trial of our second-

John McHutchison, AO, MD

generation core inhibitor candidate,  

Chief Executive Officer and President

past year, we made significant strides in 

ABI-2158, for chronic HBV infection and 

the expansion of our pipeline of research 

later receiving FDA Fast Track Designation 

programs leveraging the strength of our 

for its development and review. 

research and development expertise in 

virology and HBV specifically. Through  

an external collaboration, we obtained  

the rights to a develop a novel class 

of HBV cccDNA disruptors targeting 

different phases of the HBV viral 

replication cycle distinct f rom and 

complementary to those targeted by 

our existing pipeline. In addition to 

the fourth CI compound, the team 

identified two additional novel targets, 

and we are focusing discovery efforts 

on generating compounds against 

them. We believe that our internal and 

external discovery programs and targets 

are differentiated in the space and have 

the potential to accelerate our progress 

toward the development of finite and 

curative therapies.

Continued Corporate and Scientific 

Momentum: 2020 in Retrospect

other important goals, including: 

•  Continuing to strengthen our leadership 

team and board of directors with the 

appointments of Chief Scientific Officer, 

Virology, William Delaney, PhD; Chief Legal 

and Business Officer, Jason Okazaki; Senior 

Vice President of Corporate Development, 

Carl Enell; Senior Vice President of 

Pharmaceutical Development and 

Manufacturing, Nicole White, PhD;  

and board member, Gina Consylman. 

•  Forming new partnerships, including: a 

licensing and collaboration agreement 

with BeiGene for our three clinical-stage 

core inhibitors in the China Territory 

(including Taiwan, Macau and Hong 

Kong); a clinical collaboration agreement 

to evaluate VBR in combination with 

Arbutus Biopharma’s AB-729 and Nrtl 

therapy; and a collaboration and option 

agreement with Door Pharmaceuticals  

for a novel class of cccDNA disruptors.

•  Winding-down our microbiome program 

in the first quarter of 2021, focusing our 

strategy and resources on finite and 

curative therapies for HBV.

As I look back, I’m reminded of the tenacity 

and flexibility that our team showed while 

navigating 2020’s personal and professional 

challenges. It’s a privilege to work alongside 

our talented and experienced team that 

brings years of extensive HBV and virology 

experience to the company, as well as a track 

record executing in viral hepatitis. 

With our refined strategy, strong resources, 

and focused discovery and development 

programs, I am excited for what the future 

brings along our path to developing finite 

and curative HBV therapies. We look forward 

to updating you as things progress. 

Wishing you good health, 

Our HBV Program:  

Where We Are Today

POTENT NEXT-GENERATION  

CORE INHIBITORS

•  ABI-H2158 (2158): Phase 2 study 

is ongoing with interim data 

anticipated in the second half  

of 2021. 

•  ABI-H3733 (3733): Phase 1a study 

completed in healthy subjects.

•  Fourth Core Inhibitor Candidate: 

New candidate on track to be 

nominated during the first half  

of 2021 with a potential best-in-

class profile. 

PROOF-OF-CONCEPT COMBINATION 

STUDIES WITH OTHER 

COMPLEMENTARY MECHANISMS

•  VBR + NrtI + interferon (peg-IFNα): 

Phase 2a initiated.

•  VBR + NrtI + RNAi: Phase 2 initiated. 

•  Additional Combinations: Further 

potential studies are under review 

to build upon the VBR + NrtI 

antiviral backbone by evaluating 

the addition of one or more 

complementary mechanisms  

of action.

RESEARCH PROGRAMS ON NEW 

TARGETS

•  Core Protein cccDNA Disruptors: 

Complementary to our portfolio of 

core inhibitors. 

•  Novel HBV Targets: Initiation of 

two additional internal programs 

evaluating differentiated and 

undisclosed targets.

Updated Pipeline Strategy: Three 

Key Components to Drive Progress

Our HBV pipeline of core inhibitors is 

comprised of the most advanced and 

potentially best-in-class core inhibitors 

in development. We believe that core 

inhibitors administered with NrtI will form 

the backbone for finite and curative HBV 

combination therapies, and this approach is 

central to the three key components of our 

updated pipeline strategy:  

•  Data-driven advancement of our core 

inhibitor candidates. We have three core 

inhibitors in various stages of clinical 

development, VBR, ABI-H2128 and 

ABI-H3733, as well as a fourth discovery 

compound that we plan to nominate 

during the first half of 2021. With different 

chemical scaffolds, each candidate offers 

a unique profile and opportunity to more 

deeply suppress viral replication and 

prevent the formation of new cccDNA. The 

ultimate goal is to choose the best core 

inhibitors to move forward in future studies 

of finite and curative combinations. 

•  Advancement of proof-of-concept 

multi-drug combination studies. With 

a favorable safety profile and Phase 2 

data already in hand, we are initially 

evaluating VBR combined with Nrtl as the 

antiviral backbone in triple-combination 

studies with a third mechanism in 

treating patients with chronic HBV. We 

initiated two of these studies during the 

first quarter of 2021, one with Arbutus 

Biopharma’s GalNAc delivered RNAi 

therapeutic candidate, AB-729, and the 

other with interferon. 

past year, we made significant strides in 
the expansion of our pipeline of research 
programs leveraging the strength of our 
research and development expertise in 
virology and HBV specifically. Through  
an external collaboration, we obtained  
the rights to a develop a novel class 
of HBV cccDNA disruptors targeting 
different phases of the HBV viral 
replication cycle distinct f rom and 
complementary to those targeted by 
our existing pipeline. In addition to 
the fourth CI compound, the team 
identified two additional novel targets, 
and we are focusing discovery efforts 
on generating compounds against 
them. We believe that our internal and 
external discovery programs and targets 
are differentiated in the space and have 
the potential to accelerate our progress 
toward the development of finite and 
curative therapies.

Continued Corporate and Scientific 
Momentum: 2020 in Retrospect

In 2020, we also accomplished a number of 
other important goals, including: 

•  Continuing to strengthen our leadership 
team and board of directors with the 
appointments of Chief Scientific Officer, 
Virology, William Delaney, PhD; Chief Legal 
and Business Officer, Jason Okazaki; Senior 
Vice President of Corporate Development, 
Carl Enell; Senior Vice President of 
Pharmaceutical Development and 
Manufacturing, Nicole White, PhD;  
and board member, Gina Consylman. 

ABI-2158, for chronic HBV infection and 
later receiving FDA Fast Track Designation 
for its development and review. 

•  Forming new partnerships, including: a 
licensing and collaboration agreement 
with BeiGene for our three clinical-stage 
core inhibitors in the China Territory 
(including Taiwan, Macau and Hong 
Kong); a clinical collaboration agreement 
to evaluate VBR in combination with 
Arbutus Biopharma’s AB-729 and Nrtl 
therapy; and a collaboration and option 
agreement with Door Pharmaceuticals  
for a novel class of cccDNA disruptors.

•  Winding-down our microbiome program 
in the first quarter of 2021, focusing our 
strategy and resources on finite and 
curative therapies for HBV.

As I look back, I’m reminded of the tenacity 
and flexibility that our team showed while 
navigating 2020’s personal and professional 
challenges. It’s a privilege to work alongside 
our talented and experienced team that 
brings years of extensive HBV and virology 
experience to the company, as well as a track 
record executing in viral hepatitis. 

With our refined strategy, strong resources, 
and focused discovery and development 
programs, I am excited for what the future 
brings along our path to developing finite 
and curative HBV therapies. We look forward 
to updating you as things progress. 

Wishing you good health, 

•  Expansion of our discovery programs, 

both internally and externally. During the 

•  Initiating a Phase 2 trial of our second-
generation core inhibitor candidate,  

John McHutchison, AO, MD
Chief Executive Officer and President

UNITED STATES
SECURITIES AND EXCHANGE COMMISSION
WASHINGTON, DC 20549
FORM 10-K

☒ ANNUAL REPORT PURSUANT TO SECTION 13 OR 15(d) OF THE SECURITIES EXCHANGE ACT OF 1934

For the fiscal year ended December 31, 2020
or

☐ TRANSITION REPORT PURSUANT TO SECTION 13 OR 15(d) OF THE SECURITIES EXCHANGE ACT OF 1934

For the Transition Period from __________ to __________

Commission File Number: 001-35005
ASSEMBLY BIOSCIENCES, INC.
(Exact name of registrant specified in its charter)

Delaware
(State or Other Jurisdiction of
Incorporation or Organization)

20-8729264
(I.R.S. Employer
Identification No.)

331 Oyster Point Blvd., Fourth Floor
South San Francisco, California 94080
(Address of Principal Executive Offices)

Registrant’s telephone number, including area code: (833) 509-4583

Securities Registered Pursuant to Section 12(b) of the Exchange Act:

Title of Each Class
Common Stock, $0.001 Par Value

Trading Symbol(s)
ASMB

Name of Exchange on which Registered
The Nasdaq Global Select Market

Securities Registered Pursuant to Section 12(g) of the Act: None

 No   ☒

Indicate by check mark if the registrant is a well-known seasoned issuer, as defined in Rule 405 of the Securities Act. Yes   ☐    No     ☒
Indicate  by  check  mark  if  the  registrant  is  not  required  to  file  reports  pursuant  to  Section 13  or  Section 15(d)  of  the  Exchange  Act. 
Yes   ☐  
Indicate by check mark whether the registrant (1) has filed all reports required to be filed by Section 13 or 15(d) of the Securities Exchange Act 
of 1934 during the preceding 12 months (or for such shorter period that the registrant was required to file such reports), and (2) has been subject 
to such filing requirements for the past 90 days.  Yes     ☒  
Indicate by check mark whether the registrant has submitted electronically every Interactive Data File required to be submitted pursuant to Rule 
405 of Regulation S-T (§ 232.45 of this chapter) during the preceding 12 months (or for such shorter period that the registrant was required to 
submit such files). Yes     ☒  
Indicate  by  check  mark  whether  the  registrant  is  a  large  accelerated  filer,  an  accelerated  filer,  a  non-accelerated  filer,  a  smaller  reporting 
company, or an emerging growth company. See the definitions of “large accelerated filer,” “accelerated filer,” “smaller reporting company,” and 
“emerging growth company” in Rule 12b-2 of the Exchange Act:

 No     ☐

 No     ☐

Large accelerated filer

Non-accelerated filer

☒

☐

Accelerated filer

Smaller reporting company

Emerging growth company

☐

☐

☐

If an emerging growth company, indicate by check mark if the registrant has elected not to use the extended transition period for complying with 
any new or revised financial accounting standards provided pursuant to Section 13(a) of the Exchange Act.   ☐
Indicate  by  check  mark  whether  the  registrant  has  filed  a  report  on  and  attestation  to  its  management’s  assessment  of  the  effectiveness  of  its 
internal control over financial reporting under Section 404(b) of the Sarbanes-Oxley Act (15 U.S.C. 7262 (b)) by the registered public accounting 
firm that prepared or issued its audit report.    ☒

Indicate by check mark whether the registrant is a shell company (as defined in Rule 12b-2 of the Exchange Act). Yes   ☐   No       ☒
The aggregate market value of the voting stock held by non-affiliates of the registrant, as of June 30, 2020, was $756.9 million. Such aggregate 
market value was computed by reference to the closing price of the common stock as reported on the Nasdaq Global Select Market on June 30, 
2020. For purposes of making this calculation only, the registrant has defined affiliates as including only (1) directors, (2) executive officers and 
(3) certain  stockholders,  if  any,  that  hold  greater  than  10%  of  the  voting  stock  of  the  registrant,  in  each  case,  as  of  June  30,  2020.  Shares  of 
common stock held by other persons, including certain other holders of more than 10% of the registrant’s outstanding common stock, if any, have 
not  been  excluded  from  the  above  calculation  in  that  such  persons  are  not  deemed  to  be  affiliates.  The  determination  of  affiliate  status  is  not 
necessarily a conclusive determination for other purposes.
As of February 22, 2021, there were 38,246,092 shares of the registrant’s common stock, $0.001 par value per share, outstanding.

DOCUMENTS INCORPORATED BY REFERENCE
Part III  of  this  Annual  Report  on  Form  10-K  incorporates  information  by  reference  to  portions  of  the  definitive  proxy  statement  for  the 
Company’s Annual Meeting of Stockholders to be held in 2021, to be filed within 120 days of the registrant’s fiscal year ended December 31, 
2020.

 
 
 
 
 
 
 
ASSEMBLY BIOSCIENCES, INC.
TABLE OF CONTENTS

PART I
Item 1.
Business.......................................................................................................................................
Item 1A. Risk Factors .................................................................................................................................
Item 1B. Unresolved Staff Comments........................................................................................................
Properties.....................................................................................................................................
Item 2.
Legal Proceedings .......................................................................................................................
Item 3.
Item 4.
Mine Safety Disclosures..............................................................................................................
PART II
Item 5.

Market for Registrant’s Common Equity, Related Stockholder Matters and Issuer
Purchases of Equity Securities ....................................................................................................
Selected Financial Data ...............................................................................................................
Item 6.
Management’s Discussion and Analysis of Financial Condition and Results of Operation.......
Item 7.
Item 7A. Quantitative and Qualitative Disclosures about Market Risk .....................................................
Financial Statements and Supplementary Data ...........................................................................
Item 8.
Item 9.
Changes in and Disagreements with Accountants on Accounting and Financial Disclosure .....
Item 9A. Controls and Procedures..............................................................................................................
Item 9B. Other Information........................................................................................................................
PART III
Item 10. Directors, Executive Officers and Corporate Governance ..........................................................
Executive Compensation .............................................................................................................
Item 11.
Security Ownership of Certain Beneficial Owners and Management and Related
Item 12.
Stockholder Matters.....................................................................................................................
Certain Relationships and Related Transactions, and Director Independence............................
Item 13.
Principal Accounting Fees and Services .....................................................................................
Item 14.
Exhibits, Financial Statement Schedules.....................................................................................
Item 15.
Item 16.
Form 10-K Summary...................................................................................................................
Financial Statements ......................................................................................................................................

Page

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33
36
37
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54
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55

56
56

56
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56
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58
F-1

i

References to Assembly Biosciences, Inc.

Throughout this Annual Report on Form 10-K, the “Company,” “Assembly,” “we,” “us,” and “our,” except where 
the context requires otherwise, refer to Assembly Biosciences, Inc. and its consolidated subsidiaries, and “our board 
of directors” refers to the board of directors of Assembly Biosciences, Inc.

Forward-Looking Statements

This  Annual  Report  on  Form 10-K  contains  “forward-looking  statements”  that  are  subject  to  certain  risks  and 
uncertainties, including, without limitation, those set forth in Part I, Item 1A under the heading “Risk Factors,” that 
could cause actual results to materially differ. The forward-looking statements in this Annual Report on Form 10-K 
include, among other things, statements about:

(cid:129)

(cid:129)

(cid:129)

(cid:129)

(cid:129)

(cid:129)

our ability to initiate and complete clinical trials involving our chronic hepatitis B virus (HBV) therapeutic 
product candidates in the currently anticipated timeframes;

safety  and  efficacy  data  from  clinical  studies  may  not  warrant  further  development  of  our  product 
candidates;

clinical  and  nonclinical  data  presented  at  conferences  may  not  differentiate  our  product  candidates  from 
other companies’ candidates;

continued development and commercialization of our HBV product candidates will be dependent on, and 
subject to, our collaboration agreement governing our activity in the China territory;

our  ability  to  maintain  financial  resources  necessary  to  continue  our  clinical  studies  and  fund  business 
operations; and

any impact that the COVID-19 pandemic may have on our business and operations, including initiation and 
continuation of our clinical studies or timing of discussions with regulatory authorities.

You are urged to consider statements that include the words may, will, would, could, should, might, believes, hopes, 
estimates, projects, potential, expects, plans, anticipates, intends, continues, forecast, designed, goal or the negative 
of  those  words  or  other  comparable  words  to  be  uncertain  and  forward-looking.  We  intend  such  forward-looking 
statements to be covered by the safe harbor provisions contained in Section 27A of the Securities Act of 1933, as 
amended (the Securities Act), and Section 21E of the Securities Exchange Act of 1934, as amended (the Exchange 
Act).  Except  as  required  by  law,  we  assume  no  obligation  to  update  publicly  any  forward-looking  statements, 
whether as a result of new information, future events or otherwise.

ii

PART I

Item 1. Business

Overview

We  are  a  clinical-stage  biotechnology  company  advancing  a  novel  class  of  oral  therapeutic  candidates  for  the 
treatment  of  chronic  hepatitis  B  virus  (HBV)  infection.  According  to  the  World  Health  Organization  (WHO), 
approximately  270  million  people  worldwide  are  chronically  infected  with  HBV.  Our  research  and  development 
programs  are  pursuing  multiple  drug  candidates  designed  to  inhibit  the  HBV  replication  cycle  and  block  the 
generation  of  covalently  closed  circular  DNA  (cccDNA),  with  the  aim  of  discovering  and  developing  finite  and 
curative  therapies  for  patients  with  HBV.  We  have  discovered  several  novel  core  inhibitors,  which  are  small 
molecules that directly target and allosterically modulate the HBV core (HBc) protein in a way that affects assembly 
and stability of HBV nucleocapsids.

The  ongoing  COVID-19  pandemic  has  affected  certain  aspects  of  our  business.  As  further  detailed  below,  those 
effects  have  been  primarily  limited  to  where  and  how  our  employees  work  in  our  labs  and  offices.  To  date,  our 
current  and  future  planned  clinical  trials  and  pre-clinical  studies  have  not  been  subject  to  significant  impact  as  a 
result of the COVID-19 pandemic.

As previously announced, in January 2021, we wound down our Microbiome program to prioritize and focus our 
resources on discovering and developing finite and curative therapies for HBV. Our Microbiome program had been 
developing a novel class of oral live microbial biotherapeutics candidates designed to treat disorders associated with 
the microbiome.

HBV Background

HBV is a leading global cause of chronic liver disease and liver transplants. The WHO estimates that approximately 
270 million people worldwide are infected with HBV and 887,000 people died in 2015 as a result of HBV, mostly 
from complications, including cirrhosis and hepatocellular carcinoma. HBV is a global epidemic and infects more 
than  twice  the  number  of  people  infected  with  hepatitis  C  virus  and  HIV  infections  combined,  according  to  the 
WHO  as  of  the  end  of  2019.  Of  the  approximately  270  million  people  living  with  HBV  infection,  only 
approximately  30  million  were  aware  of  their  infection,  and  only  approximately  5  million  of  those  diagnosed 
received treatment. Few treated patients exhibit cure, defined herein as sustained viral suppression (more than six 
months) of HBV DNA (less than the lower limit of quantification (LLOQ)) after a finite duration of therapy.

Current Treatments

There have been no new mechanisms used to treat chronic HBV approved in 25 years. Current therapeutic options 
for HBV include:

antiviral  medications—including 

(cid:129) Direct  Acting  Antiviral  medications  (Nucelos(t)ide  analog  reverse  transcriptase  inhibitors  (NrtIs)). 
Several 
(Hepsera®), 
telbivudine (Tyzeka®),  tenofovir  alafenamide  (Vemlidy®),  tenofovir  disoproxil  fumarate  (Viread®)  and 
entecavir  (Baraclude®)—effectively  reduce  circulating  virus  levels  by  inhibiting  reverse  transcription. 
Chronic  therapy  with  these  agents  can  result  in  reduced  liver  inflammation  and  fibrosis.  Unfortunately, 
these are rarely curative, even after years of therapy, and viral replication resumes when therapy is stopped.

lamivudine 

(Epivir®), 

adefovir 

(cid:129)

Pegylated Interferon alfa (Peg-IFNα or interferon). This synthetic version of a substance produced by 
the body to fight infection is used mainly for people infected with HBV who do not want to undergo long-
term treatment (e.g., patients who might want to become pregnant within a few years). It is administered by 
injection.  Cure  rates  are  relatively  low  and  side  effects  may  be  severe,  including  flu-like  symptoms  and 
depression.

1

Business Strategy

Our  goal  is  to  discover  and  develop  finite  and  curative  therapies  for  those  chronically  infected  with  HBV.  Our 
efforts to forge a new and differentiated path to develop finite and curative therapies for chronic HBV infection are 
inspired by the millions living with this condition worldwide. While we have learned that combination therapy of 
our first-generation core inhibitor product candidate, vebicorvir (VBR), with NrtIs alone will not result in a finite 
and  curative  treatment,  we  believe  that  a  regimen  of  core  inhibitors  in  combination  with  NrtI  therapy  will  be  the 
antiviral  backbone  of  future  finite  and  curative  therapies.  As  a  result,  our  business  strategy  is  focused  on  three 
parallel paths:

(cid:129) Developing  and  advancing  VBR,  ABI-H2158  (2158)  and  ABI-H3733  (3733),  our  current  clinical-stage 
core inhibitor product candidates, and identifying and selecting a fourth-generation core inhibitor product 
candidate with a profile superior to 2158 and 3733;

(cid:129) Assessing core inhibitors in multi-drug combination studies, adding non-overlapping mechanisms of action 

to the core inhibitor + NrtI backbone; and

(cid:129) Discovering and developing additional compounds beyond core inhibitors, including a cccDNA disruptor 

and a number of other recently initiated novel pre-clinical programs.

With respect to our core inhibitor pipeline, we have concise, data-driven development plans to enable selection of 
the  optimal  core  inhibitor  to  advance  for  finite  and  curative  combination  therapies  for  HBV.  We  intend  to 
complement  our  core  inhibitor  programs  with  additional  new  mechanisms  of  action  discovered  and  developed 
internally  as  well  as  externally  through  collaborations,  licenses,  partnerships  and  other  types  of  business 
arrangements.

Our Primary Focus: Targeting HBV Core Protein to Achieve a Cure 

HBV  is  a  DNA  virus  that  infects  hepatocytes  and  establishes  a  reservoir  of  cccDNA,  a  unique  DNA  moiety  that 
resides  in  the  cell  nucleus  of  HBV-infected  hepatocytes  and  is  associated  with  viral  persistence  and  chronic 
infection.  No  currently  approved  oral  therapies  target  cccDNA  activity  directly,  which  makes  molecules  that  can 
modulate  cccDNA  generation  or  disrupt  its  function  highly  sought  in  the  HBV  field.  As  a  result,  most  of  our 
research and development efforts to date have focused on discovering and developing compounds targeting the core 
protein,  a  highly  conserved  viral  structural  protein  that  has  no  human  homologue  and  is  involved  in  numerous 
aspects of the HBV replication cycle, including the generation of HBV cccDNA. Through our research efforts, we 
have  discovered  several  chemically  distinct  series  of  small  molecule  core  inhibitors  that  directly  target  and 
allosterically  inhibit  core  protein  functions.  Our  pipeline  therefore  offers  the  potential  for  both  first-in-class  and 
best-in-class  compounds  that  target  critical  steps  involved  in  cccDNA  generation  and  the  HBV  viral  replication 
cycle.  We  believe  that  our  approach  of  targeting  viral  core  protein  and  its  related  functions  provides  a  promising 
foundation for finite and curative HBV treatment regimens.

A  benchmark  for  therapeutic  agents  aiming  to  decrease  cccDNA  levels  is  the  use  of  several  key  viral  antigens  as 
surrogate biomarkers of active cccDNA. The same biomarkers can be used in both primary human hepatocyte cells 
and patients. On this basis, our core inhibitors have shown preclinical proof of principle. In a variety of cell culture 
models, core inhibitors have demonstrated the ability to reduce production of viral HBV DNA levels as well as the 
surrogate markers for cccDNA establishment: HBV e antigen (HBeAg), HBV core related antigen (HBcrAg), and 
viral pre-genomic RNA (pgRNA). 

In pursuit of our goal of developing finite and curative therapies for patients with chronic HBV infection, we plan on 
advancing  the  optimal  core  inhibitor  in  our  portfolio  for  use  as  an  anti-viral  backbone  with  NrtI.  While  we  have 
three candidates in clinical studies and are working towards identifying a fourth-generation candidate later this year, 
we will follow a disciplined, data-driven approach to identify the optimal candidate(s) to produce potentially higher 
cure rates than are currently obtainable for patients with chronic HBV infection under the current standard of care.

Our Core Inhibitor Product Candidates

Our clinical strategy encompasses testing core inhibitors first as a monotherapy in Phase 1, as required by regulatory 
agencies, to demonstrate their intrinsic antiviral activity and safety and subsequently in Phase 2 in combination with 
NrtI and potentially other classes of HBV therapies.

2

Vebicorvir

VBR,  our  lead  core  inhibitor  product  candidate,  is  licensed  from  Indiana  University.  The  conduct  of  the  Phase  2 
studies, Study 201 and 202 and our open-label extension study, Study 211, are all complete. We presented interim 
updates on our clinical studies at a variety of conferences, including at the European Association for the Study of the 
Liver’s (EASL) Digital International Liver CongressTM in August 2020 and the American Association for the Study 
of Liver Diseases (AASLD) Annual Meeting in November 2020.

Our  most  recently  completed  study  for  VBR,  Study  211,  involved  transitioning  patients  who  met  the  requisite 
stopping criteria, as determined with our lead investigators and the U.S. Food and Drug Administration (FDA), off 
of therapy to test for sustained virologic response (SVR). SVR refers to sustained viral suppression (more than six 
months)  of  HBV  DNA  below  LLOQ  and  would  be  consistent  with  a  successful  finite  treatment  for  HBV.  In 
November 2020, it became clear that patients who stopped therapy in Study 211 had not achieved meaningful SVR 
rates as 39 of 41 patients relapsed, meaning they had detectable HBV. We continue to analyze Study 211 data and 
intend to submit more detailed findings to a future medical meeting; however, it is clear that combination therapy of 
VBR  plus  NrtI  alone  is  not  sufficient  to  cure  HBV.  Based  on  these  results,  we  terminated  Study  211  prior  to  its 
completion.

Despite the off-treatment results in Study 211, the Phase 2 studies demonstrated on-treatment that subjects receiving 
VBR plus NrtI achieved faster and deeper suppression of viral replication compared to placebo. Based on this data, 
we  believed  that  the  addition  of  VBR  to  NrtI  therapy  could  potentially  help  two  patient  populations  as  a  chronic 
suppressive  treatment  (CST):  (1)  treatment-naïve  patients,  for  whom  addition  of  VBR  to  NrtI  could  lead  to  faster 
and  deeper  viral  suppression  and  (2)  partially  virologically  suppressed  patients  who  continue  to  have  viral  levels 
above LLOQ by commercial assays, for whom the addition of VBR to NrtI could suppress viral levels below what 
could be achieved by NrtI alone.

In connection with preparation for registrational studies for VBR in CST in 2020, we held a number of discussions 
with leading viral hepatitis experts regarding use of VBR as a CST. In addition, we initiated an additional Phase 2 
study  of  VBR,  Study  205,  to  evaluate  treatment  intensification  with  VBR  in  patients  with  chronic  HBV  infection 
who are only partially virologically suppressed on NrtI. 

In  the  second  half  of  2020,  we  also  held  an  End-of-Phase  2  meeting  with  the  National  Medical  Products 
Administration, Center for Drug Evaluation, China, and reached agreement on a Phase 3 registrational program for 
CST  use  of  VBR  plus  NrtI.  We  also  had  discussions  with  the  FDA  regarding  the  same  Phase  3  registrational 
program.

Based  on  discussions  with  leading  viral  hepatitis  experts,  global  regulatory  discussions  and  feedback,  and,  with 
respect to the China territory, discussions and agreement with our collaboration partner, BeiGene, Ltd. (BeiGene), 
we  recently  decided  to  not  move  forward  with  the  global  registrational  studies  for  VBR  as  a  chronic  suppressive 
treatment (CST) with NrtI. The decision was made to focus on the greatest unmet medical need of patients, which 
lies  predominantly  in  cure,  rather  than  CST.  As  a  result,  we  also  expect  to  terminate  Study  205,  as  we  focus  our 
efforts with VBR moving forward in combination with NrtI and additional mechanisms targeting finite and curative 
combination therapy.

ABI-H2158

Our  second-generation  core  inhibitor  product  candidate,  2158,  was  internally  discovered  and  developed  and  is 
chemically distinct from VBR.

We  reported  the  final  data  from  dose-ranging  cohorts  of  the  Phase  1b  portion  of  the  Phase  1a/1b  dose-ranging 
clinical study at EASL in August 2020. Based on data from the Phase 1b dose-ranging study, we initiated a Phase 2 
clinical study in June 2020 using a 300 mg daily dose of 2158. This study is being conducted in approximately ten 
countries in Asia, North America and Europe. We expect interim data from this study in the second half of 2021. 
While we will continue to monitor the situation closely, at this time, we do not expect our timelines for this study to 
be significantly impacted by the COVID-19 pandemic. 

ABI-H3733

Our third core inhibitor product candidate, 3733, has completed Investigational New Drug (IND) enabling studies. 
3733  has  a  novel  chemical  scaffold  separate  from  both  VBR  and  2158.  We  presented  a  preclinical  profile  of  this 
candidate in the first quarter of 2019.

3

In  the  first  quarter  of  2020,  we  initiated  a  Phase  1a  clinical  study  to  evaluate  safety,  tolerability  and 
pharmacokinetics  (PK)  following  single  ascending  dose  and  multiple  ascending  dose  administration  of  3733  in 
healthy subjects in New Zealand. Conduct for the study was completed in the fourth quarter of 2020 and preliminary 
data indicate that 3733 was generally well-tolerated and had favorable PK.

Additional Product Candidates

In  addition  to  our  three  clinical-stage  product  candidates,  our  research  discovery  team  is  actively  focused  on 
identifying and selecting a fourth-generation core inhibitor candidate, which we anticipate in the first half of 2021.

Core Inhibitor Collaboration and License Agreements

Indiana University Research and Technology Corporation

In September 2013, we entered into an exclusive license agreement (the IURTC License Agreement) with Indiana 
University  Research  and  Technology  Corporation  (IURTC)  pursuant  to  which  we  acquired,  with  rights  to 
sublicense,  the  rights  to  develop  and  commercialize  products  associated  with  multiple  patents  and  patent 
applications covering aspects of our HBV program held by IURTC. As part of this agreement, we are obligated to 
make  milestone  payments  based  upon  the  successful  accomplishment  of  clinical  and  regulatory  milestones.  The 
aggregate  amount  of  all  performance  milestone  payments  under  the  IURTC  License  Agreement,  should  all 
performance milestones through development be met, is $0.8 million, with a portion related to the first performance 
milestone having been paid. Under the IURTC License Agreement, we are also obligated to pay IURTC royalties 
based on net sales of the licensed technology ranging from 0.5% to 1.75%. In addition, under the IURTC License 
Agreement, we pay annual diligence maintenance fees of $0.1 million. Milestone payments received by IURTC are 
fully  creditable  against  the  annual  diligence  maintenance  fee  for  the  year  in  which  the  milestone  payments  are 
received.

The  IURTC  License  Agreement  may  be  terminated  by  us,  with  or  without  cause,  upon  90  days  advance  written 
notice,  by  IURTC  upon  our  material  breach  with  60  days  advance  written  notice  or  by  IURTC,  in  certain  cases, 
upon our insolvency or bankruptcy immediately upon written notice.

BeiGene, Ltd.

In  July  2020,  we  entered  into  a  Collaboration  Agreement  with  BeiGene,  granting  BeiGene  an  exclusive,  royalty-
bearing license to develop and commercialize products containing VBR, 2158 and 3733 (the BeiGene Agreement) 
in the People’s Republic of China, Hong Kong, Taiwan and Macau (the Territory).

Under  the  BeiGene  Agreement,  we  and  BeiGene  will  collaborate  on  development  activities  with  respect  to  the 
licensed products in accordance with a mutually agreed upon development plan. 

Pursuant to the terms of the BeiGene Agreement, BeiGene paid us an upfront amount of $40.0 million, and we are 
eligible to receive up to approximately $500.0 million in milestone payments, comprised of up to $113.8 million in 
development  and  regulatory  and  $385.0  million  in  net  sales  milestone  payments.  In  addition,  we  are  eligible  to 
receive  tiered  royalties  at  percentages  ranging  from  the  mid-teens  to  the  low  30s  of  net  sales.  BeiGene  has  also 
agreed to pay all development and regulatory costs up to an aggregate of $45.0 million in the Territory for VBR, 
2158  and  3733.  Following  this  initial  investment,  we  and  BeiGene  will  share  development  costs  for  the  Territory 
equally.

The BeiGene Agreement also contains provisions such as representations and warranties of the parties, terms as to 
governance of the collaboration, commercialization and regulatory responsibilities of the parties, and manufacturing 
and supply, including potential adjustments in the event supply costs exceed certain levels. In addition, during the 
term of the BeiGene Agreement, neither party will commercialize any competing products in the Territory.

If, after 2158 and 3733 reach the end of Phase 2 clinical trials, we and BeiGene are unable to mutually agree on the 
terms of a Phase 3 global study, BeiGene may elect to terminate the BeiGene Agreement solely as it relates to that 
compound, as applicable. Such a termination would result in us regaining all rights to the applicable compound in 
the  Territory.  In  addition,  BeiGene  may  terminate  the  BeiGene  Agreement  for  convenience  at  any  time  upon  90 
days’ advance written notice to us. The BeiGene Agreement also contains customary provisions for termination by 
either party, including in the event of breach of the BeiGene Agreement, subject to cure.

4

Multi-Drug Combination Studies

We believe that core inhibitors and NrtI will be central to finite and curative therapies for chronic HBV infection. 
Therefore, as we continue to develop and advance our current and future core inhibitors through clinical studies, we 
plan  to  conduct  multi-drug  combination  studies  in  parallel  that  add  additional  drugs  (or  compounds)  with  non-
overlapping  mechanisms  of  action  to  the  core  inhibitor  +  NrtI  antiviral  backbone.  Specifically,  we  plan  on  only 
incorporating our current and future core inhibitors that have demonstrated they are well-tolerated and effective in 
clinical  studies  in  dual  combination  with  NrtI.  As  the  300  mg  daily  dose  of  VBR  has  been  observed  to  be  well-
tolerated in all studies conducted to date, with no serious adverse effects or dose-limiting toxicities identified and no 
pattern  of  treatment-emergent  clinical  or  laboratory  abnormalities  observed  and  has  progressed  beyond  dual 
combination studies, we currently have two triple combination studies planned to study VBR in combination with 
NrtI and a third mechanism of action. 

In  August  2020,  we  entered  into  a  Clinical  Trial  Agreement  with  Arbutus  Biopharma  Corporation  (Arbutus), 
pursuant  to  which  we  and  Arbutus  will  conduct  a  randomized,  multi-center,  open-label  Phase  2  clinical  trial  to 
explore  the  safety,  PK  and  antiviral  activity  of  the  triple  combination  of  VBR,  NrtI  and  AB-729  compared  to  the 
double  combinations  of  VBR  plus  NrtI  and  AB-729  plus  NrtI  in  virologically  suppressed  patients.  This  clinical 
study is projected to initiate in the first half of 2021.

Our  second  triple  combination  study  evaluates  VBR  and  NrtI  in  combination  with  interferon  in  treatment-naïve 
HBeAg positive subjects and was initiated in the first quarter of 2021.

In  addition  to  the  above  studies,  we  expect  to  continue  to  pursue  additional  multi-drug  combinations  that  include 
other or additional non-overlapping mechanisms of action to the core inhibitor + NrtI antiviral backbone.

Beyond Core Inhibitors

In addition to the development and advancement of our core inhibitor portfolio and our current and future multi-drug 
combination studies, our research and development team is working on discovering and developing a potent fourth-
generation core inhibitor, cccDNA disruptors and small molecules targeting novel undisclosed targets to add to the 
core inhibitor + NrtI antiviral backbone to achieve cure. In November 2020, we entered into an exclusive, two-year 
collaboration  and  option  agreement  with  Door  Pharmaceuticals  (Door  Pharma)  focused  on  the  development  of  a 
novel  class  of  HBV  inhibitors.  Door  Pharma’s  discovery  platform  targets  functions  of  core  protein  distinct  from 
viral assembly and have the potential to interfere with viral nucleic acid including intra-nuclear cccDNA, providing 
a strong complement to our current portfolio. Together with Door Pharma, we are working on identifying cccDNA 
disruptors,  which  will  be  aimed  at  inhibiting  different  intra-nuclear  steps  in  the  viral  replication  cycle  that 
complement the activity of our core inhibitors.

Under  the  terms  of  the  agreement,  Door  Pharma  will  build  upon  its  previous  efforts  to  lead  and  conduct  new 
discovery  research,  which  we  will  fund.  In  return  for  an  up-front  payment  and  success-based  milestones  and 
royalties, we will be granted an exclusive option to license compounds arising from the collaboration and will be 
responsible for the continued development and commercialization of optioned compounds.

Intellectual Property

In regard to our HBV patent estate, we co-own with and exclusively license from Indiana University two issued U.S. 
patents and related foreign patents and patent applications that relate to compositions of matter and methods of using 
VBR. The issued U.S. patents are expected to expire in 2035 and 2036. In addition, we own a pending U.S. patent 
application and related foreign applications directed to a process for preparing VBR; any patents issuing therefrom 
are expected to expire in 2038. Finally, we own an international (PCT) patent application directed to formulations of 
VBR; any patents issuing therefrom are expected to expire in 2040.

We own a pending U.S. patent application and related foreign applications that relate to compositions of matter and 
methods of using 2158; any patents issuing therefrom are expected to expire in 2038. 

We  own  a  PCT  patent  application  that  relates  to  compositions  of  matter  and  methods  of  using  3733;  any  patents 
issuing therefrom are expected to expire in 2039.

5

Microbiome Program

Following  the  termination  of  the  Research,  Development,  Collaboration  and  License  Agreement  between  the 
Company and Allergan Pharmaceuticals International Limited, which was acquired by AbbVie, Inc. in May 2020, 
we  began  an  extensive  process  to  identify  strategic  alternatives  to  continue  the  development  of  the  Microbiome 
program upon the return of the related intellectual property rights. This process did not result in us receiving any 
bids on any portion of the Microbiome program, including our facility in Groton, Connecticut. 

As a result, in December 2020, we and our Board of Directors (the Board) decided to wind down our Microbiome 
program as of January 31, 2021, including our facility in Groton, Connecticut, to prioritize and focus our resources 
on our HBV programs.

Government Regulation

Government authorities in the United States, at the federal, state and local level, and in other countries extensively 
regulate,  among  other  things,  the  research,  development,  testing,  manufacture,  including  any  manufacturing 
changes, packaging, storage, recordkeeping, labeling, advertising, promotion, distribution, marketing, post-approval 
monitoring and reporting, import and export of pharmaceutical products, such as those we are developing.   

U.S. drug approval process

In  the  United  States,  the  FDA  regulates  drugs  under  the  Federal  Food,  Drug,  and  Cosmetic  Act  (FDCA)  and 
implementing  regulations.  The  process  of  obtaining  regulatory  approvals  and  subsequent  compliance  with 
appropriate federal, state, local and foreign statutes and regulations requires the expenditure of substantial time and 
financial  resources.  Failure  to  comply  with  the  applicable  U.S.  requirements  at  any  time  during  the  product 
development process, approval process or after approval may subject an applicant to a variety of administrative or 
judicial  sanctions,  such  as  the  FDA’s  refusal  to  approve  pending  applications,  withdrawal  of  an  approval,  license 
revocation,  imposition  of  a  clinical  hold,  issuance  of  warning  letters  and  untitled  letters,  product  recalls,  product 
seizures,  total  or  partial  suspension  of  production  or  distribution,  injunctions,  fines,  refusals  of  government 
contracts, restitution, disgorgement of profits or civil or criminal penalties.

The  process  required  by  the  FDA  before  a  drug  may  be  marketed  in  the  United  States  generally  involves  the 
following:

(cid:129)

(cid:129)

(cid:129)

(cid:129)

(cid:129)

(cid:129)

(cid:129)

completion  of  nonclinical  laboratory  tests  and  animal  studies  in  compliance  with  the  FDA’s  good 
laboratory  practice  (GLP)  regulations  and  applicable  requirements  for  the  humane  use  of  laboratory 
animals or other applicable requirements;

submission to the FDA of an IND which must become effective before human clinical studies may begin;

approval by an independent institutional review board (IRB) or ethics committee at each clinical site before 
each trial may be initiated;

performance  of  adequate  and  well-controlled  human  clinical  studies  in  accordance  with  good  clinical 
practices  (GCP),  and  any  additional  requirements  for  the  protection  of  human  research  patients  and  their 
health information, to establish the safety and efficacy of the proposed drug for each indication;

submission to the FDA of a new drug application (NDA);

satisfactory completion of an FDA inspection of the manufacturing facility or facilities at which the product 
is produced to assess compliance with current good manufacturing practices (cGMP) requirements and to 
assure  that  the  facilities,  methods  and  controls  are  adequate  to  preserve  the  product’s  identity,  strength, 
quality and purity; and

FDA review and approval of the NDA.

6

Nonclinical studies and IND

Nonclinical  studies  include  laboratory  evaluation  of  product  chemistry  and  formulation,  as  well  as in  vitro and 
animal  studies  to  assess  the  potential  for  adverse  events  and  in  some  cases  to  establish  a  rationale  for  therapeutic 
use. The conduct of nonclinical studies is subject to federal regulations and requirements, including GLP regulations 
for  safety/toxicology  studies.  An  IND  sponsor  must  submit  the  results  of  the  nonclinical  tests,  together  with 
manufacturing  information,  analytical  data,  any  available  clinical  data  or  literature  and  plans  for  clinical  studies, 
among  other  things,  to  the  FDA  as  part  of  an  IND.  Some  long-term  nonclinical  testing,  such  as  animal  tests  of 
reproductive adverse events and carcinogenicity, may continue after the IND is submitted. For some products, the 
FDA may waive the need for certain nonclinical tests. An IND automatically becomes effective 30 days after receipt 
by the FDA, unless before that time the FDA raises concerns or questions related to one or more proposed clinical 
studies and places the trial on clinical hold. If an IND or clinical study is placed on clinical hold, the IND sponsor 
and the FDA must resolve any outstanding concerns before the clinical study can begin. As a result, submission of 
an IND may not result in the FDA allowing clinical studies to commence.

Clinical studies

Clinical studies involve the administration of the investigational new drug to human subjects under the supervision 
of qualified investigators in accordance with GCP requirements, which include, among other things, the requirement 
that all research subjects provide their informed consent in writing before their participation in any clinical study. 
Clinical  studies  are  conducted  under  written  study  protocols  detailing,  among  other  things,  the  objectives  of  the 
study, the parameters to be used in monitoring safety, and the effectiveness criteria to be evaluated. A protocol for 
each clinical study and any subsequent protocol amendments must be submitted to the FDA as part of the IND. In 
addition,  an  IRB  at  each  institution  participating  in  the  clinical  study  must  review  and  approve  the  plan  for  any 
clinical study before it commences at that institution, and the IRB must conduct continuing review. The IRB must 
review  and  approve,  among  other  things,  the  study  protocol  and  informed  consent  information  to  be  provided  to 
study subjects. An IRB must operate in compliance with FDA regulations. Information about certain clinical studies 
must  be  submitted  within  specific  timeframes  to  the  National  Institutes  of  Health  for  public  dissemination  at 
www.clinicaltrials.gov.

Human clinical studies are typically conducted in three sequential phases, which may overlap or be combined:

(cid:129)

(cid:129)

(cid:129)

Phase 1: The drug is initially introduced into healthy human subjects or patients with the target disease or 
condition  and  tested  for  safety,  dosage  tolerance,  absorption,  metabolism,  distribution,  excretion  and,  if 
possible, to gain an early indication of its effectiveness.

Phase 2: The drug is administered to a limited patient population to identify possible adverse effects and 
safety  risks,  to  preliminarily  evaluate  the  efficacy  of  the  product  for  specific  targeted  diseases  and  to 
determine dosage tolerance and optimal dosage.

Phase  3: The  drug  is  administered  to  an  expanded  patient  population  in  adequate  and  well-controlled 
clinical studies to generate sufficient data to statistically confirm the efficacy and safety of the product for 
approval, to establish the overall risk-benefit profile of the product and to provide adequate information for 
the labeling of the product.

Progress  reports  detailing  the  results  of  the  clinical  studies  must  be  submitted  at  least  annually  to  the  FDA. 
Additionally, IND safety reports must be submitted to the FDA and the investigators within 15 calendar days after 
determining that the information qualifies for reporting. IND safety reports are required for serious and unexpected 
suspected adverse reactions, findings from animal or in vitro testing or other studies that suggest a significant risk to 
humans, and any clinically important increase in the rate of a serious suspected adverse reaction over that listed in 
the protocol or investigator brochure. In addition, a sponsor must notify the FDA within seven calendar days after 
receiving information concerning any unexpected fatal or life-threatening suspected adverse reaction. Phase 1, Phase 
2 and Phase 3 clinical studies may not be completed successfully within any specified period, or at all. Furthermore, 
the  FDA  or  the  sponsor  may  suspend  or  terminate  a  clinical  study  at  any  time  on  various  grounds,  including  a 
finding that the research subjects are being exposed to an unacceptable health risk. Similarly, an IRB can suspend or 
terminate approval of a clinical study at its institution if the clinical study is not being conducted in accordance with 
the IRB’s requirements or if the drug has been associated with unexpected serious harm to patients.

7

A manufacturer of an investigational drug for a serious disease or condition is required to make available, such as by 
posting  on  its  website,  its  policy  regarding  evaluating  and  responding  to  requests  for  individual  patient  access  to 
such investigational drug. This requirement applies on the earlier of the first initiation of a Phase 2 or Phase 3 trial of 
the investigational drug or, as applicable, 15 days after the drug receives a designation as a breakthrough therapy, 
fast track product, or regenerative advanced therapy.

Marketing approval

After the completion of required clinical testing, the results of the nonclinical studies and clinical studies, together 
with detailed information relating to the product’s chemistry, manufacture, controls and proposed labeling, among 
other things, are submitted to the FDA as part of an NDA requesting approval to market the product for one or more 
indications. Under federal law, the submission of most NDAs is additionally subject to a substantial application user 
fee, currently $2.9 million and the sponsor of an approved NDA is also subject to an annual program fee currently 
set at $0.3 million through September 30, 2021. These fees are typically adjusted on October 1 each year.

The FDA conducts a preliminary review of all NDAs within the first 60 days after submission before accepting them 
for filing to determine whether they are sufficiently complete to permit substantive review. The FDA may request 
additional information rather than accept an NDA for filing. In this event, the application must be resubmitted with 
the additional information. The resubmitted application is also subject to review before the FDA accepts it for filing. 
Once the submission is accepted for filing, the FDA begins an in-depth substantive review. The FDA has agreed to 
specified  performance  goals  in  the  review  of  NDAs.  Under  these  goals,  the  FDA  has  committed  to  review  most 
original applications for non-priority products within ten months, and most original applications for priority review 
products,  that  is,  drugs  for  a  serious  or  life-threatening  condition  that  the  FDA  determines  represent  a  significant 
improvement over existing therapy, within six months. For NDAs for novel products, the ten- and six-month time 
periods runs from the filing date; for all other original applications, the ten- and six-month time periods run from the 
submission date. The review process may be extended by the FDA for three additional months to consider certain 
information or clarification regarding information already provided in the submission. Despite these review goals, it 
is not uncommon for FDA review of an NDA to extend beyond the goal date. The FDA may also refer applications 
for novel drugs or products that present difficult questions of safety or efficacy to an advisory committee, typically a 
panel  that  includes  clinicians  and  other  experts,  for  review,  evaluation  and  a  recommendation  as  to  whether  the 
application should be approved. The FDA is not bound by the recommendations of an advisory committee, but it 
considers such recommendations carefully when making decisions.

Before  approving  an  NDA,  the  FDA  typically  will  inspect  the  facility  or  facilities  where  the  product  is 
manufactured. The FDA will not approve an application unless it determines that the manufacturing processes and 
facilities  are  in  compliance  with  cGMP  requirements  and  adequate  to  assure  consistent  production  of  the  product 
within required specifications. In addition, before approving an NDA, the FDA will typically inspect one or more 
clinical sites to assure compliance with GCP and integrity of the clinical data submitted.

After  the  FDA’s  evaluation  of  the  NDA  and  inspection  of  the  manufacturing  facilities,  the  FDA  may  issue  an 
approval letter or a complete response letter. An approval letter authorizes commercial marketing of the drug with 
specific  prescribing  information  for  specific  indications.  A  complete  response  letter  generally  outlines  the 
deficiencies in the submission and may require substantial additional testing or information in order for the FDA to 
reconsider  the  application.  If  and  when  those  deficiencies  have  been  addressed  to  the  FDA’s  satisfaction  in  a 
resubmission  of  the  NDA,  the  FDA  will  issue  an  approval  letter.  The  FDA  has  committed  to  reviewing  such 
resubmissions in two or six months depending on the type of information included. Even with submission of this 
additional information, the FDA ultimately may decide that the application does not satisfy the regulatory criteria for 
approval and refuse to approve the NDA. Even if the FDA approves a product, it may limit the approved indications 
for use for the product, require that contraindications, warnings or precautions be included in the product labeling, 
require that post-approval studies, including Phase 4 clinical studies, be conducted to further assess a drug’s safety 
after approval, require testing and surveillance programs to monitor the product after commercialization, or impose 
other conditions, including distribution and use restrictions or other risk management mechanisms, including Risk 
Evaluation and Mitigation Strategies (REMS), which can materially affect the potential market and profitability of 
the  product  or  impose  new  labeling,  testing  or  distribution  and  use  requirements.  The  FDA  may  prevent  or  limit 
further marketing of a product based on the results of post-market studies or surveillance programs. After approval, 
some  types  of  changes  to  the  approved  product,  such  as  adding  new  indications,  manufacturing  changes  and 
additional labeling claims, are subject to further testing requirements and FDA review and approval. 

8

Fast track designation

The  FDA  is  required  to  facilitate  and  expedite  the  development  and  review  of  drugs  that  are  intended  for  the 
treatment  of  a  serious  or  life-threatening  disease  or  condition  for  which  there  is  no  effective  treatment  and  which 
demonstrate the potential to address unmet medical needs for the disease or condition. Under the fast track program, 
the sponsor of a new product candidate may request the FDA to designate the product for a specific indication as a 
fast track product concurrent with or after the filing of the IND for the product candidate. The FDA must determine 
if  the  product  candidate  qualifies  for  fast  track  designation  within  60  calendar  days  after  receipt  of  the  sponsor’s 
request.

In  addition  to  other  benefits,  such  as  the  ability  to  have  greater  interactions  with  the  FDA,  the  FDA  may  initiate 
review of sections of a fast track product’s NDA before the application is complete. This rolling review is available 
if the applicant provides and the FDA approves a schedule for the submission of the remaining information and the 
applicant pays applicable user fees. However, the FDA’s time period goal for reviewing a fast track application does 
not begin until the last section of the NDA is submitted. In addition, the fast track designation may be withdrawn by 
the  FDA  if  the  FDA  believes  that  the  designation  is  no  longer  supported  by  data  emerging  in  the  clinical  study 
process. In 2018 and 2020, the FDA granted fast track designation to VBR and 2158, respectively, for the treatment 
of patients with chronic HBV infection.

Priority review

Under FDA policies, a product candidate may be eligible for priority review, a review generally within a six-month 
time  frame  from  the  time  a  complete  application  is  received  or  filed.  Products  generally  are  eligible  for  priority 
review  if  they  are  intended  for  treatment  of  a  serious  or  life-threatening  disease  or  condition  and  provide  a 
significant  improvement  in  safety  or  effectiveness  compared  to  marketed  products  in  the  treatment,  diagnosis  or 
prevention  of  a  serious  disease  or  condition.  A  fast  track  designated  product  candidate  would  ordinarily  meet  the 
FDA’s criteria for priority review.

Accelerated approval

Under  the  FDA’s  accelerated  approval  regulations,  the  FDA  may  approve  a  drug  for  a  serious  or  life-threatening 
illness  that  provides  meaningful  therapeutic  benefit  to  patients  over  existing  treatments  based  upon  a  surrogate 
endpoint  that  is  reasonably  likely  to  predict  clinical  benefit  or  on  a  clinical  endpoint  that  can  be  measured  earlier 
than  irreversible  morbidity  or  mortality  (IMM).  In  clinical  studies,  a  surrogate  endpoint  is  a  measurement  of 
laboratory or clinical signs of a disease or condition that substitutes for a direct measurement of how a patient feels, 
functions  or  survives.  Surrogate  endpoints  can  often  be  measured  more  easily  or  more  rapidly  than  clinical 
endpoints.  A  product  candidate  approved  on  this  basis  is  subject  to  rigorous  post-marketing  compliance 
requirements,  including  the  completion  of  Phase  4  or  post-approval  clinical  studies  to  confirm  the  effect  on  the 
clinical  endpoint.  Failure  to  conduct  required  post-approval  studies,  or  confirm  a  clinical  benefit  during  post-
marketing  studies,  would  allow  the  FDA  to  withdraw  the  drug  from  the  market  on  an  expedited  basis.  All 
promotional materials for drug candidates approved under accelerated regulations are subject to prior review by the 
FDA.

Breakthrough therapy designation

A sponsor can request designation of a product candidate as a “breakthrough therapy.” A breakthrough therapy is 
defined as a drug that is intended, alone or in combination with one or more other drugs, to treat a serious or life-
threatening  disease  or  condition,  and  preliminary  clinical  evidence  indicates  that  the  drug  may  demonstrate 
substantial improvement over existing therapies on one or more clinically significant endpoints, such as substantial 
treatment effects observed early in clinical development. Drugs designated as breakthrough therapies also may be 
eligible  for  priority  review.  The  FDA  must  take  certain  actions,  such  as  holding  timely  meetings  and  providing 
advice, intended to expedite the development and review of an application for approval of a breakthrough therapy. 
Even if a product qualifies for one or more of these programs, the FDA may later decide that the product no longer 
meets  the  conditions  for  qualification  or  decide  that  the  time  period  for  FDA  review  or  approval  will  not  be 
shortened.

9

Orphan drugs

Under the Orphan Drug Act, as amended, the FDA may grant orphan drug designation to drugs intended to treat a 
rare  disease  or  condition,  which  is  generally  defined  as  a  disease  or  condition  that  affects  fewer  than  200,000 
individuals  in  the  United  States  or  that  affects  more  than  200,000  individuals  in  the  United  States  and  for  which 
there  is  no  reasonable  expectation  that  the  cost  of  developing  and  making  available  the  drug  for  the  disease  or 
condition  will  be  recovered  from  sales  of  the  product  in  the  United  States.  Orphan  drug  designation  must  be 
requested  before  submitting  an  NDA  or  BLA.  After  the  FDA  grants  orphan  drug  designation,  the  identity  of  the 
product and its potential orphan use are disclosed publicly by the FDA. Orphan drug designation does not shorten 
the  duration  of  the  regulatory  review  and  approval  process.  The  first  NDA  or  BLA  applicant  to  receive  FDA 
approval for a particular active moiety to treat a particular disease with FDA orphan drug designation is entitled to a 
seven-year exclusive marketing period in the United States for that product and indication. During the seven-year 
exclusivity period, the FDA may not approve any other applications to market the same drug for the same orphan 
indication, except in limited circumstances, such as a showing of clinical superiority to the product with orphan drug 
exclusivity. A drug will be considered clinically superior if it is shown to be safer, more effective or makes a major 
contribution to patient care. Orphan drug exclusivity does not prevent the FDA from approving a different drug for 
the same orphan disease or condition, or the same drug for a different disease or condition. Among the other benefits 
of orphan drug designation are tax credits for certain research and a waiver of the NDA/BLA application user fee.

Pediatric information

Under  the  Pediatric  Research  Equity  Act  of  2003,  as  amended,  an  NDA  or  supplement  to  an  NDA  for  drug  with 
certain novel features (e.g., new active ingredient, new indication) must contain data that are adequate to assess the 
safety  and  effectiveness  of  the  drug  for  the  claimed  indications  in  all  relevant  pediatric  subpopulations,  and  to 
support dosing and administration for each pediatric subpopulation for which the product is safe and effective. The 
FDA  may,  on  its  own  initiative  or  at  the  request  of  the  applicant,  grant  deferrals  for  submission  of  some  or  all 
pediatric data until after approval of the product for use in adults, or full or partial waivers from the pediatric data 
requirements. A sponsor of a new drug subject to the above pediatric testing requirements also is required to submit 
to the FDA a pediatric study plan generally 60 days after an end-of-Phase 2 meeting with the agency. Generally, the 
pediatric data requirements do not apply to products with orphan drug designation.

Other regulatory requirements

Any drug manufactured or distributed by us pursuant to FDA approvals will be subject to pervasive and continuing 
regulation  by  the  FDA,  including,  among  other  things,  requirements  relating  to  recordkeeping,  periodic  reporting, 
product sampling and distribution, advertising and promotion and reporting of adverse experiences with the product. 
After approval, most changes to the approved product, such as adding new indications or other labeling claims, are 
subject to prior FDA review and approval.

The FDA may impose a number of post-approval requirements, including REMS, as a condition of approval of an 
NDA  or  BLA.  For  example,  the  FDA  may  require  post-marketing  testing,  including  Phase  4  clinical  studies,  and 
surveillance to further assess and monitor the product’s safety and effectiveness after commercialization.

In addition, drug manufacturers and other entities involved in the manufacture and distribution of approved drugs 
are  required  to  register  their  establishments  with  the  FDA  and  state  agencies  and  are  subject  to  periodic 
unannounced inspections by the FDA and these state agencies for compliance with cGMP requirements. Changes to 
the  manufacturing  process  are  strictly  regulated  and  often  require  prior  FDA  approval  before  being  implemented. 
FDA regulations also require investigation and correction of any deviations from cGMP and impose reporting and 
documentation  requirements  upon  us  and  any  third-party  manufacturers  that  we  may  decide  to  use.  Accordingly, 
manufacturers  must  continue  to  expend  time,  money  and  effort  in  the  areas  of  production  and  quality  control  to 
maintain cGMP compliance.

10

Once an approval is granted, the FDA may withdraw the approval if compliance with regulatory requirements and 
standards is not maintained or if problems occur after the product reaches the market. Later discovery of previously 
unknown  problems  with  a  product,  including  adverse  events  of  unanticipated  severity  or  frequency,  or  with 
manufacturing processes, or failure to comply with regulatory requirements, may result in revisions to the approved 
labeling  to  add  new  safety  information,  imposition  of  post-market  studies  or  clinical  studies  to  assess  new  safety 
risks or imposition of distribution or other restrictions under a REM program. Other potential consequences include, 
among other things:

(cid:129)

(cid:129)

(cid:129)

(cid:129)

(cid:129)

restrictions on the marketing or manufacturing of the product, complete withdrawal of the product from the 
market or product recalls;

fines, warning letters or holds on post-approval clinical studies;

refusal of the FDA to approve pending applications or supplements to approved applications, or suspension 
or revocation of product approvals;

product seizure or detention, or refusal to permit the import or export of products; or

consent decrees, injunctions or the imposition of civil or criminal penalties.

The FDA strictly regulates marketing, labeling, advertising and promotion of products that are placed on the market. 
Drugs generally may be promoted only for the approved indications and in accordance with the provisions of the 
approved labeling. The FDA and other agencies actively enforce the laws and regulations prohibiting the promotion 
of  off  label  uses,  and  a  company  that  is  found  to  have  improperly  promoted  off  label  uses  may  be  subject  to 
significant liability.

Physician Drug Samples

As part of the sales and marketing process, pharmaceutical companies frequently provide samples of approved drugs 
to  physicians.  The  Prescription  Drug  Marketing  Act  (PDMA)  regulates  the  distribution  of  drug  samples  at  the 
federal level and sets minimum standards for the registration and regulation of drug distributors by the states. Both 
the  PDMA  and  state  laws  limit  the  distribution  of  prescription  pharmaceutical  product  samples  and  impose 
requirements to ensure accountability in distribution. In addition, the PDMA sets forth civil and criminal penalties 
for violations.

Foreign Regulation

In order to market any product outside of the United States, we would need to comply with numerous and varying 
regulatory requirements of other countries regarding safety and efficacy and governing, among other things, clinical 
studies, marketing authorization, commercial sales and distribution of our products. Whether or not we obtain FDA 
approval for a product, we would need to obtain the necessary approvals by the comparable regulatory authorities of 
foreign  countries  before  we  can  commence  clinical  studies  or  marketing  of  the  product  in  those  countries.  The 
approval  process  varies  from  country  to  country  and  can  involve  additional  product  testing  and  additional 
administrative  review  periods.  The  time  required  to  obtain  approval  in  other  countries  might  differ  from  and  be 
longer  than  that  required  to  obtain  FDA  approval.  Regulatory  approval  in  one  country  does  not  ensure  regulatory 
approval in another, but a failure or delay in obtaining regulatory approval in one country may negatively impact the 
regulatory process in others.

New Legislation and Regulations

From  time  to  time,  legislation  is  drafted,  introduced  and  passed  in  Congress  that  could  significantly  change  the 
statutory  provisions  governing  the  testing,  approval,  manufacturing  and  marketing  of  products  regulated  by  the 
FDA. In addition to new legislation, FDA regulations and policies are often revised or interpreted by the agency in 
ways  that  may  significantly  affect  our  business  and  our  products.  It  is  impossible  to  predict  whether  further 
legislative changes will be enacted or whether FDA regulations, guidance, policies or interpretations will be changed 
or what the effect of such changes, if any, may be.

11

Pharmaceutical Coverage, Pricing and Reimbursement

Significant uncertainty exists as to the coverage and reimbursement status of any drug products for which we may 
obtain regulatory approval. Sales of any of our product candidates, if approved, will depend, in part, on the extent to 
which the costs of the products will be covered by third-party payors, including government health programs such as 
Medicare and Medicaid, commercial health insurers and managed care organizations. The process for determining 
whether a payor will provide coverage for a drug product may be separate from the process for setting the price or 
reimbursement rate that the payor will pay for the drug product once coverage is approved. Third-party payors may 
limit  coverage  to  specific  drug  products  on  an  approved  list,  or  formulary,  which  might  not  include  all  of  the 
approved drugs for a particular indication.

In  order  to  secure  coverage  and  reimbursement  for  any  product  that  might  be  approved  for  sale,  we  may  need  to 
conduct expensive pharmacoeconomic studies in order to demonstrate the medical necessity and cost-effectiveness 
of  the  product,  in  addition  to  the  trials  required  to  obtain  FDA  or  other  comparable  regulatory  approvals.  Our 
product  candidates  may  not  be  considered  medically  necessary  or  cost-effective.  A  payor’s  decision  to  provide 
coverage for a drug product does not imply that an adequate reimbursement rate will be approved. Companies may 
also need to provide discounts to purchasers, private health plans or government healthcare programs. Third-party 
reimbursement  may  not  be  sufficient  to  enable  us  to  maintain  price  levels  high  enough  to  realize  an  appropriate 
return  on  our  investment  in  product  development.  Further,  one  payor’s  determination  to  provide  coverage  for  a 
product  does  not  assure  that  other  payors  will  also  provide  coverage  and  reimbursement  for  the  product,  and  the 
level of coverage and reimbursement can differ significantly from payor to payor.

The containment of healthcare costs has become a priority of federal, state and foreign governments, and the prices 
of  drugs  have  been  a  focus  in  this  effort.  Third-party  payors  are  increasingly  challenging  the  prices  charged  for 
medical products and services and examining the medical necessity and cost-effectiveness of medical products and 
services, in addition to their safety and efficacy. If these third-party payors do not consider our products to be cost-
effective compared to other available therapies, they may not cover our products after approval as a benefit under 
their plans or, if they do, the level of payment may not be sufficient to allow us to sell our products at a profit. The 
U.S. government, state legislatures and foreign governments have shown significant interest in implementing cost 
containment programs to limit the growth of government-paid health care costs, including price controls, restrictions 
on reimbursement and requirements for substitution of generic products for branded prescription drugs. Adoption of 
such controls and measures and tightening of restrictive policies in jurisdictions with existing controls and measures, 
could limit payments for pharmaceuticals such as the drug candidates that we are developing and could adversely 
affect our net revenue and results. Even if favorable coverage and reimbursement status is attained for one or more 
products for which we may receive regulatory approval, less favorable coverage policies and reimbursement rates 
may be implemented in the future.

Pricing  and  reimbursement  schemes  vary  widely  from  country  to  country.  Some  countries  provide  that  drug 
products  may  be  marketed  only  after  a  reimbursement  price  has  been  agreed.  Some  countries  may  require  the 
completion  of  additional  studies  that  compare  the  cost-effectiveness  of  a  particular  product  candidate  to  currently 
available therapies. For example, the European Union provides options for its member states to restrict the range of 
drug products for which their national health insurance systems provide reimbursement and to control the prices of 
medicinal products for human use. European Union member states may approve a specific price for a drug product 
or may instead adopt a system of direct or indirect controls on the profitability of us placing the drug product on the 
market.  Other  member  states  allow  companies  to  fix  their  own  prices  for  drug  products  but  monitor  and  control 
company profits. The downward pressure on health care costs in general, particularly prescription drugs, has become 
very intense. As a result, increasingly high barriers are being erected to the entry of new products. In addition, in 
some countries, cross-border imports from low-priced markets exert competitive pressure that may reduce pricing 
within a country. There can be no assurance that any country that has price controls or reimbursement limitations for 
drug products will allow favorable reimbursement and pricing arrangements for any of our products.

The marketability of any products for which we may receive regulatory approval for commercial sale is dependent 
on  the  availability  of  adequate  coverage  and  reimbursement  from  government  and  third-party  payors.  In  addition, 
the  emphasis  on  managed  care  in  the  United  States  has  increased  and  we  expect  will  continue  to  increase  the 
pressure  on  drug  pricing.  Coverage  policies,  third-party  reimbursement  rates  and  drug  pricing  regulation  may 
change  at  any  time.  In  particular,  in  the  United  States,  the  Affordable  Care  Act  (ACA)  and  its  amendment,  the 
Health  Care  and  Education  Reconciliation  Act,  contains  provisions  that  may  reduce  the  profitability  of  drug 

12

products,  including,  for  example,  increased  rebates  for  drugs  sold  to  Medicaid  programs,  extension  of  Medicaid 
rebates to Medicaid managed care plans, mandatory discounts for certain Medicare Part D beneficiaries and annual 
fees based on pharmaceutical companies’ share of sales to federal health care programs.

Among the provisions of the ACA of importance to our potential drug candidates are the following:

(cid:129)

(cid:129)

(cid:129)

(cid:129)

(cid:129)

(cid:129)

(cid:129)

(cid:129)

(cid:129)

(cid:129)

an  annual,  nondeductible  fee  on  any  entity  that  manufactures  or  imports  specified  branded  prescription 
drugs;

an  increase  in  the  statutory  minimum  rebates  a  manufacturer  must  pay  under  the  Medicaid  Drug  Rebate 
Program;

expansion  of  healthcare  fraud  and  abuse  laws,  including  the  False  Claims  Act  and  the  Anti-Kickback 
Statute, new government investigative powers, and enhanced penalties for noncompliance;

a new Medicare Part D coverage gap discount program, in which manufacturers must agree to offer 70% 
point-of-sale discounts off negotiated prices of applicable brand drugs under the Bipartisan Budget Act of 
2018 (BBA);

extension of manufacturers’ Medicaid rebate liability;

expansion of eligibility criteria for Medicaid programs;

expansion of the entities eligible for discounts under the Public Health Service Act pharmaceutical pricing 
program;

requirements to report financial arrangements with physicians and teaching hospitals;

a  requirement  to  annually  report  drug  samples  that  manufacturers  and  distributors  provide  to  physicians; 
and

a Patient-Centered Outcomes Research Institute to oversee, identify priorities in, and conduct comparative 
clinical effectiveness research, along with funding for such research.

Since its enactment, there have been many judicial, Presidential, and Congressional challenges to numerous aspects 
of the ACA. For example, former President Trump issued several executive orders and other directives designed to 
delay, circumvent, or loosen certain requirements or implementation of certain requirements mandated by the ACA. 
Concurrently, Congress has considered legislation that would repeal, or repeal and replace all or part of the ACA. 
While  Congress  has  not  passed  comprehensive  repeal  legislation,  several  bills  affecting  the  implementation  of 
certain taxes under the ACA have been signed into law. For example, the Tax Cuts and Jobs Act, signed into law in 
2017,  effectively  repealed  the  individual  health  insurance  mandate,  which  is  considered  a  key  component  of  the 
ACA, and the U.S. Supreme Court recently heard oral arguments regarding the constitutionality of the ACA and the 
individual mandate, with a decision expected during the current term in 2021. Further, the Trump Administration’s 
2020  federal  spending  package  permanently  eliminated,  effective  January  1,  2020,  the  ACA-mandated  “Cadillac” 
tax on certain high-cost employer-sponsored insurance plans and, on January 1, 2021, eliminated the health insurer 
tax. Moreover, the BBA, among other things, amended the ACA to close the coverage gap in most Medicare drug 
plans, commonly referred to as the “donut hole”. 

In addition, other legislative changes have been proposed and adopted since the ACA was enacted. These changes 
included aggregate reductions to Medicare payments to providers of up to 2% per fiscal year, and, due to subsequent 
legislative amendments, will remain in effect through 2030, with the exception of a temporary suspension from May 
1,  2020  through  March  2021,  unless  additional  Congressional  action  is  taken.  Further,  in  January  2013,  then 
President Obama signed into law the American Taxpayer Relief Act of 2012, which, among other things, reduced 
Medicare  payments  to  several  providers,  and  increased  the  statute  of  limitations  period  for  the  government  to 
recover  overpayments  to  providers  from  three  to  five  years.  These  laws  may  result  in  additional  reductions  in 
Medicare and other healthcare funding.

13

Additionally, there has been increasing legislative and enforcement interest in the United States with respect to drug 
pricing  practices.  Specifically,  there  have  been  several  recent  United  States  Congressional  inquiries  and  proposed 
and enacted federal legislation designed to, among other things, bring more transparency to drug pricing, reduce the 
cost  of  prescription  drugs  under  Medicare,  review  the  relationship  between  pricing  and  manufacturer  patient 
programs,  and  reform  government  program  reimbursement  methodologies  for  drugs.  For  example,  at  the  federal 
level,  the  Trump  Administration  issued  several  executive  orders  related  to  prescription  drug  pricing  and  sent 
“principles” for drug pricing to Congress. In addition, in September 2020, the FDA issued a final rule that sets up a 
legal  framework  for  allowing  the  importation  of  certain  prescription  drugs  from  Canada,  and  the  Centers  for 
Medicare & Medicaid Services (CMS) issued guidance that addresses the treatment of certain imported drugs under 
the  Medicaid  Drug  Rebate  Program.  In  November  2020,  the  Trump  Administration  and  the  U.S.  Department  of 
Health and Human Services (HHS) announced regulations tying certain Medicare Part B drug prices to international 
drug  prices,  modifying  certain  federal  Anti-Kickback  Statute  (AKS)  safe  harbors,  including  removing  safe  harbor 
protection for rebates negotiated between drug manufacturers and pharmacy benefit managers (PBMs) or health plan 
sponsors in Medicare Part D, and making further changes to the rules implementing the Stark Law, other AKS safe 
harbors  and  the  beneficiary  inducements  provision  in  the  civil  monetary  penalties  law.  On  November  20,  2020, 
CMS  issued  an  interim  final  rule  implementing  President  Trump’s  Most  Favored  Nation  executive  order,  which 
would  tie  Medicare  Part  B  payments  for  certain  physician-administered  drugs  to  the  lowest  price  paid  in  other 
economically  advanced  countries.  However,  on  December  28,  2020,  the  United  States  District  Court  in  Northern 
California  issued  a  nationwide  preliminary  injunction  against  implementation  of  the  interim  final  rule,  and  CMS 
announced  that  the  Most  Favored  Nation  Model  will  not  be  implemented  without  further  rulemaking.  There  also 
have been legal challenges to the modified AKS safe harbor for drug rebates, which delayed implementation of the 
modified safe harbor until January 1, 2023, pending HHS’s review, and gave the Biden Administration until April 1, 
2021 to decide whether to defend the rebate rule in court. The Biden Administration also has issued a final rule to 
delay the effective date of other provisions of the rebate rule that were scheduled to take effect on January 29, 2021 
to March 22, 2021. The likelihood of implementation of any of the other Trump Administration reform initiatives is 
uncertain,  particularly  in  light  of  the  change  in  presidential  administrations.  Individual  states  in  the  United  States 
have  also  become  increasingly  active  in  passing  legislation  and  implementing  regulations  designed  to  control 
pharmaceutical  and  biological  product  pricing,  including  price  or  patient  reimbursement  constraints,  discounts, 
restrictions  on  certain  product  access  and  marketing  cost  disclosure  and  transparency  measures.  Accordingly,  the 
ultimate content, timing or effect of healthcare reform legislation on the United States healthcare industry is unclear.

Other Healthcare Laws

In the United States, our activities are potentially subject to regulation by various federal, state and local authorities 
in  addition  to  the  FDA,  including  but  not  limited  to,  CMS,  other  divisions  of  the  U.S.  Department  of  Health  and 
Human Services (e.g., the Office of Inspector General), the U.S. Department of Justice (DOJ), and individual U.S. 
Attorney offices within the DOJ, and state and local governments. For example, the Company’s business practices, 
including  its  research  and  sales,  marketing  and  scientific/  educational  grant  programs  may  be  required  to  comply 
with federal and state fraud and abuse laws, false claims laws, the data privacy and security provisions of the Health 
Insurance  Portability  and  Accountability  Act  (HIPAA),  federal  transparency  requirements  and  similar  state  laws, 
each as amended. The laws that may affect our ability to operate include:

(cid:129)

(cid:129)

the federal Anti-Kickback Statute, which prohibits, among other things, knowingly and willfully soliciting, 
receiving,  offering  or  paying  any  remuneration  (including  any  kickback,  bribe,  or  rebate),  directly  or 
indirectly,  overtly  or  covertly,  in  cash  or  in  kind,  to  induce,  or  in  return  for,  either  the  referral  of  an 
individual, or the purchase, lease, order or recommendation of any good, facility, item or service for which 
payment may be made, in whole or in part, under a federal healthcare program, such as the Medicare and 
Medicaid  programs.  A  person  or  entity  can  be  found  guilty  of  violating  the  statute  without  actual 
knowledge of the statute or specific intent to violate it. The Anti-Kickback Statute has been interpreted to 
apply to arrangements between pharmaceutical manufacturers on the one hand and prescribers, purchasers, 
and formulary managers on the other;

federal  civil  and  criminal  false  claims  laws  and  civil  monetary  penalty  laws,  such  as  the  federal  False 
Claims Act, which impose criminal and civil penalties and authorize civil whistleblower or qui tam actions, 
against individuals or entities for, among other things: knowingly presenting, or causing to be presented, to 
the federal government, claims for payment that are false or fraudulent; making a false statement or record 
material  to  a  false  or  fraudulent  claim  or  obligation  to  pay  or  transmit  money  or  property  to  the  federal 

14

government; or knowingly concealing or knowingly and improperly avoiding or decreasing an obligation to 
pay money to the federal government. In addition, the government may assert that a claim including items 
and services resulting from a violation of the federal Anti-Kickback Statute constitutes a false or fraudulent 
claim for purposes of the False Claims Act. Manufacturers can be held liable under the False Claims Act 
even  when  they  do  not  submit  claims  directly  to  government  payors  if  they  are  deemed  to  “cause”  the 
submission of false or fraudulent claims;

(cid:129) HIPAA,  which  created  new  federal  criminal  statutes  that  prohibit  knowingly  and  willfully  executing,  or 
attempting to execute, a scheme to defraud any healthcare benefit program or obtain, by means of false or 
fraudulent  pretenses,  representations,  or  promises,  any  of  the  money  or  property  owned  by,  or  under  the 
custody or control of, any healthcare benefit program, regardless of the payor (e.g., public or private) and 
knowingly  and  willfully  falsifying,  concealing  or  covering  up  by  any  trick  or  device  a  material  fact  or 
making  any  materially  false  statements  in  connection  with  the  delivery  of,  or  payment  for,  healthcare 
benefits,  items  or  services  relating  to  healthcare  matters.  Similar  to  the  federal  Anti-Kickback  Statute,  a 
person or entity can be found guilty of violating HIPAA without actual knowledge of the statute or specific 
intent to violate it;

(cid:129) HIPAA,  as  amended  by  HITECH,  and  their  respective  implementing  regulations,  which  impose 
requirements on certain covered healthcare providers, health plans, and healthcare clearinghouses as well as 
their  respective  business  associates  that  perform  services  for  them  that  involve  the  use,  or  disclosure  of, 
individually  identifiable  health  information,  relating  to  the  privacy,  security  and  transmission  of 
individually  identifiable  health  information.  HITECH  also  created  new  tiers  of  civil  monetary  penalties, 
amended HIPAA to make civil and criminal penalties directly applicable to business associates, and gave 
state  attorneys  general  new  authority  to  file  civil  actions  for  damages  or  injunctions  in  federal  courts  to 
enforce the federal HIPAA laws and seek attorneys’ fees and costs associated with pursuing federal civil 
actions;

(cid:129)

(cid:129)

(cid:129)

(cid:129)

the federal false statements statute prohibits knowingly and willfully falsifying, concealing or covering up a 
material  fact  or  making  any  materially  false  statement  in  connection  with  the  delivery  of  or  payment  for 
healthcare benefits, items or services;

the  U.S.  federal  Food,  Drug  and  Cosmetic  Act  (FDCA),  which  prohibits,  among  other  things,  the 
adulteration or misbranding of drugs, biologics and medical devices;

the federal transparency requirements under the ACA, including the provision commonly referred to as the 
Physician Payments Sunshine Act, which requires manufacturers of drugs, devices, biologics and medical 
supplies  for  which  payment  is  available  under  Medicare,  Medicaid  or  the  Children’s  Health  Insurance 
Program to report annually to the U.S. Department of Health and Human Services information related to 
payments or other transfers of value made to physicians and teaching hospitals, as well as ownership and 
investment  interests  held  by  physicians  and  their  immediate  family  members.  Effective  January  1,  2022, 
these reporting obligations will extend to include transfers of value made to certain non-physician providers 
such as physician assistants and nurse practitioners; and

federal consumer protection and unfair competition laws, which broadly regulate marketplace activities and 
activities that potentially harm consumers.

Additionally,  we  are  subject  to  state  and  non-U.S.  equivalents  of  each  of  the  healthcare  laws  described  above, 
among  others,  some  of  which  may  be  broader  in  scope  and  may  apply  regardless  of  the  payor.  Many  U.S.  states 
have adopted laws similar to the federal Anti-Kickback Statute, some of which apply to the referral of patients for 
healthcare services reimbursed by any source, not just governmental payors, including private insurers. In addition, 
some  states  have  passed  laws  that  require  pharmaceutical  companies  to  comply  with  the  April 2003  Office  of 
Inspector  General  Compliance  Program  Guidance  for  Pharmaceutical  Manufacturers  and/or  the  Pharmaceutical 
Research and Manufacturers of America’s Code on Interactions with Healthcare Professionals. Several states also 
impose other marketing restrictions or require pharmaceutical companies to make marketing or price disclosures to 
the  state.  There  are  ambiguities  as  to  what  is  required  to  comply  with  these  state  requirements  and  if  we  fail  to 
comply with an applicable state law requirement, we could be subject to penalties.

15

In addition, regulators globally are also imposing greater monetary fines for privacy violations. The General Data 
Protection Regulation (GDPR), which went into effect on May 25, 2018, applies to any company established in the 
European Union (EU) as well as to those outside the EU if they collect and use personal data in connection with the 
offering goods or services to individuals in the EU or the monitoring of their behavior. The GDPR enhances data 
protection obligations for processors and controllers of personal data, including, for example, expanded disclosures 
about  how  personal  information  is  to  be  used,  limitations  on  retention  of  information,  mandatory  data  breach 
notification requirements and onerous new obligations on services providers. Noncompliance with the GDPR may 
result in monetary penalties of up to €20 million or 4% of worldwide revenue, whichever is higher. The GDPR also 
confers a private right of action on data subjects and consumer associations to lodge complaints with supervisory 
authorities, seek judicial remedies, and obtain compensation for damages resulting from violations. In addition, the 
GDPR includes restrictions on cross-border data transfers. The GDPR may increase our responsibility and liability 
in relation to personal data that we process where such processing is subject to the GDPR, and we may be required 
to put in place additional mechanisms to ensure compliance with the GDPR, including as implemented by individual 
countries.

California  recently  enacted  the  California  Consumer  Privacy  Act  (CCPA)  which  creates  new  individual  privacy 
rights  for  California  consumers  (as  defined  in  the  law)  and  places  increased  privacy  and  security  obligations  on 
entities handling personal data of consumers or households. The CCPA will require covered companies to provide 
certain  disclosures  to  consumers  about  its  data  collection,  use  and  sharing  practices,  and  to  provide  affected 
California residents with ways to opt-out of certain sales or transfers of personal information. The CCPA went into 
effect  on  January  1,  2020,  and  the  California  Attorney  General  began  taking  enforcement  action  against  violators 
beginning  July  1,  2020.  While  there  is  currently  an  exception  for  protected  health  information  that  is  subject  to 
HIPAA and clinical trial regulations, as currently written, the CCPA may impact our business activities. 

Competition

The pharmaceutical and biotechnology industry is very competitive, and the development and commercialization of 
new  drugs  is  influenced  by  rapid  technological  developments  and  innovation.  We  face  competition  from  several 
companies  developing  and  commercializing  products  that  will  be  competitive  with  our  drug  candidates,  including 
large  pharmaceutical  and  smaller  biotechnology  companies.  Additionally,  new  entrants  may  potentially  enter  the 
market.  Potential  competitors  include  Johnson  &  Johnson,  Roche,  Gilead  Sciences  Inc.,  GlaxoSmithKline  plc, 
Enanta Pharmaceuticals, Inc., HEC Pharma, Arbutus, Vir Bio and Aligos Therapeutics, among others. Additionally, 
we may face competition from currently available HBV treatments. Some of the competitive development programs 
from  these  companies  may  be  based  on  scientific  approaches  that  are  similar  to  our  approach,  and  others  may  be 
based  on  entirely  different  approaches.  Potential  competitors  also  include  academic  institutions,  government 
agencies  and  other  public  and  private  research  organizations  that  conduct  research,  seek  patent  protection  and 
establish  collaborative  arrangements  for  research,  development,  manufacturing  and  commercialization  of  products 
similar to ours or that otherwise target indications that we are pursuing.

Manufacturing

We currently rely on third-party manufacturers to supply the quantities of VBR, 2158 and 3733 used in our clinical 
and  nonclinical  studies.  We  currently  have  no  plans  to  establish  any  manufacturing  facilities  for  our  product 
candidates. 

Human Capital Management

Employees

As  of  December  31,  2020,  we  had  139  total  employees  and  contracts  with  a  number  of  temporary  contractors, 
consultants and contract research organizations. Our employees are spread across facilities in South San Francisco, 
California, Groton, Connecticut and a small facility in China. We also have a small number of remote employees 
spread across the United States. During 2020, we increased our headcount by adding 51 new employees. The new 
employees were hired to support, extend and grow our clinical and preclinical pipeline, with new hires in clinical 
development and operations, research, manufacturing and general and administrative functions, including expanding 
our corporate development team. Following the wind-down of our Microbiome program on January 31, 2021, we 
had  95  total  employees,  with  one  employee  remaining  in  Groton,  Connecticut  to  manage  the  shutdown  of  that 
facility.

16

While we wound down our Microbiome program in early 2021, we expect to continue to add employees to support 
our  HBV  programs  in  2021,  with  a  focus  on  continuing  to  build  out  our  clinical  team  to  support  ongoing  and 
planned clinical development studies and building out our preclinical research and development team under our new 
Chief Scientific Officer, who joined us in May 2020. We continually evaluate our needs and make strategic choices 
regarding whether to hire internal teams or outsource certain functions to contract research organizations (CROs) or 
contract  manufacturing  organizations  (CMOs),  as  appropriate.  We  currently  outsource  our  clinical  study 
management  to  various  CROs  and  utilize  certain  CMOs  to  manufacture  both  the  drug  substance  and  the  drug 
product used in our ongoing and planned clinical studies.

We compete with both large and small companies in our industry for a limited number of qualified applicants to fill 
highly specialized needs. We generally target our base salaries and annual performance-based cash bonuses at the 
50th percentile of our peers and our long-term equity incentive compensation, which all employees receive, between 
the 50th and 75th percentiles of our peers. In certain circumstances, we offer compensation above these levels, based 
on  a  candidate’s  experience,  criticality,  amount  of  responsibility  and  either  individual  or  Company-wide 
performance.  Both  annual  performance-based  cash  bonuses  and  long-term  equity  compensation  increase  as  a 
percentage  of  total  compensation  based  on  employees’  levels  of  responsibility.  We  also  offer  comprehensive 
benefits packages to all of our employees, including: 100% Company-covered medical, dental and vision coverage 
for  employees  and  their  families;  a  401k  program  with  a  Company  match;  an  employee  stock  purchase  plan;  and 
paid family leave.

A large majority of our employees have advanced degrees, and we also offer an educational assistance program that 
reimburses  employees  up  to  a  maximum  amount  per  year  for  courses  that  directly  enhance  his  or  her  area  of 
professional work or contribute to his or her immediate career growth. This program demonstrates our commitment 
to analytical growth, enhanced knowledge and professional development.

COVID-19 Response

Shortly after the counties in the San Francisco Bay Area implemented a shelter-in-place order, followed quickly by 
California’s similar statewide order, we established a COVID-19 Task Force (the Task Force) that has held regular 
meetings since it was established. The Task Force, in conjunction with our Human Resources department, has taken 
the following actions in our effort to curb the pandemic:

(cid:129) Drafting  and  distributing  comprehensive  COVID-19  office  and  exposure  policies,  and  lab  and  safety 
protocols,  each  of  which  have  been  modified  as  federal,  state  and  local  governments  have  updated  their 
guidance;

(cid:129)

Requiring all employees who are able to do so to work remotely;

(cid:129) Holding Company-wide virtual Town Hall meetings at least monthly to foster a sense of community given 

that the majority of our employees worked remotely;

(cid:129)

(cid:129)

(cid:129)

(cid:129)

Increasing cleaning protocols at U.S. office and lab facilities;

Providing  all  employees  with  cloth  face  coverings  and  increasing  availability  of  personal  protective 
equipment to lab employees;

Prohibiting all work-related domestic and international travel; and

Requiring masks to be worn at all Company locations.

The Task Force will continue to hold regular meetings to discuss and update internal guidance and protocols until 
we determine that meetings are no longer necessary.

Corporate History

We  were  incorporated  in  Delaware  in  October  2005  under  the  name  South  Island  Biosciences,  Inc.  (which  was 
changed  to  Ventrus  Biosciences,  Inc.  in  April  2007).  On  July  11,  2014,  we  acquired  Assembly  Pharmaceuticals, 
Inc., a private company, through a merger with our wholly owned subsidiary (the Merger). In connection with the 
Merger, we changed our name from Ventrus Biosciences, Inc. to Assembly Biosciences, Inc.

17

Corporate Information

Our principal executive office is at 331 Oyster Point Blvd., Fourth Floor, South San Francisco, California 94080. 
Our telephone number is (833) 409-4583.

Available Information

Our  website  address  is  www.assemblybio.com.  We  routinely  post,  or  have  posted,  important  information  for 
investors  on  our  website  in  the  “Investors”  section.  We  use  this  website  as  a  means  of  disclosing  material 
information  in  compliance  with  our  disclosure  obligations  under  Regulation  FD.  Accordingly,  investors  should 
monitor the “Investors” section of our website, in addition to following our press releases, Securities and Exchange 
Commission (SEC) filings, presentations and webcasts. We make available free of charge through our website our 
press releases, Annual Reports on Form 10-K, Quarterly Reports on Form 10-Q, Current Reports on Form 8-K and 
all amendments to those reports as soon as reasonably practicable after electronically filed with or furnished to the 
SEC.

The  information  contained  on  our  website  is  not  a  part  of,  and  should  not  be  construed  as  being  incorporated  by 
reference, into this report.

The  reports  filed  with  the  SEC  by  us  and  by  our  officers,  directors  and  significant  shareholders  are  available  for 
review on the SEC’s website at www.sec.gov.

Item 1A. Risk Factors

You should carefully consider the following risk factors, together with all other information in this report, including 
our consolidated financial statements and notes thereto, and in our other filings with the Securities and Exchange 
Commission. If any of the following risks, or other risks not presently known to us or that we currently believe to not 
be  material,  develop  into  actual  events,  then  our  business,  financial  condition,  results  of  operations  or  prospects 
could  be  materially  adversely  affected.  If  that  happens,  the  market  price  of  our  common  stock  could  decline,  and 
stockholders may lose all or part of their investment.

Risks Related to Our Business

We have no approved products and depend on the future success of our HBV program. We cannot be certain that 
we  or  our  collaborators  will  be  able  to  obtain  regulatory  approval  for,  or  successfully  commercialize,  product 
candidates from our current pipeline or any other product candidates that we may subsequently identify, license 
or otherwise acquire.

We  and  our  collaborators  are  not  permitted  to  market  or  promote  any  product  candidates  in  the  United  States, 
Europe,  China  or  other  countries  before  we  receive  regulatory  approval  from  the  FDA  or  comparable  foreign 
regulatory authorities, and we may never receive such regulatory approval for our current product candidates. We 
have  not  submitted  a  new  drug  application  (NDA)  to  the  FDA  or  comparable  applications  to  other  regulatory 
authorities and do not expect to be in a position to do so in the near future.

All  of  our  product  candidates  are  in  clinical  development  or  in  varying  stages  of  nonclinical  development.  Data 
supporting  our  drug  discovery  and  nonclinical  and  clinical  development  programs  are  derived  from  laboratory 
studies,  nonclinical  studies  and  Phase  1  and  Phase  2  clinical  studies.  It  may  be  years  before  the  larger,  pivotal 
studies necessary to support regulatory approval of our current product candidates are completed, if ever. 

In addition to our current product pipeline, we may identify, license or otherwise acquire rights to other technologies 
or product candidates. Any such transactions would involve numerous risks, and we may be unsuccessful in entering 
into any such transactions or developing any such technologies or product candidates.

For these reasons, our drug discovery and development may not be successful, and we may be unable to continue 
clinical development of our product candidates and may not generate product approvals or product revenue, any of 
which could have a material adverse impact on our business, results of operations and financial condition. 

18

The COVID-19 pandemic may materially and adversely affect our business.

The  continued  spread  of  COVID-19  could  adversely  impact  our  research  and  development  through  delay, 
modification or suspension of our clinical and/or nonclinical studies. Other clinical-stage biotechnology companies, 
like us, have had their clinical and nonclinical studies affected by the COVID-19 pandemic.

The  COVID-19  pandemic  has  and  may  continue  to:  (1)  impact  patient  enrollment,  retention  or  compliance  with 
clinical study protocols; (2) require modifications to, or deviations from, study protocols and procedures, such as the 
use of telehealth and home health visits instead of on-site monitoring and treatment, which could increase the cost 
of,  and  time  for,  conducting  clinical  studies;  (3) disrupt  or  suspend  the  business  operations  of  our  third-party 
contract research organizations (CROs), manufacturers of our drug candidates and the clinical sites conducting our 
clinical  studies;  (4) delay  regulatory  meetings  and  filings  with  regulatory  agencies  in  the  United  States  and  other 
countries; and (5) disrupt supply chains and cause delays of shipments of critical reagents, PPE and disinfectants, 
each of which are necessary for our laboratories and the laboratories of our CROs to maintain normal workflows. 
Even if we are able to timely collect clinical data while the outbreak is ongoing, COVID-19 may negatively affect 
the quality, completeness, integrity, interpretability and cost of obtaining such clinical study data. 

The  full  extent  of  the  pandemic’s  impact  on  our  business  will  depend  on  future  developments,  which  are  highly 
uncertain  and  cannot  be  predicted  with  confidence,  such  as  the  duration  and  severity  of  the  pandemic  and  the 
effectiveness of actions for containment, treatment and prevention of COVID-19. However, any COVID-19-related 
business  interruptions  or  delays  could  materially  and  adversely  affect  our  ability  to  conduct  our  research  and 
development activities in the manner and on the timelines presently planned as well as negatively affect the accuracy 
of our estimates regarding capital requirements, needs for additional financing and our ability to produce accurate 
and  timely  financial  statements.  Any  of  these  disruptions  could  have  a  material  adverse  impact  on  our  business, 
results of operations, financial condition and share price. 

As a result of the COVID-19 pandemic, governments around the world implemented significant measures to control 
the spread of the virus, including quarantines, travel restrictions, stay-at-home orders and business shutdowns. While 
governments have relaxed these measures as cases numbers go down, periodic surges in COVID-19 cases have, and 
may  in  the  future,  prompted  many  governments  to  reimplement  these  restrictions,  including  in  Europe  and  the 
United States. We continue to take precautionary measures intended to minimize our employees’ potential exposure 
to the virus, including temporarily requiring all employees who are able to do so to work remotely and suspending 
all  non-essential  business  travel  worldwide  for  our  employees.  Requiring  all  employees  to  work  remotely  may 
disrupt our operations, increase the risk of a cybersecurity incident or otherwise negatively affect our business.

In addition to the risks related to the COVID-19 pandemic discussed above, the uncertainty surrounding, and risks 
created  by,  the  pandemic  may  have  the  effect  of  heightening  many  of  the  other  risks  discussed  in  this  section 
impacting our operations.

We  are  not  currently  profitable  and  might  never  become  profitable,  and  we  will  need  additional  financing  to 
complete the development of any product candidates and fund our activities into the future.

We do not have any approved products, and we have a history of losses. We expect to continue to incur substantial 
operating and capital expenditures to advance our current product candidates through clinical development, continue 
research and discovery efforts to identify potential additional product candidates and seek regulatory approvals for 
our current and future product candidates. All operations and capital expenditures will be funded from cash on hand, 
securities  offerings  or  debt  financings  and  payments  we  may  receive  from  out-licensing,  collaborations  or  other 
strategic arrangements. However, there is no assurance that we will be successful in raising any necessary additional 
capital  on  terms  that  are  acceptable  to  us,  or  at  all.  If  we  are  unable  to  develop  and  commercialize  any  product 
candidates and generate sufficient revenue or raise capital, we could be forced to delay, scale back or discontinue 
product  development  and  clinical  studies,  sacrifice  attractive  business  opportunities,  cease  operations  entirely  and 
sell, or otherwise transfer, all or substantially all of our remaining assets, which would likely have a material adverse 
impact on our business, results of operations, financial condition and share price.

19

Nonclinical and clinical testing required for our product candidates is expensive and time-consuming and may 
fail to demonstrate the level of safety and efficacy necessary for product approval. 

Before we or any commercial partners can obtain FDA approval (or other foreign approvals) necessary to sell any of 
our  product  candidates,  we  must  show  that  each  potential  product  is  safe  and  effective  in  humans.  To  meet  these 
requirements, we must conduct extensive nonclinical testing and sufficient, well-controlled clinical studies. 

The results of nonclinical studies may not be representative of disease behavior in a clinical setting and thus may not 
be  predictive  of  the  outcomes  of  our  clinical  studies.  In  addition,  the  results  of  early  clinical  studies  of  product 
candidates may not be predictive of the results of later-stage clinical studies.

Conducting nonclinical and clinical studies is a lengthy, time consuming and expensive process. The length of time 
varies substantially according to the type, complexity, novelty, and intended use of the product candidate, and often 
can be several years or more. In addition, failure or delays can occur at any time during the nonclinical and clinical 
study process, resulting in additional operating expenses or harm to our business. 

The  commencement  and  rate  of  completion  of  clinical  studies  might  be  delayed  by  many  factors,  including,  for 
example:

(cid:129)

(cid:129)

(cid:129)

(cid:129)

(cid:129)

(cid:129)

delays in reaching agreement with regulatory authorities on trial design;

delays in reaching agreement on acceptable terms with prospective CROs and clinical study sites;

failure to demonstrate efficacy or the emergence of unforeseen safety issues;

insufficient quantities of qualified materials under cGMP for use in clinical studies due to manufacturing 
challenges, delays or interruptions in the supply chain;

slower  than  expected  rates  of  patient  recruitment  or  failure  to  recruit  a  sufficient  number  of  eligible 
patients,  which  may  be  due  to  a  number  of  reasons,  including  the  size  of  the  patient  population,  the 
proximity of patients to clinical sites, the eligibility criteria for the study, the design of the clinical study, 
and other potential drug candidates being studied;

delays in patients completing participation in a trial or return for post-treatment follow-up for any reason, 
including, product side effects or disease progression;

(cid:129) modification of clinical study protocols;

(cid:129)

(cid:129)

delays, suspension, or termination of clinical studies by the institutional review board or ethics committee 
responsible for overseeing the study at a particular study site; and

government or other regulatory agency delays or clinical holds requiring suspension or termination of our 
clinical studies due to safety, tolerability or other issues related to our product candidates.

The failure of nonclinical and clinical studies to demonstrate safety and effectiveness of a product candidate for the 
desired indications, whether conducted by us or by a CRO, would harm the development of that product candidate 
and potentially other product candidates. This failure could cause us to abandon a product candidate and could delay 
development of other product candidates. Any delay in, or failure of, our nonclinical studies or clinical studies could 
delay,  or  preclude,  the  filing  of  our  NDAs  and  comparable  applications  with  the  FDA  and  foreign  regulatory 
agencies, as applicable, and materially harm our business, prospects, financial condition and results of operations.

We rely on CROs to conduct some of this testing due to our lack of suitable facilities and resources.

We  do  not  have  sufficient  facilities  or  resources  to  conduct  all  of  our  anticipated  nonclinical  and  clinical  testing 
internally. As a result, we contract with CROs to conduct a significant portion of the nonclinical and clinical testing 
required for regulatory approval for our product candidates. Our reliance on CROs reduces our control over these 
activities but does not relieve us of our responsibilities. For example, we are responsible for ensuring that each of 
our studies is conducted in accordance with the applicable protocol, legal and regulatory requirements and scientific 
standards, including, in the case of clinical studies, good clinical practices, even if the study is conducted by a CRO. 

20

In the event CROs fail to perform their duties in such a fashion or we are unable to retain or continue with CROs on 
acceptable terms, we may not be able to complete our clinical studies and may fail to obtain regulatory approval for 
our product candidates.

Furthermore, these CROs may also have relationships with other entities, some of which may be our competitors. 
CRO personnel are not our employees, and except for remedies available to us under our agreements with such third 
parties,  we  cannot  control  whether  they  devote  sufficient  time  and  resources  to  our  clinical  and  nonclinical 
programs.  If  the  CROs  do  not  successfully  carry  out  their  contractual  duties  or  obligations  or  meet  expected 
deadlines, if they need to be replaced or if the quality or accuracy of the clinical data they obtain is compromised 
due  to  the  failure  to  adhere  to  our  clinical  protocols,  regulatory  requirements  or  for  other  reasons,  our  research, 
nonclinical studies or clinical studies may be extended, delayed or terminated and we may not be able to obtain, or 
may be delayed in obtaining, regulatory approvals for our product candidates, any of which could materially harm 
our business, prospects, financial condition and results of operations.

Top-line or preliminary data may not accurately reflect the final results of a particular study or trial.

We may publicly disclose top-line or preliminary data based on analysis of then-available efficacy, tolerability, PK 
and  safety  data,  and  the  results  and  related  findings  and  conclusions  are  subject  to  change  following  a  more 
comprehensive  review  of  the  data  related  to  the  particular  study  or  trial.  We  also  make  assumptions,  estimates, 
calculations and conclusions as part of our data analyses, and we may not have received or had the opportunity to 
fully and carefully evaluate all data prior to release.  As a  result,  the top-line or preliminary results that we report 
may differ from final results of the same studies or different conclusions or considerations may qualify such results 
once  additional  data  have  been  received  and  fully  evaluated.  Top-line  data  also  remains  subject  to  audit  and 
verification procedures that may result in the final data differing materially from previously published preliminary 
data. As a result, top-line and preliminary data should be viewed with caution until the final data are available.

In  addition  to  top-line  or  preliminary  results,  the  information  we  may  publicly  disclose  regarding  a  particular 
nonclinical  or  clinical  study  is  based  on  extensive  information,  and  you  or  others  may  not  agree  with  what  we 
determine  is  the  material  or  otherwise  appropriate  information  to  include  in  our  disclosure.  In  addition,  any 
information  we  determine  not  to  disclose  may  ultimately  be  deemed  significant  with  respect  to  future  decisions, 
conclusions, views, activities or otherwise regarding a particular drug, drug candidate or our business. If the top-line 
or  preliminary  data  that  we  report  differ  from  final  results,  or  if  others,  including  regulatory  authorities,  disagree 
with, or do not accept, the data or conclusions reached, our ability to obtain approval for, and commercialize, our 
product candidates may be harmed or delayed, which could harm our business, financial condition, operating results 
or prospects.

We  rely  on  third  parties  to  formulate  and  manufacture  our  product  candidates  and  products  that  we  study  in 
combination  with  our  product  candidates.  Our  use  of  third  parties  may  increase  the  risk  that  we  will  not  have 
sufficient quantities of our product candidates or other products on time or at an acceptable cost.

We  rely  on  third-party  manufacturers  to  supply  the  quantities  of  VBR,  2158  and  3733  used  in  our  clinical  and 
nonclinical studies. If any product candidate we develop or acquire in the future receives FDA or other regulatory 
approval, we expect to continue our reliance on one or more third-party contractors to manufacture our products. If, 
for  any  reason,  we  are  unable  to  rely  on  any  third-party  sources  we  have  identified  to  manufacture  our  product 
candidates,  we  would  need  to  identify  and  contract  with  additional  or  replacement  third-party  manufacturers  to 
manufacture compounds, drug substances and drug products for nonclinical, clinical and commercial purposes. We 
may  not  be  successful  in  identifying  additional  or  replacement  third-party  manufacturers,  or  in  negotiating 
acceptable terms with any that we do identify. If we are unable to establish and maintain manufacturing capacity, the 
development and sales of our products and our financial performance may be materially and adversely affected.

We are exposed to the following risks with respect to the manufacture of our product candidates:

(cid:129) We will need to identify manufacturers for commercial supply on acceptable terms, which we may not be 
able  to  do  because  the  number  of  potential  manufacturers  is  limited,  and  the  FDA  must  evaluate  and 
approve any new or replacement contractor. 

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(cid:129) Any third-party manufacturers with whom we contract might be unable to formulate and manufacture our 
product  candidates  in  the  volume  and  quality  required  to  meet  our  clinical  and,  if  approved,  commercial 
needs in a timely manner.

(cid:129) Any third-party manufacturers with whom we contract might not perform as agreed or might not remain in 

the contract manufacturing business for the time required to supply our products.

(cid:129) One or more of any third-party manufacturers with whom we contract could be foreign, which increases the 

risk of shipping delays and adds the risk of import restrictions.

(cid:129) We do not have complete control over, and cannot ensure, any third-party manufacturers’ compliance with 
cGMP and other government regulations and corresponding foreign requirements, including periodic FDA 
and state regulatory inspections.

(cid:129) We  may  be  required  to  obtain  intellectual  property  rights  from  third  parties  in  order  to  manufacture  our 
product candidates, and if any third-party manufacturer makes improvements in the manufacturing process 
for our product candidates, we may not own, or may have to share, the intellectual property rights to the 
innovation.

(cid:129) We  may  be  required  to  share  our  trade  secrets  and  know-how  with  third  parties,  thereby  risking  the 

misappropriation or disclosure of our intellectual property by or to third parties.

(cid:129) When  contracting  with  third-party  manufacturers,  we  might  compete  with  other  companies  for  access  to 
these manufacturers’ facilities and might be subject to manufacturing delays if the manufacturers give other 
clients higher priority than we are given.

Each of these risks could delay our development efforts, nonclinical studies and clinical studies or the approval, if 
any, of our product candidates by the FDA or applicable non-U.S. regulatory authorities and the commercialization 
of  our  product  candidates.  This  could  result  in  higher  costs  or  deprive  us  of  potential  product  revenues  and 
materially harm our business, financial condition and results of operations.

If  we  lose  key  management  personnel  and  cannot  recruit  and  retain  similarly  qualified  replacements,  our 
business may materially suffer.

We are highly dependent on the services of our executive officers. Our employment agreements with our executive 
officers do not ensure their retention. We do not currently maintain, nor do we intend to obtain in the future, “key 
person” life insurance that would compensate us in the event of the death or disability of any of the members of our 
management team. Our executive officers are critical to our success, and loss of any of these key employees could 
have a material adverse impact on our business, financial condition and results of operations.

Fast Track designations for VBR and 2158 may not result in faster development, regulatory review or approval.

If nonclinical or clinical data demonstrate potential to address unmet medical needs for a serious or life-threatening 
condition,  the  sponsor  may  apply  for  FDA  Fast  Track  designation.  Fast  Track  designation  provides  increased 
opportunities  for  sponsor  meetings  with  the  FDA  during  nonclinical  and  clinical  development,  in  addition  to  the 
potential  for  rolling  review  once  a  marketing  application  is  filed.  Both  VBR  and  2158  have  received  Fast  Track 
designation for the treatment of patients with chronic HBV infection. However, even with Fast Track designation, 
we  may  not  experience  a  faster  development  process,  review  or  approval  compared  to  conventional  FDA 
procedures.  Fast  Track  designation  does  not  assure  ultimate  approval  by  the  FDA.  The  FDA  may  withdraw  Fast 
Track designation if it believes that the designation is no longer supported by data from our product development 
program. Any such withdrawal could adversely affect our business.

We are dependent on an in-license relationship for VBR.

Our  license  agreement  with  IURTC  imposes  diligence  requirements  on  us  and  requires  us  to  make  milestone 
payments based upon the successful accomplishment of clinical and regulatory milestones related to VBR, royalty 
payments if VBR is approved and diligence maintenance fees. These payments will make it less profitable for us to 
develop VBR than if we owned the technology outright. In addition, if we breach any of our obligations under our 
license  agreement,  IURTC  may  have  a  right  to  terminate  the  license,  in  which  event  we  could  lose  our  rights  to 
VBR. 

22

Our collaboration partners might delay, prevent, or undermine the success of our product candidates.

Our  operating  and  financial  strategy  for  the  development,  nonclinical  and  clinical  testing,  manufacture,  and 
commercialization  of  drug  candidates  heavily  depends  on  collaborating  with  corporations,  academic  institutions, 
licensors,  licensees,  and  other  parties.  However,  there  can  be  no  assurance  that  we  will  successfully  establish  or 
maintain these collaborations. If a collaboration is terminated, replacement collaborators might not be available on 
attractive terms, or at all. 

The  activities  of  any  collaborator  will  not  be  within  our  control  and  might  not  be  within  our  power  to  influence. 
There can be no assurance that any collaborator will perform its obligations to our satisfaction or at all, that we will 
derive  any  revenue  or  profits  from  these  collaborations,  or  that  any  collaborator  will  not  compete  with  us.  If  any 
collaboration is unsuccessful, we might require substantially greater capital to undertake development and marketing 
of  our  proposed  products  and  might  not  be  able  to  develop  and  market  these  products  effectively,  if  at  all.  In 
addition,  a  lack  of  development  and  marketing  collaborations  might  lead  to  significant  delays  in  introducing 
proposed products into certain markets and/or reduced sales of proposed products in such markets.

We rely on data provided by third parties that has not been independently verified and could prove to be false, 
misleading, or incomplete.

We  rely  on  third-party  vendors,  scientists,  investigators  and  collaborators  to  provide  us  with  significant  data  and 
other  information  related  to  our  projects,  nonclinical  studies  and  clinical  studies,  and  our  business.  If  these  third 
parties provide inaccurate, misleading, or incomplete data, our business, prospects, and results of operations could 
be materially adversely affected.

Significant  disruptions  of  information  technology  systems  or  breaches  of  data  security  could  materially  and 
adversely affect our business, results of operations and financial condition.

We  collect  and  maintain  information  in  digital  form  and  are  increasingly  dependent  on  information  technology 
systems  and  infrastructure  to  operate  our  business.  In  the  ordinary  course  of  our  business,  we  collect,  store  and 
transmit large amounts of confidential information, including intellectual property, proprietary business information 
and personal information. It is critical that we do so in a secure manner to maintain the confidentiality and integrity 
of such confidential information. We have outsourced elements of our information technology infrastructure and, as 
a  result,  a  number  of  third-party  vendors  may  or  could  have  access  to  our  confidential  information.  Our  internal 
information technology systems and infrastructure, and those of our current and any future collaborators, contractors 
and consultants and other third parties on which we rely, are vulnerable to damage from computer viruses, malware, 
natural disasters, terrorism, war, telecommunication and electrical failures, cyberattacks or cyber intrusions over the 
Internet,  attachments  to  emails,  persons  inside  our  organization,  or  persons  with  access  to  systems  inside  our 
organization.

The risk of a security breach or disruption, particularly through cyberattacks or cyber intrusion, has escalated as the 
number, intensity and sophistication of attempted attacks and intrusions from around the world have increased. In 
addition, the prevalent use of mobile devices that access confidential information increases the risk of data security 
breaches, which could lead to the loss of confidential information or other intellectual property. The costs to us to 
mitigate network security problems, bugs, viruses, worms, malicious software programs and security vulnerabilities 
could  be  significant,  and  our  efforts  to  address  these  problems  may  not  be  successful.  If  unsuccessful,  these 
problems could cause interruptions, delays, cessation of service and other harm to our business and our competitive 
position, including material disruption of our product development programs. For example, any loss of clinical study 
data from completed or ongoing or planned clinical studies could result in delays in our regulatory approval efforts 
and significantly increase our costs to recover or reproduce the data.

If  a  computer  security  breach  affects  our  systems  or  results  in  the  unauthorized  release  of  personally  identifiable 
information,  our  reputation  could  be  materially  damaged.  In  addition,  such  a  breach  may  require  notification  to 
governmental agencies, the media or individuals pursuant to various federal, state and non-U.S. privacy and security 
laws, if applicable, including the Health Insurance Portability and Accountability Act of 1996 (HIPAA), as amended 
by the Health Information Technology for Clinical Health Act of 2009 (HITECH), and its implementing rules and 
regulations, as well as regulations promulgated by the Federal Trade Commission, state breach notification law and 
the European Union’s General Data Protection Regulation (GDPR). We would also be exposed to a risk of loss or 
litigation  and  potential  liability,  which  could  materially  adversely  affect  our  business,  results  of  operations  and 
financial condition.

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Research,  development  and  commercialization  goals  may  not  be  achieved  in  the  timeframes  that  we  publicly 
estimate, which could have an adverse impact on our business and could cause our stock price to decline.

We  set  goals,  and  make  public  statements  regarding  our  expectations,  regarding  the  timing  of  certain 
accomplishments, developments and milestones under our research and development programs. The actual timing of 
these events can vary significantly due to a number of factors, including, the amount of time, effort and resources 
committed to our programs by us and any collaborators and the uncertainties inherent in the clinical development 
and regulatory approval process. As a result, there can be no assurance that we or any collaborators will initiate or 
complete clinical development activities, make regulatory submissions or receive regulatory approvals as planned or 
that we or any collaborators will be able to adhere to our current schedule for the achievement of key milestones 
under any of our programs. If we or any collaborators fail to achieve one or more of the milestones as planned, our 
business could be materially adversely affected, and the price of our common stock could decline.

Developments by competitors might render our product candidates or technologies obsolete or non-competitive.

The pharmaceutical and biotechnology industries are intensely competitive. In addition, the clinical and commercial 
landscape  for  HBV  is  rapidly  changing;  we  expect  new  data  from  commercial  and  clinical-stage  products  to 
continue to emerge. We compete with organizations, some with significantly more resources, who are developing 
competitive product candidates. If our competitors develop effective treatments for HBV or any other indication or 
field  we  might  pursue,  and  successfully  commercialize  those  treatments,  our  business  and  prospects  could  be 
materially harmed.  

Companies with core inhibitor products may produce negative clinical data, which would adversely affect public 
and clinical communities’ perceptions of our product candidates, and may negatively impact regulatory approval 
of, or demand for, our potential products.

Our HBV therapy research and development efforts involve therapeutics based on modulating forms of HBV core 
proteins with core inhibitors. Negative data from clinical studies using a competitor’s core inhibitors could adversely 
impact the perception of the therapeutic use of our product candidates and our ability to enroll patients in clinical 
studies. 

The  clinical  and  commercial  success  of  our  potential  products  will  depend  in  part  on  the  public  and  clinical 
communities’  acceptance  of  core  inhibitors,  a  novel  class  of  product  candidates.  Moreover,  our  success  depends 
upon  physicians  prescribing,  and  their  patients  being  willing  to  receive,  treatments  that  involve  the  use  of  core 
inhibitor product candidates we may develop in lieu of, or in addition to, existing treatments with which they are 
already  familiar  and  for  which  more  clinical  data  may  be  available.  Adverse  events  in  our  nonclinical  or  clinical 
studies  or  those  of  our  competitors  or  of  academic  researchers  utilizing  core  inhibitor  therapies,  even  if  not 
ultimately attributable to our product candidates, and any resulting publicity could result in increased governmental 
regulation,  unfavorable  public  perception,  potential  regulatory  delays  in  the  testing  or  approval  of  our  product 
candidates,  stricter  labeling  requirements  for  our  product  candidates  that  are  approved,  if  any,  and  a  decrease  in 
demand for any such products.

Risks Related to Our Regulatory and Legal Environment

We  are  and  will  be  subject  to  extensive  and  costly  government  regulation  and  the  failure  to  comply  with  these 
regulations may have a material adverse effect on our operations and business.

Our product candidates are subject to extensive and rigorous domestic government regulation including regulation 
by the FDA, the Centers for Medicare and Medicaid Services, other divisions of the U.S. Department of Health and 
Human  Services,  the  U.S.  Department  of  Justice,  state  and  local  governments,  and  their  respective  foreign 
equivalents.  Both  before  and  after  approval  of  any  product,  we  and  our  collaborators,  suppliers,  contract 
manufacturers  and  clinical  investigators  are  subject  to  extensive  regulation  by  governmental  authorities  in  the 
United  States  and  other  countries,  covering,  among  other  things,  testing,  manufacturing,  quality  control,  clinical 
studies,  post-marketing  studies,  labeling,  advertising,  promotion,  distribution,  import  and  export,  governmental 
pricing, price reporting and rebate requirements. Failure to comply with applicable requirements could result in one 
or  more  of  the  following  actions:  warning  or  untitled  letters;  unanticipated  expenditures;  delays  in  approval  or 
refusal  to  approve  a  product  candidate;  voluntary  or  mandatory  product  recall;  product  seizure;  interruption  of 
manufacturing or clinical studies; operating or marketing restrictions; injunctions; criminal prosecution and civil or 

24

criminal penalties including fines and other monetary penalties; exclusion from federal health care programs such as 
Medicare and Medicaid; adverse publicity; and disruptions to our business. 

If we or our collaborators are able to obtain regulatory approval for a particular product, the approval might limit the 
intended medical uses for the product, limit our ability to promote, sell, and distribute the product, require that we 
conduct  costly  post-marketing  surveillance,  and/or  require  that  we  conduct  ongoing  post-marketing  studies.  Once 
obtained,  any  approvals  might  be  withdrawn,  including,  for  example,  if  there  is  a  later  discovery  of  previously 
unknown problems with the product, such as a previously unknown safety issue.

If we, our collaborators, or our contract manufacturers fail to comply with applicable regulatory requirements at any 
stage  during  the  regulatory  process,  such  noncompliance  could  result  in  delays  in  the  approval  of  applications  or 
supplements  to  approved  applications,  refusal  by  a  regulatory  authority  (including  the  FDA)  to  review  pending 
market  approval  applications  or  supplements  to  approved  applications,  untitled  letters  or  warning  letters,  fines, 
import and export restrictions, product recalls or seizures, injunctions, total or partial suspension of production, civil 
penalties,  withdrawals  of  previously  approved  marketing  applications,  recommendations  by  the  FDA  or  other 
regulatory authorities against governmental contracts, and/or criminal prosecutions.

The regulatory approval processes of the FDA and comparable foreign authorities are lengthy, time consuming 
and inherently unpredictable, and if we or our collaborators are ultimately unable to obtain regulatory approval 
for our product candidates, our business will be substantially harmed.

We,  or  any  current  or  future  collaborators,  cannot  assure  you  that  we  will  receive  the  approvals  necessary  to 
commercialize for sale any of our product candidates, or any product candidate we acquire or develop in the future. 
We will need FDA approval to commercialize our product candidates in the United States and approvals from the 
applicable  regulatory  authorities  in  foreign  jurisdictions  to  commercialize  our  product  candidates  in  those 
jurisdictions.  In  order  to  obtain  FDA  approval  of  any  product  candidate,  we  must  submit  to  the  FDA  an  NDA 
demonstrating that the product candidate is safe and effective for its intended use. This requires significant research, 
nonclinical  studies,  and  clinical  studies.  Satisfaction  of  the  FDA’s  regulatory  requirements  typically  takes  many 
years, depends upon the type, complexity and novelty of the product candidate and requires substantial resources for 
research,  development  and  testing.  We  cannot  predict  whether  our  research  and  clinical  approaches  will  result  in 
drugs that the FDA considers safe and effective for their indicated uses. The FDA has substantial discretion in the 
approval process and might require us to conduct additional nonclinical and clinical testing, perform post-marketing 
studies or otherwise limit or impose conditions on any approval we obtain.

The  approval  process  might  also  be  delayed  by  changes  in  government  regulation,  future  legislation  or 
administrative  action  or  changes  in  FDA  policy  that  occur  prior  to  or  during  our  regulatory  review.  Delays  in 
obtaining regulatory approvals might: delay commercialization of, and our ability to derive product revenues from, 
our  product  candidates;  impose  costly  procedures  on  us;  and  diminish  any  competitive  advantages  that  we  might 
otherwise enjoy.

Even if we comply with all FDA requests, the FDA might ultimately reject one or more of our NDAs. We cannot be 
sure that we will ever obtain regulatory approval and commercialize any of our current or future product candidates. 
In foreign jurisdictions, we are subject to regulatory approval processes and risks similar to those associated with the 
FDA  described  above.  We  cannot  assure  you  that  we  will  receive  the  approvals  necessary  to  commercialize  our 
product candidates for sale outside the United States.

We and our collaborators may be subject, directly or indirectly, to applicable U.S. federal and state anti-kickback, 
false claims laws, physician payment transparency laws, fraud and abuse laws or similar healthcare and security 
laws  and  regulations,  and  health  information  privacy  and  security  laws,  which  could  expose  us  or  them  to 
criminal  sanctions,  civil  penalties,  contractual  damages,  reputational  harm  and  diminished  profits  and  future 
earnings.

Healthcare  providers,  physicians  and  others  play  a  primary  role  in  the  recommendation  and  prescription  of  any 
products for which we obtain regulatory approval. If we obtain FDA approval for any of our drug candidates and 
begin commercializing those drugs in the United States, our operations may be subject to various federal and state 
fraud  and  abuse  laws,  including  the  federal  Anti-Kickback  Statute,  the  federal  False  Claims  Act,  and  physician 
payment sunshine laws and regulations. Additionally, we are subject to state and non-U.S. equivalents of each of the 
healthcare laws described above, among others, some of which may be broader in scope and may apply regardless of 

25

the payor. These laws may impact, among other things, our proposed sales, marketing and education programs. In 
addition, we may be subject to patient privacy regulation by both the federal government and the states and foreign 
jurisdictions  in  which  we  conduct  our  business.  If  we  fail  to  comply  with  any  applicable  federal,  state  or  foreign 
legal requirement, we could be subject to penalties.

Regulators globally are imposing greater monetary fines for privacy violations. The GDPR applies to any company 
established in the European Union (EU) as well as to those outside the EU if they collect and use personal data in 
connection  with  the  offering  goods  or  services  to  individuals  in  the  EU  or  the  monitoring  of  their  behavior.  The 
GDPR enhances data protection obligations for processors and controllers of personal data, including, for example, 
expanded  disclosures  about  how  personal  information  is  to  be  used,  limitations  on  retention  of  information, 
mandatory data breach notification requirements and onerous new obligations on services providers. Noncompliance 
with the GDPR may result in monetary penalties of up to €20 million or 4% of worldwide revenue, whichever is 
higher. The GDPR may increase our responsibility and liability in relation to personal data that we process and we 
may  be  required  to  put  in  place  additional  mechanisms  to  ensure  compliance  with  the  GDPR,  including  as 
implemented  by  individual  countries.  Compliance  with  the  GDPR  and  other  changes  in  laws  or  regulations 
associated with the enhanced protection of certain types of personal data, such as healthcare data or other sensitive 
information,  could  greatly  increase  our  cost  of  developing  our  products  or  even  prevent  us  from  offering  certain 
products in jurisdictions that we may operate in. 

California  recently  enacted  the  CCPA,  which  creates  new  individual  privacy  rights  for  California  consumers  (as 
defined  in  the  law)  and  places  increased  privacy  and  security  obligations  on  entities  handling  personal  data  of 
consumers or households. The CCPA requires covered companies to provide certain disclosures to consumers about 
its  data  collection,  use  and  sharing  practices,  and  to  provide  affected  California  residents  with  ways  to  opt-out  of 
certain  sales  or  transfers  of  personal  information.  While  there  is  currently  an  exception  for  protected  health 
information that is subject to HIPAA and clinical trial regulations, as currently written, the CCPA may impact our 
business  activities.  The  uncertainty  surrounding  the  implementation  of  CCPA  exemplifies  the  vulnerability  of  our 
business to the evolving regulatory environment related to personal data and protected health information.

Because of the breadth of these laws and the narrowness of the statutory exceptions and safe harbors available, it is 
possible that some of our business activities could be subject to challenge under one or more of such laws. 

Violations  of  these  laws  may  be  punishable  by  criminal  and/or  civil  sanctions,  including  penalties,  fines  and/or 
exclusion or suspension from federal and state healthcare programs such as Medicare and Medicaid and debarment 
from  contracting  with  the  U.S.  government.  In  addition,  private  individuals  have  the  ability  to  bring  actions  on 
behalf of the U.S. government under the federal False Claims Act as well as under the false claims laws of several 
states.

If any of the physicians or other providers or entities with whom we expect to do business with are found to be not 
in  compliance  with  applicable  laws,  they  may  be  subject  to  criminal,  civil  or  administrative  sanctions,  including 
exclusions from government funded healthcare programs, which may also adversely affect our business.

We face the risk of product liability claims and might not be able to obtain insurance.

Our business exposes us to the risk of product liability claims that are inherent in drug development. If the use of 
one or more of our product candidates or approved drugs, if any, harms people, we might be subject to costly and 
damaging product liability claims brought against us by clinical study participants, consumers, health care providers, 
pharmaceutical companies or others selling our products. Our inability to obtain sufficient product liability/clinical 
study insurance at an acceptable cost to protect against potential product liability claims could prevent or inhibit the 
commercialization  of  pharmaceutical  products  we  develop.  We  cannot  predict  all  of  the  possible  harms  or  side 
effects  that  might  result  and,  therefore,  the  amount  of  insurance  coverage  we  maintain  might  not  be  adequate  to 
cover all liabilities we might incur. If we are unable to obtain insurance at an acceptable cost or otherwise protect 
against  potential  product  liability  claims,  we  will  be  exposed  to  significant  liabilities,  which  might  materially  and 
adversely affect our business and financial position. If we are sued for any injury allegedly caused by our products, 
our  liability  could  exceed  our  total  assets  and  our  ability  to  pay.  Any  successful  product  liability  claims  brought 
against us would decrease our cash and may adversely affect our business, stock price and financial condition.

26

We might be exposed to liability claims associated with the use of hazardous materials and chemicals.

Our research, development and manufacturing activities and/or those of our third-party contractors might involve the 
controlled  use  of  hazardous  materials  and  chemicals.  Although  we  will  strive  to  have  our  safety  procedures,  and 
those of our contractors, comply with federal, state and local laws and regulations for using, storing, handling and 
disposing  of  these  materials,  we  cannot  completely  eliminate  the  risk  of  accidental  injury  or  contamination  from 
these materials. In the event of such an accident, we could be held liable for any resulting damages, and any liability 
could  materially  and  adversely  affect  our  business,  financial  condition  and  results  of  operations.  In  addition,  the 
federal,  state  and  local  laws  and  regulations  governing  the  use,  manufacture,  storage,  handling  and  disposal  of 
hazardous  or  radioactive  materials  and  waste  products  might  require  us  to  incur  substantial  compliance  costs  that 
could  materially  and  adversely  affect  our  business,  financial  condition  and  results  of  operations.  We  do  not  carry 
hazardous  materials  liability  insurance.  We  intend  to  obtain  such  insurance  in  the  future,  if  necessary,  but  cannot 
give assurance that we will obtain such coverage.

Our  employees,  independent  contractors,  consultants,  collaborators  and  contract  research  organizations  may 
engage  in  misconduct  or  other  improper  activities,  including  noncompliance  with  regulatory  standards  and 
requirements, which could result in significant liability for us and harm our reputation.

We are exposed to the risk of fraud or other misconduct, including failure to:

(cid:129)

(cid:129)

(cid:129)

(cid:129)

(cid:129)

comply with applicable regulations of, and provide accurate information to, the FDA or comparable foreign 
regulatory authorities;

comply  with  federal  and  state  healthcare  fraud  and  abuse  laws  and  regulations  and  similar  laws  and 
regulations established and enforced by comparable foreign regulatory authorities;

comply with the United States Foreign Corrupt Practices Act (the FCPA), the U.K. Bribery Act 2010, the 
PRC Criminal Law, the PRC Anti-unfair Competition Law and other anti-bribery and trade laws;

report financial information and data accurately; or

disclose unauthorized activities.

Misconduct  could  also  involve  the  improper  use  or  misrepresentation  of  information  obtained  in  the  course  of 
clinical studies, creating fraudulent data in our nonclinical studies or clinical studies or illegal misappropriation of 
product  materials,  which  could  result  in  regulatory  sanctions,  delays  in  clinical  studies,  or  serious  harm  to  our 
reputation. 

It is not always possible to identify and deter misconduct. The precautions we take to detect and prevent this activity 
may not be effective in controlling unknown or unmanaged risks or losses or in protecting us from governmental 
investigations  or  other  actions  or  lawsuits  stemming  from  a  failure  to  be  in  compliance  with  such  laws  or 
regulations.  Additionally,  we  are  subject  to  the  risk  that  a  person  or  government  could  allege  such  fraud  or  other 
misconduct,  even  if  none  occurred.  If  any  such  actions  are  instituted  against  us  and  we  are  not  successful  in 
defending ourselves or asserting our rights, those actions could harm our business, results of operations, financial 
condition and cash flows, including through the imposition of significant fines or other sanctions.

We have international operations, including in China, and conduct clinical studies outside of the United States. A 
number of risks associated with international operations could materially and adversely affect our business.

We  expect  to  be  subject  to  a  number  of  risks  related  with  our  international  operations,  many  of  which  may  be 
beyond our control. These risks include:

(cid:129)

(cid:129)

(cid:129)

different regulatory requirements for drug approvals in foreign countries;

different  standards  of  care  in  various  countries  that  could  complicate  the  evaluation  of  our  product 
candidates;

different U.S. and foreign drug import and export rules;

27

(cid:129)

(cid:129)

(cid:129)

(cid:129)

(cid:129)

(cid:129)

(cid:129)

(cid:129)

different reimbursement systems and different competitive drugs indicated to treat the indication for which 
our product candidates are being developed;

reduced protection for intellectual property rights in certain countries;

unexpected changes in tariffs, trade barriers and regulatory requirements;

compliance with the FCPA and other anti-corruption and anti-bribery laws;

compliance with tax, employment, immigration and labor laws for employees living or traveling abroad;

foreign taxes, including withholding of payroll taxes;

foreign currency fluctuations and compliance with foreign currency exchange rules, which could result in 
increased  operating  expenses  and  reduced  revenues,  and  other  obligations  incident  to  doing  business  in 
another country; and

business  interruptions  resulting  from  geopolitical  actions,  including  tariffs,  war  and  terrorism,  natural 
disasters or outbreaks of disease.

Risks Related to Our Intellectual Property

Our business depends on protecting our intellectual property.

If we and our licensors do not obtain protection for our respective intellectual property rights, our competitors might 
be  able  to  take  advantage  of  our  research  and  development  efforts  to  develop  competing  drugs.  Our  success, 
competitive position and future revenues, if any, depend in part on our ability and the abilities of our licensors to 
obtain and maintain patent protection for our products, methods, processes and other technologies, to preserve our 
trade secrets, to prevent third parties from infringing on our proprietary rights and to operate without infringing the 
proprietary rights of third parties.

We  rely  upon  a  combination  of  patents,  trade  secret  protection  and  contractual  arrangements  to  protect  the 
intellectual  property  related  to  our  technologies.  We  will  only  be  able  to  protect  our  products  and  proprietary 
information  and  technology  by  preventing  unauthorized  use  by  third  parties  to  the  extent  that  our  patents,  trade 
secrets, and contractual position allow us to do so. We cannot be certain that we will secure any rights to any issued 
patents with claims that cover any of our proprietary product candidates and technologies. The patent prosecution 
process is expensive and time-consuming, and we may not be able to file and prosecute all necessary or desirable 
patent  applications  at  a  reasonable  cost  or  in  a  timely  manner.  It  is  also  possible  that  we  will  fail  to  identify 
patentable aspects of our research and development output before it is too late to obtain patent protection or before 
our competitors secure patents covering such discoveries. The patent process also is subject to numerous risks and 
uncertainties, and there can be no assurance that we will be successful in protecting our products by obtaining and 
defending patents.

Composition-of-matter patents relating to the active pharmaceutical ingredient (API) are generally considered to be 
the strongest form of intellectual property protection for pharmaceutical products. Such patents provide protection 
not limited to any one method of use. Method-of-use patents protect the use of a product for the specified method(s) 
and  do  not  prevent  a  competitor  from  making  and  marketing  a  product  that  is  identical  to  our  product  for  an 
indication that is outside the scope of the patented method. We rely on a combination of these and other types of 
patents to protect our product candidates, and there can be no assurance that our intellectual property will create and 
sustain the competitive position of our product candidates.

Biotechnology  and  pharmaceutical  product  patents  involve  highly  complex  legal  and  scientific  questions.  Any 
patent  applications  that  we  own  or  license  may  fail  to  result  in  issued  patents.  In  addition,  the  U.S.  Patent  and 
Trademark  Office  (the  USPTO)  and  patent  offices  in  other  jurisdictions  often  require  that  patent  applications 
concerning  pharmaceutical  and/or  biotechnology-related  inventions  are  limited  or  narrowed  substantially  to  cover 
only the specific innovations exemplified in the patent application, thereby limiting the scope of protection against 
competitive  challenges.  Thus,  even  if  we  or  our  licensors  are  able  to  obtain  patents,  the  patents  might  be 
substantially narrower than anticipated. 

28

If  patents  do  successfully  issue  from  our  applications,  third  parties  may  challenge  their  validity  or  enforceability, 
which may result in such patents being narrowed, invalidated, or held unenforceable. Even if our patents and patent 
applications are not challenged by third parties, those patents and patent applications may not prevent others from 
designing around our claims and may not otherwise adequately protect our product candidates. 

Patent and other intellectual property protection is crucial to the success of our business and prospects, and there is a 
substantial  risk  that  such  protections,  if  obtained,  will  prove  inadequate.  The  legal  systems  of  certain  countries, 
including China, do not always favor the enforcement of patents, trade secrets, and other intellectual property rights, 
particularly those relating to pharmaceutical and biotechnology products, which could make it difficult for us to stop 
infringement of our patents, misappropriation of our trade secrets, or marketing of competing products in violation 
of our proprietary rights. 

Beyond the protection afforded by patents, we seek to rely on trade secret protection and confidentiality agreements 
to  protect  proprietary  know-how,  information,  or  technology  that  is  not  covered  by  our  patents.  Although  our 
agreements  require  all  of  our  employees  to  assign  their  inventions  to  us,  and  we  require  all  of  our  employees, 
consultants,  advisors,  collaborators,  contractors  and  any  third  parties  who  have  access  to  our  trade  secrets, 
proprietary  know-how  and  other  confidential  information  and  technology  to  enter  into  appropriate  confidentiality 
agreements,  we  cannot  be  certain  that  our  trade  secrets,  proprietary  know-how  and  other  confidential  information 
and technology will not be subject to unauthorized disclosure or that our competitors will not otherwise gain access 
to or independently develop substantially equivalent trade secrets, proprietary know-how and other information and 
technology. If we are unable to prevent unauthorized disclosure of our intellectual property related to our product 
candidates and technology to third parties, we may not be able to establish or maintain a competitive advantage in 
our market, which could materially adversely affect our business and operations.

We  may  incur  substantial  costs  as  a  result  of  litigation  or  other  proceedings  relating  to  our  patents  and  other 
intellectual property rights.

We  may  in  the  future  be  involved  in  legal  or  administrative  proceedings  involving  our  intellectual  property, 
including infringement of our intellectual property by third parties. These lawsuits or proceedings likely would be 
expensive, consume time and resources and divert the attention of managerial and scientific personnel, even if we 
were successful in stopping the infringement of such patents. There is a risk that these proceedings will decide that 
such  patents  or  other  intellectual  property  rights  are  not  valid  and  that  we  do  not  have  the  right  to  stop  the  other 
party from using our inventions. There is also the risk that, even if the validity of such patents is upheld, the court or 
administrative  agency  will  refuse  to  stop  the  other  party  on  the  ground  that  such  other  party’s  activities  do  not 
infringe our rights to such patents. If we were not successful in defending our intellectual property, our competitors 
could develop and market products based on our discoveries, which may reduce demand for our products.

We may infringe the intellectual property rights of others, which may prevent or delay our product development 
efforts and stop us from commercializing or increase the costs of commercializing our product candidates.

Our success will depend in part on our ability to operate without infringing the proprietary rights of third parties. 
Our competitors may have filed, and may in the future file, patent applications covering products and technologies 
similar  to  ours.  Any  such  patent  application  may  have  priority  over  our  patent  applications,  which  could  further 
require us to obtain rights from third parties to issued patents covering such products and technologies. We cannot 
guarantee that the manufacture, use or marketing of any product candidates that we develop will not infringe third-
party patents.

If a patent infringement suit were brought against us, we may be forced to stop or delay developing, manufacturing, 
or selling potential products that are claimed to infringe a third party’s intellectual property, unless that third party 
grants us rights to use its intellectual property. In such cases, we may be required to obtain licenses to patents or 
proprietary rights of others in order to continue development, manufacture or sale of our products. If we are unable 
to  obtain  a  license  or  develop  or  obtain  non-infringing  technology,  or  if  we  fail  to  defend  an  infringement  action 
successfully,  or  if  we  are  found  to  have  infringed  a  valid  patent,  we  may  incur  substantial  costs  and  monetary 
damages,  encounter  significant  delays  in  bringing  our  product  candidates  to  market  and  be  precluded  from 
manufacturing or selling our product candidates, any of which could harm our business significantly.

29

The cost of maintaining our patent protection globally is high and requires continuous review and compliance. 
We may not be able to effectively maintain our intellectual property position throughout the major markets of the 
world.

The  USPTO  and  foreign  patent  authorities  require  maintenance  fees,  payments  and  continued  compliance  with  a 
number of procedural and documentary requirements. Noncompliance may result in abandonment or lapse of patents 
or patent applications and a partial or complete loss of patent rights in the relevant jurisdiction. Such a loss could 
reduce royalty payments for lack of patent coverage from our collaboration partners or may result in competition, 
either of which could have a material adverse effect on our business.

We  have  made,  and  will  continue  to  make,  certain  strategic  decisions  in  balancing  the  costs  and  the  potential 
protections afforded by the patent laws of certain countries. As a result, we may not be able to prevent third parties 
from practicing our inventions in all countries, or from selling or importing products made using our inventions in 
and into the United States or other countries. Third parties may use our technologies in territories in which we have 
not  obtained  patent  protection  to  develop  their  own  products  and  may  infringe  our  patents  in  territories  which 
provide inadequate enforcement mechanisms. Such third-party products may compete with our product candidates, 
and  our  patents  or  other  intellectual  property  rights  may  not  be  effective  or  sufficient  to  prevent  them  from 
competing. Such competition could materially and adversely affect our business and financial condition.

Intellectual property rights do not address all potential threats to any competitive advantage we may have.

The degree of future protection afforded by our intellectual property rights is uncertain because intellectual property 
rights  have  limitations,  and  intellectual  property  rights  may  not  adequately  protect  our  business  or  permit  us  to 
maintain our competitive advantage. The following examples are illustrative:

(cid:129) Others may be able to make compounds that are the same as, or similar to, our current or future product 
candidates but that are not covered by the claims of the patents that we own or have exclusively licensed.

(cid:129) We  or  any  of  our  licensors  or  strategic  partners  might  not  have  been  the  first  to  make  the  inventions 
covered by the issued patents or pending patent applications that we own or have exclusively licensed.

(cid:129) We  or  any  of  our  licensors  or  strategic  partners  might  not  have  been  the  first  to  file  patent  applications 

covering certain of our inventions.

(cid:129) Others may independently develop similar or alternative technologies or duplicate any of our technologies 

without infringing our intellectual property rights.

(cid:129)

The prosecution of our pending patent applications may not result in granted patents.

(cid:129) Granted  patents  that  we  own  or  have  exclusively  licensed  may  not  provide  us  with  any  competitive 
advantages, or may be held invalid or unenforceable, as a result of legal challenges by our competitors.

(cid:129)

Patent protection on our product candidates may expire before we are able to develop and commercialize 
the product, or before we are able to recover our investment in the product.

(cid:129) Our competitors might conduct research and development activities in the United States and other countries 
that  provide  a  safe  harbor  from  patent  infringement  claims  for  such  activities,  as  well  as  in  countries  in 
which  we  do  not  have  patent  rights  and  may  then  use  the  information  learned  from  such  activities  to 
develop competitive products for sale in markets where we intend to market our product candidates.

The  existence  of  counterfeit  pharmaceutical  products  in  pharmaceutical  markets  may  damage  our  brand  and 
reputation and have a material adverse effect on our business, operations and prospects.

Counterfeit products, including counterfeit pharmaceutical products, are a significant problem, particularly in China. 
Counterfeit  pharmaceuticals  are  products  sold  or  used  for  research  under  the  same  or  similar  names,  or  similar 
mechanism of action or product class, but which are sold without proper licenses or approvals. The proliferation of 
counterfeit pharmaceuticals has grown in recent years and may continue to grow in the future. Such products may be 

30

used for indications or purposes that are not recommended or approved or for which there is no data or inadequate 
data with regard to safety or efficacy. Such products divert sales from genuine products, often are of lower cost and 
lower  quality  (having  different  ingredients  or  formulations,  for  example),  and  have  the  potential  to  damage  the 
reputation for quality and effectiveness of the genuine product. 

If  counterfeit  pharmaceuticals  illegally  sold  or  used  for  research  result  in  adverse  events  or  side  effects  to 
consumers, we may be associated with any negative publicity resulting from such incidents. In addition, counterfeit 
products could be used in nonclinical studies or clinical studies or could otherwise produce undesirable side effects 
or adverse events that may be attributed to our products as well, which could cause us or regulatory authorities to 
interrupt, delay or halt clinical studies and could result in the delay or denial of regulatory approval by the FDA or 
other regulatory authorities and potential product liability claims.  

In China, although the government has recently increased the lower and upper limits on penalties on producers of 
counterfeit and substandard pharmaceuticals, these penalties have not eliminated counterfeit pharmaceuticals. As a 
result,  we  may  not  be  able  to  prevent  third  parties  from  selling  or  purporting  to  sell  our  products  in  China.  The 
existence  of,  and  any  increase  in,  the  sales  and  production  of  counterfeit  pharmaceuticals,  or  the  technological 
capabilities  of  counterfeiters,  could  negatively  impact  our  revenues,  brand  reputation,  business  and  results  of 
operations.

Risks Related to Our Common Stock

Our amended and restated bylaws provide that the Court of Chancery of the State of Delaware will be the sole 
and exclusive forum for certain types of actions and proceedings that may be initiated by our stockholders, which 
could limit our stockholders’ ability to bring a claim in a judicial forum they find favorable for disputes with us 
or our directors, officers or other employees.

Our amended and restated bylaws provide that, with certain limited exceptions, unless we consent to the selection of 
an  alternative  forum,  the  Court  of  Chancery  of  the  State  of  Delaware  (the  Court  of  Chancery)  is  the  sole  and 
exclusive forum for (1) any derivative action or proceeding brought on our behalf; (2) any action asserting a claim of 
breach of fiduciary duty owed by any of our current or former directors, officers or other employees to us or to our 
stockholders;  (3)  any  action  asserting  a  claim  arising  pursuant  to  the  Delaware  General  Corporation  Law,  or  our 
certificate  of  incorporation  or  bylaws  (as  each  may  be  amended  from  time  to  time);  or  (4)  any  action  asserting  a 
claim governed by the internal affairs doctrine. Alternatively, if such court does not have jurisdiction, the Superior 
Court of Delaware, or, if such other court does not have jurisdiction, the United States District Court for the District 
of Delaware, will be the sole and exclusive forum for such actions and proceedings. The choice of forum provision 
may limit a stockholder’s ability to bring a claim in a judicial forum that it finds favorable for disputes with us or 
our  directors,  officers,  or  other  employees,  which  may  discourage  such  lawsuits  against  us  and  our  directors, 
officers, and other employees. Alternatively, if a court were to find the choice of forum provision contained in our 
amended  and  restated  bylaws  to  be  inapplicable  or  unenforceable  in  an  action,  we  may  incur  additional  costs 
associated  with  resolving  such  action  in  other  jurisdictions,  which  could  have  a  material  adverse  impact  on  our 
business. The choice of forum provision in our amended and restated bylaws will not preclude or contract the scope 
of  exclusive  federal  or  concurrent  jurisdiction  for  actions  brought  under  the  federal  securities  laws,  including  the 
Exchange Act or the Securities Act, or the respective rules and regulations promulgated thereunder.

The price of our common stock might fluctuate significantly, and you could lose all or part of your investment.

The  price  of  our  common  stock  fluctuates  widely.  Continued  volatility  in  the  market  price  of  our  common  stock 
might prevent a stockholder from being able to sell shares of our common stock at or above the price paid for such 
shares. The trading price of our common stock may continue to be volatile and subject to wide price fluctuations in 
response to various factors, many of which are beyond our control, such as the progress, results and timing of our 
clinical studies and nonclinical studies and other studies involving our product candidates, the success or failure of 
our  product  candidates,  the  receipt  or  loss  of  required  regulatory  approvals  for  our  product  candidates,  the 
availability of capital or the other risks discussed in this “Risk Factors” section. 

31

Item 1B. Unresolved Staff Comments

None.

Item 2. Properties

We  lease  office  space  for  corporate  and  administrative  functions  and  laboratory  space  in  South  San  Francisco, 
California under a sub-sublease that expires in December 2023. Prior to moving into the South San Francisco office 
and laboratory space in February 2019, we leased office and laboratory space in San Francisco, California under a 
sublease  that  expired  on  February  28,  2019.  The  leased  location  in  San  Francisco,  California  supported  both  the 
HBV and Microbiome programs. We also conducted research, development and small-scale manufacturing activities 
for  the  Microbiome  program  at  office  and  laboratory  space  in  Groton,  Connecticut  under  a  lease  that  expires  in 
March 2021. We also lease office space that was used for administrative functions in Carmel, Indiana under a lease 
agreement that expires in August 2023. In February 2021, we subleased substantially all of the office space under 
this lease.

We believe these leased facilities are adequate for our current needs and that additional space will be available in the 
future on commercially reasonable terms as needed.

Item 3. Legal Proceedings

We are not a party to any material legal proceedings at this time. From time to time, we may be subject to various 
legal  proceedings  and  claims  that  arise  in  the  ordinary  course  of  our  business  activities.  Although  the  results  of 
litigation and claims cannot be predicted with certainty, we do not believe we are party to any claim or litigation the 
outcome of which, if determined adversely to us, would individually or in the aggregate be reasonably expected to 
have a material adverse effect on our business. Regardless of the outcome, litigation can have an adverse effect on 
us because of defense and settlement costs, diversion of management resources and other factors.

Item 4. Mine Safety Disclosures

Not applicable.

32

PART II

Item  5.  Market  for  Registrant’s  Common  Equity,  Related  Stockholder  Matters  and  Issuer  Purchases  of 
Equity Securities

Market Information for Common Stock

Our common stock is traded under the symbol “ASMB” and is quoted on The Nasdaq Global Select Market.

Holders of Record

As of February 22, 2021, there were 67 stockholders of record, which excludes stockholders whose shares were held 
in nominee or street name by brokers.

Dividend Policy

We have never declared or paid any dividends and do not anticipate paying any dividends on our common stock in 
the foreseeable future.

Comparative Stock Performance Graph

The information included under the heading “Comparative Stock Performance Graph” in this Item 5 of Part II of this 
Form 10-K shall not be deemed to be “soliciting material” or subject to Regulation 14A or 14C, shall not be deemed 
“filed”  for  purposes  of  Section  18  of  the  Exchange  Act,  or  otherwise  subject  to  the  liabilities  of  that  section,  nor 
shall it be deemed incorporated by reference in any filing under the Securities Act or the Exchange Act.

Set  forth  below  is  a  graph  comparing  the  total  cumulative  returns  of  our  common  stock,  the  Nasdaq  Composite 
Index and the Nasdaq Biotechnology Index. The graph assumes $100 was invested in our common stock and each of 
the indices on December 31, 2015 and that all dividends, if any, are reinvested.  

* $100 invested on December 31, 2015 in stock or index, including reinvestment of dividends.

Assembly Biosciences, Inc. .........................   
Nasdaq Composite .......................................   
Nasdaq Biotechnology.................................   

 12/31/2015  12/31/2016  12/31/2017  12/31/2018  12/31/2019  12/31/2020 
80.56 
257.38 
134.42  

272.44   
179.19   
106.95   

100.00   
100.00   
100.00   

161.78   
107.50   
78.32   

602.53   
137.86   
94.81   

301.20   
132.51   
85.97   

33

 
 
Securities Authorized for Issuance Under Equity Compensation Plans

The  following  table  sets  forth  the  indicated  information  as  of  December  31,  2020  with  respect  to  our  equity 
compensation plans.

Number of
securities
to be issued
upon
exercise of
outstanding
options,
warrants
and rights
(a)

Weighted
average
exercise
price of
outstanding
options,
warrants
and
rights(1)
(b)

Number of
securities
remaining
available for
future
issuance
under equity
compensation
plans
(excluding
securities
reflected in
column (a))
(c)
2,355,332  (3)

Plan Category
Equity compensation plans approved by securityholders .............     5,515,752  (2)   $

14.39     

Equity compensation plans not approved by securityholders .......     2,067,708  (4)   $
Total ..............................................................................................     7,583,460   

18.86     

24,020  (5)

2,379,352   

(1) The weighted average exercise price is calculated solely based on the exercise prices of the outstanding stock 
options and does not reflect the shares that will be issued upon the vesting of outstanding awards of restricted 
stock units (RSUs), which have no exercise price.

(2) This  number  includes  the  following:  363,161  shares  subject  to  stock  options  granted  under  the  2010  Equity 
Incentive  Plan  (2010  Plan);  2,453,335  shares  subject  to  outstanding  awards  granted  under  the  Assembly 
Biosciences,  Inc.  Amended  and  Restated  2014  Stock  Incentive  Plan  (2014  Plan),  of  which  2,296,823  were 
subject to outstanding stock options and 156,512 were subject to outstanding RSUs; 2,269,503 shares subject to 
outstanding awards granted under the Assembly Biosciences, Inc. 2018 Stock Incentive Plan, as amended (2018 
Plan), of which 1,608,912 were subject to outstanding stock options, 624,106 were subject to outstanding RSUs 
and 36,485 are underlying stock appreciation rights (which are not included in column (a) but are reflected in 
column  (c));  and  466,238  options  assumed  by  us  in  connection  with  our  merger  with  Assembly 
Pharmaceuticals.  This  number  excludes  purchase  rights  currently  accruing  under  the  Assembly  Biosciences, 
Inc. 2018 Employee Stock Purchase Plan (2018 ESPP).

(3) This  number  includes:  no  shares  under  the  2010  Plan,  which  has  been  frozen;  85,968  shares  available  for 
issuance under the 2014 Plan; 2,037,029 shares available for issuance under the 2018 Plan and; 232,335 shares 
reserved for issuance under the 2018 ESPP. As of February 22, 2021, assuming each participant purchases the 
maximum number of shares in the current offering period, no more than 51,000 shares are subject to purchase in 
the current offering, which ends on May 14, 2021.

(4) This number includes 791,028 shares subject to outstanding awards granted under the 2017 Inducement Award 
Plan  (2017  Inducement  Plan),  of  which  779,778  were  subject  to  outstanding  stock  options  and  11,250  were 
subject to outstanding RSUs; 500,000 shares subject to stock options granted under the 2019 Inducement Award 
Plan (2019 Inducement Plan).

(5) This number includes: 700 shares available for issuance under the 2017 Inducement Plan and no shares under 

the 2019 Inducement Plan.

34

 
   
 
   
 
 
 
   
    
   
      
    
     
     
Our  stockholder-approved  equity  compensation  plans  consist  of  the  2018  Plan,  2014  Plan,  the  2010  Plan,  stock 
options assumed in our merger with Assembly Pharmaceuticals and the 2018 ESPP. Effective on June 2, 2016, the 
2010 Plan was frozen, and no further grants will be made under the 2010 Plan. Shares that are forfeited under the 
2010 Plan on or after June 2, 2016 will become available for issuance under the 2014 Plan. An “Award” under the 
2018  Plan,  2014  Plan  or  2010  Plan  is  any  right  to  receive  our  common  stock  consisting  of  non-statutory  stock 
options, incentive stock options, stock appreciation rights, RSUs, or any other stock award.

In May 2018, our stockholders approved the 2018 ESPP. The 2018 ESPP provides for the purchase by employees of 
up to an aggregate of 400,000 shares of the Company’s common stock. Eligible employees can purchase shares of 
our common stock at the end of a predetermined offering period at 85% of the lower of the fair market value at the 
beginning or end of the offering period.

Our outstanding equity compensation arrangements that have not been approved by our stockholders consist of the 
2017 Inducement Plan, the 2019 Inducement Plan and warrants to purchase shares of our common stock issued to 
one consultant. In April 2017, our board of directors adopted the 2017 Inducement Plan and reserved 800,000 shares 
of our common stock for issuance under the Inducement Plan, and in August 2019, our board of directors adopted 
the  2019  Inducement  Plan  and  reserved  500,000  shares  of  our  common  stock  for  issuance  under  the  2019 
Inducement Award Plan. The only persons eligible to receive grants of awards under the either the 2017 Inducement 
Plan  or  the  2019  Inducement  Plan  are  individuals  who  satisfy  the  standards  for  inducement  grants  under  Nasdaq 
Marketplace  Rule  5635(c)(4)  and  the  related  guidance  under  Nasdaq  IM  5635-1-that  is,  generally,  a  person  not 
previously an employee or director of ours, or following a bona fide period of non-employment, as an inducement 
material to the individual's entering into employment with us. An “Award” is any right to receive our common stock 
pursuant to the Inducement Plan, consisting of nonstatutory stock options, stock appreciation rights, restricted stock 
awards, RSUs, or any other stock award.

Recent Sales of Unregistered Securities

There were no unregistered sales of equity securities in 2020.

Purchases of Equity Securities by the Issuer and Affiliated Purchasers

We  did  not  purchase  any  of  our  registered  equity  securities  during  the  period  covered  by  this  Annual  Report  on 
Form 10-K.

35

Item 6. Selected Financial Data

The  following  selected  balance  sheet  data  for  the  years  ended  December  31,  2020  and  2019  and  the  statement  of 
operations data for the years ended December 31, 2020, 2019 and 2018 should be read in conjunction with Part II, 
Item  7  “Management’s  Discussion  and  Analysis  of  Financial  Condition  and  Results  of  Operations”  and  in 
conjunction  with  the  consolidated  financial  statements,  related  notes  and  other  financial  information  included 
elsewhere  in  this  Annual  Report.  The  selected  consolidated  results  of  operation  data  for  the  years  ended 
December 31,  2017  and  2016  and  the  balance  sheet  data  for  the  years  ended  December  31,  2018,  2017  and  2016 
have been derived from audited consolidated financial statements not included herein. Our historical results are not 
necessarily indicative of the results to be expected in the future.   

($ in thousands except for per share amounts)
Balance Sheet Data:
Total assets ................................................................  $ 283,254    $ 339,907    $ 268,045    $ 169,303    $
Total stockholders’ equity .........................................    240,578      273,217      210,653      113,120     

2020

2019

2017

December 31,
2018

2016

98,119 
79,878 

Statement of Operations Data:
Collaboration revenue ...............................................  $ 79,105    $ 15,963    $ 14,804    $
Operating expenses....................................................    143,881      118,676      107,539     
(92,735)    
Loss from operations .................................................   
3,083     
Interest and other income, net ...................................   
(89,652)    
Loss before income taxes ..........................................   

(64,776)     (102,713)    
4,295     
(98,408)    

2,624     
(62,152)    

9,019    $
61,246     
(52,227)    
368     
(51,859)    

— 
45,278 
(45,278)
399 
(44,879)

Income tax (expenses) benefit ...................................   
618 
Net loss ......................................................................  $ (62,152)   $ (97,634)   $ (90,751)   $ (42,809)   $ (44,261)
Unrealized gain/loss on marketable securities, net
of tax..........................................................................   
Basic and dilutive loss per share ...............................  $

45     
(3.98)   $

209     
(2.41)   $

146     
(3.72)   $

(69)    
(1.75)   $

221 
(2.57)

(1,099)    

9,050     

774     

—     

The increase in total assets from $98.1 million as of December 31, 2016 to $169.3 million as of December 31, 2017 
was primarily due to a capital raise of $64.8 million in net proceeds in November 2017 and receipt from Allergan of 
an  upfront  payment  of  $50.0  million  in  February  2017.  The  increase  in  total  assets  from  $169.3  million  as  of 
December 31, 2017 to $268.0 million as of December 31, 2018 was primarily due to a capital raise of $155.4 million 
in  net  proceeds  to  us  in  July  2018.  The  increase  in  total  assets  from  $268.0  million  as  of  December  31,  2018  to 
$339.9  million  as  of  December  31,  2019  is  primarily  due  to  a  capital  raise  of  $134.7  million  in  net  proceeds  in 
December 2019. The decrease in total assets from $339.9 million as of December 31, 2019 to $283.3 million as of 
December 31, 2020 is primarily due to cash used in operations. Our operating expenses have increased year over 
year primarily due to increases in research and development activities and an increase in our total headcount. See 
Part  II,  Item  7  “Management’s  Discussion  and  Analysis  of  Financial  Condition  and  Results  of  Operations”  for  a 
discussion on results of operations and financing activities since 2018.

36

  
 
 
 
   
   
   
   
 
   
      
      
      
      
  
 
   
      
      
      
      
  
   
      
      
      
      
  
 
   
      
      
      
      
  
Item 7. Management’s Discussion and Analysis of Financial Condition and Results of Operation

The  following  discussion  and  analysis  of  our  financial  condition  and  results  of  operations  should  be  read  in 
conjunction with “Selected Financial Data”, our consolidated financial statements and the related notes thereto and 
other  financial  information  appearing  elsewhere  in  this  Annual  Report  on  Form  10-K.  The  following  discussion 
contains forward-looking statements that involve risks and uncertainties. Our actual results could differ materially 
from those expressed or implied in any forward-looking statements as a result of various factors, including those set 
forth in this Form 10-K under “Item 1A. Risk Factors.”

Overview

We  are  a  clinical-stage  biotechnology  company  advancing  a  novel  class  of  oral  therapeutic  candidates  for  the 
treatment  of  chronic  hepatitis  B  virus  (HBV)  infection.  According  to  the  World  Health  Organization  (WHO), 
approximately  270  million  people  worldwide  are  chronically  infected  with  HBV.  Our  research  and  development 
programs  are  pursuing  multiple  drug  candidates  designed  to  inhibit  the  HBV  replication  cycle  and  block  the 
generation  of  covalently  closed  circular  DNA  (cccDNA),  with  the  aim  of  discovering  and  developing  finite  and 
curative  therapies  for  patients  with  HBV.  We  have  discovered  several  novel  core  inhibitors,  which  are  small 
molecules that directly target and allosterically modulate the HBV core (HBc) protein in a way that affects assembly 
and stability of HBV nucleocapsids.

The  ongoing  COVID-19  pandemic  has  affected  certain  aspects  of  our  business.  As  further  detailed  below,  those 
effects  have  been  primarily  limited  to  where  and  how  our  employees  work  in  our  labs  and  offices.  To  date,  our 
current  and  future  planned  clinical  trials  and  pre-clinical  studies  have  not  been  subject  to  significant  impact  as  a 
result of the COVID-19 pandemic.

As previously announced, in January 2021, we wound down our Microbiome program to prioritize and focus our 
resources on discovering and developing finite and curative therapies for HBV. Our Microbiome program had been 
developing a novel class of oral live microbial biotherapeutics candidates designed to treat disorders associated with 
the microbiome.

Our Primary Focus: Targeting HBV Core Protein to Achieve a Cure 

HBV  is  a  DNA  virus  that  infects  hepatocytes  and  establishes  a  reservoir  of  cccDNA,  a  unique  DNA  moiety  that 
resides  in  the  cell  nucleus  of  HBV-infected  hepatocytes  and  is  associated  with  viral  persistence  and  chronic 
infection.  No  currently  approved  oral  therapies  target  cccDNA  activity  directly,  which  makes  molecules  that  can 
modulate  cccDNA  generation  or  disrupt  its  function  highly  sought  in  the  HBV  field.  As  a  result,  most  of  our 
research and development efforts to date have focused on discovering and developing compounds targeting the core 
protein,  a  highly  conserved  viral  structural  protein  that  has  no  human  homologue  and  is  involved  in  numerous 
aspects of the HBV replication cycle, including the generation of HBV cccDNA. Through our research efforts, we 
have  discovered  several  chemically  distinct  series  of  small  molecule  core  inhibitors  that  directly  target  and 
allosterically inhibit core protein functions.

Vebicorvir

Vebicorvir (VBR), our lead core inhibitor product candidate, is licensed from Indiana University. The conduct of the 
Phase 2 studies, Study 201 and 202 and our open-label extension study, Study 211, are all complete. We presented 
interim  updates  on  our  clinical  studies  at  a  variety  of  conferences,  including  at  the  European  Association  for  the 
Study of the Liver’s (EASL) Digital International Liver CongressTM in August 2020 and the American Association 
for the Study of Liver Diseases (AASLD) Annual Meeting in November 2020.

Our  most  recently  completed  study  for  VBR,  Study  211,  involved  transitioning  patients  who  met  the  requisite 
stopping criteria, as determined with our lead investigators and the U.S. Food and Drug Administration (FDA), off 
of therapy to test for sustained virologic response (SVR). SVR refers to sustained viral suppression (more than six 
months) of HBV DNA below the lower limit of quantification (LLOQ) and would be consistent with a successful 
finite treatment for HBV. In November 2020, it became clear that patients who stopped therapy in Study 211 had not 
achieved meaningful SVR rates as 39 of 41 patients relapsed, meaning they had detectable HBV. We continue to 
collect  and  analyze  Study  211  data  and  intend  to  submit  more  detailed  findings  to  a  future  medical  meeting; 
however, it is clear that combination therapy of VBR plus nucelos(t)ide analog reverse transcriptase inhibitors (NrtI) 
alone is not sufficient to cure HBV. Based on these results, we terminated Study 211 prior to its completion.

Based  on  discussions  with  leading  viral  hepatitis  experts,  global  regulatory  discussions  and  feedback,  and,  with 
respect to the China territory, discussions and agreement with our collaboration partner, BeiGene, Ltd. (BeiGene), 

37

we  recently  decided  to  not  move  forward  with  the  global  registrational  studies  for  VBR  as  a  chronic  suppressive 
treatment (CST) with NrtI. The decision was made to focus on the greatest unmet medical need of patients, which 
lies  predominantly  in  cure,  rather  than  CST.  As  a  result,  we  also  expect  to  terminate  Study  205,  as  we  focus  our 
efforts with VBR moving forward in combination with NrtI and additional mechanisms targeting finite and curative 
combination therapy.

ABI-H2158

Our  second-generation  core  inhibitor  product  candidate,  ABI-H2158  (2158),  was  internally  discovered  and 
developed and is chemically distinct from VBR.

We  reported  the  final  data  from  dose-ranging  cohorts  of  the  Phase  1b  portion  of  the  Phase  1a/1b  dose-ranging 
clinical study at EASL in August 2020. Based on data from the Phase 1b dose-ranging study, we initiated a Phase 2 
clinical study in June 2020 using a 300 mg daily dose of 2158. This study is being conducted in approximately ten 
countries in Asia, North America and Europe. We expect interim data from this study in the second half of 2021. 
While we will continue to monitor the situation closely, at this time, we do not expect our timelines for this study to 
be significantly impacted by the COVID-19 pandemic. 

ABI-H3733

Our  third  core  inhibitor  product  candidate,  ABI-H3733  (3733),  has  completed  Investigational  New  Drug  (IND) 
enabling studies. 3733 has a novel chemical scaffold separate from both VBR and 2158. We presented a preclinical 
profile of this candidate in the first quarter of 2019.

In  the  first  quarter  of  2020,  we  initiated  a  Phase  1a  clinical  study  to  evaluate  safety,  tolerability  and 
pharmacokinetics  (PK)  following  single  ascending  dose  and  multiple  ascending  dose  administration  of  3733  in 
healthy subjects in New Zealand. Conduct for the study was completed in the fourth quarter of 2020 and preliminary 
data indicate that 3733 was generally well-tolerated and had favorable PK.

Additional Product Candidates

In  addition  to  our  three  clinical-stage  product  candidates,  our  research  discovery  team  is  actively  focused  on 
identifying and selecting a fourth-generation core inhibitor candidate, which we anticipate in the first half of 2021.

Multi-Drug Combination Studies

We believe that core inhibitors and NrtI will be central to finite and curative therapies for chronic HBV infection. 
Therefore, as we continue to develop and advance our current and future core inhibitors through clinical studies, we 
plan  to  conduct  multi-drug  combination  studies  in  parallel  that  add  additional  drugs  (or  compounds)  with  non-
overlapping  mechanisms  of  action  to  the  core  inhibitor  +  NrtI  antiviral  backbone.  Specifically,  we  plan  on  only 
incorporating our current and future core inhibitors that have demonstrated they are well-tolerated and effective in 
clinical  studies  in  dual  combination  with  NrtI.  As  the  300  mg  daily  dose  of  VBR  has  been  observed  to  be  well-
tolerated in all studies conducted to date, with no serious adverse effects or dose-limiting toxicities identified and no 
pattern  of  treatment-emergent  clinical  or  laboratory  abnormalities  observed  and  has  progressed  beyond  dual 
combination studies, we currently have two triple combination studies planned to study VBR in combination with 
NrtI and a third mechanism of action.

Beyond Core Inhibitors

In addition to the development and advancement of our core inhibitor portfolio and our current and future multi-drug 
combination studies, our research and development team is working on discovering and developing a potent fourth-
generation core inhibitor, cccDNA disruptors and small molecules targeting novel undisclosed targets to add to the 
core inhibitor + NrtI antiviral backbone to achieve cure.

Operations

We  currently  have  corporate  and  administrative  offices  and  research  laboratory  space  in  South  San  Francisco, 
California, Groton, Connecticut and a small office in China.

Since our inception, we have had no revenue from product sales and have funded our operations principally through 
debt  financings  prior  to  our  initial  public  offering  in  2010  and  through  equity  financings  and  collaborations  since 
then.  Our  operations  to  date  have  been  primarily  limited  to  organizing  and  staffing  our  company,  licensing  our 
product  candidates,  discovering  and  developing  our  product  candidates,  maintaining  and  improving  our  patent 

38

portfolio  and  raising  capital.  We  have  generated  significant  losses  to  date,  and  we  expect  to  continue  to  generate 
losses as we continue to develop our product candidates. As of December 31, 2020, we had an accumulated deficit 
of $501.6 million. Because we do not generate revenue from any of our product candidates, our losses will continue 
as we further develop and seek regulatory approval for, and commercialize, our product candidates. As a result, our 
operating  losses  are  likely  to  be  substantial  over  the  next  several  years  as  we  continue  the  development  of  our 
product candidates and thereafter if none are approved or successfully launched. We are unable to predict the extent 
of any future losses or when we will become profitable, if at all.

Financial Operations Overview

Research and Development Expense

Research  and  development  expenses  consist  primarily  of  costs  incurred  for  our  research  activities,  including  our 
drug  discovery  efforts,  target  validation,  lead  optimization  and  the  development  of  our  product  candidates,  which 
include:

(cid:129)

(cid:129)

(cid:129)

(cid:129)

(cid:129)

employee-related expenses including salaries, benefits, and stock-based compensation expense;

expenses  incurred  under  agreements  with  third  parties,  including  contract  research  organizations  (CROs) 
that  conduct  research  and  development,  nonclinical  and  clinical  activities  on  our  behalf  and  the  cost  of 
consultants, and contract manufacturing organizations (CMOs) that manufacture all of our drug substance 
and the drug product used in our HBV program;

the cost of lab supplies and acquiring, developing, and manufacturing nonclinical and, in the case of our 
Microbiome program, early stage clinical study materials;

fees related to our license agreements; and

facilities,  depreciation,  and  other  expenses,  which  include  direct  and  allocated  expenses  for  rent  and 
maintenance of facilities, insurance, and other operating costs.

Research and development costs are expensed as incurred. Nonrefundable advance payments for goods or services 
to  be  received  in  the  future  for  use  in  research  and  development  activities  are  deferred  and  capitalized.  The 
capitalized amounts are expensed as the related goods are delivered or the services are rendered.

We  use  our  employee  and  infrastructure  resources  across  multiple  research  and  development  programs,  and  we 
allocate  internal  employee-related  and  infrastructure  costs,  as  well  as  certain  third-party  costs,  to  each  of  our 
programs based on the personnel resources allocated to such program. Our research and development expenses, by 
major program, are outlined in the table below (in thousands):

HBV(1)..........................................................................  $
Microbiome(2) ..............................................................   

2020
71,957   $
34,866    
Total .......................................................................  $ 106,823   $

Year Ended December 31,
2019
57,534   $
28,223    
85,757   $

2018
49,416 
23,325 
72,741  

(1) Expenses  presented  for  HBV  include  reimbursement  of  expenses  of  $0.2  million  under  the  Clinical  Trial 
Collaboration Agreement (Arbutus Agreement) with Arbutus Biopharma Corporation (Arbutus), as discussed in 
Note 9 to the Consolidated Financial Statements.

(2) Expenses  presented  for  Microbiome  do  not  reflect  reimbursement  of  expenses  under  the  Research, 
Development,  Collaboration  and  License  Agreement  (Allergan  Agreement)  with  Allergan  Pharmaceuticals 
International Limited (Allergan), as discussed in Note 9 to the Consolidated Financial Statements.

39

 
 
 
 
 
  
   
 
The successful discovery and development of our product candidates is highly uncertain. As such, at this time, we 
cannot reasonably estimate, or know the nature, timing and estimated costs, of the efforts that will be necessary to 
complete the remainder of their development. We are also unable to predict when, if ever, material net cash inflows 
will  commence  from  our  product  candidates.  This  is  due  to  the  numerous  risks  and  uncertainties  associated  with 
developing medicines, including the uncertainty of:

(cid:129)

(cid:129)

(cid:129)

the  timing,  progress  and  success  of  our  clinical  trials  and  research  discovery  team  in  identifying  new 
product candidates;

establishing  an  appropriate  safety  profile  with  IND-enabling  toxicology  studies  sufficient  to  advance 
additional product candidates into clinical development;

successful enrollment in, and completion of, clinical studies;

(cid:129) making arrangements with third-party manufacturers; and

(cid:129)

obtaining  and  maintaining  patent  and  trade  secret  protection  and  regulatory  exclusivity  for  our  product 
candidates.

A change in the outcome of any of these variables or variables discussed in “Item 1A. Risk Factors” with respect to 
the development of any of our product candidates would significantly change the costs and timing associated with 
the development of that product candidate.

Research and development activities are central to our business model. Product candidates in later stages of clinical 
development generally have higher development costs than those in earlier stages of clinical development, primarily 
due to the increased size and duration of later-stage clinical studies. However, we do not believe that it is possible at 
this  time  to  accurately  project  total  program-specific  expenses  through  commercialization.  There  are  numerous 
factors  associated  with  the  successful  commercialization  of  any  of  our  product  candidates,  including  future  trial 
design and various regulatory requirements, many of which cannot be determined with accuracy at this time based 
on our stage of development. Additionally, future commercial and regulatory factors beyond our control will impact 
our clinical development programs and plans.

General and administrative expenses

General  and  administrative  expenses  consist  primarily  of  salaries  and  other  related  costs,  including  stock-based 
compensation,  for  personnel  in  executive,  finance,  accounting,  business  development,  legal  and  human  resources 
functions.  Other  significant  costs  include  facility  costs  not  otherwise  included  in  research  and  development 
expenses, insurance costs, legal fees relating to patents and corporate matters and fees for accounting and consulting 
services.

We anticipate that our general and administrative expenses will increase in the future to support continued research 
and development activities, potential commercialization of our product candidates and costs of operating as a public 
company. These increases will likely include increased costs related to the hiring of additional personnel and fees to 
outside  consultants,  lawyers  and  accountants,  among  other  expenses.  Additionally,  we  anticipate  increased  costs 
associated  with  being  a  public  company,  including  expenses  related  to  services  associated  with  maintaining 
compliance  with  exchange  listing  and  U.S.  Securities  and  Exchange  Commission  (SEC)  requirements,  insurance, 
and investor relations costs.

Interest income

Interest income consists of interest earned on our cash and cash equivalents and available-for-sale securities.

Critical Accounting Policies and Significant Judgments and Estimates

Our  management’s  discussion  and  analysis  of  our  financial  condition  and  results  of  operations  is  based  on  our 
consolidated  financial  statements,  which  we  have  prepared  in  accordance  with  accounting  principles  generally 
accepted  in  the  United  States.  The  preparation  of  these  consolidated  financial  statements  requires  us  to  make 
estimates and assumptions that affect the reported amounts of assets and liabilities and the disclosure of contingent 
assets and liabilities at the date of the financial statements, as well as the reported amounts of revenues and expenses 
during the reporting periods. We evaluate our estimates and judgments, including those described in greater detail 

40

below,  on  an  ongoing  basis.  We  base  our  estimates  on  historical  experience  and  on  various  other  factors  that  we 
believe are reasonable under the circumstances, the results of which form the basis for making judgments about the 
carrying  value  of  assets  and  liabilities  that  are  not  readily  apparent  from  other  sources.  Actual  results  may  differ 
from these estimates under different assumptions or conditions.

While  our  significant  accounting  policies  are  described  in  more  detail  in  the  notes  to  our  consolidated  financial 
statements  included  elsewhere  in  this  Annual  Report  on  Form  10-K,  we  believe  that  the  following  accounting 
policies are the most critical to aid you in fully understanding and evaluating our financial condition and results of 
operations.

Revenue Recognition and Accounts Receivable from Collaboration

We  analyze  our  collaboration  arrangements  to  assess  whether  such  arrangements,  or  transactions  between 
arrangement participants, involve joint operating activities performed by parties that are both active participants in 
the activities and exposed to significant risks and rewards dependent on the commercial success of such activities or 
are more akin to a vendor-customer relationship. In making this evaluation, we consider whether the activities of the 
collaboration  are  considered  to  be  distinct  and  deemed  to  be  within  the  scope  of  the  collaborative  arrangement 
accounting standard and those that are more reflective of a vendor-customer relationship and, therefore, within the 
scope of the revenue with contracts with customers accounting standard. This assessment is performed throughout 
the life of the arrangement based on changes in the responsibilities of all parties in the arrangement.

For elements of collaboration arrangements that are not accounted for pursuant to the revenue from contracts with 
customers accounting standard, an appropriate recognition method is determined and applied consistently, generally 
by analogy to the revenue from contracts with customers accounting standard. Amounts related to transactions with 
a counterparty in a collaborative arrangement that is not a customer are presented as collaboration revenue and on a 
separate line item from revenue recognized from contracts with customers, if any, in our consolidated statements of 
operations and comprehensive loss.

Under  certain  collaborative  arrangements,  we  are  reimbursed  for  a  portion  of  our  research  and  development 
expenses  or  participate  in  the  cost-sharing  of  such  research  and  development  expenses.  Such  reimbursements  and 
cost-sharing  arrangements  are  reflected  as  a  reduction  of  research  and  development  expense  our  consolidated 
statements  of  operations  and  comprehensive  loss,  as  we  do  not  consider  performing  these  activities  for 
reimbursement to be a part of our ongoing major or central operations.

For  arrangements  or  transactions  between  arrangement  participants  determined  to  be  within  the  scope  of  the 
contracts with customers accounting standard, we evaluate the term of the arrangement and recognize revenue when 
the customer obtains control of promised goods or services in a contract for an amount that reflects the consideration 
we expect to receive in exchange for those goods or services. For contracts with customers, we apply the following 
five-step  model  in  order  to  determine  this  amount:  (1)  identification  of  the  promised  goods  or  services  in  the 
contract;  (2)  determination  of  whether  the  promised  goods  or  services  are  performance  obligations,  including 
whether  they  are  distinct  in  the  context  of  the  contract;  (3)  measurement  of  the  transaction  price,  including  the 
constraint on variable consideration; (4) allocation of the transaction price to the performance obligations; and (5) 
recognition of revenue when (or as) we satisfy each performance obligation. 

We have provided standard indemnification and protection of licensed intellectual property for our customers. These 
provisions  are  part  of  assurance  that  the  licenses  meet  the  agreements,  representations  and  are  not  obligations  to 
provide goods or services.

We only apply the five-step model to contracts when it is probable we will collect the consideration we are entitled 
to  in  exchange  for  the  goods  or  services  it  transfers  to  the  customer.  As  part  of  the  accounting  for  contracts  with 
customers,  we  must  develop  assumptions  that  require  judgment  to  determine  the  standalone  selling  price  of  each 
performance obligation identified in the contract. We then allocate the total transaction price to each performance 
obligation  based  on  the  estimated  standalone  selling  prices  of  each  performance  obligation.  We  recognize  the 
amount  of  the  transaction  price  that  is  allocated  to  the  respective  performance  obligation  when  the  performance 
obligation is satisfied or as it is satisfied as revenue. 

Upfront License Fees

If a license to our intellectual property is determined to be distinct from the other performance obligations identified 
in  the  arrangement,  we  recognize  revenues  from  nonrefundable,  upfront  license  fees  based  on  the  relative  value 
prescribed to the license compared to the total value of the arrangement. The revenue is recognized when the license 

41

is transferred to the collaborator and the collaborator is able to use and benefit from the license.  For licenses that are 
not  distinct  from  other  obligations  identified  in  the  arrangement,  we  utilize  judgment  to  assess  the  nature  of  the 
combined performance obligation to determine whether the combined performance obligation is satisfied over time 
or at a point in time. If the combined performance obligation is satisfied over time, we apply an appropriate method 
of measuring progress for purposes of recognizing revenue from nonrefundable, upfront license fees.  We evaluate 
the  measure  of  progress  each  reporting  period  and,  if  necessary,  adjust  the  measure  of  performance  and  related 
revenue recognition.

Research and Development Service Payments

Under  the  Allergan  Agreement,  we  were  reimbursed  at  a  certain  percentage  for  performing  research  and 
development services based on hours worked by our employees at a fixed contractual rate per hour and third-party 
pass-through costs we incurred on a quarterly basis. Research and development service payments were included in 
the transaction price in the reporting period we concluded it was probable that recording revenue in the period would 
not result in a significant reversal in amounts recognized in future periods. Accounts receivable were recorded when 
the right to the research and development service payment consideration became unconditional. We recorded the full 
reimbursed  portion  of  these  expenses  accounted  for  under  the  contract  with  customer  accounting  standard  as 
collaboration  revenue  in  our  consolidated  statements  of  operations  as  we  consider  performing  research  and 
development services to be a part of our ongoing and central operations.

Development and Regulatory Milestone Payments

Depending on facts and circumstances, we may record revenues from certain milestones in a reporting period before 
the  milestone  is  achieved  if  we  conclude  that  achievement  of  the  milestone  is  probable  and  that  recognition  of 
revenue related to the milestone will not result in a significant reversal in amounts recognized in future periods. We 
record  a  corresponding  contract  asset  when  this  conclusion  is  reached.  Milestone  payments  that  have  not  been 
included in the transaction price to date are fully constrained. We re-evaluate the probability of achievement of such 
milestones and any related constraint each reporting period. We adjust our estimate of the overall transaction price, 
including the amount of collaborative revenue that was recorded, if necessary.   

Sales-based Milestone and Royalty Payments

Our customer may be required to pay us sales-based milestone payments or royalties on future sales of commercial 
products.  We recognize revenues related to sales-based milestone and royalty payments upon the later to occur of 
(1) achievement of the collaborator’s underlying sales or (2) satisfaction of any performance obligation(s) related to 
these sales, in each case assuming our licensed intellectual property is deemed to be the predominant item to which 
the sales-based milestones and/or royalties relate.

We receive payments from our customer based on billing schedules established in each contract.  Upfront payments 
and  fees  are  recorded  as  deferred  revenue  upon  receipt  or  when  due  until  we  perform  our  obligations  under  the 
arrangement.  If  the  related  performance  obligation  is  expected  to  be  satisfied  within  the  next  12  months,  these 
amounts  will  be  classified  in  current  liabilities.  We  recognize  a  contract  asset  relating  to  our  conditional  right  to 
consideration  that  is  not  subject  to  a  constraint.  Amounts  are  recorded  as  accounts  receivable  when  our  right  to 
consideration is unconditional.  

A net contract asset or liability is presented for each contract with a customer. We do not assess whether a contract 
has  a  significant  financing  component  if  the  expectation  at  contract  inception  is  such  that  the  period  between 
payment by the customer and the transfer of the promised goods or services to the customer will be one year or less.

We may be required to exercise considerable judgment in estimating revenue to be recognized. Judgment is required 
in identifying performance obligations, estimating the transaction price, estimating the standalone selling prices of 
identified  performance  obligations,  which  may  include  forecasted  revenue,  development  timelines,  reimbursement 
rates  for  personnel  and  other  research  and  development  costs,  discount  rates  and  probabilities  of  technical  and 
regulatory success, and estimating the progress towards satisfaction of performance obligations.

On  January  1,  2018,  we  adopted  ASU  No.  2014-09,  Revenue  from  Contracts  with  Customers,  as  amended 
(Accounting Standards Codification Topic 606) (ASC 606) using the modified retrospective method applied to those 
contracts which were not completed as of January 1, 2018. We also elected to use the practical expedient that allows 

42

an  entity  to  expense  the  incremental  cost  of  obtaining  a  contract  as  an  expense  when  incurred  if  the  amortization 
period of the asset that an entity otherwise would have recognized is less than one year. Results for the year ended 
December 31, 2018 are presented under ASC 606, while prior period amounts are not adjusted and continue to be 
reported in accordance with historic accounting under the previous revenue recognition accounting standard. As of 
the  adoption  date  of  ASC  606,  we  had  only  one  contract  with  a  customer,  Allergan,  that  had  not  been 
completed.  Based  on  our  analysis,  we  concluded  there  was  no  significant  change  in  applying  ASC  606  to  our 
agreement  with  Allergan  and  no  amounts  have  been  recognized  within  “accumulated  deficit”  in  the  consolidated 
balance sheet related to the adoption of the new standard.

Goodwill and Indefinite-Lived Intangible Assets

Goodwill and indefinite-lived intangible assets are reviewed for impairment at least annually in the fourth quarter 
and more frequently if events or other changes in circumstances indicate that the carrying amount of the assets may 
not  be  recoverable.  Impairment  of  goodwill  and  indefinite-lived  intangibles  is  determined  to  exist  when  the  fair 
value is less than the carrying value of the net assets being tested.

43

Goodwill

We determined that we have only one operating segment and reporting unit. Accordingly, our review of goodwill 
impairment indicators is performed at the entity-wide level. In performing each annual impairment assessment and 
any interim impairment assessment, we determine if we should qualitatively assess whether it is more likely than not 
that the fair value of goodwill is less than its carrying amount (the qualitative impairment test). Some of the factors 
considered  in  the  assessment  include  general  macroeconomic  conditions,  conditions  specific  to  the  industry  and 
market, cost factors, the overall financial performance and whether there have been sustained declines in our share 
price.  If  we  conclude  it  is  more  likely  than  not  that  the  fair  value  of  the  reporting  unit  is  less  than  its  carrying 
amount,  or  elect  not  to  use  the  qualitative  impairment  test,  a  quantitative  impairment  test  is  performed.  Effective 
January 1, 2020, we early adopted ASU 2017-04, Intangibles-Goodwill and Other (Topic 350): Simplifying the Test 
for Goodwill Impairment (ASU 2017-04), which simplifies how an entity is required to test goodwill for impairment 
by  eliminating  Step  2  from  the  goodwill  impairment  test.  Under  this  accounting  standard,  annual  or  interim 
quantitative  impairment  testing  is  performed  by  comparing  the  estimated  fair  value  of  the  reporting  unit  to  its 
carrying  value.  An  impairment  charge  is  recognized  for  the  amount  by  which  the  carrying  amount  exceeds  the 
reporting  unit’s  fair  value,  not  to  exceed  the  carrying  value  of  goodwill.  We  use  our  market  capitalization  as  an 
indicator  of  fair  value.  We  believe  that  since  our  reporting  unit  is  publicly  traded,  the  ability  of  a  controlling 
stockholder to benefit from synergies and other intangible assets that arise from control might cause the fair value of 
our  reporting  unit  as  a  whole  to  exceed  our  market  capitalization.  However,  we  believe  that  the  fair  value 
measurement need not be based solely on the quoted market price of an individual share of our common stock, but 
also  can  consider  the  impact  of  a  control  premium  in  measuring  the  fair  value  of  its  reporting  unit.  The  control 
premium  utilized  is  based  on  control  premiums  observed  in  recent  acquisitions  of  entities  similar  to  us  that  were 
made on a non-minority basis. Should our market capitalization be less than our total stockholders’ equity as of our 
annual test date or as of any interim impairment testing date, we would also consider market comparables, recent 
trends  in  our  stock  price  over  a  reasonable  period  and,  if  appropriate,  use  an  income  approach  (discounted  cash 
flow) to determine whether the fair value of our reporting unit is greater than our carrying amount. If we were to use 
an  income  approach,  we  would  establish  a  fair  value  by  estimating  the  present  value  of  our  projected  future  cash 
flows expected to be generated from our business. The discount rate applied to the projected future cash flows to 
arrive at the present value would be intended to reflect all risks of ownership and the associated risks of realizing the 
stream  of  projected  future  cash  flows.  Our  discounted  cash  flow  methodology  would  consider  projections  of 
financial performance for a period of several years combined with an estimated residual value. The most significant 
assumptions  we  would  use  in  a  discounted  cash  flow  methodology  are  the  discount  rate,  the  residual  value  and 
expected future revenues, gross margins and operating costs, along with considering any implied control premium. 
In  2020,  we  elected  to bypass the qualitative goodwill  impairment  assessment.  As  of  October 1,  2020,  we  have 
determined through a quantitative impairment test that the fair value significantly exceeded the carrying value of our 
single  reporting  unit,  and  concluded  that  goodwill  was  not  impaired.  In  November  2020,  after  our  public 
announcement  that  it  became  clear  that  patients  who  stopped  therapy  in  Study  211  had  not  achieved  meaningful 
SVR  rates  as  39  of  41  patients  relapsed,  our  stock  price  declined  152%  closing  on  November  5  at  $15.90  and 
opening on November 6 at $6.30. Due to a sustained decline in our stock price during the remainder of the fourth 
quarter of 2020, we determined these factors were an indication of a triggering event of impairment and an interim 
goodwill impairment test was performed as of December 31, 2020. However, our interim quantitative impairment 
test  still  determined  the  fair  value  exceeded  the  carrying  value  of  our  single  reporting  unit  and  concluded  that 
goodwill was still not impaired. We did not recognize any goodwill impairment in any of the years presented.

Indefinite-Lived Intangible Asset

Our indefinite-lived intangible asset consists of in-process research and development (IPR&D) projects acquired in a 
business  combination  that  are  used  in  research  and  development  activities  but  have  not  yet  reached  technological 
feasibility,  regardless  of  whether  they  have  alternative  future  use.  The  primary  basis  for  determining  the 
technological feasibility or completion of these projects is obtaining regulatory approval to market the underlying 
products  in  an  applicable  geographic  region.  We  classify  in-process  research  and  development  acquired  in  a 
business combination as an indefinite-lived intangible asset until the completion or abandonment of the associated 
research and development efforts. Upon completion of the associated research and development efforts, we perform 
a final test for impairment and will determine the useful life of the technology and begin amortizing the assets to 
reflect  their  use  over  their  remaining  lives.  Upon  permanent  abandonment,  we  would  write  off  the  remaining 
carrying amount of the associated IPR&D intangible asset.

In  performing  each  annual  impairment  assessment  and  any  interim  impairment  assessment,  we  determine  if  we 
should qualitatively assess whether it is more likely than not that the fair value of our IPR&D asset is less than its 
carrying  amount  (the  qualitative  impairment  test).  If  we  conclude  that  is  the  case,  or  elect  not  to  use  qualitative 
impairment test, we would proceed with quantitatively determining the fair value of the IPR&D asset and comparing 
its fair value to its carrying value to determine the amount of impairment, if any (the quantitative impairment test).

44

In performing the qualitative impairment test, we consider the results of the most recent quantitative impairment test 
and identify the most relevant drivers of the fair value for the IPR&D asset. The most relevant drivers of fair value 
we  have  identified  are  consistent  with  the  assumptions  used  in  the  quantitative  estimate  of  the  IPR&D  asset 
discussed below. Using these drivers, we identify events and circumstances that may have an effect on the fair value 
of the IPR&D asset since the last time the IPR&D’s fair value was quantitatively determined. We then weigh these 
factors to determine and conclude if it is not more likely than not that the IPR&D asset is impaired. If it is more 
likely  than  not  that  the  IPR&D  asset  is  impaired  we  proceed  with  quantitatively  determining  the  fair  value  of  the 
IPR&D asset.

We use the income approach to determine the fair value of our IPR&D asset. This approach calculates fair value by 
estimating the after-tax cash flows attributable to an in-process project over its useful life and then discounting these 
after-tax cash flows back to a present value. This estimate includes significant assumptions regarding the estimates 
that  market  participants  would  make  in  evaluating  the  IPR&D  asset,  including  the  probability  of  successfully 
completing  clinical  trials  and  obtaining  regulatory  approval  to  market  the  IPR&D  asset,  the  timing  of  and  the 
expected  costs  to  complete  IPR&D  projects,  future  net  cash  flows  from  potential  drug  sales,  which  are  based  on 
estimates  of  the  sales  price  of  the  drug,  the  number  of  patients  who  will  be  diagnosed  and  treated  and  our 
competitive position in the marketplace, and appropriate discount and tax rates. Any impairment to be recorded is 
calculated  as  the  difference  between  the  fair  value  of  the  IPR&D  asset  as  of  the  date  of  the  assessment  with  the 
carrying value of the IPR&D asset on our consolidated balance sheet.

For our 2020 impairment test, we performed a qualitative test and concluded it was more-likely-than-not that the fair 
value  of  our  IPR&D  asset  exceeded  its  carrying  value  and  no  further  testing  was  required.  This  was  based  on  a 
decrease  in  the  probability  of  success  based  on  the  impact  of  the  Study  211  and  dual  combination  VBR  and  NrtI 
therapy’s  ability  to  serve  as  a  finite  and  curative  therapy  for  chronic  HBV  infection  offset  by  an  increase  in  the 
probability of success of 2158 and 3733 based on their advancement into Phase 2 and Phase 1 trials during 2020, 
respectively  and  the  significance  of  the  future  net  cash  flows  from  potential  drug  sales  for  a  finite  and  curative 
therapy for chronic HBV infection as primarily driven by the number of patients who will be diagnosed and treated 
and our competitive position in the marketplace. We did not recognize any IPR&D impairment in any of the years 
presented.

For asset purchases outside of business combinations, we expense any purchased research and development assets as 
of the acquisition date if they have no alternative future uses.

Research and Development Expense and Accruals 

Research and development costs include personnel-related costs, outside contracted services including clinical study 
costs, facilities costs, fees paid to consultants, milestone payments prior to FDA approval, license fees prior to FDA 
approval, professional services, travel costs, dues and subscriptions, depreciation and materials used in clinical trials 
as  well  as  research  and  development  and  costs  incurred  under  our  collaboration  agreements.  Research  and 
development  costs  are  expensed  as  incurred  unless  there  is  an  alternative  future  use  in  other  research  and 
development  projects.  Payments  made  prior  to  the  receipt  of  goods  or  services  to  be  used  in  research  and 
development  are  capitalized  until  the  goods  or  services  are  received.  Such  payments  are  evaluated  for  current  or 
long-term  classification  based  on  when  they  will  be  realized  or  consumed.  Assets  acquired  as  part  of  an  asset 
acquisition  that  are  used  in  research  and  development  or  are  IPR&D  are  immediately  expensed  as  research  and 
development unless there is an alternative future use in other research and development projects. 

As  part  of  the  process  of  preparing  our  consolidated  financial  statements,  we  are  required  to  estimate  certain 
research and development expenses. This process involves reviewing quotations and contracts, reviewing the terms 
of our license agreements, communicating with our vendors and applicable personnel to identify services that have 
been performed on our behalf and estimating the level of service performed and the associated cost incurred for the 
service  when  we  have  not  yet  been  invoiced  or  otherwise  notified  of  the  actual  cost.  The  majority  of  our  service 
providers invoice us monthly in arrears for services performed or when contractual milestones are met. Payments 
made prior to the receipt of goods or services to be used in research and development are capitalized until the goods 
or  services  are  received.  Such  payments  are  evaluated  for  current  or  long-term  classification  based  on  when  they 
will  be  realized  or  consumed.  Examples  of  estimated  amortized  or  accrued  research  and  development  expenses 
include fees to:

(cid:129)

(cid:129)

(cid:129)

CROs and other service providers in connection with clinical studies;

CMOs in connection with the production of clinical trial materials; and

vendors in connection with preclinical development activities.

45

We  base  our  expenses  related  to  clinical  studies  on  our  estimates  of  the  services  received  and  efforts  expended 
pursuant  to  contracts  with  multiple  research  institutions  and  contract  research  organizations  that  conduct  and 
manage clinical studies on our behalf. The financial terms of these agreements are subject to negotiation, vary from 
contract  to  contract  and  may  result  in  uneven  payment  flows  and  expense  recognition.  Payments  under  some  of 
these contracts depend on factors such as the successful enrollment of patients and the completion of clinical trial 
milestones. In either amortizing or accruing service fees, we estimate the time period over which services will be 
performed and the level of effort to be expended in each period. If the actual timing of the performance of services 
or  the  level  of  effort  varies  from  our  estimate,  we  adjust  the  related  prepayment  or  accrual  accordingly.  Our 
understanding  of  the  status  and  timing  of  services  performed  relative  to  the  actual  status  and  timing  of  services 
performed may vary and may result in our reporting changes in estimates in any particular period. Adjustments to 
prior period estimates have not been material for the years ended December 31, 2020 and 2019.

We have and may continue to enter into license agreements to access and utilize certain technology. In each case, we 
evaluate  if  the  license  agreement  results  in  the  acquisition  of  an  asset  or  a  business.  To  date,  none  of  our  license 
agreements have been considered to be acquisitions of businesses. For asset acquisitions, the upfront payments to 
acquire  such  licenses,  as  well  as  any  future  milestone  payments,  are  immediately  recognized  as  research  and 
development  expense  when  paid,  provided  there  is  no  alternative  future  use  of  the  rights  in  other  research  and 
development  projects.  These  license  agreements  may  also  include  contingent  consideration  in  the  form  of  cash 
payments  to  be  made  for  future  milestone  events.  We  assess  whether  such  contingent  consideration  meets  the 
definition of a derivative and to date we have determined that such contingent consideration are not derivatives.

Restructuring Charges 

We  recognize  restructuring  charges  related  to  reorganization  plans  that  have  been  committed  to  by  us  and  when 
liabilities have been incurred. In connection with these activities, we record restructuring charges at fair value for (1) 
contractual  employee  termination  benefits  when  obligations  are  associated  to  services  already  rendered,  rights  to 
such  benefits  have  vested,  and  payment  of  benefits  is  probable  and  can  be  reasonably  estimated,  (2)  one-time 
employee termination benefits when we have committed to a plan of termination, the plan identifies the employees 
and their expected termination dates, the details of termination benefits are complete, it is unlikely changes to the 
plan  will  be  made  or  the  plan  will  be  withdrawn  and  communication  to  such  employees  has  occurred,  and  (3) 
contract termination costs when a contract is terminated before the end of its term. 

One-time  employee  termination  benefits  are  recognized  in  their  entirety  when  communication  has  occurred and 
future  services  are  not  required.  If  future  services  are  required,  the  costs  are  recorded  ratably  over  the  remaining 
period  of  service.  Contract  termination  costs  to  be  incurred  over  the  remaining  contract  term  without  economic 
benefit are recorded in their entirety when the contract is canceled.

The recognition of restructuring charges requires us to make certain judgments and estimates regarding the nature, 
timing and amount of costs associated with the planned reorganization plan. To the extent the actual results differ 
from  its  estimates  and  assumptions,  we  may  be  required  to  revise  the  estimates  of  future  accrued  restructuring 
liabilities,  requiring  the  recognition  of  additional  restructuring  charges  or  the  reduction  of  accrued  restructuring 
liabilities previously recognized. Such changes to previously estimated amounts may be material to our consolidated 
financial statements. Changes in the estimates of the restructuring charges are recorded in the period in which the 
change is determined. 

At  the  end  of  each  reporting  period,  we  evaluate  the  remaining  accrued  restructuring  balances  to  ensure  that  no 
excess accruals are retained and the utilization of the provisions are for their intended purpose in accordance with 
developed restructuring plans.

Off-Balance Sheet Arrangements

Since our inception, we have not engaged in any off-balance sheet arrangements.   

Contractual Obligations

We  have  contractual  and  commercial  obligations  under  our  operating  lease  commitments  and  licenses.  The 
following table summarizes our future contractual obligations and commercial commitments at December 31, 2020 
(in thousands): 

46

Operating lease obligations .......................................   $
Total contractual obligations ...............................   $

4,369    $
4,369    $

7,407    $
7,407    $

—    $
—    $

    Total
—    $ 11,776 
—    $ 11,776  

Payments Due By Period

Less than

1 year     1-3 years     3-5 years    

More than
5 years

In general, milestone, royalty and other contingent fees associated with certain collaboration and license agreements 
have not been included in the above table of contractual obligations, because we cannot reasonably estimate if or 
when they will occur. The milestone payments included in the table of contractual obligations above are payments 
we believe are reasonably likely to occur during the indicated time periods. We enter into contracts in the normal 
course of business with CROs for clinical trials and CMO’s for clinical supply manufacturing and with vendors for 
preclinical  research  studies  and  other  services  and  products  for  operating  purposes,  which  generally  provide  for 
termination  within  30  days  of  notice,  and  therefore,  are  cancelable  contracts  and  not  included  in  the  table  above. 
Further, we anticipate that our operating lease obligations will be higher than projected as we renew existing real 
estate leases that expire in 2020 and enter into new or expanded real estate leases.

Results of Operations

General

At  December  31,  2020,  we  had  an  accumulated  deficit  of  $501.6  million  primarily  as  a  result  of  research  and 
development expenses and general and administrative expenses. While we may in the future generate revenue from 
a variety of sources, including license fees, milestone payments, research and development payments in connection 
with strategic partnerships and/or product sales, our product candidates are in the clinical stage of development and 
may  never  be  successfully  developed  or  commercialized.  Accordingly,  we  expect  to  continue  to  incur  substantial 
losses from operations for the foreseeable future and there can be no assurance that we will ever generate significant 
revenues.

Comparison of the Years Ended December 31, 2020 and 2019

Collaboration Revenue

The following table summarizes the period-over-period changes in our collaboration revenue (in thousands, except 
for percentages):

Collaboration revenue..........................................   $

79,105    $

15,963    $

Year ended December 31,
2019
2020

$ Change

2020 vs. 2019  
63,142 

  % Change
  2020 vs. 2019  

396%

Collaboration revenue for the year ended December 31, 2020 includes the remaining deferred revenue balance of 
$37.0  million  and  reimbursements  incurred  under  the  Allergan  Agreement,  for  which  AbbVie  Inc.  gave  written 
notice  of  termination  in  June  2020  following  its  acquisition  of  Allergan,  and  $31.0  million  recognized  for  the 
transfer of the VBR License upon entering into the Collaboration Agreement with BeiGene (BeiGene Agreement). 

Research and Development Expense 

The  following  table  summarizes  the  period-over-period  changes  in  our  research  and  development  expenses  (in 
thousands, except for percentages):

Year ended December 31,

$ Change

  % Change

Program/Description
HBV(1) ..................................................................   $
25%
Microbiome(2).......................................................    
24%
25%
Total research and development expenses...........   $
(1) Expenses presented for HBV include reimbursement of expenses of $0.2 million under the Arbutus Agreement, 

2020 vs. 2019  
14,423 
6,643 
21,066 

71,957    $
34,866     
106,823    $

57,534    $
28,223     
85,757    $

  2020 vs. 2019  

2019

2020

as discussed in Note 9 to the Consolidated Financial Statements.

(2) Expenses  presented  for  the  Microbiome  program  exclude  collaboration  revenue  related  to  expense 
reimbursements under the Allergan Agreement as discussed in Note 9 to the Consolidated Financial Statements.

47

 
 
 
 
 
 
   
   
 
 
  
   
   
  
   
   
 
 
 
   
   
  
  
  
Research and development expenses were $106.8 million for the year ended December 31, 2020 compared to $85.8 
million for the year ended December 31, 2019. The increase was due to an increase of $14.4 million in research and 
development  expenses  related  to  the  HBV  program  and  an  increase  of  $6.6  million  in  research  and  development 
expenses related to the Microbiome program. These increases were primarily due to increases in clinical activities, 
chemistry  and  manufacturing  control  activities  to  support  VBR,  2158,  3733  and  Microbiome  clinical  trials  and 
increased  salary  and  benefits  due  to  additional  employees.  In  December  2020,  we  and  our  Board  of  Directors 
determined that it was in our best interest to wind down the Microbiome program, enabling us to prioritize resources 
and  focus  on  the  advancement  of  our  pipeline  of  novel  core  inhibitors  for  chronic  HBV  infection.  We  expect  to 
complete  the  wind-down  of  the  Microbiome  program  in  early  2021.  Microbiome  expenses  for  the  year  ended 
December  31,  2020  includes  $5.5  million  in  restructuring  costs  related  to  the  wind-down,  which  consists  of  $3.9 
million in employee severance and related benefits and $1.6 million in asset impairment and other costs. Refer to 
Note  6  to  the  Consolidated  Financial  Statements  for  additional  information.  Research  and  development  expenses 
include non-cash stock-based compensation expenses of $11.4 million for both the years ended December 31, 2020 
and 2019. 

General and Administrative Expense

The  following  table  summarizes  the  period-over-period  change  in  our  general  and  administrative  expenses  (in 
thousands, except for percentages):

General and administrative expenses...................   $

37,058    $

32,919    $

Year ended December 31,
2019
2020

$ Change

2020 vs. 2019  
4,139 

  % Change
  2020 vs. 2019  

13%

General  and  administrative  expense  consists  primarily  of  salaries,  consulting  fees  and  other  related  costs, 
professional  fees  for  legal  services,  accounting  and  tax  services,  insurance  and  travel  expenses,  as  well  as  stock-
based compensation expense associated with equity awards to our employees, consultants and directors.

General and administrative expenses were $37.1 million for the year ended December 31, 2020, compared to $32.9 
million for the year ended December 31, 2019. The increase in general and administrative expenses was primarily 
due to an increase of $3.1 million in professional expenses mostly attributable to the amortized incremental contract 
costs  associated  with  entering  into  the  BeiGene  Agreement,  $1.3  million  in  stock-based  compensation  expense,  
$0.5  million  in  equipment  rental  and  $0.3  million  in  recruitment  costs  due  to  an  increase  in  headcount  partially 
offset  by  a  decrease  of  $0.9  million  in  travel  related  expenses  due  to  state  and  local  laws  restricting  travel  in 
response  to  the  COVID-19  pandemic.  General  and  administrative  expenses  includes  non-cash  stock-based 
compensation  expense  of  $10.5  million  and  $9.2  million  for  the  years  ended  December  31,  2020  and  2019, 
respectively. Stock-based  compensation  expense  for  the  year  ended  December  31,  2020  includes  the  reversal  of 
previously recognized expense of $1.7 million related to forfeited awards resulting from the departure of one of our 
former officers during the period, while stock-based compensation expense for the year ended December 31, 2019 
includes  the  reversal  of  previously  recognized  expense  of  $3.6  million  related  to  forfeited  awards  resulting  from 
another our former officers during the period.  

Interest and Other Income

The  following  table  summarizes  the  period-over-period  changes  in  our  interest  and  other  income  (in  thousands, 
except for percentages):

Interest and other income.....................................   $

2,624    $

4,305    $

(1,681)   

-39%

Year ended December 31,
2019
2020

$ Change

2020 vs. 2019  

  % Change
  2020 vs. 2019  

Interest and other income was $2.6 million for the year ended December 31, 2020 compared to $4.3 million for the 
same  period  in  2019.  Interest  income  for  the  years  ended  December  31,  2020  and  2019  was  primarily  related  to 
interest  income  earned  on  marketable  securities,  corporate  bonds  and  money  market  funds  and  the  decrease  is  a 
result of lower balances and lower yields carried in 2020.  

48

 
 
   
 
 
  
   
   
  
 
 
   
 
 
  
   
   
Income Tax (Expense) Benefit

The following table summarizes the period-over-period change in our income tax benefit (in thousands, except for 
percentages):

Year ended December 31,
2019
2020

$ Change

2020 vs. 2019  

  % Change
  2020 vs. 2019  

Income tax benefit................................................   $

—    $

774    $

(774)   

-100%

Income tax benefit for the year ended December 31, 2020 was nominal compared to an income tax benefit for year 
ended December 31, 2019 of $0.8 million. The income tax benefit in the prior year is primarily due to a change in 
our  state  and  local  effective  tax  rate  and  recording  the  impact  of  certain  indefinite-lived  deferred  tax  asset 
carryforwards. 

Comparison of the Years Ended December 31, 2019 and 2018

Collaboration Revenue

The following table summarizes the period-over-period changes in our collaboration revenue (in thousands, except 
for percentages):

Collaboration revenue..........................................   $

15,963    $

14,804    $

Year ended December 31,
2018
2019

$ Change

2019 vs. 2018  
1,159 

  % Change
  2019 vs. 2018  

8%

During the year ended December 31, 2019, we generated $16.0 million of collaboration revenue, which included the 
amortization of deferred revenue and reimbursement revenue in each case incurred under the Allergan Agreement, 
an increase of $1.2 million from $14.8 million for the same period in 2018. The increase was based on increased 
research efforts performed during 2019 for our Microbiome program.

Research and Development Expense 

The  following  table  summarizes  the  period-over-period  changes  in  our  research  and  development  expenses  (in 
thousands, except for percentages):

Year ended December 31,

$ Change

  % Change

Program/Description
HBV(1) ..................................................................   $
16%
Microbiome(2).......................................................    
21%
18%
Total research and development expenses...........   $
(1)  Expenses  presented  for  the  Microbiome  program  exclude  collaboration  revenue  related  to  expense 
reimbursements under the Allergan Agreement as discussed in Note 9 to the Consolidated Financial Statements.

2019 vs. 2018  
8,118 
4,898 
13,016 

49,416    $
23,325     
72,741    $

57,534    $
28,223     
85,757    $

  2019 vs. 2018  

2019

2018

Research and development expenses were $85.8 million for the year ended December 31, 2019 compared to $72.7 
million for the year ended December 31, 2018. The increase was due to an increase of $8.1 million in research and 
development  expenses  related  to  the  HBV  program  and  an  increase  of  $4.9  million  in  research  and  development 
expenses related to the Microbiome program. These increases were primarily due to increases in clinical activities, 
chemistry and manufacturing control activities to support VBR, 2158 and Microbiome clinical trials and increased 
salary and benefits due to additional employees. Research and development expenses include non-cash stock based 
compensation  expenses  of  $11.4  million  for  the  year  ended  December  31,  2019,  a  decrease  of  $0.4  million  from 
$11.8 million for the year ended December 31, 2018.

General and Administrative Expense

The  following  table  summarizes  the  period-over-period  change  in  our  general  and  administrative  expenses  (in 
thousands, except for percentages):

Year ended December 31,
2018
2019

$ Change

2019 vs. 2018  

  % Change
  2019 vs. 2018  

General and administrative expenses...................   $

32,919    $

34,798    $

(1,879)   

-5%

General  and  administrative  expense  consists  primarily  of  salaries,  consulting  fees  and  other  related  costs, 
professional  fees  for  legal  services,  accounting  and  tax  services,  insurance  and  travel  expenses,  as  well  as  stock-
based compensation expense associated with equity awards to our employees, consultants and directors.

49

 
 
   
 
 
  
   
   
 
 
   
 
 
  
   
   
  
   
   
 
 
 
   
   
  
  
  
 
 
   
 
 
  
   
   
General and administrative expenses were $32.9 million for the year ended December 31, 2019, compared to $34.8 
million for the year ended December 31, 2018. The increase in general and administrative expenses was primarily 
due  to  an  increase  of  $3.5  million  in  employee  related  expenses  due  to  the  addition  of  employees  in  executive 
management,  finance  and  human  resources.  This  increase  also  includes  a  one-time  expense  of  $1.7  million  for 
severance  packages  in  conjunction  with  the  relocation  of  our  corporate  headquarters  to  South  San  Francisco, 
California effective January 1, 2020, the departure of one of our former executives, $0.9 million in rent expenses for 
our new office in South San Francisco and $0.3 million in professional expenses.

Stock-based  compensation  expense  was  $9.2  million  for  the  year  ended  December  31,  2019,  a  decrease  of  $7.5 
million from $16.7 million for the year ended December 31, 2018. The decrease was primarily due to a $4.3 million 
one-time expense related to the departure and transition to consultant of one of our former executive officers in 2018 
coupled with the reversal of previously recognized expense of $3.6 million related to forfeited awards resulting from 
the departure of one of our former executive officers in 2019. 

Interest and Other Income

The  following  table  summarizes  the  period-over-period  changes  in  our  interest  and  other  income  (in  thousands, 
except for percentages):

Interest and other income.....................................   $

4,305    $

3,083    $

Year ended December 31,
2018
2019

$ Change

2019 vs. 2018  
1,222 

  % Change
  2019 vs. 2018  

40%

Interest and other income was $4.3 million for the year ended December 31, 2019 compared to $3.1 million for the 
same  period  in  2018.  Interest  income  for  the  years  ended  December  31,  2019  and  2018  was  primarily  related  to 
interest  income  earned  on  marketable  securities,  corporate  bonds  and  money  market  funds,  and  the  increase  is  a 
result of higher balances carried in 2019.  

Income Tax (Expense) Benefit

The following table summarizes the period-over-period change in our income tax benefit (in thousands, except for 
percentages):

Income tax benefit (expense) ...............................   $

774    $

(1,099)  $

Year ended December 31,
2018
2019

$ Change

2019 vs. 2018  
1,873 

  % Change
  2019 vs. 2018  

170%

Income tax benefit for the year ended December 31, 2019 was $0.8 million compared to an income tax expense for 
year ended December 31, 2018 of $1.1 million. The income tax benefit in 2019 is primarily due to a change in our 
state  and  local  effective  tax  rate  and  recording  the  impact  of  certain  indefinite-lived  deferred  tax  asset 
carryforwards. The  income  tax  expense  recognized  in  2018  is  primarily  due  to  a  change  in  our  state  and  local 
effective tax rate.

Liquidity and Capital Resources

As a result of our significant research and development expenditures and the lack of any FDA-approved products to 
generate  product  sales  revenue,  we  have  not  been  profitable  and  have  generated  operating  losses  since  we  were 
incorporated  in  October  2005.  We  have  funded  our  operations  through  December  31,  2020  principally  with  debt 
prior to our initial public offering, and thereafter with equity financing, raising an aggregate of $551.8 million in net 
proceeds  from  public  offerings  and  private  placements  from  inception  to  December  31,  2020.  Additionally,  in 
February  2017,  we  received  a  $50.0  million  upfront  payment  in  connection  with  the  execution  of  the  Allergan 
Agreement and in July 2020, we received a $40.0 million upfront payment in connection with the execution of the 
BeiGene Agreement.

In July 2018, we sold to various investors an aggregate of 4,600,000 shares of common stock in a public offering at 
$36.00  per  share,  which  included  the  exercise  in  full  by  the  underwriters  of  their  option  to  purchase  600,000 
additional shares of common stock. We received aggregate net proceeds of $155.4 million from the offering and the 
option exercise, after deducting underwriting discounts and commissions and offering expenses payable.

50

 
 
   
 
 
  
   
   
  
 
 
   
 
 
  
   
   
  
In  December  2019,  we  sold  to  various  investors  an  aggregate  of  6,287,878  shares  of  common  stock  at  a  public 
offering price of $16.50 per share, which included the exercise in full by the underwriters of their option to purchase 
1,136,363  shares  of  common  stock,  and  pre-funded  warrants  to  purchase  2,424,242  shares  of  common  stock  at  a 
public offering price of $16.499. We received aggregate net proceeds of $134.7 million from the offering and the 
option exercise, after deducting underwriting discounts and commissions and offering expenses payable.

In  December  2020,  we  sold  an  aggregate  of  892,840  shares  of  common  stock  through  “at-the-market”  offerings 
(2020 ATM), resulting in net proceeds of $5.5 million. 

Cash Flows 

A summary of our cash flows for the periods presented was as follows (in thousands):

Operating activities ...........................................................................   $
Investing activities ............................................................................    
Financing activities ...........................................................................    
Net increase (decrease) in cash and cash equivalents..................   $

(62,957)   $
68,070     
7,599     
12,712    $

(84,067)   $
(50,318)    
139,646     
5,261    $

(64,958)
(135,397)
159,793 
(40,562)

Year Ended December 31,
2019

2018

2020

Net Cash Used in Operating Activities

Net cash used in operating activities was $63.0 million for the year ended December 31, 2020. This was primarily 
due to $62.2 million of net loss and a decrease of $30.3 million of operating assets and liabilities, which were offset 
by  a  $21.9  million  non-cash  expense  recorded  for  stock-based  compensation,  $5.2  million  of  amortization  of 
operating  lease  right-of-use  assets,  $1.8  million  in  non-cash  expense  for  acquired  IPR&D  and  $0.7  million  of 
depreciation and amortization expense. 

Net cash used in operating activities was $84.1 million for the year ended December 31, 2019. This was primarily 
due to $97.6 million of net loss, a decrease of $9.5 million of operating assets and liabilities, $0.8 million of deferred 
income  tax  benefit  and  $1.7  million  of  amortization  of  discount  on  marketable  securities,  which  were  offset  by  a 
$20.6 million non-cash expense recorded for stock-based compensation, $4.5 million of amortization of operating 
lease right-of-use assets and $0.5 million of depreciation and amortization expense. 

Net cash used in operating activities was $65.0 million for the year ended December 31, 2018. This was primarily 
due  to  $90.8  million  of  net  loss,  a  decrease  of  $4.2  million  of  operating  assets  and  liabilities  and  $0.2  million  of 
amortization of discount on marketable securities, which were offset by a $28.5 million non-cash expense recorded 
for stock-based compensation, $0.6 million of depreciation and amortization expense and $1.1 million of deferred 
income tax expenses.

Net Cash Provided by (Used in) Investing Activities

Net cash provided by investing activities for the year ended December 31, 2020 was $68.1 million primarily due to a 
purchase  of  $193.2  million  marketable  securities,  $0.5  million  of  fixed  assets  and  $1.8  million  of  IPR&D,  which 
were  offset  by  $221.6  million  for  the  redemption  of  marketable  securities  and  $41.9  million  for  the  sale  of 
marketable securities.

Net  cash  used  in  investing  activities  for  the  year  ended  December  31,  2019  was  $50.3  million  primarily  due  to  a 
purchase  of  $281.3  million  marketable  securities  and  $1.6  million  of  fixed  assets,  which  were  offset  by  $203.9 
million for the redemption of marketable securities and $28.7 million for the sale of marketable securities.

Net cash used in investing activities for the year ended December 31, 2018 was $135.4 million primarily due to a 
purchase of $183.9 million marketable securities and $0.3 million of fixed assets and construction in progress, which 
were offset by $48.9 million for the redemption of marketable securities.

51

 
 
 
 
 
   
   
 
Net Cash Provided by Financing Activities

Net cash provided by financing activities for the year ended December 31, 2020 was $7.6 million resulting from the 
net  proceeds  of  $5.5  million  from  the  sale  of  892,840  shares  of  our  common  stock  under  the  2020  ATM,  $1.5 
million from the exercise of stock options to purchase 175,579 shares of common stock and $0.7 million from the 
issuance of 86,812 shares of common stock under our 2018 ESPP.

Net cash provided by financing activities for the year ended December 31, 2019 was $139.6 million resulting from 
the net proceeds of $134.7 million from our public offering of 6,287,878 shares of common stock and 2,424,242 pre-
funded  warrants  to  purchase  2,424,242  shares  of  common  stock  at  a  public  offering  price  of  $16.499,  including 
1,136,363  shares  of  common  stock  purchased  by  the  underwriters  pursuant  to  their  30-day  option  to  purchase 
additional shares, $4.2 million from the exercise of stock options to purchase 585,292 shares of common stock and 
$0.7 million from the issuance of 59,370 shares of common stock under our 2018 ESPP.

Net cash provided by financing activities for the year ended December 31, 2018 was $159.8 million, resulting from 
the net proceeds of $155.4 million from our public offering of 4,600,000 shares of common stock, including 600,000 
shares of common stock purchased by the underwriters pursuant to their 30-day option to purchase additional shares, 
and $4.0 million from the exercise of stock options to purchase 775,224 shares of common stock.

Future Funding Requirements

We  expect  our  expenses  related  to  HBV  program  to  remain  flat  in  2021  but  to  generally  increase  over  time  in 
connection with our ongoing activities, particularly as we continue the research, development and clinical studies of 
our product candidates and pursue our intellectual property strategy. Accordingly, we will need to obtain substantial 
additional funding in connection with our continuing operations. If we are unable to raise capital when needed or on 
attractive terms, we could be forced to delay, reduce or eliminate our research and development programs or future 
commercialization efforts.

We  monitor  our  cash  needs  and  the  status  of  the  capital  markets  on  a  continuous  basis.  From  time  to  time,  we 
opportunistically raise capital and have done so numerous times since our initial public offering by issuing equity 
securities, most recently in December 2020. We expect to continue to raise capital when and as needed and at the 
time and in the manner most advantageous to us.

We expect that our existing cash, cash equivalents and marketable securities, will enable us to fund our operating 
expenses and capital expenditure requirements for at least the next twelve months. Our future capital requirements 
will depend on many factors, including:

(cid:129)

(cid:129)

(cid:129)

(cid:129)

(cid:129)

(cid:129)

the scope, progress, results and costs of our ongoing drug discovery, nonclinical development, laboratory 
testing and clinical studies of our product candidates and any additional clinical studies we may conduct in 
the future;

the extent to which we further acquire or in-license other product candidates and technologies;

our  ability  to  manufacture,  and  to  contract  with  third  parties  to  manufacture,  adequate  supplies  of  our 
product candidates for our clinical studies and any eventual commercialization;

the costs, timing and outcome of regulatory review of our product candidates;

the  costs  of  preparing,  filing  and  prosecuting  patent  applications  in  the  United  States  and  abroad, 
maintaining  and  enforcing  our  intellectual  property  rights  and  defending  intellectual  property-related 
claims; and

our ability to establish and maintain collaborations on favorable terms, if at all.

Identifying potential product candidates and conducting nonclinical testing and clinical studies is a time-consuming, 
expensive  and  uncertain  process  that  takes  years  to  complete,  and  we  may  never  generate  the  necessary  data  or 
results  required  to  obtain  marketing  approval  and  achieve  product  sales.  In  addition,  our  product  candidates,  if 
approved,  may  not  achieve  commercial  success.  Our  commercial  revenues,  if  any,  will  be  derived  from  sales  of 
medicines  that  we  do  not  expect  to  be  commercially  available  for  years,  if  at  all.  Accordingly,  we  will  need  to 

52

continue to rely on additional financings to achieve our business objectives. Adequate additional financings may not 
be available to us on acceptable terms, or at all.

Until  such  time,  if  ever,  as  we  can  generate  substantial  product  revenues,  we  expect  to  finance  our  cash  needs 
through  a  combination  of  equity  offerings,  debt  financings,  collaborations,  strategic  alliances  and  licensing 
arrangements. We do not have any committed external source of funds. To the extent that we raise additional capital 
through the sale of equity or convertible debt securities, the ownership interest of our stockholders will be diluted, 
and the terms of these securities may include liquidation or other preferences that adversely affect the rights of our 
common  stockholders.  Debt  financing,  if  available,  may  involve  agreements  that  include  covenants  limiting  or 
restricting  our  ability  to  take  specific  actions,  such  as  incurring  additional  debt,  making  capital  expenditures  or 
declaring dividends.

If we raise funds through additional collaborations, strategic alliances or licensing arrangements with third parties, 
we may have to relinquish valuable rights to our technologies, future revenue streams, research programs or product 
candidates or to grant licenses on terms that may not be favorable to us. If we are unable to raise additional funds 
through equity or debt financings when needed, we may be required to delay, limit, reduce or terminate our product 
development or future commercialization efforts or grant rights to develop and market product candidates that we 
would otherwise prefer to develop and market ourselves.

Recent Accounting Pronouncements

See  Note  2  of  notes  to  the  consolidated  financial  statements  for  a  discussion  of  recent  accounting  standards  and 
pronouncements.

Cautionary Statement

We  operate  in  a  highly  competitive  environment  that  involves  a  number  of  risks,  some  of  which  are  beyond  our 
control. The following statement highlights some of these risks. For more detail, see “Item 1A. Risk Factors.”

Statements  contained  in  this  Form  10-K  that  are  not  historical  facts,  are  or  might  constitute  forward-looking 
statements under the safe harbor provisions of the Private Securities Litigation Reform Act of 1995. Although we 
believe  the  expectations  reflected  in  such  forward-looking  statements  are  based  on  reasonable  assumptions,  our 
expectations might not be attained. Forward-looking statements involve known and unknown risks that could cause 
actual results to differ materially from expected results. Factors that could cause actual results to differ materially 
from  our  expectations  expressed  in  the  report  include,  among  others:  risks  related  to  the  costs,  timing,  regulatory 
review and results of our nonclinical studies and clinical studies; our ability to obtain FDA approval of our product 
candidates; our anticipated capital expenditures, our estimates regarding our capital requirements, and our need for 
future  capital;  our  liquidity  and  working  capital  requirements;  our  expectations  regarding  our  revenues,  expenses 
and other results of operations; the unpredictability of the size of the markets for, and market acceptance of, any of 
our products; our ability to sell any approved products and the price we are able realize; our ability to establish and 
maintain collaborations on favorable terms; our ability to obtain future funding on acceptable terms; our ability to 
hire and retain necessary employees and to staff our operations appropriately; our ability to compete in our industry 
and  innovation  by  our  competitors;  our  ability  to  stay  abreast  of  and  comply  with  new  or  modified  laws  and 
regulations that currently apply or become applicable to our business; estimates and estimate methodologies used in 
preparing  our  financial  statements;  the  future  trading  prices  of  our  common  stock  and  the  impact  of  securities 
analysts’ reports on these prices; and the risks set out in our filings with the SEC.

53

Item 7A. Quantitative and Qualitative Disclosures about Market Risk

Our primary exposure to market risk is interest income sensitivity, which is affected by changes in the general level 
of U.S. interest rates.

We  do  not  believe  that  our  cash  and  equivalents  have  significant  risk  of  default  or  illiquidity.  Under  our  current 
investment policies, we invest our cash and cash equivalents in money market funds which invest in short-term U.S. 
Treasury  securities  with  insignificant  rates  of  return.  We  also  invest  our  cash  and  cash  equivalents  in  readily 
marketable,  high-quality  securities  that  are  diversified  and  structured  to  minimize  market  risks.  Our  exposure  to 
market  risk  for  changes  in  interest  rates  relates  primarily  to  our  investments  in  marketable  securities.  Marketable 
securities held in our investment portfolio are subject to changes in market value in response to changes in interest 
rates  and  liquidity.  A  significant  change  in  market  interest  rates  could  have  a  material  impact  on  interest  income 
earned from our investment portfolio. Changes in interest rates may affect the fair value of our investment portfolio; 
however, we will not recognize such gains or losses in our statement of operations and comprehensive income (loss) 
unless the investments are sold.  

While we believe our cash and equivalents do not contain excessive risk, we cannot provide absolute assurance that 
in  the  future  our  investments  will  not  be  subject  to  adverse  changes  in  market  value.  In  addition,  we  maintain 
significant  amounts  of  cash  and  equivalents  at  one  or  more  financial  institutions  that  are  in  excess  of  federally 
insured limits.  

Inflation generally affects us by increasing our cost of labor and clinical study costs. We do not believe that inflation 
has had a material effect on our results of operations during 2020, 2019 or 2018.

Item 8. Financial Statements and Supplementary Data

The financial statements required to be filed pursuant to this Item 8 are appended to this report. An index of those 
financial statements is found on page F-1.

Item 9. Changes in and Disagreements with Accountants on Accounting and Financial Disclosure

None.

Item 9A. Controls and Procedures

Evaluation of Disclosure Controls and Procedures

We maintain a system of disclosure controls and procedures, as defined in Rule 13a-15(e) promulgated under the 
Securities  and  Exchange  Act  of  1934,  as  amended  (the  Exchange  Act),  that  is  designed  to  provide  reasonable 
assurance that information, which is required to be disclosed in our reports filed pursuant to the Exchange Act, is 
accumulated and communicated to management in a timely manner. At the end of fiscal year ending December 31, 
2020, we carried out an evaluation, under the supervision, and with the participation of, our management, including 
our Chief Executive Officer and our Chief Financial Officer, of the effectiveness of the design and operation of our 
disclosure controls and procedures pursuant to Exchange Act Rule 13a-15(b). Based upon that evaluation, our Chief 
Executive Officer and Chief Financial Officer concluded that our disclosure controls and procedures for the fiscal 
year ending as of December 31, 2020 were effective at reasonable assurance levels.

Management’s Annual Report on Internal Control over Financial Reporting

Our management is responsible for establishing and maintaining adequate internal control over financial reporting, 
as such term is defined in Exchange Act Rule 13a-15(f). Our internal control over financial reporting is designed to 
provide  reasonable  assurance  to  our  management  and  Board  of  Directors  regarding  the  preparation  and  fair 
presentation  of  published  financial  statements.  A  control  system,  no  matter  how  well  designed  and  operated,  can 
only provide reasonable, not absolute, assurance that the objectives of the control system are met. Because of these 
inherent limitations, management does not expect that our internal controls over financial reporting will prevent all 
error  and  all  fraud.  Under  the  supervision  and  with  the  participation  of  our  management,  including  our  Chief 
Executive Officer and our Chief Financial Officer, we conducted an evaluation of the effectiveness of our internal 
control over financial reporting based on the framework in Internal Control-Integrated Framework issued in 2013 by 
the  Committee  of  Sponsoring  Organizations  of  the  Treadway  Commission.  Based  on  our  evaluation  under  the 

54

framework  in  Internal  Control-Integrated  Framework,  our  management  concluded  that  our  internal  control  over 
financial reporting was effective as of December 31, 2020.

Our independent registered public accounting firm, Ernst & Young LLP has issued an opinion on the effectiveness 
of  our  internal  control  over  financial  reporting  as  of  December  31,  2020.  The  report  of  Ernst  &  Young  LLP  is 
included with the financial statements appended to this Form 10-K pursuant to Item 8.

Changes in Internal Control over Financial Reporting

There were no changes in our internal control over financial reporting in the fourth quarter of 2020 that materially 
affected, or are reasonably likely to materially affect, our internal control over financial reporting.

Item 9B. Other Information

Not applicable.

55

PART III

ITEM 10.  Directors, Executive Officers and Corporate Governance

Except as set forth below, the information required by this item will be contained in our definitive proxy statement 
to be filed with the SEC in connection with the Annual Meeting of Stockholders (Proxy Statement) within 120 days 
after the conclusion of our fiscal year ended December 31, 2020 and is incorporated in this Annual Report on Form 
10-K by reference.

Code of Ethics

Our Board has adopted a Code of Ethics for our principal executive officer and all senior financial officers and a 
Code  of  Conduct  applicable  to  all  of  our  employees  and  our  directors.  Both  Codes  are  available  under  the 
“Investors—Corporate Governance” section of our website at www.assemblybio.com. If we make any substantive 
amendments to, or grant any waivers from, the Code of Ethics for our principal executive officer, principal financial 
officer, principal accounting officer, controller or persons performing similar functions, or any officer or director, 
we will disclose the nature of such amendment or waiver on our website or in a Current Report on Form 8-K.

ITEM 11.  Executive Compensation

The information required by this item will be contained in the Proxy Statement and is incorporated into this Annual 
Report on Form 10-K by reference.

ITEM  12.  Security  Ownership  of  Certain  Beneficial  Owners  and  Management  and  Related  Stockholder 
Matters

Except for the table regarding equity compensation plans, which is included in Part II, Item 5 of this Annual Report 
on Form 10-K, the information required by this item will be contained in the Proxy Statement and is incorporated 
into this Annual Report on Form 10-K by reference.

ITEM 13.  Certain Relationships and Related Party Transactions, and Director Independence

The information required by this item will be contained in the Proxy Statement and is incorporated into this Annual 
Report on Form 10-K by reference.

ITEM 14.  Principal Accounting Fees and Services

The information required by this item will be contained in the Proxy Statement and is incorporated into this Annual 
Report on Form 10-K by reference.

ITEM 15.  Exhibits, Financial Statement Schedules

(a) Exhibits.   The following exhibits are filed as part of this registration statement:

Exhibit
Number  

  3.1

  3.2

  4.1
  4.2
  4.3
10.1

10.2*

Description of Document
 Fifth Amended and Restated Certificate of Incorporation 
dated June 11, 2020.
 Amended and Restated Bylaws as amended through 
January 22, 2021.
 Specimen of Common Stock Certificate.
Form of Pre-Funded Warrant.
Description of Securities.
 Sub-Sublease, dated as of July 18, 2018, between 
Prothena Biosciences, Inc., as Sub-Sublandlord, and 
Assembly Biosciences, Inc., as Sub-Subtenant.
 Exclusive License Agreement dated September 3, 2013 
by and between The Indiana University Research and 
Technology Corporation and Assembly Pharmaceuticals, 
Inc.

Registrant’s
Form
8-K

8-K

S-3
8-K

Dated
 06/01/2018 

 01/27/2021 

 12/30/2015 
12/16/2019

Exhibit
No.
3.1

Filed
Herewith

3.1

4.1
4.1

10-Q

 11/08/2018 

10.1

X

10-Q

 11/17/2014  10.29  

56

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Exhibit
Number  

10.3†

10.4†

10.5†‡

10.6#

10.7#

10.8#

10.9#

10.10#

10.11#

10.12#

10.13#
10.14#

10.15#

10.16#

10.17#

10.18#

10.19#

10.20#

10.21#
10.22#

10.23#

10.24#

10.25#

10.26#

Description of Document
Amendment No. 1 to Exclusive License Agreement, by 
and between Assembly Biosciences, Inc. and the Indiana 
University Research and Technology Corporation.
Amendment No. 2 to Exclusive License Agreement, by 
and between Assembly Biosciences, Inc. and the Indiana 
University Research and Technology Corporation.
Collaboration Agreement, dated as of July 17, 2020, by 
and between Assembly Biosciences, Inc. and BeiGene, 
Ltd.
 Employment Agreement, dated August 6, 2019, between 
Assembly Biosciences, Inc. and John G. McHutchison, 
A.O., M.D.
 Employment Agreement, dated September 30, 2019, 
between Assembly Biosciences, Inc. and Thomas J. 
Russo, effective as of October 28, 2019.
Amendment No. 1 to Employment Agreement, dated 
February 26, 2020, between Assembly Biosciences, Inc. 
and Thomas J. Russo.
 Employment Agreement, dated October 22, 2019, 
between Assembly Biosciences, Inc. and Luisa M. 
Stamm, M.D., Ph.D. effective as of November 6, 2019.
Amendment No. 1 to Employment Agreement, dated 
February 26, 2020, between Assembly Biosciences, Inc. 
and Luisa M. Stamm, M.D., Ph.D.
 Employment Agreement, dated March 23, 2020, between 
Assembly Biosciences, Inc. and Jason A. Okazaki, 
effective as of March 26, 2020.
 Employment Agreement, dated May 1, 2020, between 
Assembly Biosciences, Inc. and William E. Delaney IV, 
Ph.D., effective as of May 27, 2020.
 2010 Equity Incentive Plan.
 Assembly Biosciences, Inc. Amended and Restated 2014 
Stock Incentive Plan.
Omnibus Amendment to Assembly Biosciences, Inc. 
Stock Incentive Plans.
 Form of Notice of Stock Option Grant and Stock Option 
Agreement under Amended and Restated 2014 Stock 
Incentive Plan.
 Form of Restricted Stock Unit Award Notice and 
Restricted Stock Unit Award Agreement under the 
Amended and Restated 2014 Stock Incentive Plan.
 Assembly Biosciences, Inc. 2017 Inducement Award 
Plan.
 Form of Notice of Stock Option Grant and Stock Option 
Agreement under the 2017 Inducement Award Plan.
 Form of Restricted Stock Unit Award Notice and 
Restricted Stock Unit Award Agreement under the 2017 
Inducement Award Plan.
 Assembly Biosciences, Inc. 2018 Stock Incentive Plan.
Amendment No. 1 to Assembly Biosciences, Inc. 2018 
Stock Incentive Plan.
Amendment No. 3 to Assembly Biosciences, Inc. 2018 
Stock Incentive Plan.
 Form of Notice of Stock Option Grant and Stock Option 
Agreement under the 2018 Stock Incentive Plan.
 Form of Restricted Stock Unit Award Notice and 
Restricted Stock Unit Award Agreement under the 2018 
Stock Incentive Plan.
 Form of Stock Appreciation Right Award Agreement for 
Non-U.S. Grantees under the Assembly Biosciences, Inc. 
2018 Stock Incentive Plan.

Registrant’s
Form
10-Q

Dated
11/05/2020

Exhibit
No.
10.1

Filed
Herewith

X

X

10-Q

11/05/2020

10.2

10-Q

11/05/2020

10.3

10-Q

 11/07/2019 

10.1

10-Q

 11/07/2019 

10.6

10-Q

05/08/2020

10.6

10-K

 03/04/2020 

10.7

10-Q

05/08/2020

10.7

S-1/A
8-K

  10/4/2010   10.14  
  6/6/2016  

10.1

10-Q

05/08/2020

10.2

S-8

  9/17/2014   10.28  

10-Q

 11/01/2017 

10.1

10-Q

 08/09/2017 

10.1

10-Q

 08/09/2017 

10.2

10-Q

 08/09/2017 

10.3

8-K
8-K

8-K

8-K

8-K

  6/1/2018  
05/21/2019

10.1
10.2

06/16/2020

10.1

  6/1/2018  

10.2

  6/1/2018  

10.3

8-K

 10/12/2018 

10.4

57

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
Registrant’s
Form
8-K

Dated
  6/1/2018  

Exhibit
No.
10.4

Filed
Herewith

10-Q

 11/07/2019 

10.4

10-Q

11/07/2019

10.5

10-Q

05/08/2020

10.3

10-Q

05/08/2020

10.4

10-Q

05/08/2020

10.5

8-K

02/11/2020

10.1

X
X

X
X

X

X

X

Exhibit
Number  

Description of Document

10.27#

10.28#

10.29#

10.30#

10.31#

10.32#

10.33#
21.1
23.1

24.1
31.1

31.2

32.1**

32.2**

 Assembly Biosciences, Inc. 2018 Employee Stock 
Purchase Plan.
 Assembly Biosciences, Inc. 2019 Inducement Award 
Plan.
Form of Notice of Stock Option Grant and Stock Option 
Agreement under the 2019 Inducement Award Plan.
Assembly Biosciences, Inc. 2020 Inducement Award 
Plan.
Form of Notice of Stock Option Grant and Stock Option 
Agreement under the 2020 Inducement Award Plan. 
Form of Restricted Stock Unit Award Notice and 
Restricted Stock Unit Award Agreement under the 2020 
Inducement Award Plan.
Assembly Biosciences, Inc. 2020 Corporate Bonus Plan. 
 List of Subsidiaries of Assembly Biosciences, Inc.
 Consent of Independent Registered Public Accounting 
Firm.
 Power of Attorney (included on signature page).
 Certification of the Chief Executive Officer Pursuant to 
Section 302 of the Sarbanes-Oxley Act of 2002.
 Certification of the Chief Financial Officer Pursuant to 
Section 302 of the Sarbanes-Oxley Act of 2002.
 Certification of the Chief Executive Officer Pursuant to 
18 U.S.C. Section 1350 as Adopted Pursuant to Section 
906 of the Sarbanes-Oxley Act of 2002.
 Certification of the Chief Financial Officer Pursuant to 18 
U.S.C. Section 1350 as Adopted Pursuant to Section 906 
of the Sarbanes-Oxley Act of 2002.

101.INS   Inline XBRL Instance Document.
101.SCH  Inline XBRL Taxonomy Extension Schema Document.
101.CAL  Inline XBRL Taxonomy Extension Calculation Linkbase 

Document.

101.DEF  Inline XBRL Taxonomy Extension Definitions Linkbase 

Document.

101.LAB  Inline XBRL Taxonomy Extension Label Linkbase 

Document.

101.PRE  Inline XBRL Taxonomy Extension Presentation Linkbase 

104

Document.
Cover Page Interactive Data File (embedded within the 
Inline XBRL document).

* Certain  information  in  this  exhibit  has  been  omitted  and  filed  separately  with  the  Securities  and  Exchange 

†
‡

Commission pursuant to a confidential treatment request.
The schedules to this exhibit have been omitted pursuant to Item 601(a)(5) of Regulation S-K.
Portions of this exhibit that are both not material and would likely cause competitive harm to the registrant if 
publicly disclosed have been omitted pursuant to Item 601(b)(10)(iv) of Regulation S-K.
Represents management contracts or compensatory plans or arrangements.

#
** The certifications attached as Exhibits 32.1 and 32.2 that accompany this Annual Report on Form 10-K are to 
be deemed furnished and shall not be deemed “filed” with the SEC and are not to be incorporated by reference 
into any filing of Assembly Biosciences, Inc. under the Securities Act of 1933, as amended, or the Securities 
Exchange Act of 1934, as amended, whether made before or after the date of this Annual Report on Form 10-K, 
irrespective of any general incorporation language contained in such filing.

Item 16.  Form 10-K Summary.

None

58

 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
In accordance with Section 13 or 15(d) of the Securities Exchange Act, the Registrant caused this report to be signed 
on its behalf by the undersigned, thereunto duly authorized.

SIGNATURES

Date: February 25, 2021

ASSEMBLY BIOSCIENCES, INC.

/s/ John G. McHutchison, A.O., M.D.

By:
Name:John G. McHutchison, A.O., M.D.
Title: Chief Executive Officer and President

POWER OF ATTORNEY

KNOW ALL PERSONS BY THESE PRESENTS, that each person whose signature appears below constitutes and 
appoints John G. McHutchison, A.O., M.D., Thomas J. Russo, CFA and Jason A. Okazaki, jointly and severally, his 
or  her  attorneys-in-fact,  each  with  the  power  of  substitution,  for  him  or  her  in  any  and  all  capacities,  to  sign  any 
amendments to this report, and to file the same, with exhibits thereto and other documents in connection therewith 
with the Securities and Exchange Commission, hereby ratifying and confirming all that each of said attorneys-in-
fact, or his or her substitute or substitutes may do or cause to be done by virtue hereof.

Pursuant to the requirements of the Securities Exchange Act of 1934, this report has been signed by the following 
persons on behalf of the registrant in the capacities and on the dates indicated.

Signature

Title

/s/ John G. McHutchison, A.O., M.D.  Chief Executive Officer, President and Director
John G. McHutchison, A.O., M.D.

  (Principal Executive Officer)

Date

  February 25, 2021

/s/ Thomas J. Russo, CFA
Thomas J. Russo, CFA

/s/ William R. Ringo, Jr.
William R. Ringo, Jr.

/s/ Anthony E. Altig
Anthony E. Altig

/s/ Gina Consylman
Gina Consylman

/s/ Richard D. DiMarchi, Ph.D.
Richard D. DiMarchi, Ph.D.

/s/ Myron Z. Holubiak
Myron Z. Holubiak

/s/ Susan Mahony, Ph.D.
Susan Mahony, Ph.D.

  Chief Financial Officer
  (Principal Financial and Principal Accounting Officer)

  February 25, 2021

  Chairman of the Board

  February 25, 2021

  February 25, 2021

  February 25, 2021

  February 25, 2021

  February 25, 2021

  February 25, 2021

  Director

  Director

  Director

  Director

  Director

59

 
 
 
 
 
 
 
 
 
 
 
 
 
   
 
 
 
 
 
   
 
 
 
 
 
   
   
 
 
 
 
 
   
   
 
 
 
 
 
   
   
 
 
 
 
 
   
   
 
 
 
 
 
   
   
 
 
 
 
 
   
   
 
 
 
 
[This page intentionally left blank] 

ASSEMBLY BIOSCIENCES, INC.
FINANCIAL STATEMENTS

Reports of Independent Registered Public Accounting Firm.............................................................................

Consolidated Balance Sheets as of December 31, 2020 and 2019.....................................................................

Consolidated Statements of Operations and Comprehensive Loss for the Years Ended December 31, 2020, 
2019 and 2018 ....................................................................................................................................................

Consolidated Statements of Changes in Stockholders’ Equity for the Years Ended December 31, 2020, 2019 
and 2018 .............................................................................................................................................................

Page

F-2

F-7

F-8

F-9

Consolidated Statements of Cash Flows for the Years Ended December 31, 2020, 2019 and 2018.................

F-10

Notes to Consolidated Financial Statements ......................................................................................................

F-11

F-1

Report of Independent Registered Public Accounting Firm

To the Stockholders and the Board of Directors of Assembly Biosciences, Inc.

Opinion on the Financial Statements

We have audited the accompanying consolidated balance sheets of Assembly Biosciences, Inc. (the Company) as of 
December 31, 2020 and 2019, the related consolidated statements of operations and comprehensive loss, changes in 
stockholders’  equity  and  cash  flows  for  each  of  the  three  years  in  the  period  ended  December  31,  2020,  and  the 
related  notes  (collectively  referred  to  as  the  “consolidated  financial  statements”).  In  our  opinion,  the  consolidated 
financial statements present fairly, in all material respects, the financial position of the Company at December 31, 
2020 and 2019, and the results of its operations and its cash flows for each of the three years in the period ended 
December 31, 2020, in conformity with U.S. generally accepted accounting principles. 

We also have audited, in accordance with the standards of the Public Company Accounting Oversight Board (United 
States)  (PCAOB),  the  Company's  internal  control  over  financial  reporting  as  of  December  31,  2020,  based  on 
criteria  established  in  Internal  Control—Integrated  Framework  issued  by  the  Committee  of  Sponsoring 
Organizations of the Treadway Commission (2013 Framework) and our report dated February 25, 2021 expressed 
an unqualified opinion thereon.

Basis for Opinion

These financial statements are the responsibility of the Company’s management. Our responsibility is to express an 
opinion on the Company’s financial statements based on our audits. We are a public accounting firm registered with 
the  PCAOB  and  are  required  to  be  independent  with  respect  to  the  Company  in  accordance  with  the  U.S.  federal 
securities  laws  and  the  applicable  rules  and  regulations  of  the  Securities  and  Exchange  Commission  and  the 
PCAOB. 

We conducted our audits in accordance with the standards of the PCAOB. Those standards require that we plan and 
perform  the  audit  to  obtain  reasonable  assurance  about  whether  the  financial  statements  are  free  of  material 
misstatement,  whether  due  to  error  or  fraud.  Our  audits  included  performing  procedures  to  assess  the  risks  of 
material  misstatement  of  the  financial  statements,  whether  due  to  error  or  fraud,  and  performing  procedures  that 
respond  to  those  risks.  Such  procedures  included  examining,  on  a  test  basis,  evidence  regarding  the  amounts  and 
disclosures  in  the  financial  statements.  Our  audits  also  included  evaluating  the  accounting  principles  used  and 
significant estimates made by management, as well as evaluating the overall presentation of the financial statements. 
We believe that our audits provide a reasonable basis for our opinion. 

Critical Audit Matters 

The  critical  audit  matters  communicated  below  are  matters  arising  from  the  current  period  audit  of  the  financial 
statements that were communicated or required to be communicated to the audit committee and that: (1) relate to 
accounts  or  disclosures  that  are  material  to  the  financial  statements  and  (2)  involved  our  especially  challenging, 
subjective or complex judgments. The communication of critical audit matters does not alter in any way our opinion 
on  the  consolidated  financial  statements,  taken  as  a  whole,  and  we  are  not,  by  communicating  the  critical  audit 
matters below, providing separate opinions on the critical audit matters or on the accounts or disclosures to which 
they relate.

F-2

Description of 
the Matter

Accrued clinical trial expenses
For  the  year  ended  December  31,  2020,  the  Company  incurred  $106.8  million  of  research  and 
development expenses and recorded $4.4 million for accrued clinical trial expenses at December 
31,  2020.  As  described  in  Note  2  to  the  consolidated  financial  statements,  the  Company’s 
expense  accruals  for  clinical  trials  are  based  on  estimates  of  the  services  received  and  efforts 
expended  pursuant  to  contracts  with  multiple  contract  research  organizations  (CROs)  and 
manufacturing vendors that conduct and manage these activities on its behalf. When billing terms 
under such contracts do not coincide with the timing of when the work is performed, management 
is  required  to  make  estimates  of  outstanding  obligations  to  those  third  parties  as  of  period  end. 
The accrual is based on a number of factors, including the time period over which services will be 
performed,  enrollment  of  subjects,  number  of  sites  activated,  and  the  level  of  effort  to  be 
expended in each period. At period end, accrued clinical trial expenses are recorded based upon 
estimates of the proportion of work completed over the  term of the  individual  clinical trial and 
manufacturing activities in accordance with signed agreements with the third parties. If possible, 
the  Company  obtains  information  regarding  unbilled  services  directly  from  these  service 
providers  and  performs  procedures  to  challenge  these  estimates  based  on  their  internal 
understanding of the services provided to date. However, the Company may also be required to 
estimate  these  services  based  on  information  available  to  its  internal  clinical  or  administrative 
staff if such information is not able to be obtained timely from its services providers.

Auditing  accrued  clinical  trial  expenses  is  complex  because  of  the  judgments  applied  by 
management to determine the commencement and completion date of vendor tasks and the cost 
and extent of work performed during the reporting period for services not yet billed by contracted 
third-party  vendors.  The  testing  of  the  Company’s  accrued  clinical  trial  expense  models  also 
involves  a  high  level  of  effort  to  test  the  high  volume  of  data  used  to  determine  the  estimated 
accrual.

How We 
Addressed the 
Matter in Our 
Audit

We  obtained  an  understanding,  evaluated  the  design  and  tested  the  operating  effectiveness  of 
controls over the Company’s process for estimating the accrued clinical trial expenses including 
controls  over  management’s  assessment  and  measurement  of  clinical  trial  progress  and  related 
estimates  of  accrued  clinical  trial  costs  and  the  completeness  and  accuracy  of  underlying  data 
used in the analysis.

To  test  the  estimate  of  accrued  clinical  trial  expenses,  we  performed  audit  procedures  that 
included, among others, direct confirmation of contract terms and conditions with a sample of the 
Company’s third-party vendors. We also confirmed the progress of contracted clinical activities 
with these third-party vendors and compared such data to the Company’s estimates of progress as 
reflected  in  their  accrual  models.  We  further  tested  the  accuracy  of  the  calculations,  the 
completeness  of  the  data  utilized,  and  the  reasonableness  of  the  assumptions  used  in 
management’s  accrual  models  by  testing  actual  invoices  paid  to  date,  agreeing  inputs  back  to 
contractual  terms  and  holding  discussions  with  clinical  or  administrative  staff  outside  of  the 
finance  function.  Procedures  were  performed  to  evaluate  the  reliability,  completeness  and 
relevance  of  management’s  data  by  testing  actual  invoices  paid  and  holding  discussions  with 
clinical  or  administrative  staff  outside  of  the  finance  function  to  corroborate  progress  and 
estimated  level  of  expended  effort  incurred  by  the  Company’s  third-party  vendors.  Further,  we 
inspected material invoices received from third parties after the balance sheet date and evaluated 
whether  services  performed  prior  to  the  consolidated  balance  sheet  date  had  been  properly 
included in the accrual.

F-3

Description of 
the Matter

How We 
Addressed the 
Matter in Our 
Audit

Revenue Recognition for the Collaborative Arrangement with BeiGene, Ltd.
As  described  in  Note  9  to  the  consolidated  financial  statements,  in  July  2020,  the  Company 
entered  into  a  collaboration  agreement  with  BeiGene,  Ltd.  (BeiGene)  to  develop  and 
commercialize the Company’s product candidates in China for the treatment of chronic Hepatitis 
B  virus  infection  (the  BeiGene  Agreement).  The  BeiGene  Agreement  includes  up-front  fees, 
milestones,  royalties,  expense  reimbursement,  and  potential  cost  share  and  profit  sharing. 
Management  was  required  to  use  judgment  to  determine  what  part  of  the  BeiGene  Agreement 
was within the scope of the contract with customers guidance and what part of the agreement was 
within  the  scope  of  the  collaborative  arrangement  guidance.  For  the  year  ended  December  31, 
2020, the Company recognized $31.0 million as collaboration revenue and $9.0 million of long-
term deferred revenue from the BeiGene Agreement. 

Auditing  the  Company’s  accounting  for  revenues  from  its  BeiGene  Agreement  was  especially 
challenging  due  to  the  complex  and  highly  judgmental  nature  of  evaluating  the  terms  of  the 
agreement, evaluating whether analogies to the revenue accounting or collaborative arrangements 
guidance are appropriate, and allocating the transaction price to the performance obligations.

We  obtained  an  understanding,  evaluated  the  design  and  tested  the  operating  effectiveness  of 
controls over management’s assessment of the accounting treatment of the BeiGene Agreement 
and identification of performance obligations and application of the accounting guidance. 

To  test  the  accounting  for  revenue  from  the  BeiGene  Agreement,  among  other  procedures,  we 
tested and evaluated, the performance obligations identified and the allocation of transaction price 
to performance obligations. We also assessed whether management’s evaluation of the portions 
of  the  BeiGene  Agreement  subject  to  the  scope  of  the  contract  with  customers  accounting 
standard  and  collaborative  arrangements  accounting  standard,  as  well  as  their  analogies  to  the 
revenue  from  contracts  with  customers  accounting  standard  or  the  portion  of  the  BeiGene 
Agreement subject to the collaborative arrangements guidance, was an appropriate application of 
an accounting policy.  

/s/ Ernst & Young LLP
We have served as the Company’s auditor since 2015.

Redwood City, California
February 25, 2021

F-4

Report of Independent Registered Public Accounting Firm

To the Stockholders and the Board of Directors of Assembly Biosciences, Inc.

Opinion on Internal Control over Financial Reporting 

We have audited Assembly Biosciences, Inc.’s internal control over financial reporting as of December 31, 2020, 
based  on  criteria  established  in  Internal  Control—Integrated  Framework  issued  by  the  Committee  of  Sponsoring 
Organizations  of  the  Treadway  Commission  (2013  framework)  (the  COSO  criteria).  In  our  opinion,  Assembly 
Biosciences,  Inc.  (the  Company)  maintained,  in  all  material  respects,  effective  internal  control  over  financial 
reporting as of December 31, 2020, based on the COSO criteria. 

We also have audited, in accordance with the standards of the Public Company Accounting Oversight Board (United 
States) (PCAOB), the consolidated balance sheets of the Company as of December 31, 2020 and 2019, the related 
consolidated statements of operations and comprehensive loss, changes in stockholders’ equity and cash flows for 
each of the three years in the period ended December 31, 2020, and the related notes and our report dated February 
25, 2021 expressed an unqualified opinion thereon. 

Basis for Opinion 

The  Company’s  management  is  responsible  for  maintaining  effective  internal  control  over  financial  reporting  and 
for  its  assessment  of  the  effectiveness  of  internal  control  over  financial  reporting  included  in  the  accompanying 
Management's  Annual  Report  on  Internal  Control  Over  Financial  Reporting.  Our  responsibility  is  to  express  an 
opinion on the Company’s internal control over financial reporting based on our audit. We are a public accounting 
firm registered with the PCAOB and are required to be independent with respect to the Company in accordance with 
the U.S. federal securities laws and the applicable rules and regulations of the Securities and Exchange Commission 
and the PCAOB. 

We conducted our audit in accordance with the standards of the PCAOB. Those standards require that we plan and 
perform  the  audit  to  obtain  reasonable  assurance  about  whether  effective  internal  control  over  financial  reporting 
was maintained in all material respects. 

Our audit included obtaining an understanding of internal control over financial reporting, assessing the risk that a 
material weakness exists, testing and evaluating the design and operating effectiveness of internal control based on 
the  assessed  risk,  and  performing  such  other  procedures  as  we  considered  necessary  in  the  circumstances.  We 
believe that our audit provides a reasonable basis for our opinion. 

Definition and Limitations of Internal Control Over Financial Reporting 

A  company’s  internal  control  over  financial  reporting  is  a  process  designed  to  provide  reasonable  assurance 
regarding  the  reliability  of  financial  reporting  and  the  preparation  of  financial  statements  for  external  purposes  in 
accordance  with  generally  accepted  accounting  principles.  A  company’s  internal  control  over  financial  reporting 
includes  those  policies  and  procedures  that  (1)  pertain  to  the  maintenance  of  records  that,  in  reasonable  detail, 
accurately and fairly reflect the transactions and dispositions of the assets of the company; (2) provide reasonable 
assurance  that  transactions  are  recorded  as  necessary  to  permit  preparation  of  financial  statements  in  accordance 
with  generally  accepted  accounting  principles,  and  that  receipts  and  expenditures  of  the  company  are  being  made 
only  in  accordance  with  authorizations  of  management  and  directors  of  the  company;  and  (3)  provide  reasonable 
assurance regarding prevention or timely detection of unauthorized acquisition, use, or disposition of the company’s 
assets that could have a material effect on the financial statements. 

F-5

Because of its inherent limitations, internal control over financial reporting may not prevent or detect misstatements. 
Also, projections of any evaluation of effectiveness to future periods are subject to the risk that controls may become 
inadequate because of changes in conditions, or that the degree of compliance with the policies or procedures may 
deteriorate. 

/s/ Ernst & Young LLP

Redwood City, California
February 25, 2021

F-6

ASSEMBLY BIOSCIENCES, INC.
CONSOLIDATED BALANCE SHEETS
(In thousands except for share amounts and par value)

ASSETS
Current assets

Cash and cash equivalents .............................................................................  $
Marketable securities .....................................................................................   
Accounts receivable from collaborations ......................................................   
Prepaid expenses and other current assets .....................................................   
Total current assets..............................................................................................   

Property and equipment, net..........................................................................   
Operating lease right-of-use (ROU) assets ....................................................   
Other assets....................................................................................................   
Indefinite-lived intangible asset.....................................................................   
Goodwill ........................................................................................................   
Total assets.........................................................................................................  $

LIABILITIES AND STOCKHOLDERS' EQUITY
Current liabilities

Accounts payable...........................................................................................  $
Accrued clinical expenses .............................................................................   
Other accrued expenses .................................................................................   
Deferred revenue - short-term .......................................................................   
Operating lease liabilities - short-term ..........................................................   
Total current liabilities ........................................................................................   

Deferred tax liabilities ...................................................................................   
Deferred revenue - long-term ........................................................................   
Operating lease liabilities - long-term ...........................................................   
Total liabilities ...................................................................................................   

Commitments and contingencies

Stockholders' equity

As of December 31,

2020

2019

59,444    $
156,969     
1,230     
6,850     
224,493     

1,600     
9,131     
6,392     
29,000     
12,638     
283,254    $

4,598    $
4,444     
11,987     
—     
3,404     
24,433     

2,531     
8,987     
6,725     
42,676     

46,732 
227,311 
3,374 
5,363 
282,780 

1,830 
11,975 
1,684 
29,000 
12,638 
339,907 

1,731 
4,826 
8,286 
6,411 
3,186 
24,440 

2,531 
30,637 
9,082 
66,690 

Preferred stock, $0.001 par value; 5,000,000 shares authorized; no shares 
issued or outstanding .....................................................................................   
Common stock, $0.001 par value; 100,000,000 shares authorized as of 
December 31, 2020 and 2019; 34,026,680 and 32,558,307 shares issued 
and outstanding as of December 31, 2020 and 2019, respectively................   
Additional paid-in capital ..............................................................................   
Accumulated other comprehensive loss ........................................................   
Accumulated deficit.......................................................................................   
Total stockholders' equity..............................................................................   
Total liabilities and stockholders' equity ........................................................  $

—     

— 

34     
742,387     
(270)    
(501,573)    
240,578     
283,254    $

32 
712,807 
(201)
(439,421)
273,217 
339,907  

See Accompanying Notes to the Consolidated Financial Statements 

F-7

 
 
 
 
 
   
 
     
       
 
     
       
 
 
   
      
  
 
     
       
 
     
       
 
     
       
 
 
   
      
  
 
     
       
 
     
       
 
 
     
       
 
     
       
 
ASSEMBLY BIOSCIENCES, INC. 
CONSOLIDATED STATEMENTS OF OPERATIONS AND COMPREHENSIVE LOSS 
(In thousands except for share and per share amounts)

Year ended December 31,
2019

2018

2020

Collaboration revenue ....................................................................  $

79,105    $

15,963    $

14,804 

Operating expenses:

Research and development ..........................................................   
General and administrative ..........................................................   
Total operating expenses...................................................................   
Loss from operations ......................................................................   

106,823     
37,058     
143,881     
(64,776)    

85,757     
32,919     
118,676     
(102,713)    

72,741 
34,798 
107,539 
(92,735)

Other income

Interest and other income ............................................................   
Total other income ............................................................................   
Loss before income taxes ................................................................   

2,624     
2,624     
(62,152)    

4,305     
4,305     
(98,408)    

3,083 
3,083 
(89,652)

Income tax benefit (expense) ............................................................   
Net loss .............................................................................................  $

—     
(62,152)   $

774     
(97,634)   $

(1,099)
(90,751)

Other comprehensive income

Unrealized gain (loss) on marketable securities, net of tax .........   
Comprehensive loss.........................................................................  $

(69)    
(62,221)   $

146     
(97,488)   $

45 
(90,706)

Net loss per share, basic and diluted .................................................  $
Weighted average common shares outstanding, basic
and diluted.........................................................................................    35,427,120      26,258,790      22,801,644  

(3.72)   $

(1.75)   $

(3.98)

See Accompanying Notes to the Consolidated Financial Statements 

F-8

 
 
 
 
 
   
   
 
 
   
      
      
  
   
      
      
  
 
   
      
      
  
   
      
      
  
 
   
      
      
  
 
   
      
      
  
   
      
      
  
 
   
      
      
  
ASSEMBLY BIOSCIENCES, INC. 
CONSOLIDATED STATEMENTS OF CHANGES IN STOCKHOLDERS’ EQUITY 
(In thousands except for share amounts)

Balance as of December 31, 2017 .............
Sale of common stock, net of
underwriters' discount and costs..................
Issuance of common stock upon
exercise of stock options .............................
Issuance of common stock under
Employee Stock Purchase Plan (ESPP) ......
Issuance of shares of common stock for
settlement of restricted stock units
(RSUs) .........................................................
Unrealized gain on marketable securities,
net of tax ......................................................
Stock-based compensation ..........................
Net loss ........................................................
Balance as of December 31, 2018 .............
Sale of common stock and pre-funded
warrants, net of underwriters' discount
and costs ......................................................
Issuance of common stock upon exercise
of stock options............................................
Settlement of RSUs for cash........................
Issuance of common stock under ESPP ......
Issuance of shares of common stock for
settlement of RSUs ......................................
Unrealized gain on marketable securities,
net of tax ......................................................
Stock-based compensation ..........................
Net loss ........................................................
Balance as of December 31, 2019 .............
Sale of common stock, net of
commissions and fees ..................................
Issuance of common stock upon
exercise of stock options .............................
Issuance of common stock under
ESPP ............................................................
Issuance of shares of common stock for
settlement of RSUs ......................................
Unrealized loss on marketable
securities ......................................................
Stock-based compensation ..........................
Net loss ........................................................
Balance as of December 31, 2020 .............

Additional

Accumulated
Other

  Common Stock   
  Shares
  20,137,974  $

20  $ 364,528   $

Paid-in    

Comprehensive   Accumulated   

  Amount    Capital

Loss

    Deficit

Total
Stockholders' 
Equity

(392) $

(251,036) $

113,120 

—    

—    

—    

—    

155,425 

—    

—    

3,960 

408 

   4,600,000   

4   

155,421    

735,030   

1   

3,959    

21,483   

—   

408    

938   

—   

—    

—    

—    

— 

—   
—   
—   
  25,495,425  $

—   
—    
—   
28,446    
—    
—   
25  $ 552,762   $

45    
—    
—    
(347) $

—    
—    
(90,751)  
(341,787) $

45 
28,446 
(90,751)
210,653 

   6,287,878   

6   

134,655    

585,292   
—   
59,370   

130,342   

1   
—   
—   

—   

4,237    
(4)  
747    

—    

—    

—    
—    
—    

—    

—    

134,661 

—    
—    
—    

—    

4,238 
(4)
747 

— 

—   
—   
—   
  32,558,307  $

—   
—    
—   
20,410    
—    
—   
32  $ 712,807   $

146    
—    
—    
(201) $

—    
—    
(97,634)  
(439,421) $

146 
20,410 
(97,634)
273,217 

892,840   

175,579   

86,812   

313,142   

1   

1   

—   

—   

5,451    

1,466    

680    

—    

—    

—    

—    

—    

—    

—    

—    

—    

5,452 

1,467 

680 

— 

—   
—   
—   
  34,026,680  $

—    
—   
21,983    
—   
—    
—   
34  $ 742,387   $

(69)  
—    
—    
(270) $

—    
—    
(62,152)  
(501,573) $

(69)
21,983 
(62,152)
240,578  

See Accompanying Notes to the Consolidated Financial Statements

F-9

 
 
   
   
 
  
  
  
  
  
  
  
  
  
  
  
  
  
  
  
  
  
  
  
  
ASSEMBLY BIOSCIENCES, INC. 
CONSOLIDATED STATEMENTS OF CASH FLOWS
(In thousands)

Cash flows from operating activities
Net loss ...................................................................................................   $
Adjustments to reconcile net loss to net cash used in operating 
activities:

Depreciation and amortization ..........................................................
Non-cash IPR&D expense ................................................................
Stock-based compensation................................................................
Net accretion and amortization of investments in marketable
securities ...........................................................................................
Non-cash rent expense ......................................................................
Deferred income tax (benefit) expense .............................................
Loss on disposal of fixed assets ........................................................
Other .................................................................................................
Changes in operating assets and liabilities:

Accounts receivable from collaborations....................................
Prepaid expenses and other current assets...................................
Other assets .................................................................................
Accounts payable ........................................................................
Accrued clinical expenses ...........................................................
Other accrued expenses...............................................................
Deferred revenue .........................................................................
Deferred rent ...............................................................................
Operating lease liabilities ............................................................
Net cash used in operating activities ......................................................  

Year Ended December 31,
2019

2018

2020

(62,152)   $

(97,634)   $

(90,751)

691     
1,750     
21,853     

(13)    
5,214     
—     
9     
—     

2,144     
(1,487)    
(4,708)    
2,867     
(382)    
3,831     
(28,061)    
—     
(4,513)    
(62,957)    

494     
— 
20,558     

(1,735)    
4,454     
(774)    
102     
(5)    

(944)    
(3,685)    
1,664     
(1,962)    
1,265     
2,016     
(3,612)    
—     
(4,269)    
(84,067)    

643 
— 
28,485 

(229)
— 
1,099 
— 
— 

(156)
(1,094)
(3,008)
1,569 
3,119 
382 
(5,125)
108 
— 
(64,958)

Cash flows from investing activities

Purchases of property and equipment .........................................
Purchase of IPR&D.....................................................................
Purchases of marketable securities..............................................
Proceeds from maturities of marketable securities .....................
Proceeds from sale of marketable securities ...............................
Net cash provided by (used in) investing activities ................................  

(470)    
(1,750)    
(193,188)    
221,617     
41,861     
68,070     

(1,554)    
—     
(281,334)    
203,911     
28,659     
(50,318)    

(340)
— 
(183,941)
48,884 
— 
(135,397)

Cash flows from financing activities

Proceeds from common stock and pre-funded warrants sold,
net of underwriters' discount, commissions and costs ................  
Proceeds from the issuance of common stock under ESPP ........  
Proceeds from the exercise of stock options ...............................
Net cash provided by financing activities...............................................  

Net increase (decrease) in cash and cash equivalents.............................  
Cash and cash equivalents at the beginning of the period ......................  
Cash and cash equivalents at the end of the period...........................   $
Supplemental non-cash investing and financing activities
Operating lease liabilities arising from obtaining right-of-use assets ....   $

5,452     
680     
1,467     
7,599     

134,661     
747     
4,238     
139,646     

12,712     
46,732     
59,444    $

5,261     
41,471     
46,732    $

155,425 
408 
3,960 
159,793 

(40,562)
82,033 
41,471 

1,302    $

15,261    $

—  

See Accompanying Notes to the Consolidated Financial Statements

F-10

 
 
 
 
 
   
   
 
 
 
      
      
  
 
 
      
      
  
  
  
  
  
  
  
  
  
  
  
      
      
  
  
  
  
  
  
  
  
  
  
 
 
 
 
      
      
  
 
 
      
      
  
  
  
  
  
  
 
 
 
 
      
      
  
 
 
      
      
  
 
 
  
 
 
 
 
      
      
  
 
 
 
 
      
      
  
ASSEMBLY BIOSCIENCES, INC. 
Notes to Consolidated Financial Statements

Note 1 - Nature of Business

Overview

Assembly Biosciences, Inc., together with its subsidiaries (Assembly or the Company), incorporated in Delaware in 
October 2005, is a clinical-stage biotechnology company advancing a novel class of oral therapeutic candidates for 
the treatment of hepatitis B virus (HBV) infection. The Company operates in one segment and is headquartered in 
South San Francisco, California with operations in California, Connecticut and China. 

The  Company’s  research  and  development  programs  are  pursuing  multiple  drug  candidates  that  inhibit  the  HBV 
replication cycle and block the generation of covalently closed circular DNA (cccDNA), with the aim of discovering 
and developing finite and curative therapies for patients with HBV. Assembly has discovered multiple novel core 
inhibitors, which are small molecules that directly target and allosterically modify the HBV core (HBc) protein.

In December 2020, the Company and its Board of Directors approved a plan to wind down its Microbiome program 
in order to prioritize and focus its resources entirely on discovering and developing finite and curative therapies for 
HBV. The Microbiome program had been developing a novel class of oral live microbial biotherapeutics candidates 
designed to treat disorders associated with the microbiome.

Liquidity

The Company has not derived any revenue from product sales to date and currently has no approved products. Once 
a product has been developed, it will need to be approved for sale by the U.S. Food and Drug Administration (FDA) 
or an applicable foreign regulatory agency. Since inception, the Company’s operations have been financed primarily 
through the sale of equity securities, the proceeds from the exercise of warrants and stock options, the issuance of 
debt, and upfront payments related to collaboration agreements. The Company has incurred losses from operations 
since  inception  and  expects  to  continue  to  incur  substantial  losses  for  the  next  several  years  as  it  continues  its 
product development efforts. Management believes the Company currently has sufficient funds to meet its operating 
requirements for at least the next twelve months following the date that these consolidated financial statements are 
issued.  If  the  Company  cannot  generate  significant  cash  from  its  operations,  it  intends  to  obtain  any  additional 
funding  it  requires  through  strategic  relationships,  public  or  private  equity  or  debt  financings,  grants  or  other 
arrangements (see  Note  7  for  recent  sales  of  common  stock).  The  Company  cannot  assure  such  funding  will  be 
available on reasonable terms, if at all. Market volatility resulting from the novel coronavirus disease (COVID-19) 
pandemic or other factors could also adversely impact the Company’s ability to access capital when and as needed.

If the Company is unable to generate enough revenue from its collaborations, secure additional sources of funding or 
receive  full  and  timely  collections  of  amounts  due,  it  may  be  necessary  to  significantly  reduce  the  current  rate  of 
spending  through  reductions  in  staff  and  delaying,  scaling  back,  or  stopping  certain  research  and  development 
programs, including more costly clinical trials.

F-11

Note 2 - Summary of Significant Accounting Policies and Recent Accounting Pronouncements

Basis of Presentation

These  consolidated  financial  statements  have  been  prepared  in  accordance  with  accounting  principles  generally 
accepted  in  the  United  States  (U.S.  GAAP)  and  include  the  accounts  of  the  Company  and  its  wholly  owned 
subsidiaries. All intercompany balances and transactions have been eliminated in consolidation.

Use of Estimates

The preparation of consolidated financial statements in conformity with the accounting principles generally accepted 
in  the  United  States  of  America  (U.S.  GAAP)  requires  management  to  make  estimates  and  assumptions  that  may 
affect the reported amounts of assets and liabilities and disclosure of contingent assets and liabilities at the date of 
the financial statements and reported amounts of expenses during the reporting period. Actual results could differ 
from those estimates.

Significant  estimates  inherent  in  the  preparation  of  the  accompanying  consolidated  financial  statements  include 
estimates  for  the  cost-based  input  of  revenue  recognition  and  standalone  selling  price  estimates  for  allocation  of 
transaction price to performance obligations revenue recognition, estimates of costs incurred but not yet invoiced for 
clinical  trial  accruals,  recoverability  and  useful  lives  of  our  long-lived  assets,  the  estimated  fair  value  of  our 
indefinite-lived intangible assets, the estimated fair value of our reporting unit for purposes of evaluating goodwill 
impairment,  provisions  for  income  taxes,  amounts  receivable  under  collaboration  agreements,  measurement  of 
operating  lease  liabilities,  and  the  fair  value  of  stock  options, stock  appreciation  rights,  and  RSUs  granted  to 
employees, directors, and consultants.

The  Company’s  estimates  could  be  affected  by  external  conditions,  including  those  unique  to  the  Company  and 
general  economic  conditions.  It  is  reasonably  possible  that  these  external  factors  could  have  an  effect  on  the 
Company’s estimates and could cause actual results to differ from those estimates and assumptions.

Other Risks and Uncertainties

In  March  2020,  the  World  Health  Organization  declared  the  COVID-19  outbreak  a  pandemic.  To  date,  the 
Company’s operations have not been significantly impacted by the COVID-19 pandemic. However, the Company 
cannot  at  this  time  predict  the  specific  extent,  duration,  or  full  impact  the  COVID-19  pandemic  will  have  on  its 
business, operations, strategy, prospects and financial condition and results. The impact of the COVID-19 pandemic 
on the Company’s financial performance will depend on future developments, including the duration and spread of 
the  outbreak  and  related  governmental  advisories  and  restrictions.  These  developments  and  the  impact  of  the 
COVID-19 pandemic on the financial markets and the overall economy are highly uncertain. If the financial markets 
and/or the overall economy are impacted for an extended period, the Company’s results may be adversely affected.

Cash and Cash Equivalents

All highly liquid investments, including money market funds, with original maturities of three months or less at the 
time of purchase are considered to be cash equivalents.  All of the Company’s cash equivalents have liquid markets 
and high credit ratings.  The Company maintains its cash in bank deposits and other accounts, the balances of which, 
at times and at December 31, 2020 and 2019, exceed federally insured limits.

Investments in Marketable Securities

The Company invests its excess cash in debt securities with high credit ratings including but not limited to money 
market funds classified as cash equivalents, asset backed securities, securities issued by the U.S. government and its 
agencies,  corporate  debt  securities  and  commercial  paper.  The  Company  has  designated  its  investments  in 
marketable securities as available-for-sale and measures these securities at their respective fair values. Marketable 
securities are classified as short-term or long-term based on the maturity date and their availability to meet current 
operating requirements. Marketable securities that mature in one year or less are classified as short-term available-
for-sale securities and are reported as a component of current assets.

F-12

Securities  that  are  classified  as  available-for-sale  are  measured  at  fair  value  with  temporary  unrealized  gains  and 
losses reported in other comprehensive loss, and as a component of stockholders' equity until their disposition. The 
Company reviews all available-for-sale securities at each period end to determine if they remain available-for-sale 
based on their current intent and ability to sell the security if it is required to do so. Realized gains and losses from 
the sale of marketable securities, if any, are calculated using the specific-identification method.

Marketable  securities  are  subject  to  a  periodic  impairment  review.  The  Company  may  recognize  an  impairment 
charge when a decline in the fair value of investments below the cost basis is determined to be other-than-temporary. 
In determining whether a decline in market value is other-than-temporary, various factors are considered, including 
the cause, duration of time and severity of the impairment, any adverse changes in the investees’ financial condition, 
and the Company’s intent and ability to hold the security for a period of time sufficient to allow for an anticipated 
recovery in market value. To date, there have been no declines in value deemed to be other than temporary for any 
of our investments in marketable securities.

Goodwill and Indefinite-Lived Intangible Asset

Goodwill and indefinite-lived intangible assets are reviewed for impairment at least annually in the fourth quarter, 
and more frequently if events or other changes in circumstances indicate that the carrying amount of the assets may 
not  be  recoverable.  Impairment  of  goodwill  and  indefinite-lived  intangibles  is  determined  to  exist  when  the  fair 
value is less than the carrying value of the net assets being tested.

Goodwill

The difference between the purchase price and the fair value of assets acquired and liabilities assumed in a business 
combination is allocated to goodwill. Goodwill is evaluated for impairment on an annual basis as of October 1, and 
more  frequently  if  indicators  are  present  or  changes  in  circumstances  suggest  that  impairment  may  exist.  In 
performing each annual impairment assessment and any interim impairment assessment, the Company determines if 
it should qualitatively assess whether it is more likely than not that the fair value of goodwill is less than its carrying 
amount (the qualitative impairment test). If the Company concludes it is more likely than not that the fair value of 
the reporting unit is less than its carrying amount, or elect not to use the qualitative impairment test, a quantitative 
impairment  test  is  performed  The  Company  annual  or  interim  quantitative  impairment  testing  is  performed  by 
comparing the estimated fair value of the reporting unit to its carrying value. An impairment charge is recognized 
for  the  amount  by  which  the  carrying  amount  exceeds  the  reporting  unit’s  fair  value,  not  to  exceed  the  carrying 
value of goodwill.

As of October 1, 2020 the Company has determined through its quantitative impairment test that the fair value of its 
goodwill significantly exceeded the carrying value of its single reporting unit and concluded that goodwill was not 
impaired.  In  November  2020,  after  the  Company’s  public  announcement  that  it  became  clear  that  patients  who 
stopped therapy in Study 211 had not achieved meaningful sustained virologic response rates most of the patients 
had relapsed, the Company’s stock price declined significantly. Due to a sustained decline in the Company’s stock 
price during the remainder of the fourth quarter of 2020, the Company determined these factors were an indication 
of  a  triggering  event  of  impairment  and  an  interim  goodwill  impairment  test  was  performed  as  of  December  31, 
2020. However, the interim quantitative impairment test still determined the fair value, when considering a control 
premium  based  on  a  range  of  recent  acquisitions  of  entities  similar  to  the  Company  which  were  made  on  a  non-
minority  basis,  exceeded  the  carrying  value  of  its  single  reporting  unit,  and  concluded  that  goodwill  was  still  not 
impaired. The Company has not recognized any goodwill impairment in any of the periods presented.

Indefinite-Lived Intangible Asset

The Company’s indefinite-lived intangible asset consists of IPR&D acquired in a business combination that are used 
in research and development activities but have not yet reached technological feasibility, regardless of whether they 
have alternative future use. The primary basis for determining the technological feasibility or completion of these 
projects is obtaining regulatory approval to market the underlying products in an applicable geographic region. The 
Company  classifies  IPR&D  acquired  in  a  business  combination  as  an  indefinite-lived  intangible  asset  until  the 
completion or abandonment of the associated research and development efforts. Upon completion of the associated 
research and development efforts, the Company performed a final test for impairment and will determine the useful 
life of the technology and begin amortizing the assets to reflect their use over their remaining lives. Upon permanent 

F-13

abandonment,  the  Company  would  write-off  the  remaining  carrying  amount  of  the  associated  IPR&D  intangible 
asset.

Indefinite-lived  intangible  assets  are  not  amortized,  but  instead  are  reviewed  for  impairment  at  least  annually,  or 
more frequently if events occur or circumstances change that would indicate the carrying amount may be impaired. 
In performing each annual impairment assessment and any interim impairment assessment, the Company determines 
if it should qualitatively assess whether it is more likely than not that the fair value of its IPR&D asset is less than its 
carrying  amount  (the  qualitative  impairment  test).  If  the  Company  concludes  that  is  the  case,  or  elect  not  to  use 
qualitative  impairment  test,  the  Company  would  proceed  with  quantitatively  determining  the  fair  value  of  the 
IPR&D asset and comparing its fair value to its carrying value to determine the amount of impairment, if any (the 
quantitative impairment test).

When performing the quantitative impairment assessment, the Company uses the income approach to determine the 
fair value of its IPR&D asset. This approach calculates fair value by estimating the after-tax cash flows attributable 
to an in-process project over its useful life and then discounting these after-tax cash flows back to a present value. 
This  estimate  includes  judgmental  assumptions  regarding  the  estimates  that  market  participants  would  make  in 
evaluating  the  IPR&D  asset,  including  the  probability  of  successfully  completing  clinical  trials  and  obtaining 
regulatory approval to market the IPR&D asset, the timing of and the expected costs to complete IPR&D projects, 
future net cash flows from potential drug sales, which are based on estimates of the sales price of the drug, the size 
of the patient population and cure rate, our competitive position in the marketplace, and appropriate discount and tax 
rates. Any impairment to be recorded is calculated as the difference between the fair value of the IPR&D asset as of 
the date of the assessment with the carrying value of the IPR&D asset on its consolidated balance sheet.

In  performing  the  qualitative  impairment  test,  the  Company  considers  the  results  of  the  most  recent  quantitative 
impairment  test  and  identifies  the  most  relevant  drivers  of  the  fair  value  for  the  IPR&D  asset.  The  most  relevant 
drivers of fair value identified are consistent with the assumptions used in the quantitative estimate of the IPR&D 
asset discussed below. Using these drivers of fair value, the Company identifies events and circumstances that may 
have an effect on the fair value of the IPR&D asset since the last time the IPR&D’s fair value was quantitatively 
determined. The Company then weighs these factors to determine and conclude if it is not more likely than not that 
the IPR&D asset is impaired. If it is more likely than not that the IPR&D asset is impaired, the Company proceeds 
with quantitatively determining the fair value of the IPR&D asset.

For  the  Company’s  2020  impairment  test,  the  Company  performed  a  qualitative  test  and  concluded  it  was  more-
likely-than-not that the fair value of its IPR&D asset exceeded its carrying value and no further testing was required. 
This  was  based  on  a  decrease  in  the  probability  of  success  based  on  the  impact  of  the  Study  211  and  dual 
combination  VBR  and  NrtI  therapy’s  ability  to  serve  as  a  finite  and  curative  therapy  for  chronic  HBV  infection 
offset by an increase in the probability of success of 2158 and 3733 based on their advancement into Phase 2 and 
Phase 1 trials during 2020, respectively and the significance of the future net cash flows from potential drug sales 
for a finite and curative therapy for chronic HBV infection as primarily driven by the number of patients who will be 
diagnosed and treated and the Company’s competitive position in the marketplace. The Company did not recognize 
any IPR&D impairment in any of the periods presented.

Leases

All of the Company’s leases are operating leases for facilities and equipment. Prior to January 1, 2019, the Company 
recognized  related  rent  expense  on  a  straight-line  basis  over  the  term  of  the  lease.  Incentives  granted  under  the 
Company’s facilities lease, including allowances for leasehold improvements and rent holidays, were recognized as 
reductions  to  rental  expense  on  a  straight-line  basis  over  the  term  of  the  lease.  Deferred  rent  consisted  of  the 
difference between cash payments and the rent expense recognized.

Subsequent to the adoption of the new leasing standard on January 1, 2019, the Company recognizes a lease asset 
for  its  right  to  use  the  underlying  asset  and  a  lease  liability  for  the  corresponding  lease  obligation.  The  Company 
determines  whether  an  arrangement  is  or  contains  a  lease  at  contract  inception.  Operating  leases  with  a  duration 
greater than one year are included in operating lease right-of-use assets, operating lease liabilities - short-term, and 
operating  lease  liabilities -  long-term  in  the  Company’s  consolidated  balance  sheets.  Operating  lease  right-of-use 
assets and liabilities are recognized at the lease commencement date based on the present value of lease payments 
over  the  lease  term.  In  determining  the  net  present  value  of  lease  payments,  the  Company  uses  its  incremental 

F-14

borrowing rate based on the information available at the lease commencement date. The incremental borrowing rate 
represents the interest rate the Company would incur at lease commencement to borrow an amount equal to the lease 
payments  on  a  collateralized  basis  over  the  term  of  a  lease.  The  Company  considers  a  lease  term  to  be  the 
noncancelable period that it has the right to use the underlying asset, including any periods where it is reasonably 
assured  the  Company  will  exercise  the  option  to  extend  the  contract.  Periods  covered  by  an  option  to  extend  are 
included in the lease term if the lessor controls the exercise of that option. 

The operating lease right-of-use assets also include any lease payments made and exclude lease incentives. Lease 
expense  is  recognized  on  a  straight-line  basis  over  the  expected  lease  term.  Variable  lease  expenses  are  recorded 
when incurred. The Company has elected not to separate lease and non-lease components for its leased assets and 
accounts for all lease and non-lease components of its agreements as a single lease component.

Impairment of Long-Lived Assets

The Company monitors the carrying value of long-lived assets, including ROU operating lease assets, for potential 
impairment and tests the recoverability of such assets whenever events or changes in circumstances indicate that the 
carrying  amounts  may  not  be  recoverable.  If  a  change  in  circumstance  occurs,  the  Company  performs  a  test  of 
recoverability by comparing the carrying value of the asset or asset group to its undiscounted expected future cash 
flows.  If  cash  flows  cannot  be  separately  and  independently  identified  for  a  single  asset,  the  Company  will 
determine  whether  impairment  has  occurred  for  the  group  of  assets  for  which  the  Company  can  identify  the 
projected cash flows. If the carrying values are in excess of undiscounted expected future cash flows, the Company 
measures any impairment by comparing the fair value of the asset or asset group to its carrying value. In conjunction 
with the decision to wind down the Microbiome program in December 2020, the Company evaluated its ROU assets 
and  property  and  equipment  used  in  the  Microbiome  program  for  impairment.  The  Company  determined  the 
carrying value was no longer recoverable and, based on a fair value of the assets determined from market quotes, 
recorded an impairment loss of $0.7 million included in research and development expenses. The Company did not 
recognize any impairment on its long-lived assets in 2019 or 2018.

Property and Equipment, Net

Property  and  equipment  are  stated  at  cost  and  consist  of  lab  and  office  equipment,  leasehold  improvements  and 
computer  hardware  and  software.  The  Company  records  depreciation  under  the  straight-line  method  over  the 
estimated useful lives of its property and equipment ranging from three to seven years.

Leasehold improvements are amortized over the remaining terms of the respective leases or the estimated useful life 
of the leasehold improvements, whichever is less. Maintenance and repair costs are expensed as incurred.

Fair Value Measurements

The  Company  follows  accounting  guidance  on  fair  value  measurements  for  financial  instruments  measured  on  a 
recurring basis, as well as for certain assets and liabilities that are initially recorded at their estimated fair values. 
Fair value is defined as the exit price, or the amount that would be received from selling an asset or paid to transfer a 
liability  in  an  orderly  transaction  between  market  participants  at  the  measurement  date.  The  Company  uses  the 
following three-level hierarchy that maximizes the use of observable inputs and minimizes the use of unobservable 
inputs to value its financial instruments:

Level 1: Observable inputs such as unadjusted quoted prices in active markets for identical instruments.

Level 2: Quoted prices for similar instruments that are directly or indirectly observable in the marketplace.

Level  3:  Significant  unobservable  inputs  which  are  supported  by  little  or  no  market  activity  and  that  are 
financial instruments whose values are determined using pricing models, discounted cash flow methodologies, 
or  similar  techniques,  as  well  as  instruments  for  which  the  determination  of  fair  value  requires  significant 
judgment or estimation.

Financial instruments measured at fair value are classified in their entirety based on the lowest level of input that is 
significant to the fair value measurement. The assessment of the significance of a particular input to the fair value 
measurement in its entirety requires us to make judgments and consider factors specific to the asset or liability. The 
use of different assumptions and/or estimation methodologies may have a material effect on estimated fair values. 
Accordingly, the fair value estimates disclosed or initial amounts recorded may not be indicative of the amount that 
the Company or holders of the instruments could realize in a current market exchange.

F-15

The carrying amounts of cash equivalents and marketable securities approximate their fair value based upon quoted 
market prices. Certain of the Company’s financial instruments are not measured at fair value on a recurring basis, 
but are recorded at amounts that approximate their fair value due to their liquid or short-term nature, such as cash, 
accounts receivable, accounts payable and accrued expenses.   

The following tables present the fair value of the Company’s financial assets measured at fair value on a recurring 
basis using the above input categories (in thousands):

December 31, 2020

Level 1

Level 2

Level 3

Cash equivalents

Money market funds .........................................   $
U.S. and foreign commercial paper ..................    
Total cash equivalents ............................................    
Short-term investments

U.S. and foreign corporate debt securities........    
Asset-backed securities.....................................    
U.S. treasury securities .....................................    
U.S. and foreign commercial paper ..................    
Total short-term investments..................................    
Total assets measured at fair value.........................   $

47,553    $
—     
47,553     

—     
—     
—     
—     
—     
47,553    $

—    $
6,498     
6,498     

16,939     
12,675     
23,999     
103,356     
156,969     
163,467    $

December 31, 2019

Level 1

Level 2

Level 3

Cash equivalents

Money market fund...........................................   $
U.S. and foreign corporate debt securities........    
U.S. and foreign commercial paper ..................    
Total cash equivalents ............................................    
Short-term investments

U.S. and foreign corporate debt securities........    
Asset-backed securities.....................................    
U.S. treasury securities .....................................    
U.S. and foreign commercial paper ..................    
Total short-term investments..................................    
Total assets measured at fair value.........................   $

33,095    $
—     
—     
33,095     

—     
—     
—     
—     
—     
33,095    $

—    $
4,999     
4,484     
9,483     

72,486     
34,025     
44,714     
76,086     
227,311     
236,794    $

Estimated
Fair Value  

—    $
—     
—     

—     
—     
—     
—     
—     
—    $

47,553 
6,498 
54,051 

16,939 
12,675 
23,999 
103,356 
156,969 
211,020  

Estimated
Fair Value  

—    $
—     
—     
—     

—     
—     
—     
—     
—     
—    $

33,095 
4,999 
4,484 
42,578 

72,486 
34,025 
44,714 
76,086 
227,311 
269,889  

Money  market  funds  are  highly  liquid  and  actively  traded  marketable  securities  that  generally  transact  at  a  stable 
$1.00  net  asset  value  representing  its  estimated  fair  value.  The  Company  estimates  the  fair  value  of  its  U.S.  and 
foreign corporate debt securities, asset backed securities, U.S. treasury securities and U.S. and foreign commercial 
paper by taking into consideration valuations obtained from third-party pricing services. The pricing services utilize 
industry standard valuation models, including both income and market-based approaches, for which all significant 
inputs are observable, either directly or indirectly, to estimate fair value. These inputs include reported trades of and 
broker/dealer  quotes  on 
issuer  credit  spreads;  benchmark  securities; 
prepayment/default projections based on historical data; and other observable inputs.

the  same  or  similar  securities, 

There have been no transfers between Level 1, Level 2 or Level 3 for any of the periods presented. See Note 3 for 
further information regarding the carrying value of our investments in marketable securities.

F-16

 
 
 
 
 
   
   
   
     
       
       
       
 
   
      
      
      
  
 
 
 
 
 
   
   
   
     
       
       
       
 
   
      
      
      
  
Revenue Recognition and Accounts Receivable from Collaborations

The Company analyzes its collaboration arrangements to assess whether such arrangements, or transactions between 
arrangement participants, involve joint operating activities performed by parties that are both active participants in 
the activities and exposed to significant risks and rewards dependent on the commercial success of such activities or 
are  more  akin  to  a  vendor-customer  relationship.  In  making  this  evaluation,  the  Company  considers  whether  the 
activities of the collaboration are considered to be distinct and deemed to be within the scope of the collaborative 
arrangement accounting standard and those that are more reflective of a vendor-customer relationship and, therefore, 
within the scope of the revenue with contracts with customers accounting standard. This assessment is performed 
throughout the life of the arrangement based on changes in the responsibilities of all parties in the arrangement.

For elements of collaboration arrangements that are not accounted for pursuant to the revenue from contracts with 
customers accounting standard, an appropriate recognition method is determined and applied consistently, generally 
by analogy to the revenue from contracts with customers accounting standard. Amounts related to transactions with 
a counterparty in a collaborative arrangement that is not a customer are presented as collaboration revenue and on a 
separate line item from revenue recognized from contracts with customers, if any, in the Company’s consolidated 
statements of operations and comprehensive loss.

Under  certain  collaborative  arrangements,  the  Company  has  been  reimbursed  for  a  portion  of  its  research  and 
development  expenses  or  participates  in  the  cost-sharing  of  such  research  and  development  expenses.  Such 
reimbursements and cost-sharing arrangements are reflected as a reduction of research and development expense in 
the  Company’s  consolidated  statements  of  operations  and  comprehensive  loss,  as  the  Company  does  not  consider 
performing these activities for reimbursement to be a part of its ongoing major or central operations.

For  arrangements  or  transactions  between  arrangement  participants  determined  to  be  within  the  scope  of  the 
contracts with customers accounting standard, the Company evaluates the term of the arrangement and recognizes 
revenue when the customer obtains control of promised goods or services in a contract for an amount that reflects 
the  consideration  the  Company  expects  to  receive  in  exchange  for  those  goods  or  services.  For  contracts  with 
customers, the Company applies the following five-step model in order to determine this amount: (1) identification 
of the promised goods or services in the contract; (2) determination of whether the promised goods or services are 
performance obligations, including whether they are distinct in the context of the contract; (3) measurement of the 
transaction  price,  including  the  constraint  on  variable  consideration;  (4)  allocation  of  the  transaction  price  to  the 
performance  obligations;  and  (5)  recognition  of  revenue  when  (or  as)  the  Company  satisfies  each  performance 
obligation. 

The  Company  has  provided  standard  indemnification  and  protection  of  licensed  intellectual  property  for  its 
customer. These provisions are part of assurance that the licenses meet the agreements, representations and are not 
obligations to provide goods or services.

The  Company  only  applies  the  five-step  model  to  contracts  when  it  is  probable  the  Company  will  collect  the 
consideration  it  is  entitled  to  in  exchange  for  the  goods  or  services  it  transfers  to  the  customer.  As  part  of  the 
accounting for contracts with customers, the Company must develop assumptions that require judgment to determine 
the standalone selling price of each performance obligation identified in the contract. The Company then allocates 
the total transaction price to each performance obligation based on the estimated standalone selling prices of each 
performance  obligation.  The  Company  recognizes  the  amount  of  the  transaction  price  that  is  allocated  to  the 
respective performance obligation when the performance obligation is satisfied or as it is satisfied as revenue. 

Upfront License Fees

If  a  license  to  the  Company’s  intellectual  property  is  determined  to  be  distinct  from  the  other  performance 
obligations  identified  in  the  arrangement,  the  Company  recognizes  revenues  from  nonrefundable,  upfront  license 
fees  based  on  the  relative  value  prescribed  to  the  license  compared  to  the  total  value  of  the  arrangement.  The 
revenue  is  recognized  when  the  license  is  transferred  to  the  collaborator  and  the  collaborator  is  able  to  use  and 
benefit from the license.  For licenses that are not distinct from other obligations identified in the arrangement, the 
Company utilizes judgment to assess the nature of the combined performance obligation to determine whether the 
combined performance obligation is satisfied over time or at a point in time. If the combined performance obligation 
is  satisfied  over  time,  the  Company  applies  an  appropriate  method  of  measuring  progress  for  purposes  of 
recognizing  revenue  from  nonrefundable,  upfront  license  fees.  The  Company  evaluates  the  measure  of  progress 
each reporting period and, if necessary, adjusts the measure of performance and related revenue recognition.

F-17

Development and Regulatory Milestone Payments

Depending  on  facts  and  circumstances,  the  Company  may  record  revenues  from  certain  milestones  in  a  reporting 
period  before  the  milestone  is  achieved  if  the  Company  concludes  achievement  of  the  milestone  is  probable  and 
recognition  of  revenue  related  to  the  milestone  will  not  result  in  a  significant  reversal  in  amounts  recognized  in 
future  periods.  The  Company  records  a  corresponding  contract  asset  when  this  conclusion  is  reached.  Milestone 
payments  that  have  not  been  included  in  the  transaction  price  to  date  are  fully  constrained.  The  Company  re-
evaluates the probability of achievement of such milestones and any related constraint each reporting period. The 
Company adjusts its estimate of the overall transaction price, including the amount of collaborative revenue that was 
recorded, if necessary.  

Research and Development Service Payments

Under  the  Research,  Development,  Collaboration  and  License  Agreement  (Allergan  Agreement)  with  Allergan 
Pharmaecuticals  International  Limited  (Allergan),  the  Company  was  reimbursed  at  a  certain  percentage  for 
performing  research  and  development  services  based  on  hours  worked  by  the  Company’s  employees,  at  a  fixed 
contractual rate per hour, and third-party pass-through costs the Company incurred on a quarterly basis. Research 
and  development  service  payments  were  included  in  the  transaction  price  in  the  reporting  period  the  Company 
concluded it was probable that recording revenue in the period would not result in a significant reversal in amounts 
recognized  in  future  periods.  Accounts  receivable  were  recorded  when  the  right  to  the  research  and  development 
service payment consideration became unconditional. The Company recorded the full reimbursed portion of these 
expenses  as  collaboration  revenue  associated  with  the  Allergan  Agreement  in  its  consolidated  statements  of 
operations as the Company consider performing research and development services to be a part of its ongoing and 
central operations.

Sales-based Milestone and Royalty Payments

The  Company’s  customer  may  be  required  to  pay  the  Company  sales-based  milestone  payments  or  royalties  on 
future  sales  of  commercial  products.   The  Company  recognizes  revenues  related  to  sales-based  milestone  and 
royalty payments upon the later to occur of (i) achievement of the collaborator’s underlying sales or (ii) satisfaction 
of any performance obligation(s) related to these sales, in each case assuming the Company’s licensed intellectual 
property is deemed to be the predominant item to which the sales-based milestones and/or royalties relate.

The Company receives payments from its customer based on billing schedules established in each contract.  Upfront 
payments  and  fees  are  recorded  as  deferred  revenue  upon  receipt  or  when  due  until  the  Company  performs  its 
obligations under the arrangement.  If the related performance obligation is expected to be satisfied within the next 
twelve  months,  these  amounts  will  be  classified  in  current  liabilities.  The  Company  recognizes  a  contract  asset 
relating to its conditional right to consideration that is not subject to a constraint. Amounts are recorded as accounts 
receivable when the Company’s right to consideration is unconditional.  

A  net  contract  asset  or  liability  is  presented  for  each  contract  with  a  customer.  The  Company  does  not  assess 
whether  a  contract  has  a  significant  financing  component  if  the  expectation  at  contract  inception  is  such  that  the 
period between payment by the customer and the transfer of the promised goods or services to the customer will be 
one year or less.

At December 31, 2020 and 2019, all accounts receivable are deemed collectible. 

Stock-Based Compensation

The Company measures stock-based compensation to employees, consultants, and Board members at fair value on 
the grant date of the award. The fair value of RSUs is determined based on the number of shares granted and the 
quoted  market  price  of  the  Company’s  common  stock  on  the  date  of  grant.  Compensation  cost  is  recognized  as 
expense  on  a  straight-line  basis  over  the  requisite  service  period  of  the  award.  Stock-based  awards  with  graded 
vesting schedules are recognized using the accelerated attribution method on a straight-line basis over the requisite 
service  period  for  each  separately  vesting  portion  of  the  award.  For  awards  that  have  a  performance  condition, 
compensation cost is measured based on the fair value of the award on the grant date, the date performance targets 
are  established,  and  is  expensed  over  the  requisite  service  period  for  each  separately  vesting  tranche  when 
achievement  of  the  performance  condition  becomes  probable.  The  Company  assesses  the  probability  of  the 
performance conditions being met on a continuous basis. Forfeitures are recognized when they occur.

F-18

The  Company  estimates  the  fair  value  of  stock  option  grants  that  do  not  contain  market-based  vesting  conditions 
using the Black-Scholes option pricing model. The assumptions used in estimating the fair value of these awards, 
such  as  expected  term,  expected  dividend  yield,  volatility  and  risk-free  interest  rate,  represent  management’s  best 
estimates and involve inherent uncertainties and the application of management’s judgment. The Company is also 
required to make estimates as to the probability of achieving the specific performance conditions. If actual results 
are  not  consistent  with  the  Company’s  assumptions  and  judgments  used  in  making  these  estimates,  the  Company 
may  be  required  to  increase  or  decrease  compensation  expense,  which  could  be  material  to  the  Company’s 
consolidated results of operations.

Prior  to  January  1,  2019,  the  Company  remeasured  the  fair  value  of  the  non-employee  awards  at  each  reporting 
period prior to vesting and finally at the vesting date of the award. Changes in the estimated fair value of these non-
employee  awards  were  recognized  as  compensation  expense  in  the  period  of  change.  After  January  1,  2019,  the 
Company recognizes non-employee compensation costs over the requisite service period based on a measurement of 
fair value for each stock award.

Research and Development Expense and Accruals

Research and development costs include personnel-related costs, outside contracted services including clinical study 
costs, facilities costs, fees paid to consultants, milestone payments prior to FDA approval, license fees prior to FDA 
approval, professional services, travel costs, dues and subscriptions, depreciation and materials used in clinical trials 
and  research  and  development  and  costs  incurred  under  the  Collaboration  Agreement.  Research  and  development 
costs are expensed as incurred unless there is an alternative future use in other research and development projects. 
Payments made prior to the receipt of goods or services to be used in research and development are capitalized until 
the  goods  or  services  are  received.  Such  payments  are  evaluated  for  current  or  long-term  classification  based  on 
when they will be realized or consumed. Assets acquired as part of an asset acquisition that are used in research and 
development  or  are  IPR&D  are  immediately  expensed  as  research  and  development  unless  there  is  an  alternative 
future use in other research and development projects.

The  Company  records  expenses  related  to  clinical  studies  and  manufacturing  development  activities  based  on  its 
estimates  of  the  services  received  and  efforts  expended  pursuant  to  contracts  with  multiple  contract  research 
organizations  (CROs)  and  manufacturing  vendors  that  conduct  and  manage  these  activities  on  its  behalf.  The 
financial  terms  of  these  agreements  are  subject  to  negotiation,  vary  from  contract  to  contract,  and  may  result  in 
uneven payment flows. There may be instances in which payments made to the Company’s vendors will exceed the 
level  of  services  provided  and  result  in  a  prepayment  of  the  expense.  Payments  under  some  of  these  contracts 
depend on factors such as the successful enrollment of subjects and the completion of clinical study milestones. In 
amortizing or accruing service fees, the Company estimates the time period over which services will be performed, 
enrollment of subjects, number of sites activated and the level of effort to be expended in each period. If the actual 
timing of the performance of services or the level of effort varies from the Company’s estimate, the Company will 
adjust the accrued or prepaid expense balance accordingly. To date, there have been no material differences from the 
Company’s estimates to the amounts actually incurred.

The  Company  has  entered  and  may  continue  to  enter  into  license  agreements  to  access  and  utilize  certain 
technology. In each case, the Company evaluates if the license agreement results in the acquisition of an asset or a 
business. To date, none of the Company’s license agreements have been considered to be acquisitions of businesses. 
For asset acquisitions, the upfront payments to acquire such licenses, as well as any future milestone payments, are 
immediately recognized as research and development expense when paid, provided there is no alternative future use 
of  the  rights  in  other  research  and  development  projects.  These  license  agreements  may  also  include  contingent 
consideration in the form of cash payments to be made for future milestone events. The Company assesses whether 
such contingent consideration meets the definition of a derivative and to date the Company has determined that such 
contingent consideration are not derivatives.

Restructuring Charges 

The  Company  recognizes  restructuring  charges  related  to  reorganization  plans  that  have  been  committed  to  by 
management  and  when  liabilities  have  been  incurred.  In  connection  with  these  activities,  the  Company  records 
restructuring charges at fair value for (1) contractual employee termination benefits when obligations are associated 
to  services  already  rendered,  rights  to  such  benefits  have  vested,  and  payment  of  benefits  is  probable  and  can  be 
reasonably  estimated,  (2)  one-time  employee  termination  benefits  when  management  has  committed  to  a  plan  of 
termination,  the  plan  identifies  the  employees  and  their  expected  termination  dates,  the  details  of  termination 
benefits  are  complete,  it  is  unlikely  changes  to  the  plan  will  be  made  or  the  plan  will  be  withdrawn  and 

F-19

communication  to  such  employees  has  occurred,  and  (3)  contract  termination  costs  when  a  contract  is  terminated 
before the end of its term. 

One-time  employee  termination  benefits  are  recognized  in  their  entirety  when  communication  has  occurred, and 
future  services  are  not  required.  If  future  services  are  required,  the  costs  are  recorded  ratably  over  the  remaining 
period  of  service.  Contract  termination  costs  to  be  incurred  over  the  remaining  contract  term  without  economic 
benefit are recorded in their entirety when the contract is canceled.

The recognition of restructuring charges requires the Company to make certain judgments and estimates regarding 
the nature, timing and amount of costs associated with the planned reorganization plan. To the extent the Company’s 
actual  results  differ  from  its  estimates  and  assumptions,  the  Company  may  be  required  to  revise  the  estimates  of 
future accrued restructuring liabilities, requiring the recognition of additional restructuring charges or the reduction 
of  accrued  restructuring  liabilities  already  recognized.  Such  changes  to  previously  estimated  amounts  may  be 
material to the consolidated financial statements. Changes in the estimates of the restructuring charges are recorded 
in the period the change is determined. 

At the end of each reporting period, the Company evaluates the remaining accrued restructuring balances to ensure 
that no excess accruals are retained, and the utilization of the provisions are for their intended purpose in accordance 
with developed restructuring plans.

Variable Interest Entities

The Company reviews agreements it enters into with third party entities, pursuant to which we may have a variable 
interest in the entity, in order to determine if the entity is a variable interest entity (VIE). If the entity is a VIE, the 
Company assesses whether or not it is the primary beneficiary of that entity. In determining whether the Company is 
the primary beneficiary of an entity, the Company applies a qualitative approach that determines whether it has both 
(1) the power to direct the economically significant activities of the entity and (2) the obligation to absorb losses of, 
or the right receive benefits from, the entity that could potentially be significant to that entity. If the Company were 
to determine it is the primary beneficiary of a VIE, the Company would consolidate the statements of operations and 
financial condition of the VIE into its consolidated financial statements.

The Company’s determination about whether it should consolidate such VIEs is made continuously as changes to 
existing  relationships  or  future  transactions  may  result  in  a  consolidation  event.  As  of  December  31,  2020,  the 
Company did not consolidate any entities it had determined to be VIEs.

Income Taxes

The Company records income taxes using the asset and liability method. Deferred income tax assets and liabilities 
are  recognized  for  the  future  tax  effects  attributable  to  temporary  differences  between  the  financial  statement 
carrying amounts of existing assets and liabilities and their respective income tax bases, and operating loss and tax 
credit carryforwards. The effect of a change in tax rates on deferred tax assets and liabilities is recognized in income 
in the period that includes the enactment date. The Company establishes a valuation allowance if it is more likely 
than not that the deferred tax assets will not be realized based on an evaluation of objective verifiable evidence. For 
tax positions that are more likely than not of being sustained upon audit, the Company recognizes the largest amount 
of the benefit that is greater than 50% likely of being realized. For tax positions that are not more likely than not of 
being sustained upon audit, the Company does not recognize any portion of the benefit.

The Company recognizes and measures uncertain tax positions using a two-step approach set forth in authoritative 
guidance.  The  first  step  is  to  evaluate  the  tax  position  taken  or  expected  to  be  taken  by  determining  whether  the 
weight  of  available  evidence  indicates  that  it  is  more  likely  than  not  that  the  tax  position  will  be  sustained  in  an 
audit,  including  resolution  of  any  related  appeals  or  litigation  processes.  The  second  step  is  to  measure  the  tax 
benefit  as  the  largest  amount  that  is  more  than  50%  likely  to  be  realized  upon  ultimate  settlement.  Significant 
judgment is required to evaluate uncertain tax positions. The Company evaluates uncertain tax positions on a regular 
basis. The evaluations are based on a number of factors, including changes in facts and circumstances, changes in 
tax law, correspondence with tax authorities during the course of the audit, and effective settlement of audit issues. 
The provision for income taxes includes the effects of any accruals that the Company believes are appropriate. It is 
the Company’s policy to recognize interest and penalties related to income tax matters in income tax expense. No 
interest or penalties related to uncertain tax positions has been incurred or accrued for any periods presented.  

F-20

In  March  2020,  the  Families  First  Coronavirus  Response  Act  (FFCR  Act)  and  the  Coronavirus  Aid,  Relief,  and 
Economic Security Act (CARES Act) were each enacted in response to the COVID-19 pandemic. The FFCR Act 
and the CARES Act contain numerous income tax provisions relating to refundable payroll tax credits, deferment of 
employer  side  social  security  payments,  net  operating  loss  carryback  periods,  alternative  minimum  tax  credit 
refunds, modifications to the net interest deduction limitations and technical corrections to tax depreciation methods 
for qualified improvement property. 

In  June  2020,  Assembly  Bill  85  (A.B.  85)  was  signed  into  California  law.  A.B.  85  provides  for  a  three-year 
suspension of the use of net operating losses for medium and large businesses and a three-year cap on the use of 
business incentive tax credits to offset no more than $5.0 million of tax per year. A.B. 85 suspends the use of net 
operating losses for taxable years 2020, 2021 and 2022 for certain taxpayers with taxable income of $1.0 million or 
more. The carryover period for any net operating losses that are suspended under this provision will be extended. 
A.B. 85 also requires that business incentive tax credits including carryovers may not reduce the applicable tax by 
more than $5.0 million for taxable years 2020, 2021 and 2022. 

In  December  2020,  the  Consolidated  Appropriations  Act,  2021  (CAA)  was  signed  into  law.  The  CAA  included 
additional funding through tax credits as part of its economic package for 2021. 

The  FFCR  Act,  CARES  Act,  A.B.  85  did  and  CAA  not  have  a  material  impact  on  the  Company’s  consolidated 
financial statements; however, the Company continues to examine the impacts the FFCR Act, CARES Act, A.B. 85 
and CAA may have on its business, results of operations, financial condition and liquidity.

Net Loss per Share

Basic net loss per common share excludes dilution and is computed by dividing net loss by the weighted average 
number of common shares outstanding during the period.  Diluted net loss per common share reflects the potential 
dilution  that  could  occur  if  securities  or  other  contracts  to  issue  common  stock  were  exercised  or  converted  into 
common  stock  or  resulted  in  the  issuance  of  common  stock  that  then  shared  in  the  earnings  of  the  entity  unless 
inclusion of such shares would be anti-dilutive.  Since the Company has only incurred losses, basic and diluted net 
loss per share is the same.

In December 2019, the Company sold 6,287,878 shares of common stock as well as pre-funded warrants to purchase 
up  to  2,424,242  shares  of  common  stock  (see  Note  7).  The  pre-funded  warrants  are  exercisable  for  shares  of 
common stock at a price of $0.001 per share. The shares of common stock into which the pre-funded warrants may 
be exercised are considered outstanding for the purposes of computing earnings per share because the shares may be 
issued for little or no consideration, they are fully vested, and are exercisable after the original issuance date.

Securities excluded from the computation of diluted loss from per share because including them would have been 
antidilutive are as follows:

Warrants to purchase common stock..............................................    
Options to purchase common stock................................................    
Common stock subject to purchase under our ESPP......................    
Unvested RSUs...............................................................................    
Total ..........................................................................................    

—     
6,696,592     
44,223     
746,868     
7,487,683     

15,296     
5,613,353     
11,342     
630,384     
6,270,375     

15,296 
4,637,145 
21,483 
568,005 
5,241,929  

Year Ended December 31,
2019

2018

2020

Comprehensive Loss

Comprehensive  loss  is  comprised  of  net  loss  and  adjustments  for  the  change  in  unrealized  gains  and  losses  on 
investments  in  available-for-sale  marketable  securities.  The  Company  displays  comprehensive  loss  and  its 
components in the consolidated statements of operations and comprehensive loss, net of tax effects if any.

F-21

 
 
 
 
 
   
   
 
Concentrations of Risk

Credit Risk

Financial  instruments  which  potentially  subject  the  Company  to  credit  risk  consist  primarily  of  cash,  cash 
equivalents and marketable securities. The Company holds these investments in highly rated financial institutions, 
and, by policy, limits the amounts of credit exposure to any one financial institution. These amounts at times may 
exceed federally insured limits. The Company has not experienced any credit losses in such accounts and does not 
believe  it  is  exposed  to  any  significant  credit  risk  on  these  funds.  The  Company  has  no  off-balance  sheet 
concentrations  of  credit  risk,  such  as  foreign  currency  exchange  contracts,  option  contracts  or  other  hedging 
arrangements.

Supplier Risk

Certain materials and key components the Company utilizes in its operations are obtained through single suppliers. 
Since the suppliers of key components and materials must be named in a New Drug Application (NDA) filed with 
the FDA for a product, significant delays can occur if the qualification of a new supplier is required. If delivery of 
material from the Company’s suppliers were interrupted for any reason, the Company may be unable to supply any 
of its product candidates for clinical trials. 

Adoption of Recent Accounting Pronouncements

In January 2017, the Financial Accounting Standards Board (FASB) issued ASU 2017-04, Intangibles-Goodwill and 
Other (Topic 350): Simplifying the Test for Goodwill Impairment (ASU 2017-04), which simplifies how an entity is 
required to test goodwill for impairment by eliminating Step 2 from the goodwill impairment test. Step 2 measures a 
goodwill  impairment  loss  by  comparing  the  implied  fair  value  of  a  reporting  unit's  goodwill  with  the  carrying 
amount of that goodwill. Under the amendments in ASU 2017-04, an entity should recognize an impairment charge 
for the amount by which the carrying amount of a reporting unit exceeds its fair value; however, the loss recognized 
should  not  exceed  the  total  amount  of  goodwill  allocated  to  that  reporting  unit.  The  updated  accounting  standard 
requires a prospective adoption. In November 2019, the FASB issued ASU 2019-10, Financial Instruments – Credit 
Losses (Topic 326), Derivatives and Hedging (Topic 815), and Leases (Topic 842): Effective Dates (ASU 2019-10), 
which  deferred  the  effective  date  of  this  standard  for  all  entities  except  SEC  filers  that  are  not  smaller  reporting 
companies to fiscal years beginning after December 15, 2022, including interim periods within those fiscal years. 
Early  adoption  is  permitted  for  goodwill  impairment  tests  performed  on  testing  dates  after  January  1,  2017.  The 
Company  early  adopted  ASU  2017-04  effective  January  1,  2020.  The  adoption  of  this  standard  had  no  material 
impact on the Company’s consolidated financial statements.

On  January  1,  2020,  the  Company  adopted  ASU  2018-13,  Fair  Value  Measurement  (Topic  820):   Disclosure 
Framework -  Changes  to  the  Disclosure  Requirements  for  Fair  Value  Measurement,  which  makes  a  number  of 
changes meant to add, modify or remove certain disclosure requirements associated with the movement amongst or 
hierarchy associated with Level 1, Level 2 and Level 3 fair value measurements. The adoption of this standard had 
no material impact on the Company’s consolidated financial statements and related disclosures.

On January 1, 2020, the Company adopted ASU 2018-18, Collaborative Arrangements (Topic 808): Clarifying the 
Interaction  between  Topic  808  and  Topic  606,  which  clarifies  that  certain  transactions  between  collaborative 
arrangement participants should be accounted for as revenue under Topic 606 when the collaborative arrangement 
participant is a customer in the context of a unit of account. In those situations, all the guidance in Topic 606 should 
be applied, including recognition, measurement, presentation, and disclosure requirements. The standard adds unit-
of-account guidance in Topic 808 to align with the guidance in Topic 606 (that is, a distinct good or service) when 
an entity is assessing whether the collaborative arrangement or a part of the arrangement is within the scope of Topic 
606 and requires that in a transaction with a collaborative arrangement participant that is not directly related to sales 
to  third  parties,  presenting  the  transaction  together  with  revenue  recognized  under  Topic  606  is  precluded  if  the 
collaborative  arrangement  participant  is  not  a  customer.  Amendments  in  the  standard  should  be  applied 
retrospectively  to  the  date  of  initial  application  of  Topic  606,  but  entities  may  elect  to  apply  the  amendments  in 
Topic  808  retrospectively  either  to  all  contracts  or  only  to  contracts  that  are  not  completed  at  the  date  of  initial 
application of Topic 606, and should disclose the election. An entity may also elect to apply the practical expedient 
for contract modifications that is permitted for entities using the modified retrospective transition method in Topic 

F-22

606. The adoption of this standard had no impact on the Company’s consolidated financial statements and related 
disclosures.

In December 2019, the FASB issued ASU No. 2019-12, Simplifying the Accounting for Income Taxes (ASU 2019-
12),  which  eliminates  certain  exceptions  to  the  guidance  in  Income  Taxes  (Topic  740)  related  to  the  approach  for 
intraperiod tax allocation, the methodology for calculating income taxes in an interim period and the recognition of 
deferred  tax  liabilities  for  outside  basis  differences.  The  new  accounting  standard  also  simplifies  aspects  of  the 
accounting for franchise taxes and enacted changes in tax laws or rates and clarifies the accounting for transactions 
that  result  in  a  step-up  in  the  tax  basis  of  goodwill.  The  standard  is  effective  for  fiscal  years  beginning  after 
December 15, 2020 and interim periods within those fiscal years. Early adoption is permitted in an interim or annual 
period. Entities that elect to early adopt the amendments in an interim period should reflect any adjustments as of the 
beginning of the annual period that includes that interim period. Additionally, entities that elect early adoption must 
adopt all the amendments in the same period. Entities will apply the accounting standard prospectively, except for 
certain  amendments.  The  Company  early  adopted  ASU  2019-12  effective  January  1,  2020.  The  adoption  of  this 
standard did not have a material impact on the Company’s consolidated financial statements and related disclosures.

Accounting Pronouncements to Be Adopted

In June 2016, the FASB issued ASU 2016-13, Financial Instruments - Credit Losses: Measurement of Credit Losses 
on  Financial  Instruments  (ASU  2016-13),  which  requires  that  expected  credit  losses  relating  to  financial  assets 
measured  on  an  amortized  cost  basis  and  available-for-sale  debt  securities  be  recorded  through  an  allowance  for 
credit losses. ASU 2016-13 limits the amount of credit losses to be recognized for available-for-sale debt securities 
to  the  amount  by  which  carrying  value  exceeds  fair  value  and  also  requires  the  reversal  of  previously  recognized 
credit losses if fair value increases. In April, May and November 2019, the FASB issued additional amendments to 
the new accounting standard related to transition and clarification. In November 2019, the FASB issued ASU 2019-
10,  Financial  Instruments—Credit  Losses  (Topic  326),  Derivatives  and  Hedging  (Topic  815),  and  Leases  (Topic 
842): Effective Dates (ASU 2019-10), which deferred the effective date of this standard for all entities except SEC 
filers that are not smaller reporting companies to fiscal years beginning after December 15, 2022, including interim 
periods within those fiscal years. Early adoption is permitted. The Company is currently evaluating the timing and 
impact of adopting this new accounting standard on its consolidated financial statements and related disclosures.

In August 2020, the FASB issued ASU 2020-06, Debt—Debt with Conversion and Other Options (Subtopic 470-20) 
and  Derivatives  and  Hedging—Contracts  in  Entity’s  Own  Equity  (Subtopic  815-40):  Accounting  for  Convertible 
Instruments and Contracts in an Entity’s Own Equity (ASU 2020-06), which simplifies the accounting for certain 
financial instruments with characteristics of liabilities and equity, including convertible instruments and contracts on 
an entity’s own equity. Specifically, ASU 2020-06 simplifies accounting for convertible instruments by removing 
major  separation  models  in  ASC  470-20  that  require  separate  accounting  for  embedded  conversion  features.  The 
ASU also removes certain settlement conditions in ASC 815-40 that are required for equity contracts to qualify for 
the  derivative  scope  exception,  which  will  permit  more  equity  contracts  to  qualify  for  the  scope  exception  and 
simplifies  the  diluted  EPS  calculation  in  certain  areas.  The  ASU  is  effective  for  interim  and  annual  periods 
beginning after December 15, 2021, with early adoption permitted after December 15, 2020. Adoption of the ASU 
can  either  be  on  a  modified  retrospective  or  full  retrospective  basis.  The  Company  is  currently  evaluating  the 
impacts of ASU 2020-06 on its consolidated financial statements and related disclosures.

In  October  2020,  the  FASB  issued  ASU  2020-10,  Codification  Improvements  –  Disclosures.  This  ASU  improves 
consistency  by  amending  the  codification  to  include  all  disclosure  guidance  in  the  appropriate  disclosure  sections 
and  clarifies  application  of  various  provisions  in  the  Codification  by  amending  and  adding  new  headings,  cross 
referencing  to  other  accounting  standards,  and  refining  or  correcting  termination.  This  ASU  is  effective  for  fiscal 
years  beginning  after  December  15,  2020.  The  adoption  of  the  ASU  will  not  impact  the  Company’s  consolidated 
financial statements or related disclosures.

F-23

Note 3 - Investments in Marketable Securities

Investments in marketable available-for-sale securities consisted of the following (in thousands):

December 31, 2020
Gross
Unrealized
Gain (1)

Gross
Unrealized
Loss (1)

Amortized
Cost

Estimated
Fair Value  

Cash equivalents

Money market funds .........................................   $
U.S. and foreign commercial paper ..................    
Total cash equivalents ............................................    
Short-term investments

U.S. and foreign corporate debt securities........    
Asset-backed securities.....................................    
U.S. treasury securities .....................................    
U.S. and foreign commercial paper ..................    
Total short-term investments..................................    
Total cash equivalents and investments .................   $

47,553    $
6,498     
54,051     

16,939     
12,674     
23,997     
103,356     
156,966     
211,017    $

—    $
—     
—     

3     
2     
2     
—     
7     
7    $

—    $
—     
—     

(3)    
(1)    
—     
—     
(4)    
(4)   $

47,553 
6,498 
54,051 

16,939 
12,675 
23,999 
103,356 
156,969 
211,020  

December 31, 2019
Gross
Unrealized
Gain (1)

Gross
Unrealized
Loss (1)

Amortized
Cost

Estimated
Fair Value  

Cash equivalents

Money market funds .........................................   $
U.S. and foreign corporate debt securities........    
U.S. and foreign commercial paper ..................    
Total cash equivalents ............................................    
Short-term investments

U.S. and foreign corporate debt securities........    
Asset-backed securities.....................................    
U.S. treasury securities .....................................    
U.S. and foreign commercial paper ..................    
Total short-term investments..................................    
Total cash equivalents and investments .................   $

33,095    $
5,000     
4,484     
42,579     

72,452     
34,008     
44,692     
76,086     
227,238     
269,817    $

(1) Gross unrealized gain (loss) is pre-tax.

—    $
—     
—     
—     

38     
17     
24     
—     
79     
79    $

—    $
(1)    
—     
(1)    

(4)    
—     
(2)    
—     
(6)    
(7)   $

33,095 
4,999 
4,484 
42,578 

72,486 
34,025 
44,714 
76,086 
227,311 
269,889  

As of December 31, 2020, the contractual term to maturity of short-term marketable securities held by the Company 
is less than one year. There were no long-term marketable securities held by the Company as of December 31, 2020.

Realized gains and losses for the years ended December 31, 2020, 2019 and 2018 were not significant. None of the 
Company’s investments have been in a continuous unrealized loss position for more than 12 months as of December 
31, 2020.

See Note 2 for further information regarding the fair value of our investments in marketable securities.

F-24

 
 
 
 
 
   
   
   
     
       
       
       
 
     
       
       
       
 
 
 
 
 
 
   
   
   
     
       
       
       
 
     
       
       
       
 
Note 4 - Property and Equipment, Net

Property and equipment consist of the following (in thousands):

As of December 31,

2020

2019

Lab equipment..................................................................................  $
Office equipment.............................................................................. 
Leasehold improvement................................................................... 
Total property and equipment ............................................................... 
Less: Accumulated depreciation............................................................ 
Property and equipment, net..................................................................  $

247    $
699   
2,490   
3,436   
(1,836)  
1,600    $

247 
699 
2,084 
3,030 
(1,200)
1,830  

Depreciation expense for the years ended December 31, 2020, 2019 and 2018 was $0.7 million, $0.5 million, and 
$0.6  million,  respectively,  and  was  recorded  in  both  research  and  development  expense  and  general  and 
administrative  expense  in  the  consolidated  statements  of  operations  and  comprehensive  loss.  Primarily  all  of 
property and equipment is located in the U.S.

Note 5 – Other Accrued Expenses 

Other accrued expenses consist of the following (in thousands): 

Other accrued expenses:

Accrued compensation.....................................................................  $ 
Accrued restructuring charges ......................................................... 
Accrued professional fees and other ................................................ 
Total other accrued expenses.................................................................  $

7,016    $
4,164   
807   
11,987    $

5,312 
2,094 
880 
8,286  

As of December 31,

2020

2019

Note 6 – Restructurings

2019 Restructuring

In  November  2019,  the  Company’s  Board  of  Directors  approved  the  relocation  of  the  Company  corporate 
headquarters  to  South  San  Francisco,  California  which  became  effective  January  1,  2020.  The  Company  accrued 
restructuring  charges  of  $2.1  million  in  2019  related  to  one-time  termination  severance  payments  and  other 
employee-related costs associated with the relocation plan. This represents the total amount expected to be incurred 
in connection with the relocation. 

2020 Restructuring

In December 2020, the Company and its Board of Directors determined that it was in the Company’s best interest to 
wind down its Microbiome program, enabling the Company to prioritize resources and focus on the advancement of 
its pipeline of novel core inhibitors for chronic HBV infection. The Company expects to complete the wind-down of 
the Microbiome program in early 2021. 

F-25

 
 
 
 
 
   
 
 
 
 
 
 
 
 
 
 
 
 
 
 
   
 
 
 
    
 
  
 
 
 
 
The  following  table  summarizes  the  Company’s  estimates  of  costs  incurred  and  expected  to  be  incurred  (in 
thousands):

Total 
Restructuring 
Cost

Employee 
Severance and 
Related 
Benefits

Asset 
Impairment 
and Other 
Costs

Total estimated restructuring costs to be incurred..............   $
Restructuring costs incurred during the period:
Total restructuring costs incurred for the year ended
December 31, 2019.............................................................    
Total restructuring costs incurred for the year ended
December 31, 2020.............................................................    
Cumulative restructuring costs incurred through
December 31, 2020.............................................................   $

8,040    $

6,461    $

1,579 

2,094     

2,094     

5,684     

4,105     

7,778    $

6,199    $

— 

1,579 

1,579  

The  following  table  presents  the  activity  in  the  accrued  restructuring  charges  during  the  period,  all  of  which  are 
related to employee severance and related benefits (in thousands):

Accrued balance as of January 1, 2019..............................................................................  $
Costs incurred............................................................................................................... 
Accrued balance as of December 31, 2019........................................................................  $
Costs incurred............................................................................................................... 
Reductions for cash payments ...................................................................................... 
Accrued balance as of December 31, 2020........................................................................  $

— 
2,094 
2,094 
3,843 
(1,773)
4,164  

The  Company  also  recognized  $0.3  million  of  accelerated  vesting  for  stock-based  compensation  for  employees 
subject to the restructuring activities during 2020.

The Company expects the accrued restructuring liability to be fully paid in 2021.

The following table presents where the restructuring charges were recognized (in thousands):

Year Ended December 31,
2019
2020

Research and development ....................................................................  $
General and administrative.................................................................... 
Total.......................................................................................................  $

5,486    $
198   
5,684    $

433 
1,661 
2,094  

Note 7 - Stockholders’ Equity

The  Company  is  authorized  to  issue  5,000,000  shares  of  preferred  stock  as  of  December  31,  2020  and  2019, 
respectively.  As  of  December  31,  2020  and  2019,  no  shares  of  preferred  stock  were  issued  and  outstanding.  The 
Company  is  authorized  to  issue  100,000,000  shares  of  common  stock  as  of  December  31,  2020  and  2019, 
respectively.

Sale of Common Stock and Pre-Funded Warrants

In December 2017, the Company filed a registration statement on Form S-3 with the SEC, File No. 333-222366, that 
became  effective  January  10,  2018  (the  2018  Registration  Statement).  The  2018  Registration  Statement  gave  the 
Company the ability to sell any combination of the securities described in the 2018 Registration Statement in one or 
more  offerings  up  to  an  aggregate  offering  price  of  $250.0  million.  In  connection  with  the  filing  of  the  2018 
Registration Statement, the Company entered into a sales agreement that gave the Company the ability to sell shares 
of its common stock having an aggregate offering price of up to $75.0 million through “at the market offerings” (the 
2017 ATM). The 2017 ATM was terminated effective September 6, 2020, and no shares were sold under the 2017 
ATM prior to the termination. 

F-26

 
 
   
   
 
   
      
      
  
 
 
 
 
 
 
 
 
   
 
 
 
In July 2018, the Company sold to various investors an aggregate of 4,600,000 shares of common stock in a public 
offering  at  $36.00  per  share,  which  included  the  exercise  in  full  by  the  underwriters  of  their  option  to  purchase 
600,000 additional shares of common stock. The Company received aggregate net proceeds of $155.4 million from 
the offering and the option exercise, after deducting underwriting discounts and commissions and offering expenses 
payable by the Company.

In December 2019, the Company sold to various investors an aggregate of 6,287,878 shares of common stock at a 
public offering price of $16.50 per share, which included the exercise in full by the underwriters of their option to 
purchase  1,136,363  shares  of  common  stock,  and  pre-funded  warrants  to  purchase  2,424,242  shares  of  common 
stock at a public offering price of $16.499. The Company received aggregate net proceeds of $134.7 million from 
the offering and the option exercise, after deducting underwriting discounts and commissions and offering expenses 
payable  by  the  Company.  The  pre-funded  warrants  became  immediately  exercisable  upon  issuance  at  an  exercise 
price  of  $0.001  per  share,  but  under  their  terms,  the  outstanding  pre-funded  warrants  to  purchase  shares  of  the 
Company’s  common  stock  generally  may  not  be  exercised  if  the  holder’s  ownership  of  the  Company’s  common 
stock  would  exceed  19.99%  following  such  exercise.  The  exercise  price  and  number  of  shares  of  common  stock 
issuable upon the exercise of the pre-funded warrants (Warrant Shares) are subject to adjustment in the event of any 
stock dividends and splits, reverse stock split, recapitalization, reorganization or similar transaction, as described in 
the pre-funded warrant agreements. Under certain circumstances, the pre-funded warrants may be exercisable on a 
“cashless” basis. Both the pre-funded warrants and the Warrant Shares are registered securities.

The pre-funded warrants were classified as a component of permanent stockholders’ equity within additional paid-
in-capital  and  were  recorded  at  the  issuance  date  using  a  relative  fair  value  allocation  method.  The  pre-funded 
warrants  are  equity  classified  because  they  are  freestanding  financial  instruments  that  are  legally  detachable  and 
separately exercisable from the equity instruments, are immediately exercisable, do not embody an obligation for the 
Company to repurchase its shares, permit the holders to receive a fixed number of common shares upon exercise, are 
indexed  to  the  Company’s  common  stock  and  meet  the  equity  classification  criteria.  In  addition,  such  pre-funded 
warrants do not provide any guarantee of value or return. The Company valued the pre-funded warrants at issuance, 
concluding their sales price approximated their fair value, and allocated net proceeds from the sale proportionately 
to  the  common  stock  and  pre-funded  warrants  of  which  $37.5  million  allocated  to  the  pre-funded  warrants  and 
recorded as a component of additional paid-in-capital.

In August 2020, the Company filed a shelf registration statement on Form S-3 with the SEC, File No. 333-248469, 
that became effective on September 4, 2020 (the 2020 Registration Statement). The Company may from time to time 
sell any combination of the securities described in the 2020 Registration Statement in one or more offerings up to an 
aggregate  offering  price  of  $300.0  million.  In  connection  with  the  filing  of  the  2020  Registration  Statement,  the 
Company entered into a sales agreement under which the Company may offer and sell shares of its common stock 
having an aggregate offering price of up to $100.0 million through “at-the-market” offerings (2020 ATM), which 
shares are included in the $300.0 million of securities registered pursuant to the 2020 Registration Statement. During 
the year ended December 31, 2020, the Company issued and sold 892,840 shares of common stock under the 2020 
Registration Statement, for which the Company received net proceeds of $5.5 million, after deducting commissions, 
fees and expenses. 

The  Company  carried  forward  registration  fees  paid  with  respect  to  $21.4  million  of  securities  that  remained 
available under the 2018 Registration Statement. As such, as of the effectiveness of the 2020 Registration Statement, 
the 2018 Registration Statement was deemed terminated.

Common Stock Warrants

As of December 31, 2020, the following warrants to purchase shares of the Company’s common stock were issued 
and outstanding:

Issue date

Expiration
date

Exercise Price
per Share

December 31, 
2020

December 31, 
2019

September 10, 2010 ...  September 10, 2020   $
  $
December 16, 2019 .... 

None

30.000   
0.001   

—   
2,424,242   
2,424,242   

15,296 
2,424,242 
2,439,538  

F-27

 
 
   
   
 
 
 
 
 
 
 
 
 
 
    
 
 
There were no warrants exercised during the years ended December 31, 2020, 2019 and 2018. During the year ended 
December  31,  2020,  15,296  warrants  to  purchase  common  stock  expired  unexercised.  During  the  year  ended 
December 31, 2018, 1,613 warrants to purchase common stock expired unexercised.

Note 8 - Stock-Based Compensation

Equity Incentive Plans

In May 2018, the Company’s stockholders approved (1) the Assembly Biosciences, Inc. 2018 Stock Incentive Plan 
(the  2018  Plan)  pursuant  to  which  the  Company  reserved  1,900,000  shares  of  its  common  stock  for  issuance  in 
connection with equity incentive awards and (2) the Assembly Biosciences, Inc. Employee Stock Purchase Plan (the 
2018  ESPP)  pursuant  to  which  the  Company  reserved  400,000  shares  of  its  common  stock  for  issuance  in 
connection with purchases by employees pursuant to this plan.

In May 2019, the Company’s stockholders approved an amendment to the 2018 Plan that increased the aggregate 
shares of common stock reserved under the 2018 Plan to 3,000,000.

In June 2020, the Company’s stockholders approved an amendment to the 2018 Plan that increased the aggregate 
number of shares of common stock reserved under the 2018 Plan to 4,600,000.

As of December 31, 2020, the Company had awards outstanding under the following shareholder approved plans: 
2010  Equity  Incentive  Plan  (the  2010  Plan),  which  has  been  frozen;  the  Amended  and  Restated  2014  Stock 
Incentive  Plan  (the  2014  Plan);  and  the  2018  Plan.  Shares  of  common  stock  underlying  awards  that  are  forfeited 
under  the  2010  Plan  on  or  after  June  2,  2016  will  become  available  for  issuance  under  the  2014  Plan.  As  of 
December  31,  2020,  the  Company  also  had  awards  outstanding  under  the  Assembly  Biosciences,  Inc.  2017 
Inducement  Award  Plan  (the  2017  Plan),  the  2019  Inducement  Award  Plan  (the  2019  Plan)  and  the  Assembly 
Biosciences, Inc. 2020 Inducement Award Plan (the 2020 Plan).

The Company issues new shares of common stock to settle options exercised or vested RSUs. The Company also 
issues new shares of common stock in connection with purchases of shares of common stock by eligible employees 
under the Company’s 2018 ESPP.

Stock Plan Activity

Stock Options

The following table summarizes the stock option activity and related information for 2020:

Weighted
Average
Exercise
Price

Weighted
Average
Remaining
Contractual
Term (Years)   

Total
Intrinsic
Value
(in thousands) 

Number
of Shares

Outstanding as of December 31, 2019 ...................   
Granted ...................................................................   
Exercised ................................................................   
Forfeited .................................................................   
Outstanding as of December 31, 2020 ...................   
Exercisable as of December 31, 2020 ....................   

5,613,353    $
1,649,340     
(175,579)   
(390,522)   
6,696,592    $
3,926,732    $

Per Share    
15.90     
16.07     
9.75     
22.81     
15.70     
14.70     

6.9    $
5.5    $

1,856 
1,813  

The  weighted-average  grant-date  fair  value  of  options  granted  was  $10.64,  $10.55  and  $30.84  during  the  years 
ended December 31, 2020, 2019 and 2018, respectively. The total intrinsic value of options exercised in 2020, 2019 
and 2018 was $2.0 million, $5.0 million and $31.1 million, respectively.  

F-28

 
 
   
      
  
      
  
      
  
      
  
RSUs

The following table summarizes RSU activity and related information for 2020:

Nonvested as of December 31, 2019 ...............................................................    
Granted.............................................................................................................    
Vested ..............................................................................................................    
Forfeited...........................................................................................................    
Nonvested as of December 31, 2020 ...............................................................    

Number
of RSU's

758,718    $
536,164   
(297,133)  
(110,881)  
886,868  (1) $

Weighted
Average Fair
Value Per RSU
at Grant Price  
25.47 
16.21 
23.65 
26.46 
20.36  

(1)

Includes 140,000 RSUs that have vested but are subject to deferred settlement, which have a weighted average 
remaining contractual term of 2.2 years.

The total fair value of RSUs vested and settled during 2020, 2019 and 2018 was $7.8 million, $5.7 million, and $5.3 
million, respectively. The total intrinsic value of RSUs vested and settled during 2020 and 2019 was $4.4 million 
and $2.9 million, respectively. The total intrinsic value of RSUs vested and settled during 2018 was nominal.

As of December 31, 2020, RSUs outstanding include 100,000 RSUs granted in September 2019 to the Company’s 
chief executive officer with performance-based conditions. The 100,000 awards with an aggregate fair value of $1.2 
million vest upon performance conditions not yet deemed probable and accordingly no stock-based compensation 
expense has been recognized as of December 31, 2020. In July 2020, the performance condition for 45,000 RSUs 
granted in December 2017 to a former executive officer was met associated with the execution of an HBV business 
development transaction. The Company recognized $0.7 million as a cumulative catch-up adjustment of stock-based 
compensation expense for this award for the year ended December 31, 2020. In the second quarter of 2019, 100,000 
RSUs granted to a former officer were forfeited due to his departure. These RSUs had a grant date fair value of $2.4 
million and were vesting over time but would have accelerated upon the achievement of certain performance-based 
conditions.  The  Company  reversed  the  previously  recognized  expense  of  $0.5  million  related  to  these  forfeited 
awards upon the departure of the former officer in 2019. 

Employee Stock Purchase Plan

The 2018 ESPP provides for the purchase by employees of up to an aggregate of 400,000 shares of the Company’s 
common stock at a discount to the market price. Subject to the annual statutory limits and the 2018 ESPP’s limit of 
1,000 shares of common stock per offering, an eligible employee may participate through payroll deductions of up 
to 15% of such employee’s compensation for each pay period

Eligible  employees  can  purchase  the  Company’s  common  stock  at  the  end  of  a  predetermined  offering  period  at 
85% of the lower of the fair market value at the beginning or end of the offering period. Under the 2018 ESPP, the 
offering  periods  end  on  the  last  business  day  occurring  on  or  before  May  14  or  November  14.  The  ESPP  is 
compensatory and results in stock-based compensation expense.

In  November  2018,  employees  purchased  21,483  shares  of  common  stock  under  the  2018  ESPP.  In  May  and 
November  2019,  employees  purchased  36,804  and  22,566  shares  of  common  stock,  respectively,  under  the  2018 
ESPP. In May and November 2020, employees purchased 42,266 and 44,546 shares of common stock, respectively, 
under the 2018 ESPP. As of December 31, 2020, 232,335 shares of common stock are available for future sale under 
the  Company’s  2018  ESPP.  Stock-based  compensation  expense  recorded  in  connection  with  the  2018  ESPP  was 
$0.5 million, $0.4 million and $0.2 million for the years December 31, 2020, 2019 and 2018, respectively.

F-29

 
 
   
 
 
 
Valuation Assumptions

The Company used the Black-Scholes option-pricing model for determining the estimated fair value and stock-based 
compensation related to stock options and ESPP purchase rights. 

A summary of the assumptions used to estimate the fair values of stock options grants for the years presented is as 
follows: 

Year Ended December 31,
2019

2018

2020

Exercise price......................................................................   $5.62 - $23.30     $9.31 - $23.04     $23.78 - $57.53  
Expected volatility ..............................................................   66.4% - 92.3%     66.5% - 83.2%     75.6% - 86.1%  
Risk-free interest rate..........................................................   0.26% - 1.44%     1.36% - 2.65%     2.56% - 3.04%  
Expected term (years) .........................................................  
Expected dividend yield .....................................................  

5.5 - 7.5
0%

5.5 - 7.5
0%

5.5 - 7.0
0%

The risk-free interest rate assumption was based on the rates for U.S. Treasury zero-coupon bonds with maturities 
similar to those of the expected term of the stock option being valued. The expected dividend yield was zero as the 
Company currently does not intend to pay dividends in the foreseeable future. The weighted average expected term 
of  options  was  calculated  using  the  simplified  method  as  prescribed  by  accounting  guidance  for  stock-based 
compensation  due  to  the  Company’s  limited  history  of  relevant  stock  option  exercise  activity.  The  expected 
volatility was calculated based on the Company’s historical stock prices, supplemented as necessary with historical 
volatility of the common stock of several peer companies with characteristics similar to those of the Company.

The fair value of ESPP purchase rights were not material for any period presented.

Stock-Based Compensation Expense

The Company recognized stock-based compensation expense included in the consolidated statement of operations 
and comprehensive loss for the periods presented (in thousands):

Year Ended December 31,
2019

2018

2020

Research and development .................................................  $
General and administrative .................................................   
Total stock-based compensation expense .......................  $

11,380    $
10,473  (1) 
21,853    $

11,376    $
9,182  (2) 
20,558    $

11,820 
16,665 
28,485  

(1)

(2)

Includes the reversal of previously recognized expense of $1.7 million related to forfeited awards resulting from 
the departure of one of our former executive officers during the year.

Includes the reversal of previously recognized expense of $3.6 million related to forfeited awards resulting from 
the departure of one of our former executive officers during the year.

As  of  December  31,  2020,  there  was  $20.4  million  of  total  unrecognized  stock-based  compensation  related  to 
outstanding  equity  awards  which  is  expected  to  be  recognized  over  a  weighted  average  remaining  amortization 
period of 1.8 years.

F-30

 
 
 
 
 
   
   
 
   
   
 
   
   
 
 
 
 
 
 
   
   
 
Note 9 - Collaboration Agreements

Allergan Agreement

In  January  2017,  the  Company  and  Allergan  entered  into  the  Allergan  Agreement  to  develop  and  commercialize 
select  microbiome  gastrointestinal  disease  therapies.  Pursuant  to  the  Allergan  Agreement,  the  Company  granted 
Allergan  an  exclusive  worldwide  license  to  certain  of  its  intellectual  property,  including  its  intellectual  property 
arising  under  the  Allergan  Agreement,  to  develop  and  commercialize  licensed  compounds  for  ulcerative  colitis 
(UC),  Crohn’s  disease,  and  two  compounds  for  irritable  bowel  syndrome  (IBS).  Allergan  and  the  Company  also 
agreed to collaborate on research and development activities with respect to the licensed compounds in accordance 
with  a  mutually  agreed  upon  research  and  development  plan.  Per  the  terms  of  the  Allergan  Agreement,  Allergan 
could select backups and additional target indications to add to the licenses granted for additional consideration and 
also had the ability to enter into a contract manufacturing agreement with the Company for compound supply at cost 
plus an agreed upon margin. In addition, the Company participated on a Joint Development Committee (JDC) and 
Joint Patent Committee (JPC). Allergan had the right to terminate the Allergan Agreement at any time upon advance 
written notice.

In  June  2020,  following  its  acquisition  of  Allergan,  AbbVie  Inc.  (AbbVie),  on  behalf  of  Allergan,  gave  written 
notice of termination of the Allergan Agreement effective 120 days following the delivery of notice, on October 10, 
2020. Upon termination, the licenses granted by the Company and its know-how reverted to the Company. Under 
the  terms  of  the  Allergan  Agreement,  AbbVie  was  obligated  to  continue  to  reimburse  the  Company  for  certain 
research  and  development  costs  through  October  10,  2020.  Upon  effectiveness  of  the  termination,  such 
reimbursements  ceased.  Due  to  the  delivery  of  the  termination  notice,  the  Company  determined  there  were  no 
further enforceable rights and obligations under the Allergan Agreement beyond June 2020 and the remaining $36.0 
million of deferred revenue was recognized in 2020. 

Allergan  paid  the  Company  an  upfront  non-refundable  payment  of  $50.0  million  which  was  received  in  2017. 
Additionally, the Company was eligible to receive variable consideration in the form of research and development 
cost reimbursements, up to $631.0 million related to seven development milestones and up to $2.14 billion related to 
12  commercial  development  and  sales  milestones  in  connection  with  the  successful  development  and 
commercialization of licensed compounds. In addition, the Company was eligible to receive tiered royalties at rates 
ranging from the mid-single digits to the mid-teens based on net sales.

Allergan  and  the  Company  agreed  to  share  research  and  development  costs  up  to  an  aggregate  of  $75.0  million 
through proof-of-concept (POC) studies on a ⅔, ⅓ basis, respectively, and Allergan agreed to assume all post-POC 
development  costs.  In  the  event  any  pre-POC  development  costs  would  have  exceeded  $75.0  million  in  the 
aggregate,  the  Company  may  have  elected  either  (a)  to  fund  ⅓  of  such  costs  in  excess  of  $75.0  million  or  (b)  to 
allow  Allergan  to  deduct  from  future  development  milestone  payments  ⅓  of  the  development  costs  funded  by 
Allergan in excess of $75.0 million plus a premium of 25%. The Company had an option to co-promote the licensed 
programs in the U.S. and China, subject to certain conditions set forth in the Allergan Agreement.

The Company concluded that Allegan was a customer, and the contract was not subject to accounting literature on 
collaborative arrangements. This is because the Company granted to Allergan licenses to its intellectual property and 
agreed to perform research and development services, all of which are outputs of the Company’s ongoing activities, 
in  exchange  for  consideration.  The  Company  identified  the  following  material  promises  under  the  Allergan 
Agreement:  (1)  grant  of  a  licenses  to  intellectual  property  for  the  four  initial  indications,  inclusive  of  the  related 
technology  know-how  (Licenses)  and  (2) the  obligation  to  perform  research  development  services  through  POC 
(Development Services). The Company’s participation on the JDC and JPC were considered to be immaterial in the 
context  of  the  contract.  The  Company’s  co-promotion  option  was  not  considered  to  be  a  performance  obligation. 
Allergan’s  selection  of  backups  or  additional  target  indications  to  add  to  the  licenses  granted  for  additional 
consideration and ability to enter into a contract manufacturing agreement with the Company for compound supply 
at cost plus an agreed upon margin were not considered to be performance obligations as the Company concluded 
the options were not offered at a discount that exceeds discounts available to other customers, and therefore were not 
material  rights.  The  grant  of  additional  licensing  rights  upon  option  exercises  and  contract  manufacturing 
agreements were to be accounted for as separate contracts when or if they occurred.

F-31

The  Company  concluded  the  Licenses  each  were  considered  to  be  functional  as  they  had  significant  standalone 
functionality  and  were  capable  of  being  distinct.  However,  the  Company  determined  that  each  of  the  Licenses 
individually were not distinct from the Development Services within the context of the agreement. This is because 
Allergan  was  dependent  on  the  Company  to  execute  the  Development  Services,  which  it  was  uniquely  able  to 
perform,  in  order  for  Allergan  to  benefit  from  the  Licenses.  As  such,  the  Company  determined  that  it  had  four 
performance  obligations  under  the  Allergan  Agreement  associated  with  the  grant  of  the  four  compound  Licenses 
combined  with  the  performance  of  the  Development  Services  for  each  of  the  four  compound  indications.  The 
Company  determined  that  the  four  performance  obligations  would  have  been  performed  over  the  duration  of  the 
contract, which began in February 2017 and ends upon receipt of the termination notice. The Company used a cost-
based input method to measure proportional performance and to calculate the corresponding amount of revenue to 
recognize. The Company believed this was the best measure of progress because other measures do not reflect how 
the Company transfers its performance obligation to Allegan. In applying the cost-based input method of revenue 
recognition,  the  Company  measured  costs  incurred  relative  to  budgeted  costs  to  fulfill  the  four  performance 
obligations. These costs consisted primarily of third-party contract costs and internal labor costs. Revenue will be 
recognized  based  on  actual  costs  incurred  as  a  percentage  of  total  budgeted  costs  as  the  Company  completed  its 
performance obligations.

To  allocate  transaction  price  among  the  four  performance  obligations,  the  Company  estimated  their  standalone 
selling price (SSP) using an income-based valuation approach for the estimated value a licensor of the compounds 
would  receive  considering  the  stage  of  the  compounds’  development.  A  change  in  the  assumptions  used  to 
determine  its  best  estimate  of  selling  price  for  the  four  performance  obligations  would  not  have  had  a  significant 
effect on the allocation of consideration received to the four performance obligations.

The  transaction  price  at  the  inception  of  the  agreement  and  upon  adoption  of  the  revenue  from  contracts  with 
customers guidance was limited to the $50.0 million upfront payment. Of this amount, the Company allocated $12.5 
million to each of the four performance obligations. Research and development cost reimbursement payments were 
included  in  the  transaction  price  in  the  reporting  period  that  the  Company  concludes  that  it  was  probable  that 
recording  revenue  in  the  period  would  not  have  resulted  in  a  significant  reversal  in  amounts  recognized.  The 
variable  consideration  related  to  the  remaining  development  and  commercialization  milestone  payments  was  not 
included  in  the  transaction  price  as  these  were  fully  constrained.  As  part  of  the  Company’s  evaluation  of  the 
development  and  commercialization  milestones  constraint,  the  Company  determined  the  achievement  of  such 
milestones was contingent upon success in future clinical trials and regulatory approvals which was not within its 
control and uncertain at this stage.  Any variable consideration related to sales-based milestones (including royalties) 
would  have  been  recognized  when  the  related  sales  occur  as  they  were  determined  to  relate  predominantly  to  the 
license  granted  to  Allergan. The  Company  re-evaluated  the  transaction  price  in  each  reporting  period  and  as 
uncertain events were resolved or other changes in circumstances occurred.

The Company did not incur any significant incremental costs of obtaining the Allergan contract.

For the year ended December 31, 2020, 2019, and 2018 the Company recognized $48.1 million, $16.0 million and 
$14.8 million respectively, in collaboration revenue associated with the Allergan Agreement. Short-term and long-
term deferred revenue contract liabilities related to the Allergan Agreement were $6.4 million and $30.6 million at 
December 31, 2019, respectively. There were no deferred revenue contract liabilities as of December 31, 2020 due 
to the Company recognizing a cumulative catch-up adjustment of the remaining deferred revenue balance during the 
year ended December 31, 2020 for the determined completion of the Company’s performance obligations under the 
Allergan Agreement upon receipt of the notice of termination from AbbVie. Contract asset balances of $1.0 million 
and $3.4 million were recorded as of December 31, 2020 and 2019, respectively. 

BeiGene Agreement

In  July  2020,  the  Company  and  BeiGene,  Ltd.  (BeiGene)  entered  into  a  Collaboration  Agreement  (the  BeiGene 
Agreement)  to  develop  and  commercialize  the  Company’s  novel  core  inhibitor  product  candidates  VBR,  ABI-
H2158 and ABI-H3733 for chronic HBV infection (the Licensed Product Candidates) in the People’s Republic of 
China,  Hong  Kong,  Taiwan  and  Macau  (the  Territory).  Under  the  agreement,  the  Company  and  BeiGene  are 
collaborating on certain global clinical studies and both the Company and BeiGene will independently conduct other 
clinical studies in their own respective territories. 

BeiGene agreed to pay all development and regulatory costs for the Licensed Product Candidates in the Territory up 
to  an  aggregate  of  $45.0  million.  Development  and  regulatory  costs  for  the  Licensed  Product  Candidates  for  the 
Territory in excess of $45.0 million will be shared equally by the Company and BeiGene. If the Company conducts 

F-32

certain ancillary trials outside of the plan to develop these candidates in the Territory, BeiGene may elect to obtain 
access  to  the  know-how  and  clinical  data  resulting  for  such  ancillary  trials  and  shall  reimburse  the  Company 
proportionally  for  the  Territory  of  the  costs  of  such  trials.    Activities  under  the  BeiGene  Agreement  will  be 
governed by a joint steering committee (JSC) consisting of equal representatives from each party to the agreement. 
All  decisions  of  the  JSC  are  to  be  made  by  consensus  with  final  decision-making  authority  granted  to  each  party 
based on key areas of the collaboration for which they are responsible.   During the term of the BeiGene Agreement, 
neither party will commercialize any competing products in the Territory.    The Company will be responsible for 
manufacturing  and  supply  of  the  candidates  to  be  used  in  and  outside  of  the  Territory,  although  the  parties  may 
approve BeiGene to take on some or all of the commercial supply activities of the applicable Licensed Products in 
the Territory.

The Company is not obligated to perform pre-phase 3 clinical trial development work outside the Territory on ABI-
H2158 and ABI-H3733 but must provide BeiGene pre-Phase 3 clinical trial know-how and development results if 
and when such development efforts are completed. If, after ABI-H2158 and ABI-H3733 reach the end of Phase 2 
clinical  trials,  the  Company  and  BeiGene  are  unable  to  mutually  agree  on  the  terms  of  a  Phase  3  global  study, 
BeiGene may elect to terminate the BeiGene Agreement solely as it relates to that compound, as applicable. Such a 
termination  would  result  in  the  Company  regaining  all  rights  to  the  applicable  compound  in  the  Territory.  In 
addition,  BeiGene  may  terminate  the  BeiGene  Agreement  for  convenience  at  any  time  upon  90  days’  advance 
written  notice  to  us.  The  BeiGene  Agreement  also  contains  customary  provisions  for  termination  by  either  party, 
including in the event of breach of the BeiGene Agreement, subject to cure.

Pursuant to the terms of the BeiGene Agreement, the Company received an upfront cash payment of $40.0 million 
from  BeiGene  for  the  delivery  of  exclusive,  royalty-bearing  licenses  to  develop  and  commercialize  the  Licensed 
Product Candidates in the Territory, and the Company is eligible to receive up to approximately $500.0 million in 
cash milestone payments, comprised of up to $113.8 million for development and regulatory milestones and up to 
$385.0 million in net sales milestones. In addition, the Company is eligible to receive tiered royalties at percentages 
ranging from the mid-teens to the low thirties of net sales. 

The BeiGene Agreement is within the scope of the collaborative arrangements guidance as both parties are active 
participants  and  are  exposed  to  significant  risks  and  rewards  dependent  on  the  success  of  commercializing  the 
Licensed Product Candidates in the Territory but that the unit of account related to the delivery of Licensed Product 
Candidates is within the scope of the contract with customers guidance.    The remaining units of account related to 
participation on the JSC and subcommittees, clinical supply and other in Territory and global development activities 
(the Collaboration Activities) are within the scope of the collaborative arrangements guidance. Commercial supply 
will  be  evaluated  as  a  separate  contract  when  the  agreement  is  executed  and  a  purchase  order  is  received  from 
BeiGene.

The  Company  identified  the  following  material  promises  related  to  the  contract  with  customers  unit  of  account 
under the BeiGene Agreement: 1) the transfer of the VBR License, 2) the transfer of the ABI-H2158 License, and 3) 
the transfer of the ABI-H3733 License. The Company concluded each of these licenses to be functional as they have 
significant  standalone  functionality  and  grants  BeiGene  the  right  to  use  the  Company’s  intellectual  property  as  it 
exists on the effective date of the license. The ABI-H2158 and ABI-H3733 Licenses have a continuing technology 
transfer obligation that is considered to be an attribute of these licenses.    The agreed upon prices for the clinical and 
commercial supply of the Licensed Product Candidates to BeiGene do not represent material rights, and therefore 
are not performance obligations, and such pricing on an aggregate basis represents the standalone selling price an 
entity  would  typically  pay  for  such  a  product  in  that  region  or  market.  There  are  also  no  minimum  purchase 
commitments.

The  Company  estimated  the  standalone  selling  price  (SSP)  of  the  Licenses  using  an  income-based  valuation 
approach  for  the  estimated  value  a  licensor  of  the  compounds  would  receive  considering  the  stage  of  the 
compound’s development. The Company believes a change in the assumptions used to determine its best estimate of 
SSP would not have a significant value on the allocation of consideration received.

The  transaction  price  at  the  inception  of  the  agreement  was  limited  to  the  $40.0  million  upfront  payment.  The 
variable  consideration  related  to  the  remaining  development  and  commercialization  milestone  payments  has  not 
been  included  in  the  transaction  price  as  these  were  fully  constrained  as  of  December  31,  2020.  As  part  of  the 
Company’s evaluation of the development and commercialization milestones constraint, the Company determined 
the  achievement  of  such  milestones  are  contingent  upon  success  in  future  clinical  trials  and  regulatory  approvals 
which  are  not  within  its  control  and  uncertain  at  this  stage.  Any  variable  consideration  related  to  sales-based 
milestones (including royalties) will be recognized when the related sales occur as they were determined to relate 

F-33

predominantly to the Licensed Product Candidates granted to BeiGene. The Company will reevaluate the transaction 
price in each reporting period as uncertain events are resolved or other changes in circumstances occur.

During the year ended December 31, 2020, the Company recognized $31.0 million as collaboration revenue for the 
amount allocated to the VBR License as substantial completion of the license technology transfer has occurred. The 
remaining transaction price allocated to the ABI-H2158 and ABI-H3733 Licenses of $9.0 million was recorded as a 
long-term deferred revenue contract liability on the consolidated balance sheet as of December 31, 2020. Revenue 
for these performance obligations will be recognized when the Company provides pre-Phase 3 clinical trial know-
how and development results for these compounds to BeiGene or a termination of the BeiGene Agreement for the 
respective compound.

Payments to, or reimbursements from, BeiGene related to the Collaboration Activities will be accounted for as an 
increase to or reduction of research and development expenses when incurred or realized, respectively. During the 
year  ended  December  31,  2020,  the  Company  did  not  recognize  any  increase  or  reduction  of  research  and 
development expense under the BeiGene Agreement. 

The Company incurred $3.5 million in incremental costs of obtaining the BeiGene Agreement. These contract costs 
have been capitalized and are being recognized consistent with the pattern of recognition of revenue associated with 
the  Licensed  Product  Candidates.  As  of  December  31,  2020,  $2.7  million  has  been  amortized  to  general  and 
administrative expenses and $0.8 million is included in other assets on the condensed consolidated balance sheet. 

Arbutus Agreement

In  August  2020,  the  Company  and  Arbutus  Biopharma  Corporation  (Arbutus)  entered  into  a  Collaboration 
Agreement (Arbutus Agreement) to conduct a randomized, multi-center, open-label Phase 2 clinical trial to explore 
the safety, PK and antiviral activity of the triple combination of VBR, AB-729 and an NrtI compared to the double 
combinations of VBR with an NrtI and AB-729 with an NrtI. Assembly and Arbutus will share responsibility for the 
costs of the trial equally, excluding manufacturing supply which will be the burden of each company to supply their 
respective drugs VBR and AB-729.

The  Arbutus  Agreement  is  within  the  scope  of  the  collaborative  arrangements  guidance  as  both  parties  are  active 
participants and are exposed to significant risks and rewards dependent on the success of the collaborative activity. 
Arbutus is not a customer as it does not obtain an output from the collaborative activities as they were not provided 
an  exclusive  license  to  VBR  or  the  ability  to  manufacture  VBR,  and  the  Company  does  not  consider  performing 
such collaborative activities to be a part of its ongoing activities.

The revenue from contracts with customers guidance was considered by analogy in determining the unit of account, 
and  the  recognition  and  measurement  of  such  unit  of  account  for  collaborative  activities  under  the  Arbutus 
Agreement  and  concluded  there  is  one  activity,  to  run  an  open-label  Phase  2  clinical  trial,  which  is  akin  to 
performance  obligation  related  to  collaborative  activities.  Reimbursements  and  cost-sharing  portions  of  this 
performance obligation will be reflected as a reduction of research and development expense when realized in the 
Company’s  consolidated  statements  of  operations,  as  the  Company  does  not  consider  performing  research  and 
development  services  for  reimbursement  to  be  a  part  of  its  ongoing  major  or  central  operations.  During  the  year 
ended  December  31,  2020,  the  Company  recognized  a  reduction  of  research  and  development  expense  of  $0.2 
million under the Arbutus Agreement.

Contract Liabilities

The following tables present changes in the Company’s contract liabilities (in thousands):

Balance at
Beginning
of Period     Additions     Deductions    

Balance at
End of
Period  

Year Ended December 31, 2020
Contract liabilities:

Deferred revenue ............................................................  $

37,048    $

40,000    $

(68,061)  $

8,987 

Year Ended December 31, 2019
Contract liabilities:

Deferred revenue ............................................................  $

40,660    $

—    $

(3,612)  $

37,048  

F-34

 
 
     
       
       
       
 
     
       
       
       
 
 
     
       
       
       
 
     
       
       
       
 
     
       
       
       
 
Collaboration revenue recognized in the period from    
Amounts included in deferred revenue at the beginning
of the period........................................................................  $
Performance obligations satisfied in previous periods .......   

Note 10 – Strategic License Agreements 

HBV Research Agreement with Indiana University

Year Ended December 31,
2019

2018

2020

37,048    $
—     

3,612    $
—     

5,125 
—  

Since September 2013, the Company has been party to an exclusive License Agreement dated September 3, 2013 
with Indiana University Research and Technology Corporation (IURTC) from whom it has licensed aspects of the 
Company’s  HBV  program  held  by  IURTC.  The  license  agreement  requires  the  Company  to  make  milestone 
payments based upon the successful accomplishment of clinical and regulatory milestones. The aggregate amount of 
all  performance  milestone  payments  under  the  IURTC  license  agreement,  should  all  milestones  through 
development be met, is $0.8 million, with a portion related to the first performance milestone having been paid. The 
Company is obligated to pay IURTC royalty payments based on net sales of the licensed technology as well as a 
portion of any sublicensing revenue Assembly receives. The Company is also required to pay diligence maintenance 
fees  each  year  to  the  extent  that  the  royalty,  sublicensing,  and  milestone  payments  to  IURTC  are  less  than  the 
diligence  maintenance  fee  for  that  year.  A  performance  milestone  totaling  $0.1  million  was  determined  to  have 
occurred under this agreement and was paid during the year ended December 31, 2020. Additionally, the Company 
paid IURTC $0.7 million as a sublicensing fee during the year ended December 31, 2020. The Company made $0.1 
million  in  milestone  payments  for  the  year  ended  December  31,  2018.  No  milestone  payments  were  incurred  or 
accrued for under this agreement as of and for the year ended December 31, 2019. The milestone and license fees 
are included in research and development expenses in the consolidated statements of operations and comprehensive 
loss. 

Microbiome Targeted Colonic Delivery Platform

In  November  2013,  the  Company  entered  into  a  License  and  Collaboration  Agreement  with  Therabiome,  LLC 
(Therabiome),  for  all  intellectual  property  and  know-how  owned  or  controlled  by  Therabiome  relating  to  the  oral 
delivery of pharmaceutical drugs to specific sites in the intestine, using a pH sensitive controlled release capsule-in-
capsule technology. The Company will be solely responsible for all research and development activities with respect 
to any product it develops under the license.

The Company must pay Therabiome clinical and regulatory milestones for each product or therapy advanced from 
the  platform  for  U.S.  regulatory  milestones.  The  Company  also  must  pay  Therabiome  lesser  amounts  for  foreign 
regulatory  milestones,  which  vary  by  country  and  region.  The  Company  also  must  pay  Therabiome  royalties  on 
annual net sales of a product in the low to mid-single digit percentages plus, once annual net sales exceed certain 
thresholds, a one-time cash payment upon reaching the thresholds.

Therabiome must pay the Company royalties on annual net sales of any product Therabiome is permitted to develop 
using  the  intellectual  property  in  the  low  double  to  mid-double  digit  percentages,  depending  on  the  level  of 
development  or  involvement  the  Company  had  in  the  product.  Two  regulatory  milestones  resulting  in  payments 
totaling  $0.4  million  were  determined  to  have  occurred  under  this  agreement  and  were  paid  in  the  year  ended 
December  31,  2019.  No  amounts  were  incurred  or  accrued  for  this  agreement  as  of  and  for  the  years  ended 
December 31, 2020 and 2018. 

In  connection  with  the  wind-down  of  the  Microbiome  program,  the  License  and  Collaboration  Agreement  with 
Therabiome was terminated in January 2021.

F-35

 
 
 
 
 
   
   
 
      
      
  
Door Agreement

In  November  2020,  the  Company  and  Door  Pharmaceuticals,  LLC  (Door)  entered  into  an  exclusive,  two-year 
Collaboration Agreement and Sublicense Agreement (collectively, Door Agreement) focused on the development of 
a novel class of HBV inhibitors. Under the terms of the agreement, Door will build upon its previous efforts to lead 
and conduct new discovery research, which Assembly will fund. In return for an up-front payment of $1.8 million, 
success-based milestones up to $35.0 million, exercise and annual fees ranging from $0.1 million to $2.0 million and 
royalties  in  the  low  to  mid-single  digits,  the  Company  will  be  granted  an  exclusive  option  to  license  compounds 
arising  from  the  collaboration  and  will  be  responsible  for  the  continued  development  and  commercialization  of 
optioned compounds. For the period ended December 31, 2020, the Company incurred $0.3 million of research and 
development funding in addition to the $1.8 million up-front payment.

Under the consolidation accounting standard, the Company determined that Door is a VIE. The Company does not 
have the power to direct the activities that most significantly affect the economic performance of Door and as such 
the  Company  is  not  the  primary  beneficiary  and  consolidation  is  not  required.  As  of  December  31,  2020,  the 
Company has not provided financial or other support to Door that was not contractually required.

Note 11 - Income Taxes

There was no current income tax provision for the years ended December 31, 2020, 2019 and 2018. The deferred 
income  tax  expense  for  the  year  ended  December  31,  2020  was  not  material.  The  Company  recognized  deferred 
income tax benefit of $0.8 million for the year ended December 31, 2019 and a deferred income tax expense of $1.1 
million for the year ended December 31, 2018.

The effective tax rate of our provision for income taxes differs from the federal statutory rate as follows:

2020

As of December 31,
2019

2018

Statutory federal income tax rate .......................................   
State taxes, net of federal tax benefit .................................   
Stock based compensation .................................................   
Research and development tax credits ...............................   
State rate change.................................................................   
Uncertain tax positions.......................................................   
Return to provision adjustments.........................................   
Other...................................................................................   
Change in valuation allowance ..........................................   
Income taxes provision (benefit)........................................   

21.0%   
6.1 
0.7 
2.2 
— 
2.2 
4.3 
0.1 
(36.6)    
0.0%   

21.0%   
5.6 
(3.8)    
5.6 
(1.4)    
(2.1)    
(2.5)    
(0.2)    
(21.4)    
0.8%   

21.0%
7.1 
6.7 
2.4 
2.5 
(4.8)
4.4 
0.8 
(41.3)
(1.2)%

F-36

 
 
 
 
 
 
 
 
 
 
   
   
   
   
   
   
   
   
   
Significant components of the Company’s deferred taxes are as follows (in thousands):

As of December 31,

2020

2019

Deferred tax assets:

Federal and state-operating loss carryforwards..........................................  $
Stock-based compensation .........................................................................   
Intangible assets .........................................................................................   
Deferred revenue ........................................................................................   
Operating lease liabilities ...........................................................................   
Research and development credits .............................................................   
Other ...........................................................................................................   
Total deferred tax assets...................................................................................   
Valuation allowance.........................................................................................   
Deferred tax asset, net of valuation allowance ................................................  $

108,236    $
16,563   
1,463   
—   
2,600   
8,872   
854   
138,588   
(131,332)  

7,256    $

Deferred tax liabilities:

In-process research and development.........................................................  $
Operating lease right-of-use assets.............................................................   
Total deferred tax liabilities .............................................................................   
Net deferred tax liability ..................................................................................  $

(7,443)   $
(2,344)  
(9,787)  
(2,531)   $

81,584 
12,347 
1,774 
9,503 
3,147 
7,499 
702 
116,556 
(108,577)
7,979 

(7,439)
(3,071)
(10,510)
(2,531)

The Company maintains a valuation allowance on deferred tax assets due to the uncertainty regarding the ability to 
utilize  these  deferred  tax  assets  in  the  future.  The  increase  in  the  valuation  allowance  for  both  the  years  ended 
December  31,  2020  and  2019  is  primarily  due  to  an  increase  in  the  Company’s  federal  and  state-operating  loss 
carryforwards. The in-process research and development deferred tax liability was recorded in connection with the 
merger with Assembly Pharmaceuticals, Inc. in 2014 and relates to the difference between the carrying amount of 
in-process  research  and  development  for  financial  statement  purposes  relative  to  the  amount  used  for  income  tax 
purposes.

As of December 31, 2020, the Company had potentially utilizable gross federal net operating loss carryforwards of 
$378.8 million with $264.1 million of net operating losses that carry forward indefinitely and $114.7 million of net 
operating  losses  which  begin  to  expire  in  2027  if  not  utilized. There  are  state  net  operating  loss  carryforwards  of 
$446.8 million with $0.7 million carrying forward indefinitely and $446.1 million beginning to expire in 2031.  In 
addition,  the  Company  has  federal  research  and  development  credit  carryforwards  of  $8.5  million  which  begin  to 
expire in 2028 if not utilized and California research and development credit carryforwards of $3.6 million, which 
will carryforward indefinitely.

Pursuant  to  Internal  Revenue  Code  (IRC),  Section 382  and  383,  use  of  the  Company’s  U.S.  federal  and  state  net 
operating  loss  and  research  and  development  income  tax  credit  carryforwards  may  be  limited  in  the  event  of  a 
cumulative  change  in  ownership  of  more  than  50.0%  within  a  three-year  period.  The  Company  has  performed  an 
ownership change study through December 31, 2019 and has determined that a “change in ownership” as defined by 
IRC Section 382 and the rules and regulations promulgated thereunder, did occur in December 2010, January 2013 
and October 2014. The Company has adjusted its net operating loss carryovers to appropriately reflect any attributes 
which  will  expire  due  to  the  limitation.  The  Company  has  not  performed  any  additional  analysis  for  IRC 
Sections 382 and 383 and there is a risk that additional changes in ownership could have occurred since December 
31, 2018. If a change in ownership were to have occurred, additional net operating loss and tax credit carryforwards 
could  be  eliminated  or  restricted.  If  eliminated,  the  related  asset  would  be  removed  from  the  deferred  tax  asset 
schedule with a corresponding reduction in the valuation allowance.

F-37

 
 
 
 
 
   
 
   
    
 
  
 
 
 
 
 
 
 
 
 
   
    
 
  
   
    
 
  
 
 
The following table summarizes activity related to the Company’s gross unrecognized tax benefits (in thousands):

2020

As of December 31,
2019

2018

  Balances as of beginning of year ......................................  $
Increases related to prior year tax positions .....................   
  Decreases related to prior year tax positions ....................   
Increases related to current year tax positions..................   
  Balances as of end of year ................................................  $

6,070    $
—     
(4,162)    
747     
2,655    $

4,613    $
15     
(934)    
2,376     
6,070    $

— 
3,679 
— 
934 
4,613  

The  unrecognized  tax  benefits,  if  recognized,  would  not  have  an  impact  on  the  Company’s  effective  tax  rate 
assuming the Company continues to maintain a full valuation allowance position. Based on prior year’s operations 
and  experience,  the  Company  does  not  expect  a  significant  change  to  its  unrecognized  tax  benefits  over  the  next 
twelve  months.  The  unrecognized  tax  benefits  may  increase  or  change  during  the  next  year  for  unexpected  or 
unusual  items  for  items  that  arise  in  the  ordinary  course  of  business.  In  subsequent  periods,  any  interest  and 
penalties related to uncertain tax positions will be recognized as a component of income tax expense.

The Company files income tax returns in the U.S. federal, California and other state jurisdictions and is not currently 
under  examination  by  federal,  state,  or  local  taxing  authorities  for  any  open  tax  years.  Due  to  net  operating  loss 
carryforwards, all years effectively remain open for income tax examination by tax authorities in the U.S. and states 
in which the Company files tax returns.

Note 12 - Leases

Operating Leases

The Company leases corporate office and laboratory space in South San Francisco, California under a sub-sublease 
that  expires  in  December 2023.  The  sub-sublease  contains  scheduled  rent  increases  over  the  lease  term.  Prior  to 
moving into the South San Francisco office and laboratory space in February 2019, the Company leased office and 
laboratory space in San Francisco, California, under a sublease that expired in February 2019. The Company also 
leases  office  space  for  administrative  functions  in  Carmel,  Indiana  under  a  lease  agreement  that  expires  in 
August 2023.  In  February  2021,  the  Company  subleased  substantially  all  of  the  office  space  under  the  Carmel, 
Indiana  lease.  The  Company  also  leases  office  and  laboratory  space  in  Groton,  Connecticut  that  supports  the 
Microbiome program under a lease that expires in March 2021. Due to the wind-down of the Microbiome program, 
the lease will not be renewed. The Company’s China subsidiary leases office space and lab space in Shanghai. The 
lab space expired in December 2020 and the office space expires March 2021, neither of which are being renewed. 
Additionally, the Company’s China subsidiary leases office space in Beijing under a lease agreement that expires in 
December 2021. Certain lease contracts contain renewal clauses that the Company assesses on a case by case basis. 
The Company also leases certain laboratory equipment accounted for as operating leases expiring at various dates, 
with  the  final  lease  expiring  in  2023.  In  February  2021,  the  Company  purchased  substantially  all  of  the  leased 
equipment used for the Microbiome program from its leasing agency and sold them to a third party. The loss on the 
sale is equal to the impairment loss the Company recognized on these assets for the year ended December 31, 2020 
of $0.7 million. 

When the Company cannot determine the implicit rate in its leasing arrangements, the Company uses its incremental 
borrowing  rate  as  the  discount  rate  when  measuring  operating  lease  liabilities.  The  incremental  borrowing  rate 
represents an estimate of the interest rate the Company would incur at lease commencement to borrow an amount 
equal  to  the  lease  payments  on  a  collateralized  basis  over  the  term  of  a  lease  within  a  particular  currency 
environment.

F-38

 
 
 
 
 
 
 
   
   
 
 
 
At December 31, 2020, the Company had operating lease liabilities of $10.1 million and right-of-use assets of $9.1 
million.

The following summarizes quantitative information about the Company’s operating leases (in thousands):

Lease cost

Operating lease cost .........................................................................  $
Short-term lease cost........................................................................ 
Variable lease cost ........................................................................... 
Total lease cost ......................................................................................  $

5,214    $
401   
1,468   
7,083    $

4,454 
609 
1,193 
6,256  

Year Ended December 31,
2019
2020

Year Ended December 31,
2019
2020

Operating cash flows from operating leases..........................................  $
Right-of-use assets exchanged for new operating lease liabilities ........  $

4,513    $
1,302    $

4,269 
15,261  

As  of  December  31,  2020,  the  weighted-average  remaining  lease  term  for  operating  leases  was  2.7  years  and  the 
weighted-average discount rate for operating leases was 9.2%.

As of December 31, 2020, the maturities of the Company’s operating lease liabilities were as follows (in thousands):

2021....................................................................................................................................  $
2022.................................................................................................................................... 
2023.................................................................................................................................... 
Total ................................................................................................................................... 
Less: present value discount .............................................................................................. 
Operating lease liabilities...................................................................................................  $

4,369 
3,905 
3,502 
11,776 
(1,647)
10,129  

Operating lease costs were $7.1 million, $6.3 million and $4.2 million for the years ended December 31, 2020, 2019 
and 2018, respectively.

Note 13 - Employee Benefit Plan

In January 2018, the Company established a defined contribution 401(k) plan (the Plan) for all employees who are at 
least 21 years of age. Employees are eligible to participate in the Plan upon commencement of employment. Under 
the terms of the Plan, employees may make voluntary contributions as a percentage of compensation. The Plan also 
permits the Company to make discretionary matching contributions. In 2020, 2019 and 2018, the Company made 
discretionary matching contributions of $0.9 million, $0.7 million and $0.7 million, respectively.

F-39

 
 
 
 
 
   
 
 
   
   
   
 
 
 
 
 
 
 
 
 
 
   
 
 
 
 
 
Note 14 - Selected Quarterly Financial Data (Unaudited)

The following table contains quarterly financial information for the four quarters of 2020 and 2019 which has been 
prepared  in  accordance  with  GAAP  for  interim  financial  information.  The  Company  believes  that  the  following 
information reflects all normal recurring adjustments necessary for a fair statement of the information for the periods 
presented.

  March 31    

June 30

    September 30     December 31  

2020 Quarter Ended

Collaboration revenue ............................................  $
Operating expenses ................................................  $
Interest and other income .......................................  $
Net income (loss) ...................................................  $
Unrealized gain (loss) from marketable
securities, net of tax................................................  $
Basic net income (loss) per common share ............  $
Diluted net income (loss) per common share.........  $

(in thousands except for per share amounts)
4,081    $
31,775    $
1,039    $
(26,655)  $

34,611    $
38,630    $
670    $
(3,349)  $

39,376    $
32,797    $
691    $
7,270    $

115    $
(0.76)  $
(0.76)  $

190    $
0.21    $
0.19    $

(262)  $
(0.09)  $
(0.09)  $

1,037 
40,679 
224 
(39,418)

(112)
(1.11)
(1.11)

  March 31    

June 30

    September 30     December 31  

2019 Quarter Ended

Collaboration revenue ............................................  $
Operating expenses ................................................  $
Interest and other income .......................................  $
Net loss...................................................................  $
Unrealized gain (loss) from marketable
securities, net of tax................................................  $
Basic and diluted net loss per common share ........  $

Note 15 – Subsequent Events

(in thousands except for per share amounts)
3,885    $
32,221    $
1,276    $
(27,052)  $

3,080    $
22,780    $
1,182    $
(18,503)  $

4,231    $
30,224    $
983    $
(24,995)  $

4,767 
33,451 
859 
(27,084)

108    $
(1.05)  $

52    $
(0.72)  $

(18)  $
(0.96)  $

4 
(0.99)

Subsequent  to  December  31,  2020,  the  Company  sold  4,177,080  shares  of  common  stock  through  its  2020  ATM 
resulting in net proceeds of $25.5 million.

F-40

 
 
 
 
 
 
 
 
   
      
      
      
  
 
 
 
 
 
 
 
CORPORATE INFORMATION 

Directors  

Anthony E. Altig 
Former Chief Financial Officer, Biotix 
Holdings, Inc. 

Gina Consylman 
Chief Financial Officer, Ironwood 
Pharmaceuticals, Inc. 

Richard D. DiMarchi, Ph.D. 
Distinguished Professor of Biochemistry and 
Gill Chair in Biomolecular Sciences at Indiana 
University 

Myron Z. Holubiak 
President and Chief Executive Officer, Citius 
Pharmaceuticals, Inc. 

Susan Mahony, Ph.D. 
Former Senior Vice President and President of 
Lilly Oncology, Eli Lilly and Company 

John G. McHutchison, A.O., M.D. 
Chief Executive Officer and President, Assembly 
Biosciences, Inc. 

William R. Ringo, Jr. 
Chairman of the Board, Five Prime 
Therapeutics, Inc. 

Corporate Headquarters 
331 Oyster Point Blvd., Fourth Floor 
South San Francisco, California 94080 
+1.833.509.4583

Website 
www.assemblybio.com  

Stock Listing 
Assembly Biosciences, Inc. common stock is 
listed on The Nasdaq Global Select Market and 
quoted under the symbol “ASMB” 

Executive Officers 

John G. McHutchison, A.O., M.D. 
Chief Executive Officer and President 

Thomas J. Russo, CFA 
Chief Financial Officer 

Jason A. Okazaki 
Chief Legal and Business Officer 

Luisa Stamm, M.D., Ph.D. 
Chief Medical Officer 

William E. Delaney IV, Ph.D. 
Chief Scientific Officer 

Transfer Agent 
American Stock Transfer & Trust Company 
6201 15th Avenue 
Brooklyn, New York 11219 

331 Oyster Point Boulevard
4th Floor
South San Francisco, CA 94080

assemblybio.com

2020 Annual Report